Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cc		LIM class homeoboxes GOF	-			
2	100	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
3	100	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
4	99.99	oe	ccsbBroad304_00036	AFP	-			
5	99.99	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
6	99.99	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
7	99.97	oe	ccsbBroad304_01651	TCF7L2	-			
8	99.97	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
9	99.97	oe	ccsbBroad304_01066	NDUFA4	-			
10	99.97	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
11	99.97	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
12	99.97	oe	ccsbBroad304_01880	LAGE3	-			
13	99.97	oe	ccsbBroad304_00833	IFNG	Interferons			
14	99.97	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
15	99.97	oe	ccsbBroad304_03604	ENOSF1	-			
16	99.97	oe	ccsbBroad304_00464	DTNA	-			
17	99.97	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
18	99.97	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
19	99.97	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
20	99.97	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
21	99.97	oe	ccsbBroad304_05547	TMEM110	-			
22	99.97	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
23	99.97	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
24	99.97	oe	ccsbBroad304_12106	PXK	Slob family			
25	99.97	oe	ccsbBroad304_01163	PDHA1	-			
26	99.97	oe	ccsbBroad304_06665	OAT	-			
27	99.97	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
28	99.97	oe	ccsbBroad304_06569	MCM5	-			
29	99.97	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
30	99.97	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
31	99.97	oe	ccsbBroad304_02052	KYNU	-			
32	99.97	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
33	99.97	oe	ccsbBroad304_00809	HUS1	-			
34	99.97	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
35	99.97	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
36	99.97	oe	ccsbBroad304_06294	GNAZ	-			
37	99.97	oe	ccsbBroad304_00515	ERH	-			
38	99.97	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
39	99.97	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
40	99.97	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
41	99.97	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
42	99.97	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
43	99.97	oe	ccsbBroad304_00060	AMBP	Lipocalins			
44	99.97	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
45	99.97	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
46	99.97	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
47	99.97	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
48	99.97	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
49	99.97	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
50	99.97	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
51	99.97	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
52	99.97	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
53	99.97	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
54	99.97	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
55	99.97	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
56	99.97	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
57	99.97	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
58	99.97	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
59	99.97	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
60	99.97	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
61	99.97	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
62	99.97	kd	CGS001-10221	TRIB1	Trbl family			
63	99.97	kd	CGS001-89882	TPD52L3	-			
64	99.97	kd	CGS001-8576	STK16	NAK family			
65	99.97	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
66	99.97	kd	CGS001-340371	NRBP2	NRBP family			
67	99.97	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
68	99.97	kd	CGS001-389421	LIN28B	-			
69	99.97	kd	CGS001-5653	KLK6	Chymotrypsin			
70	99.97	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
71	99.97	kd	CGS001-9709	HERPUD1	-			
72	99.97	kd	CGS001-2882	GPX7	-			
73	99.97	kd	CGS001-2770	GNAI1	-			
74	99.97	kd	CGS001-9638	FEZ1	-			
75	99.97	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
76	99.97	kd	CGS001-1786	DNMT1	Methyltransferases			
77	99.97	kd	CGS001-79947	DHDDS	-			
78	99.97	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
79	99.97	kd	CGS001-84433	CARD11	-			
80	99.97	kd	CGS001-717	C2	Complement system			
81	99.97	kd	CGS001-10973	ASCC3	-			
82	99.97	kd	CGS001-367	AR	Nuclear hormone receptors			
83	99.97	kd	CGS001-328	APEX1	-			
84	99.97	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
85	99.96	cc		Beta-adrenergic receptor agonist	-			
86	99.96	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
87	99.96	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
88	99.96	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
89	99.96	oe	ccsbBroad304_12226	NAGK	-			
90	99.96	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
91	99.96	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
92	99.96	oe	ccsbBroad304_02551	CPSF4	-			
93	99.96	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
94	99.96	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
95	99.96	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
96	99.96	kd	CGS001-10474	TADA3	-			
97	99.96	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
98	99.96	kd	CGS001-4781	NFIB	-			
99	99.96	kd	CGS001-9787	DLGAP5	-			
100	99.95	kd	CGS001-5163	PDK1	-			
101	99.95	kd	CGS001-10289	EIF1B	-			
102	99.94	oe	ccsbBroad304_01008	KITLG	-			
103	99.94	oe	ccsbBroad304_01618	STXBP1	-			
104	99.94	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
105	99.94	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
106	99.94	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
107	99.94	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
108	99.94	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
109	99.94	kd	CGS001-9967	THRAP3	-			
110	99.94	kd	CGS001-1495	CTNNA1	Catenins			
111	99.94	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
112	99.93	oe	ccsbBroad304_02843	FTSJ1	-			
113	99.93	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
114	99.93	oe	ccsbBroad304_14242	MCCC2	-			
115	99.93	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
116	99.93	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
117	99.93	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
118	99.93	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
119	99.93	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
120	99.93	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
121	99.93	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
122	99.93	kd	CGS001-51002	TPRKB	-			
123	99.93	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
124	99.93	kd	CGS001-4801	NFYB	-			
125	99.93	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
126	99.93	kd	CGS001-665	BNIP3L	-			
127	99.93	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
128	99.91	cc		Homeobox Gene GOF	-			
129	99.91	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
130	99.91	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
131	99.91	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
132	99.91	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
133	99.91	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
134	99.91	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
135	99.91	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
136	99.91	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
137	99.91	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
138	99.91	kd	CGS001-9943	OXSR1	FRAY subfamily			
139	99.91	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
140	99.91	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
141	99.91	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
142	99.9	cc		Cyclooxygenase inhibitor	-			
143	99.9	oe	ccsbBroad304_03268	GMPR2	-			
144	99.9	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
145	99.9	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
146	99.9	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
147	99.9	kd	CGS001-4605	MYBL2	-			
148	99.9	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
149	99.9	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
150	99.9	kd	CGS001-79581	GPR172A	-			
151	99.88	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
152	99.88	kd	CGS001-9833	MELK	MELK subfamily			
153	99.88	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
154	99.87	oe	ccsbBroad304_07140	XPC	-			
155	99.87	oe	ccsbBroad304_01374	RAP1A	-			
156	99.87	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
157	99.87	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
158	99.87	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
159	99.86	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
160	99.85	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
161	99.85	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
162	99.85	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
163	99.85	oe	ccsbBroad304_06382	HMGCL	-			
164	99.85	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
165	99.85	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
166	99.85	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
167	99.85	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
168	99.85	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
169	99.85	kd	CGS001-5966	REL	NFkappaB transcription factor family			
170	99.85	kd	CGS001-2244	FGB	Endogenous ligands			
171	99.85	kd	CGS001-1606	DGKA	EF-hand domain containing			
172	99.85	kd	CGS001-965	CD58	CD molecules			
173	99.85	kd	CGS001-10096	ACTR3	-			
174	99.85	oe	ccsbBroad304_01974	RNASET2	-			
175	99.84	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
176	99.84	oe	ccsbBroad304_00644	GCLC	-			
177	99.84	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
178	99.84	kd	CGS001-8720	MBTPS1	Subtilisin			
179	99.84	kd	CGS001-7919	DDX39B	DEAD-boxes			
180	99.84	kd	CGS001-27241	BBS9	-			
181	99.82	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
182	99.82	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
183	99.81	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
184	99.81	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
185	99.81	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
186	99.81	oe	ccsbBroad304_01013	MIF	-			
187	99.81	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
188	99.81	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
189	99.79	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
190	99.79	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
191	99.78	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
192	99.78	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
193	99.78	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
194	99.78	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
195	99.78	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
196	99.78	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
197	99.78	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
198	99.78	kd	CGS001-7353	UFD1L	-			
199	99.78	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
200	99.78	kd	CGS001-1374	CPT1A	-			
201	99.77	kd	CGS001-6513	SLC2A1	Solute carriers			
202	99.76	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
203	99.75	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
204	99.75	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
205	99.75	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
206	99.75	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
207	99.75	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
208	99.75	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
209	99.75	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
210	99.73	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
211	99.73	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
212	99.73	kd	CGS001-1763	DNA2	-			
213	99.72	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
214	99.72	oe	ccsbBroad304_02572	SERINC3	-			
215	99.72	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
216	99.72	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
217	99.72	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
218	99.72	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
219	99.72	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
220	99.71	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
221	99.71	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
222	99.71	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
223	99.7	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
224	99.69	oe	ccsbBroad304_00469	DUT	-			
225	99.69	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
226	99.69	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
227	99.69	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
228	99.68	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
229	99.68	oe	ccsbBroad304_00570	FIGF	-			
230	99.68	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
231	99.68	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
232	99.68	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
233	99.67	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
234	99.66	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
235	99.66	oe	ccsbBroad304_06098	DHCR24	-			
236	99.66	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
237	99.66	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
238	99.66	kd	CGS001-3980	LIG3	-			
239	99.66	kd	CGS001-2771	GNAI2	-			
240	99.66	kd	CGS001-2353	FOS	basic leucine zipper proteins			
241	99.66	kd	CGS001-23536	ADAT1	-			
242	99.65	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
243	99.65	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
244	99.65	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
245	99.64	kd	CGS001-4522	MTHFD1	-			
246	99.63	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
247	99.63	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
248	99.63	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
249	99.63	kd	CGS001-2639	GCDH	-			
250	99.62	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
251	99.62	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
252	99.6	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
253	99.6	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
254	99.6	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
255	99.6	kd	CGS001-3169	FOXA1	Forkhead boxes			
256	99.59	oe	ccsbBroad304_02741	PDS5A	-			
257	99.59	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
258	99.59	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
259	99.59	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
260	99.59	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
261	99.59	kd	CGS001-10423	CDIPT	-			
262	99.57	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
263	99.57	kd	CGS001-5992	RFX4	-			
264	99.57	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
265	99.56	cc		Adenosine receptor agonist	-			
266	99.56	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
267	99.54	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
268	99.54	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
269	99.54	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
270	99.54	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
271	99.54	oe	ccsbBroad304_05756	ACAA1	-			
272	99.53	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
273	99.53	kd	CGS001-9847	KIAA0528	-			
274	99.51	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
275	99.51	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
276	99.5	oe	ccsbBroad304_08322	UFM1	-			
277	99.5	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
278	99.5	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
279	99.48	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
280	99.47	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
281	99.47	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
282	99.47	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
283	99.45	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
284	99.44	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
285	99.44	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
286	99.43	kd	CGS001-1376	CPT2	-			
287	99.42	kd	CGS001-51593	SRRT	-			
288	99.41	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
289	99.41	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
290	99.4	oe	ccsbBroad304_01787	YES1	Src family			
291	99.4	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
292	99.4	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
293	99.4	kd	CGS001-629	CFB	Complement system			
294	99.38	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
295	99.38	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
296	99.38	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
297	99.37	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
298	99.37	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
299	99.36	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
300	99.34	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
301	99.33	oe	ccsbBroad304_01872	DGCR14	-			
302	99.32	oe	ccsbBroad304_00370	CS	-			
303	99.32	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
304	99.31	kd	CGS001-23212	RRS1	-			
305	99.3	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
306	99.29	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
307	99.26	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
308	99.25	oe	ccsbBroad304_07890	CBX7	-			
309	99.25	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
310	99.25	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
311	99.24	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
312	99.23	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
313	99.23	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
314	99.22	oe	ccsbBroad304_01203	PIM1	PIM family			
315	99.22	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
316	99.22	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
317	99.22	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
318	99.22	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
319	99.21	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
320	99.2	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
321	99.17	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
322	99.16	kd	CGS001-6204	RPS10	S ribosomal proteins			
323	99.15	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
324	99.15	kd	CGS001-2212	FCGR2A	CD molecules			
325	99.14	oe	ccsbBroad304_08116	TBK1	IKK family			
326	99.14	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
327	99.14	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
328	99.13	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
329	99.12	oe	ccsbBroad304_00221	CASP3	Caspases			
330	99.12	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
331	99.11	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
332	99.11	kd	CGS001-22954	TRIM32	-			
333	99.09	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
334	99.09	oe	ccsbBroad304_00359	CPT1A	-			
335	99.09	kd	CGS001-55179	FAIM	-			
336	99.08	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
337	99.07	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
338	99.07	oe	ccsbBroad304_02443	HAX1	-			
339	99.06	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
340	99.06	kd	CGS001-79109	MAPKAP1	-			
341	99.04	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
342	99.04	oe	ccsbBroad304_06458	IRF3	-			
343	99.04	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
344	99.03	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
345	99.03	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
346	99.03	kd	CGS001-29984	RHOD	-			
347	99.02	kd	CGS001-9158	FIBP	-			
348	99.01	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
349	98.99	oe	ccsbBroad304_13903	MTAP	-			
350	98.96	oe	ccsbBroad304_03405	CHRAC1	-			
351	98.95	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
352	98.94	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
353	98.93	oe	ccsbBroad304_04619	GNG8	-			
354	98.91	kd	CGS001-1676	DFFA	-			
355	98.89	oe	ccsbBroad304_00795	HSF2	-			
356	98.89	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
357	98.88	oe	ccsbBroad304_02485	STAMBP	-			
358	98.88	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
359	98.86	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
360	98.86	kd	CGS001-391013	PLA2G2C	-			
361	98.86	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
362	98.85	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
363	98.85	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
364	98.83	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
365	98.82	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
366	98.82	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
367	98.8	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
368	98.78	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
369	98.77	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
370	98.76	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
371	98.76	kd	CGS001-7423	VEGFB	-			
372	98.76	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
373	98.73	oe	ccsbBroad304_02837	BHMT2	-			
374	98.72	oe	ccsbBroad304_00164	BLMH	-			
375	98.71	kd	CGS001-1465	CSRP1	-			
376	98.7	kd	CGS001-1120	CHKB	-			
377	98.69	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
378	98.68	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
379	98.67	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
380	98.66	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
381	98.65	kd	CGS001-4170	MCL1	-			
382	98.63	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
383	98.62	kd	CGS001-10190	TXNDC9	-			
384	98.61	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
385	98.61	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
386	98.58	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
387	98.52	kd	CGS001-2023	ENO1	-			
388	98.51	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
389	98.51	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
390	98.51	kd	CGS001-3927	LASP1	-			
391	98.5	kd	CGS001-4610	MYCL1	-			
392	98.48	kd	CGS001-8089	YEATS4	-			
393	98.46	oe	ccsbBroad304_06695	PCK2	-			
394	98.45	oe	ccsbBroad304_10437	STMN1	-			
395	98.45	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
396	98.44	oe	ccsbBroad304_07097	TRAF1	-			
397	98.43	oe	ccsbBroad304_03113	DSE	-			
398	98.41	kd	CGS001-55810	FOXJ2	Forkhead boxes			
399	98.38	oe	ccsbBroad304_07018	SUPT5H	-			
400	98.38	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
401	98.37	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
402	98.37	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
403	98.35	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
404	98.34	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
405	98.34	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
406	98.33	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
407	98.33	kd	CGS001-8531	CSDA	-			
408	98.27	oe	ccsbBroad304_07569	TRIB1	Trbl family			
409	98.26	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
410	98.26	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
411	98.25	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
412	98.25	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
413	98.25	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
414	98.23	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
415	98.18	kd	CGS001-1949	EFNB3	Ephrins			
416	98.15	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
417	98.15	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
418	98.14	oe	ccsbBroad304_00001	NAT1	-			
419	98.13	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
420	98.12	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
421	98.12	kd	CGS001-54915	YTHDF1	-			
422	98.08	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
423	98.07	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
424	98.06	kd	CGS001-435	ASL	-			
425	98.01	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
426	98	kd	CGS001-6652	SORD	-			
427	98	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
428	97.99	oe	ccsbBroad304_06718	PFN2	-			
429	97.99	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
430	97.95	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
431	97.93	kd	CGS001-3032	HADHB	-			
432	97.92	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
433	97.92	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
434	97.9	oe	ccsbBroad304_00964	SMAD7	SMADs			
435	97.88	kd	CGS001-89910	UBE3B	-			
436	97.87	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
437	97.86	kd	CGS001-5091	PC	Carboxylases			
438	97.85	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
439	97.83	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
440	97.82	oe	ccsbBroad304_13939	MOK	RCK family			
441	97.8	kd	CGS001-5428	POLG	DNA polymerases			
442	97.79	kd	CGS001-9807	IP6K1	-			
443	97.77	kd	CGS001-9870	KIAA0317	-			
444	97.76	oe	ccsbBroad304_03129	ERO1L	-			
445	97.75	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
446	97.74	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
447	97.74	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
448	97.73	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
449	97.72	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
450	97.72	kd	CGS001-1892	ECHS1	-			
451	97.71	oe	ccsbBroad304_07704	SUB1	-			
452	97.7	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
453	97.69	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
454	97.69	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
455	97.68	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
456	97.67	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
457	97.66	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
458	97.65	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
459	97.62	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
460	97.62	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
461	97.61	oe	ccsbBroad304_06013	CLPTM1	-			
462	97.61	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
463	97.61	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
464	97.59	kd	CGS001-4077	NBR1	-			
465	97.59	kd	CGS001-64077	LHPP	-			
466	97.58	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
467	97.58	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
468	97.57	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
469	97.55	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
470	97.55	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
471	97.55	kd	CGS001-2247	FGF2	Endogenous ligands			
472	97.54	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
473	97.49	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
474	97.47	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
475	97.47	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
476	97.44	kd	CGS001-3098	HK1	-			
477	97.42	oe	ccsbBroad304_02045	BUD31	-			
478	97.41	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
479	97.4	kd	CGS001-150094	SIK1	QIK subfamily			
480	97.39	kd	CGS001-4946	OAZ1	-			
481	97.37	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
482	97.37	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
483	97.35	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
484	97.35	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
485	97.35	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
486	97.34	oe	ccsbBroad304_00116	ASS1	-			
487	97.32	kd	CGS001-10284	SAP18	-			
488	97.31	cc		Thymidylate synthase inhibitor	-			
489	97.3	kd	CGS001-56654	NPDC1	-			
490	97.3	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
491	97.29	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
492	97.29	kd	CGS001-7311	UBA52	L ribosomal proteins			
493	97.27	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
494	97.27	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
495	97.26	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
496	97.22	kd	CGS001-2475	MTOR	FRAP subfamily			
497	97.22	kd	CGS001-51292	GMPR2	-			
498	97.19	kd	CGS001-1659	DHX8	DEAH-boxes			
499	97.17	kd	CGS001-10434	LYPLA1	-			
500	97.16	oe	ccsbBroad304_01371	RALA	-			
501	97.16	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
502	97.15	kd	CGS001-701	BUB1B	Bub family			
503	97.14	oe	ccsbBroad304_00650	GNA11	-			
504	97.14	kd	CGS001-26277	TINF2	-			
505	97.11	oe	ccsbBroad304_00459	DPYD	-			
506	97.08	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
507	97.07	kd	CGS001-4482	MSRA	-			
508	97.07	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
509	97.06	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
510	97.05	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
511	97.03	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
512	97.01	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
513	97	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
514	97	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
515	96.97	oe	ccsbBroad304_08104	MED4	-			
516	96.97	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
517	96.97	kd	CGS001-2745	GLRX	-			
518	96.97	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
519	96.96	oe	ccsbBroad304_02737	JMJD6	-			
520	96.93	oe	ccsbBroad304_06424	IFI16	-			
521	96.93	kd	CGS001-9231	DLG5	-			
522	96.92	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
523	96.91	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
524	96.89	kd	CGS001-64863	METTL4	-			
525	96.88	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
526	96.87	kd	CGS001-5590	PRKCZ	Iota subfamily			
527	96.86	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
528	96.84	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
529	96.82	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
530	96.81	cc		FOS transcription factor family GOF	-			
531	96.81	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
532	96.8	kd	CGS001-9404	LPXN	-			
533	96.77	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
534	96.73	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
535	96.73	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
536	96.72	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
537	96.68	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
538	96.66	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
539	96.65	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
540	96.63	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
541	96.62	oe	ccsbBroad304_01845	RDBP	-			
542	96.62	kd	CGS001-23530	NNT	-			
543	96.61	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
544	96.61	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
545	96.56	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
546	96.56	kd	CGS001-2550	GABBR1	GABA receptors			
547	96.51	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
548	96.5	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
549	96.49	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
550	96.46	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
551	96.44	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
552	96.44	kd	CGS001-11129	CLASRP	-			
553	96.41	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
554	96.4	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
555	96.38	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
556	96.37	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
557	96.35	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
558	96.35	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
559	96.35	kd	CGS001-25913	POT1	-			
560	96.35	kd	CGS001-55893	ZNF395	Zinc fingers, C2H2-type			
561	96.33	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
562	96.3	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
563	96.3	kd	CGS001-55556	ENOSF1	-			
564	96.27	oe	ccsbBroad304_08266	PIPOX	-			
565	96.27	oe	ccsbBroad304_04170	PANK2	-			
566	96.26	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
567	96.24	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
568	96.23	kd	CGS001-4700	NDUFA6	LYR motif containing			
569	96.22	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
570	96.22	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
571	96.22	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
572	96.18	cc		Serotonin receptor agonist	-			
573	96.17	oe	ccsbBroad304_00941	LIG3	-			
574	96.17	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
575	96.14	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
576	96.12	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
577	96.1	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
578	96.09	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
579	96.09	kd	CGS001-10670	RRAGA	-			
580	96.06	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
581	96.06	kd	CGS001-57222	ERGIC1	-			
582	96.04	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
583	96.03	kd	CGS001-116443	GRIN3A	Glutamate receptors			
584	96.02	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
585	96	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
586	96	oe	ccsbBroad304_06255	LRRC32	-			
587	95.99	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
588	95.96	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
589	95.94	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
590	95.94	kd	CGS001-10928	RALBP1	-			
591	95.93	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
592	95.87	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
593	95.83	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
594	95.74	oe	ccsbBroad304_01208	PITPNA	-			
595	95.74	kd	CGS001-5018	OXA1L	-			
596	95.72	oe	ccsbBroad304_08386	SMOX	-			
597	95.72	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
598	95.7	oe	ccsbBroad304_01613	STK11	LKB subfamily			
599	95.7	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
600	95.69	cc		Rho associated kinase inhibitor	-			
601	95.69	kd	CGS001-1725	DHPS	-			
602	95.69	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
603	95.61	kd	CGS001-64223	MLST8	WD repeat domain containing			
604	95.6	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
605	95.44	kd	CGS001-3689	ITGB2	Integrins			
606	95.43	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
607	95.41	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
608	95.4	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
609	95.39	kd	CGS001-6884	TAF13	-			
610	95.38	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
611	95.37	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
612	95.34	oe	ccsbBroad304_06642	NIT1	-			
613	95.33	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
614	95.3	kd	CGS001-23585	TMEM50A	-			
615	95.3	kd	CGS001-7001	PRDX2	-			
616	95.22	kd	CGS001-79006	METRN	-			
617	95.21	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
618	95.21	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
619	95.21	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
620	95.21	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
621	95.21	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
622	95.2	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
623	95.18	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
624	95.18	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
625	95.16	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
626	95.12	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
627	95.1	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
628	95.1	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
629	95.06	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
630	95.06	kd	CGS001-230	ALDOC	-			
631	95.06	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
632	95.05	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
633	95.01	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
634	95	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
635	94.99	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
636	94.99	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
637	94.97	kd	CGS001-597	BCL2A1	-			
638	94.92	kd	CGS001-5223	PGAM1	-			
639	94.89	kd	CGS001-4193	MDM2	-			
640	94.86	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
641	94.86	oe	ccsbBroad304_02686	COPZ1	-			
642	94.86	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
643	94.86	kd	CGS001-55715	DOK4	Pleckstrin homology (PH) domain containing			
644	94.84	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
645	94.82	cc		MDM inhibitor	-			
646	94.81	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
647	94.78	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
648	94.73	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
649	94.68	oe	ccsbBroad304_03874	UBL5	-			
650	94.67	oe	ccsbBroad304_01623	SUPT4H1	-			
651	94.67	oe	ccsbBroad304_03237	LEF1	-			
652	94.64	kd	CGS001-5092	PCBD1	-			
653	94.62	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
654	94.61	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
655	94.59	kd	CGS001-23463	ICMT	-			
656	94.58	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
657	94.58	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
658	94.54	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
659	94.52	oe	ccsbBroad304_01395	RFX5	-			
660	94.5	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
661	94.47	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
662	94.4	kd	CGS001-25874	BRP44	-			
663	94.38	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
664	94.37	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
665	94.36	kd	CGS001-63948	DMRTB1	-			
666	94.34	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
667	94.33	kd	CGS001-4255	MGMT	-			
668	94.3	kd	CGS001-6520	SLC3A2	SLC3 family			
669	94.3	kd	CGS001-51268	PIPOX	-			
670	94.28	oe	ccsbBroad304_01139	PA2G4	-			
671	94.28	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
672	94.23	oe	ccsbBroad304_07029	TADA2A	-			
673	94.23	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
674	94.22	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
675	94.2	oe	ccsbBroad304_03232	VPS28	-			
676	94.2	kd	CGS001-1512	CTSH	Cathepsins			
677	94.17	oe	ccsbBroad304_06235	G6PD	-			
678	94.13	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
679	94.08	kd	CGS001-5927	KDM5A	Histone demethylases			
680	94.07	kd	CGS001-2098	ESD	-			
681	94.05	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
682	94.01	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
683	93.98	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
684	93.97	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
685	93.95	kd	CGS001-10671	DCTN6	-			
686	93.94	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
687	93.89	kd	CGS001-6647	SOD1	-			
688	93.87	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
689	93.82	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
690	93.79	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
691	93.77	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
692	93.74	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
693	93.68	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
694	93.65	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
695	93.65	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
696	93.62	oe	ccsbBroad304_04626	EGLN3	-			
697	93.6	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
698	93.6	kd	CGS001-1488	CTBP2	-			
699	93.59	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
700	93.56	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
701	93.56	kd	CGS001-873	CBR1	Prostaglandin synthases			
702	93.54	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
703	93.53	kd	CGS001-1605	DAG1	-			
704	93.5	kd	CGS001-23142	DCUN1D4	-			
705	93.47	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
706	93.46	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
707	93.44	oe	ccsbBroad304_02956	EHF	-			
708	93.25	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
709	93.25	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
710	93.23	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
711	93.22	oe	ccsbBroad304_07662	NPRL2	-			
712	93.21	oe	ccsbBroad304_02231	USP6NL	-			
713	93.2	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
714	93.19	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
715	93.16	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
716	93.16	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
717	93.16	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
718	93.08	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
719	93.08	oe	ccsbBroad304_06159	CTTN	-			
720	93.08	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
721	93.01	oe	ccsbBroad304_08553	STAP2	-			
722	92.98	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
723	92.87	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
724	92.87	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
725	92.83	kd	CGS001-8805	TRIM24	TIF1 family			
726	92.8	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
727	92.78	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
728	92.77	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
729	92.73	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
730	92.71	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
731	92.66	kd	CGS001-572	BAD	-			
732	92.64	kd	CGS001-111	ADCY5	Adenylate cyclases			
733	92.61	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
734	92.57	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
735	92.52	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
736	92.51	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
737	92.48	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
738	92.47	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
739	92.38	kd	CGS001-55837	EAPP	-			
740	92.35	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
741	92.33	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
742	92.33	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
743	92.31	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
744	92.3	oe	ccsbBroad304_06654	NPM1	-			
745	92.24	kd	CGS001-8896	BUD31	-			
746	92.21	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
747	92.2	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
748	92.19	kd	CGS001-9180	OSMR	IL-6 receptor family			
749	92.16	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
750	92.14	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
751	92.11	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
752	92.1	kd	CGS001-23710	GABARAPL1	-			
753	92.02	kd	CGS001-3248	HPGD	Prostaglandin synthases			
754	92.01	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
755	92	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
756	91.94	kd	CGS001-53340	SPA17	-			
757	91.86	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
758	91.81	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
759	91.81	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
760	91.8	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
761	91.78	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
762	91.77	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
763	91.77	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
764	91.7	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
765	91.7	kd	CGS001-1195	CLK1	CDC-like kinases			
766	91.7	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
767	91.7	oe	ccsbBroad304_05948	CCND2	-			
768	91.68	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
769	91.66	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
770	91.6	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
771	91.58	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
772	91.55	oe	ccsbBroad304_08346	COQ3	-			
773	91.54	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
774	91.53	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
775	91.49	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
776	91.48	kd	CGS001-1211	CLTA	-			
777	91.44	oe	ccsbBroad304_02287	GNPDA1	-			
778	91.33	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
779	91.33	kd	CGS001-10084	PQBP1	-			
780	91.29	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
781	91.26	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
782	91.2	oe	ccsbBroad304_00709	GUK1	-			
783	91.19	oe	ccsbBroad304_02058	PLOD3	-			
784	91.19	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
785	91.07	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
786	91.06	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
787	91.05	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
788	91.03	kd	CGS001-1788	DNMT3A	Methyltransferases			
789	90.93	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
790	90.88	kd	CGS001-57787	MARK4	MARK subfamily			
791	90.87	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
792	90.86	oe	ccsbBroad304_08045	NOX1	-			
793	90.85	oe	ccsbBroad304_05528	TICAM2	-			
794	90.83	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
795	90.79	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
796	90.78	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
797	90.77	cc		Lysine acetyltransferases LOF	-			
798	90.77	kd	CGS001-498	ATP5A1	ATPases / F-type			
799	90.72	kd	CGS001-54442	KCTD5	-			
800	90.71	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
801	90.65	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
802	90.57	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
803	90.54	kd	CGS001-1509	CTSD	Cathepsins			
804	90.52	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
805	90.49	oe	ccsbBroad304_01215	PLAUR	CD molecules			
806	90.47	oe	ccsbBroad304_06975	SMARCC2	-			
807	90.45	oe	ccsbBroad304_03506	AURKAIP1	-			
808	90.45	kd	CGS001-4282	MIF	-			
809	90.43	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
810	90.42	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
811	90.42	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
812	90.41	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
813	90.4	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
814	90.39	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
815	90.34	kd	CGS001-8050	PDHX	-			
816	90.32	oe	ccsbBroad304_06645	NQO2	-			
817	90.27	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
818	90.19	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
819	90.17	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
820	90.13	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
821	90.13	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
822	90.12	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
823	90.07	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
824	90.02	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
825	90	oe	ccsbBroad304_03266	ERGIC2	-			
826	89.98	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
827	89.97	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
828	89.96	kd	CGS001-80347	COASY	-			
829	89.93	oe	ccsbBroad304_01234	POLB	DNA polymerases			
830	89.89	oe	ccsbBroad304_03357	RASD1	-			
831	89.88	kd	CGS001-4016	LOXL1	-			
832	89.82	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
833	89.8	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
834	89.76	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
835	89.67	oe	ccsbBroad304_02674	STK38	NDR family			
836	89.67	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
837	89.66	oe	ccsbBroad304_00170	BNIP1	-			
838	89.64	oe	ccsbBroad304_02048	BCL10	-			
839	89.64	oe	ccsbBroad304_04891	TMEM174	-			
840	89.55	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
841	89.53	oe	ccsbBroad304_01131	OXCT1	-			
842	89.5	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
843	89.37	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
844	89.36	kd	CGS001-900	CCNG1	-			
845	89.35	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
846	89.31	kd	CGS001-5682	PSMA1	Proteasome subunits			
847	89.28	oe	ccsbBroad304_09225	BUD13	-			
848	89.27	kd	CGS001-10672	GNA13	-			
849	89.24	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
850	89.2	oe	ccsbBroad304_07561	YAF2	-			
851	89.15	oe	ccsbBroad304_05887	CFB	Complement system			
852	89.11	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
853	89.04	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
854	89.02	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
855	89.02	kd	CGS001-9817	KEAP1	Kelch-like proteins			
856	88.99	oe	ccsbBroad304_06089	DDIT3	-			
857	88.98	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
858	88.95	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
859	88.93	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
860	88.91	kd	CGS001-25793	FBXO7	F-boxes / other			
861	88.88	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
862	88.87	oe	ccsbBroad304_03191	NOSIP	-			
863	88.87	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
864	88.84	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
865	88.84	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
866	88.82	kd	CGS001-7248	TSC1	-			
867	88.81	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
868	88.77	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
869	88.75	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
870	88.74	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
871	88.73	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
872	88.6	kd	CGS001-624	BDKRB2	Bradykinin receptors			
873	88.56	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
874	88.54	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
875	88.5	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
876	88.5	kd	CGS001-399664	MEX3D	Mex-3 homologs			
877	88.5	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
878	88.49	oe	ccsbBroad304_06998	SRPK1	SRPK family			
879	88.48	oe	ccsbBroad304_07616	ZNF238	-			
880	88.42	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
881	88.37	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
882	88.31	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
883	88.29	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
884	88.26	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
885	88.26	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
886	88.22	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
887	88.2	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
888	88.18	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
889	88.17	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
890	88.15	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
891	88	cc		HIV protease inhibitor	-			
892	88	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
893	88	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
894	87.98	oe	ccsbBroad304_02869	ASF1A	-			
895	87.98	kd	CGS001-56675	NRIP3	-			
896	87.96	cc		ATP synthase inhibitor	-			
897	87.96	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
898	87.94	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
