Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
2	100	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
3	100	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
4	99.99	cc		LIM class homeoboxes GOF	-			
5	99.97	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
6	99.97	oe	ccsbBroad304_01880	LAGE3	-			
7	99.97	oe	ccsbBroad304_02432	IFI30	-			
8	99.97	oe	ccsbBroad304_00464	DTNA	-			
9	99.97	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
10	99.97	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
11	99.97	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
12	99.97	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
13	99.97	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
14	99.97	oe	ccsbBroad304_01618	STXBP1	-			
15	99.97	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
16	99.97	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
17	99.97	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
18	99.97	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
19	99.97	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
20	99.97	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
21	99.97	oe	ccsbBroad304_00809	HUS1	-			
22	99.97	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
23	99.97	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
24	99.97	oe	ccsbBroad304_06294	GNAZ	-			
25	99.97	oe	ccsbBroad304_00515	ERH	-			
26	99.97	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
27	99.97	oe	ccsbBroad304_02551	CPSF4	-			
28	99.97	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
29	99.97	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
30	99.97	oe	ccsbBroad304_02837	BHMT2	-			
31	99.97	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
32	99.97	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
33	99.97	oe	ccsbBroad304_00036	AFP	-			
34	99.97	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
35	99.97	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
36	99.97	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
37	99.97	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
38	99.97	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
39	99.97	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
40	99.97	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
41	99.97	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
42	99.97	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
43	99.97	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
44	99.97	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
45	99.97	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
46	99.97	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
47	99.97	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
48	99.97	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
49	99.97	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
50	99.97	kd	CGS001-22954	TRIM32	-			
51	99.97	kd	CGS001-10474	TADA3	-			
52	99.97	kd	CGS001-8576	STK16	NAK family			
53	99.97	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
54	99.97	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
55	99.97	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
56	99.97	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
57	99.97	kd	CGS001-4947	OAZ2	-			
58	99.97	kd	CGS001-340371	NRBP2	NRBP family			
59	99.97	kd	CGS001-4801	NFYB	-			
60	99.97	kd	CGS001-9833	MELK	MELK subfamily			
61	99.97	kd	CGS001-3690	ITGB3	Integrins			
62	99.97	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
63	99.97	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
64	99.97	kd	CGS001-2771	GNAI2	-			
65	99.97	kd	CGS001-2770	GNAI1	-			
66	99.97	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
67	99.97	kd	CGS001-1606	DGKA	EF-hand domain containing			
68	99.97	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
69	99.97	kd	CGS001-84433	CARD11	-			
70	99.97	kd	CGS001-701	BUB1B	Bub family			
71	99.97	kd	CGS001-27241	BBS9	-			
72	99.97	kd	CGS001-328	APEX1	-			
73	99.97	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
74	99.97	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
75	99.96	oe	ccsbBroad304_02653	PRAF2	-			
76	99.96	oe	ccsbBroad304_02443	HAX1	-			
77	99.96	oe	ccsbBroad304_00170	BNIP1	-			
78	99.96	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
79	99.96	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
80	99.96	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
81	99.96	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
82	99.96	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
83	99.96	kd	CGS001-10670	RRAGA	-			
84	99.96	kd	CGS001-5992	RFX4	-			
85	99.96	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
86	99.96	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
87	99.96	kd	CGS001-1786	DNMT1	Methyltransferases			
88	99.96	kd	CGS001-79947	DHDDS	-			
89	99.94	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
90	99.94	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
91	99.94	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
92	99.94	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
93	99.94	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
94	99.94	kd	CGS001-9709	HERPUD1	-			
95	99.94	kd	CGS001-717	C2	Complement system			
96	99.93	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
97	99.93	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
98	99.93	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
99	99.93	kd	CGS001-8805	TRIM24	TIF1 family			
100	99.93	kd	CGS001-89882	TPD52L3	-			
101	99.93	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
102	99.93	kd	CGS001-8720	MBTPS1	Subtilisin			
103	99.93	kd	CGS001-5653	KLK6	Chymotrypsin			
104	99.93	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
105	99.92	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
106	99.92	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
107	99.91	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
108	99.91	oe	ccsbBroad304_07029	TADA2A	-			
109	99.91	oe	ccsbBroad304_00615	GAPDH	-			
110	99.91	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
111	99.91	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
112	99.91	oe	ccsbBroad304_01872	DGCR14	-			
113	99.91	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
114	99.91	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
115	99.91	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
116	99.91	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
117	99.91	kd	CGS001-7079	TIMP4	-			
118	99.9	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
119	99.9	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
120	99.9	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
121	99.9	oe	ccsbBroad304_06518	LDHA	-			
122	99.9	oe	ccsbBroad304_00795	HSF2	-			
123	99.9	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
124	99.9	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
125	99.9	kd	CGS001-10289	EIF1B	-			
126	99.9	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
127	99.89	oe	ccsbBroad304_00709	GUK1	-			
128	99.89	kd	CGS001-665	BNIP3L	-			
129	99.88	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
130	99.88	oe	ccsbBroad304_07080	TM7SF2	-			
131	99.88	oe	ccsbBroad304_00986	MCM2	-			
132	99.88	kd	CGS001-89910	UBE3B	-			
133	99.88	kd	CGS001-9943	OXSR1	FRAY subfamily			
134	99.88	kd	CGS001-1211	CLTA	-			
135	99.87	oe	ccsbBroad304_08553	STAP2	-			
136	99.87	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
137	99.87	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
138	99.87	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
139	99.87	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
140	99.85	oe	ccsbBroad304_01651	TCF7L2	-			
141	99.85	oe	ccsbBroad304_03874	UBL5	-			
142	99.85	kd	CGS001-9374	PPT2	-			
143	99.85	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
144	99.84	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
145	99.84	oe	ccsbBroad304_01845	RDBP	-			
146	99.84	oe	ccsbBroad304_00120	ATOX1	-			
147	99.84	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
148	99.84	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
149	99.84	kd	CGS001-63948	DMRTB1	-			
150	99.82	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
151	99.82	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
152	99.82	oe	ccsbBroad304_00459	DPYD	-			
153	99.82	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
154	99.82	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
155	99.82	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
156	99.82	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
157	99.82	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
158	99.82	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
159	99.82	kd	CGS001-1374	CPT1A	-			
160	99.81	kd	CGS001-8089	YEATS4	-			
161	99.81	kd	CGS001-6347	CCL2	Chemokine ligands			
162	99.79	oe	ccsbBroad304_00957	M6PR	-			
163	99.79	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
164	99.79	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
165	99.79	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
166	99.78	oe	ccsbBroad304_08104	MED4	-			
167	99.78	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
168	99.78	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
169	99.76	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
170	99.76	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
171	99.76	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
172	99.76	oe	ccsbBroad304_06255	LRRC32	-			
173	99.75	cc		Beta-adrenergic receptor agonist	-			
174	99.75	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
175	99.75	kd	CGS001-26277	TINF2	-			
176	99.73	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
177	99.72	cc		Retinoid receptor agonist	-			
178	99.72	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
179	99.72	oe	ccsbBroad304_07890	CBX7	-			
180	99.72	oe	ccsbBroad304_00006	ACADM	-			
181	99.72	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
182	99.72	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
183	99.7	oe	ccsbBroad304_00033	ADSS	-			
184	99.7	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
185	99.7	kd	CGS001-5163	PDK1	-			
186	99.69	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
187	99.69	kd	CGS001-8649	LAMTOR3	-			
188	99.68	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
189	99.68	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
190	99.68	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
191	99.68	kd	CGS001-4610	MYCL1	-			
192	99.68	kd	CGS001-2152	F3	CD molecules			
193	99.66	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
194	99.66	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
195	99.66	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
196	99.66	kd	CGS001-55179	FAIM	-			
197	99.65	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
198	99.65	kd	CGS001-7423	VEGFB	-			
199	99.65	kd	CGS001-2037	EPB41L2	-			
200	99.63	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
201	99.63	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
202	99.63	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
203	99.63	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
204	99.62	oe	ccsbBroad304_02485	STAMBP	-			
205	99.62	oe	ccsbBroad304_06424	IFI16	-			
206	99.62	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
207	99.62	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
208	99.62	kd	CGS001-6829	SUPT5H	-			
209	99.62	kd	CGS001-391013	PLA2G2C	-			
210	99.61	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
211	99.6	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
212	99.6	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
213	99.6	kd	CGS001-4700	NDUFA6	LYR motif containing			
214	99.59	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
215	99.59	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
216	99.59	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
217	99.58	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
218	99.57	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
219	99.57	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
220	99.57	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
221	99.57	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
222	99.57	kd	CGS001-23463	ICMT	-			
223	99.57	kd	CGS001-10007	GNPDA1	-			
224	99.57	kd	CGS001-60528	ELAC2	-			
225	99.57	kd	CGS001-1488	CTBP2	-			
226	99.56	oe	ccsbBroad304_03604	ENOSF1	-			
227	99.56	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
228	99.56	oe	ccsbBroad304_02438	FAM3C	-			
229	99.56	kd	CGS001-4522	MTHFD1	-			
230	99.54	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
231	99.54	kd	CGS001-10973	ASCC3	-			
232	99.53	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
233	99.52	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
234	99.52	kd	CGS001-57804	POLD4	DNA polymerases			
235	99.51	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
236	99.51	kd	CGS001-6601	SMARCC2	-			
237	99.51	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
238	99.51	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
239	99.51	kd	CGS001-481	ATP1B1	ATPases / P-type			
240	99.5	cc		Mitogen activated protein kinases LOF	-			
241	99.5	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
242	99.5	oe	ccsbBroad304_00568	FHL2	-			
243	99.5	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
244	99.5	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
245	99.5	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
246	99.48	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
247	99.48	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
248	99.48	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
249	99.47	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
250	99.47	oe	ccsbBroad304_01395	RFX5	-			
251	99.47	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
252	99.47	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
253	99.47	oe	ccsbBroad304_00020	ACY1	-			
254	99.46	kd	CGS001-2678	GGT1	CD molecules			
255	99.45	kd	CGS001-54442	KCTD5	-			
256	99.44	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
257	99.43	kd	CGS001-3418	IDH2	-			
258	99.42	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
259	99.41	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
260	99.41	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
261	99.41	kd	CGS001-10672	GNA13	-			
262	99.41	kd	CGS001-25874	BRP44	-			
263	99.4	kd	CGS001-170463	SSBP4	-			
264	99.39	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
265	99.38	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
266	99.38	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
267	99.38	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
268	99.36	kd	CGS001-9638	FEZ1	-			
269	99.34	kd	CGS001-51564	HDAC7	Histone deacetylases			
270	99.33	cc		Bile acid	-			
271	99.33	kd	CGS001-9787	DLGAP5	-			
272	99.33	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
273	99.32	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
274	99.32	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
275	99.32	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
276	99.32	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
277	99.31	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
278	99.31	kd	CGS001-965	CD58	CD molecules			
279	99.29	oe	ccsbBroad304_01215	PLAUR	CD molecules			
280	99.29	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
281	99.28	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
282	99.28	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
283	99.28	kd	CGS001-64943	NT5DC2	-			
284	99.28	kd	CGS001-23142	DCUN1D4	-			
285	99.26	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
286	99.25	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
287	99.25	kd	CGS001-7057	THBS1	-			
288	99.25	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
289	99.22	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
290	99.22	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
291	99.2	cc		MDM inhibitor	-			
292	99.2	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
293	99.19	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
294	99.19	kd	CGS001-389421	LIN28B	-			
295	99.16	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
296	99.15	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
297	99.15	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
298	99.15	kd	CGS001-151306	GPBAR1	Bile acid receptor			
299	99.13	oe	ccsbBroad304_00961	SMAD2	SMADs			
300	99.13	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
301	99.13	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
302	99.13	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
303	99.13	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
304	99.12	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
305	99.1	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
306	99.09	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
307	99.09	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
308	99.09	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
309	99.09	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
310	99.08	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
311	99.08	kd	CGS001-9988	DMTF1	-			
312	99.06	kd	CGS001-1314	COPA	Endogenous ligands			
313	99.05	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
314	99.04	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
315	99.03	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
316	99.02	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
317	99.02	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
318	99.02	kd	CGS001-51292	GMPR2	-			
319	99.01	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
320	99.01	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
321	99	oe	ccsbBroad304_07280	LAMTOR3	-			
322	99	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
323	99	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
324	98.98	oe	ccsbBroad304_00652	GNAS	-			
325	98.98	kd	CGS001-5682	PSMA1	Proteasome subunits			
326	98.98	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
327	98.97	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
328	98.97	kd	CGS001-1647	GADD45A	-			
329	98.94	oe	ccsbBroad304_02604	B3GNT1	-			
330	98.94	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
331	98.94	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
332	98.93	oe	ccsbBroad304_00116	ASS1	-			
333	98.93	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
334	98.92	oe	ccsbBroad304_00155	CCND1	-			
335	98.92	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
336	98.92	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
337	98.9	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
338	98.9	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
339	98.89	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
340	98.88	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
341	98.87	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
342	98.86	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
343	98.86	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
344	98.85	oe	ccsbBroad304_02633	LSM6	-			
345	98.85	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
346	98.85	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
347	98.82	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
348	98.81	kd	CGS001-4193	MDM2	-			
349	98.8	kd	CGS001-2475	MTOR	FRAP subfamily			
350	98.79	cc		Apolipoproteins LOF	-			
351	98.79	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
352	98.78	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
353	98.77	kd	CGS001-3032	HADHB	-			
354	98.74	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
355	98.74	kd	CGS001-9231	DLG5	-			
356	98.72	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