899	87.9	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
900	87.84	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
901	87.83	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
902	87.82	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
903	87.74	oe	ccsbBroad304_07851	FAM120A	-			
904	87.73	kd	CGS001-10493	VAT1	-			
905	87.68	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
906	87.67	kd	CGS001-6347	CCL2	Chemokine ligands			
907	87.65	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
908	87.59	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
909	87.58	kd	CGS001-7097	TLR2	Toll-like receptor family			
910	87.58	kd	CGS001-51564	HDAC7	Histone deacetylases			
911	87.53	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
912	87.5	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
913	87.49	oe	ccsbBroad304_00969	MAGEA10	-			
914	87.42	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
915	87.4	cc		Mitogen activated protein kinases LOF	-			
916	87.38	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
917	87.37	kd	CGS001-11340	EXOSC8	-			
918	87.35	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
919	87.33	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
920	87.31	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
921	87.31	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
922	87.24	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
923	87.19	oe	ccsbBroad304_01054	GADD45B	-			
924	87.05	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
925	87.05	kd	CGS001-6857	SYT1	Synaptotagmins			
926	87.01	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
927	86.98	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
928	86.88	cc		Bile acid	-			
929	86.88	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
930	86.84	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
931	86.79	oe	ccsbBroad304_07920	NUP62	-			
932	86.79	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
933	86.78	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
934	86.75	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
935	86.74	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
936	86.7	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
937	86.68	oe	ccsbBroad304_00003	ABAT	GABA turnover			
938	86.65	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
939	86.62	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
940	86.62	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
941	86.6	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
942	86.57	kd	CGS001-2079	ERH	-			
943	86.55	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
944	86.55	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
945	86.53	kd	CGS001-25819	CCRN4L	-			
946	86.52	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
947	86.52	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
948	86.4	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
949	86.4	kd	CGS001-3034	HAL	-			
950	86.32	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
951	86.29	oe	ccsbBroad304_03555	PANK4	-			
952	86.1	oe	ccsbBroad304_00615	GAPDH	-			
953	86.09	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
954	86.07	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
955	86.04	kd	CGS001-2538	G6PC	-			
956	85.98	oe	ccsbBroad304_09035	COASY	-			
957	85.98	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
958	85.93	oe	ccsbBroad304_04387	MKI67IP	-			
959	85.92	oe	ccsbBroad304_07798	EXOC3	-			
960	85.89	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
961	85.83	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
962	85.81	kd	CGS001-11124	FAF1	UBX domain containing			
963	85.8	kd	CGS001-91433	RCCD1	-			
964	85.79	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
965	85.76	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
966	85.7	kd	CGS001-8895	CPNE3	-			
967	85.68	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
968	85.66	oe	ccsbBroad304_06670	OGG1	-			
969	85.65	kd	CGS001-1647	GADD45A	-			
970	85.63	kd	CGS001-10111	RAD50	-			
971	85.62	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
972	85.56	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
973	85.53	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
974	85.52	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
975	85.51	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
976	85.49	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
977	85.43	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
978	85.36	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
979	85.35	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
980	85.34	kd	CGS001-7728	ZNF175	Zinc fingers, C2H2-type			
981	85.33	oe	ccsbBroad304_01560	SNAPC1	-			
982	85.33	oe	ccsbBroad304_01101	NME1	-			
983	85.31	oe	ccsbBroad304_02845	PRPF6	-			
984	85.28	oe	ccsbBroad304_00957	M6PR	-			
985	85.27	cc		X linked mental retardation group 2 LOF	-			
986	85.27	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
987	85.26	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
988	85.18	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
989	85.14	kd	CGS001-64135	IFIH1	-			
990	85.13	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
991	85.11	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
992	85.09	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
993	85.04	kd	CGS001-10691	GMEB1	-			
994	85.03	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
995	84.98	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
996	84.96	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
997	84.94	oe	ccsbBroad304_02633	LSM6	-			
998	84.86	kd	CGS001-6778	STAT6	SH2 domain containing			
999	84.84	kd	CGS001-306	ANXA3	Annexins			
1000	84.82	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
1001	84.79	kd	CGS001-2931	GSK3A	GSK subfamily			
1002	84.78	kd	CGS001-3251	HPRT1	-			
1003	84.76	oe	ccsbBroad304_06282	GLDC	-			
1004	84.73	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
1005	84.73	kd	CGS001-587	BCAT2	-			
1006	84.68	oe	ccsbBroad304_00034	AES	-			
1007	84.67	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
1008	84.66	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
1009	84.6	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
1010	84.59	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
1011	84.51	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
1012	84.5	kd	CGS001-23161	SNX13	Sorting nexins			
1013	84.47	oe	ccsbBroad304_00995	MECP2	-			
1014	84.4	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
1015	84.39	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
1016	84.32	oe	ccsbBroad304_00532	F11	Chymotrypsin			
1017	84.32	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
1018	84.23	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
1019	84.21	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
1020	84.19	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1021	84.16	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
1022	84.15	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1023	84.12	oe	ccsbBroad304_03848	METTL14	-			
1024	84.11	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
1025	84.09	oe	ccsbBroad304_01576	SOAT1	-			
1026	84.09	kd	CGS001-2752	GLUL	-			
1027	84.08	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
1028	84.04	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
1029	84	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
1030	83.97	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
1031	83.91	kd	CGS001-3033	HADH	-			
1032	83.87	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
1033	83.87	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
1034	83.81	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
1035	83.72	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
1036	83.72	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
1037	83.71	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
1038	83.67	kd	CGS001-54505	DHX29	DEAH-boxes			
1039	83.61	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
1040	83.6	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
1041	83.6	kd	CGS001-6603	SMARCD2	-			
1042	83.5	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1043	83.49	oe	ccsbBroad304_02578	EBNA1BP2	-			
1044	83.49	kd	CGS001-80135	RPF1	-			
1045	83.42	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
1046	83.41	kd	CGS001-55437	STRADB	STLK subfamily			
1047	83.41	kd	CGS001-308	ANXA5	Annexins			
1048	83.33	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
1049	83.31	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
1050	83.28	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
1051	83.25	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
1052	83.24	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
1053	83.23	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
1054	83.18	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
1055	83.13	kd	CGS001-50813	COPS7A	-			
1056	83.11	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
1057	83.1	oe	ccsbBroad304_02386	EIF1B	-			
1058	83.1	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
1059	83.06	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
1060	82.94	kd	CGS001-200734	SPRED2	-			
1061	82.93	kd	CGS001-7771	ZFP112	-			
1062	82.92	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
1063	82.91	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1064	82.89	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
1065	82.89	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
1066	82.87	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
1067	82.83	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
1068	82.83	kd	CGS001-29937	NENF	-			
1069	82.82	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
1070	82.81	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
1071	82.76	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
1072	82.71	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
1073	82.71	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
1074	82.69	kd	CGS001-253430	IPMK	-			
1075	82.67	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
1076	82.65	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
1077	82.57	kd	CGS001-5446	PON3	Paraoxonases			
1078	82.54	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
1079	82.52	cc		Tachykinin antagonist	-			
1080	82.52	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
1081	82.5	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
1082	82.5	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
1083	82.49	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
1084	82.48	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
1085	82.48	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
1086	82.46	kd	CGS001-6256	RXRA	Retinoid X receptors			
1087	82.42	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
1088	82.42	kd	CGS001-378	ARF4	ADP-ribosylation factors			
1089	82.39	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
1090	82.23	oe	ccsbBroad304_08481	CEP55	-			
1091	82.2	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1092	82.19	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
1093	82.18	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
1094	82.15	kd	CGS001-23223	RRP12	-			
1095	82.15	kd	CGS001-57804	POLD4	DNA polymerases			
1096	82.13	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
1097	82.07	oe	ccsbBroad304_06720	PHYH	-			
1098	82	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
1099	81.97	oe	ccsbBroad304_06291	GNAI1	-			
1100	81.78	kd	CGS001-4292	MLH1	-			
1101	81.77	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1102	81.73	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
1103	81.72	cp	BRD-A71009679	KUC103420N	-666			-666
1104	81.65	oe	ccsbBroad304_01413	RPA2	-			
1105	81.65	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
1106	81.61	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
1107	81.6	kd	CGS001-8829	NRP1	CD molecules			
1108	81.58	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
1109	81.56	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
1110	81.55	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
1111	81.52	oe	ccsbBroad304_04153	PHF17	-			
1112	81.46	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
1113	81.45	kd	CGS001-60528	ELAC2	-			
1114	81.44	oe	ccsbBroad304_02653	PRAF2	-			
1115	81.44	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
1116	81.43	oe	ccsbBroad304_02500	RRAGA	-			
1117	81.43	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1118	81.42	oe	ccsbBroad304_04404	TUBB6	Tubulins			
1119	81.32	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
1120	81.32	kd	CGS001-115	ADCY9	Adenylyl cyclases			
1121	81.25	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
1122	81.24	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
1123	81.2	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
1124	81.19	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
1125	81.16	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
1126	81.1	oe	ccsbBroad304_01247	POU2AF1	-			
1127	81.08	kd	CGS001-36	ACADSB	-			
1128	81.03	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
1129	80.99	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
1130	80.96	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
1131	80.95	kd	CGS001-23139	MAST2	MAST family			
1132	80.94	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
1133	80.93	oe	ccsbBroad304_03097	CNOT7	-			
1134	80.9	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
1135	80.82	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
1136	80.76	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
1137	80.65	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
1138	80.63	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1139	80.62	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1140	80.61	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
1141	80.58	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
1142	80.57	oe	ccsbBroad304_08684	CXCR7	-			
1143	80.55	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
1144	80.54	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
1145	80.5	oe	ccsbBroad304_03772	CCNL1	-			
1146	80.5	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
1147	80.48	kd	CGS001-5144	PDE4D	Phosphodiesterases			
1148	80.46	kd	CGS001-9170	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1149	80.38	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
1150	80.21	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
1151	80.21	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
1152	80.2	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
1153	80.14	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
1154	80.08	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
1155	80.07	oe	ccsbBroad304_02566	MORF4L1	-			
1156	80	kd	CGS001-51441	YTHDF2	-			
1157	79.98	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
1158	79.89	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
1159	79.86	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
1160	79.79	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
1161	79.77	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
1162	79.77	kd	CGS001-25942	SIN3A	-			
1163	79.73	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
1164	79.72	kd	CGS001-5743	PTGS2	Cyclooxygenase			
1165	79.7	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
1166	79.7	kd	CGS001-10613	ERLIN1	-			
1167	79.67	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
1168	79.67	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
1169	79.66	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
1170	79.66	kd	CGS001-100	ADA	Adenosine turnover			
1171	79.63	cc		Retinoid receptor agonist	-			
1172	79.62	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
1173	79.57	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
1174	79.55	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
1175	79.5	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
1176	79.44	kd	CGS001-2768	GNA12	-			
1177	79.43	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
1178	79.42	kd	CGS001-51001	MTERFD1	-			
1179	79.37	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
1180	79.36	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
1181	79.3	oe	ccsbBroad304_02496	MTX2	-			
1182	79.3	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
1183	79.3	kd	CGS001-10329	TMEM5	-			
1184	79.23	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
1185	79.22	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
1186	79.22	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
1187	79.16	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
1188	79.15	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
1189	79.04	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
1190	79.01	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
1191	79	kd	CGS001-6757	SSX2	-			
1192	78.99	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
1193	78.98	kd	CGS001-84647	PLA2G12B	-			
1194	78.97	kd	CGS001-29110	TBK1	IKK family			
1195	78.94	kd	CGS001-3690	ITGB3	Integrins			
1196	78.91	kd	CGS001-10018	BCL2L11	-			
1197	78.86	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
1198	78.82	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
1199	78.78	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
1200	78.76	cc		Leucine rich repeat kinase inhibitor	-			
1201	78.73	kd	CGS001-29105	C16ORF80	-			
1202	78.7	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
1203	78.64	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
1204	78.6	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
1205	78.59	kd	CGS001-5105	PCK1	-			
1206	78.57	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
1207	78.57	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
1208	78.57	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
1209	78.49	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
1210	78.48	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
1211	78.48	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
1212	78.47	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
1213	78.45	kd	CGS001-2159	F10	Chymotrypsin			
1214	78.42	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1215	78.4	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
1216	78.34	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
1217	78.26	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1218	78.22	kd	CGS001-9412	MED21	-			
1219	78.21	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
1220	78.17	kd	CGS001-9374	PPT2	-			
1221	78.16	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
1222	78.08	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
1223	78.07	kd	CGS001-3664	IRF6	-			
1224	78.02	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
1225	78.01	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
1226	77.99	oe	ccsbBroad304_01271	PPT1	-			
1227	77.99	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
1228	77.97	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
1229	77.92	oe	ccsbBroad304_03853	LSM2	-			
1230	77.82	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
1231	77.79	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
1232	77.74	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
1233	77.74	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1234	77.74	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1235	77.73	oe	ccsbBroad304_00250	CD19	CD molecules			
1236	77.69	cc		Estrogen receptor agonist	-			
1237	77.69	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
1238	77.67	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
1239	77.65	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
1240	77.61	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
1241	77.61	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
1242	77.6	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
1243	77.57	oe	ccsbBroad304_00661	GNGT2	-			
1244	77.57	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
1245	77.49	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
1246	77.47	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
1247	77.47	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
1248	77.46	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
1249	77.44	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
1250	77.36	oe	ccsbBroad304_00836	IGF2	-			
1251	77.32	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
1252	77.18	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
1253	77.16	kd	CGS001-170463	SSBP4	-			
1254	77.12	kd	CGS001-51128	SAR1B	-			
1255	77.02	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
1256	76.99	oe	ccsbBroad304_01841	BAG6	-			
1257	76.98	kd	CGS001-3035	HARS	Aminoacyl tRNA synthetases / Class II			
1258	76.97	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
1259	76.93	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
1260	76.79	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
1261	76.79	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
1262	76.75	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
1263	76.74	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
1264	76.69	kd	CGS001-23678	SGK3	SGK family			
1265	76.68	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
1266	76.68	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
1267	76.67	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
1268	76.67	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
1269	76.63	kd	CGS001-2113	ETS1	ETS Transcription Factors			
1270	76.61	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
1271	76.57	kd	CGS001-1128	CHRM1	Cholinergic receptors			
1272	76.56	kd	CGS001-9318	COPS2	-			
1273	76.55	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
1274	76.54	oe	ccsbBroad304_06048	CRYZ	-			
1275	76.47	kd	CGS001-8864	PER2	-			
1276	76.41	oe	ccsbBroad304_02057	P4HA2	-			
1277	76.39	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
1278	76.34	oe	ccsbBroad304_00150	BAX	-			
1279	76.27	oe	ccsbBroad304_05985	CFL1	-			
1280	76.26	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1281	76.26	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
1282	76.26	kd	CGS001-161725	OTUD7A	OTU domain containing			
1283	76.26	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
1284	76.24	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
1285	76.24	kd	CGS001-10325	RRAGB	-			
1286	76.24	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
1287	76.16	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
1288	76.14	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
1289	76.13	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
1290	76.12	kd	CGS001-7157	TP53	-			
1291	76.05	kd	CGS001-7295	TXN	-			
1292	76.05	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
1293	75.98	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
1294	75.98	kd	CGS001-5575	PRKAR1B	Protein kinase A			
1295	75.97	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
1296	75.9	oe	ccsbBroad304_08536	PARL	-			
1297	75.8	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
1298	75.75	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
1299	75.73	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
1300	75.73	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
1301	75.72	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1302	75.62	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
1303	75.6	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
1304	75.59	kd	CGS001-51734	SEPX1	-			
1305	75.55	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
1306	75.53	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
1307	75.51	oe	ccsbBroad304_07834	GGA2	-			
1308	75.48	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
1309	75.48	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
1310	75.48	kd	CGS001-9767	PHF16	-			
1311	75.47	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
1312	75.42	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
1313	75.37	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
1314	75.24	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
1315	75.24	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1316	75.24	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
1317	75.23	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
1318	75.17	kd	CGS001-64781	CERK	Ceramide kinase			
1319	75.16	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
1320	75.16	kd	CGS001-6223	RPS19	S ribosomal proteins			
1321	75.16	kd	CGS001-8431	NR0B2	DAX-like receptors			
1322	75.06	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
1323	75.05	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
1324	75.02	cp	BRD-K34508425	KUC103898N	-666			-666
1325	75.01	kd	CGS001-10465	PPIH	-			
1326	74.94	oe	ccsbBroad304_00880	IRF2	-			
1327	74.94	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
1328	74.93	kd	CGS001-8692	HYAL2	-			
1329	74.91	kd	CGS001-1951	CELSR3	Cadherins / Major cadherins			
1330	74.88	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
1331	74.83	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
1332	74.8	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
1333	74.72	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
1334	74.71	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
1335	74.55	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
1336	74.55	kd	CGS001-2773	GNAI3	-			
1337	74.49	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
1338	74.45	kd	CGS001-8985	PLOD3	-			
1339	74.43	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
1340	74.4	kd	CGS001-3925	STMN1	-			
1341	74.39	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
1342	74.34	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
1343	74.34	kd	CGS001-116519	APOA5	Apolipoproteins			
1344	74.31	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
1345	74.28	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
1346	74.28	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
1347	74.27	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
1348	74.23	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
1349	74.22	kd	CGS001-4299	AFF1	-			
1350	74.15	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
1351	74.12	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
1352	74.12	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
1353	74.11	oe	ccsbBroad304_02708	TRIM32	-			
1354	74.1	kd	CGS001-4048	LTA4H	Hydrolases			
1355	73.91	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
1356	73.9	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
1357	73.88	oe	ccsbBroad304_00392	CTLA4	CD molecules			
1358	73.78	oe	ccsbBroad304_00100	RHOA	-			
1359	73.76	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
1360	73.7	kd	CGS001-3066	HDAC2	Histone deacetylases			
1361	73.67	oe	ccsbBroad304_00819	IDH3B	-			
1362	73.67	kd	CGS001-23636	NUP62	-			
1363	73.6	kd	CGS001-813	CALU	EF-hand domain containing			
1364	73.57	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
1365	73.55	kd	CGS001-3995	FADS3	Fatty acid desaturases			
1366	73.52	cc		Ubiquitin-specific peptidases LOF	-			
1367	73.47	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
1368	73.47	kd	CGS001-4947	OAZ2	-			
1369	73.33	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
1370	73.22	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1371	73.14	kd	CGS001-835	CASP2	Caspases			
1372	73.13	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
1373	73.11	kd	CGS001-24140	FTSJ1	-			
1374	73.08	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
1375	72.93	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
1376	72.91	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
1377	72.89	kd	CGS001-481	ATP1B1	ATPases / P-type			
1378	72.84	kd	CGS001-27034	ACAD8	-			
1379	72.82	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1380	72.77	kd	CGS001-1837	DTNA	-			
1381	72.71	kd	CGS001-661	POLR3D	RNA polymerase subunits			
1382	72.58	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
1383	72.57	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
1384	72.53	oe	ccsbBroad304_14047	TACC3	-			
1385	72.52	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
1386	72.49	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
1387	72.44	oe	ccsbBroad304_00552	FEN1	-			
1388	72.37	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
1389	72.34	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
1390	72.31	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
1391	72.31	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
1392	72.28	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
1393	72.26	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
1394	72.26	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
1395	72.25	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
1396	72.24	oe	ccsbBroad304_07548	TSSC4	-			
1397	72.22	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
1398	72.13	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
1399	72.05	kd	CGS001-7292	TNFSF4	CD molecules			
1400	71.98	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
1401	71.93	kd	CGS001-64943	NT5DC2	-			
1402	71.86	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
1403	71.85	oe	ccsbBroad304_02133	CD83	CD molecules			
1404	71.75	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
1405	71.73	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
1406	71.59	oe	ccsbBroad304_06287	GM2A	-			
1407	71.55	kd	CGS001-4190	MDH1	-			
1408	71.51	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1409	71.44	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
1410	71.44	kd	CGS001-6727	SRP14	-			
1411	71.42	oe	ccsbBroad304_00120	ATOX1	-			
1412	71.34	cc		DNA synthesis inhibitor	-			
1413	71.31	kd	CGS001-30836	DNTTIP2	-			
1414	71.29	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
1415	71.28	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
1416	71.24	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
1417	71.22	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
1418	71.17	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
1419	71.16	kd	CGS001-5906	RAP1A	-			
1420	71.15	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
1421	71.11	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
1422	71.08	oe	ccsbBroad304_03859	ENOPH1	-			
1423	71.07	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1424	71	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
1425	70.96	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
1426	70.94	kd	CGS001-2184	FAH	-			
1427	70.92	oe	ccsbBroad304_01661	TFCP2	-			
1428	70.92	kd	CGS001-83448	PUS7L	-			
1429	70.91	kd	CGS001-1362	CPD	Carboxypeptidase A			
1430	70.9	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
1431	70.87	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
1432	70.85	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
1433	70.85	kd	CGS001-51070	NOSIP	-			
1434	70.84	kd	CGS001-6210	RPS15A	S ribosomal proteins			
1435	70.81	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
1436	70.73	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
1437	70.6	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
1438	70.55	oe	ccsbBroad304_02361	MFSD10	-			
1439	70.5	oe	ccsbBroad304_00549	FDX1	-			
1440	70.48	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
1441	70.42	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
1442	70.38	oe	ccsbBroad304_00818	IDH3A	-			
1443	70.31	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
1444	70.29	kd	CGS001-3155	HMGCL	-			
1445	70.28	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
1446	70.27	oe	ccsbBroad304_03878	SENP2	-			
1447	70.13	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
1448	70.13	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1449	70.1	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
1450	70.09	oe	ccsbBroad304_02425	CDIPT	-			
1451	70.04	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
1452	69.99	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
1453	69.92	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
1454	69.86	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
1455	69.85	kd	CGS001-801	CALM1	EF-hand domain containing			
1456	69.84	kd	CGS001-7917	BAG6	-			
1457	69.82	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
1458	69.79	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
1459	69.74	kd	CGS001-3998	LMAN1	-			
1460	69.7	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
1461	69.67	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
1462	69.67	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
1463	69.66	kd	CGS001-6598	SMARCB1	-			
1464	69.58	kd	CGS001-8914	TIMELESS	-			
1465	69.57	oe	ccsbBroad304_06855	RDX	-			
1466	69.55	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
1467	69.5	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
1468	69.48	kd	CGS001-8220	DGCR14	-			
1469	69.47	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
1470	69.47	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
1471	69.45	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1472	69.42	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
1473	69.42	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
1474	69.42	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
1475	69.41	oe	ccsbBroad304_06711	PFAS	-			
1476	69.4	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
1477	69.28	kd	CGS001-6282	S100A11	EF-hand domain containing			
1478	69.28	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
1479	69.27	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
1480	69.17	oe	ccsbBroad304_03641	ASF1B	-			
1481	69.17	kd	CGS001-23344	ESYT1	Synaptotagmins			
1482	69.15	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
1483	69.1	kd	CGS001-7374	UNG	-			
1484	69.03	cc		Aromatase inhibitor	-			
1485	68.99	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
1486	68.96	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1487	68.95	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
1488	68.92	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
1489	68.86	kd	CGS001-185	AGTR1	Angiotensin receptors			
1490	68.85	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
1491	68.85	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
1492	68.84	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1493	68.82	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1494	68.8	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
1495	68.73	oe	ccsbBroad304_00418	CD55	CD molecules			
1496	68.69	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
1497	68.68	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
1498	68.64	oe	ccsbBroad304_03933	CARD9	-			
1499	68.62	kd	CGS001-10390	CEPT1	-			
1500	68.41	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
1501	68.38	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
1502	68.31	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
1503	68.3	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
1504	68.3	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
1505	68.28	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
1506	68.21	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
1507	68.15	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1508	67.99	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
1509	67.98	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
1510	67.97	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
1511	67.96	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
1512	67.96	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
1513	67.93	kd	CGS001-11164	NUDT5	Nudix motif containing			
1514	67.92	kd	CGS001-397	ARHGDIB	Endogenous ligands			
1515	67.89	kd	CGS001-7029	TFDP2	-			
1516	67.89	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
1517	67.88	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
1518	67.87	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
1519	67.87	kd	CGS001-103	ADAR	-			
1520	67.86	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
1521	67.85	oe	ccsbBroad304_00155	CCND1	-			
1522	67.81	oe	ccsbBroad304_02110	VAPB	-			
1523	67.8	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
1524	67.76	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
1525	67.75	oe	ccsbBroad304_14174	CDKAL1	-			
1526	67.74	oe	ccsbBroad304_03910	CCDC90A	-			
1527	67.7	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
1528	67.69	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
1529	67.63	kd	CGS001-6714	SRC	Src family			
1530	67.58	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
1531	67.55	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
1532	67.52	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
1533	67.52	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
1534	67.49	kd	CGS001-348	APOE	Apolipoproteins			
1535	67.47	oe	ccsbBroad304_07478	CCP110	-			
1536	67.43	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
1537	67.4	kd	CGS001-7298	TYMS	Methyltransferases			
1538	67.37	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
1539	67.37	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
1540	67.28	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
1541	67.26	cc		Potassium channel blocker	-			
1542	67.25	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
1543	67.21	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
1544	67.19	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
1545	67.17	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1546	67.14	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
1547	67.04	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
1548	67.01	oe	ccsbBroad304_03386	SPA17	-			
1549	67.01	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
1550	67.01	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
1551	66.98	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1552	66.97	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
1553	66.93	kd	CGS001-57057	TBX20	T-boxes			
1554	66.86	kd	CGS001-9447	AIM2	-			
1555	66.8	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1556	66.77	kd	CGS001-6732	SRPK1	SRPK family			
1557	66.67	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
1558	66.65	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
1559	66.58	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
1560	66.47	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
1561	66.42	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
1562	66.42	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
1563	66.41	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
1564	66.38	oe	ccsbBroad304_03640	CEP72	-			
1565	66.38	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
1566	66.36	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1567	66.24	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
1568	66.17	kd	CGS001-571	BACH1	BTB/POZ domain containing			
1569	66.15	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
1570	66.13	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
1571	66.07	oe	ccsbBroad304_06745	PNN	-			
1572	66.07	kd	CGS001-7405	UVRAG	-			
1573	65.96	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
1574	65.95	kd	CGS001-57819	LSM2	-			
1575	65.9	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
1576	65.81	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
1577	65.8	kd	CGS001-29763	PACSIN3	-			
1578	65.79	kd	CGS001-9474	ATG5	-			
1579	65.78	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
1580	65.75	kd	CGS001-3418	IDH2	-			
1581	65.73	oe	ccsbBroad304_00471	E2F6	-			
1582	65.72	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
1583	65.69	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
1584	65.69	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
1585	65.67	oe	ccsbBroad304_01933	TEAD2	-			
1586	65.67	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
1587	65.65	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
1588	65.61	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
1589	65.6	kd	CGS001-345	APOC3	Apolipoproteins			
1590	65.59	kd	CGS001-23378	RRP8	-			
1591	65.57	oe	ccsbBroad304_13998	PDXK	-			
1592	65.56	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
1593	65.56	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
1594	65.56	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
1595	65.55	oe	ccsbBroad304_03652	EXOC2	-			
1596	65.54	oe	ccsbBroad304_08825	LHPP	-			
1597	65.51	kd	CGS001-53632	PRKAG3	AMPK subfamily			
1598	65.49	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
1599	65.43	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
1600	65.42	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
1601	65.41	oe	ccsbBroad304_00033	ADSS	-			
1602	65.4	oe	ccsbBroad304_03808	ERGIC1	-			
1603	65.4	kd	CGS001-7525	YES1	Src family			
1604	65.4	kd	CGS001-10400	PEMT	-			
1605	65.38	kd	CGS001-5359	PLSCR1	-			
1606	65.36	kd	CGS001-4303	FOXO4	Forkhead boxes			
1607	65.34	kd	CGS001-4151	MB	-			
1608	65.27	oe	ccsbBroad304_02875	BRP44	-			
1609	65.24	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
1610	65.11	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
1611	65.1	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
1612	64.99	kd	CGS001-7849	PAX8	Paired boxes			
1613	64.99	kd	CGS001-11151	CORO1A	Coronins			
1614	64.97	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
1615	64.93	oe	ccsbBroad304_01164	PDHB	-			
1616	64.92	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1617	64.89	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
1618	64.89	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
1619	64.85	cc		Tumor necrosis factor superfamily LOF	-			
1620	64.77	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
1621	64.76	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
1622	64.75	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
1623	64.7	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
1624	64.69	kd	CGS001-8535	CBX4	-			
1625	64.67	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
1626	64.65	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
1627	64.59	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
1628	64.57	cc		Protein phosphatase catalytic subunits LOF	-			
1629	64.49	oe	ccsbBroad304_05937	CASP7	Caspases			
1630	64.47	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
1631	64.46	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
1632	64.41	kd	CGS001-337867	UBAC2	-			
1633	64.28	oe	ccsbBroad304_07531	TANK	-			
1634	64.21	cc		C2 domain containing LOF	-			
1635	64.21	oe	ccsbBroad304_02589	COPS5	-			
1636	64.2	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
1637	64.18	kd	CGS001-10007	GNPDA1	-			
1638	64.06	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
1639	64.04	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
1640	64.02	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
1641	63.92	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
1642	63.89	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
1643	63.88	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
1644	63.75	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
1645	63.74	oe	ccsbBroad304_00568	FHL2	-			
1646	63.72	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1647	63.68	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
1648	63.67	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
1649	63.65	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
1650	63.64	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
1651	63.6	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
1652	63.56	oe	ccsbBroad304_01855	NCOA4	-			
1653	63.5	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
1654	63.38	cc		PI3K Signaling LOF	-			
1655	63.25	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
1656	63.22	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
1657	63.21	cc		Toll like receptors LOF	-			
1658	63.11	kd	CGS001-5562	PRKAA1	AMPK subfamily			
1659	63.06	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
1660	63.04	kd	CGS001-5050	PAFAH1B3	-			
1661	63.02	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1662	62.98	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
1663	62.98	oe	ccsbBroad304_00874	INS	-			
1664	62.97	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
1665	62.97	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
1666	62.96	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1667	62.94	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
1668	62.92	kd	CGS001-58472	SQRDL	-			
1669	62.89	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
1670	62.89	kd	CGS001-6829	SUPT5H	-			
1671	62.8	kd	CGS001-3421	IDH3G	-			
1672	62.79	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
1673	62.75	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
1674	62.68	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
1675	62.68	kd	CGS001-4194	MDM4	-			
1676	62.66	kd	CGS001-4734	NEDD4	-			
1677	62.62	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
1678	62.58	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
1679	62.57	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1680	62.56	kd	CGS001-8974	P4HA2	-			
1681	62.54	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
1682	62.48	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
1683	62.45	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
1684	62.44	oe	ccsbBroad304_01061	NAB2	-			
1685	62.44	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
1686	62.36	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
1687	62.34	kd	CGS001-3131	HLF	-			
1688	62.31	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
1689	62.25	cc		Na-K-Cl transporter inhibitor	-			
1690	62.2	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
1691	62.13	oe	ccsbBroad304_03573	BRF2	-			
1692	62.12	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
1693	62.04	oe	ccsbBroad304_06349	HAGH	-			
1694	61.96	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
1695	61.93	cc		HRH1 antagonist	-			
1696	61.92	oe	ccsbBroad304_00492	EIF5A	-			
1697	61.77	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
1698	61.74	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
1699	61.74	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
1700	61.68	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
1701	61.67	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
1702	61.64	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
1703	61.61	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
1704	61.54	oe	ccsbBroad304_01148	PCBD1	-			
1705	61.48	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
1706	61.46	kd	CGS001-5037	PEBP1	-			
1707	61.41	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
1708	61.35	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
1709	61.34	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
1710	61.28	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
1711	61.27	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
1712	61.27	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1713	61.21	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
1714	61.2	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
1715	61.11	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
1716	61.05	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
1717	61.03	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
1718	61.02	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
1719	61	oe	ccsbBroad304_01257	PPOX	-			
1720	60.95	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
1721	60.88	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
1722	60.87	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
1723	60.85	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
1724	60.79	kd	CGS001-9500	MAGED1	-			
1725	60.76	kd	CGS001-64080	RBKS	-			
1726	60.64	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
1727	60.58	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
1728	60.5	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
1729	60.43	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
1730	60.37	kd	CGS001-4232	MEST	-			
1731	60.31	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
1732	60.23	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
1733	60.22	oe	ccsbBroad304_02115	PTTG1	-			
1734	60.2	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
1735	60.2	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
1736	60.12	kd	CGS001-8848	TSC22D1	-			
1737	60.09	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1738	60.05	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1739	60.02	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
1740	60	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
1741	59.91	cc		Targets of VEGFR inhibitors GOF	-			
1742	59.9	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1743	59.88	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
1744	59.85	kd	CGS001-2078	ERG	ETS Transcription Factors			
1745	59.82	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
1746	59.8	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
1747	59.66	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
1748	59.65	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
1749	59.57	kd	CGS001-3630	INS	-			
1750	59.55	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
1751	59.51	kd	CGS001-5898	RALA	-			
1752	59.51	kd	CGS001-255738	PCSK9	Subtilisin			
1753	59.47	kd	CGS001-2295	FOXF2	Forkhead boxes			
1754	59.42	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
1755	59.41	oe	ccsbBroad304_00658	GNG5	-			
1756	59.4	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
1757	59.35	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
1758	59.34	oe	ccsbBroad304_03415	GFOD1	-			
1759	59.34	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
1760	59.33	oe	ccsbBroad304_04194	ELL3	-			
1761	59.32	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
1762	59.3	kd	CGS001-51071	DERA	-			
1763	59.22	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
1764	59.19	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
1765	59.19	kd	CGS001-55206	SBNO1	-			
1766	59.16	kd	CGS001-1026	CDKN1A	-			
1767	59.05	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
1768	59.03	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
1769	59.01	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
1770	58.97	kd	CGS001-5624	PROC	Endogenous ligands			
1771	58.96	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
1772	58.94	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
1773	58.94	oe	ccsbBroad304_05135	PARP15	-			
1774	58.9	kd	CGS001-79600	TCTN1	Tectonic proteins			
1775	58.88	oe	ccsbBroad304_05194	LIPH	-			
1776	58.87	kd	CGS001-317705	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
1777	58.78	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
1778	58.75	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
1779	58.7	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
1780	58.66	oe	ccsbBroad304_06237	GAA	Glycosidases			
1781	58.63	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
1782	58.59	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
1783	58.57	kd	CGS001-2678	GGT1	CD molecules			
1784	58.56	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
1785	58.55	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
1786	58.54	cc		Akt Signaling GOF	-			
1787	58.53	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
1788	58.52	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
1789	58.52	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
1790	58.51	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
1791	58.51	oe	ccsbBroad304_09358	MAPK1IP1L	-			
1792	58.48	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1793	58.38	kd	CGS001-2108	ETFA	-			
1794	58.29	oe	ccsbBroad304_05763	ACTB	-			
1795	58.28	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
1796	58.26	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
1797	58.26	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
1798	58.24	oe	ccsbBroad304_08093	DCPS	-			
1799	58.16	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
1800	58.16	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
1801	58.15	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
1802	58.14	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
1803	58.1	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
1804	58.08	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
1805	58	oe	ccsbBroad304_01930	CUL2	-			
1806	57.91	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
1807	57.84	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
1808	57.83	oe	ccsbBroad304_13891	LCK	Src family			
1809	57.82	oe	ccsbBroad304_05758	ACADSB	-			
1810	57.82	kd	CGS001-2524	FUT2	Fucosyltransferases			
1811	57.81	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
1812	57.8	kd	CGS001-55968	NSFL1C	UBX domain containing			
1813	57.79	kd	CGS001-6601	SMARCC2	-			
1814	57.78	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
1815	57.77	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
1816	57.72	kd	CGS001-818	CAMK2G	CAMK2 family			
1817	57.66	kd	CGS001-169841	ZNF169	Zinc fingers, C2H2-type			
1818	57.63	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
1819	57.63	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
1820	57.6	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1821	57.54	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
1822	57.4	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
1823	57.34	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
1824	57.29	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
1825	57.17	kd	CGS001-2242	FES	Fer family			
1826	57.15	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
1827	57.13	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
1828	57.11	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
1829	57.08	oe	ccsbBroad304_06292	GNAI2	-			
1830	57.06	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
1831	57.05	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
1832	56.99	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
1833	56.96	cc		TGF beta receptor inhibitor	-			
1834	56.96	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
1835	56.92	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
1836	56.87	cc		BCL inhibitor	-			
1837	56.82	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
1838	56.81	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
1839	56.77	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
1840	56.76	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
1841	56.72	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
1842	56.71	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
1843	56.71	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1844	56.66	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
1845	56.62	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
1846	56.62	kd	CGS001-9415	FADS2	Fatty acid desaturases			
1847	56.61	kd	CGS001-4173	MCM4	-			
1848	56.59	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
1849	56.56	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
1850	56.55	kd	CGS001-57680	CHD8	-			
1851	56.52	kd	CGS001-10447	FAM3C	-			
1852	56.44	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
1853	56.43	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
1854	56.4	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
1855	56.35	oe	ccsbBroad304_07280	LAMTOR3	-			
1856	56.29	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
1857	56.22	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
1858	56.21	kd	CGS001-578	BAK1	-			
1859	56.2	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
1860	56.17	oe	ccsbBroad304_02306	PQBP1	-			
1861	56.16	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
1862	56.05	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
1863	56.02	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
1864	56.01	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
1865	55.91	kd	CGS001-5236	PGM1	-			
1866	55.83	kd	CGS001-2987	GUK1	-			
1867	55.82	kd	CGS001-1604	CD55	CD molecules			
1868	55.8	oe	ccsbBroad304_04064	PRR15L	-			
1869	55.8	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
1870	55.69	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
1871	55.66	oe	ccsbBroad304_01166	PDK2	PDHK family			
1872	55.65	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
1873	55.63	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
1874	55.58	kd	CGS001-161	AP2A2	-			
1875	55.57	kd	CGS001-8835	SOCS2	SH2 domain containing			
1876	55.56	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
1877	55.54	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
1878	55.52	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
1879	55.47	kd	CGS001-10452	TOMM40	-			
1880	55.45	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
1881	55.44	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
1882	55.39	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
1883	55.39	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1884	55.37	oe	ccsbBroad304_08605	PBK	TOPK family			
1885	55.34	kd	CGS001-1119	CHKA	-			
1886	55.33	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
1887	55.32	kd	CGS001-30	ACAA1	-			
1888	55.29	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
1889	55.28	kd	CGS001-8480	RAE1	WD repeat domain containing			
1890	55.28	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
1891	55.26	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
1892	55.25	oe	ccsbBroad304_02502	GNA13	-			
1893	55.24	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
1894	55.23	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
1895	55.23	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
1896	55.22	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
1897	55.2	kd	CGS001-663	BNIP2	-			
1898	55.17	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1899	55.13	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
1900	55.1	kd	CGS001-32	ACACB	Carboxylases			
1901	55.02	oe	ccsbBroad304_00237	CCND3	-			
1902	54.95	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
1903	54.91	kd	CGS001-5062	PAK2	PAKA subfamily			
1904	54.9	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
1905	54.8	cc		Sodium channel blocker	-			
1906	54.8	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
1907	54.79	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
1908	54.78	oe	ccsbBroad304_00509	EPHX1	-			
1909	54.77	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
1910	54.76	oe	ccsbBroad304_10431	HADHB	-			
1911	54.76	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
1912	54.73	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
1913	54.7	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
1914	54.7	kd	CGS001-9124	PDLIM1	-			
1915	54.66	oe	ccsbBroad304_02862	CCRN4L	-			
1916	54.63	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
1917	54.48	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
1918	54.45	oe	ccsbBroad304_06574	MDH2	-			
1919	54.37	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
1920	54.36	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
1921	54.36	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
1922	54.34	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
1923	54.34	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
1924	54.29	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
1925	54.29	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
1926	54.22	oe	ccsbBroad304_00424	DBI	-			
1927	54.21	kd	CGS001-7083	TK1	-			
1928	54.19	kd	CGS001-55111	PLEKHJ1	Pleckstrin homology (PH) domain containing			
1929	54.16	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
1930	54.14	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
1931	54.1	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
1932	54.08	kd	CGS001-4837	NNMT	-			
1933	54.07	kd	CGS001-116832	RPL39L	L ribosomal proteins			
1934	54.07	kd	CGS001-3978	LIG1	-			
1935	54.01	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
1936	53.97	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
1937	53.97	kd	CGS001-5164	PDK2	PDHK family			
1938	53.96	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
1939	53.89	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
1940	53.87	oe	ccsbBroad304_03428	EXOSC4	-			
1941	53.86	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
1942	53.85	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
1943	53.84	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
1944	53.84	kd	CGS001-4088	SMAD3	SMADs			
1945	53.83	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
1946	53.83	kd	CGS001-1840	DTX1	-			
1947	53.81	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
1948	53.75	oe	ccsbBroad304_00832	IFNB1	Interferons			
1949	53.74	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
1950	53.7	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
1951	53.69	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
1952	53.68	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
1953	53.68	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
1954	53.62	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
1955	53.61	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
1956	53.53	oe	ccsbBroad304_06435	RBPJ	-			
1957	53.48	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
1958	53.47	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
1959	53.45	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
1960	53.45	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
1961	53.43	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
1962	53.42	kd	CGS001-5373	PMM2	-			
1963	53.41	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
1964	53.37	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
1965	53.32	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
1966	53.3	kd	CGS001-9443	MED7	-			
1967	53.28	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
1968	53.27	oe	ccsbBroad304_03372	CAB39	-			
1969	53.23	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
1970	53.22	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
1971	53.22	kd	CGS001-593	BCKDHA	-			
1972	53.21	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
1973	53.2	oe	ccsbBroad304_01143	PAFAH1B3	-			
1974	53.17	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
1975	53.16	oe	ccsbBroad304_01624	SUPV3L1	-			
1976	53.16	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
1977	53.14	kd	CGS001-1727	CYB5R3	-			
1978	53.13	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1979	53.04	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
1980	53.01	kd	CGS001-1869	E2F1	-			
1981	52.98	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
1982	52.97	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
1983	52.95	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
1984	52.94	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
1985	52.93	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
1986	52.92	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
1987	52.89	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
1988	52.87	oe	ccsbBroad304_02239	RASSF2	-			
1989	52.86	oe	ccsbBroad304_09881	RFX6	-			
1990	52.86	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
1991	52.83	oe	ccsbBroad304_00397	CTSK	Cathepsins			
1992	52.8	kd	CGS001-55802	DCP1A	-			
1993	52.78	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
1994	52.76	kd	CGS001-3479	IGF1	Endogenous ligands			
1995	52.74	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
1996	52.74	kd	CGS001-2523	FUT1	Fucosyltransferases			
1997	52.71	kd	CGS001-81848	SPRY4	-			
1998	52.68	oe	ccsbBroad304_01373	RAN	-			
1999	52.61	oe	ccsbBroad304_03565	ADI1	-			
2000	52.61	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
2001	52.52	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2002	52.4	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
2003	52.4	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
2004	52.32	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
2005	52.32	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
2006	52.26	kd	CGS001-83440	ADPGK	-			
2007	52.26	oe	ccsbBroad304_06172	EPS8	-			
2008	52.25	oe	ccsbBroad304_04675	ATG4A	-			
2009	52.24	oe	ccsbBroad304_02756	RRP8	-			
2010	52.24	kd	CGS001-1212	CLTB	-			
2011	52.22	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
2012	52.13	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
2013	52.12	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
2014	52.11	oe	ccsbBroad304_01699	TPD52L2	-			
2015	52.1	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
2016	52.09	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
2017	52.07	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
2018	52	kd	CGS001-10475	TRIM38	-			
2019	52	kd	CGS001-3682	ITGAE	Integrins			
2020	51.9	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
2021	51.89	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
2022	51.89	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
2023	51.82	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
2024	51.82	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
2025	51.8	cc		KCNJ11 modulator	-			
2026	51.74	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
2027	51.73	kd	CGS001-1440	CSF3	Endogenous ligands			
2028	51.7	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
2029	51.66	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
2030	51.65	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
2031	51.65	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
2032	51.62	oe	ccsbBroad304_00006	ACADM	-			
2033	51.51	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
2034	51.5	oe	ccsbBroad304_02922	TES	-			
2035	51.49	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
2036	51.49	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
2037	51.48	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
2038	51.4	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
2039	51.36	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
2040	51.35	kd	CGS001-2115	ETV1	ETS Transcription Factors			
2041	51.28	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
2042	51.27	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
2043	51.26	kd	CGS001-23658	LSM5	-			
2044	51.14	oe	ccsbBroad304_02432	IFI30	-			
2045	51.11	kd	CGS001-84617	TUBB6	Tubulins			
2046	51.11	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
2047	51.04	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
2048	50.95	oe	ccsbBroad304_08339	CMPK1	-			
2049	50.91	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
2050	50.87	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
2051	50.8	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
2052	50.77	oe	ccsbBroad304_07252	DGKZ	-			
2053	50.77	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
2054	50.71	oe	ccsbBroad304_02026	NRP1	CD molecules			
2055	50.69	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
2056	50.68	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
2057	50.6	kd	CGS001-10617	STAMBP	-			
2058	50.6	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
2059	50.6	kd	CGS001-2896	GRN	-			
2060	50.58	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
2061	50.58	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
2062	50.55	kd	CGS001-10398	MYL9	EF-hand domain containing			
2063	50.47	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
2064	50.47	kd	CGS001-8802	SUCLG1	-			
2065	50.43	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
2066	50.41	oe	ccsbBroad304_08452	PIH1D1	-			
2067	50.3	kd	CGS001-54899	PXK	Slob family			
2068	50.29	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
2069	50.29	kd	CGS001-901	CCNG2	-			
2070	50.26	oe	ccsbBroad304_09615	LACC1	-			
2071	50.26	oe	ccsbBroad304_06420	ICAM3	CD molecules			
2072	50.22	oe	ccsbBroad304_00738	HINT1	-			
2073	50.21	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
2074	50.19	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
2075	50.15	oe	ccsbBroad304_00933	LDHB	-			
2076	50.15	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
2077	50.13	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
2078	50.13	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
2079	50.09	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
2080	50.07	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
2081	50.04	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
2082	50	kd	CGS001-6469	SHH	-			
2083	49.99	cc		Serine proteases GOF	-			
2084	49.98	oe	ccsbBroad304_01205	PIN1	-			
2085	49.96	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
2086	49.94	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
2087	49.88	oe	ccsbBroad304_06462	ITGAE	Integrins			
2088	49.88	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
2089	49.86	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
2090	49.81	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
2091	49.79	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
2092	49.77	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
2093	49.73	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
2094	49.7	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
2095	49.69	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
2096	49.62	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
2097	49.58	kd	CGS001-5831	PYCR1	-			
2098	49.55	kd	CGS001-5579	PRKCB	Alpha subfamily			
2099	49.54	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
2100	49.52	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
2101	49.49	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
2102	49.48	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
2103	49.4	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
2104	49.39	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
2105	49.39	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
2106	49.39	kd	CGS001-64094	SMOC2	EF-hand domain containing			
2107	49.38	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
2108	49.36	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
2109	49.32	kd	CGS001-29978	UBQLN2	Ubiquilin family			
2110	49.3	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
2111	49.28	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2112	49.23	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
2113	49.22	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
2114	49.2	kd	CGS001-6117	RPA1	-			
2115	49.16	kd	CGS001-823	CAPN1	EF-hand domain containing			
2116	49.15	oe	ccsbBroad304_09195	MCM8	-			
2117	49.14	oe	ccsbBroad304_03080	C16ORF80	-			
2118	49.1	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
2119	49.09	kd	CGS001-10476	ATP5H	ATPases / F-type			
2120	49.02	oe	ccsbBroad304_06226	FTL	-			
2121	48.98	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
2122	48.98	kd	CGS001-4300	MLLT3	-			
2123	48.98	kd	CGS001-1962	EHHADH	-			
2124	48.94	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
2125	48.86	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2126	48.84	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
2127	48.83	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
2128	48.83	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2129	48.82	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
2130	48.79	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
2131	48.74	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
2132	48.73	kd	CGS001-93185	IGSF8	CD molecules			
2133	48.72	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
2134	48.71	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2135	48.67	oe	ccsbBroad304_07017	SUOX	-			
2136	48.62	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
2137	48.6	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2138	48.59	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
2139	48.57	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
2140	48.56	oe	ccsbBroad304_02368	TIMM17B	-			
2141	48.51	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
2142	48.4	kd	CGS001-58528	RRAGD	-			
2143	48.38	oe	ccsbBroad304_12008	NLK	nmo subfamily			
2144	48.36	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
2145	48.34	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
2146	48.29	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
2147	48.28	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
2148	48.27	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
2149	48.19	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
2150	48.18	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
2151	48.15	kd	CGS001-23014	FBXO21	F-boxes / other			
2152	48.11	oe	ccsbBroad304_01105	PNP	-			
2153	48.08	kd	CGS001-5934	RBL2	-			
2154	48.07	kd	CGS001-8453	CUL2	-			
2155	48.06	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
2156	48.03	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
2157	47.99	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
2158	47.95	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
2159	47.93	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
2160	47.92	kd	CGS001-387	RHOA	-			
2161	47.88	oe	ccsbBroad304_00171	BNIP3L	-			
2162	47.82	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
2163	47.8	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
2164	47.78	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
2165	47.69	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
2166	47.66	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
2167	47.62	oe	ccsbBroad304_07511	KIF14	Kinesins			
2168	47.58	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
2169	47.52	kd	CGS001-23464	GCAT	-			
2170	47.5	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
2171	47.5	oe	ccsbBroad304_00231	CBFB	-			
2172	47.48	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
2173	47.47	kd	CGS001-9813	KIAA0494	-			
2174	47.43	kd	CGS001-6009	RHEB	-			
2175	47.41	oe	ccsbBroad304_07102	TSG101	-			
2176	47.3	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
2177	47.29	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
2178	47.28	oe	ccsbBroad304_03739	NRIP3	-			
2179	47.25	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
2180	47.24	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
2181	47.21	oe	ccsbBroad304_01186	PHB	-			
2182	47.17	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
2183	47.17	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
2184	47.12	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
2185	47.1	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
2186	47.09	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
2187	47.06	oe	ccsbBroad304_03773	CIAPIN1	-			
2188	47.02	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
2189	47	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
2190	46.97	oe	ccsbBroad304_14020	SH3BP5	-			
2191	46.92	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
2192	46.92	oe	ccsbBroad304_00652	GNAS	-			
2193	46.83	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
2194	46.8	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2195	46.75	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
2196	46.69	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
2197	46.67	oe	ccsbBroad304_02831	SGK3	SGK family			
2198	46.64	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
2199	46.62	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
2200	46.6	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
2201	46.6	kd	CGS001-2017	CTTN	-			
2202	46.58	kd	CGS001-25966	C2CD2	-			
2203	46.55	oe	ccsbBroad304_00783	HPRT1	-			
2204	46.52	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
2205	46.52	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
2206	46.52	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
2207	46.5	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
2208	46.48	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
2209	46.41	kd	CGS001-3725	JUN	basic leucine zipper proteins			
2210	46.4	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
2211	46.4	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
2212	46.38	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
2213	46.34	cc		Zinc fingers RanBP2 type LOF	-			
2214	46.33	kd	CGS001-253260	RICTOR	-			
2215	46.3	cc		Supressors of cytokine signaling GOF	-			
2216	46.3	kd	CGS001-3659	IRF1	-			
2217	46.28	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2218	46.27	kd	CGS001-4086	SMAD1	SMADs			
2219	46.24	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
2220	46.24	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
2221	46.23	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
2222	46.2	oe	ccsbBroad304_01002	METTL1	-			
2223	46.2	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2224	46.19	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
2225	46.16	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
2226	46.15	oe	ccsbBroad304_00876	INSIG1	-			
2227	46.15	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
2228	46.07	kd	CGS001-6285	S100B	EF-hand domain containing			
2229	46.07	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
2230	46.05	oe	ccsbBroad304_00816	IDE	Pitrilysin			
2231	46.03	oe	ccsbBroad304_02484	PAICS	-			
2232	46.03	kd	CGS001-1950	EGF	-			
2233	45.9	kd	CGS001-9670	IPO13	Importins			
2234	45.89	oe	ccsbBroad304_01923	UXT	-			
2235	45.88	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
2236	45.84	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
2237	45.83	kd	CGS001-3676	ITGA4	Integrins			
2238	45.74	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
2239	45.67	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
2240	45.64	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
2241	45.6	kd	CGS001-51271	UBAP1	-			
2242	45.58	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
2243	45.57	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
2244	45.57	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
2245	45.54	kd	CGS001-4171	MCM2	-			
2246	45.53	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
2247	45.51	kd	CGS001-949	SCARB1	-			
2248	45.45	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
2249	45.43	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2250	45.43	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
2251	45.38	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
2252	45.38	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
2253	45.36	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
2254	45.3	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2255	45.3	oe	ccsbBroad304_06852	RBP4	Lipocalins			
2256	45.3	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
2257	45.3	kd	CGS001-5306	PITPNA	-			
2258	45.3	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
2259	45.27	oe	ccsbBroad304_04788	OVCA2	-			
2260	45.21	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
2261	45.2	oe	ccsbBroad304_04465	RERG	-			
2262	45.15	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
2263	45.09	oe	ccsbBroad304_00423	DAXX	-			
2264	45.07	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
2265	44.99	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
2266	44.98	kd	CGS001-2731	GLDC	-			
2267	44.97	cc		RNA Polymerase Enzymes LOF	-			
2268	44.94	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
2269	44.92	oe	ccsbBroad304_02203	MAD2L1BP	-			
2270	44.9	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
2271	44.87	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
2272	44.87	kd	CGS001-11284	PNKP	-			
2273	44.83	cc		Wnt family LOF	-			
2274	44.8	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2275	44.8	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
2276	44.78	kd	CGS001-23650	TRIM29	-			
2277	44.74	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
2278	44.73	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
2279	44.7	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
2280	44.68	oe	ccsbBroad304_08167	DNTTIP2	-			
2281	44.64	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
2282	44.64	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
2283	44.63	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
2284	44.61	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
2285	44.58	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
2286	44.55	oe	ccsbBroad304_02668	PNKP	-			
2287	44.54	oe	ccsbBroad304_01091	NFIB	-			
2288	44.52	cc		Estrogen receptor antagonist	-			
2289	44.5	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
2290	44.49	kd	CGS001-3456	IFNB1	Interferons			
2291	44.46	oe	ccsbBroad304_02955	MYCBP	-			
2292	44.42	kd	CGS001-7105	TSPAN6	Tetraspanins			
2293	44.41	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
2294	44.37	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
2295	44.37	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
2296	44.31	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
2297	44.29	kd	CGS001-2961	GTF2E2	General transcription factors			
2298	44.24	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
2299	44.21	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
2300	44.13	kd	CGS001-27297	CRCP	-			
2301	44.12	oe	ccsbBroad304_08662	MCCC1	-			
2302	44.08	kd	CGS001-5883	RAD9A	-			
2303	44.01	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
2304	43.99	oe	ccsbBroad304_09708	PNLDC1	-			
2305	43.99	kd	CGS001-55082	ARGLU1	-			
2306	43.97	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
2307	43.93	oe	ccsbBroad304_00614	GAMT	-			
2308	43.91	kd	CGS001-151306	GPBAR1	Bile acid receptor			
2309	43.91	kd	CGS001-58478	ENOPH1	-			
2310	43.9	kd	CGS001-5366	PMAIP1	-			
2311	43.9	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
2312	43.89	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
2313	43.87	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
2314	43.86	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
2315	43.78	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
2316	43.76	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
2317	43.75	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
2318	43.72	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
2319	43.7	oe	ccsbBroad304_04786	CANT1	-			
2320	43.7	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
2321	43.68	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
2322	43.63	oe	ccsbBroad304_07238	STK24	YSK subfamily			
2323	43.62	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
2324	43.56	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
2325	43.55	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
2326	43.54	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
2327	43.52	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
2328	43.35	oe	ccsbBroad304_06870	RNH1	-			
2329	43.3	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
2330	43.3	kd	CGS001-11182	SLC2A6	Solute carriers			
2331	43.23	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
2332	43.18	kd	CGS001-3590	IL11RA	IL-6 receptor family			
2333	43.17	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
2334	43.17	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
2335	43.12	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
2336	43.12	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
2337	43.12	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
2338	43.1	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
2339	43.08	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
2340	43.04	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
2341	43.02	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
2342	42.98	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
2343	42.98	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
2344	42.97	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
2345	42.93	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2346	42.92	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
2347	42.88	oe	ccsbBroad304_03164	MTERFD1	-			
2348	42.86	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
2349	42.86	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
2350	42.85	oe	ccsbBroad304_06562	MAT1A	-			
2351	42.85	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
2352	42.81	oe	ccsbBroad304_00987	MCM3	-			
2353	42.76	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
2354	42.73	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
2355	42.71	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2356	42.61	oe	ccsbBroad304_02553	BLCAP	-			
2357	42.56	oe	ccsbBroad304_03308	YTHDF2	-			
2358	42.51	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
2359	42.5	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
2360	42.49	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
2361	42.49	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
2362	42.48	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2363	42.45	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
2364	42.44	oe	ccsbBroad304_02838	SDF2L1	-			
2365	42.42	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
2366	42.41	oe	ccsbBroad304_04294	ATG10	-			
2367	42.4	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
2368	42.4	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
2369	42.37	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
2370	42.32	kd	CGS001-2037	EPB41L2	-			
2371	42.3	oe	ccsbBroad304_07053	TFPI	-			
2372	42.29	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
2373	42.23	oe	ccsbBroad304_05152	SSBP4	-			
2374	42.23	kd	CGS001-6871	TADA2A	-			
2375	42.22	kd	CGS001-2356	FPGS	-			
2376	42.18	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
2377	42.17	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
2378	42.15	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
2379	42.1	oe	ccsbBroad304_07515	GFPT2	-			
2380	42.09	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
2381	42.06	oe	ccsbBroad304_01962	STK16	NAK family			
2382	42.03	oe	ccsbBroad304_00210	CALR	-			
2383	42.03	kd	CGS001-6050	RNH1	-			
2384	41.99	oe	ccsbBroad304_09281	TPD52L3	-			
2385	41.99	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
2386	41.91	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
2387	41.9	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
2388	41.9	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2389	41.84	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
2390	41.84	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
2391	41.83	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
2392	41.83	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
2393	41.83	kd	CGS001-4287	ATXN3	Ataxins			
2394	41.82	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
2395	41.81	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
2396	41.81	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2397	41.8	kd	CGS001-6461	SHB	SH2 domain containing			
2398	41.78	kd	CGS001-64422	ATG3	-			
2399	41.74	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2400	41.74	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
2401	41.6	kd	CGS001-10657	KHDRBS1	-			
2402	41.58	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
2403	41.55	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
2404	41.55	kd	CGS001-26298	EHF	-			
2405	41.48	oe	ccsbBroad304_02884	POT1	-			
2406	41.46	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
2407	41.43	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
2408	41.43	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
2409	41.42	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
2410	41.41	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
2411	41.35	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
2412	41.35	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
2413	41.25	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
2414	41.22	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
2415	41.19	kd	CGS001-9128	PRPF4	WD repeat domain containing			
2416	41.17	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
2417	41.14	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
2418	41.11	oe	ccsbBroad304_01659	TERF1	-			
2419	41.1	oe	ccsbBroad304_08365	CYCS	-			
2420	41.09	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
2421	41.08	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
2422	41.07	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
2423	41.05	cc		C2 domain containing protein kinases LOF	-			
2424	41.05	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
2425	41.02	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
2426	40.99	cc		IL4 Pathway LOF	-			
2427	40.94	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
2428	40.94	kd	CGS001-4668	NAGA	-			
2429	40.87	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
2430	40.86	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
2431	40.85	kd	CGS001-51655	RASD1	-			
2432	40.85	kd	CGS001-523	ATP6V1A	ATPases / V-type			
2433	40.85	oe	ccsbBroad304_06739	PLOD1	-			
2434	40.84	oe	ccsbBroad304_03173	TMED7	-			
2435	40.84	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
2436	40.82	kd	CGS001-10969	EBNA1BP2	-			
2437	40.81	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
2438	40.81	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
2439	40.81	kd	CGS001-65123	INTS3	-			
2440	40.79	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
2441	40.79	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
2442	40.79	kd	CGS001-9159	PCSK7	Subtilisin			
2443	40.79	kd	CGS001-4267	CD99	CD molecules			
2444	40.77	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
2445	40.75	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
2446	40.71	kd	CGS001-5004	ORM1	Lipocalins			
2447	40.65	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
2448	40.64	kd	CGS001-5053	PAH	Amino acid hydroxylases			
2449	40.62	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
2450	40.6	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
2451	40.58	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
2452	40.57	oe	ccsbBroad304_07808	RAB11FIP2	-			
2453	40.56	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
2454	40.56	kd	CGS001-9797	TATDN2	-			
2455	40.51	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
2456	40.51	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
2457	40.51	kd	CGS001-8678	BECN1	-			
2458	40.43	oe	ccsbBroad304_02501	DCTN6	-			
2459	40.42	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
2460	40.41	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
2461	40.4	kd	CGS001-4846	NOS3	Nitric oxide synthases			
2462	40.34	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
2463	40.29	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
2464	40.28	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
2465	40.26	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
2466	40.25	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2467	40.2	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2468	40.2	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
2469	40.19	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2470	40.16	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
2471	40.13	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
2472	40.04	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
2473	40.01	kd	CGS001-2335	FN1	Endogenous ligands			
2474	39.99	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
2475	39.96	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
2476	39.93	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
2477	39.9	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
2478	39.9	kd	CGS001-93594	WDR67	-			
2479	39.89	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
2480	39.89	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
2481	39.89	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
2482	39.89	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
2483	39.85	oe	ccsbBroad304_02716	NMNAT2	-			
2484	39.83	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
2485	39.83	kd	CGS001-5073	PARN	-			
2486	39.81	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
2487	39.8	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
2488	39.79	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
2489	39.73	kd	CGS001-6832	SUPV3L1	-			
2490	39.7	oe	ccsbBroad304_02367	CALCOCO2	-			
2491	39.68	oe	ccsbBroad304_02857	BAMBI	-			
2492	39.64	oe	ccsbBroad304_00954	LYN	Src family			
2493	39.59	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
2494	39.59	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
2495	39.56	oe	ccsbBroad304_08325	LIPT1	-			
2496	39.55	kd	CGS001-3660	IRF2	-			
2497	39.53	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
2498	39.46	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2499	39.45	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
2500	39.35	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
2501	39.34	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
2502	39.34	kd	CGS001-4836	NMT1	-			
2503	39.31	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
2504	39.31	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
2505	39.31	kd	CGS001-3800	KIF5C	Kinesins			
2506	39.28	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
2507	39.24	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
2508	39.23	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
2509	39.21	kd	CGS001-10810	WASF3	-			
2510	39.2	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
2511	39.17	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
2512	39.13	kd	CGS001-51380	CSAD	-			
2513	39.1	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
2514	39.08	kd	CGS001-545	ATR	ATR subfamily			
2515	39.01	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2516	38.99	oe	ccsbBroad304_00854	IL8	-			
2517	38.97	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
2518	38.97	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
2519	38.93	kd	CGS001-2309	FOXO3	Forkhead boxes			
2520	38.92	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
2521	38.88	oe	ccsbBroad304_05098	MAGEB6	-			
2522	38.78	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
2523	38.76	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
2524	38.75	kd	CGS001-1314	COPA	Endogenous ligands			
2525	38.74	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
2526	38.72	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
2527	38.71	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
2528	38.7	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
2529	38.68	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
2530	38.62	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
2531	38.57	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
2532	38.54	oe	ccsbBroad304_04202	MED28	-			
2533	38.52	oe	ccsbBroad304_02414	IRF9	-			
2534	38.49	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
2535	38.43	kd	CGS001-5198	PFAS	-			
2536	38.4	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
2537	38.4	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
2538	38.4	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
2539	38.39	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
2540	38.35	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
2541	38.34	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
2542	38.32	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
2543	38.29	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
2544	38.27	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
2545	38.22	kd	CGS001-8624	PSMG1	-			
2546	38.2	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
2547	38.19	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
2548	38.19	kd	CGS001-22908	SACM1L	-			
2549	38.14	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
2550	38.12	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
2551	38.12	kd	CGS001-6499	SKIV2L	-			
2552	38.1	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
2553	38.1	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
2554	38.08	kd	CGS001-51727	CMPK1	-			
2555	38.05	kd	CGS001-8435	SOAT2	-			
2556	38.01	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
2557	37.99	oe	ccsbBroad304_06008	AP2M1	-			
2558	37.97	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
2559	37.95	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2560	37.92	oe	ccsbBroad304_02438	FAM3C	-			
2561	37.88	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
2562	37.87	oe	ccsbBroad304_03023	CRCP	-			
2563	37.85	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
2564	37.82	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
2565	37.82	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
2566	37.82	kd	CGS001-54584	GNB1L	WD repeat domain containing			
2567	37.81	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
2568	37.78	oe	ccsbBroad304_03625	HIF1AN	-			
2569	37.72	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
2570	37.7	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
2571	37.69	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
2572	37.68	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
2573	37.61	oe	ccsbBroad304_07362	NMI	-			
2574	37.6	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
2575	37.58	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
2576	37.57	oe	ccsbBroad304_00268	CD81	CD molecules			
2577	37.56	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
2578	37.53	kd	CGS001-3566	IL4R	IL-2 receptor family			
2579	37.51	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
2580	37.47	cc		Vitamin D receptor agonist	-			
2581	37.44	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
2582	37.41	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
2583	37.41	kd	CGS001-3909	LAMA3	Laminins			
2584	37.29	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
2585	37.26	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
2586	37.26	oe	ccsbBroad304_04399	PGBD1	-			
2587	37.25	cc		Akt Signaling LOF	-			
2588	37.21	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
2589	37.19	oe	ccsbBroad304_09954	PTRF	-			
2590	37.17	oe	ccsbBroad304_02834	GABARAPL1	-			
2591	37.15	oe	ccsbBroad304_06324	GPX7	-			
2592	37.15	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
2593	37.12	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
2594	37.11	kd	CGS001-51097	SCCPDH	-			
2595	37.1	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
2596	37.07	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
2597	37.06	oe	ccsbBroad304_02554	TRAFD1	-			
2598	36.95	kd	CGS001-2956	MSH6	-			
2599	36.93	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
2600	36.91	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
2601	36.89	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
2602	36.87	oe	ccsbBroad304_07875	SPECC1L	-			
2603	36.87	kd	CGS001-3161	HMMR	CD molecules			
2604	36.85	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
2605	36.84	oe	ccsbBroad304_07888	CBX6	-			
2606	36.81	cc		BMP Signaling LOF	-			
2607	36.81	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
2608	36.8	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
2609	36.8	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
2610	36.79	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
2611	36.79	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
2612	36.78	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
2613	36.76	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
2614	36.75	kd	CGS001-29940	DSE	-			
2615	36.7	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
2616	36.7	kd	CGS001-6722	SRF	-			
2617	36.68	kd	CGS001-11319	ECD	-			
2618	36.65	kd	CGS001-64750	SMURF2	-			
2619	36.63	oe	ccsbBroad304_04053	DERL1	-			
2620	36.63	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
2621	36.62	kd	CGS001-5982	RFC2	ATPases / AAA-type			
2622	36.54	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
2623	36.51	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
2624	36.46	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
2625	36.46	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
2626	36.46	kd	CGS001-8872	CDC123	-			
2627	36.43	oe	ccsbBroad304_02534	UTP14A	-			
2628	36.41	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
2629	36.4	kd	CGS001-1528	CYB5A	Cytochrome b genes			
2630	36.38	kd	CGS001-3895	KTN1	-			
2631	36.38	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
2632	36.36	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
2633	36.32	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
2634	36.32	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
2635	36.31	kd	CGS001-55176	SEC61A2	-			
2636	36.27	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
2637	36.26	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
2638	36.22	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
2639	36.19	oe	ccsbBroad304_07080	TM7SF2	-			
2640	36.16	kd	CGS001-7099	TLR4	Toll-like receptor family			
2641	36.14	oe	ccsbBroad304_06523	LIG1	-			
2642	36.14	kd	CGS001-861	RUNX1	-			
2643	36.12	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
2644	36.01	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
2645	36	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
2646	35.99	kd	CGS001-55612	FERMT1	Fermitins			
2647	35.98	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2648	35.98	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2649	35.94	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
2650	35.92	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
2651	35.9	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
2652	35.87	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2653	35.86	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
2654	35.86	kd	CGS001-2717	GLA	-			
2655	35.85	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