357	98.7	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
358	98.64	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
359	98.64	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
360	98.64	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
361	98.63	oe	ccsbBroad304_02741	PDS5A	-			
362	98.61	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
363	98.61	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
364	98.58	cc		Zinc fingers RanBP2 type LOF	-			
365	98.58	kd	CGS001-7849	PAX8	Paired boxes			
366	98.57	kd	CGS001-25836	NIPBL	-			
367	98.56	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
368	98.54	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
369	98.54	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
370	98.53	oe	ccsbBroad304_00150	BAX	-			
371	98.52	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
372	98.51	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
373	98.49	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
374	98.48	kd	CGS001-6256	RXRA	Retinoid X receptors			
375	98.48	kd	CGS001-6196	RPS6KA2	RSK subfamily			
376	98.46	oe	ccsbBroad304_07569	TRIB1	Trbl family			
377	98.46	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
378	98.46	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
379	98.45	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
380	98.44	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
381	98.43	oe	ccsbBroad304_00060	AMBP	Lipocalins			
382	98.43	kd	CGS001-572	BAD	-			
383	98.43	kd	CGS001-523	ATP6V1A	ATPases / V-type			
384	98.41	oe	ccsbBroad304_03859	ENOPH1	-			
385	98.39	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
386	98.38	kd	CGS001-1509	CTSD	Cathepsins			
387	98.37	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
388	98.36	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
389	98.36	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
390	98.35	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
391	98.34	oe	ccsbBroad304_02565	RALBP1	-			
392	98.34	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
393	98.33	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
394	98.32	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
395	98.32	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
396	98.32	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
397	98.31	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
398	98.3	kd	CGS001-11129	CLASRP	-			
399	98.27	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
400	98.26	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
401	98.25	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
402	98.25	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
403	98.24	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
404	98.24	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
405	98.23	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
406	98.22	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
407	98.22	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
408	98.21	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
409	98.17	oe	ccsbBroad304_07888	CBX6	-			
410	98.17	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
411	98.17	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
412	98.16	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
413	98.15	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
414	98.14	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
415	98.14	oe	ccsbBroad304_02956	EHF	-			
416	98.14	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
417	98.11	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
418	98.05	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
419	98.04	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
420	98.02	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
421	98	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
422	98	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
423	97.98	oe	ccsbBroad304_05948	CCND2	-			
424	97.95	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
425	97.95	oe	ccsbBroad304_06449	ILF3	-			
426	97.94	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
427	97.94	kd	CGS001-79581	GPR172A	-			
428	97.93	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
429	97.93	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
430	97.92	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
431	97.89	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
432	97.88	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
433	97.87	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
434	97.86	oe	ccsbBroad304_02875	BRP44	-			
435	97.86	kd	CGS001-9412	MED21	-			
436	97.85	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
437	97.83	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
438	97.83	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
439	97.79	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
440	97.76	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
441	97.74	oe	ccsbBroad304_03573	BRF2	-			
442	97.73	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
443	97.73	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
444	97.72	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
445	97.67	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
446	97.66	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
447	97.63	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
448	97.61	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
449	97.59	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
450	97.56	kd	CGS001-79109	MAPKAP1	-			
451	97.55	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
452	97.54	kd	CGS001-7771	ZFP112	-			
453	97.52	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
454	97.5	oe	ccsbBroad304_00995	MECP2	-			
455	97.5	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
456	97.47	oe	ccsbBroad304_02231	USP6NL	-			
457	97.47	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
458	97.45	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
459	97.45	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
460	97.44	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
461	97.42	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
462	97.42	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
463	97.41	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
464	97.41	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
465	97.4	kd	CGS001-3169	FOXA1	Forkhead boxes			
466	97.39	cc		Rho associated kinase inhibitor	-			
467	97.38	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
468	97.36	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
469	97.34	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
470	97.33	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
471	97.33	kd	CGS001-1892	ECHS1	-			
472	97.32	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
473	97.31	oe	ccsbBroad304_00644	GCLC	-			
474	97.29	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
475	97.26	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
476	97.25	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
477	97.25	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
478	97.24	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
479	97.24	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
480	97.23	oe	ccsbBroad304_03652	EXOC2	-			
481	97.21	cc		Potassium channel blocker	-			
482	97.21	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
483	97.19	oe	ccsbBroad304_01013	MIF	-			
484	97.18	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
485	97.13	oe	ccsbBroad304_08346	COQ3	-			
486	97.13	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
487	97.13	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
488	97.11	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
489	97.09	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
490	97.06	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
491	97.05	kd	CGS001-6009	RHEB	-			
492	97.04	kd	CGS001-1949	EFNB3	Ephrins			
493	97.04	kd	CGS001-64422	ATG3	-			
494	97.03	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
495	97.01	oe	ccsbBroad304_03173	TMED7	-			
496	96.99	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
497	96.97	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
498	96.95	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
499	96.93	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
500	96.92	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
501	96.92	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
502	96.91	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
503	96.89	cc		FXR antagonist	-			
504	96.86	oe	ccsbBroad304_00532	F11	Chymotrypsin			
505	96.86	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
506	96.85	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
507	96.83	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
508	96.83	kd	CGS001-2639	GCDH	-			
509	96.78	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
510	96.76	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
511	96.76	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
512	96.76	kd	CGS001-4811	NID1	-			
513	96.73	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
514	96.72	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
515	96.7	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
516	96.7	kd	CGS001-5092	PCBD1	-			
517	96.69	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
518	96.68	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
519	96.66	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
520	96.6	oe	ccsbBroad304_03555	PANK4	-			
521	96.6	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
522	96.58	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
523	96.57	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
524	96.57	kd	CGS001-348	APOE	Apolipoproteins			
525	96.56	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
526	96.54	kd	CGS001-4781	NFIB	-			
527	96.5	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
528	96.5	kd	CGS001-11325	DDX42	DEAD-boxes			
529	96.49	kd	CGS001-790	CAD	-			
530	96.48	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
531	96.47	cc		HSP inhibitor	-			
532	96.46	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
533	96.4	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
534	96.4	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
535	96.4	kd	CGS001-3248	HPGD	Prostaglandin synthases			
536	96.34	kd	CGS001-51268	PIPOX	-			
537	96.33	kd	CGS001-51380	CSAD	-			
538	96.27	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
539	96.26	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
540	96.25	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
541	96.25	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
542	96.25	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
543	96.23	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
544	96.23	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
545	96.19	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
546	96.18	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
547	96.16	kd	CGS001-10084	PQBP1	-			
548	96.13	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
549	96.13	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
550	96.11	oe	ccsbBroad304_09708	PNLDC1	-			
551	96.06	oe	ccsbBroad304_00819	IDH3B	-			
552	96.05	kd	CGS001-23223	RRP12	-			
553	96.02	cc		Thymidylate synthase inhibitor	-			
554	96	oe	ccsbBroad304_02668	PNKP	-			
555	95.98	oe	ccsbBroad304_02047	AP1S2	-			
556	95.94	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
557	95.94	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
558	95.93	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
559	95.9	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
560	95.9	kd	CGS001-10447	FAM3C	-			
561	95.89	kd	CGS001-9817	KEAP1	Kelch-like proteins			
562	95.88	oe	ccsbBroad304_01163	PDHA1	-			
563	95.88	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
564	95.88	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
565	95.87	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
566	95.86	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
567	95.85	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
568	95.85	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
569	95.81	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
570	95.81	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
571	95.8	oe	ccsbBroad304_03129	ERO1L	-			
572	95.8	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
573	95.8	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
574	95.79	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
575	95.72	oe	ccsbBroad304_00397	CTSK	Cathepsins			
576	95.71	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
577	95.71	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
578	95.71	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
579	95.71	kd	CGS001-1212	CLTB	-			
580	95.7	oe	ccsbBroad304_06645	NQO2	-			
581	95.7	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
582	95.69	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
583	95.68	kd	CGS001-2098	ESD	-			
584	95.65	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
585	95.65	kd	CGS001-10928	RALBP1	-			
586	95.63	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
587	95.63	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
588	95.62	kd	CGS001-10096	ACTR3	-			
589	95.61	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
590	95.61	kd	CGS001-2353	FOS	basic leucine zipper proteins			
591	95.58	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
592	95.58	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
593	95.56	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
594	95.55	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
595	95.54	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
596	95.49	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
597	95.47	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
598	95.46	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
599	95.45	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
600	95.44	cc		Vitamin D receptor agonist	-			
601	95.42	oe	ccsbBroad304_01413	RPA2	-			
602	95.41	kd	CGS001-2538	G6PC	-			
603	95.39	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
604	95.38	oe	ccsbBroad304_07140	XPC	-			
605	95.38	kd	CGS001-29883	CNOT7	-			
606	95.37	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
607	95.37	kd	CGS001-2745	GLRX	-			
608	95.36	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
609	95.35	kd	CGS001-1376	CPT2	-			
610	95.28	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
611	95.28	kd	CGS001-367	AR	Nuclear hormone receptors			
612	95.27	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
613	95.27	oe	ccsbBroad304_06089	DDIT3	-			
614	95.2	kd	CGS001-4846	NOS3	Nitric oxide synthases			
615	95.14	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
616	95.13	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
617	95.1	oe	ccsbBroad304_06090	DDOST	-			
618	95.09	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
619	95.08	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
620	95.07	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
621	95.06	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
622	95.05	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
623	95.02	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
624	95.01	kd	CGS001-1605	DAG1	-			
625	94.96	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
626	94.93	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
627	94.87	oe	ccsbBroad304_03772	CCNL1	-			
628	94.84	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
629	94.81	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
630	94.81	kd	CGS001-873	CBR1	Prostaglandin synthases			
631	94.74	oe	ccsbBroad304_01271	PPT1	-			
632	94.74	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
633	94.73	oe	ccsbBroad304_03506	AURKAIP1	-			
634	94.72	kd	CGS001-6513	SLC2A1	Solute carriers			
635	94.7	oe	ccsbBroad304_06291	GNAI1	-			
636	94.69	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
637	94.68	kd	CGS001-5144	PDE4D	Phosphodiesterases			
638	94.67	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
639	94.64	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
640	94.6	cc		Aromatase inhibitor	-			
641	94.58	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
642	94.58	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
643	94.43	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
644	94.42	kd	CGS001-5966	REL	NFkappaB transcription factor family			
645	94.42	kd	CGS001-2882	GPX7	-			
646	94.39	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
647	94.38	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
648	94.35	oe	ccsbBroad304_12226	NAGK	-			
649	94.34	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
650	94.33	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
651	94.32	kd	CGS001-64863	METTL4	-			
652	94.26	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
653	94.25	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
654	94.24	oe	ccsbBroad304_06870	RNH1	-			
655	94.21	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
656	94.21	kd	CGS001-10111	RAD50	-			
657	94.15	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
658	94.15	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
659	94.14	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
660	94.1	kd	CGS001-51655	RASD1	-			
661	94.08	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
662	94.06	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
663	94.04	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
664	94.03	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
665	94.02	kd	CGS001-5018	OXA1L	-			
666	94.01	kd	CGS001-399664	MEX3D	Mex-3 homologs			
667	94.01	kd	CGS001-1119	CHKA	-			
668	93.98	kd	CGS001-84647	PLA2G12B	-			
669	93.98	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
670	93.94	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
671	93.93	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
672	93.9	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
673	93.87	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
674	93.73	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
675	93.66	oe	ccsbBroad304_00469	DUT	-			
676	93.65	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
677	93.65	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
678	93.63	kd	CGS001-7083	TK1	-			
679	93.56	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
680	93.53	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
681	93.51	oe	ccsbBroad304_04544	RCCD1	-			
682	93.47	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
683	93.47	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
684	93.47	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
685	93.46	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
686	93.45	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
687	93.44	oe	ccsbBroad304_00818	IDH3A	-			
688	93.41	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
689	93.4	oe	ccsbBroad304_02058	PLOD3	-			
690	93.39	kd	CGS001-9670	IPO13	Importins			
691	93.38	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
692	93.38	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
693	93.37	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
694	93.34	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
695	93.31	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
696	93.26	kd	CGS001-257397	TAB3	-			
697	93.26	kd	CGS001-4048	LTA4H	Hydrolases			
698	93.25	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
699	93.25	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
700	93.25	kd	CGS001-7001	PRDX2	-			
701	93.19	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
702	93.15	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
703	93.13	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
704	93.08	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
705	93.04	kd	CGS001-9474	ATG5	-			
706	93.01	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
707	93.01	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
708	92.98	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
709	92.94	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
710	92.89	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
711	92.85	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
712	92.81	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
713	92.79	kd	CGS001-25819	CCRN4L	-			
714	92.78	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
715	92.76	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
716	92.76	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
717	92.73	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
718	92.72	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
719	92.72	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
720	92.72	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
721	92.66	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
722	92.65	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
723	92.64	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
724	92.62	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
725	92.62	kd	CGS001-56654	NPDC1	-			
726	92.61	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
727	92.52	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
728	92.51	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
729	92.5	kd	CGS001-9807	IP6K1	-			
730	92.5	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
731	92.49	oe	ccsbBroad304_00549	FDX1	-			
732	92.44	cc		Na-K-Cl transporter inhibitor	-			
733	92.43	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
734	92.41	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
735	92.4	kd	CGS001-23047	PDS5B	-			
736	92.39	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
737	92.37	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
738	92.37	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
739	92.36	kd	CGS001-1495	CTNNA1	Catenins			
740	92.32	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
741	92.31	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
742	92.3	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
743	92.3	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
744	92.26	kd	CGS001-80347	COASY	-			
745	92.24	oe	ccsbBroad304_00987	MCM3	-			
746	92.2	kd	CGS001-10390	CEPT1	-			
747	92.15	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
748	92.14	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
749	92.11	oe	ccsbBroad304_02270	FAM20B	-			
750	92.1	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
751	92.05	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
752	92.04	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
753	91.95	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
754	91.94	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
755	91.89	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
756	91.86	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
757	91.79	kd	CGS001-2731	GLDC	-			
758	91.78	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
759	91.78	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
760	91.75	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
761	91.75	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
762	91.69	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
763	91.57	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
764	91.55	kd	CGS001-79006	METRN	-			
765	91.5	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
766	91.48	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
767	91.48	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
768	91.48	kd	CGS001-818	CAMK2G	CAMK2 family			
769	91.43	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
770	91.41	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
771	91.4	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
772	91.4	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
773	91.35	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
774	91.35	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
775	91.31	oe	ccsbBroad304_06282	GLDC	-			
776	91.31	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
777	91.23	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
778	91.21	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
779	91.17	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
780	91.17	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
781	91.16	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
782	91.14	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
783	91.06	oe	ccsbBroad304_06458	IRF3	-			
784	91.03	oe	ccsbBroad304_06718	PFN2	-			
785	90.99	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
786	90.98	kd	CGS001-2108	ETFA	-			
787	90.92	kd	CGS001-8864	PER2	-			
788	90.89	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
789	90.87	kd	CGS001-2247	FGF2	Endogenous ligands			
790	90.77	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
791	90.77	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
792	90.77	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
793	90.76	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
794	90.76	kd	CGS001-10423	CDIPT	-			
795	90.74	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
796	90.74	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
797	90.72	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
798	90.7	kd	CGS001-4734	NEDD4	-			
799	90.67	oe	ccsbBroad304_07922	TRIM29	-			
800	90.65	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
801	90.62	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
802	90.56	cc		Estrogen receptor agonist	-			
803	90.53	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
804	90.52	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
805	90.47	kd	CGS001-23585	TMEM50A	-			
806	90.45	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
807	90.44	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
808	90.43	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
809	90.38	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
810	90.29	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
811	90.28	kd	CGS001-64781	CERK	Ceramide kinase			
812	90.25	oe	ccsbBroad304_09006	RPF1	-			
813	90.25	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
814	90.09	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
815	90.06	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
816	90.05	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
817	90.04	kd	CGS001-54623	PAF1	-			
818	89.99	cp	BRD-K65910366	KUC103904N	-666			-666
819	89.98	kd	CGS001-6757	SSX2	-			
820	89.95	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
821	89.82	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
822	89.81	oe	ccsbBroad304_02157	MED21	-			
823	89.81	kd	CGS001-5624	PROC	Endogenous ligands			
824	89.77	oe	ccsbBroad304_13939	MOK	RCK family			
825	89.76	oe	ccsbBroad304_00221	CASP3	Caspases			
826	89.76	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
827	89.76	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
828	89.74	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
829	89.74	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
830	89.73	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
831	89.72	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
832	89.72	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
833	89.7	oe	ccsbBroad304_06665	OAT	-			
834	89.69	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
835	89.63	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
836	89.54	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
837	89.53	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
838	89.52	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
839	89.51	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
840	89.47	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
841	89.4	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
842	89.39	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
843	89.31	cp	BRD-K15842202	eudesmic-acid	-666			-666
844	89.27	cc		Gamma secretase inhibitor	-			
845	89.26	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
846	89.15	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
847	89.11	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
848	89.1	oe	ccsbBroad304_00810	HYAL1	-			
849	89.1	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
850	89.08	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
851	89.05	kd	CGS001-91433	RCCD1	-			
852	88.93	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
853	88.92	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
854	88.82	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
855	88.82	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
856	88.76	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
857	88.75	kd	CGS001-6647	SOD1	-			
858	88.7	oe	ccsbBroad304_01787	YES1	Src family			
859	88.66	kd	CGS001-115	ADCY9	Adenylyl cyclases			
860	88.59	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
861	88.57	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
862	88.56	kd	CGS001-2773	GNAI3	-			
863	88.53	kd	CGS001-5566	PRKACA	Protein kinase A			
864	88.5	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
865	88.48	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
866	88.39	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
867	88.38	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
868	88.36	kd	CGS001-5223	PGAM1	-			
869	88.28	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
870	88.27	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
871	88.25	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
872	88.23	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
873	88.2	kd	CGS001-1659	DHX8	DEAH-boxes			
874	88.13	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
875	88.11	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
876	88.08	oe	ccsbBroad304_02239	RASSF2	-			
877	88.02	oe	ccsbBroad304_02110	VAPB	-			
878	88	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
879	87.96	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
880	87.94	kd	CGS001-2159	F10	Chymotrypsin			
881	87.94	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
882	87.93	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
883	87.93	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
884	87.87	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
885	87.86	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
886	87.85	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
887	87.84	oe	ccsbBroad304_06670	OGG1	-			
888	87.83	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
889	87.83	kd	CGS001-58478	ENOPH1	-			
890	87.81	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
891	87.76	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
892	87.75	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
893	87.49	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
894	87.49	kd	CGS001-397	ARHGDIB	Endogenous ligands			
895	87.46	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
896	87.46	kd	CGS001-2987	GUK1	-			
897	87.38	oe	ccsbBroad304_06085	DCK	-			
898	87.33	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
899	87.2	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
900	87.17	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
901	87.16	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
902	87.15	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
903	87.13	oe	ccsbBroad304_00949	LRPAP1	-			
904	87.12	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
905	87.12	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
906	87.1	kd	CGS001-25793	FBXO7	F-boxes / other			
907	87.02	kd	CGS001-3035	HARS	Aminoacyl tRNA synthetases / Class II			
908	86.99	oe	ccsbBroad304_00231	CBFB	-			
909	86.97	cc		Androgen receptor modulator	-			
910	86.97	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
911	86.92	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
912	86.9	kd	CGS001-9318	COPS2	-			
913	86.9	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
914	86.89	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
915	86.86	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
916	86.84	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
917	86.83	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
918	86.78	oe	ccsbBroad304_07616	ZNF238	-			
919	86.75	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
920	86.74	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
921	86.72	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
922	86.67	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
923	86.61	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
924	86.47	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
925	86.47	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
926	86.44	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
927	86.43	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
928	86.43	kd	CGS001-51015	ISOC1	-			
929	86.41	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
930	86.38	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
931	86.36	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
932	86.3	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
933	86.24	oe	ccsbBroad304_13598	NRBP2	NRBP family			
934	86.14	oe	ccsbBroad304_05749	A2M	-			
935	86.14	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
936	86.1	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
937	86.08	oe	ccsbBroad304_00164	BLMH	-			
938	86.04	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
939	86.03	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
940	86.02	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
941	86.01	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
942	85.93	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
943	85.88	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
944	85.87	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
945	85.87	kd	CGS001-23536	ADAT1	-			
946	85.86	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
947	85.79	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
948	85.79	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
949	85.76	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
950	85.65	oe	ccsbBroad304_00620	GCDH	-			
951	85.65	oe	ccsbBroad304_03641	ASF1B	-			
952	85.64	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
953	85.6	oe	ccsbBroad304_03878	SENP2	-			
954	85.59	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
955	85.59	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
956	85.59	oe	ccsbBroad304_01855	NCOA4	-			
957	85.57	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
958	85.56	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
959	85.51	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
960	85.48	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
961	85.45	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
962	85.45	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
963	85.42	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
964	85.4	kd	CGS001-5428	POLG	DNA polymerases			
965	85.4	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
966	85.37	oe	ccsbBroad304_02115	PTTG1	-			
967	85.36	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
968	85.31	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
969	85.29	oe	ccsbBroad304_06174	ERCC1	-			
970	85.29	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
971	85.28	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
972	85.27	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
973	85.25	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
974	85.2	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
975	85.19	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
976	85.15	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
977	85.15	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
978	85.1	cc		Supressors of cytokine signaling GOF	-			
979	85.08	oe	ccsbBroad304_07920	NUP62	-			
980	85.04	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
981	85.04	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
982	85.03	oe	ccsbBroad304_05937	CASP7	Caspases			
983	84.99	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
984	84.95	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
985	84.95	kd	CGS001-27113	BBC3	-			
986	84.93	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
987	84.92	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
988	84.89	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
989	84.89	kd	CGS001-3909	LAMA3	Laminins			
990	84.88	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
991	84.87	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
992	84.87	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
993	84.86	kd	CGS001-30836	DNTTIP2	-			
994	84.85	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
995	84.8	kd	CGS001-10221	TRIB1	Trbl family			
996	84.79	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
997	84.78	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
998	84.74	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
999	84.72	cc		Serine proteases GOF	-			
1000	84.72	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
1001	84.7	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
1002	84.51	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
1003	84.49	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
1004	84.47	kd	CGS001-11142	PKIG	-			
1005	84.46	kd	CGS001-116832	RPL39L	L ribosomal proteins			
1006	84.42	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
1007	84.42	kd	CGS001-8220	DGCR14	-			
1008	84.41	kd	CGS001-111	ADCY5	Adenylate cyclases			
1009	84.39	oe	ccsbBroad304_06287	GM2A	-			
1010	84.38	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
1011	84.26	oe	ccsbBroad304_06349	HAGH	-			
1012	84.25	oe	ccsbBroad304_08481	CEP55	-			
1013	84.18	oe	ccsbBroad304_02674	STK38	NDR family			
1014	84.13	oe	ccsbBroad304_01008	KITLG	-			
1015	84.12	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
1016	84.08	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
1017	84.06	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
1018	83.98	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
1019	83.96	kd	CGS001-10078	TSSC4	-			
1020	83.91	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
1021	83.91	oe	ccsbBroad304_06683	FURIN	Subtilisin			
1022	83.9	kd	CGS001-23131	GPATCH8	G patch domain containing			
1023	83.89	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
1024	83.83	kd	CGS001-2752	GLUL	-			
1025	83.81	oe	ccsbBroad304_01035	MSH5	-			
1026	83.81	kd	CGS001-7353	UFD1L	-			
1027	83.81	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
1028	83.7	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
1029	83.69	kd	CGS001-7311	UBA52	L ribosomal proteins			
1030	83.66	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1031	83.57	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
1032	83.57	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
1033	83.49	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
1034	83.47	kd	CGS001-2002	ELK1	ETS Transcription Factors			
1035	83.38	oe	ccsbBroad304_09954	PTRF	-			
1036	83.33	oe	ccsbBroad304_01054	GADD45B	-			
1037	83.28	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
1038	83.2	kd	CGS001-23212	RRS1	-			
1039	83.11	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
1040	83.1	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