2656	35.83	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
2657	35.81	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
2658	35.79	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
2659	35.78	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
2660	35.74	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
2661	35.73	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
2662	35.71	kd	CGS001-4830	NME1	-			
2663	35.69	kd	CGS001-4312	MMP1	Matrix metallopeptidase			
2664	35.68	oe	ccsbBroad304_04471	C5ORF62	-			
2665	35.67	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
2666	35.64	kd	CGS001-56922	MCCC1	-			
2667	35.62	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
2668	35.61	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2669	35.56	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
2670	35.56	kd	CGS001-29775	CARD10	-			
2671	35.54	kd	CGS001-694	BTG1	-			
2672	35.52	cc		Sigma receptor antagonist	-			
2673	35.52	oe	ccsbBroad304_02157	MED21	-			
2674	35.47	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
2675	35.43	oe	ccsbBroad304_04655	TRIM9	-			
2676	35.36	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
2677	35.35	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
2678	35.32	oe	ccsbBroad304_02002	RNMT	-			
2679	35.3	kd	CGS001-10298	PAK4	PAKB subfamily			
2680	35.28	oe	ccsbBroad304_07401	TXNL1	-			
2681	35.26	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
2682	35.25	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2683	35.25	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
2684	35.23	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
2685	35.21	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
2686	35.19	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
2687	35.18	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
2688	35.17	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
2689	35.16	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
2690	35.13	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
2691	35.07	kd	CGS001-2057	EPOR	Prolactin receptor family			
2692	35.02	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
2693	35.02	kd	CGS001-133690	CAPSL	EF-hand domain containing			
2694	35.01	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
2695	35	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
2696	34.99	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
2697	34.94	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
2698	34.93	kd	CGS001-56889	TM9SF3	-			
2699	34.88	kd	CGS001-3669	ISG20	-			
2700	34.87	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
2701	34.84	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2702	34.79	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
2703	34.76	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
2704	34.73	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
2705	34.73	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
2706	34.69	oe	ccsbBroad304_02772	ICMT	-			
2707	34.68	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
2708	34.67	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
2709	34.66	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
2710	34.64	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
2711	34.61	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
2712	34.59	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
2713	34.58	oe	ccsbBroad304_00063	AMPD2	-			
2714	34.56	kd	CGS001-727	C5	Endogenous ligands			
2715	34.55	kd	CGS001-56616	DIABLO	-			
2716	34.52	oe	ccsbBroad304_01723	TTK	TTK family			
2717	34.51	kd	CGS001-8525	DGKZ	-			
2718	34.5	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
2719	34.49	oe	ccsbBroad304_03269	CD320	CD molecules			
2720	34.48	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
2721	34.48	kd	CGS001-23077	MYCBP2	-			
2722	34.47	kd	CGS001-11142	PKIG	-			
2723	34.45	kd	CGS001-896	CCND3	-			
2724	34.44	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
2725	34.42	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
2726	34.42	kd	CGS001-114609	TIRAP	-			
2727	34.37	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
2728	34.37	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
2729	34.36	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
2730	34.33	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
2731	34.31	oe	ccsbBroad304_01150	PCCB	Carboxylases			
2732	34.31	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
2733	34.27	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
2734	34.26	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
2735	34.21	kd	CGS001-23743	BHMT2	-			
2736	34.15	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
2737	34.14	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
2738	34.14	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
2739	34.13	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
2740	34.12	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2741	34.12	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
2742	34.12	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
2743	34.09	oe	ccsbBroad304_01146	PARN	-			
2744	34.07	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
2745	34.05	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
2746	34.03	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
2747	34.01	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
2748	34.01	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
2749	34	cc		Interleukin receptors LOF	-			
2750	33.99	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
2751	33.97	kd	CGS001-11168	PSIP1	-			
2752	33.96	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
2753	33.93	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
2754	33.92	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
2755	33.91	kd	CGS001-54623	PAF1	-			
2756	33.9	kd	CGS001-4125	MAN2B1	-			
2757	33.9	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
2758	33.86	oe	ccsbBroad304_03112	NENF	-			
2759	33.8	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
2760	33.79	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
2761	33.79	kd	CGS001-54108	CHRAC1	-			
2762	33.78	kd	CGS001-4436	MSH2	-			
2763	33.77	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
2764	33.76	oe	ccsbBroad304_08775	SQRDL	-			
2765	33.73	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2766	33.71	oe	ccsbBroad304_01485	SC5DL	-			
2767	33.66	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
2768	33.62	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
2769	33.61	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2770	33.6	kd	CGS001-56731	SLC2A4RG	-			
2771	33.58	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
2772	33.55	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
2773	33.54	oe	ccsbBroad304_06136	ECHS1	-			
2774	33.54	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
2775	33.53	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
2776	33.51	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
2777	33.46	oe	ccsbBroad304_00961	SMAD2	SMADs			
2778	33.46	kd	CGS001-79094	CHAC1	-			
2779	33.45	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2780	33.43	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
2781	33.42	kd	CGS001-944	TNFSF8	CD molecules			
2782	33.38	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
2783	33.36	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2784	33.29	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
2785	33.24	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
2786	33.18	oe	ccsbBroad304_04544	RCCD1	-			
2787	33.18	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
2788	33.16	kd	CGS001-5427	POLE2	DNA polymerases			
2789	33.15	oe	ccsbBroad304_00865	ILF2	-			
2790	33.14	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
2791	33.03	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
2792	32.99	kd	CGS001-1611	DAP	-			
2793	32.95	oe	ccsbBroad304_00101	RHOC	-			
2794	32.95	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
2795	32.92	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
2796	32.9	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
2797	32.89	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
2798	32.89	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2799	32.88	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
2800	32.85	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
2801	32.82	kd	CGS001-9788	MTSS1	-			
2802	32.8	oe	ccsbBroad304_02446	TADA3	-			
2803	32.78	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
2804	32.74	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
2805	32.67	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
2806	32.61	oe	ccsbBroad304_02565	RALBP1	-			
2807	32.55	kd	CGS001-10827	FAM114A2	-			
2808	32.47	kd	CGS001-2002	ELK1	ETS Transcription Factors			
2809	32.39	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
2810	32.33	kd	CGS001-4795	NFKBIL1	-			
2811	32.32	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
2812	32.28	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
2813	32.26	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2814	32.25	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2815	32.24	kd	CGS001-7020	TFAP2A	-			
2816	32.17	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2817	32.13	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
2818	32.09	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
2819	32.06	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
2820	32.03	kd	CGS001-122809	SOCS4	SH2 domain containing			
2821	32.02	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2822	31.99	oe	ccsbBroad304_07766	RASSF1	-			
2823	31.97	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
2824	31.9	oe	ccsbBroad304_01754	UCK2	-			
2825	31.9	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
2826	31.87	kd	CGS001-55604	LRRC16A	-			
2827	31.85	oe	ccsbBroad304_03767	TOMM22	-			
2828	31.82	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
2829	31.77	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
2830	31.76	oe	ccsbBroad304_02357	SSX3	-			
2831	31.74	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
2832	31.73	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
2833	31.73	kd	CGS001-353	APRT	-			
2834	31.69	kd	CGS001-1356	CP	-			
2835	31.68	oe	ccsbBroad304_07024	SYK	Syk family			
2836	31.66	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
2837	31.66	kd	CGS001-55191	NADSYN1	-			
2838	31.65	kd	CGS001-4176	MCM7	-			
2839	31.61	oe	ccsbBroad304_00572	FKBP3	-			
2840	31.59	kd	CGS001-10013	HDAC6	Histone deacetylases			
2841	31.56	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
2842	31.55	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2843	31.51	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
2844	31.49	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
2845	31.37	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
2846	31.33	oe	ccsbBroad304_03072	GTPBP8	-			
2847	31.28	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
2848	31.27	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
2849	31.26	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
2850	31.26	oe	ccsbBroad304_06765	PRCC	-			
2851	31.19	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
2852	31.14	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
2853	31.13	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
2854	31.12	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
2855	31.12	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
2856	31.09	kd	CGS001-6118	RPA2	-			
2857	31.06	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
2858	31.04	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2859	31	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
2860	30.99	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2861	30.99	kd	CGS001-351	APP	Endogenous ligands			
2862	30.98	kd	CGS001-4121	MAN1A1	-			
2863	30.96	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
2864	30.94	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
2865	30.9	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
2866	30.85	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
2867	30.83	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
2868	30.8	oe	ccsbBroad304_00986	MCM2	-			
2869	30.78	kd	CGS001-1198	CLK3	CDC-like kinases			
2870	30.76	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
2871	30.68	kd	CGS001-5645	PRSS2	Serine peptidases			
2872	30.68	kd	CGS001-708	C1QBP	-			
2873	30.66	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
2874	30.64	kd	CGS001-7471	WNT1	Endogenous ligands			
2875	30.61	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
2876	30.6	kd	CGS001-26292	MYCBP	-			
2877	30.58	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
2878	30.57	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
2879	30.56	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
2880	30.54	kd	CGS001-94234	FOXQ1	Forkhead boxes			
2881	30.53	oe	ccsbBroad304_03951	NARFL	-			
2882	30.51	oe	ccsbBroad304_00102	RND3	-			
2883	30.51	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
2884	30.49	kd	CGS001-10046	MAMLD1	-			
2885	30.48	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
2886	30.44	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
2887	30.41	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
2888	30.39	oe	ccsbBroad304_00262	CD59	CD molecules			
2889	30.36	kd	CGS001-26993	AKAP8L	-			
2890	30.32	kd	CGS001-644	BLVRA	-			
2891	30.31	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
2892	30.31	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
2893	30.26	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
2894	30.2	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
2895	30.17	oe	ccsbBroad304_05821	ANXA1	Annexins			
2896	30.16	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
2897	30.07	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
2898	30.06	oe	ccsbBroad304_05038	HORMAD2	-			
2899	30.01	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
2900	30	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
2901	29.89	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
2902	29.74	kd	CGS001-7852	CXCR4	Chemokine receptors			
2903	29.73	kd	CGS001-54499	TMCO1	-			
2904	29.72	kd	CGS001-4144	MAT2A	-			
2905	29.7	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
2906	29.67	cc		Apolipoproteins LOF	-			
2907	29.61	kd	CGS001-2152	F3	CD molecules			
2908	29.58	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
2909	29.57	kd	CGS001-9697	TRAM2	-			
2910	29.55	kd	CGS001-23102	TBC1D2B	-			
2911	29.55	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
2912	29.52	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
2913	29.47	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
2914	29.45	kd	CGS001-6196	RPS6KA2	RSK subfamily			
2915	29.42	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
2916	29.36	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
2917	29.36	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
2918	29.35	kd	CGS001-3551	IKBKB	IKK family			
2919	29.35	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
2920	29.33	kd	CGS001-23030	KDM4B	Histone demethylases			
2921	29.31	cc		Topoisomerase inhibitor	-			
2922	29.3	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
2923	29.28	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
2924	29.23	kd	CGS001-257397	TAB3	-			
2925	29.2	oe	ccsbBroad304_06174	ERCC1	-			
2926	29.18	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
2927	29.08	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
2928	29.03	kd	CGS001-7251	TSG101	-			
2929	29.02	kd	CGS001-54407	SLC38A2	System A-like transporters			
2930	29.01	kd	CGS001-57026	PDXP	-			
2931	29.01	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
2932	28.99	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
2933	28.97	oe	ccsbBroad304_00648	GLRX	-			
2934	28.96	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
2935	28.92	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
2936	28.91	oe	ccsbBroad304_09006	RPF1	-			
2937	28.9	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
2938	28.86	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
2939	28.85	oe	ccsbBroad304_07557	NAMPT	-			
2940	28.85	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
2941	28.81	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
2942	28.76	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
2943	28.73	kd	CGS001-57147	SCYL3	-			
2944	28.7	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
2945	28.67	kd	CGS001-6850	SYK	Syk family			
2946	28.67	kd	CGS001-57018	CCNL1	-			
2947	28.65	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
2948	28.63	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2949	28.59	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
2950	28.55	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
2951	28.55	kd	CGS001-11116	FGFR1OP	-			
2952	28.45	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
2953	28.39	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
2954	28.33	kd	CGS001-8634	RTCD1	-			
2955	28.32	oe	ccsbBroad304_07923	LSM5	-			
2956	28.31	oe	ccsbBroad304_03047	BZW2	-			
2957	28.29	kd	CGS001-28511	NKIRAS2	-			
2958	28.24	kd	CGS001-7466	WFS1	-			
2959	28.2	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
2960	28.19	kd	CGS001-22889	KIAA0907	-			
2961	28.18	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
2962	28.11	kd	CGS001-1196	CLK2	CDC-like kinases			
2963	28.1	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
2964	28.1	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
2965	28.1	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
2966	28.1	kd	CGS001-50943	FOXP3	Forkhead boxes			
2967	28.07	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
2968	28.07	kd	CGS001-1154	CISH	SH2 domain containing			
2969	28.06	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
2970	27.97	oe	ccsbBroad304_04038	ELOVL6	-			
2971	27.95	kd	CGS001-9218	VAPA	-			
2972	27.94	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
2973	27.9	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
2974	27.86	kd	CGS001-670	BPHL	-			
2975	27.84	oe	ccsbBroad304_04649	ADC	-			
2976	27.8	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
2977	27.76	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
2978	27.69	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
2979	27.67	kd	CGS001-24148	PRPF6	-			
2980	27.64	kd	CGS001-7477	WNT7B	Endogenous ligands			
2981	27.57	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
2982	27.54	oe	ccsbBroad304_07012	STK3	MST subfamily			
2983	27.51	oe	ccsbBroad304_07320	SQSTM1	-			
2984	27.51	kd	CGS001-283450	C12ORF51	-			
2985	27.48	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
2986	27.46	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
2987	27.44	oe	ccsbBroad304_03311	EVL	-			
2988	27.43	oe	ccsbBroad304_03696	C19ORF10	-			
2989	27.42	oe	ccsbBroad304_04775	NTAN1	-			
2990	27.35	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
2991	27.34	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
2992	27.3	kd	CGS001-91304	C19ORF6	-			
2993	27.24	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
2994	27.1	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
2995	27.05	oe	ccsbBroad304_04616	ORMDL3	-			
2996	26.99	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
2997	26.94	oe	ccsbBroad304_01152	PCNA	-			
2998	26.89	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
2999	26.87	kd	CGS001-57157	PHTF2	-			
3000	26.86	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
3001	26.78	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
3002	26.78	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
3003	26.77	oe	ccsbBroad304_07094	TPMT	-			
3004	26.74	kd	CGS001-388	RHOB	-			
3005	26.73	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
3006	26.73	kd	CGS001-5566	PRKACA	Protein kinase A			
3007	26.67	oe	ccsbBroad304_07827	STK38L	NDR family			
3008	26.62	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
3009	26.58	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
3010	26.57	kd	CGS001-1737	DLAT	-			
3011	26.56	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
3012	26.47	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
3013	26.44	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
3014	26.44	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
3015	26.43	kd	CGS001-9926	LPGAT1	-			
3016	26.32	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
3017	26.28	oe	ccsbBroad304_06663	OAS1	-			
3018	26.26	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3019	26.25	oe	ccsbBroad304_00390	CTGF	-			
3020	26.2	kd	CGS001-255877	BCL6B	BTB/POZ domain containing			
3021	26.14	kd	CGS001-23492	CBX7	-			
3022	26.11	oe	ccsbBroad304_03182	GLOD4	-			
3023	26.03	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
3024	25.96	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
3025	25.91	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
3026	25.89	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
3027	25.89	kd	CGS001-4976	OPA1	-			
3028	25.85	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3029	25.84	kd	CGS001-2592	GALT	-			
3030	25.8	oe	ccsbBroad304_02416	TUBB4B	-			
3031	25.74	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
3032	25.74	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3033	25.67	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
3034	25.61	kd	CGS001-9156	EXO1	-			
3035	25.56	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
3036	25.53	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
3037	25.49	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
3038	25.46	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
3039	25.4	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
3040	25.38	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
3041	25.38	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
3042	25.35	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
3043	25.31	kd	CGS001-634	CEACAM1	CD molecules			
3044	25.26	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
3045	25.21	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
3046	25.09	cc		VEGFR inhibitor	-			
3047	25.09	kd	CGS001-29883	CNOT7	-			
3048	25.06	kd	CGS001-60493	FASTKD5	-			
3049	24.96	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
3050	24.92	oe	ccsbBroad304_02270	FAM20B	-			
3051	24.73	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
3052	24.66	kd	CGS001-53343	NUDT9	Nudix motif containing			
3053	24.64	kd	CGS001-4616	GADD45B	-			
3054	24.64	kd	CGS001-283	ANG	Ribonucleases, RNase A			
3055	24.63	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
3056	24.61	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
3057	24.57	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
3058	24.43	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
3059	24.27	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
3060	24.24	kd	CGS001-63892	THADA	-			
3061	24.21	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
3062	24.1	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
3063	24.06	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
3064	24.04	kd	CGS001-1643	DDB2	WD repeat domain containing			
3065	23.93	kd	CGS001-7504	XK	Blood group antigens			
3066	23.83	kd	CGS001-2588	GALNS	Arylsulfatase family			
3067	23.82	kd	CGS001-1111	CHEK1	CHK1 subfamily			
3068	23.82	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
3069	23.79	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
3070	23.79	kd	CGS001-1429	CRYZ	-			
3071	23.75	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
3072	23.72	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
3073	23.62	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
3074	23.56	oe	ccsbBroad304_03119	C16ORF5	-			
3075	23.54	oe	ccsbBroad304_01372	RALB	-			
3076	23.43	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3077	23.38	oe	ccsbBroad304_06367	HK1	-			
3078	23.38	kd	CGS001-2664	GDI1	-			
3079	23.26	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
3080	23.24	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
3081	23.2	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
3082	23.2	kd	CGS001-23509	POFUT1	Fucosyltransferases			
3083	23.16	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
3084	23.13	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
3085	23.1	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
3086	23.09	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
3087	23.09	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
3088	23	kd	CGS001-8826	IQGAP1	-			
3089	22.98	oe	ccsbBroad304_04257	SPRY4	-			
3090	22.97	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
3091	22.88	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
3092	22.86	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
3093	22.73	kd	CGS001-2161	F12	Chymotrypsin			
3094	22.65	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
3095	22.6	kd	CGS001-4602	MYB	-			
3096	22.6	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
3097	22.47	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
3098	22.44	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
3099	22.39	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
3100	22.34	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
3101	22.2	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
3102	22.17	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
3103	22.17	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
3104	21.75	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
3105	21.73	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
3106	21.49	kd	CGS001-182	JAG1	CD molecules			
3107	21.42	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
3108	21.37	kd	CGS001-10614	HEXIM1	-			
3109	21.34	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3110	21.31	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
3111	21.23	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
3112	21.17	kd	CGS001-10078	TSSC4	-			
3113	21.04	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
3114	20.96	oe	ccsbBroad304_05745	CD24	CD molecules			
3115	20.9	kd	CGS001-54498	SMOX	-			
3116	20.86	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
3117	20.85	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3118	20.8	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
3119	20.76	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3120	20.7	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
3121	20.68	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
3122	20.65	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
3123	20.5	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3124	20.39	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
3125	20.37	cc		GATA Zinc finger domain containing LOF	-			
3126	20.33	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3127	20.31	oe	ccsbBroad304_00966	MAFG	-			
3128	20.18	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3129	20.16	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
3130	20.14	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
3131	20	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
3132	19.98	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
3133	19.97	oe	ccsbBroad304_00239	CCNG1	-			
3134	19.95	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
3135	19.91	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
3136	19.61	kd	CGS001-7057	THBS1	-			
3137	19.58	kd	CGS001-205	AK4	Adenylate kinases			
3138	19.58	kd	CGS001-7187	TRAF3	-			
3139	19.48	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
3140	19.47	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
3141	19.32	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
3142	19.12	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
3143	18.91	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
3144	18.91	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
3145	18.8	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
3146	18.76	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
3147	18.71	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
3148	18.71	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
3149	18.67	kd	CGS001-10198	MPHOSPH9	-			
3150	18.4	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
3151	18.34	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3152	18.2	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3153	18.19	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
3154	18.13	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
3155	17.77	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
3156	17.73	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
3157	17.67	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
3158	17.64	cc		Androgen receptor modulator	-			
3159	17.62	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
3160	17.59	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
3161	17.51	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
3162	17.24	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3163	17.08	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
3164	16.97	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
3165	16.91	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
3166	16.88	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
3167	16.86	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
3168	16.82	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
3169	16.7	kd	CGS001-54957	TXNL4B	-			
3170	16.68	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
3171	16.67	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
3172	16.6	cc		Tubulin inhibitor	-			
3173	16.57	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
3174	16.56	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
3175	16.5	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
3176	16.38	kd	CGS001-5688	PSMA7	Proteasome subunits			
3177	16.24	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
3178	16.09	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
3179	15.92	cc		Progesterone receptor antagonist	-			
3180	15.72	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
3181	15.63	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
3182	15.48	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
3183	15.4	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
3184	15.26	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
3185	15.07	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
3186	14.64	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
3187	14.59	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
3188	14.47	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
3189	14.44	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
3190	14.44	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
3191	14.4	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
3192	14.24	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
3193	13.89	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3194	13.8	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
3195	13.67	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
3196	13.46	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
3197	13.25	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
3198	13.06	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
3199	12.52	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
3200	12.49	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
3201	12.34	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
3202	12.31	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3203	12.27	cc		Mediator complex LOF	-			
3204	11.89	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
3205	11.7	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
3206	11.37	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
3207	11.29	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
3208	11.05	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3209	10.89	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
3210	10.83	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
3211	10.07	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
3212	8.85	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
3213	8.46	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
3214	7.87	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
3215	7.34	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
3216	7.28	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
3217	6.68	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
3218	6.59	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
3219	4.57	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
3220	-5.49	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
3221	-7.51	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
3222	-7.67	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
3223	-8.97	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
3224	-9.14	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3225	-9.21	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3226	-9.32	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
3227	-9.57	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
3228	-9.63	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3229	-9.77	kd	CGS001-2288	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
3230	-10.22	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
3231	-10.63	cc		Cannabinoid receptor agonist	-			
3232	-10.66	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
3233	-10.76	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
3234	-11.29	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
3235	-11.72	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
3236	-11.93	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
3237	-12.05	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
3238	-12.39	cc		Cyclin dependent kinases LOF	-			
3239	-12.5	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
3240	-12.53	oe	ccsbBroad304_02175	MAGED1	-			
3241	-12.74	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
3242	-12.89	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
3243	-13.02	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
3244	-13.29	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
3245	-13.34	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
3246	-13.39	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3247	-13.89	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
3248	-13.96	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
3249	-13.98	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
3250	-14.02	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
3251	-14.16	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
3252	-14.18	kd	CGS001-8743	TNFSF10	CD molecules			
3253	-14.26	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
3254	-14.39	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
3255	-14.4	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
3256	-14.42	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
3257	-14.5	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
3258	-14.58	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
3259	-14.72	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
3260	-14.99	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
3261	-15.03	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
3262	-15.36	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
3263	-15.39	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
3264	-15.4	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
3265	-15.4	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
3266	-15.46	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
3267	-15.54	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
3268	-15.54	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
3269	-15.56	kd	CGS001-2957	GTF2A1	General transcription factors			
3270	-15.58	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
3271	-15.62	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
3272	-15.67	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
3273	-15.75	kd	CGS001-50808	AK3	-			
3274	-15.79	kd	CGS001-84669	USP32	EF-hand domain containing			
3275	-15.94	kd	CGS001-54861	SNRK	SNRK subfamily			
3276	-15.96	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
3277	-15.98	oe	ccsbBroad304_01483	SAT1	-			
3278	-16.07	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
3279	-16.08	kd	CGS001-7965	AIMP2	-			
3280	-16.1	cc		HOXL subclass homeoboxes LOF	-			
3281	-16.11	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3282	-16.23	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
3283	-16.24	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
3284	-16.35	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
3285	-16.37	kd	CGS001-375449	MAST4	MAST family			
3286	-16.6	cp	BRD-K15842202	eudesmic-acid	-666			-666
3287	-16.64	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
3288	-16.84	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
3289	-16.95	kd	CGS001-6622	SNCA	Parkinson disease			
3290	-17	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
3291	-17.01	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
3292	-17.03	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
3293	-17.04	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
3294	-17.08	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
3295	-17.08	kd	CGS001-144811	LACC1	-			
3296	-17.12	cc		Interleukins GOF	-			
3297	-17.47	oe	ccsbBroad304_02579	YWHAQ	-			
3298	-17.52	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3299	-17.54	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
3300	-17.54	kd	CGS001-6774	STAT3	SH2 domain containing			
3301	-17.56	oe	ccsbBroad304_02497	YKT6	-			
3302	-17.76	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
3303	-18.02	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3304	-18.14	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
3305	-18.27	kd	CGS001-3663	IRF5	-			
3306	-18.32	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
3307	-18.4	oe	ccsbBroad304_04292	INHBE	-			
3308	-18.46	oe	ccsbBroad304_06180	ESD	-			
3309	-18.49	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3310	-18.49	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
3311	-18.57	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
3312	-18.88	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
3313	-18.94	kd	CGS001-1036	CDO1	-			
3314	-19.08	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
3315	-19.08	kd	CGS001-1028	CDKN1C	-			
3316	-19.09	kd	CGS001-10544	PROCR	CD molecules			
3317	-19.1	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
3318	-19.17	oe	ccsbBroad304_02452	NXF1	-			
3319	-19.18	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
3320	-19.18	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
3321	-19.21	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
3322	-19.28	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
3323	-19.33	kd	CGS001-10314	LANCL1	-			
3324	-19.44	kd	CGS001-18	ABAT	GABA turnover			
3325	-19.49	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
3326	-19.54	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
3327	-19.56	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
3328	-19.56	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
3329	-19.6	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
3330	-19.65	kd	CGS001-5338	PLD2	Hydrolases			
3331	-19.68	kd	CGS001-5110	PCMT1	-			
3332	-19.71	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
3333	-19.75	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
3334	-19.76	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
3335	-19.82	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
3336	-19.84	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
3337	-19.86	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
3338	-19.91	cc		Gamma secretase inhibitor	-			
3339	-19.97	oe	ccsbBroad304_01327	PSPH	-			
3340	-20	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
3341	-20.04	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
3342	-20.05	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
3343	-20.05	kd	CGS001-6446	SGK1	SGK family			
3344	-20.13	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
3345	-20.16	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
3346	-20.17	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
3347	-20.17	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
3348	-20.2	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
3349	-20.24	kd	CGS001-790	CAD	-			
3350	-20.24	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
3351	-20.31	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
3352	-20.33	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
3353	-20.33	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
3354	-20.33	kd	CGS001-6611	SMS	-			
3355	-20.36	kd	CGS001-9232	PTTG1	-			
3356	-20.37	kd	CGS001-147179	WIPF2	-			
3357	-20.37	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3358	-20.42	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
3359	-20.5	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
3360	-20.52	kd	CGS001-6201	RPS7	S ribosomal proteins			
3361	-20.59	oe	ccsbBroad304_05907	BUB1B	Bub family			
3362	-20.6	kd	CGS001-3065	HDAC1	Histone deacetylases			
3363	-20.62	kd	CGS001-11344	TWF2	Twinfilin subfamily			
3364	-20.7	kd	CGS001-662	BNIP1	-			
3365	-20.76	kd	CGS001-3608	ILF2	-			
3366	-20.8	kd	CGS001-1948	EFNB2	Ephrins			
3367	-21	kd	CGS001-5962	RDX	-			
3368	-21.02	kd	CGS001-11007	CCDC85B	-			
3369	-21.05	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3370	-21.11	cc		Wnt family GOF	-			
3371	-21.15	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
3372	-21.24	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
3373	-21.29	kd	CGS001-4069	LYZ	-			
3374	-21.36	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
3375	-21.37	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
3376	-21.38	kd	CGS001-2203	FBP1	-			
3377	-21.44	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
3378	-21.47	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
3379	-21.49	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
3380	-21.56	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3381	-21.58	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
3382	-21.58	kd	CGS001-6776	STAT5A	SH2 domain containing			
3383	-21.59	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
3384	-21.62	kd	CGS001-5894	RAF1	RAF family			
3385	-21.63	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
3386	-21.65	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
3387	-21.66	oe	ccsbBroad304_04379	LZIC	-			
3388	-21.74	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
3389	-21.8	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
3390	-21.8	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
3391	-21.83	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
3392	-21.83	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
3393	-21.89	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
3394	-21.9	oe	ccsbBroad304_06178	ERCC5	-			
3395	-21.91	kd	CGS001-2099	ESR1	Estrogen receptors			
3396	-21.96	kd	CGS001-3242	HPD	Oxidoreductases			
3397	-22.02	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
3398	-22.03	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
3399	-22.11	kd	CGS001-84923	FAM104A	-			
3400	-22.11	kd	CGS001-5167	ENPP1	-			
3401	-22.16	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
3402	-22.17	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
3403	-22.2	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
3404	-22.23	kd	CGS001-2877	GPX2	-			
3405	-22.3	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
3406	-22.38	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
3407	-22.39	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3408	-22.44	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
3409	-22.44	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
3410	-22.47	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
3411	-22.53	kd	CGS001-10214	SSX3	-			
3412	-22.59	kd	CGS001-23369	PUM2	-			
3413	-22.62	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
3414	-22.69	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
3415	-22.69	kd	CGS001-399694	SHC4	SH2 domain containing			
3416	-22.7	kd	CGS001-4683	NBN	-			
3417	-22.71	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
3418	-22.72	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
3419	-22.78	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3420	-22.79	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
3421	-22.8	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
3422	-22.81	oe	ccsbBroad304_04534	HN1L	-			
3423	-22.82	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
3424	-22.87	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
3425	-23	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
3426	-23.01	oe	ccsbBroad304_02086	PDLIM1	-			
3427	-23.04	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3428	-23.05	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
3429	-23.06	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
3430	-23.08	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
3431	-23.08	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
3432	-23.12	kd	CGS001-2067	ERCC1	-			
3433	-23.16	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
3434	-23.17	oe	ccsbBroad304_08055	ATP5S	-			
3435	-23.2	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
3436	-23.25	kd	CGS001-10312	TCIRG1	ATPases / V-type			
3437	-23.29	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
3438	-23.29	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3439	-23.32	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
3440	-23.34	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
3441	-23.37	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
3442	-23.38	kd	CGS001-80349	WDR61	WD repeat domain containing			
3443	-23.39	oe	ccsbBroad304_01605	SSX2	-			
3444	-23.39	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
3445	-23.45	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
3446	-23.45	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
3447	-23.46	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
3448	-23.49	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
3449	-23.5	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
3450	-23.52	cc		Vesicular Transport LOF	-			
3451	-23.54	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
3452	-23.58	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
3453	-23.66	kd	CGS001-3420	IDH3B	-			
3454	-23.67	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
3455	-23.69	kd	CGS001-5727	PTCH1	-			
3456	-23.75	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
3457	-23.79	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
3458	-23.85	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
3459	-23.9	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
3460	-23.94	kd	CGS001-5925	RB1	Endogenous ligands			
3461	-23.96	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
3462	-24	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
3463	-24.04	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
3464	-24.06	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
3465	-24.06	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
3466	-24.07	kd	CGS001-27125	AFF4	-			
3467	-24.1	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
3468	-24.12	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
3469	-24.15	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
3470	-24.17	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
3471	-24.19	kd	CGS001-5355	PLP2	-			
3472	-24.2	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
3473	-24.22	oe	ccsbBroad304_07754	FGFR1OP	-			
3474	-24.25	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
3475	-24.26	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3476	-24.29	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
3477	-24.36	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
3478	-24.38	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
3479	-24.39	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
3480	-24.41	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
3481	-24.42	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
3482	-24.43	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
3483	-24.46	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
3484	-24.47	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
3485	-24.49	kd	CGS001-4245	MGAT1	-			
3486	-24.56	kd	CGS001-10755	GIPC1	-			
3487	-24.6	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
3488	-24.62	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
3489	-24.64	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
3490	-24.65	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
3491	-24.65	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
3492	-24.67	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
3493	-24.69	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
3494	-24.7	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
3495	-24.76	oe	ccsbBroad304_01392	TRIM27	-			
3496	-24.78	kd	CGS001-9552	SPAG7	-			
3497	-24.79	kd	CGS001-4833	NME4	-			
3498	-24.8	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
3499	-24.81	oe	ccsbBroad304_01527	SGK1	SGK family			
3500	-24.82	kd	CGS001-83729	INHBE	-			
3501	-24.85	oe	ccsbBroad304_07528	DMTF1	-			
3502	-24.86	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
3503	-24.88	oe	ccsbBroad304_06996	SRM	-			
3504	-24.89	kd	CGS001-1997	ELF1	ETS Transcription Factors			
3505	-24.93	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
3506	-24.94	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
3507	-24.95	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
3508	-25.01	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
3509	-25.02	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
3510	-25.02	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
3511	-25.02	kd	CGS001-2645	GCK	Hexokinases			
3512	-25.03	kd	CGS001-4637	MYL6	EF-hand domain containing			
3513	-25.05	kd	CGS001-7035	TFPI	-			
3514	-25.09	oe	ccsbBroad304_07491	IP6K1	-			
3515	-25.09	kd	CGS001-10247	HRSP12	-			
3516	-25.09	kd	CGS001-8192	CLPP	ATPases / AAA-type			
3517	-25.12	kd	CGS001-8669	EIF3J	-			
3518	-25.15	kd	CGS001-23647	ARFIP2	-			
3519	-25.16	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
3520	-25.17	kd	CGS001-57521	RPTOR	WD repeat domain containing			
3521	-25.17	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
3522	-25.2	kd	CGS001-5621	PRNP	CD molecules			