1041	83.07	kd	CGS001-8678	BECN1	-			
1042	83.05	oe	ccsbBroad304_00390	CTGF	-			
1043	83.04	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
1044	82.97	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1045	82.96	oe	ccsbBroad304_01374	RAP1A	-			
1046	82.93	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
1047	82.93	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
1048	82.93	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
1049	82.9	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
1050	82.84	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1051	82.78	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
1052	82.75	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
1053	82.75	kd	CGS001-56616	DIABLO	-			
1054	82.66	oe	ccsbBroad304_06264	GBP2	-			
1055	82.6	kd	CGS001-1763	DNA2	-			
1056	82.58	kd	CGS001-9415	FADS2	Fatty acid desaturases			
1057	82.54	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
1058	82.51	kd	CGS001-506	ATP5B	ATPases / F-type			
1059	82.48	oe	ccsbBroad304_07267	PDLIM4	-			
1060	82.45	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
1061	82.43	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1062	82.42	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
1063	82.41	oe	ccsbBroad304_02496	MTX2	-			
1064	82.38	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
1065	82.37	kd	CGS001-53340	SPA17	-			
1066	82.29	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
1067	82.22	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
1068	82.15	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
1069	82.13	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
1070	82.11	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1071	82.11	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
1072	82.07	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
1073	82.03	kd	CGS001-2078	ERG	ETS Transcription Factors			
1074	81.85	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1075	81.84	oe	ccsbBroad304_04675	ATG4A	-			
1076	81.78	cc		Lysine acetyltransferases LOF	-			
1077	81.76	oe	ccsbBroad304_07834	GGA2	-			
1078	81.74	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
1079	81.73	oe	ccsbBroad304_09195	MCM8	-			
1080	81.71	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
1081	81.69	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
1082	81.62	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
1083	81.62	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
1084	81.55	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
1085	81.54	kd	CGS001-8743	TNFSF10	CD molecules			
1086	81.5	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
1087	81.49	oe	ccsbBroad304_14174	CDKAL1	-			
1088	81.41	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
1089	81.4	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
1090	81.38	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1091	81.38	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
1092	81.33	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
1093	81.23	oe	ccsbBroad304_02869	ASF1A	-			
1094	81.21	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
1095	81.17	kd	CGS001-139135	PASD1	-			
1096	81.16	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
1097	81.15	kd	CGS001-4255	MGMT	-			
1098	81.08	oe	ccsbBroad304_02572	SERINC3	-			
1099	81.07	oe	ccsbBroad304_06226	FTL	-			
1100	81.04	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
1101	80.96	oe	ccsbBroad304_02857	BAMBI	-			
1102	80.88	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
1103	80.87	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
1104	80.86	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
1105	80.86	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
1106	80.86	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
1107	80.71	kd	CGS001-4077	NBR1	-			
1108	80.67	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
1109	80.61	kd	CGS001-1362	CPD	Carboxypeptidase A			
1110	80.58	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
1111	80.58	kd	CGS001-29110	TBK1	IKK family			
1112	80.55	kd	CGS001-1512	CTSH	Cathepsins			
1113	80.53	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
1114	80.47	kd	CGS001-6520	SLC3A2	SLC3 family			
1115	80.47	kd	CGS001-338	APOB	Apolipoproteins			
1116	80.46	cc		Norepinephrine reuptake inhibitor	-			
1117	80.4	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
1118	80.37	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
1119	80.36	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
1120	80.36	oe	ccsbBroad304_07478	CCP110	-			
1121	80.25	kd	CGS001-25913	POT1	-			
1122	80.24	oe	ccsbBroad304_00210	CALR	-			
1123	80.19	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
1124	80.19	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1125	80.18	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
1126	80.07	kd	CGS001-51271	UBAP1	-			
1127	80.05	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
1128	80.05	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
1129	80.01	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
1130	80.01	kd	CGS001-8531	CSDA	-			
1131	80	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
1132	79.98	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1133	79.96	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
1134	79.94	oe	ccsbBroad304_03853	LSM2	-			
1135	79.93	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
1136	79.92	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
1137	79.91	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
1138	79.9	oe	ccsbBroad304_03268	GMPR2	-			
1139	79.89	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
1140	79.89	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
1141	79.88	kd	CGS001-3251	HPRT1	-			
1142	79.87	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
1143	79.83	kd	CGS001-64135	IFIH1	-			
1144	79.8	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
1145	79.78	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
1146	79.78	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
1147	79.76	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
1148	79.76	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
1149	79.71	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
1150	79.71	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
1151	79.69	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
1152	79.62	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
1153	79.6	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
1154	79.58	kd	CGS001-4605	MYBL2	-			
1155	79.55	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
1156	79.52	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
1157	79.48	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
1158	79.46	oe	ccsbBroad304_03113	DSE	-			
1159	79.42	oe	ccsbBroad304_03080	C16ORF80	-			
1160	79.39	oe	ccsbBroad304_00424	DBI	-			
1161	79.34	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
1162	79.33	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
1163	79.29	kd	CGS001-10434	LYPLA1	-			
1164	79.28	kd	CGS001-30	ACAA1	-			
1165	79.21	kd	CGS001-8895	CPNE3	-			
1166	79.18	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
1167	79.12	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
1168	79.11	oe	ccsbBroad304_00115	ASPH	-			
1169	79.07	oe	ccsbBroad304_04626	EGLN3	-			
1170	79.07	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
1171	79.05	oe	ccsbBroad304_01962	STK16	NAK family			
1172	79.02	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
1173	79	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
1174	79	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
1175	78.99	kd	CGS001-813	CALU	EF-hand domain containing			
1176	78.99	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
1177	78.97	kd	CGS001-5091	PC	Carboxylases			
1178	78.89	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
1179	78.86	kd	CGS001-230	ALDOC	-			
1180	78.85	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
1181	78.78	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
1182	78.77	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
1183	78.74	oe	ccsbBroad304_04053	DERL1	-			
1184	78.69	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
1185	78.62	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
1186	78.5	oe	ccsbBroad304_14047	TACC3	-			
1187	78.5	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
1188	78.43	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
1189	78.33	kd	CGS001-629	CFB	Complement system			
1190	78.32	kd	CGS001-11004	KIF2C	Kinesins			
1191	78.31	kd	CGS001-10465	PPIH	-			
1192	78.23	oe	ccsbBroad304_06765	PRCC	-			
1193	78.2	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
1194	78.19	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
1195	78.19	kd	CGS001-8624	PSMG1	-			
1196	78.19	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
1197	78.17	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
1198	78.16	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
1199	78.14	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
1200	78.14	kd	CGS001-3161	HMMR	CD molecules			
1201	78.13	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
1202	78.12	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
1203	78.1	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
1204	78.03	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1205	77.99	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
1206	77.98	oe	ccsbBroad304_08045	NOX1	-			
1207	77.95	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
1208	77.94	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
1209	77.93	oe	ccsbBroad304_00249	CD14	CD molecules			
1210	77.91	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
1211	77.84	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
1212	77.74	oe	ccsbBroad304_05887	CFB	Complement system			
1213	77.7	oe	ccsbBroad304_03237	LEF1	-			
1214	77.68	oe	ccsbBroad304_00874	INS	-			
1215	77.62	kd	CGS001-36	ACADSB	-			
1216	77.57	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
1217	77.5	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
1218	77.47	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
1219	77.46	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
1220	77.45	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
1221	77.42	kd	CGS001-9500	MAGED1	-			
1222	77.38	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
1223	77.35	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
1224	77.31	oe	ccsbBroad304_01164	PDHB	-			
1225	77.27	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
1226	77.22	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
1227	77.19	oe	ccsbBroad304_04465	RERG	-			
1228	77.19	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
1229	77.18	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
1230	77.07	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
1231	77	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
1232	76.97	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
1233	76.94	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
1234	76.89	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
1235	76.87	oe	ccsbBroad304_00570	FIGF	-			
1236	76.86	kd	CGS001-51002	TPRKB	-			
1237	76.85	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
1238	76.84	cc		Tumor necrosis factor superfamily LOF	-			
1239	76.72	oe	ccsbBroad304_00836	IGF2	-			
1240	76.67	oe	ccsbBroad304_02576	MLLT11	-			
1241	76.67	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
1242	76.66	oe	ccsbBroad304_03428	EXOSC4	-			
1243	76.65	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
1244	76.62	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
1245	76.61	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1246	76.59	oe	ccsbBroad304_12106	PXK	Slob family			
1247	76.57	kd	CGS001-3551	IKBKB	IKK family			
1248	76.56	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
1249	76.56	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
1250	76.56	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
1251	76.5	kd	CGS001-10691	GMEB1	-			
1252	76.45	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
1253	76.41	oe	ccsbBroad304_00053	ALDOA	-			
1254	76.41	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1255	76.28	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1256	76.26	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
1257	76.2	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1258	76.07	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
1259	76.07	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
1260	76.05	oe	ccsbBroad304_01234	POLB	DNA polymerases			
1261	75.99	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
1262	75.99	kd	CGS001-1465	CSRP1	-			
1263	75.95	cc		Kruppel like transcription factors LOF	-			
1264	75.93	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
1265	75.86	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
1266	75.81	kd	CGS001-124583	CANT1	-			
1267	75.8	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
1268	75.78	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
1269	75.73	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
1270	75.73	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
1271	75.56	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
1272	75.54	kd	CGS001-9404	LPXN	-			
1273	75.5	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
1274	75.35	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
1275	75.35	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1276	75.32	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
1277	75.32	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
1278	75.31	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
1279	75.31	kd	CGS001-8848	TSC22D1	-			
1280	75.29	kd	CGS001-26298	EHF	-			
1281	75.26	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
1282	75.21	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1283	75.21	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
1284	75.21	kd	CGS001-7295	TXN	-			
1285	75.19	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
1286	75.15	kd	CGS001-2523	FUT1	Fucosyltransferases			
1287	75.13	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
1288	75.06	kd	CGS001-3664	IRF6	-			
1289	75.03	oe	ccsbBroad304_01101	NME1	-			
1290	74.99	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
1291	74.95	kd	CGS001-133690	CAPSL	EF-hand domain containing			
1292	74.9	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1293	74.88	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
1294	74.86	oe	ccsbBroad304_13903	MTAP	-			
1295	74.84	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
1296	74.84	kd	CGS001-6732	SRPK1	SRPK family			
1297	74.81	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
1298	74.79	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
1299	74.72	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
1300	74.7	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
1301	74.69	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
1302	74.65	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
1303	74.62	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
1304	74.61	kd	CGS001-25966	C2CD2	-			
1305	74.53	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
1306	74.53	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
1307	74.5	kd	CGS001-57048	PLSCR3	-			
1308	74.48	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
1309	74.47	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
1310	74.36	kd	CGS001-3659	IRF1	-			
1311	74.33	kd	CGS001-9156	EXO1	-			
1312	74.31	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
1313	74.24	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1314	74.23	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
1315	74.21	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1316	74.18	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
1317	74.13	kd	CGS001-1195	CLK1	CDC-like kinases			
1318	74.12	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
1319	74.11	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
1320	74.11	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
1321	74.06	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
1322	74.06	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
1323	74.04	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
1324	74.03	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
1325	73.95	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
1326	73.89	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
1327	73.81	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
1328	73.72	kd	CGS001-2717	GLA	-			
1329	73.62	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
1330	73.61	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
1331	73.59	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
1332	73.53	kd	CGS001-57787	MARK4	MARK subfamily			
1333	73.42	oe	ccsbBroad304_14242	MCCC2	-			
1334	73.41	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
1335	73.36	oe	ccsbBroad304_08167	DNTTIP2	-			
1336	73.35	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
1337	73.32	oe	ccsbBroad304_02578	EBNA1BP2	-			
1338	73.31	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
1339	73.28	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
1340	73.21	kd	CGS001-56731	SLC2A4RG	-			
1341	73.15	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
1342	73.05	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
1343	72.99	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
1344	72.99	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
1345	72.9	kd	CGS001-60493	FASTKD5	-			
1346	72.86	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
1347	72.84	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
1348	72.8	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
1349	72.8	kd	CGS001-4292	MLH1	-			
1350	72.77	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
1351	72.77	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
1352	72.75	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
1353	72.72	oe	ccsbBroad304_00963	SMAD5	SMADs			
1354	72.7	kd	CGS001-2896	GRN	-			
1355	72.66	oe	ccsbBroad304_00650	GNA11	-			
1356	72.65	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
1357	72.64	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
1358	72.62	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
1359	72.56	kd	CGS001-2768	GNA12	-			
1360	72.55	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
1361	72.5	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
1362	72.49	oe	ccsbBroad304_08536	PARL	-			
1363	72.43	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
1364	72.4	kd	CGS001-9158	FIBP	-			
1365	72.38	kd	CGS001-3689	ITGB2	Integrins			
1366	72.33	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
1367	72.31	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
1368	72.26	kd	CGS001-8835	SOCS2	SH2 domain containing			
1369	72.25	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
1370	72.23	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
1371	72.19	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
1372	72.18	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
1373	72.05	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
1374	72.05	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
1375	72.02	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
1376	72.02	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
1377	72.01	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
1378	72	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
1379	71.96	kd	CGS001-23161	SNX13	Sorting nexins			
1380	71.91	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
1381	71.91	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
1382	71.84	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
1383	71.84	kd	CGS001-900	CCNG1	-			
1384	71.83	kd	CGS001-58472	SQRDL	-			
1385	71.79	oe	ccsbBroad304_02203	MAD2L1BP	-			
1386	71.77	kd	CGS001-54108	CHRAC1	-			
1387	71.76	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
1388	71.73	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
1389	71.73	kd	CGS001-571	BACH1	BTB/POZ domain containing			
1390	71.71	kd	CGS001-147179	WIPF2	-			
1391	71.66	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
1392	71.64	kd	CGS001-944	TNFSF8	CD molecules			
1393	71.5	kd	CGS001-5927	KDM5A	Histone demethylases			
1394	71.32	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
1395	71.31	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
1396	71.25	oe	ccsbBroad304_00370	CS	-			
1397	71.18	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
1398	71.16	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
1399	71.15	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
1400	71.13	kd	CGS001-5446	PON3	Paraoxonases			
1401	71.12	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
1402	71.06	oe	ccsbBroad304_14020	SH3BP5	-			
1403	70.96	kd	CGS001-7251	TSG101	-			
1404	70.92	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
1405	70.91	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
1406	70.89	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
1407	70.85	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
1408	70.85	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
1409	70.85	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
1410	70.77	oe	ccsbBroad304_03497	TXNL4B	-			
1411	70.7	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
1412	70.62	kd	CGS001-10493	VAT1	-			
1413	70.6	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
1414	70.58	oe	ccsbBroad304_02045	BUD31	-			
1415	70.55	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
1416	70.55	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1417	70.52	oe	ccsbBroad304_02502	GNA13	-			
1418	70.52	kd	CGS001-9813	KIAA0494	-			
1419	70.51	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
1420	70.48	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
1421	70.46	oe	ccsbBroad304_07704	SUB1	-			
1422	70.42	oe	ccsbBroad304_07219	CDC7	CDC7 family			
1423	70.4	kd	CGS001-10476	ATP5H	ATPases / F-type			
1424	70.38	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
1425	70.33	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
1426	70.25	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
1427	70.23	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1428	70.14	kd	CGS001-22887	FOXJ3	Forkhead boxes			
1429	70.13	kd	CGS001-9967	THRAP3	-			
1430	70.11	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
1431	70.11	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
1432	70.02	kd	CGS001-5164	PDK2	PDHK family			
1433	70.01	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
1434	70.01	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
1435	69.93	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
1436	69.89	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
1437	69.87	oe	ccsbBroad304_08266	PIPOX	-			
1438	69.86	oe	ccsbBroad304_02386	EIF1B	-			
1439	69.85	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
1440	69.85	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
1441	69.85	kd	CGS001-2244	FGB	Endogenous ligands			
1442	69.84	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
1443	69.81	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
1444	69.81	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
1445	69.79	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
1446	69.79	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
1447	69.74	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
1448	69.74	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
1449	69.66	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
1450	69.59	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1451	69.5	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
1452	69.47	oe	ccsbBroad304_00359	CPT1A	-			
1453	69.46	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
1454	69.45	cp	BRD-A71009679	KUC103420N	-666			-666
1455	69.44	oe	ccsbBroad304_06048	CRYZ	-			
1456	69.41	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
1457	69.41	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
1458	69.4	kd	CGS001-5645	PRSS2	Serine peptidases			
1459	69.4	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
1460	69.39	kd	CGS001-3065	HDAC1	Histone deacetylases			
1461	69.31	oe	ccsbBroad304_02845	PRPF6	-			
1462	69.31	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
1463	69.29	kd	CGS001-8634	RTCD1	-			
1464	69.29	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
1465	69.28	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
1466	69.1	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
1467	69.09	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
1468	69.08	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
1469	69.07	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
1470	69.02	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
1471	68.83	kd	CGS001-54584	GNB1L	WD repeat domain containing			
1472	68.76	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
1473	68.75	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
1474	68.7	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
1475	68.69	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
1476	68.66	oe	ccsbBroad304_08116	TBK1	IKK family			
1477	68.63	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
1478	68.63	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
1479	68.55	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
1480	68.52	oe	ccsbBroad304_02195	SPAG7	-			
1481	68.5	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
1482	68.46	kd	CGS001-378	ARF4	ADP-ribosylation factors			
1483	68.32	oe	ccsbBroad304_04170	PANK2	-			
1484	68.24	oe	ccsbBroad304_06663	OAS1	-			
1485	68.21	kd	CGS001-10190	TXNDC9	-			
1486	68.16	kd	CGS001-54957	TXNL4B	-			
1487	68.14	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1488	68.13	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
1489	68.12	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1490	68.12	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
1491	68.09	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
1492	68.04	kd	CGS001-5982	RFC2	ATPases / AAA-type			
1493	68	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
1494	67.99	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
1495	67.98	kd	CGS001-116443	GRIN3A	Glutamate receptors			
1496	67.96	oe	ccsbBroad304_07662	NPRL2	-			
1497	67.91	oe	ccsbBroad304_06642	NIT1	-			
1498	67.89	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
1499	67.89	kd	CGS001-26292	MYCBP	-			
1500	67.87	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
1501	67.85	kd	CGS001-5590	PRKCZ	Iota subfamily			
1502	67.82	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
1503	67.81	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
1504	67.78	kd	CGS001-8896	BUD31	-			
1505	67.77	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
1506	67.73	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
1507	67.65	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
1508	67.64	kd	CGS001-150094	SIK1	QIK subfamily			
1509	67.6	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1510	67.6	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
1511	67.58	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
1512	67.56	kd	CGS001-80135	RPF1	-			
1513	67.54	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
1514	67.51	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
1515	67.48	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
1516	67.47	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
1517	67.45	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
1518	67.45	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
1519	67.45	kd	CGS001-3171	FOXA3	Forkhead boxes			
1520	67.43	oe	ccsbBroad304_01131	OXCT1	-			
1521	67.42	oe	ccsbBroad304_07851	FAM120A	-			
1522	67.38	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
1523	67.33	oe	ccsbBroad304_00941	LIG3	-			
1524	67.33	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1525	67.31	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
1526	67.3	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
1527	67.07	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
1528	66.93	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
1529	66.92	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
1530	66.86	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
1531	66.76	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
1532	66.73	kd	CGS001-3980	LIG3	-			
1533	66.72	cc		C2 domain containing LOF	-			
1534	66.65	kd	CGS001-23464	GCAT	-			
1535	66.62	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
1536	66.59	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
1537	66.59	kd	CGS001-4125	MAN2B1	-			
1538	66.56	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
1539	66.54	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
1540	66.52	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
1541	66.48	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
1542	66.46	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
1543	66.46	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
1544	66.45	oe	ccsbBroad304_04619	GNG8	-			
1545	66.36	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
1546	66.32	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1547	66.28	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
1548	66.28	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
1549	66.27	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
1550	66.25	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
1551	66.24	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
1552	66.21	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
1553	66.2	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
1554	66.14	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
1555	66.13	kd	CGS001-10969	EBNA1BP2	-			
1556	66.1	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
1557	66.07	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
1558	66.04	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
1559	66	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
1560	65.98	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
1561	65.97	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
1562	65.93	kd	CGS001-84617	TUBB6	Tubulins			
1563	65.9	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
1564	65.88	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
1565	65.85	cc		ATP synthase inhibitor	-			
1566	65.81	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
1567	65.8	kd	CGS001-55111	PLEKHJ1	Pleckstrin homology (PH) domain containing			
1568	65.79	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
1569	65.78	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
1570	65.77	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
1571	65.76	kd	CGS001-10468	FST	-			
1572	65.73	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
1573	65.69	kd	CGS001-79094	CHAC1	-			
1574	65.66	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
1575	65.62	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
1576	65.6	kd	CGS001-55082	ARGLU1	-			
1577	65.51	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
1578	65.42	oe	ccsbBroad304_05098	MAGEB6	-			
1579	65.42	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
1580	65.42	kd	CGS001-955	ENTPD6	-			
1581	65.41	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
1582	65.39	cc		X linked mental retardation group 2 LOF	-			
1583	65.39	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
1584	65.32	kd	CGS001-253260	RICTOR	-			
1585	65.31	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
1586	65.29	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
1587	65.29	kd	CGS001-3895	KTN1	-			
1588	65.26	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
1589	65.15	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
1590	65.12	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
1591	65.06	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
1592	65.03	oe	ccsbBroad304_02138	TRIP10	-			
1593	65.03	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
1594	65.03	kd	CGS001-7919	DDX39B	DEAD-boxes			
1595	65	oe	ccsbBroad304_05194	LIPH	-			
1596	64.96	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
1597	64.86	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
1598	64.85	kd	CGS001-4173	MCM4	-			
1599	64.84	oe	ccsbBroad304_00658	GNG5	-			
1600	64.83	oe	ccsbBroad304_02287	GNPDA1	-			
1601	64.69	kd	CGS001-9767	PHF16	-			
1602	64.69	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
1603	64.67	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1604	64.64	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
1605	64.63	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
1606	64.63	kd	CGS001-154197	PNLDC1	-			
1607	64.6	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
1608	64.59	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
1609	64.58	kd	CGS001-801	CALM1	EF-hand domain containing			
1610	64.54	kd	CGS001-5306	PITPNA	-			
1611	64.48	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
1612	64.4	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
1613	64.4	kd	CGS001-25942	SIN3A	-			
1614	64.33	oe	ccsbBroad304_00964	SMAD7	SMADs			
1615	64.31	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
1616	64.29	kd	CGS001-835	CASP2	Caspases			
1617	64.24	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
1618	64.24	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
1619	64.23	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
1620	64.22	kd	CGS001-8692	HYAL2	-			
1621	64.19	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
1622	64.17	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
1623	64.16	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1624	64.08	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
1625	64.06	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
1626	64.05	kd	CGS001-5962	RDX	-			
1627	64.04	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
1628	64.04	kd	CGS001-1725	DHPS	-			
1629	64	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
1630	63.85	kd	CGS001-8829	NRP1	CD molecules			
1631	63.82	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
1632	63.76	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
1633	63.75	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1634	63.73	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
1635	63.72	oe	ccsbBroad304_03266	ERGIC2	-			
1636	63.7	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
1637	63.66	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
1638	63.61	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
1639	63.6	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
1640	63.59	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
1641	63.51	kd	CGS001-3630	INS	-			
1642	63.5	kd	CGS001-3925	STMN1	-			
1643	63.47	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
1644	63.44	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1645	63.32	oe	ccsbBroad304_04202	MED28	-			
1646	63.3	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
1647	63.25	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
1648	63.22	kd	CGS001-7097	TLR2	Toll-like receptor family			
1649	63.14	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
1650	63.11	kd	CGS001-5575	PRKAR1B	Protein kinase A			
1651	63.1	kd	CGS001-3482	IGF2R	CD molecules			
1652	63.01	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
1653	63.01	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
1654	62.99	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
1655	62.98	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
1656	62.93	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
1657	62.88	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
1658	62.86	oe	ccsbBroad304_03640	CEP72	-			
1659	62.84	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
1660	62.79	oe	ccsbBroad304_00783	HPRT1	-			
1661	62.79	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
1662	62.78	oe	ccsbBroad304_00738	HINT1	-			
1663	62.7	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
1664	62.62	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
1665	62.61	kd	CGS001-205	AK4	Adenylate kinases			
1666	62.61	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
1667	62.59	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
1668	62.53	oe	ccsbBroad304_06383	HMMR	CD molecules			
1669	62.48	kd	CGS001-822	CAPG	-			
1670	62.47	oe	ccsbBroad304_09881	RFX6	-			
1671	62.45	kd	CGS001-64077	LHPP	-			
1672	62.43	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
1673	62.4	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
1674	62.33	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
1675	62.3	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
1676	62.29	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
1677	62.28	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
1678	62.24	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
1679	62.22	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
1680	62.22	kd	CGS001-3416	IDE	Pitrilysin			
1681	62.17	cc		NFkB pathway inhibitor	-			
1682	62.12	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
1683	62.08	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1684	62.06	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
1685	62.06	kd	CGS001-7029	TFDP2	-			
1686	62.05	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
1687	61.96	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
1688	61.94	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
1689	61.94	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1690	61.94	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
1691	61.93	cc		C2 domain containing protein kinases LOF	-			
1692	61.92	oe	ccsbBroad304_01576	SOAT1	-			
1693	61.92	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
1694	61.92	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
1695	61.89	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
1696	61.87	kd	CGS001-64333	ARHGAP9	Rho GTPase activating proteins			
1697	61.77	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
1698	61.76	kd	CGS001-1951	CELSR3	Cadherins / Major cadherins			
1699	61.74	kd	CGS001-5664	PSEN2	Presenilin			
1700	61.74	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1701	61.73	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
1702	61.72	kd	CGS001-22938	SNW1	-			
1703	61.7	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1704	61.7	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1705	61.67	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
1706	61.64	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
1707	61.61	oe	ccsbBroad304_05763	ACTB	-			
1708	61.54	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1709	61.5	oe	ccsbBroad304_08775	SQRDL	-			
1710	61.48	kd	CGS001-5300	PIN1	-			
1711	61.45	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
1712	61.34	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
1713	61.32	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
1714	61.31	kd	CGS001-1869	E2F1	-			
1715	61.28	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
1716	61.17	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
1717	61.12	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
1718	61.12	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1719	61.1	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1720	61	oe	ccsbBroad304_07798	EXOC3	-			