3523	-25.21	kd	CGS001-8804	CREG1	-			
3524	-25.25	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
3525	-25.25	kd	CGS001-29116	MYLIP	-			
3526	-25.25	oe	ccsbBroad304_05981	CDO1	-			
3527	-25.26	kd	CGS001-10468	FST	-			
3528	-25.27	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
3529	-25.28	kd	CGS001-83593	RASSF5	-			
3530	-25.31	oe	ccsbBroad304_07887	GCAT	-			
3531	-25.33	kd	CGS001-7360	UGP2	-			
3532	-25.34	oe	ccsbBroad304_03934	LEPRE1	-			
3533	-25.4	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
3534	-25.48	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3535	-25.52	kd	CGS001-51805	COQ3	-			
3536	-25.54	kd	CGS001-2072	ERCC4	-			
3537	-25.54	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3538	-25.58	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
3539	-25.59	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
3540	-25.6	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
3541	-25.67	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
3542	-25.7	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
3543	-25.71	oe	ccsbBroad304_00491	EIF4EBP2	-			
3544	-25.71	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
3545	-25.73	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
3546	-25.83	kd	CGS001-4817	NIT1	-			
3547	-25.86	oe	ccsbBroad304_00226	CAV1	-			
3548	-25.87	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3549	-25.89	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
3550	-25.9	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
3551	-25.9	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
3552	-25.91	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
3553	-25.94	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
3554	-25.97	kd	CGS001-1756	DMD	-			
3555	-25.98	oe	ccsbBroad304_13880	IDH3G	-			
3556	-26.01	oe	ccsbBroad304_00098	ARG1	Arginase			
3557	-26.04	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
3558	-26.06	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
3559	-26.06	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
3560	-26.06	kd	CGS001-23621	BACE1	Pepsin			
3561	-26.08	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
3562	-26.11	kd	CGS001-3988	LIPA	-			
3563	-26.18	kd	CGS001-55379	LRRC59	-			
3564	-26.19	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
3565	-26.23	oe	ccsbBroad304_00053	ALDOA	-			
3566	-26.27	oe	ccsbBroad304_02012	FADD	-			
3567	-26.27	kd	CGS001-664	BNIP3	-			
3568	-26.31	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
3569	-26.32	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
3570	-26.33	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
3571	-26.33	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
3572	-26.34	kd	CGS001-6895	TARBP2	-			
3573	-26.39	kd	CGS001-10681	GNB5	WD repeat domain containing			
3574	-26.45	cc		DNA Replication LOF	-			
3575	-26.55	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
3576	-26.57	kd	CGS001-116931	MED12L	-			
3577	-26.64	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
3578	-26.67	oe	ccsbBroad304_09354	IGSF8	CD molecules			
3579	-26.67	kd	CGS001-10253	SPRY2	-			
3580	-26.7	oe	ccsbBroad304_00510	EPHX2	-			
3581	-26.71	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
3582	-26.72	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
3583	-26.74	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
3584	-26.76	kd	CGS001-7296	TXNRD1	-			
3585	-26.79	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
3586	-26.81	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
3587	-26.87	oe	ccsbBroad304_02318	KIF20A	Kinesins			
3588	-26.87	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
3589	-26.88	kd	CGS001-5979	RET	Type XIV RTKs: RET			
3590	-26.89	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
3591	-26.9	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
3592	-26.91	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
3593	-26.93	oe	ccsbBroad304_00115	ASPH	-			
3594	-26.93	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
3595	-26.94	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
3596	-26.95	kd	CGS001-5933	RBL1	-			
3597	-26.95	kd	CGS001-54884	RETSAT	-			
3598	-27.02	kd	CGS001-64428	NARFL	-			
3599	-27.02	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
3600	-27.03	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
3601	-27.05	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
3602	-27.07	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
3603	-27.09	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
3604	-27.1	kd	CGS001-11336	EXOC3	-			
3605	-27.11	oe	ccsbBroad304_03812	PBXIP1	-			
3606	-27.16	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
3607	-27.19	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
3608	-27.19	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
3609	-27.25	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
3610	-27.25	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
3611	-27.26	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
3612	-27.27	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
3613	-27.27	kd	CGS001-55214	LEPREL1	-			
3614	-27.28	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
3615	-27.3	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
3616	-27.33	kd	CGS001-23028	KDM1A	Histone demethylase			
3617	-27.34	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
3618	-27.36	kd	CGS001-5188	PET112	-			
3619	-27.37	kd	CGS001-403	ARL3	ADP-ribosylation factors			
3620	-27.38	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
3621	-27.43	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
3622	-27.43	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
3623	-27.43	kd	CGS001-11200	CHEK2	CHK1 subfamily			
3624	-27.44	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
3625	-27.46	oe	ccsbBroad304_08292	IP6K2	-			
3626	-27.46	kd	CGS001-4439	MSH5	-			
3627	-27.49	kd	CGS001-5106	PCK2	-			
3628	-27.52	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
3629	-27.53	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
3630	-27.57	kd	CGS001-29102	DROSHA	-			
3631	-27.6	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
3632	-27.6	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
3633	-27.62	kd	CGS001-5498	PPOX	-			
3634	-27.65	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
3635	-27.66	cc		FLT3 inhibitor	-			
3636	-27.67	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
3637	-27.68	oe	ccsbBroad304_10846	GGT1	CD molecules			
3638	-27.68	oe	ccsbBroad304_03728	DIABLO	-			
3639	-27.7	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
3640	-27.72	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
3641	-27.75	kd	CGS001-1029	CDKN2A	-			
3642	-27.76	oe	ccsbBroad304_08839	IFIH1	-			
3643	-27.76	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
3644	-27.77	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
3645	-27.78	kd	CGS001-7090	TLE3	WD repeat domain containing			
3646	-27.84	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
3647	-27.85	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
3648	-27.86	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
3649	-27.91	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
3650	-27.94	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
3651	-27.95	oe	ccsbBroad304_06264	GBP2	-			
3652	-27.96	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
3653	-27.99	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
3654	-28.05	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
3655	-28.05	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
3656	-28.09	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
3657	-28.11	kd	CGS001-8313	AXIN2	-			
3658	-28.12	kd	CGS001-25836	NIPBL	-			
3659	-28.19	kd	CGS001-7078	TIMP3	-			
3660	-28.21	kd	CGS001-23131	GPATCH8	G patch domain containing			
3661	-28.22	kd	CGS001-8841	HDAC3	Histone deacetylases			
3662	-28.24	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
3663	-28.24	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
3664	-28.24	kd	CGS001-2077	ERF	ETS Transcription Factors			
3665	-28.26	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
3666	-28.26	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
3667	-28.27	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
3668	-28.29	kd	CGS001-178	AGL	-			
3669	-28.29	kd	CGS001-87	ACTN1	EF-hand domain containing			
3670	-28.3	kd	CGS001-59286	UBL5	-			
3671	-28.32	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
3672	-28.33	oe	ccsbBroad304_07267	PDLIM4	-			
3673	-28.35	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3674	-28.36	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
3675	-28.4	oe	ccsbBroad304_00430	GADD45A	-			
3676	-28.4	kd	CGS001-10972	TMED10	-			
3677	-28.42	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
3678	-28.42	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
3679	-28.43	oe	ccsbBroad304_02229	TRAM2	-			
3680	-28.45	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
3681	-28.46	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
3682	-28.47	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
3683	-28.49	kd	CGS001-427	ASAH1	Acid ceramidase			
3684	-28.5	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
3685	-28.54	kd	CGS001-117154	DACH2	-			
3686	-28.55	kd	CGS001-10497	UNC13B	-			
3687	-28.58	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
3688	-28.58	kd	CGS001-843	CASP10	Caspases			
3689	-28.6	oe	ccsbBroad304_00212	CAMLG	-			
3690	-28.6	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
3691	-28.64	oe	ccsbBroad304_08511	RFK	-			
3692	-28.65	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
3693	-28.66	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
3694	-28.66	kd	CGS001-65243	ZNF643	-			
3695	-28.67	kd	CGS001-1445	CSK	Csk family			
3696	-28.67	kd	CGS001-350	APOH	Apolipoproteins			
3697	-28.68	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
3698	-28.69	kd	CGS001-4087	SMAD2	SMADs			
3699	-28.7	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
3700	-28.73	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3701	-28.74	kd	CGS001-2010	EMD	-			
3702	-28.76	oe	ccsbBroad304_03040	NKIRAS2	-			
3703	-28.78	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
3704	-28.79	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
3705	-28.83	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
3706	-28.85	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
3707	-28.89	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
3708	-28.89	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
3709	-28.97	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
3710	-28.98	kd	CGS001-4179	CD46	CD molecules			
3711	-28.99	oe	ccsbBroad304_06350	HAL	-			
3712	-29.01	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
3713	-29.04	kd	CGS001-5378	PMS1	-			
3714	-29.1	oe	ccsbBroad304_03121	NRBF2	-			
3715	-29.1	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
3716	-29.1	kd	CGS001-26227	PHGDH	-			
3717	-29.11	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
3718	-29.16	kd	CGS001-22794	CASC3	-			
3719	-29.26	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
3720	-29.28	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
3721	-29.29	kd	CGS001-7039	TGFA	-			
3722	-29.3	kd	CGS001-5565	PRKAB2	AMPK subfamily			
3723	-29.3	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3724	-29.31	cc		PDGFR/KIT inhibitor	-			
3725	-29.34	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
3726	-29.38	cc		Bacterial cell wall synthesis inhibitor	-			
3727	-29.38	kd	CGS001-7832	BTG2	-			
3728	-29.45	kd	CGS001-57048	PLSCR3	-			
3729	-29.46	cc		Bacterial 30S ribosomal subunit inhibitor	-			
3730	-29.46	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
3731	-29.48	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
3732	-29.5	kd	CGS001-149428	BNIPL	-			
3733	-29.53	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
3734	-29.54	kd	CGS001-4811	NID1	-			
3735	-29.56	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
3736	-29.58	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
3737	-29.59	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
3738	-29.6	kd	CGS001-6258	RXRG	Retinoid X receptors			
3739	-29.6	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
3740	-29.63	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
3741	-29.65	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
3742	-29.68	kd	CGS001-271	AMPD2	-			
3743	-29.72	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
3744	-29.73	kd	CGS001-10250	SRRM1	-			
3745	-29.73	kd	CGS001-6632	SNRPD1	-			
3746	-29.73	kd	CGS001-1105	CHD1	-			
3747	-29.74	kd	CGS001-22938	SNW1	-			
3748	-29.75	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
3749	-29.78	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3750	-29.8	kd	CGS001-8467	SMARCA5	-			
3751	-29.82	oe	ccsbBroad304_03118	NRBP1	NRBP family			
3752	-29.85	kd	CGS001-23670	TMEM2	-			
3753	-29.86	kd	CGS001-4665	NAB2	-			
3754	-29.88	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
3755	-29.89	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
3756	-29.89	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
3757	-29.9	kd	CGS001-22887	FOXJ3	Forkhead boxes			
3758	-29.92	kd	CGS001-9380	GRHPR	-			
3759	-29.92	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
3760	-29.93	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
3761	-29.94	kd	CGS001-10513	APPBP2	-			
3762	-29.95	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
3763	-29.96	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
3764	-30	kd	CGS001-388677	NOTCH2NL	-			
3765	-30.01	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
3766	-30.01	kd	CGS001-3569	IL6	Interferons			
3767	-30.01	kd	CGS001-29083	GTPBP8	-			
3768	-30.04	oe	ccsbBroad304_00222	CASP6	Caspases			
3769	-30.05	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
3770	-30.06	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
3771	-30.06	kd	CGS001-80212	CCDC92	-			
3772	-30.08	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
3773	-30.08	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
3774	-30.08	kd	CGS001-10105	PPIF	-			
3775	-30.09	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
3776	-30.09	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
3777	-30.12	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
3778	-30.15	kd	CGS001-9111	NMI	-			
3779	-30.17	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
3780	-30.22	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
3781	-30.22	kd	CGS001-149233	IL23R	IL-12 receptor family			
3782	-30.23	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
3783	-30.24	kd	CGS001-29982	NRBF2	-			
3784	-30.28	oe	ccsbBroad304_00447	DLD	-			
3785	-30.28	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
3786	-30.29	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
3787	-30.31	oe	ccsbBroad304_08461	CDCA4	-			
3788	-30.32	kd	CGS001-8649	LAMTOR3	-			
3789	-30.37	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
3790	-30.37	kd	CGS001-5170	PDPK1	PDK1 family			
3791	-30.38	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
3792	-30.39	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
3793	-30.41	kd	CGS001-7086	TKT	-			
3794	-30.42	oe	ccsbBroad304_01084	NEU1	-			
3795	-30.42	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
3796	-30.45	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
3797	-30.47	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3798	-30.51	kd	CGS001-56916	SMARCAD1	-			
3799	-30.51	kd	CGS001-29911	HOOK2	-			
3800	-30.54	kd	CGS001-1981	EIF4G1	Parkinson disease			
3801	-30.55	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
3802	-30.55	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
3803	-30.56	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
3804	-30.62	oe	ccsbBroad304_01640	TAF12	-			
3805	-30.62	kd	CGS001-8295	TRRAP	TRRAP subfamily			
3806	-30.63	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
3807	-30.64	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
3808	-30.72	kd	CGS001-3171	FOXA3	Forkhead boxes			
3809	-30.75	oe	ccsbBroad304_00949	LRPAP1	-			
3810	-30.75	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
3811	-30.76	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
3812	-30.76	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
3813	-30.76	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
3814	-30.77	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
3815	-30.78	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
3816	-30.81	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
3817	-30.83	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
3818	-30.9	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
3819	-30.93	kd	CGS001-11004	KIF2C	Kinesins			
3820	-30.94	kd	CGS001-5045	FURIN	Subtilisin			
3821	-30.97	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
3822	-30.98	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
3823	-31	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
3824	-31.01	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
3825	-31.04	oe	ccsbBroad304_08217	SCCPDH	-			
3826	-31.07	kd	CGS001-6364	CCL20	Chemokine ligands			
3827	-31.09	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
3828	-31.09	oe	ccsbBroad304_00112	ASNA1	-			
3829	-31.14	kd	CGS001-513	ATP5D	ATPases / F-type			
3830	-31.15	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
3831	-31.16	oe	ccsbBroad304_07326	EIF2B2	-			
3832	-31.16	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
3833	-31.16	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
3834	-31.17	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
3835	-31.18	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
3836	-31.18	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
3837	-31.18	kd	CGS001-22978	NT5C2	Adenosine turnover			
3838	-31.25	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
3839	-31.28	oe	ccsbBroad304_00225	CAT	-			
3840	-31.3	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3841	-31.32	oe	ccsbBroad304_02220	MTFR1	-			
3842	-31.34	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
3843	-31.34	kd	CGS001-433	ASGR2	C-type lectin domain containing			
3844	-31.34	oe	ccsbBroad304_00183	C1S	Complement system			
3845	-31.36	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
3846	-31.36	kd	CGS001-3460	IFNGR2	Interferon receptor family			
3847	-31.4	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
3848	-31.4	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
3849	-31.42	kd	CGS001-9200	PTPLA	-			
3850	-31.43	kd	CGS001-7276	TTR	-			
3851	-31.46	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
3852	-31.48	oe	ccsbBroad304_01832	PAX8	Paired boxes			
3853	-31.48	oe	ccsbBroad304_06783	LGMN	Legumain			
3854	-31.48	kd	CGS001-7263	TST	-			
3855	-31.56	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
3856	-31.58	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
3857	-31.59	oe	ccsbBroad304_01114	NUP88	-			
3858	-31.59	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
3859	-31.59	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
3860	-31.59	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
3861	-31.6	oe	ccsbBroad304_07922	TRIM29	-			
3862	-31.62	kd	CGS001-8428	STK24	YSK subfamily			
3863	-31.63	cc		GPCR Subset GOF	-			
3864	-31.63	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
3865	-31.65	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3866	-31.66	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
3867	-31.71	oe	ccsbBroad304_00993	MDM4	-			
3868	-31.75	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
3869	-31.77	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
3870	-31.78	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3871	-31.79	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
3872	-31.84	kd	CGS001-3992	FADS1	Fatty acid desaturases			
3873	-31.84	kd	CGS001-54205	CYCS	-			
3874	-31.87	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
3875	-31.88	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
3876	-32.02	kd	CGS001-23047	PDS5B	-			
3877	-32.06	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
3878	-32.06	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
3879	-32.07	kd	CGS001-56647	BCCIP	-			
3880	-32.08	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
3881	-32.09	kd	CGS001-6696	SPP1	Endogenous ligands			
3882	-32.1	kd	CGS001-10482	NXF1	-			
3883	-32.1	kd	CGS001-27113	BBC3	-			
3884	-32.14	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
3885	-32.15	kd	CGS001-162699	TCEB3C	-			
3886	-32.15	kd	CGS001-2230	FDX1	-			
3887	-32.19	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
3888	-32.24	kd	CGS001-8667	EIF3H	-			
3889	-32.25	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
3890	-32.27	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
3891	-32.34	kd	CGS001-11136	SLC7A9	SLC7 family			
3892	-32.36	cc		G2 M Checkpoint LOF	-			
3893	-32.37	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
3894	-32.37	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
3895	-32.37	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
3896	-32.38	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
3897	-32.4	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3898	-32.43	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
3899	-32.46	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
3900	-32.5	kd	CGS001-55620	STAP2	-			
3901	-32.51	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
3902	-32.51	kd	CGS001-6643	SNX2	Sorting nexins			
3903	-32.51	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
3904	-32.51	kd	CGS001-1534	CYB561	Cytochrome b genes			
3905	-32.53	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
3906	-32.53	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
3907	-32.56	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
3908	-32.59	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
3909	-32.6	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
3910	-32.65	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3911	-32.68	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
3912	-32.69	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
3913	-32.69	kd	CGS001-3560	IL2RB	IL-2 receptor family			
3914	-32.7	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
3915	-32.71	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
3916	-32.71	oe	ccsbBroad304_00725	HADHA	-			
3917	-32.71	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3918	-32.72	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
3919	-32.76	oe	ccsbBroad304_07287	HYAL2	-			
3920	-32.78	oe	ccsbBroad304_03444	PAF1	-			
3921	-32.81	kd	CGS001-6443	SGCB	-			
3922	-32.81	kd	CGS001-154197	PNLDC1	-			
3923	-32.9	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
3924	-32.93	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
3925	-32.94	kd	CGS001-11198	SUPT16H	-			
3926	-32.96	kd	CGS001-966	CD59	CD molecules			
3927	-32.97	kd	CGS001-5891	MOK	RCK family			
3928	-32.98	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
3929	-32.98	kd	CGS001-5538	PPT1	-			
3930	-33.02	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
3931	-33.04	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
3932	-33.05	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
3933	-33.05	oe	ccsbBroad304_01394	RFX4	-			
3934	-33.11	oe	ccsbBroad304_02017	PEX11A	-			
3935	-33.11	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
3936	-33.15	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
3937	-33.17	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
3938	-33.18	oe	ccsbBroad304_05936	CASP2	Caspases			
3939	-33.18	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
3940	-33.18	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
3941	-33.18	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
3942	-33.2	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
3943	-33.22	kd	CGS001-3685	ITGAV	Integrins			
3944	-33.24	kd	CGS001-10174	SORBS3	-			
3945	-33.3	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
3946	-33.32	oe	ccsbBroad304_06549	SMAD3	SMADs			
3947	-33.32	oe	ccsbBroad304_02526	POP4	-			
3948	-33.32	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
3949	-33.33	kd	CGS001-6233	RPS27A	S ribosomal proteins			
3950	-33.35	kd	CGS001-3176	HNMT	-			
3951	-33.38	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3952	-33.4	kd	CGS001-7431	VIM	Intermediate filaments type III			
3953	-33.4	kd	CGS001-29915	HCFC2	-			
3954	-33.41	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
3955	-33.42	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
3956	-33.42	kd	CGS001-89766	UMODL1	-			
3957	-33.43	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
3958	-33.44	oe	ccsbBroad304_08993	DHDDS	-			
3959	-33.44	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
3960	-33.51	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
3961	-33.52	oe	ccsbBroad304_07277	RTCD1	-			
3962	-33.52	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
3963	-33.56	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
3964	-33.61	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
3965	-33.61	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
3966	-33.62	kd	CGS001-124583	CANT1	-			
3967	-33.64	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3968	-33.65	oe	ccsbBroad304_02399	TNIP1	-			
3969	-33.69	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
3970	-33.72	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
3971	-33.73	kd	CGS001-10841	FTCD	-			
3972	-33.74	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
3973	-33.76	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
3974	-33.77	oe	ccsbBroad304_07411	LPXN	-			
3975	-33.78	oe	ccsbBroad304_03591	ETNK1	-			
3976	-33.78	oe	ccsbBroad304_06004	CKB	-			
3977	-33.79	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
3978	-33.79	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
3979	-33.8	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
3980	-33.81	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
3981	-33.83	oe	ccsbBroad304_10230	STK19	G11 family			
3982	-33.83	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
3983	-33.83	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
3984	-33.88	kd	CGS001-7389	UROD	-			
3985	-33.91	kd	CGS001-11180	WDR6	WD repeat domain containing			
3986	-33.92	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
3987	-33.93	kd	CGS001-2073	ERCC5	-			
3988	-33.94	kd	CGS001-5588	PRKCQ	Delta subfamily			
3989	-33.95	oe	ccsbBroad304_02919	KIAA1279	-			
3990	-33.96	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
3991	-33.97	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
3992	-34	kd	CGS001-6477	SIAH1	-			
3993	-34.02	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
3994	-34.11	oe	ccsbBroad304_01035	MSH5	-			
3995	-34.11	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
3996	-34.11	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
3997	-34.14	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
3998	-34.15	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
3999	-34.21	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
4000	-34.22	oe	ccsbBroad304_01142	PAFAH1B2	-			
4001	-34.22	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
4002	-34.23	oe	ccsbBroad304_06290	GNA15	-			
4003	-34.24	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
4004	-34.26	kd	CGS001-51466	EVL	-			
4005	-34.27	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
4006	-34.28	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4007	-34.29	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
4008	-34.31	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
4009	-34.33	oe	ccsbBroad304_05947	CCNC	-			
4010	-34.34	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
4011	-34.35	kd	CGS001-11325	DDX42	DEAD-boxes			
4012	-34.38	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
4013	-34.4	oe	ccsbBroad304_02195	SPAG7	-			
4014	-34.4	kd	CGS001-4122	MAN2A2	-			
4015	-34.43	kd	CGS001-10645	CAMKK2	Meta subfamily			
4016	-34.44	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4017	-34.47	kd	CGS001-11179	ZNF277	-			
4018	-34.47	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
4019	-34.49	kd	CGS001-2053	EPHX2	-			
4020	-34.5	oe	ccsbBroad304_06518	LDHA	-			
4021	-34.54	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
4022	-34.56	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
4023	-34.57	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
4024	-34.57	kd	CGS001-51015	ISOC1	-			
4025	-34.61	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
4026	-34.61	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4027	-34.61	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
4028	-34.66	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
4029	-34.66	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
4030	-34.68	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
4031	-34.78	kd	CGS001-5663	PSEN1	Presenilin			
4032	-34.8	oe	ccsbBroad304_03186	GMNN	-			
4033	-34.87	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
4034	-34.87	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4035	-34.88	kd	CGS001-4860	PNP	-			
4036	-34.88	kd	CGS001-55644	OSGEP	-			
4037	-34.89	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
4038	-34.92	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
4039	-34.92	kd	CGS001-11212	PROSC	-			
4040	-34.93	kd	CGS001-6514	SLC2A2	Solute carriers			
4041	-34.94	cc		JAK inhibitor	-			
4042	-35.02	oe	ccsbBroad304_06565	MB	-			
4043	-35.07	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
4044	-35.07	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
4045	-35.09	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
4046	-35.09	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
4047	-35.11	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
4048	-35.13	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
4049	-35.13	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
4050	-35.14	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
4051	-35.14	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
4052	-35.18	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
4053	-35.18	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
4054	-35.2	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
4055	-35.22	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
4056	-35.24	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
4057	-35.27	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
4058	-35.28	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
4059	-35.28	oe	ccsbBroad304_07349	MAP7	-			
4060	-35.29	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
4061	-35.3	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
4062	-35.33	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
4063	-35.34	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
4064	-35.37	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
4065	-35.38	oe	ccsbBroad304_05823	ANXA2	Annexins			
4066	-35.41	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
4067	-35.41	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
4068	-35.44	kd	CGS001-58533	SNX6	Sorting nexins			
4069	-35.45	kd	CGS001-7013	TERF1	-			
4070	-35.47	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
4071	-35.48	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
4072	-35.5	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
4073	-35.5	oe	ccsbBroad304_02047	AP1S2	-			
4074	-35.51	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
4075	-35.51	kd	CGS001-169436	C9ORF96	-			
4076	-35.57	kd	CGS001-2155	F7	Chymotrypsin			
4077	-35.59	kd	CGS001-1284	COL4A2	Collagens			
4078	-35.61	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
4079	-35.63	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
4080	-35.64	kd	CGS001-8569	MKNK1	MKN subfamily			
4081	-35.67	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
4082	-35.67	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
4083	-35.68	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
4084	-35.69	oe	ccsbBroad304_01985	EIF3H	-			
4085	-35.7	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4086	-35.7	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
4087	-35.71	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
4088	-35.72	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
4089	-35.72	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
4090	-35.75	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
4091	-35.82	kd	CGS001-50846	DHH	-			
4092	-35.84	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
4093	-35.9	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
4094	-35.91	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
4095	-35.98	oe	ccsbBroad304_00249	CD14	CD molecules			
4096	-35.98	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4097	-35.98	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
4098	-35.99	oe	ccsbBroad304_05192	SPRED2	-			
4099	-35.99	oe	ccsbBroad304_03850	TRIB3	Trbl family			
4100	-35.99	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
4101	-36.02	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
4102	-36.03	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
4103	-36.07	kd	CGS001-7158	TP53BP1	-			
4104	-36.08	oe	ccsbBroad304_03450	TMED9	-			
4105	-36.1	oe	ccsbBroad304_01019	MLH1	-			
4106	-36.1	oe	ccsbBroad304_00550	FDXR	-			
4107	-36.11	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
4108	-36.14	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
4109	-36.14	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
4110	-36.15	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
4111	-36.16	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
4112	-36.16	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
4113	-36.17	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
4114	-36.24	kd	CGS001-5202	PFDN2	-			
4115	-36.26	oe	ccsbBroad304_00113	ASNS	-			
4116	-36.28	kd	CGS001-5664	PSEN2	Presenilin			
4117	-36.3	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
4118	-36.31	oe	ccsbBroad304_06449	ILF3	-			
4119	-36.32	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
4120	-36.33	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
4121	-36.34	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
4122	-36.34	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
4123	-36.36	kd	CGS001-4172	MCM3	-			
4124	-36.37	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
4125	-36.38	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
4126	-36.38	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
4127	-36.38	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
4128	-36.42	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4129	-36.44	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
4130	-36.46	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
4131	-36.47	kd	CGS001-150280	HORMAD2	-			
4132	-36.54	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
4133	-36.57	oe	ccsbBroad304_08426	TEX10	-			
4134	-36.58	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
4135	-36.59	kd	CGS001-10020	GNE	-			
4136	-36.61	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
4137	-36.64	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
4138	-36.66	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4139	-36.67	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
4140	-36.71	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
4141	-36.73	kd	CGS001-54821	ERCC6L	-			
4142	-36.76	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
4143	-36.83	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
4144	-36.88	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
4145	-36.88	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
4146	-36.89	oe	ccsbBroad304_06188	F10	Chymotrypsin			
4147	-36.9	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
4148	-36.92	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
4149	-36.93	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
4150	-36.94	kd	CGS001-65263	PYCRL	-			
4151	-36.97	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
4152	-36.98	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
4153	-36.98	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
4154	-36.99	kd	CGS001-29888	STRN4	WD repeat domain containing			
4155	-37	kd	CGS001-718	C3	Endogenous ligands			
4156	-37	kd	CGS001-35	ACADS	-			
4157	-37.01	oe	ccsbBroad304_03089	PACSIN3	-			
4158	-37.01	oe	ccsbBroad304_00389	CTBP1	-			
4159	-37.01	cp	BRD-K65910366	KUC103904N	-666			-666
4160	-37.05	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
4161	-37.06	kd	CGS001-83933	HDAC10	Histone deacetylases			
4162	-37.09	oe	ccsbBroad304_00710	GUSB	-			
4163	-37.09	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
4164	-37.11	kd	CGS001-5708	PSMD2	Proteasome subunits			
4165	-37.12	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
4166	-37.12	kd	CGS001-1841	DTYMK	-			
4167	-37.13	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
4168	-37.13	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
4169	-37.15	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
4170	-37.17	kd	CGS001-839	CASP6	Caspases			
4171	-37.19	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
4172	-37.2	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
4173	-37.21	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
4174	-37.21	kd	CGS001-4758	NEU1	-			
4175	-37.22	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
4176	-37.25	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
4177	-37.27	oe	ccsbBroad304_02217	FEZ1	-			
4178	-37.29	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
4179	-37.31	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
4180	-37.36	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
4181	-37.39	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
4182	-37.42	kd	CGS001-286380	FOXD4L3	-			
4183	-37.42	kd	CGS001-2114	ETS2	ETS Transcription Factors			
4184	-37.42	kd	CGS001-183	AGT	Endogenous ligands			
4185	-37.44	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
4186	-37.47	oe	ccsbBroad304_02094	FIBP	-			
4187	-37.53	oe	ccsbBroad304_00099	ARG2	Arginase			
4188	-37.53	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
4189	-37.53	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
4190	-37.53	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4191	-37.54	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
4192	-37.55	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
4193	-37.57	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
4194	-37.57	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
4195	-37.57	kd	CGS001-9541	CIR1	-			
4196	-37.58	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
4197	-37.58	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4198	-37.6	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
4199	-37.62	oe	ccsbBroad304_02804	KLHDC2	-			
4200	-37.63	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
4201	-37.65	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
4202	-37.66	oe	ccsbBroad304_01976	EIF4EBP3	-			
4203	-37.67	cc		Histone deacetylases LOF	-			
4204	-37.75	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
4205	-37.8	kd	CGS001-3638	INSIG1	-			
4206	-37.9	oe	ccsbBroad304_07768	NISCH	-			
4207	-37.9	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
4208	-37.91	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
4209	-37.91	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
4210	-37.91	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
4211	-37.92	cc		S100 calcium binding proteins LOF	-			
4212	-37.93	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
4213	-37.94	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
4214	-37.95	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
4215	-37.97	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
4216	-38	kd	CGS001-1955	MEGF9	-			
4217	-38	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
4218	-38.01	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
4219	-38.01	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
4220	-38.02	oe	ccsbBroad304_00161	BID	Endogenous ligands			
4221	-38.04	cc		Bacterial DNA gyrase inhibitor	-			
4222	-38.04	oe	ccsbBroad304_02759	DICER1	-			
4223	-38.04	kd	CGS001-9531	BAG3	-			
4224	-38.07	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
4225	-38.09	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
4226	-38.11	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
4227	-38.12	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
4228	-38.16	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
4229	-38.17	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
4230	-38.17	oe	ccsbBroad304_05757	ACADS	-			
4231	-38.17	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
4232	-38.18	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
4233	-38.2	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
4234	-38.23	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
4235	-38.24	oe	ccsbBroad304_02458	STK25	YSK subfamily			
4236	-38.27	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
4237	-38.27	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
4238	-38.3	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
4239	-38.32	oe	ccsbBroad304_13633	PI4KAP2	-			
4240	-38.35	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
4241	-38.38	cc		Reverse transcriptase inhibitor	-			
4242	-38.38	oe	ccsbBroad304_00020	ACY1	-			
4243	-38.39	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
4244	-38.44	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
4245	-38.48	kd	CGS001-64343	AZI2	-			
4246	-38.49	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
4247	-38.52	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4248	-38.55	oe	ccsbBroad304_00960	SMAD1	SMADs			
4249	-38.65	kd	CGS001-1736	DKC1	-			
4250	-38.66	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
4251	-38.69	kd	CGS001-3046	HBE1	-			
4252	-38.7	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
4253	-38.71	oe	ccsbBroad304_02205	WTAP	-			
4254	-38.71	oe	ccsbBroad304_02419	NDRG1	-			
4255	-38.71	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
4256	-38.74	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
4257	-38.77	kd	CGS001-64333	ARHGAP9	Rho GTPase activating proteins			
4258	-38.81	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
4259	-38.83	oe	ccsbBroad304_08898	TRAK2	-			
4260	-38.83	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
4261	-38.87	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4262	-38.89	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
4263	-38.89	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
4264	-38.9	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
4265	-38.9	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
4266	-38.9	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
4267	-38.94	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
4268	-39.01	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
4269	-39.06	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
4270	-39.11	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
4271	-39.11	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
4272	-39.14	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
4273	-39.15	oe	ccsbBroad304_02345	TXNDC9	-			
4274	-39.16	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
4275	-39.21	cc		Sterol demethylase inhibitor	-			
4276	-39.21	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
4277	-39.22	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
4278	-39.23	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
4279	-39.33	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
4280	-39.39	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
4281	-39.41	oe	ccsbBroad304_06144	EFNB3	Ephrins			
4282	-39.41	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
4283	-39.45	kd	CGS001-7270	TTF1	-			
4284	-39.46	oe	ccsbBroad304_13952	SHMT2	-			
4285	-39.51	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
4286	-39.51	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
4287	-39.51	oe	ccsbBroad304_06383	HMMR	CD molecules			
4288	-39.54	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
4289	-39.55	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4290	-39.55	kd	CGS001-2782	GNB1	WD repeat domain containing			
4291	-39.56	oe	ccsbBroad304_07605	LYPLA1	-			
4292	-39.56	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
4293	-39.58	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
4294	-39.66	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
4295	-39.68	kd	CGS001-55536	CDCA7L	-			
4296	-39.69	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
4297	-39.72	oe	ccsbBroad304_06889	RPN2	-			
4298	-39.72	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
4299	-39.73	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
4300	-39.75	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
4301	-39.77	kd	CGS001-8731	RNMT	-			
4302	-39.83	cc		Progesterone receptor agonist	-			
4303	-39.84	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
4304	-39.86	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
4305	-39.87	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
4306	-39.92	oe	ccsbBroad304_06976	SMARCE1	-			
4307	-39.92	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
4308	-39.94	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
4309	-39.94	kd	CGS001-9695	EDEM1	-			
4310	-40.01	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
4311	-40.01	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
4312	-40.03	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
4313	-40.04	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
4314	-40.04	kd	CGS001-22921	MSRB2	-			
4315	-40.06	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
4316	-40.06	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
4317	-40.09	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
4318	-40.09	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
4319	-40.14	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
4320	-40.2	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
4321	-40.2	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
4322	-40.23	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
4323	-40.23	kd	CGS001-26511	CHIC2	-			
4324	-40.31	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
4325	-40.31	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
4326	-40.32	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
4327	-40.32	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
4328	-40.34	oe	ccsbBroad304_09284	UBE3B	-			
4329	-40.34	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
4330	-40.39	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
4331	-40.42	kd	CGS001-57019	CIAPIN1	-			
4332	-40.43	cc		Phospholipases LOF	-			
4333	-40.48	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
4334	-40.49	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
4335	-40.52	oe	ccsbBroad304_07119	UGP2	-			
4336	-40.53	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
4337	-40.58	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
4338	-40.59	kd	CGS001-114785	MBD6	-			
4339	-40.61	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
4340	-40.62	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
4341	-40.63	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
4342	-40.63	kd	CGS001-5209	PFKFB3	-			
4343	-40.64	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
4344	-40.66	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
4345	-40.7	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4346	-40.72	oe	ccsbBroad304_06253	GALT	-			
4347	-40.77	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
4348	-40.84	kd	CGS001-29916	SNX11	Sorting nexins			
4349	-40.84	kd	CGS001-1384	CRAT	-			
4350	-40.85	kd	CGS001-11232	POLG2	DNA polymerases			
4351	-40.87	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
4352	-40.87	kd	CGS001-1633	DCK	-			
4353	-40.88	oe	ccsbBroad304_07800	EXOSC8	-			
4354	-40.89	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
4355	-40.89	kd	CGS001-6856	SYPL1	-			
4356	-40.9	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
4357	-40.9	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
4358	-40.9	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
4359	-40.93	kd	CGS001-11157	LSM6	-			
4360	-40.96	oe	ccsbBroad304_03615	ZNF673	-			
4361	-41.02	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
4362	-41.03	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
4363	-41.04	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
4364	-41.07	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
4365	-41.11	kd	CGS001-6387	CXCL12	Endogenous ligands			
4366	-41.13	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
4367	-41.17	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
4368	-41.21	oe	ccsbBroad304_13499	KSR2	RAF family			
4369	-41.21	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
4370	-41.23	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
4371	-41.24	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
4372	-41.25	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
4373	-41.26	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
4374	-41.26	kd	CGS001-7016	TESK1	TESK subfamily			
4375	-41.28	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
4376	-41.32	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
4377	-41.37	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4378	-41.37	kd	CGS001-836	CASP3	Caspases			
4379	-41.39	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
4380	-41.4	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
4381	-41.41	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
4382	-41.46	kd	CGS001-80314	EPC1	-			
4383	-41.51	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
4384	-41.51	kd	CGS001-1493	CTLA4	CD molecules			
4385	-41.52	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
4386	-41.53	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
4387	-41.54	kd	CGS001-174	AFP	-			
4388	-41.55	cc		IGF-1 inhibitor	-			
4389	-41.55	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
4390	-41.56	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
4391	-41.6	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4392	-41.62	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
4393	-41.64	kd	CGS001-1066	CES1	Carboxylesterases			
4394	-41.66	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
4395	-41.67	kd	CGS001-533	ATP6V0B	ATPases / V-type			
4396	-41.68	cc		FXR antagonist	-			
4397	-41.7	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