1721	60.93	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
1722	60.93	kd	CGS001-578	BAK1	-			
1723	60.9	oe	ccsbBroad304_01593	SRP14	-			
1724	60.9	oe	ccsbBroad304_02220	MTFR1	-			
1725	60.77	kd	CGS001-57680	CHD8	-			
1726	60.76	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
1727	60.72	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
1728	60.68	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
1729	60.67	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
1730	60.59	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
1731	60.57	kd	CGS001-29984	RHOD	-			
1732	60.57	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1733	60.52	oe	ccsbBroad304_01148	PCBD1	-			
1734	60.52	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
1735	60.49	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
1736	60.49	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
1737	60.47	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
1738	60.46	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
1739	60.39	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
1740	60.38	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
1741	60.37	oe	ccsbBroad304_06237	GAA	Glycosidases			
1742	60.37	oe	ccsbBroad304_04387	MKI67IP	-			
1743	60.36	kd	CGS001-7248	TSC1	-			
1744	60.28	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
1745	60.25	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
1746	60.23	oe	ccsbBroad304_02772	ICMT	-			
1747	60.23	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
1748	60.23	kd	CGS001-10214	SSX3	-			
1749	60.21	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
1750	60.19	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
1751	60.09	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
1752	60.02	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1753	59.99	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
1754	59.95	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
1755	59.94	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
1756	59.91	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
1757	59.82	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
1758	59.74	oe	ccsbBroad304_06855	RDX	-			
1759	59.74	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
1760	59.71	kd	CGS001-306	ANXA3	Annexins			
1761	59.68	kd	CGS001-1198	CLK3	CDC-like kinases			
1762	59.64	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
1763	59.62	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
1764	59.6	kd	CGS001-10671	DCTN6	-			
1765	59.56	oe	ccsbBroad304_01139	PA2G4	-			
1766	59.54	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
1767	59.54	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1768	59.52	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
1769	59.52	kd	CGS001-2931	GSK3A	GSK subfamily			
1770	59.47	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
1771	59.46	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
1772	59.45	oe	ccsbBroad304_06253	GALT	-			
1773	59.38	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
1774	59.37	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
1775	59.35	kd	CGS001-54821	ERCC6L	-			
1776	59.23	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
1777	59.21	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
1778	59.17	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
1779	59.14	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
1780	59.12	kd	CGS001-23743	BHMT2	-			
1781	59.09	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
1782	59.07	kd	CGS001-3098	HK1	-			
1783	59.06	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
1784	59.03	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
1785	59.02	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
1786	58.95	kd	CGS001-6832	SUPV3L1	-			
1787	58.93	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
1788	58.89	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
1789	58.88	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
1790	58.86	kd	CGS001-51727	CMPK1	-			
1791	58.83	oe	ccsbBroad304_01146	PARN	-			
1792	58.81	kd	CGS001-427	ASAH1	Acid ceramidase			
1793	58.78	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
1794	58.68	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1795	58.6	kd	CGS001-23028	KDM1A	Histone demethylase			
1796	58.57	kd	CGS001-8985	PLOD3	-			
1797	58.55	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1798	58.51	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
1799	58.38	kd	CGS001-103	ADAR	-			
1800	58.32	kd	CGS001-5236	PGM1	-			
1801	58.3	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
1802	58.27	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
1803	58.27	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
1804	58.2	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
1805	58.07	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
1806	58.07	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
1807	58.05	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
1808	58.05	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
1809	58.05	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
1810	58.03	oe	ccsbBroad304_06066	CTSL1	-			
1811	58.03	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
1812	58.01	oe	ccsbBroad304_00648	GLRX	-			
1813	58	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1814	57.89	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
1815	57.8	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
1816	57.76	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
1817	57.73	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
1818	57.72	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
1819	57.71	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
1820	57.7	oe	ccsbBroad304_08825	LHPP	-			
1821	57.7	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
1822	57.7	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
1823	57.59	oe	ccsbBroad304_01105	PNP	-			
1824	57.46	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
1825	57.44	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
1826	57.41	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
1827	57.25	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
1828	57.21	oe	ccsbBroad304_00969	MAGEA10	-			
1829	57.15	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
1830	57.04	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
1831	56.98	oe	ccsbBroad304_08365	CYCS	-			
1832	56.96	oe	ccsbBroad304_00933	LDHB	-			
1833	56.93	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
1834	56.91	oe	ccsbBroad304_00237	CCND3	-			
1835	56.86	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1836	56.78	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
1837	56.76	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
1838	56.75	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
1839	56.69	oe	ccsbBroad304_02737	JMJD6	-			
1840	56.61	kd	CGS001-55810	FOXJ2	Forkhead boxes			
1841	56.56	kd	CGS001-4287	ATXN3	Ataxins			
1842	56.53	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
1843	56.51	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
1844	56.5	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
1845	56.5	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1846	56.45	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
1847	56.45	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
1848	56.3	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
1849	56.29	kd	CGS001-57026	PDXP	-			
1850	56.27	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
1851	56.26	kd	CGS001-7504	XK	Blood group antigens			
1852	56.23	oe	ccsbBroad304_07362	NMI	-			
1853	56.2	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
1854	56.19	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
1855	56.18	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
1856	56.16	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
1857	56.15	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
1858	56.1	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
1859	55.97	kd	CGS001-83593	RASSF5	-			
1860	55.95	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
1861	55.94	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
1862	55.91	kd	CGS001-51441	YTHDF2	-			
1863	55.9	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
1864	55.9	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
1865	55.88	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
1866	55.8	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
1867	55.76	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
1868	55.75	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
1869	55.62	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
1870	55.6	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
1871	55.55	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
1872	55.53	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
1873	55.49	oe	ccsbBroad304_03405	CHRAC1	-			
1874	55.49	kd	CGS001-23077	MYCBP2	-			
1875	55.44	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
1876	55.44	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
1877	55.37	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
1878	55.33	kd	CGS001-2114	ETS2	ETS Transcription Factors			
1879	55.32	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
1880	55.32	kd	CGS001-387	RHOA	-			
1881	55.26	oe	ccsbBroad304_07548	TSSC4	-			
1882	55.2	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
1883	55.2	oe	ccsbBroad304_01841	BAG6	-			
1884	55.2	kd	CGS001-55612	FERMT1	Fermitins			
1885	55.16	kd	CGS001-6895	TARBP2	-			
1886	55.12	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
1887	55.09	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
1888	55.07	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
1889	55.07	oe	ccsbBroad304_01373	RAN	-			
1890	55.07	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
1891	55.06	kd	CGS001-5366	PMAIP1	-			
1892	55.04	kd	CGS001-253430	IPMK	-			
1893	55	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
1894	54.94	oe	ccsbBroad304_08325	LIPT1	-			
1895	54.93	oe	ccsbBroad304_04379	LZIC	-			
1896	54.9	kd	CGS001-8974	P4HA2	-			
1897	54.89	oe	ccsbBroad304_02249	KIAA0494	-			
1898	54.87	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
1899	54.87	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
1900	54.84	kd	CGS001-23014	FBXO21	F-boxes / other			
1901	54.81	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
1902	54.78	oe	ccsbBroad304_05902	BNIP3	-			
1903	54.76	kd	CGS001-10614	HEXIM1	-			
1904	54.76	kd	CGS001-94234	FOXQ1	Forkhead boxes			
1905	54.64	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
1906	54.64	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
1907	54.62	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
1908	54.59	oe	ccsbBroad304_08093	DCPS	-			
1909	54.51	kd	CGS001-8639	AOC3	Oxidoreductases			
1910	54.48	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
1911	54.39	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
1912	54.38	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
1913	54.34	kd	CGS001-10284	SAP18	-			
1914	54.33	oe	ccsbBroad304_06654	NPM1	-			
1915	54.32	oe	ccsbBroad304_03308	YTHDF2	-			
1916	54.3	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
1917	54.28	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
1918	54.23	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
1919	54.19	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
1920	54.19	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
1921	54.13	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
1922	54.11	kd	CGS001-5062	PAK2	PAKA subfamily			
1923	54.08	kd	CGS001-2356	FPGS	-			
1924	54.07	oe	ccsbBroad304_01208	PITPNA	-			
1925	54.03	kd	CGS001-3579	CXCR2	Chemokine receptors			
1926	54.01	kd	CGS001-9170	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1927	54.01	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
1928	53.96	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
1929	53.94	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
1930	53.94	kd	CGS001-1356	CP	-			
1931	53.92	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
1932	53.92	kd	CGS001-23678	SGK3	SGK family			
1933	53.91	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
1934	53.89	kd	CGS001-6652	SORD	-			
1935	53.76	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
1936	53.7	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
1937	53.69	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
1938	53.66	kd	CGS001-3995	FADS3	Fatty acid desaturases			
1939	53.64	kd	CGS001-10018	BCL2L11	-			
1940	53.62	kd	CGS001-435	ASL	-			
1941	53.58	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
1942	53.58	kd	CGS001-3155	HMGCL	-			
1943	53.55	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
1944	53.53	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
1945	53.44	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
1946	53.44	kd	CGS001-54505	DHX29	DEAH-boxes			
1947	53.34	oe	ccsbBroad304_04153	PHF17	-			
1948	53.31	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
1949	53.31	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
1950	53.26	oe	ccsbBroad304_00100	RHOA	-			
1951	53.25	oe	ccsbBroad304_00072	ANXA7	Annexins			
1952	53.17	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
1953	53.13	oe	ccsbBroad304_08684	CXCR7	-			
1954	53.09	oe	ccsbBroad304_09358	MAPK1IP1L	-			
1955	53.04	oe	ccsbBroad304_01247	POU2AF1	-			
1956	53.04	kd	CGS001-6884	TAF13	-			
1957	53.03	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
1958	53	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
1959	52.97	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
1960	52.95	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
1961	52.94	cc		Sodium channel blocker	-			
1962	52.94	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
1963	52.92	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
1964	52.84	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
1965	52.76	oe	ccsbBroad304_01203	PIM1	PIM family			
1966	52.65	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
1967	52.62	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
1968	52.52	kd	CGS001-29916	SNX11	Sorting nexins			
1969	52.51	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1970	52.51	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
1971	52.49	kd	CGS001-10400	PEMT	-			
1972	52.45	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
1973	52.36	oe	ccsbBroad304_07808	RAB11FIP2	-			
1974	52.35	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
1975	52.2	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
1976	52.19	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
1977	52.07	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
1978	52.07	kd	CGS001-8464	SUPT3H	-			
1979	52.06	kd	CGS001-27297	CRCP	-			
1980	52	kd	CGS001-1727	CYB5R3	-			
1981	51.99	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
1982	51.97	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
1983	51.91	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
1984	51.91	kd	CGS001-54915	YTHDF1	-			
1985	51.9	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
1986	51.89	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
1987	51.85	kd	CGS001-9697	TRAM2	-			
1988	51.82	oe	ccsbBroad304_01716	TSN	-			
1989	51.82	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
1990	51.81	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
1991	51.74	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
1992	51.69	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
1993	51.68	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
1994	51.67	oe	ccsbBroad304_00747	HLF	-			
1995	51.63	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
1996	51.58	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
1997	51.58	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
1998	51.57	kd	CGS001-1036	CDO1	-			
1999	51.55	oe	ccsbBroad304_07766	RASSF1	-			
2000	51.53	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
2001	51.44	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
2002	51.43	oe	ccsbBroad304_06985	SORD	-			
2003	51.35	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
2004	51.31	oe	ccsbBroad304_01933	TEAD2	-			
2005	51.3	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
2006	51.27	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
2007	51.25	oe	ccsbBroad304_08322	UFM1	-			
2008	51.24	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
2009	51.23	cc		Cyclooxygenase inhibitor	-			
2010	51.18	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
2011	51.17	oe	ccsbBroad304_00993	MDM4	-			
2012	51.16	cc		HIV protease inhibitor	-			
2013	51.15	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
2014	51.13	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
2015	51.13	kd	CGS001-2621	GAS6	-			
2016	51.11	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
2017	50.98	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
2018	50.97	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
2019	50.96	cc		Tachykinin antagonist	-			
2020	50.96	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
2021	50.94	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2022	50.87	kd	CGS001-83448	PUS7L	-			
2023	50.74	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
2024	50.72	kd	CGS001-4668	NAGA	-			
2025	50.71	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
2026	50.69	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
2027	50.65	kd	CGS001-7039	TGFA	-			
2028	50.64	kd	CGS001-5373	PMM2	-			
2029	50.63	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
2030	50.6	kd	CGS001-587	BCAT2	-			
2031	50.58	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
2032	50.53	kd	CGS001-2184	FAH	-			
2033	50.5	oe	ccsbBroad304_01532	SIAH1	-			
2034	50.47	kd	CGS001-23621	BACE1	Pepsin			
2035	50.43	kd	CGS001-663	BNIP2	-			
2036	50.38	cp	BRD-A02189320	met-leu-phe	-666			-666
2037	50.34	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
2038	50.29	oe	ccsbBroad304_06098	DHCR24	-			
2039	50.25	kd	CGS001-839	CASP6	Caspases			
2040	50.21	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
2041	50.21	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
2042	50.19	oe	ccsbBroad304_00542	FBP1	-			
2043	50.17	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
2044	50.15	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
2045	50.09	oe	ccsbBroad304_02843	FTSJ1	-			
2046	50.04	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
2047	50	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
2048	49.92	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2049	49.9	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2050	49.89	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
2051	49.89	oe	ccsbBroad304_00816	IDE	Pitrilysin			
2052	49.88	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
2053	49.86	oe	ccsbBroad304_03848	METTL14	-			
2054	49.85	oe	ccsbBroad304_01623	SUPT4H1	-			
2055	49.85	oe	ccsbBroad304_08511	RFK	-			
2056	49.79	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2057	49.78	kd	CGS001-100	ADA	Adenosine turnover			
2058	49.77	oe	ccsbBroad304_06172	EPS8	-			
2059	49.75	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
2060	49.7	oe	ccsbBroad304_04775	NTAN1	-			
2061	49.7	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
2062	49.57	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
2063	49.56	kd	CGS001-2023	ENO1	-			
2064	49.55	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
2065	49.48	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
2066	49.47	oe	ccsbBroad304_00661	GNGT2	-			
2067	49.47	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
2068	49.4	cc		RNA Polymerase Enzymes LOF	-			