4398	-41.71	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
4399	-41.73	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
4400	-41.75	oe	ccsbBroad304_01748	UFD1L	-			
4401	-41.76	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
4402	-41.78	kd	CGS001-23588	KLHDC2	-			
4403	-41.83	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
4404	-41.84	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
4405	-41.85	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
4406	-41.89	oe	ccsbBroad304_01674	TIMP4	-			
4407	-41.89	kd	CGS001-4925	NUCB2	EF-hand domain containing			
4408	-41.9	oe	ccsbBroad304_10758	CTBP2	-			
4409	-41.92	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
4410	-41.95	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
4411	-41.95	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
4412	-42.05	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
4413	-42.05	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
4414	-42.06	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
4415	-42.06	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
4416	-42.1	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
4417	-42.11	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
4418	-42.12	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
4419	-42.14	oe	ccsbBroad304_01180	PFKFB3	-			
4420	-42.19	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
4421	-42.21	kd	CGS001-63933	CCDC90A	-			
4422	-42.22	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4423	-42.23	oe	ccsbBroad304_00881	IRF5	-			
4424	-42.35	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
4425	-42.41	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4426	-42.43	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
4427	-42.44	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
4428	-42.46	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
4429	-42.47	oe	ccsbBroad304_03433	DDIT4	-			
4430	-42.48	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
4431	-42.5	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
4432	-42.52	oe	ccsbBroad304_03155	DHH	-			
4433	-42.52	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
4434	-42.55	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
4435	-42.55	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
4436	-42.59	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
4437	-42.65	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
4438	-42.72	oe	ccsbBroad304_08888	ACD	-			
4439	-42.73	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
4440	-42.74	oe	ccsbBroad304_00072	ANXA7	Annexins			
4441	-42.81	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
4442	-42.82	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
4443	-42.88	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
4444	-42.93	oe	ccsbBroad304_00991	MDH1	-			
4445	-42.95	kd	CGS001-5257	PHKB	-			
4446	-42.98	kd	CGS001-51290	ERGIC2	-			
4447	-43	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
4448	-43.07	kd	CGS001-5245	PHB	-			
4449	-43.11	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
4450	-43.12	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
4451	-43.13	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
4452	-43.17	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
4453	-43.17	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
4454	-43.2	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
4455	-43.2	kd	CGS001-2932	GSK3B	GSK subfamily			
4456	-43.22	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
4457	-43.33	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
4458	-43.34	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
4459	-43.35	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
4460	-43.35	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
4461	-43.4	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
4462	-43.42	oe	ccsbBroad304_00501	EMD	-			
4463	-43.44	oe	ccsbBroad304_07761	CORO1A	Coronins			
4464	-43.45	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
4465	-43.47	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
4466	-43.49	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
4467	-43.5	oe	ccsbBroad304_04457	TOX2	-			
4468	-43.54	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
4469	-43.55	kd	CGS001-283150	FOXR1	Forkhead boxes			
4470	-43.58	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
4471	-43.62	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
4472	-43.63	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
4473	-43.68	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
4474	-43.69	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
4475	-43.7	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4476	-43.71	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
4477	-43.71	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
4478	-43.72	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
4479	-43.73	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
4480	-43.79	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4481	-43.8	kd	CGS001-9270	ITGB1BP1	-			
4482	-43.86	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
4483	-43.88	cc		Lipocalins GOF	-			
4484	-43.91	oe	ccsbBroad304_02576	MLLT11	-			
4485	-43.91	oe	ccsbBroad304_03179	BOLA1	-			
4486	-43.91	kd	CGS001-2747	GLUD2	-			
4487	-43.95	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
4488	-43.97	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
4489	-44	oe	ccsbBroad304_06535	LPL	-			
4490	-44.01	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
4491	-44.02	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
4492	-44.03	oe	ccsbBroad304_06090	DDOST	-			
4493	-44.03	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
4494	-44.06	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
4495	-44.07	oe	ccsbBroad304_01184	PGK1	-			
4496	-44.07	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
4497	-44.09	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
4498	-44.1	oe	ccsbBroad304_06671	OPA1	-			
4499	-44.1	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
4500	-44.11	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
4501	-44.13	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
4502	-44.18	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
4503	-44.19	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
4504	-44.21	cc		PPAR receptor agonist	-			
4505	-44.22	cc		HMGCR inhibitor	-			
4506	-44.22	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
4507	-44.22	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
4508	-44.28	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
4509	-44.29	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
4510	-44.31	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
4511	-44.42	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
4512	-44.44	kd	CGS001-84515	MCM8	-			
4513	-44.45	kd	CGS001-826	CAPNS1	EF-hand domain containing			
4514	-44.5	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
4515	-44.56	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
4516	-44.57	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
4517	-44.6	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
4518	-44.61	kd	CGS001-8464	SUPT3H	-			
4519	-44.64	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
4520	-44.68	oe	ccsbBroad304_06040	CRY1	-			
4521	-44.73	cc		NFKB Activation GOF	-			
4522	-44.74	oe	ccsbBroad304_07220	CDC45	-			
4523	-44.78	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
4524	-44.81	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
4525	-44.84	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
4526	-44.85	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4527	-44.9	kd	CGS001-7982	ST7	-			
4528	-44.95	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
4529	-44.96	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
4530	-44.97	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
4531	-45.01	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
4532	-45.05	oe	ccsbBroad304_06683	FURIN	Subtilisin			
4533	-45.1	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4534	-45.11	oe	ccsbBroad304_02349	MPHOSPH9	-			
4535	-45.17	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
4536	-45.18	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
4537	-45.23	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
4538	-45.23	oe	ccsbBroad304_07688	FAM114A2	-			
4539	-45.24	kd	CGS001-8772	FADD	-			
4540	-45.25	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
4541	-45.27	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
4542	-45.27	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
4543	-45.32	kd	CGS001-2729	GCLC	-			
4544	-45.37	kd	CGS001-1497	CTNS	-			
4545	-45.39	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
4546	-45.39	kd	CGS001-6723	SRM	-			
4547	-45.4	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
4548	-45.41	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
4549	-45.45	kd	CGS001-3269	HRH1	Histamine receptors			
4550	-45.47	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
4551	-45.49	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
4552	-45.51	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
4553	-45.51	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
4554	-45.52	kd	CGS001-10001	MED6	-			
4555	-45.53	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
4556	-45.59	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
4557	-45.64	oe	ccsbBroad304_02138	TRIP10	-			
4558	-45.65	kd	CGS001-3827	KNG1	Endogenous ligands			
4559	-45.65	kd	CGS001-23581	CASP14	Caspases			
4560	-45.68	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
4561	-45.71	oe	ccsbBroad304_09821	TMEM154	-			
4562	-45.71	oe	ccsbBroad304_01960	CASK	CASK family			
4563	-45.76	oe	ccsbBroad304_01675	TK1	-			
4564	-45.77	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
4565	-45.83	oe	ccsbBroad304_01532	SIAH1	-			
4566	-45.88	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
4567	-45.89	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
4568	-45.9	kd	CGS001-3416	IDE	Pitrilysin			
4569	-45.91	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
4570	-45.93	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
4571	-45.93	kd	CGS001-4594	MUT	-			
4572	-45.95	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
4573	-45.98	oe	ccsbBroad304_02604	B3GNT1	-			
4574	-45.99	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
4575	-46	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4576	-46.02	oe	ccsbBroad304_06301	GOT2	-			
4577	-46.12	oe	ccsbBroad304_03235	TUBD1	Tubulins			
4578	-46.13	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
4579	-46.13	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
4580	-46.19	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
4581	-46.2	kd	CGS001-26128	KIAA1279	-			
4582	-46.22	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4583	-46.25	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
4584	-46.26	oe	ccsbBroad304_00624	GCK	Hexokinases			
4585	-46.27	kd	CGS001-527	ATP6V0C	ATPases / V-type			
4586	-46.28	oe	ccsbBroad304_01701	TPI1	-			
4587	-46.28	oe	ccsbBroad304_02143	CNOT8	-			
4588	-46.29	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
4589	-46.31	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
4590	-46.31	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
4591	-46.41	kd	CGS001-11040	PIM2	PIM family			
4592	-46.43	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
4593	-46.46	cc		ATPase inhibitor	-			
4594	-46.46	oe	ccsbBroad304_06140	EEF1D	-			
4595	-46.47	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
4596	-46.48	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
4597	-46.5	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
4598	-46.51	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
4599	-46.52	cc		Bromodomain Inhibitor	-			
4600	-46.58	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
4601	-46.58	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
4602	-46.58	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
4603	-46.65	kd	CGS001-4221	MEN1	-			
4604	-46.65	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
4605	-46.74	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
4606	-46.74	kd	CGS001-27244	SESN1	-			
4607	-46.83	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4608	-46.83	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
4609	-46.84	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4610	-46.84	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
4611	-46.84	kd	CGS001-1069	CETN2	EF-hand domain containing			
4612	-46.88	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
4613	-46.9	cc		MEK inhibitor	-			
4614	-46.91	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
4615	-46.95	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4616	-46.96	kd	CGS001-90861	HN1L	-			
4617	-47	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
4618	-47.05	oe	ccsbBroad304_13598	NRBP2	NRBP family			
4619	-47.06	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
4620	-47.08	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
4621	-47.09	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
4622	-47.1	oe	ccsbBroad304_06648	CNOT3	-			
4623	-47.1	kd	CGS001-384	ARG2	Arginase			
4624	-47.12	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
4625	-47.17	oe	ccsbBroad304_00489	EHHADH	-			
4626	-47.2	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
4627	-47.26	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
4628	-47.29	oe	ccsbBroad304_00179	BTG1	-			
4629	-47.3	oe	ccsbBroad304_14143	NUSAP1	-			
4630	-47.33	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
4631	-47.35	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
4632	-47.36	kd	CGS001-338	APOB	Apolipoproteins			
4633	-47.39	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
4634	-47.4	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
4635	-47.41	oe	ccsbBroad304_01724	TTR	-			
4636	-47.41	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
4637	-47.43	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
4638	-47.44	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
4639	-47.52	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
4640	-47.52	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
4641	-47.55	kd	CGS001-5480	PPIC	-			
4642	-47.56	oe	ccsbBroad304_02018	SUCLA2	-			
4643	-47.6	cc		SRY LOF	-			
4644	-47.61	kd	CGS001-6491	STIL	-			
4645	-47.72	kd	CGS001-8833	GMPS	-			
4646	-47.74	oe	ccsbBroad304_01183	PGD	-			
4647	-47.74	kd	CGS001-6185	RPN2	-			
4648	-47.75	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
4649	-47.76	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
4650	-47.79	oe	ccsbBroad304_02373	SPRY2	-			
4651	-47.8	oe	ccsbBroad304_07374	PTPLA	-			
4652	-47.8	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
4653	-47.81	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
4654	-47.82	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
4655	-47.83	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
4656	-47.83	kd	CGS001-7185	TRAF1	-			
4657	-47.84	oe	ccsbBroad304_02402	TMEM5	-			
4658	-47.89	cc		PI3K inhibitor	-			
4659	-48.08	kd	CGS001-1398	CRK	SH2 domain containing			
4660	-48.08	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
4661	-48.15	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
4662	-48.15	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
4663	-48.16	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
4664	-48.24	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
4665	-48.25	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
4666	-48.25	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
4667	-48.27	kd	CGS001-6193	RPS5	S ribosomal proteins			
4668	-48.39	oe	ccsbBroad304_00542	FBP1	-			
4669	-48.44	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
4670	-48.44	oe	ccsbBroad304_00817	IDH2	-			
4671	-48.45	kd	CGS001-275	AMT	-			
4672	-48.56	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4673	-48.58	oe	ccsbBroad304_06862	RGS3	-			
4674	-48.6	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
4675	-48.6	kd	CGS001-10904	BLCAP	-			
4676	-48.66	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
4677	-48.68	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
4678	-48.75	oe	ccsbBroad304_08596	EAPP	-			
4679	-48.84	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
4680	-48.91	kd	CGS001-2581	GALC	-			
4681	-48.94	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
4682	-48.97	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
4683	-49.01	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
4684	-49.08	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
4685	-49.1	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
4686	-49.12	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
4687	-49.13	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
4688	-49.15	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
4689	-49.16	kd	CGS001-51160	VPS28	-			
4690	-49.2	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
4691	-49.25	oe	ccsbBroad304_05902	BNIP3	-			
4692	-49.26	oe	ccsbBroad304_00841	IKBKB	IKK family			
4693	-49.26	oe	ccsbBroad304_01617	STX4	-			
4694	-49.26	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
4695	-49.26	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
4696	-49.27	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
4697	-49.28	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
4698	-49.3	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
4699	-49.33	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
4700	-49.39	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
4701	-49.4	kd	CGS001-10494	STK25	YSK subfamily			
4702	-49.45	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
4703	-49.48	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
4704	-49.57	kd	CGS001-2597	GAPDH	-			
4705	-49.6	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
4706	-49.65	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4707	-49.69	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
4708	-49.71	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
4709	-49.72	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4710	-49.79	oe	ccsbBroad304_02298	DNM1L	-			
4711	-49.86	kd	CGS001-10412	NSA2	-			
4712	-49.9	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
4713	-49.9	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
4714	-49.91	kd	CGS001-7079	TIMP4	-			
4715	-49.94	kd	CGS001-4067	LYN	Src family			
4716	-49.96	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
4717	-50.03	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
4718	-50.05	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
4719	-50.05	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
4720	-50.06	oe	ccsbBroad304_03544	FAIM	-			
4721	-50.12	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
4722	-50.13	kd	CGS001-7088	TLE1	WD repeat domain containing			
4723	-50.16	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
4724	-50.23	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
4725	-50.34	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
4726	-50.36	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
4727	-50.38	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
4728	-50.39	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
4729	-50.4	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
4730	-50.46	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
4731	-50.48	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
4732	-50.5	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
4733	-50.57	oe	ccsbBroad304_07814	SACM1L	-			
4734	-50.58	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
4735	-50.67	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
4736	-50.68	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
4737	-50.69	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
4738	-50.78	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
4739	-50.8	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
4740	-50.81	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
4741	-50.81	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
4742	-50.85	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
4743	-50.88	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4744	-50.88	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
4745	-50.89	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
4746	-50.94	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
4747	-50.96	kd	CGS001-5997	RGS2	Endogenous ligands			
4748	-50.96	kd	CGS001-2963	GTF2F2	General transcription factors			
4749	-50.97	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
4750	-50.98	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
4751	-51	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
4752	-51	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
4753	-51.03	oe	ccsbBroad304_06318	GPER	-			
4754	-51.09	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
4755	-51.2	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4756	-51.21	oe	ccsbBroad304_01862	YEATS4	-			
4757	-51.22	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4758	-51.22	kd	CGS001-6342	SCP2	-			
4759	-51.23	oe	ccsbBroad304_07843	FCHO1	-			
4760	-51.24	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
4761	-51.26	oe	ccsbBroad304_03497	TXNL4B	-			
4762	-51.28	kd	CGS001-2109	ETFB	-			
4763	-51.35	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
4764	-51.35	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
4765	-51.36	oe	ccsbBroad304_00747	HLF	-			
4766	-51.36	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
4767	-51.36	kd	CGS001-10914	PAPOLA	-			
4768	-51.37	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
4769	-51.37	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
4770	-51.39	oe	ccsbBroad304_02163	MED7	-			
4771	-51.55	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
4772	-51.58	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
4773	-51.59	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
4774	-51.61	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
4775	-51.63	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
4776	-51.65	oe	ccsbBroad304_00963	SMAD5	SMADs			
4777	-51.65	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
4778	-51.7	oe	ccsbBroad304_02822	ARFIP2	-			
4779	-51.75	cp	BRD-A02189320	met-leu-phe	-666			-666
4780	-51.81	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
4781	-51.83	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
4782	-51.83	kd	CGS001-3281	HSBP1	-			
4783	-51.86	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
4784	-51.87	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
4785	-51.88	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
4786	-51.98	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
4787	-52	oe	ccsbBroad304_00931	LCN2	Lipocalins			
4788	-52	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
4789	-52.05	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
4790	-52.07	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
4791	-52.08	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
4792	-52.09	kd	CGS001-6788	STK3	MST subfamily			
4793	-52.16	oe	ccsbBroad304_02964	TIMM9	-			
4794	-52.2	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
4795	-52.22	kd	CGS001-930	CD19	CD molecules			
4796	-52.23	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
4797	-52.29	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
4798	-52.31	oe	ccsbBroad304_03917	RBKS	-			
4799	-52.31	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
4800	-52.34	kd	CGS001-51586	MED15	-			
4801	-52.35	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
4802	-52.36	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4803	-52.36	kd	CGS001-642	BLMH	-			
4804	-52.4	oe	ccsbBroad304_08660	SMARCAD1	-			
4805	-52.41	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
4806	-52.43	kd	CGS001-6519	SLC3A1	SLC3 family			
4807	-52.48	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
4808	-52.5	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
4809	-52.57	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
4810	-52.63	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
4811	-52.71	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
4812	-52.81	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
4813	-52.81	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
4814	-52.89	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
4815	-52.98	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
4816	-53	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
4817	-53.04	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
4818	-53.08	cc		Imidazoline ligand	-			
4819	-53.18	oe	ccsbBroad304_02626	PKIG	-			
4820	-53.2	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4821	-53.23	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
4822	-53.3	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
4823	-53.36	kd	CGS001-6195	RPS6KA1	RSK subfamily			
4824	-53.4	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
4825	-53.41	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
4826	-53.44	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
4827	-53.45	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4828	-53.46	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
4829	-53.47	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
4830	-53.63	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
4831	-53.68	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
4832	-53.69	oe	ccsbBroad304_03980	DCLRE1B	-			
4833	-53.73	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
4834	-53.76	cc		Proteasome Pathway LOF	-			
4835	-53.78	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4836	-53.9	kd	CGS001-55577	NAGK	-			
4837	-53.9	oe	ccsbBroad304_08709	SCYL3	-			
4838	-53.98	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
4839	-54	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
4840	-54	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
4841	-54.01	oe	ccsbBroad304_04752	IKBIP	-			
4842	-54.02	kd	CGS001-5362	PLXNA2	Plexins			
4843	-54.15	kd	CGS001-5690	PSMB2	Proteasome subunits			
4844	-54.19	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
4845	-54.2	oe	ccsbBroad304_09833	SENP5	-			
4846	-54.23	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
4847	-54.25	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
4848	-54.25	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
4849	-54.32	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
4850	-54.32	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4851	-54.32	oe	ccsbBroad304_03732	NPDC1	-			
4852	-54.34	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
4853	-54.34	kd	CGS001-822	CAPG	-			
4854	-54.36	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
4855	-54.45	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
4856	-54.49	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
4857	-54.49	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
4858	-54.53	kd	CGS001-7165	TPD52L2	-			
4859	-54.6	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
4860	-54.6	kd	CGS001-113451	ADC	-			
4861	-54.64	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
4862	-54.64	kd	CGS001-80274	SCUBE1	-			
4863	-54.67	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
4864	-54.68	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
4865	-54.7	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4866	-54.78	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
4867	-54.79	oe	ccsbBroad304_01654	TCTA	-			
4868	-54.84	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
4869	-54.85	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
4870	-54.85	oe	ccsbBroad304_00811	ICAM1	CD molecules			
4871	-54.87	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
4872	-54.9	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
4873	-54.96	kd	CGS001-4931	NVL	ATPases / AAA-type			
4874	-54.97	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
4875	-54.99	kd	CGS001-122402	TDRD9	Tudor domain containing			
4876	-55.05	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
4877	-55.11	kd	CGS001-9322	TRIP10	-			
4878	-55.16	cc		IMPDH inhibitor	-			
4879	-55.25	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
4880	-55.27	kd	CGS001-151126	ZNF385B	-			
4881	-55.35	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
4882	-55.4	kd	CGS001-6944	VPS72	-			
4883	-55.42	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
4884	-55.45	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
4885	-55.49	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
4886	-55.52	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
4887	-55.53	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
4888	-55.55	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
4889	-55.56	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
4890	-55.61	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
4891	-55.62	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
4892	-55.63	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
4893	-55.69	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
4894	-55.79	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
4895	-55.79	kd	CGS001-4697	NDUFA4	-			
4896	-55.83	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
4897	-55.87	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
4898	-55.98	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4899	-56.01	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
4900	-56.08	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
4901	-56.11	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
4902	-56.12	kd	CGS001-2621	GAS6	-			
4903	-56.14	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
4904	-56.18	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
4905	-56.19	kd	CGS001-6217	RPS16	S ribosomal proteins			
4906	-56.2	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
4907	-56.21	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
4908	-56.28	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
4909	-56.3	kd	CGS001-9276	COPB2	WD repeat domain containing			
4910	-56.32	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
4911	-56.34	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
4912	-56.35	kd	CGS001-216	ALDH1A1	Aldehyde dehydrogenases			
4913	-56.39	oe	ccsbBroad304_00620	GCDH	-			
4914	-56.4	oe	ccsbBroad304_01673	TIMP3	-			
4915	-56.4	oe	ccsbBroad304_00054	ALDOC	-			
4916	-56.45	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
4917	-56.45	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
4918	-56.45	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
4919	-56.47	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
4920	-56.47	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
4921	-56.51	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
4922	-56.51	kd	CGS001-327	APEH	Prolyl oligopeptidase			
4923	-56.52	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
4924	-56.57	oe	ccsbBroad304_00462	DR1	-			
4925	-56.57	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
4926	-56.62	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
4927	-56.62	kd	CGS001-5253	PHF2	Histone demethylases			
4928	-56.66	kd	CGS001-51014	TMED7	-			
4929	-56.68	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
4930	-56.71	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
4931	-56.72	oe	ccsbBroad304_02864	PRDX5	-			
4932	-56.74	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
4933	-56.74	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
4934	-56.75	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
4935	-56.78	oe	ccsbBroad304_00810	HYAL1	-			
4936	-56.78	kd	CGS001-9759	HDAC4	Histone deacetylases			
4937	-56.82	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
4938	-56.87	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
4939	-56.87	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
4940	-56.88	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
4941	-56.94	kd	CGS001-5300	PIN1	-			
4942	-57.01	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
4943	-57.01	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
4944	-57.02	oe	ccsbBroad304_06085	DCK	-			
4945	-57.07	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
4946	-57.07	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
4947	-57.13	oe	ccsbBroad304_02249	KIAA0494	-			
4948	-57.18	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
4949	-57.32	oe	ccsbBroad304_07128	VHL	-			
4950	-57.34	oe	ccsbBroad304_00564	FGR	Src family			
4951	-57.37	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
4952	-57.38	kd	CGS001-538	ATP7A	ATPases / P-type			
4953	-57.45	kd	CGS001-2197	FAU	S ribosomal proteins			
4954	-57.46	oe	ccsbBroad304_00519	ETFB	-			
4955	-57.49	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
4956	-57.54	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
4957	-57.54	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
4958	-57.55	oe	ccsbBroad304_02136	COPS2	-			
4959	-57.57	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
4960	-57.59	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
4961	-57.62	oe	ccsbBroad304_09578	PASD1	-			
4962	-57.66	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
4963	-57.67	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
4964	-57.67	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
4965	-57.71	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4966	-57.72	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
4967	-57.76	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
4968	-57.8	oe	ccsbBroad304_10207	ERLIN1	-			
4969	-57.81	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
4970	-57.83	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
4971	-57.84	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
4972	-57.84	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
4973	-57.89	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
4974	-57.92	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
4975	-57.94	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
4976	-57.94	kd	CGS001-955	ENTPD6	-			
4977	-58	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
4978	-58.02	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
4979	-58.08	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4980	-58.13	kd	CGS001-9988	DMTF1	-			
4981	-58.18	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
4982	-58.19	oe	ccsbBroad304_00651	GNAI3	-			
4983	-58.2	kd	CGS001-3939	LDHA	-			
4984	-58.21	oe	ccsbBroad304_00329	CLTA	-			
4985	-58.26	cc		HSP inhibitor	-			
4986	-58.26	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
4987	-58.27	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
4988	-58.33	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
4989	-58.36	kd	CGS001-8639	AOC3	Oxidoreductases			
4990	-58.37	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
4991	-58.39	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
4992	-58.41	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
4993	-58.44	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
4994	-58.45	kd	CGS001-3579	CXCR2	Chemokine receptors			
4995	-58.46	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
4996	-58.5	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
4997	-58.53	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
4998	-58.54	kd	CGS001-1879	EBF1	-			
4999	-58.55	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
5000	-58.57	kd	CGS001-8801	SUCLG2	-			
5001	-58.59	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
5002	-58.59	oe	ccsbBroad304_10491	PFKL	-			
5003	-58.64	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
5004	-58.64	kd	CGS001-10606	PAICS	-			
5005	-58.79	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
5006	-58.81	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
5007	-58.83	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
5008	-58.9	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
5009	-58.94	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
5010	-58.95	oe	ccsbBroad304_07592	CEPT1	-			
5011	-58.98	oe	ccsbBroad304_00626	GDI1	-			
5012	-58.99	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
5013	-58.99	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
5014	-59.04	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
5015	-59.09	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
5016	-59.12	oe	ccsbBroad304_00009	ACLY	-			
5017	-59.16	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
5018	-59.21	oe	ccsbBroad304_00472	EBF1	-			
5019	-59.23	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
5020	-59.24	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
5021	-59.27	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
5022	-59.35	kd	CGS001-5387	PMS2P3	-			
5023	-59.36	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
5024	-59.37	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
5025	-59.37	kd	CGS001-23451	SF3B1	-			
5026	-59.38	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
5027	-59.39	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
5028	-59.42	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
5029	-59.46	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5030	-59.49	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
5031	-59.55	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
5032	-59.57	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
5033	-59.61	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
5034	-59.64	oe	ccsbBroad304_07275	PSMG1	-			
5035	-59.65	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
5036	-59.68	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
5037	-59.69	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
5038	-59.69	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
5039	-59.83	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
5040	-59.89	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
5041	-59.92	kd	CGS001-5684	PSMA3	Proteasome subunits			
5042	-59.94	oe	ccsbBroad304_07045	TEAD4	-			
5043	-59.94	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
5044	-59.95	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
5045	-59.95	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
5046	-59.98	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
5047	-59.98	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
5048	-59.99	oe	ccsbBroad304_02580	TMED10	-			
5049	-60.01	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
5050	-60.09	oe	ccsbBroad304_03798	PHTF2	-			
5051	-60.13	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
5052	-60.13	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
5053	-60.14	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
5054	-60.14	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
5055	-60.24	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5056	-60.24	kd	CGS001-9871	SEC24D	-			
5057	-60.27	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
5058	-60.38	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
5059	-60.4	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
5060	-60.43	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
5061	-60.45	oe	ccsbBroad304_00600	FYN	Src family			
5062	-60.49	kd	CGS001-23244	PDS5A	-			
5063	-60.5	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
5064	-60.5	kd	CGS001-2548	GAA	Glycosidases			
5065	-60.53	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
5066	-60.54	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
5067	-60.55	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5068	-60.55	kd	CGS001-122618	PLD4	-			
5069	-60.62	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
5070	-60.65	oe	ccsbBroad304_07178	ZFP112	-			
5071	-60.69	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
5072	-60.74	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
5073	-60.75	cc		V type ATPases LOF	-			
5074	-60.75	oe	ccsbBroad304_07101	TSC2	-			
5075	-60.77	oe	ccsbBroad304_00789	HSBP1	-			
5076	-60.82	oe	ccsbBroad304_02173	ATG5	-			
5077	-60.85	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
5078	-60.85	kd	CGS001-10252	SPRY1	-			
5079	-60.98	kd	CGS001-472	ATM	Other PIKK family kinases			
5080	-61.01	kd	CGS001-9354	UBE4A	U-box domain containing			
5081	-61.11	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
5082	-61.13	oe	ccsbBroad304_14291	GDPD5	-			
5083	-61.19	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
5084	-61.2	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
5085	-61.2	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
5086	-61.22	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
5087	-61.22	kd	CGS001-2878	GPX3	-			
5088	-61.24	oe	ccsbBroad304_00070	ANXA5	Annexins			
5089	-61.29	kd	CGS001-4046	LSP1	-			
5090	-61.42	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
5091	-61.44	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
5092	-61.44	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
5093	-61.49	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
5094	-61.52	oe	ccsbBroad304_01401	RIT1	-			
5095	-61.53	oe	ccsbBroad304_02702	MSRB2	-			
5096	-61.66	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
5097	-61.73	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
5098	-61.77	kd	CGS001-4664	NAB1	-			
5099	-61.89	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
5100	-61.91	kd	CGS001-79733	E2F8	-			
5101	-61.96	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
5102	-61.98	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
5103	-62.01	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
5104	-62.12	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
5105	-62.16	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
5106	-62.17	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
5107	-62.23	kd	CGS001-1514	CTSL1	-			
5108	-62.27	cc		Serotonin receptor antagonist	-			
5109	-62.28	oe	ccsbBroad304_02109	XPR1	-			
5110	-62.34	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
5111	-62.35	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
5112	-62.37	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
5113	-62.39	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
5114	-62.4	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
5115	-62.45	oe	ccsbBroad304_06278	GK	Glycerol kinases			
5116	-62.48	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
5117	-62.48	kd	CGS001-6189	RPS3A	S ribosomal proteins			
5118	-62.48	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
5119	-62.54	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
5120	-62.57	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
5121	-62.58	oe	ccsbBroad304_01398	RHEB	-			
5122	-62.61	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5123	-62.63	cc		Non Homologous End Joining LOF	-			
5124	-62.65	kd	CGS001-4507	MTAP	-			
5125	-62.67	kd	CGS001-84547	PGBD1	-			
5126	-62.71	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
5127	-62.8	kd	CGS001-27035	NOX1	-			
5128	-62.83	kd	CGS001-5160	PDHA1	-			
5129	-62.84	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
5130	-62.85	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
5131	-62.88	oe	ccsbBroad304_06538	LSP1	-			
5132	-62.89	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
5133	-62.91	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
5134	-62.94	cc		Protein synthesis inhibitor	-			
5135	-62.96	kd	CGS001-4907	NT5E	Adenosine turnover			
5136	-63.1	kd	CGS001-4547	MTTP	-			
5137	-63.13	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
5138	-63.2	oe	ccsbBroad304_01379	RBBP6	-			
5139	-63.23	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
5140	-63.26	oe	ccsbBroad304_06225	FTH1	-			
5141	-63.27	kd	CGS001-1499	CTNNB1	Catenins			
5142	-63.36	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
5143	-63.4	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
5144	-63.44	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
5145	-63.48	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
5146	-63.51	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
5147	-63.52	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
5148	-63.55	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
5149	-63.58	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
5150	-63.6	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
5151	-63.62	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
5152	-63.63	kd	CGS001-9375	TM9SF2	-			
5153	-63.67	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
5154	-63.67	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
5155	-63.68	kd	CGS001-6197	RPS6KA3	RSK subfamily			
5156	-63.77	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
5157	-63.86	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
5158	-63.89	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
5159	-63.89	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
5160	-63.9	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
5161	-63.93	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
5162	-64.01	oe	ccsbBroad304_00032	ADSL	-			
5163	-64.05	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
5164	-64.05	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
5165	-64.06	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
5166	-64.09	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
5167	-64.1	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
5168	-64.12	kd	CGS001-2783	GNB2	WD repeat domain containing			
5169	-64.2	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
5170	-64.24	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
5171	-64.24	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
5172	-64.27	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
5173	-64.29	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5174	-64.3	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5175	-64.33	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
5176	-64.39	kd	CGS001-9805	SCRN1	-			
5177	-64.42	oe	ccsbBroad304_03554	NAT10	-			
5178	-64.47	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
5179	-64.51	cc		Angiotensin receptor antagonist	-			
5180	-64.52	kd	CGS001-5909	RAP1GAP	-			
5181	-64.54	kd	CGS001-79073	TMEM109	-			
5182	-64.57	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
5183	-64.58	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
5184	-64.62	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5185	-64.67	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
5186	-64.71	kd	CGS001-23475	QPRT	-			
5187	-64.71	kd	CGS001-5479	PPIB	-			
5188	-64.72	kd	CGS001-54681	P4HTM	-			
5189	-64.76	oe	ccsbBroad304_02815	SSBP2	-			
5190	-64.78	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
5191	-64.83	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
5192	-64.85	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5193	-64.92	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
5194	-65.01	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
5195	-65.01	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5196	-65.07	oe	ccsbBroad304_02506	EBP	-			
5197	-65.2	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
5198	-65.26	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
5199	-65.28	kd	CGS001-6827	SUPT4H1	-			
5200	-65.3	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
5201	-65.3	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
5202	-65.32	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
5203	-65.33	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
5204	-65.35	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
5205	-65.36	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
5206	-65.36	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
5207	-65.39	kd	CGS001-3956	LGALS1	Endogenous ligands			
5208	-65.39	kd	CGS001-335	APOA1	Apolipoproteins			
5209	-65.4	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
5210	-65.41	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5211	-65.41	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
5212	-65.42	oe	ccsbBroad304_00490	EIF4EBP1	-			
5213	-65.44	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
5214	-65.48	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
5215	-65.53	kd	CGS001-506	ATP5B	ATPases / F-type			
5216	-65.54	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
5217	-65.59	kd	CGS001-890	CCNA2	-			
5218	-65.6	oe	ccsbBroad304_09396	TIRAP	-			
5219	-65.6	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5220	-65.65	kd	CGS001-5686	PSMA5	Proteasome subunits			
5221	-65.74	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
5222	-65.78	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5223	-65.81	kd	CGS001-11230	PRAF2	-			
5224	-65.91	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
5225	-65.96	oe	ccsbBroad304_07632	PROCR	CD molecules			
5226	-66.01	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
5227	-66.03	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
5228	-66.04	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
5229	-66.08	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5230	-66.09	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
5231	-66.1	cc		Ribosomal 40s Subunit LOF	-			
5232	-66.11	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
5233	-66.14	kd	CGS001-375	ARF1	ADP-ribosylation factors			
5234	-66.19	oe	ccsbBroad304_06126	TSC22D3	-			
5235	-66.19	kd	CGS001-475	ATOX1	-			
5236	-66.22	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
5237	-66.29	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
5238	-66.35	oe	ccsbBroad304_00162	BIK	-			
5239	-66.4	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
5240	-66.52	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
5241	-66.54	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
5242	-66.61	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
5243	-66.62	kd	CGS001-771	CA12	Carbonic anhydrases			
5244	-66.65	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
5245	-66.67	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
5246	-66.73	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
5247	-66.75	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5248	-66.78	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
5249	-66.83	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
5250	-66.83	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
5251	-66.85	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5252	-66.86	oe	ccsbBroad304_10240	CROT	-			
5253	-66.91	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
5254	-66.94	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