2069	49.38	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
2070	49.38	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
2071	49.31	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
2072	49.3	oe	ccsbBroad304_06292	GNAI2	-			
2073	49.25	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
2074	49.21	kd	CGS001-5198	PFAS	-			
2075	49.07	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
2076	49.07	oe	ccsbBroad304_00147	BAG1	-			
2077	49.02	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
2078	48.99	oe	ccsbBroad304_02052	KYNU	-			
2079	48.99	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
2080	48.97	kd	CGS001-64080	RBKS	-			
2081	48.94	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
2082	48.93	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
2083	48.92	kd	CGS001-23451	SF3B1	-			
2084	48.91	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
2085	48.91	kd	CGS001-6499	SKIV2L	-			
2086	48.88	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
2087	48.84	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
2088	48.8	oe	ccsbBroad304_04471	C5ORF62	-			
2089	48.78	cp	BRD-K34508425	KUC103898N	-666			-666
2090	48.78	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
2091	48.76	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
2092	48.75	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
2093	48.74	cc		Targets of VEGFR inhibitors GOF	-			
2094	48.72	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
2095	48.71	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
2096	48.69	oe	ccsbBroad304_10437	STMN1	-			
2097	48.68	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
2098	48.68	kd	CGS001-1445	CSK	Csk family			
2099	48.66	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2100	48.63	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
2101	48.62	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
2102	48.62	kd	CGS001-1384	CRAT	-			
2103	48.57	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
2104	48.52	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
2105	48.5	cc		PI3K Signaling LOF	-			
2106	48.5	oe	ccsbBroad304_07511	KIF14	Kinesins			
2107	48.49	kd	CGS001-9870	KIAA0317	-			
2108	48.49	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
2109	48.48	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
2110	48.47	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
2111	48.46	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
2112	48.46	kd	CGS001-79600	TCTN1	Tectonic proteins			
2113	48.44	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
2114	48.43	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
2115	48.39	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
2116	48.38	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
2117	48.36	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2118	48.35	kd	CGS001-9443	MED7	-			
2119	48.3	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
2120	48.28	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
2121	48.27	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
2122	48.14	kd	CGS001-10325	RRAGB	-			
2123	48.06	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
2124	48.04	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
2125	48.03	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
2126	48.03	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
2127	47.98	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
2128	47.96	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
2129	47.88	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
2130	47.83	oe	ccsbBroad304_03097	CNOT7	-			
2131	47.82	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
2132	47.82	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
2133	47.78	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
2134	47.76	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2135	47.74	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
2136	47.68	kd	CGS001-1837	DTNA	-			
2137	47.67	kd	CGS001-91304	C19ORF6	-			
2138	47.65	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
2139	47.65	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
2140	47.62	oe	ccsbBroad304_07097	TRAF1	-			
2141	47.61	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
2142	47.59	oe	ccsbBroad304_06013	CLPTM1	-			
2143	47.59	kd	CGS001-51001	MTERFD1	-			
2144	47.55	oe	ccsbBroad304_06739	PLOD1	-			
2145	47.5	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
2146	47.49	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
2147	47.41	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
2148	47.41	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
2149	47.4	oe	ccsbBroad304_08386	SMOX	-			
2150	47.29	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
2151	47.24	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
2152	47.22	kd	CGS001-7090	TLE3	WD repeat domain containing			
2153	47.2	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
2154	47.16	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
2155	47.12	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
2156	47.04	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
2157	47.04	kd	CGS001-8525	DGKZ	-			
2158	47.01	kd	CGS001-949	SCARB1	-			
2159	46.98	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
2160	46.86	kd	CGS001-55556	ENOSF1	-			
2161	46.81	oe	ccsbBroad304_03910	CCDC90A	-			
2162	46.79	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
2163	46.79	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
2164	46.73	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
2165	46.68	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
2166	46.68	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
2167	46.67	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
2168	46.67	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
2169	46.65	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
2170	46.65	oe	ccsbBroad304_09354	IGSF8	CD molecules			
2171	46.63	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
2172	46.59	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
2173	46.59	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
2174	46.59	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
2175	46.58	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
2176	46.54	kd	CGS001-593	BCKDHA	-			
2177	46.52	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
2178	46.48	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
2179	46.46	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
2180	46.43	oe	ccsbBroad304_01143	PAFAH1B3	-			
2181	46.43	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
2182	46.41	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
2183	46.41	oe	ccsbBroad304_09615	LACC1	-			
2184	46.39	oe	ccsbBroad304_02526	POP4	-			
2185	46.37	oe	ccsbBroad304_02716	NMNAT2	-			
2186	46.36	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
2187	46.35	kd	CGS001-51128	SAR1B	-			
2188	46.33	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
2189	46.32	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2190	46.28	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
2191	46.23	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
2192	46.21	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
2193	46.17	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
2194	46.1	oe	ccsbBroad304_01205	PIN1	-			
2195	46.1	oe	ccsbBroad304_04788	OVCA2	-			
2196	46.1	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
2197	46.09	oe	ccsbBroad304_04404	TUBB6	Tubulins			
2198	46.01	cc		Akt Signaling GOF	-			
2199	45.99	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
2200	45.98	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
2201	45.96	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
2202	45.91	kd	CGS001-7263	TST	-			
2203	45.9	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
2204	45.9	kd	CGS001-10475	TRIM38	-			
2205	45.87	oe	ccsbBroad304_02955	MYCBP	-			
2206	45.85	oe	ccsbBroad304_03858	SRPRB	-			
2207	45.85	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
2208	45.84	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
2209	45.81	kd	CGS001-79733	E2F8	-			
2210	45.78	oe	ccsbBroad304_01002	METTL1	-			
2211	45.78	kd	CGS001-55715	DOK4	Pleckstrin homology (PH) domain containing			
2212	45.76	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
2213	45.75	kd	CGS001-694	BTG1	-			
2214	45.72	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
2215	45.71	kd	CGS001-10613	ERLIN1	-			
2216	45.68	oe	ccsbBroad304_01974	RNASET2	-			
2217	45.63	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
2218	45.61	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
2219	45.54	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
2220	45.47	oe	ccsbBroad304_08662	MCCC1	-			
2221	45.44	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
2222	45.44	kd	CGS001-2524	FUT2	Fucosyltransferases			
2223	45.42	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2224	45.39	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
2225	45.35	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
2226	45.34	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
2227	45.31	kd	CGS001-114609	TIRAP	-			
2228	45.3	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
2229	45.27	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
2230	45.24	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
2231	45.22	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
2232	45.22	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
2233	45.21	oe	ccsbBroad304_02756	RRP8	-			
2234	45.19	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
2235	45.19	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
2236	45.16	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
2237	45.12	kd	CGS001-5925	RB1	Endogenous ligands			
2238	45.09	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
2239	45.04	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
2240	45.02	oe	ccsbBroad304_00833	IFNG	Interferons			
2241	44.98	kd	CGS001-161725	OTUD7A	OTU domain containing			
2242	44.95	kd	CGS001-3066	HDAC2	Histone deacetylases			
2243	44.92	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
2244	44.89	oe	ccsbBroad304_00001	NAT1	-			
2245	44.89	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2246	44.89	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
2247	44.88	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
2248	44.84	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
2249	44.8	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
2250	44.79	oe	ccsbBroad304_00418	CD55	CD molecules			
2251	44.72	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
2252	44.71	oe	ccsbBroad304_07018	SUPT5H	-			
2253	44.71	kd	CGS001-5037	PEBP1	-			
2254	44.68	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
2255	44.67	oe	ccsbBroad304_05985	CFL1	-			
2256	44.63	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
2257	44.63	kd	CGS001-9926	LPGAT1	-			
2258	44.62	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
2259	44.61	oe	ccsbBroad304_02581	ASCC3	-			
2260	44.59	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
2261	44.59	kd	CGS001-4088	SMAD3	SMADs			
2262	44.58	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
2263	44.56	oe	ccsbBroad304_05756	ACAA1	-			
2264	44.55	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
2265	44.53	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
2266	44.53	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
2267	44.52	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
2268	44.49	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
2269	44.45	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
2270	44.44	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
2271	44.43	oe	ccsbBroad304_00471	E2F6	-			
2272	44.43	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
2273	44.42	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
2274	44.42	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
2275	44.38	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
2276	44.36	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
2277	44.28	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
2278	44.25	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
2279	44.25	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
2280	44.24	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
2281	44.21	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
2282	44.18	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
2283	44.14	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
2284	44.11	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
2285	44.06	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
2286	44.04	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
2287	44.04	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
2288	44.03	kd	CGS001-2073	ERCC5	-			
2289	44.01	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
2290	43.97	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
2291	43.94	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
2292	43.89	kd	CGS001-1676	DFFA	-			
2293	43.86	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
2294	43.72	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
2295	43.69	oe	ccsbBroad304_07800	EXOSC8	-			
2296	43.69	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
2297	43.69	kd	CGS001-200734	SPRED2	-			
2298	43.64	kd	CGS001-6603	SMARCD2	-			
2299	43.63	oe	ccsbBroad304_03951	NARFL	-			
2300	43.62	kd	CGS001-22978	NT5C2	Adenosine turnover			
2301	43.62	kd	CGS001-2877	GPX2	-			
2302	43.6	oe	ccsbBroad304_03372	CAB39	-			
2303	43.6	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
2304	43.52	kd	CGS001-7405	UVRAG	-			
2305	43.47	oe	ccsbBroad304_02219	MORF4L2	-			
2306	43.45	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
2307	43.41	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
2308	43.31	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
2309	43.29	oe	ccsbBroad304_10431	HADHB	-			
2310	43.28	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
2311	43.26	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
2312	43.24	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
2313	43.22	kd	CGS001-4312	MMP1	Matrix metallopeptidase			
2314	43.22	kd	CGS001-4171	MCM2	-			
2315	43.15	kd	CGS001-55604	LRRC16A	-			
2316	43.13	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
2317	43.13	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
2318	43.13	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
2319	43.11	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
2320	43.1	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
2321	43.08	oe	ccsbBroad304_08605	PBK	TOPK family			
2322	43.05	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
2323	43.04	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
2324	43.03	oe	ccsbBroad304_03357	RASD1	-			
2325	42.99	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
2326	42.98	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
2327	42.98	kd	CGS001-7525	YES1	Src family			
2328	42.96	oe	ccsbBroad304_02057	P4HA2	-			
2329	42.94	oe	ccsbBroad304_06382	HMGCL	-			
2330	42.94	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
2331	42.94	kd	CGS001-901	CCNG2	-			
2332	42.91	kd	CGS001-597	BCL2A1	-			
2333	42.87	kd	CGS001-1655	DDX5	DEAD-boxes			
2334	42.87	oe	ccsbBroad304_08879	CASD1	-			
2335	42.83	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
2336	42.82	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
2337	42.82	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
2338	42.82	kd	CGS001-11151	CORO1A	Coronins			
2339	42.78	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
2340	42.77	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
2341	42.72	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
2342	42.71	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
2343	42.7	kd	CGS001-11164	NUDT5	Nudix motif containing			
2344	42.67	oe	ccsbBroad304_00564	FGR	Src family			
2345	42.66	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
2346	42.66	kd	CGS001-10398	MYL9	EF-hand domain containing			
2347	42.64	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
2348	42.6	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
2349	42.58	oe	ccsbBroad304_08888	ACD	-			
2350	42.57	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
2351	42.56	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
2352	42.56	kd	CGS001-7466	WFS1	-			
2353	42.51	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
2354	42.51	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
2355	42.5	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
2356	42.49	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
2357	42.47	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
2358	42.46	kd	CGS001-7728	ZNF175	Zinc fingers, C2H2-type			
2359	42.41	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
2360	42.41	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
2361	42.39	kd	CGS001-1440	CSF3	Endogenous ligands			
2362	42.35	kd	CGS001-29775	CARD10	-			
2363	42.32	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2364	42.3	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
2365	42.29	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
2366	42.22	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
2367	42.21	oe	ccsbBroad304_06998	SRPK1	SRPK family			
2368	42.18	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
2369	42.15	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
2370	42.15	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
2371	42.15	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
2372	42.08	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
2373	42.07	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
2374	42.07	kd	CGS001-5588	PRKCQ	Delta subfamily			
2375	42.05	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
2376	42.04	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
2377	42.02	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
2378	42.02	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
2379	41.99	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
2380	41.98	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2381	41.97	kd	CGS001-51097	SCCPDH	-			
2382	41.96	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
2383	41.94	oe	ccsbBroad304_06235	G6PD	-			
2384	41.93	kd	CGS001-2242	FES	Fer family			
2385	41.9	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
2386	41.86	oe	ccsbBroad304_01699	TPD52L2	-			
2387	41.86	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
2388	41.78	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
2389	41.74	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
2390	41.73	oe	ccsbBroad304_02566	MORF4L1	-			
2391	41.72	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
2392	41.68	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
2393	41.66	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
2394	41.6	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
2395	41.53	kd	CGS001-50813	COPS7A	-			
2396	41.52	oe	ccsbBroad304_02553	BLCAP	-			
2397	41.51	oe	ccsbBroad304_00171	BNIP3L	-			
2398	41.51	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
2399	41.51	kd	CGS001-23530	NNT	-			
2400	41.44	kd	CGS001-3669	ISG20	-			
2401	41.42	cc		Sigma receptor antagonist	-			
2402	41.37	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
2403	41.36	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
2404	41.34	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
2405	41.29	kd	CGS001-6598	SMARCB1	-			
2406	41.25	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
2407	41.2	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
2408	41.2	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