5255	-66.95	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5256	-66.97	oe	ccsbBroad304_06777	PRNP	CD molecules			
5257	-66.98	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
5258	-67	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
5259	-67.01	oe	ccsbBroad304_03037	TMEM97	-			
5260	-67.13	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
5261	-67.25	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
5262	-67.28	kd	CGS001-11140	CDC37	-			
5263	-67.29	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
5264	-67.33	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
5265	-67.43	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
5266	-67.47	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
5267	-67.5	cc		Tricyclic antidepressant	-			
5268	-67.5	kd	CGS001-2864	FFAR1	Fatty acid receptors			
5269	-67.61	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
5270	-67.69	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
5271	-67.69	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
5272	-67.88	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
5273	-67.92	cc		AHSP Pathway LOF	-			
5274	-67.97	kd	CGS001-10607	TBL3	WD repeat domain containing			
5275	-68.02	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
5276	-68.09	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
5277	-68.13	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
5278	-68.17	cc		Glycogen synthase kinase inhibitor	-			
5279	-68.19	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
5280	-68.23	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
5281	-68.25	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
5282	-68.33	kd	CGS001-64786	TBC1D15	-			
5283	-68.38	oe	ccsbBroad304_03618	OSGEP	-			
5284	-68.5	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
5285	-68.53	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5286	-68.54	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
5287	-68.55	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
5288	-68.56	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
5289	-68.57	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
5290	-68.62	kd	CGS001-57721	METTL14	-			
5291	-68.63	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
5292	-68.65	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
5293	-68.7	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
5294	-68.71	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5295	-68.72	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
5296	-68.72	kd	CGS001-3029	HAGH	-			
5297	-68.73	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
5298	-68.73	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
5299	-68.77	kd	CGS001-3482	IGF2R	CD molecules			
5300	-68.78	oe	ccsbBroad304_01663	TFF2	-			
5301	-68.81	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
5302	-68.89	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
5303	-68.9	oe	ccsbBroad304_08152	PSAT1	-			
5304	-68.9	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
5305	-68.9	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
5306	-68.92	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
5307	-68.94	kd	CGS001-5827	PXMP2	-			
5308	-69	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
5309	-69.08	kd	CGS001-6016	RIT1	-			
5310	-69.1	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
5311	-69.11	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5312	-69.13	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
5313	-69.16	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
5314	-69.2	kd	CGS001-2287	FKBP3	-			
5315	-69.21	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
5316	-69.21	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
5317	-69.23	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
5318	-69.26	kd	CGS001-3832	KIF11	Kinesins			
5319	-69.33	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
5320	-69.45	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5321	-69.45	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
5322	-69.52	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5323	-69.57	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
5324	-69.59	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
5325	-69.59	kd	CGS001-5581	PRKCE	Eta subfamily			
5326	-69.6	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
5327	-69.63	kd	CGS001-2615	LRRC32	-			
5328	-69.64	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
5329	-69.66	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
5330	-69.68	kd	CGS001-2004	ELK3	ETS Transcription Factors			
5331	-69.72	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
5332	-69.79	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
5333	-69.8	oe	ccsbBroad304_06651	NOV	-			
5334	-69.81	cc		FGFR inhibitor	-			
5335	-69.86	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
5336	-69.88	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
5337	-69.88	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
5338	-69.95	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
5339	-69.95	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
5340	-69.98	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
5341	-70.05	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
5342	-70.06	oe	ccsbBroad304_06993	SRD5A1	-			
5343	-70.15	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
5344	-70.23	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
5345	-70.26	oe	ccsbBroad304_00665	GOT1	-			
5346	-70.26	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
5347	-70.27	oe	ccsbBroad304_05749	A2M	-			
5348	-70.27	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
5349	-70.37	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
5350	-70.38	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
5351	-70.47	oe	ccsbBroad304_02092	SYNGR3	-			
5352	-70.48	kd	CGS001-28960	DCPS	-			
5353	-70.52	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
5354	-70.56	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
5355	-70.58	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
5356	-70.58	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
5357	-70.65	kd	CGS001-3575	IL7R	IL-2 receptor family			
5358	-70.66	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
5359	-70.67	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
5360	-70.67	kd	CGS001-85004	RERG	-			
5361	-70.73	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
5362	-70.74	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
5363	-70.74	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
5364	-70.75	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
5365	-70.76	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
5366	-70.8	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
5367	-70.81	oe	ccsbBroad304_10487	BPHL	-			
5368	-70.81	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
5369	-70.82	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
5370	-70.83	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
5371	-70.84	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5372	-70.91	kd	CGS001-1131	CHRM3	Cholinergic receptors			
5373	-70.94	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
5374	-70.94	kd	CGS001-2852	GPER	-			
5375	-71.17	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
5376	-71.27	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
5377	-71.27	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
5378	-71.27	kd	CGS001-10472	ZNF238	-			
5379	-71.36	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
5380	-71.47	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
5381	-71.5	oe	ccsbBroad304_06134	ECH1	-			
5382	-71.51	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
5383	-71.52	oe	ccsbBroad304_01716	TSN	-			
5384	-71.53	kd	CGS001-2697	GJA1	Ion channels / Gap junction proteins (connexins)			
5385	-71.59	oe	ccsbBroad304_02533	NOXA1	-			
5386	-71.61	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
5387	-71.63	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
5388	-71.66	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
5389	-71.67	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
5390	-71.68	oe	ccsbBroad304_09095	PUS7L	-			
5391	-71.68	kd	CGS001-6793	STK10	SLK subfamily			
5392	-71.75	oe	ccsbBroad304_00728	HBE1	-			
5393	-71.75	kd	CGS001-9784	SNX17	Sorting nexins			
5394	-71.76	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
5395	-71.78	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5396	-71.85	kd	CGS001-7056	THBD	CD molecules			
5397	-71.87	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
5398	-71.91	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
5399	-71.92	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
5400	-71.93	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
5401	-71.95	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
5402	-71.95	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
5403	-72	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
5404	-72.09	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
5405	-72.28	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
5406	-72.36	kd	CGS001-1831	TSC22D3	-			
5407	-72.37	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
5408	-72.48	kd	CGS001-3932	LCK	Src family			
5409	-72.55	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
5410	-72.57	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
5411	-72.58	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
5412	-72.62	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
5413	-72.62	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
5414	-72.67	kd	CGS001-112858	TP53RK	Bud32 family			
5415	-72.68	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
5416	-72.7	oe	ccsbBroad304_08879	CASD1	-			
5417	-72.71	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
5418	-72.72	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
5419	-72.79	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
5420	-72.79	kd	CGS001-10682	EBP	-			
5421	-72.81	kd	CGS001-2235	FECH	-			
5422	-72.82	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
5423	-72.83	oe	ccsbBroad304_00147	BAG1	-			
5424	-72.86	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
5425	-72.9	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
5426	-72.92	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
5427	-72.94	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
5428	-73.01	kd	CGS001-213	ALB	-			
5429	-73.1	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
5430	-73.14	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
5431	-73.16	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
5432	-73.16	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
5433	-73.18	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
5434	-73.18	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
5435	-73.24	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
5436	-73.25	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5437	-73.26	kd	CGS001-595	CCND1	-			
5438	-73.29	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
5439	-73.31	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
5440	-73.32	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
5441	-73.39	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
5442	-73.42	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
5443	-73.42	oe	ccsbBroad304_07832	XPO7	Exportins			
5444	-73.45	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
5445	-73.46	kd	CGS001-5660	PSAP	Endogenous ligands			
5446	-73.48	kd	CGS001-2760	GM2A	-			
5447	-73.52	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
5448	-73.54	oe	ccsbBroad304_06133	TOR1A	-			
5449	-73.56	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
5450	-73.59	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
5451	-73.62	oe	ccsbBroad304_03533	CDCA8	-			
5452	-73.62	kd	CGS001-25824	PRDX5	-			
5453	-73.64	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
5454	-73.68	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
5455	-73.82	kd	CGS001-2277	FIGF	-			
5456	-73.83	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
5457	-73.89	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
5458	-73.96	oe	ccsbBroad304_06828	PYCR1	-			
5459	-73.98	kd	CGS001-4074	M6PR	-			
5460	-73.99	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
5461	-74	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
5462	-74.01	oe	ccsbBroad304_00617	GBA	-			
5463	-74.03	oe	ccsbBroad304_10212	GRHL3	-			
5464	-74.11	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5465	-74.11	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
5466	-74.11	kd	CGS001-638	BIK	-			
5467	-74.17	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
5468	-74.19	kd	CGS001-11329	STK38	NDR family			
5469	-74.2	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
5470	-74.21	oe	ccsbBroad304_06234	G6PC	-			
5471	-74.29	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
5472	-74.32	oe	ccsbBroad304_02372	SPRY1	-			
5473	-74.34	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
5474	-74.37	oe	ccsbBroad304_00645	GCLM	-			
5475	-74.38	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
5476	-74.41	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
5477	-74.41	kd	CGS001-6277	S100A6	EF-hand domain containing			
5478	-74.42	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
5479	-74.44	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
5480	-74.48	kd	CGS001-9	NAT1	-			
5481	-74.49	kd	CGS001-51022	GLRX2	-			
5482	-74.5	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
5483	-74.6	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
5484	-74.62	kd	CGS001-29946	SERTAD3	-			
5485	-74.62	kd	CGS001-776	CACNA1D	Calcium channel subunits			
5486	-74.67	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
5487	-74.68	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
5488	-74.7	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
5489	-74.71	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
5490	-74.71	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
5491	-74.81	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
5492	-74.82	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
5493	-74.85	oe	ccsbBroad304_02990	LYPD3	-			
5494	-74.92	kd	CGS001-4864	NPC1	-			
5495	-74.93	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
5496	-74.97	cc		PKC inhibitor	-			
5497	-75.03	kd	CGS001-1155	TBCB	-			
5498	-75.05	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
5499	-75.06	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
5500	-75.12	kd	CGS001-55165	CEP55	-			
5501	-75.13	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
5502	-75.17	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
5503	-75.19	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
5504	-75.25	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
5505	-75.27	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
5506	-75.39	kd	CGS001-5887	RAD23B	-			
5507	-75.39	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
5508	-75.42	cc		P38 MAPK inhibitor	-			
5509	-75.43	cc		Aminoacyl tRNA synthetases class II LOF	-			
5510	-75.43	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
5511	-75.49	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
5512	-75.5	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
5513	-75.53	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
5514	-75.59	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
5515	-75.61	cc		Aurora kinase inhibitor	-			
5516	-75.68	oe	ccsbBroad304_01347	RAD1	-			
5517	-75.73	oe	ccsbBroad304_02243	DLGAP5	-			
5518	-75.78	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
5519	-75.78	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
5520	-75.91	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
5521	-76	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
5522	-76.01	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
5523	-76.04	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
5524	-76.08	oe	ccsbBroad304_02671	ECD	-			
5525	-76.12	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
5526	-76.14	cc		Dihydrofolate reductase inhibitor	-			
5527	-76.14	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
5528	-76.15	kd	CGS001-2000	ELF4	ETS Transcription Factors			
5529	-76.16	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
5530	-76.26	kd	CGS001-6599	SMARCC1	-			
5531	-76.26	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
5532	-76.27	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
5533	-76.27	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
5534	-76.29	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
5535	-76.32	oe	ccsbBroad304_04490	RSPH1	-			
5536	-76.32	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
5537	-76.33	kd	CGS001-382	ARF6	ADP-ribosylation factors			
5538	-76.38	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
5539	-76.39	oe	ccsbBroad304_05590	NOTCH2NL	-			
5540	-76.41	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
5541	-76.45	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
5542	-76.5	oe	ccsbBroad304_08802	ELAC2	-			
5543	-76.53	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
5544	-76.54	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
5545	-76.61	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
5546	-76.64	kd	CGS001-5932	RBBP8	-			
5547	-76.66	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
5548	-76.71	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
5549	-76.73	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
5550	-76.76	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
5551	-76.78	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
5552	-76.79	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
5553	-76.85	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
5554	-76.87	oe	ccsbBroad304_07337	TAF1B	-			
5555	-76.87	kd	CGS001-2030	SLC29A1	SLC29 family			
5556	-76.88	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5557	-76.89	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
5558	-76.93	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5559	-76.93	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5560	-77.01	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
5561	-77.05	kd	CGS001-7913	DEK	-			
5562	-77.06	cc		MTOR inhibitor	-			
5563	-77.08	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5564	-77.09	kd	CGS001-9221	NOLC1	-			
5565	-77.1	kd	CGS001-9710	KIAA0355	-			
5566	-77.11	oe	ccsbBroad304_02219	MORF4L2	-			
5567	-77.15	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
5568	-77.17	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
5569	-77.17	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
5570	-77.21	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
5571	-77.22	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
5572	-77.25	kd	CGS001-4200	ME2	-			
5573	-77.32	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
5574	-77.33	kd	CGS001-5618	PRLR	Prolactin receptor family			
5575	-77.34	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
5576	-77.38	oe	ccsbBroad304_00975	MAT2A	-			
5577	-77.41	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
5578	-77.41	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
5579	-77.44	kd	CGS001-9655	SOCS5	SH2 domain containing			
5580	-77.49	kd	CGS001-2534	FYN	Src family			
5581	-77.5	kd	CGS001-3030	HADHA	-			
5582	-77.51	kd	CGS001-840	CASP7	Caspases			
5583	-77.53	oe	ccsbBroad304_02592	KIF2C	Kinesins			
5584	-77.58	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
5585	-77.65	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
5586	-77.65	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
5587	-77.7	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5588	-77.74	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
5589	-77.74	kd	CGS001-9641	IKBKE	IKK family			
5590	-77.76	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
5591	-77.82	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
5592	-77.86	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
5593	-77.91	kd	CGS001-302	ANXA2	Annexins			
5594	-77.91	kd	CGS001-47	ACLY	-			
5595	-77.98	kd	CGS001-5019	OXCT1	-			
5596	-77.98	kd	CGS001-9131	AIFM1	-			
5597	-78	oe	ccsbBroad304_02218	IKBKE	IKK family			
5598	-78.02	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
5599	-78.03	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
5600	-78.05	oe	ccsbBroad304_01211	PKM2	-			
5601	-78.12	kd	CGS001-1062	CENPE	Kinesins			
5602	-78.13	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
5603	-78.19	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
5604	-78.22	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
5605	-78.23	oe	ccsbBroad304_14011	PAPSS1	-			
5606	-78.25	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
5607	-78.28	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5608	-78.28	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
5609	-78.29	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
5610	-78.3	oe	ccsbBroad304_07889	QPRT	-			
5611	-78.31	kd	CGS001-64858	DCLRE1B	-			
5612	-78.33	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
5613	-78.36	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5614	-78.36	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
5615	-78.41	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
5616	-78.47	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
5617	-78.48	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
5618	-78.51	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
5619	-78.51	kd	CGS001-79139	DERL1	-			
5620	-78.53	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
5621	-78.55	kd	CGS001-139135	PASD1	-			
5622	-78.56	kd	CGS001-5361	PLXNA1	Plexins			
5623	-78.6	oe	ccsbBroad304_01769	VEGFB	-			
5624	-78.6	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
5625	-78.61	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
5626	-78.63	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
5627	-78.64	kd	CGS001-58477	SRPRB	-			
5628	-78.64	oe	ccsbBroad304_02605	PAPD7	-			
5629	-78.68	oe	ccsbBroad304_06094	DFFA	-			
5630	-78.68	kd	CGS001-2673	GFPT1	-			
5631	-78.7	kd	CGS001-10285	SMNDC1	Tudor domain containing			
5632	-78.75	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
5633	-78.78	kd	CGS001-6194	RPS6	S ribosomal proteins			
5634	-78.83	kd	CGS001-55038	CDCA4	-			
5635	-78.87	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
5636	-78.89	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
5637	-78.9	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
5638	-78.97	cc		GABA receptor antagonist	-			
5639	-79.06	oe	ccsbBroad304_02313	ACTR3	-			
5640	-79.06	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
5641	-79.22	oe	ccsbBroad304_01556	SMARCB1	-			
5642	-79.22	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
5643	-79.24	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
5644	-79.27	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
5645	-79.3	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
5646	-79.34	oe	ccsbBroad304_06985	SORD	-			
5647	-79.37	kd	CGS001-1632	ECI1	-			
5648	-79.51	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
5649	-79.56	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
5650	-79.57	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
5651	-79.63	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
5652	-79.65	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
5653	-79.67	kd	CGS001-5613	PRKX	Protein kinase A			
5654	-79.71	kd	CGS001-9687	GREB1	-			
5655	-79.79	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
5656	-79.81	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
5657	-79.9	kd	CGS001-51172	NAGPA	-			
5658	-79.91	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5659	-79.91	kd	CGS001-3845	KRAS	RAS subfamily			
5660	-80	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
5661	-80.02	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
5662	-80.02	kd	CGS001-54512	EXOSC4	-			
5663	-80.15	oe	ccsbBroad304_00657	GNG4	-			
5664	-80.22	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
5665	-80.23	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
5666	-80.24	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
5667	-80.31	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
5668	-80.33	oe	ccsbBroad304_03122	RHOD	-			
5669	-80.37	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
5670	-80.46	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
5671	-80.53	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5672	-80.53	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
5673	-80.55	kd	CGS001-51447	IP6K2	-			
5674	-80.56	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
5675	-80.6	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
5676	-80.61	oe	ccsbBroad304_07600	NSA2	-			
5677	-80.61	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
5678	-80.63	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
5679	-80.65	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
5680	-80.66	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
5681	-80.66	kd	CGS001-345611	IRGM	-			
5682	-80.68	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
5683	-80.7	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
5684	-80.75	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
5685	-80.86	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
5686	-80.89	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
5687	-80.97	oe	ccsbBroad304_02278	THRAP3	-			
5688	-80.98	oe	ccsbBroad304_03264	UBAP1	-			
5689	-80.99	kd	CGS001-204851	HIPK1	HIPK subfamily			
5690	-81.04	oe	ccsbBroad304_01519	SET	-			
5691	-81.08	cc		Trace amine receptors LOF	-			
5692	-81.08	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
5693	-81.12	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
5694	-81.12	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
5695	-81.16	kd	CGS001-6119	RPA3	-			
5696	-81.18	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
5697	-81.31	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
5698	-81.32	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
5699	-81.37	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
5700	-81.4	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
5701	-81.41	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
5702	-81.44	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
5703	-81.45	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
5704	-81.46	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
5705	-81.52	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
5706	-81.53	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
5707	-81.54	kd	CGS001-8536	CAMK1	CAMK1 family			
5708	-81.63	cc		SRC inhibitor	-			
5709	-81.68	oe	ccsbBroad304_01641	TAF13	-			
5710	-81.69	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
5711	-81.75	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
5712	-81.75	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
5713	-81.75	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
5714	-81.79	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
5715	-81.79	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
5716	-81.79	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
5717	-81.86	kd	CGS001-9791	PTDSS1	-			
5718	-81.88	kd	CGS001-388650	FAM69A	-			
5719	-81.99	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
5720	-82	oe	ccsbBroad304_09503	KLHDC9	-			
5721	-82.01	kd	CGS001-4849	CNOT3	-			
5722	-82.02	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
5723	-82.03	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
5724	-82.05	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
5725	-82.05	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
5726	-82.1	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
5727	-82.12	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
5728	-82.14	kd	CGS001-10587	TXNRD2	-			
5729	-82.17	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
5730	-82.18	oe	ccsbBroad304_01951	BLZF1	-			
5731	-82.19	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
5732	-82.27	cc		EGFR inhibitor	-			
5733	-82.28	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
5734	-82.33	kd	CGS001-11041	B3GNT1	-			
5735	-82.35	kd	CGS001-10427	SEC24B	-			
5736	-82.46	kd	CGS001-3163	HMOX2	Haem oxygenase			
5737	-82.5	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
5738	-82.55	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
5739	-82.59	oe	ccsbBroad304_00962	SMAD4	SMADs			
5740	-82.61	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
5741	-82.65	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
5742	-82.66	oe	ccsbBroad304_00985	MCL1	-			
5743	-82.69	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
5744	-82.76	kd	CGS001-3481	IGF2	-			
5745	-82.79	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
5746	-82.8	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
5747	-82.82	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
5748	-82.85	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
5749	-82.86	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
5750	-82.91	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
5751	-82.97	kd	CGS001-6188	RPS3	S ribosomal proteins			
5752	-83.05	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
5753	-83.06	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
5754	-83.08	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5755	-83.09	oe	ccsbBroad304_07219	CDC7	CDC7 family			
5756	-83.16	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
5757	-83.17	kd	CGS001-4175	MCM6	-			
5758	-83.18	oe	ccsbBroad304_07820	SNW1	-			
5759	-83.22	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
5760	-83.26	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5761	-83.26	kd	CGS001-7003	TEAD1	-			
5762	-83.27	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5763	-83.28	kd	CGS001-9140	ATG12	-			
5764	-83.29	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
5765	-83.3	kd	CGS001-84722	PSRC1	-			
5766	-83.32	oe	ccsbBroad304_00174	BRAF	RAF family			
5767	-83.33	kd	CGS001-25885	POLR1A	RNA polymerase subunits			
5768	-83.33	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
5769	-83.41	kd	CGS001-439	ASNA1	-			
5770	-83.43	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5771	-83.47	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
5772	-83.49	oe	ccsbBroad304_01577	SOD1	-			
5773	-83.5	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
5774	-83.55	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
5775	-83.56	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
5776	-83.62	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
5777	-83.67	kd	CGS001-54805	CNNM2	-			
5778	-83.69	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
5779	-83.69	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
5780	-83.7	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
5781	-83.7	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
5782	-83.74	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
5783	-83.74	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
5784	-83.76	oe	ccsbBroad304_07651	HEXIM1	-			
5785	-83.84	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5786	-83.87	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
5787	-83.9	oe	ccsbBroad304_03950	ATG3	-			
5788	-83.91	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
5789	-83.92	oe	ccsbBroad304_01632	SYPL1	-			
5790	-83.93	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5791	-83.96	cc		Norepinephrine reuptake inhibitor	-			
5792	-83.96	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
5793	-83.98	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
5794	-84.01	cc		Cyclins LOF	-			
5795	-84.04	oe	ccsbBroad304_07197	PDHX	-			
5796	-84.06	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
5797	-84.1	cc		General transcription factors group 2 LOF	-			
5798	-84.11	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
5799	-84.11	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
5800	-84.15	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
5801	-84.16	oe	ccsbBroad304_06836	RAD23B	-			
5802	-84.18	kd	CGS001-55662	HIF1AN	-			
5803	-84.25	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5804	-84.29	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
5805	-84.3	kd	CGS001-8681	JMJD7-PLA2G4B	-			
5806	-84.33	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
5807	-84.37	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
5808	-84.38	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
5809	-84.39	kd	CGS001-59343	SENP2	-			
5810	-84.4	oe	ccsbBroad304_07363	AIFM1	-			
5811	-84.42	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
5812	-84.44	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
5813	-84.49	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
5814	-84.5	cc		RAF inhibitor	-			
5815	-84.51	kd	CGS001-6208	RPS14	S ribosomal proteins			
5816	-84.52	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
5817	-84.53	oe	ccsbBroad304_03746	CDC42SE1	-			
5818	-84.54	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
5819	-84.55	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
5820	-84.56	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
5821	-84.58	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
5822	-84.59	cc		Purinergic receptors P2Y GOF	-			
5823	-84.59	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
5824	-84.6	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
5825	-84.61	oe	ccsbBroad304_04406	PLA2G12B	-			
5826	-84.63	kd	CGS001-57149	LYRM1	LYR motif containing			
5827	-84.63	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
5828	-84.75	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
5829	-84.76	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
5830	-84.8	cc		Serpin peptidase inhibitors LOF	-			
5831	-84.81	kd	CGS001-7485	WRB	-			
5832	-84.81	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
5833	-84.88	kd	CGS001-54106	TLR9	Toll-like receptor family			
5834	-84.97	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
5835	-84.99	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
5836	-85	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
5837	-85.01	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
5838	-85.02	oe	ccsbBroad304_08645	BCCIP	-			
5839	-85.02	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
5840	-85.04	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
5841	-85.04	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
5842	-85.08	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
5843	-85.08	kd	CGS001-1662	DDX10	DEAD-boxes			
5844	-85.14	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
5845	-85.14	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
5846	-85.19	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5847	-85.21	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
5848	-85.24	oe	ccsbBroad304_00690	GRN	-			
5849	-85.25	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
5850	-85.26	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
5851	-85.35	cc		Calmodulin antagonist	-			
5852	-85.36	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
5853	-85.36	oe	ccsbBroad304_06386	HNMT	-			
5854	-85.38	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
5855	-85.46	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
5856	-85.46	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
5857	-85.47	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
5858	-85.52	oe	ccsbBroad304_06525	LIPA	-			
5859	-85.56	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
5860	-85.57	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
5861	-85.57	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
5862	-85.57	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
5863	-85.58	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
5864	-85.59	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
5865	-85.66	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
5866	-85.68	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
5867	-85.74	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
5868	-85.77	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
5869	-85.86	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
5870	-85.87	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
5871	-85.96	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
5872	-86.07	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
5873	-86.1	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
5874	-86.11	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
5875	-86.13	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
5876	-86.15	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
5877	-86.15	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
5878	-86.18	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
5879	-86.18	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
5880	-86.24	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
5881	-86.24	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
5882	-86.3	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
5883	-86.31	oe	ccsbBroad304_06066	CTSL1	-			
5884	-86.31	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
5885	-86.33	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
5886	-86.38	kd	CGS001-8807	IL18RAP	CD molecules			
5887	-86.42	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
5888	-86.43	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
5889	-86.47	cc		Phospholipases GOF	-			
5890	-86.5	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
5891	-86.51	kd	CGS001-8996	NOL3	-			
5892	-86.53	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
5893	-86.54	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
5894	-86.58	kd	CGS001-1504	CTRB1	-			
5895	-86.59	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
5896	-86.6	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
5897	-86.64	kd	CGS001-9183	ZW10	-			
5898	-86.69	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
5899	-86.72	cp	BRD-K10065684	dantron	Laxative			Laxative
5900	-86.76	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
5901	-86.79	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
5902	-86.81	kd	CGS001-23210	JMJD6	-			
5903	-86.84	cc		Potassium channel activator	-			
5904	-86.85	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
5905	-86.86	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
5906	-86.91	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
5907	-86.96	kd	CGS001-2885	GRB2	SH2 domain containing			
5908	-87	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
5909	-87	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
5910	-87.01	oe	ccsbBroad304_05439	O3FAR1	-			
5911	-87.01	oe	ccsbBroad304_00883	ISG20	-			
5912	-87.1	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
5913	-87.13	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
5914	-87.15	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
5915	-87.23	oe	ccsbBroad304_06639	NFYB	-			
5916	-87.23	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
5917	-87.23	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
5918	-87.27	oe	ccsbBroad304_07727	LIAS	-			
5919	-87.32	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
5920	-87.34	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
5921	-87.37	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
5922	-87.39	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
5923	-87.4	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
5924	-87.43	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
5925	-87.5	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5926	-87.59	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5927	-87.61	oe	ccsbBroad304_02398	LANCL1	-			
5928	-87.62	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
5929	-87.63	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
5930	-87.64	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
5931	-87.68	kd	CGS001-56005	C19ORF10	-			
5932	-87.71	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
5933	-87.72	kd	CGS001-11019	LIAS	-			
5934	-87.73	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5935	-87.75	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
5936	-87.75	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
5937	-87.81	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
5938	-87.81	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
5939	-87.82	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
5940	-87.83	oe	ccsbBroad304_07071	TKT	-			
5941	-87.84	cc		NFkB pathway inhibitor	-			
5942	-87.84	kd	CGS001-9612	NCOR2	-			
5943	-87.87	cc		Kruppel like transcription factors LOF	-			
5944	-87.87	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
5945	-87.91	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
5946	-87.94	kd	CGS001-5411	PNN	-			
5947	-87.97	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
5948	-88.13	kd	CGS001-5900	RALGDS	-			
5949	-88.14	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
5950	-88.16	oe	ccsbBroad304_05890	BHMT	-			
5951	-88.16	kd	CGS001-3265	HRAS	RAS subfamily			
5952	-88.26	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
5953	-88.31	kd	CGS001-7018	TF	-			
5954	-88.32	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
5955	-88.32	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
5956	-88.34	kd	CGS001-2919	CXCL1	Endogenous ligands			
5957	-88.37	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
5958	-88.37	kd	CGS001-27161	EIF2C2	-			
5959	-88.38	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
5960	-88.48	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
5961	-88.48	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
5962	-88.48	kd	CGS001-8870	IER3	-			
5963	-88.49	kd	CGS001-2274	FHL2	-			
5964	-88.5	kd	CGS001-10652	YKT6	-			
5965	-88.51	oe	ccsbBroad304_06888	RPN1	-			
5966	-88.52	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
5967	-88.52	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
5968	-88.6	oe	ccsbBroad304_01052	MYB	-			
5969	-88.6	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
5970	-88.61	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5971	-88.63	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
5972	-88.63	kd	CGS001-54438	GFOD1	-			
5973	-88.65	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
5974	-88.68	oe	ccsbBroad304_07088	TP53	-			
5975	-88.68	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
5976	-88.74	oe	ccsbBroad304_00398	CTSL2	-			
5977	-88.74	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
5978	-88.75	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5979	-88.77	kd	CGS001-6500	SKP1	-			
5980	-88.79	kd	CGS001-3821	KLRC1	CD molecules			
5981	-88.88	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
5982	-88.9	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
5983	-88.92	kd	CGS001-8226	HDHD1	-			
5984	-88.95	oe	ccsbBroad304_06837	RAF1	RAF family			
5985	-88.95	kd	CGS001-55793	FAM63A	-			
5986	-88.97	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
5987	-88.98	kd	CGS001-10775	POP4	-			
5988	-88.99	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
5989	-89.02	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5990	-89.03	kd	CGS001-23192	ATG4B	Aut2 peptidase			
5991	-89.05	oe	ccsbBroad304_02738	RRS1	-			
5992	-89.07	kd	CGS001-10765	KDM5B	Histone demethylases			
5993	-89.16	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
5994	-89.16	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
5995	-89.2	oe	ccsbBroad304_05980	CDKN1B	-			
5996	-89.21	oe	ccsbBroad304_08137	HOOK2	-			
5997	-89.21	kd	CGS001-1072	CFL1	-			
5998	-89.22	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
5999	-89.22	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6000	-89.26	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
6001	-89.27	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
6002	-89.28	kd	CGS001-23118	TAB2	-			
6003	-89.34	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
6004	-89.37	oe	ccsbBroad304_07490	SCRN1	-			
6005	-89.4	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
6006	-89.52	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
6007	-89.53	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
6008	-89.54	kd	CGS001-11267	SNF8	-			
6009	-89.55	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
6010	-89.55	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
6011	-89.58	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
6012	-89.58	kd	CGS001-85442	KNDC1	-			
6013	-89.62	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
6014	-89.62	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
6015	-89.63	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
6016	-89.73	oe	ccsbBroad304_00888	ITPK1	-			
6017	-89.73	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
6018	-89.73	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6019	-89.74	oe	ccsbBroad304_02596	KDELR3	-			
6020	-89.75	oe	ccsbBroad304_07217	AXIN2	-			
6021	-89.75	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
6022	-89.76	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
6023	-89.78	oe	ccsbBroad304_03961	SMURF2	-			
6024	-89.78	kd	CGS001-9738	CCP110	-			
6025	-89.81	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
6026	-89.82	kd	CGS001-7054	TH	Amino acid hydroxylases			
6027	-89.85	kd	CGS001-11315	PARK7	Parkinson disease			
6028	-89.86	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
6029	-89.92	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6030	-89.93	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
6031	-89.97	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
6032	-89.97	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6033	-89.99	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
6034	-90.02	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
6035	-90.05	oe	ccsbBroad304_06952	SKP1	-			
6036	-90.05	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
6037	-90.07	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
6038	-90.07	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
6039	-90.07	kd	CGS001-8837	CFLAR	Endogenous ligands			
6040	-90.07	kd	CGS001-857	CAV1	-			
6041	-90.08	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
6042	-90.09	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
6043	-90.11	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
6044	-90.12	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
6045	-90.12	oe	ccsbBroad304_08797	FASTKD5	-			
6046	-90.14	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
6047	-90.15	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
6048	-90.17	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
6049	-90.2	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
6050	-90.21	kd	CGS001-1312	COMT	Catecholamine turnover			
6051	-90.23	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
6052	-90.29	oe	ccsbBroad304_02581	ASCC3	-			
6053	-90.32	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
6054	-90.34	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
6055	-90.34	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
6056	-90.34	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
6057	-90.39	oe	ccsbBroad304_02509	GMEB1	-			
6058	-90.39	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
6059	-90.41	kd	CGS001-124535	HSF5	-			
6060	-90.42	oe	ccsbBroad304_00223	CASP9	Caspases			
6061	-90.47	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
6062	-90.48	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
6063	-90.49	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
6064	-90.52	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
6065	-90.52	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
6066	-90.55	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
6067	-90.58	cc		HIF activator	-			
6068	-90.65	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
6069	-90.66	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
6070	-90.76	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
6071	-90.81	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
6072	-90.83	cc		CCK receptor antagonist	-			
6073	-90.84	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
6074	-90.87	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
6075	-90.87	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
6076	-90.89	kd	CGS001-3516	RBPJ	-			
6077	-90.89	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
6078	-90.9	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6079	-90.9	oe	ccsbBroad304_00152	BCAT2	-			
6080	-90.91	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
6081	-90.92	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
6082	-90.93	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
6083	-90.96	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
6084	-90.97	kd	CGS001-2767	GNA11	-			
6085	-90.97	kd	CGS001-23242	COBL	-			
6086	-91.04	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
6087	-91.04	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
6088	-91.06	kd	CGS001-7358	UGDH	-			
6089	-91.07	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
6090	-91.09	cc		IKK inhibitor	-			
6091	-91.1	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
6092	-91.12	oe	ccsbBroad304_00956	LYZ	-			
6093	-91.12	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
6094	-91.17	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
6095	-91.19	kd	CGS001-27097	TAF5L	WD repeat domain containing			
6096	-91.23	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
6097	-91.24	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
6098	-91.28	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
6099	-91.3	oe	ccsbBroad304_02890	SYF2	-			
6100	-91.3	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
6101	-91.38	kd	CGS001-10873	ME3	-			
6102	-91.4	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
6103	-91.43	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
6104	-91.43	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6105	-91.47	kd	CGS001-5230	PGK1	-			
6106	-91.49	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
6107	-91.49	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
6108	-91.5	kd	CGS001-4782	NFIC	-			
6109	-91.51	kd	CGS001-51053	GMNN	-			
6110	-91.55	oe	ccsbBroad304_01658	PRDX2	-			
6111	-91.56	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
6112	-91.57	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
6113	-91.57	kd	CGS001-23386	NUDCD3	-			
6114	-91.59	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
6115	-91.6	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
6116	-91.6	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
6117	-91.62	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
6118	-91.62	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
6119	-91.67	kd	CGS001-1854	DUT	-			
6120	-91.68	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
6121	-91.68	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
6122	-91.7	oe	ccsbBroad304_05931	CAPG	-			
6123	-91.7	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
6124	-91.72	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
6125	-91.74	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
6126	-91.74	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
6127	-91.75	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
6128	-91.77	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
6129	-91.77	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
6130	-91.83	cc		Proteasome inhibitor	-			
6131	-91.84	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
6132	-91.84	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
6133	-91.85	oe	ccsbBroad304_03928	RRAGC	-			
6134	-91.85	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6135	-91.85	kd	CGS001-256281	NUDT14	Nudix motif containing			
6136	-91.88	kd	CGS001-51293	CD320	CD molecules			
6137	-91.91	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
6138	-91.95	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
6139	-91.96	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
6140	-91.98	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
6141	-91.99	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
6142	-91.99	kd	CGS001-8575	PRKRA	-			
6143	-92.04	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
6144	-92.23	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
6145	-92.24	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
6146	-92.24	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
6147	-92.29	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6148	-92.29	oe	ccsbBroad304_01165	PDK1	-			
6149	-92.29	kd	CGS001-9688	NUP93	-			
6150	-92.32	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
6151	-92.35	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
6152	-92.37	kd	CGS001-6184	RPN1	-			
6153	-92.41	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
6154	-92.44	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
6155	-92.45	oe	ccsbBroad304_01662	TFDP2	-			
6156	-92.47	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
6157	-92.47	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
6158	-92.47	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
6159	-92.48	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
6160	-92.5	oe	ccsbBroad304_06916	SCP2	-			
6161	-92.51	kd	CGS001-10923	SUB1	-			
6162	-92.53	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
6163	-92.53	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
6164	-92.54	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
6165	-92.54	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
6166	-92.57	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
6167	-92.59	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
6168	-92.6	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
6169	-92.6	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
6170	-92.61	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
6171	-92.63	oe	ccsbBroad304_03056	MCTS1	-			
6172	-92.63	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
6173	-92.64	cc		PARP inhibitor	-			
6174	-92.69	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
6175	-92.72	oe	ccsbBroad304_07118	UGDH	-			
6176	-92.73	kd	CGS001-5824	PEX19	-			
6177	-92.79	oe	ccsbBroad304_03420	TOLLIP	-			
6178	-92.8	oe	ccsbBroad304_08480	PNPO	-			
6179	-92.83	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
6180	-92.84	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
6181	-92.85	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
6182	-92.9	oe	ccsbBroad304_03479	YTHDF1	-			
6183	-92.9	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
6184	-92.9	kd	CGS001-5264	PHYH	-			
6185	-92.91	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
6186	-92.96	oe	ccsbBroad304_02276	MVP	-			
6187	-92.99	oe	ccsbBroad304_00085	APRT	-			
6188	-93	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
6189	-93.03	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
6190	-93.03	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
6191	-93.04	kd	CGS001-3572	IL6ST	IL-6 receptor family			
6192	-93.06	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
6193	-93.08	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
6194	-93.1	oe	ccsbBroad304_07145	ZFP161	-			
6195	-93.11	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
6196	-93.13	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
6197	-93.13	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
6198	-93.15	kd	CGS001-55634	ZNF673	-			
6199	-93.15	kd	CGS001-51720	UIMC1	-			
6200	-93.16	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
6201	-93.17	oe	ccsbBroad304_08023	EIF2C1	-			
6202	-93.17	kd	CGS001-2781	GNAZ	-			
6203	-93.18	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
6204	-93.19	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6205	-93.2	kd	CGS001-226	ALDOA	-			
6206	-93.22	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
6207	-93.22	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
6208	-93.26	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
6209	-93.28	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
6210	-93.28	kd	CGS001-3383	ICAM1	CD molecules			
6211	-93.29	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
6212	-93.3	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
6213	-93.3	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
6214	-93.31	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
6215	-93.32	oe	ccsbBroad304_05963	CD44	CD molecules			
6216	-93.33	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
6217	-93.35	kd	CGS001-31	ACACA	Carboxylases			
6218	-93.36	oe	ccsbBroad304_02285	MED6	-			
6219	-93.36	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
6220	-93.36	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
6221	-93.37	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
6222	-93.37	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
6223	-93.41	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
6224	-93.41	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
6225	-93.44	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
6226	-93.45	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
6227	-93.48	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
6228	-93.5	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
6229	-93.51	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
6230	-93.53	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
6231	-93.53	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
6232	-93.54	kd	CGS001-1999	ELF3	ETS Transcription Factors			
6233	-93.55	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
6234	-93.58	kd	CGS001-5357	PLS1	EF-hand domain containing			
6235	-93.63	kd	CGS001-25797	QPCT	Aminopeptidase Y			
6236	-93.65	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
6237	-93.67	oe	ccsbBroad304_06820	PTS	-			
6238	-93.68	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
6239	-93.69	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
6240	-93.7	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
6241	-93.73	cc		Glucocorticoid receptor agonist	-			
6242	-93.75	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
6243	-93.79	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
6244	-93.82	oe	ccsbBroad304_03658	DCP1A	-			
6245	-93.82	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
6246	-93.83	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
6247	-93.84	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
6248	-93.84	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
6249	-93.84	cp	BRD-K53220666	trimetozine	Sedative			Sedative
6250	-93.88	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
6251	-93.91	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6252	-93.92	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
6253	-93.92	kd	CGS001-9441	MED26	-			
6254	-93.98	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
6255	-93.98	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
6256	-94.04	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
6257	-94.05	oe	ccsbBroad304_00486	EFNB2	Ephrins			
6258	-94.06	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
6259	-94.09	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
6260	-94.11	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
6261	-94.11	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
6262	-94.16	kd	CGS001-819	CAMLG	-			
6263	-94.18	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
6264	-94.19	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
6265	-94.2	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
6266	-94.21	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
6267	-94.23	oe	ccsbBroad304_02197	VPS26A	-			
6268	-94.23	oe	ccsbBroad304_07208	NRIP1	-			
6269	-94.23	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
6270	-94.24	kd	CGS001-7486	WRN	-			
6271	-94.27	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
6272	-94.27	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
6273	-94.29	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
6274	-94.31	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
6275	-94.32	cc		HDAC inhibitor	-			
6276	-94.32	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
6277	-94.34	oe	ccsbBroad304_00394	CTSD	Cathepsins			
6278	-94.34	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
6279	-94.34	kd	CGS001-10538	BATF	basic leucine zipper proteins			
6280	-94.34	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
6281	-94.41	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
6282	-94.44	oe	ccsbBroad304_01948	GAS7	-			
6283	-94.45	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
6284	-94.47	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
6285	-94.52	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
6286	-94.57	kd	CGS001-1201	CLN3	-			
6287	-94.58	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6288	-94.59	oe	ccsbBroad304_02569	BTG3	-			
6289	-94.59	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
6290	-94.6	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
6291	-94.63	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6292	-94.63	kd	CGS001-11044	PAPD7	-			
6293	-94.64	cc		Canonical high mobility group proteins LOF	-			
6294	-94.67	oe	ccsbBroad304_07598	PEMT	-			
6295	-94.72	kd	CGS001-222546	RFX6	-			
6296	-94.72	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6297	-94.75	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
6298	-94.77	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
6299	-94.8	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
6300	-94.81	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
6301	-94.81	kd	CGS001-10797	MTHFD2	-			
6302	-94.84	oe	ccsbBroad304_11405	UBE3C	-			
6303	-94.84	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
6304	-94.85	oe	ccsbBroad304_02405	TFG	-			
6305	-94.88	kd	CGS001-2810	SFN	-			
6306	-94.91	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
6307	-94.92	kd	CGS001-375133	PI4KAP2	-			
6308	-94.93	oe	ccsbBroad304_03858	SRPRB	-			
6309	-95	cc		Nucleophosmin inhibitor	-			
6310	-95.04	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
6311	-95.05	cc		PKA inhibitor	-			
6312	-95.08	kd	CGS001-7040	TGFB1	Endogenous ligands			
6313	-95.09	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
6314	-95.1	kd	CGS001-54881	TEX10	-			
6315	-95.11	kd	CGS001-9275	BCL7B	-			
6316	-95.14	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6317	-95.19	kd	CGS001-190	NR0B1	DAX-like receptors			
6318	-95.24	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
6319	-95.25	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
6320	-95.25	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
6321	-95.26	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
6322	-95.28	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
6323	-95.3	kd	CGS001-85480	TSLP	-			
6324	-95.31	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
6325	-95.34	cc		PRD class homeoboxes and psudogenes LOF	-			
6326	-95.35	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
6327	-95.35	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
6328	-95.36	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6329	-95.37	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
6330	-95.39	oe	ccsbBroad304_00238	CCNE1	-			
6331	-95.4	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
6332	-95.41	kd	CGS001-10943	MSL3	-			
6333	-95.42	cc		PKC activator	-			
6334	-95.42	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
6335	-95.47	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
6336	-95.48	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
6337	-95.49	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
6338	-95.5	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
6339	-95.5	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
6340	-95.51	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
6341	-95.53	kd	CGS001-23076	RRP1B	-			
6342	-95.54	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
6343	-95.54	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
6344	-95.55	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
6345	-95.55	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
6346	-95.58	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
6347	-95.64	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
6348	-95.64	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
6349	-95.68	oe	ccsbBroad304_02677	PDAP1	-			
6350	-95.68	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6351	-95.68	kd	CGS001-9637	FEZ2	-			
6352	-95.7	oe	ccsbBroad304_01034	MSH2	-			
6353	-95.7	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
6354	-95.71	oe	ccsbBroad304_01593	SRP14	-			
6355	-95.71	kd	CGS001-10898	CPSF4	-			
6356	-95.71	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
6357	-95.75	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
6358	-95.81	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
6359	-95.83	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
6360	-95.83	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
6361	-95.83	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6362	-95.87	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
6363	-95.93	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
6364	-95.94	cc		Structural maintenance of chromosomes proteins LOF	-			
6365	-95.94	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
6366	-95.96	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
6367	-95.98	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
6368	-95.98	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
6369	-95.99	kd	CGS001-10318	TNIP1	-			
6370	-96	oe	ccsbBroad304_00316	CKS1B	-			
6371	-96.01	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
6372	-96.01	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
6373	-96.02	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
6374	-96.09	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
6375	-96.09	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6376	-96.1	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6377	-96.12	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
6378	-96.12	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
6379	-96.18	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
6380	-96.18	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6381	-96.19	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
6382	-96.19	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
6383	-96.19	kd	CGS001-9451	EIF2AK3	PEK subfamily			
6384	-96.2	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
6385	-96.2	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
6386	-96.22	cc		Cell Cycle Inhibition GOF	-			
6387	-96.23	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
6388	-96.23	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
6389	-96.25	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
6390	-96.25	kd	CGS001-5194	PEX13	-			
6391	-96.26	kd	CGS001-5920	RARRES3	-			
6392	-96.27	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
6393	-96.27	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
6394	-96.29	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
6395	-96.29	kd	CGS001-1287	COL4A5	Collagens			
6396	-96.36	oe	ccsbBroad304_02840	PISD	Decarboxylases			
6397	-96.38	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
6398	-96.39	kd	CGS001-23510	KCTD2	-			
6399	-96.4	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
6400	-96.4	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
6401	-96.43	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6402	-96.43	kd	CGS001-84971	ATG4D	-			
6403	-96.45	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
6404	-96.48	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
6405	-96.48	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
6406	-96.48	kd	CGS001-1827	RCAN1	-			
6407	-96.49	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
6408	-96.49	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
6409	-96.49	kd	CGS001-4998	ORC1	ATPases / AAA-type			
6410	-96.54	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
6411	-96.54	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
6412	-96.56	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
6413	-96.59	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
6414	-96.6	kd	CGS001-9455	HOMER2	-			
6415	-96.64	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
6416	-96.65	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
6417	-96.66	oe	ccsbBroad304_02789	ADAT1	-			
6418	-96.66	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
6419	-96.68	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
6420	-96.69	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
6421	-96.7	kd	CGS001-6646	SOAT1	-			
6422	-96.7	kd	CGS001-1655	DDX5	DEAD-boxes			
6423	-96.73	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
6424	-96.74	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
6425	-96.78	oe	ccsbBroad304_08878	METTL4	-			
6426	-96.81	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
6427	-96.81	kd	CGS001-4905	NSF	ATPases / AAA-type			
6428	-96.82	oe	ccsbBroad304_00282	CDKN1A	-			
6429	-96.84	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
6430	-96.84	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
6431	-96.85	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
6432	-96.87	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
6433	-96.89	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
6434	-96.9	cc		Dopamine receptor antagonist	-			
6435	-96.93	oe	ccsbBroad304_07884	RYBP	-			
6436	-96.94	cc		CDK inhibitor	-			
6437	-96.96	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
6438	-96.98	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
6439	-96.99	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
6440	-96.99	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
6441	-97	oe	ccsbBroad304_01001	MEST	-			
6442	-97.02	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
6443	-97.03	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
6444	-97.03	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
6445	-97.04	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
6446	-97.05	oe	ccsbBroad304_01174	PEX13	-			
6447	-97.05	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
6448	-97.07	kd	CGS001-83999	KREMEN1	-			
6449	-97.09	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
6450	-97.12	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
6451	-97.13	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
6452	-97.17	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
6453	-97.17	kd	CGS001-7077	TIMP2	-			
6454	-97.19	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
6455	-97.19	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
6456	-97.27	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
6457	-97.27	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
6458	-97.28	oe	ccsbBroad304_09756	PAQR7	-			
6459	-97.3	oe	ccsbBroad304_06095	DFFB	-			
6460	-97.31	kd	CGS001-2232	FDXR	-			
6461	-97.32	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
6462	-97.36	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
6463	-97.37	oe	ccsbBroad304_13813	ARAF	RAF family			
6464	-97.37	kd	CGS001-23753	SDF2L1	-			
6465	-97.38	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6466	-97.39	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
6467	-97.4	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
6468	-97.43	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
6469	-97.44	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
6470	-97.45	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
6471	-97.49	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
6472	-97.49	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
6473	-97.51	cc		T-type calcium channel blocker	-			
6474	-97.51	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
6475	-97.51	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
6476	-97.53	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
6477	-97.53	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
6478	-97.54	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
6479	-97.57	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
6480	-97.58	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6481	-97.58	oe	ccsbBroad304_09054	EGFL8	-			
6482	-97.58	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6483	-97.59	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
6484	-97.6	kd	CGS001-6464	SHC1	SH2 domain containing			
6485	-97.6	kd	CGS001-126823	KLHDC9	-			
6486	-97.62	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
6487	-97.62	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
6488	-97.63	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
6489	-97.63	oe	ccsbBroad304_03570	QRSL1	-			
6490	-97.64	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
6491	-97.64	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
6492	-97.65	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
6493	-97.67	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
6494	-97.67	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
6495	-97.68	kd	CGS001-30001	ERO1L	-			
6496	-97.69	kd	CGS001-84619	ZGPAT	G patch domain containing			
6497	-97.69	kd	CGS001-2966	GTF2H2	General transcription factors			
6498	-97.71	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
6499	-97.72	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
6500	-97.74	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
6501	-97.76	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
6502	-97.77	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
6503	-97.78	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
6504	-97.79	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
6505	-97.8	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
6506	-97.8	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6507	-97.83	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
6508	-97.84	oe	ccsbBroad304_00420	DAP	-			
6509	-97.84	kd	CGS001-56993	TOMM22	-			
6510	-97.86	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
6511	-97.86	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
6512	-97.87	oe	ccsbBroad304_01222	PLP2	-			
6513	-97.87	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
6514	-97.89	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
6515	-97.89	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6516	-97.9	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
6517	-97.9	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6518	-97.91	kd	CGS001-23196	FAM120A	-			
6519	-97.93	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
6520	-97.95	cc		Minor histocompatibility antigens LOF	-			
6521	-97.96	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
6522	-97.96	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
6523	-97.96	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
6524	-97.97	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
6525	-97.97	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
6526	-97.97	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
6527	-97.99	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
6528	-97.99	kd	CGS001-125965	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
6529	-98	kd	CGS001-121599	SPIC	ETS Transcription Factors			
6530	-98.02	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
6531	-98.04	kd	CGS001-10523	CHERP	G patch domain containing			
6532	-98.05	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
6533	-98.06	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
6534	-98.06	kd	CGS001-10641	NPRL2	-			
6535	-98.07	kd	CGS001-54555	DDX49	DEAD-boxes			
6536	-98.09	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6537	-98.1	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
6538	-98.1	kd	CGS001-51741	WWOX	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6539	-98.11	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6540	-98.11	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
6541	-98.12	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
6542	-98.12	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
6543	-98.13	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
6544	-98.13	kd	CGS001-7840	ALMS1	-			
6545	-98.16	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
6546	-98.17	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6547	-98.17	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6548	-98.18	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
6549	-98.19	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
6550	-98.19	kd	CGS001-23075	SWAP70	EF-hand domain containing			
6551	-98.2	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
6552	-98.2	kd	CGS001-3920	LAMP2	CD molecules			
6553	-98.2	kd	CGS001-400	ARL1	ADP-ribosylation factors			
6554	-98.21	cc		Ribonucleotide reductase inhibitor	-			
6555	-98.23	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6556	-98.25	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
6557	-98.25	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
6558	-98.25	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6559	-98.25	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
6560	-98.25	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
6561	-98.25	kd	CGS001-637	BID	Endogenous ligands			
6562	-98.28	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
6563	-98.29	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
6564	-98.3	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
6565	-98.3	kd	CGS001-10128	LRPPRC	-			
6566	-98.31	kd	CGS001-1070	CETN3	EF-hand domain containing			
6567	-98.32	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
6568	-98.32	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6569	-98.34	oe	ccsbBroad304_02801	CASP14	Caspases			
6570	-98.34	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
6571	-98.35	kd	CGS001-23081	KDM4C	Histone demethylases			
6572	-98.35	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
6573	-98.38	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
6574	-98.39	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
6575	-98.39	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
6576	-98.39	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
6577	-98.39	kd	CGS001-1152	CKB	-			
6578	-98.41	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
6579	-98.42	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
6580	-98.43	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
6581	-98.44	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
6582	-98.44	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
6583	-98.44	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
6584	-98.45	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
6585	-98.47	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
6586	-98.48	kd	CGS001-25987	TSKU	-			
6587	-98.49	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
6588	-98.49	kd	CGS001-5162	PDHB	-			
6589	-98.52	oe	ccsbBroad304_08694	TBX20	T-boxes			
6590	-98.53	oe	ccsbBroad304_02487	TXNIP	-			
6591	-98.53	kd	CGS001-23499	MACF1	EF-hand domain containing			
6592	-98.54	kd	CGS001-3985	LIMK2	LIMK subfamily			
6593	-98.55	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
6594	-98.56	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
6595	-98.56	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
6596	-98.57	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
6597	-98.58	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
6598	-98.59	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
6599	-98.63	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
6600	-98.64	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
6601	-98.67	oe	ccsbBroad304_08952	E2F8	-			
6602	-98.69	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
6603	-98.69	kd	CGS001-2313	FLI1	ETS Transcription Factors			
6604	-98.7	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
6605	-98.7	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6606	-98.72	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
6607	-98.73	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
6608	-98.73	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
6609	-98.74	oe	ccsbBroad304_02340	SORBS3	-			
6610	-98.75	kd	CGS001-2147	F2	Endogenous ligands			
6611	-98.76	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
6612	-98.78	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
6613	-98.78	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
6614	-98.78	kd	CGS001-11243	PMF1	-			
6615	-98.8	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
6616	-98.82	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
6617	-98.82	oe	ccsbBroad304_04190	CCDC92	-			
6618	-98.82	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
6619	-98.85	cc		DNA polymerase inhibitor	-			
6620	-98.87	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
6621	-98.88	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
6622	-98.88	oe	ccsbBroad304_01664	TGFA	-			
6623	-98.88	oe	ccsbBroad304_01147	PC	Carboxylases			
6624	-98.89	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6625	-98.89	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
6626	-98.89	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
6627	-98.9	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
6628	-98.9	kd	CGS001-84365	MKI67IP	-			
6629	-98.91	kd	CGS001-8508	NIPSNAP1	-			
6630	-98.92	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6631	-98.92	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
6632	-98.92	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
6633	-98.92	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
6634	-98.94	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
6635	-98.94	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6636	-98.94	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
6637	-98.95	oe	ccsbBroad304_00118	ATIC	-			
6638	-98.96	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
6639	-98.97	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
6640	-98.97	kd	CGS001-5914	RARA	Retinoic acid receptors			
6641	-98.98	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
6642	-99	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
6643	-99	kd	CGS001-4090	SMAD5	SMADs			
6644	-99	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
6645	-99	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
6646	-99.01	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
6647	-99.01	kd	CGS001-5292	PIM1	PIM family			
6648	-99.01	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
6649	-99.03	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
6650	-99.04	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
6651	-99.05	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
6652	-99.06	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
6653	-99.06	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
6654	-99.06	kd	CGS001-9467	SH3BP5	-			
6655	-99.06	kd	CGS001-347736	NME9	-			
6656	-99.07	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
6657	-99.07	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
6658	-99.07	kd	CGS001-7316	UBC	-			
6659	-99.09	kd	CGS001-5763	PTMS	-			
6660	-99.11	oe	ccsbBroad304_01351	PEX19	-			
6661	-99.12	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
6662	-99.12	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
6663	-99.13	oe	ccsbBroad304_06845	RARRES3	-			
6664	-99.13	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
6665	-99.13	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
6666	-99.13	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
6667	-99.15	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6668	-99.15	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
6669	-99.15	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
6670	-99.16	cc		MCM family LOF	-			
6671	-99.19	oe	ccsbBroad304_02415	TUBB3	Tubulins			
6672	-99.19	kd	CGS001-383	ARG1	Arginase			
6673	-99.2	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
6674	-99.2	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
6675	-99.22	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
6676	-99.23	oe	ccsbBroad304_00794	HSF1	-			
6677	-99.25	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
6678	-99.25	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
6679	-99.26	oe	ccsbBroad304_02788	PRAME	-			
6680	-99.26	kd	CGS001-8727	CTNNAL1	Catenins			
6681	-99.27	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
6682	-99.27	oe	ccsbBroad304_06992	SRC	Src family			
6683	-99.28	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
6684	-99.29	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6685	-99.29	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
6686	-99.31	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
6687	-99.31	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
6688	-99.31	kd	CGS001-6397	SEC14L1	-			
6689	-99.31	kd	CGS001-9512	PMPCB	-			
6690	-99.32	oe	ccsbBroad304_00106	ARRB1	-			
6691	-99.32	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
6692	-99.33	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
6693	-99.34	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
6694	-99.34	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
6695	-99.35	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
6696	-99.35	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
6697	-99.35	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
6698	-99.35	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
6699	-99.35	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6700	-99.35	kd	CGS001-81539	SLC38A1	System A-like transporters			
6701	-99.35	kd	CGS001-1490	CTGF	-			
6702	-99.37	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
6703	-99.37	oe	ccsbBroad304_02676	PHB2	-			
6704	-99.37	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
6705	-99.37	kd	CGS001-847	CAT	-			
6706	-99.39	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
6707	-99.4	kd	CGS001-310	ANXA7	Annexins			
6708	-99.41	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
6709	-99.41	oe	ccsbBroad304_07124	UROD	-			
6710	-99.41	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
6711	-99.41	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
6712	-99.41	kd	CGS001-10491	CRTAP	-			
6713	-99.43	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
6714	-99.43	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
6715	-99.43	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
6716	-99.43	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
6717	-99.44	oe	ccsbBroad304_02032	TSC22D1	-			
6718	-99.44	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
6719	-99.45	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
6720	-99.46	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6721	-99.49	oe	ccsbBroad304_01038	MSRA	-			
6722	-99.49	oe	ccsbBroad304_05894	BLVRA	-			
6723	-99.5	cc		Sirtuins GOF	-			
6724	-99.5	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
6725	-99.5	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
6726	-99.5	kd	CGS001-6810	STX4	-			
6727	-99.5	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
6728	-99.5	oe	ccsbBroad304_00551	FECH	-			
6729	-99.51	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
6730	-99.52	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
6731	-99.52	kd	CGS001-79902	NUP85	-			
6732	-99.53	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
6733	-99.53	kd	CGS001-55486	PARL	-			
6734	-99.53	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
6735	-99.54	oe	ccsbBroad304_09254	PAQR8	-			
6736	-99.54	kd	CGS001-2967	GTF2H3	General transcription factors			
6737	-99.56	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
6738	-99.56	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
6739	-99.56	kd	CGS001-6275	S100A4	EF-hand domain containing			
6740	-99.56	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6741	-99.57	oe	ccsbBroad304_01672	TIMP2	-			
6742	-99.57	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
6743	-99.57	kd	CGS001-2100	ESR2	Estrogen receptors			
6744	-99.58	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6745	-99.59	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
6746	-99.59	kd	CGS001-54386	TERF2IP	-			
6747	-99.59	kd	CGS001-64121	RRAGC	-			
6748	-99.6	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
6749	-99.6	kd	CGS001-55746	NUP133	-			
6750	-99.61	kd	CGS001-7100	TLR5	Toll-like receptor family			
6751	-99.61	kd	CGS001-25842	ASF1A	-			
6752	-99.62	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
6753	-99.63	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
6754	-99.63	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
6755	-99.63	kd	CGS001-5573	PRKAR1A	Protein kinase A			
6756	-99.63	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
6757	-99.63	kd	CGS001-1738	DLD	-			
6758	-99.63	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
6759	-99.65	cc		DNA dependent protein kinase inhibitor	-			
6760	-99.65	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
6761	-99.65	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6762	-99.65	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
6763	-99.66	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
6764	-99.66	oe	ccsbBroad304_00518	ETFA	-			
6765	-99.66	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
6766	-99.68	cc		SMAD family LOF	-			
6767	-99.68	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
6768	-99.68	kd	CGS001-5423	POLB	DNA polymerases			
6769	-99.68	kd	CGS001-54541	DDIT4	-			
6770	-99.69	kd	CGS001-5881	RAC3	Endogenous ligands			
6771	-99.7	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
6772	-99.71	oe	ccsbBroad304_06286	GLUL	-			
6773	-99.71	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
6774	-99.71	kd	CGS001-8741	TNFSF13	CD molecules			
6775	-99.71	kd	CGS001-4174	MCM5	-			
6776	-99.71	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
6777	-99.72	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
6778	-99.72	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
6779	-99.73	oe	ccsbBroad304_07466	VGLL4	-			
6780	-99.73	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
6781	-99.73	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
6782	-99.73	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
6783	-99.73	kd	CGS001-8800	PEX11A	-			
6784	-99.74	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6785	-99.75	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
6786	-99.75	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
6787	-99.75	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
6788	-99.75	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
6789	-99.75	kd	CGS001-5033	P4HA1	-			
6790	-99.75	kd	CGS001-4199	ME1	-			
6791	-99.75	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
6792	-99.76	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
6793	-99.76	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
6794	-99.76	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
6795	-99.76	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
6796	-99.77	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
6797	-99.78	oe	ccsbBroad304_03310	LCMT1	-			
6798	-99.78	oe	ccsbBroad304_02230	HERPUD1	-			
6799	-99.78	kd	CGS001-6772	STAT1	SH2 domain containing			
6800	-99.78	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
6801	-99.78	kd	CGS001-4351	MPI	-			
6802	-99.79	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
6803	-99.79	oe	ccsbBroad304_01304	PSEN1	Presenilin			
6804	-99.79	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
6805	-99.79	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
6806	-99.79	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
6807	-99.79	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
6808	-99.8	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
6809	-99.81	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
6810	-99.81	oe	ccsbBroad304_00529	F3	CD molecules			
6811	-99.81	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
6812	-99.81	kd	CGS001-4089	SMAD4	SMADs			
6813	-99.81	kd	CGS001-4893	NRAS	RAS subfamily			
6814	-99.81	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
6815	-99.82	oe	ccsbBroad304_07861	COBL	-			
6816	-99.82	oe	ccsbBroad304_00313	TBCB	-			
6817	-99.82	oe	ccsbBroad304_06789	PSEN2	Presenilin			
6818	-99.82	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
6819	-99.82	kd	CGS001-10673	TNFSF13B	CD molecules			
6820	-99.82	kd	CGS001-7082	TJP1	-			
6821	-99.82	kd	CGS001-8780	RIOK3	RIO3 subfamily			
6822	-99.82	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
6823	-99.83	cc		Nucleoporin LOF	-			
6824	-99.84	oe	ccsbBroad304_00184	C2	Complement system			
6825	-99.84	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
6826	-99.84	kd	CGS001-3476	IGBP1	-			
6827	-99.84	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
6828	-99.84	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
6829	-99.84	kd	CGS001-64170	CARD9	-			
6830	-99.84	kd	CGS001-84890	ADO	-			
6831	-99.85	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
6832	-99.85	oe	ccsbBroad304_06103	DMD	-			
6833	-99.85	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
6834	-99.85	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
6835	-99.85	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
6836	-99.85	kd	CGS001-2879	GPX4	-			
6837	-99.85	kd	CGS001-25	ABL1	Abl family			
6838	-99.86	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
6839	-99.87	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
6840	-99.87	oe	ccsbBroad304_06494	KLRC1	CD molecules			
6841	-99.87	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6842	-99.87	kd	CGS001-51750	RTEL1	-			
6843	-99.87	kd	CGS001-284119	PTRF	-			
6844	-99.87	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
6845	-99.87	kd	CGS001-55163	PNPO	-			
6846	-99.87	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
6847	-99.87	kd	CGS001-158	ADSL	-			
6848	-99.88	oe	ccsbBroad304_00376	CSK	Csk family			
6849	-99.88	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
6850	-99.88	kd	CGS001-7128	TNFAIP3	OTU domain containing			
6851	-99.88	kd	CGS001-22930	RAB3GAP1	-			
6852	-99.88	kd	CGS001-79071	ELOVL6	-			
6853	-99.88	kd	CGS001-55526	DHTKD1	-			
6854	-99.9	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
6855	-99.9	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
6856	-99.9	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
6857	-99.9	kd	CGS001-5108	PCM1	-			
6858	-99.9	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
6859	-99.9	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
6860	-99.9	kd	CGS001-842	CASP9	Caspases			
6861	-99.9	kd	CGS001-673	BRAF	RAF family			
6862	-99.91	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
6863	-99.91	oe	ccsbBroad304_02271	LPGAT1	-			
6864	-99.91	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
6865	-99.91	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6866	-99.91	kd	CGS001-5829	PXN	-			
6867	-99.91	kd	CGS001-11014	KDELR2	-			
6868	-99.91	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
6869	-99.93	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
6870	-99.93	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
6871	-99.93	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
6872	-99.93	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
6873	-99.93	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
6874	-99.93	kd	CGS001-55278	QRSL1	-			
6875	-99.93	kd	CGS001-81533	ITFG1	-			
6876	-99.93	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
6877	-99.94	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
6878	-99.94	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
6879	-99.94	oe	ccsbBroad304_07724	KDELR2	-			
6880	-99.94	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
6881	-99.94	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6882	-99.94	kd	CGS001-10180	RBM6	G patch domain containing			
6883	-99.94	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
6884	-99.94	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
6885	-99.94	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
6886	-99.94	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
6887	-99.95	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
6888	-99.95	oe	ccsbBroad304_01584	SPARC	-			
6889	-99.95	oe	ccsbBroad304_06464	ITGB2	Integrins			
6890	-99.96	cc		Thromboxane receptor antagonist	-			
6891	-99.96	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
6892	-99.96	oe	ccsbBroad304_05183	TXLNA	-			
6893	-99.96	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
6894	-99.96	oe	ccsbBroad304_00446	DKC1	-			
6895	-99.96	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
6896	-99.96	oe	ccsbBroad304_08840	KIF9	Kinesins			
6897	-99.96	oe	ccsbBroad304_03177	FIS1	-			
6898	-99.96	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
6899	-99.96	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
6900	-99.96	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
6901	-99.96	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
6902	-99.96	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
6903	-99.96	kd	CGS001-5580	PRKCD	Delta subfamily			
6904	-99.96	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
6905	-99.96	kd	CGS001-2160	F11	Chymotrypsin			
6906	-99.96	kd	CGS001-1163	CKS1B	-			
6907	-99.97	kd	CGS001-22933	SIRT2	Histone deacetylases			
6908	-99.97	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
6909	-99.97	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
6910	-99.97	oe	ccsbBroad304_01102	NMT1	-			
6911	-99.97	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
6912	-99.97	oe	ccsbBroad304_00038	AGL	-			
6913	-99.97	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
6914	-99.97	oe	ccsbBroad304_07506	UBAP2L	-			
6915	-99.97	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
6916	-99.97	oe	ccsbBroad304_07050	TFAP2A	-			
6917	-99.97	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
6918	-99.97	oe	ccsbBroad304_01469	RSU1	-			
6919	-99.97	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
6920	-99.97	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
6921	-99.97	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
6922	-99.97	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6923	-99.97	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
6924	-99.97	oe	ccsbBroad304_02370	HRSP12	-			
6925	-99.97	oe	ccsbBroad304_00632	GGCX	Carboxylases			
6926	-99.97	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
6927	-99.97	oe	ccsbBroad304_08392	EXOC6	-			
6928	-99.97	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
6929	-99.97	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
6930	-99.97	oe	ccsbBroad304_00146	BAD	-			
6931	-99.97	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
6932	-99.97	oe	ccsbBroad304_00077	APEX1	-			
6933	-99.97	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
6934	-99.97	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
6935	-99.97	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
6936	-99.97	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
6937	-99.97	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
6938	-99.97	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6939	-99.97	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6940	-99.97	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
6941	-99.97	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
6942	-99.97	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
6943	-99.97	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
6944	-99.97	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
6945	-99.97	kd	CGS001-7089	TLE2	WD repeat domain containing			
6946	-99.97	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
6947	-99.97	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
6948	-99.97	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
6949	-99.97	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
6950	-99.97	kd	CGS001-5255	PHKA1	-			
6951	-99.97	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
6952	-99.97	kd	CGS001-3930	LBR	Tudor domain containing			
6953	-99.97	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
6954	-99.97	kd	CGS001-3672	ITGA1	Integrins			
6955	-99.97	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
6956	-99.97	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
6957	-99.97	kd	CGS001-2821	GPI	-			
6958	-99.97	kd	CGS001-2266	FGG	Endogenous ligands			
6959	-99.97	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
6960	-99.97	kd	CGS001-23149	FCHO1	-			
6961	-99.97	kd	CGS001-1503	CTPS	-			
6962	-99.97	kd	CGS001-1399	CRKL	SH2 domain containing			
6963	-99.97	kd	CGS001-9133	CCNB2	-			
6964	-99.97	kd	CGS001-8900	CCNA1	-			
6965	-99.97	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
6966	-99.97	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
6967	-99.97	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
6968	-99.99	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
6969	-99.99	oe	ccsbBroad304_02292	BCL2L11	-			
6970	-99.99	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
6971	-99.99	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
6972	-100	kd	CGS001-56882	CDC42SE1	-			