2409	41.19	kd	CGS001-6632	SNRPD1	-			
2410	41.18	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
2411	41.18	kd	CGS001-56916	SMARCAD1	-			
2412	41.16	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
2413	41.15	oe	ccsbBroad304_04064	PRR15L	-			
2414	41.14	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
2415	41	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
2416	40.99	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
2417	40.98	oe	ccsbBroad304_01723	TTK	TTK family			
2418	40.96	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
2419	40.96	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
2420	40.96	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
2421	40.94	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
2422	40.93	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
2423	40.89	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
2424	40.88	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
2425	40.86	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
2426	40.86	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
2427	40.84	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
2428	40.81	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
2429	40.75	kd	CGS001-7157	TP53	-			
2430	40.66	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
2431	40.66	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
2432	40.65	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2433	40.63	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
2434	40.62	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
2435	40.62	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
2436	40.59	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
2437	40.58	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2438	40.56	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
2439	40.55	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
2440	40.53	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
2441	40.53	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
2442	40.52	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
2443	40.49	kd	CGS001-9687	GREB1	-			
2444	40.45	kd	CGS001-345	APOC3	Apolipoproteins			
2445	40.43	oe	ccsbBroad304_01613	STK11	LKB subfamily			
2446	40.42	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
2447	40.41	oe	ccsbBroad304_06648	CNOT3	-			
2448	40.35	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
2449	40.29	oe	ccsbBroad304_03917	RBKS	-			
2450	40.25	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
2451	40.21	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
2452	40.2	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
2453	40.15	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
2454	40.12	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
2455	40.12	kd	CGS001-1788	DNMT3A	Methyltransferases			
2456	40.09	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
2457	40.03	oe	ccsbBroad304_03037	TMEM97	-			
2458	40	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
2459	40	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
2460	39.98	oe	ccsbBroad304_01659	TERF1	-			
2461	39.97	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2462	39.93	kd	CGS001-8872	CDC123	-			
2463	39.92	oe	ccsbBroad304_00572	FKBP3	-			
2464	39.86	kd	CGS001-255738	PCSK9	Subtilisin			
2465	39.81	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
2466	39.81	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
2467	39.78	kd	CGS001-29763	PACSIN3	-			
2468	39.77	kd	CGS001-11157	LSM6	-			
2469	39.76	oe	ccsbBroad304_07768	NISCH	-			
2470	39.76	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
2471	39.75	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
2472	39.75	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2473	39.75	kd	CGS001-8802	SUCLG1	-			
2474	39.75	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
2475	39.74	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
2476	39.73	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
2477	39.59	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
2478	39.56	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
2479	39.55	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
2480	39.55	oe	ccsbBroad304_01371	RALA	-			
2481	39.5	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
2482	39.5	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
2483	39.5	oe	ccsbBroad304_03739	NRIP3	-			
2484	39.5	kd	CGS001-6204	RPS10	S ribosomal proteins			
2485	39.46	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
2486	39.45	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
2487	39.44	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
2488	39.44	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
2489	39.42	kd	CGS001-4190	MDH1	-			
2490	39.42	kd	CGS001-56922	MCCC1	-			
2491	39.4	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
2492	39.4	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
2493	39.38	oe	ccsbBroad304_07252	DGKZ	-			
2494	39.38	oe	ccsbBroad304_08055	ATP5S	-			
2495	39.38	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
2496	39.29	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
2497	39.26	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2498	39.25	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
2499	39.22	kd	CGS001-55163	PNPO	-			
2500	39.21	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
2501	39.19	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
2502	39.19	kd	CGS001-4282	MIF	-			
2503	39.13	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
2504	39.13	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
2505	39.12	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
2506	39.09	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
2507	39.05	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
2508	39.05	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
2509	39.04	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
2510	39.04	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
2511	38.99	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
2512	38.96	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
2513	38.94	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
2514	38.91	oe	ccsbBroad304_03386	SPA17	-			
2515	38.88	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
2516	38.87	kd	CGS001-8431	NR0B2	DAX-like receptors			
2517	38.85	cc		PPAR receptor agonist	-			
2518	38.82	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
2519	38.76	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
2520	38.75	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2521	38.68	oe	ccsbBroad304_07515	GFPT2	-			
2522	38.67	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
2523	38.67	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
2524	38.65	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
2525	38.65	oe	ccsbBroad304_06720	PHYH	-			
2526	38.63	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
2527	38.62	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
2528	38.6	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
2529	38.59	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
2530	38.5	oe	ccsbBroad304_02554	TRAFD1	-			
2531	38.49	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
2532	38.46	kd	CGS001-23710	GABARAPL1	-			
2533	38.42	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
2534	38.39	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
2535	38.34	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
2536	38.34	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
2537	38.32	oe	ccsbBroad304_01150	PCCB	Carboxylases			
2538	38.32	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
2539	38.31	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
2540	38.3	oe	ccsbBroad304_02922	TES	-			
2541	38.27	oe	ccsbBroad304_07349	MAP7	-			
2542	38.27	oe	ccsbBroad304_06367	HK1	-			
2543	38.22	oe	ccsbBroad304_01066	NDUFA4	-			
2544	38.21	kd	CGS001-5579	PRKCB	Alpha subfamily			
2545	38.2	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
2546	38.12	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
2547	38.1	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
2548	38.09	oe	ccsbBroad304_01166	PDK2	PDHK family			
2549	38.08	oe	ccsbBroad304_05758	ACADSB	-			
2550	38.07	kd	CGS001-93594	WDR67	-			
2551	38.05	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
2552	38.01	kd	CGS001-29937	NENF	-			
2553	38.01	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2554	38	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
2555	37.98	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
2556	37.93	kd	CGS001-5053	PAH	Amino acid hydroxylases			
2557	37.93	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
2558	37.9	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
2559	37.83	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
2560	37.76	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
2561	37.75	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
2562	37.74	oe	ccsbBroad304_07238	STK24	YSK subfamily			
2563	37.65	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
2564	37.63	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
2565	37.62	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
2566	37.59	kd	CGS001-9847	KIAA0528	-			
2567	37.58	oe	ccsbBroad304_06695	PCK2	-			
2568	37.56	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
2569	37.55	kd	CGS001-5253	PHF2	Histone demethylases			
2570	37.53	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
2571	37.51	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
2572	37.51	kd	CGS001-4300	MLLT3	-			
2573	37.48	kd	CGS001-10329	TMEM5	-			
2574	37.47	cc		Interleukins GOF	-			
2575	37.47	oe	ccsbBroad304_03980	DCLRE1B	-			
2576	37.47	kd	CGS001-2017	CTTN	-			
2577	37.45	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
2578	37.44	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
2579	37.44	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
2580	37.43	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
2581	37.39	kd	CGS001-5898	RALA	-			
2582	37.38	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
2583	37.38	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2584	37.38	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
2585	37.35	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
2586	37.34	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
2587	37.34	kd	CGS001-51070	NOSIP	-			
2588	37.33	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
2589	37.31	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
2590	37.31	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
2591	37.28	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
2592	37.24	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
2593	37.24	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
2594	37.23	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
2595	37.22	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
2596	37.22	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
2597	37.13	kd	CGS001-7292	TNFSF4	CD molecules			
2598	37.09	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
2599	37.08	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2600	37.06	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
2601	37.04	kd	CGS001-51734	SEPX1	-			
2602	37.01	oe	ccsbBroad304_02804	KLHDC2	-			
2603	36.95	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
2604	36.95	kd	CGS001-23030	KDM4B	Histone demethylases			
2605	36.94	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
2606	36.93	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
2607	36.92	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
2608	36.91	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
2609	36.9	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
2610	36.9	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
2611	36.9	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
2612	36.89	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
2613	36.88	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
2614	36.87	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
2615	36.86	oe	ccsbBroad304_07557	NAMPT	-			
2616	36.85	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
2617	36.8	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
2618	36.79	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
2619	36.79	kd	CGS001-3033	HADH	-			
2620	36.77	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
2621	36.76	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
2622	36.73	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
2623	36.7	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
2624	36.67	kd	CGS001-3927	LASP1	-			
2625	36.67	kd	CGS001-662	BNIP1	-			
2626	36.66	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
2627	36.66	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
2628	36.64	oe	ccsbBroad304_02372	SPRY1	-			
2629	36.61	oe	ccsbBroad304_00991	MDH1	-			
2630	36.61	oe	ccsbBroad304_00063	AMPD2	-			
2631	36.61	kd	CGS001-3978	LIG1	-			
2632	36.56	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
2633	36.54	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
2634	36.53	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
2635	36.5	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
2636	36.5	kd	CGS001-6285	S100B	EF-hand domain containing			
2637	36.5	kd	CGS001-32	ACACB	Carboxylases			
2638	36.47	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
2639	36.46	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
2640	36.46	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
2641	36.46	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
2642	36.44	kd	CGS001-51071	DERA	-			
2643	36.43	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
2644	36.42	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
2645	36.39	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
2646	36.39	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
2647	36.38	kd	CGS001-93185	IGSF8	CD molecules			
2648	36.38	kd	CGS001-9131	AIFM1	-			
2649	36.37	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
2650	36.36	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
2651	36.27	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
2652	36.24	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
2653	36.22	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
2654	36.2	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
2655	36.19	kd	CGS001-2956	MSH6	-			
2656	36.09	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
2657	36.07	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
2658	36.04	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
2659	36.04	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
2660	35.96	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
2661	35.93	kd	CGS001-28511	NKIRAS2	-			
2662	35.82	kd	CGS001-84923	FAM104A	-			
2663	35.78	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
2664	35.75	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
2665	35.72	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
2666	35.61	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
2667	35.58	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
2668	35.57	oe	ccsbBroad304_01347	RAD1	-			
2669	35.56	kd	CGS001-55893	ZNF395	Zinc fingers, C2H2-type			
2670	35.55	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
2671	35.55	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
2672	35.52	oe	ccsbBroad304_07727	LIAS	-			
2673	35.47	kd	CGS001-169841	ZNF169	Zinc fingers, C2H2-type			
2674	35.42	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
2675	35.4	oe	ccsbBroad304_02838	SDF2L1	-			
2676	35.39	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
2677	35.39	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
2678	35.31	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
2679	35.29	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
2680	35.22	oe	ccsbBroad304_00423	DAXX	-			
2681	35.21	kd	CGS001-7852	CXCR4	Chemokine receptors			
2682	35.2	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
2683	35.18	kd	CGS001-1026	CDKN1A	-			
2684	35.18	kd	CGS001-6722	SRF	-			
2685	35.12	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
2686	35.11	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
2687	35.11	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
2688	35.1	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
2689	35.09	kd	CGS001-57222	ERGIC1	-			
2690	35.08	kd	CGS001-4482	MSRA	-			
2691	35.04	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2692	35.04	kd	CGS001-3034	HAL	-			
2693	35.03	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
2694	35.01	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
2695	34.98	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
2696	34.98	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
2697	34.97	oe	ccsbBroad304_07287	HYAL2	-			
2698	34.92	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
2699	34.92	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
2700	34.9	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
2701	34.89	oe	ccsbBroad304_03040	NKIRAS2	-			
2702	34.85	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
2703	34.84	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
2704	34.8	kd	CGS001-11182	SLC2A6	Solute carriers			
2705	34.77	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2706	34.74	oe	ccsbBroad304_05547	TMEM110	-			
2707	34.74	kd	CGS001-4602	MYB	-			
2708	34.73	oe	ccsbBroad304_00486	EFNB2	Ephrins			
2709	34.73	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
2710	34.69	oe	ccsbBroad304_00179	BTG1	-			
2711	34.69	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
2712	34.65	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2713	34.63	kd	CGS001-24140	FTSJ1	-			
2714	34.61	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
2715	34.6	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
2716	34.58	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
2717	34.56	oe	ccsbBroad304_03232	VPS28	-			
2718	34.56	kd	CGS001-84971	ATG4D	-			
2719	34.55	kd	CGS001-81848	SPRY4	-			
2720	34.54	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
2721	34.53	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
2722	34.51	oe	ccsbBroad304_00614	GAMT	-			
2723	34.48	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
2724	34.48	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
2725	34.41	oe	ccsbBroad304_07024	SYK	Syk family			
2726	34.38	cc		KCNJ11 modulator	-			
2727	34.38	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
2728	34.34	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
2729	34.33	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
2730	34.32	oe	ccsbBroad304_06435	RBPJ	-			
2731	34.27	kd	CGS001-3676	ITGA4	Integrins			
2732	34.26	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
2733	34.23	oe	ccsbBroad304_03808	ERGIC1	-			
2734	34.2	oe	ccsbBroad304_02368	TIMM17B	-			
2735	34.18	kd	CGS001-8435	SOAT2	-			
2736	34.18	kd	CGS001-5906	RAP1A	-			
2737	34.15	kd	CGS001-6117	RPA1	-			
2738	34.12	kd	CGS001-57018	CCNL1	-			
2739	34.11	kd	CGS001-5891	MOK	RCK family			
2740	34.1	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
2741	34.07	oe	ccsbBroad304_02500	RRAGA	-			
2742	34.05	oe	ccsbBroad304_03112	NENF	-			
2743	34.02	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
2744	34.01	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
2745	34	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
2746	33.94	oe	ccsbBroad304_08023	EIF2C1	-			
2747	33.94	kd	CGS001-5831	PYCR1	-			
2748	33.92	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
2749	33.91	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
2750	33.89	kd	CGS001-55837	EAPP	-			
2751	33.89	kd	CGS001-8453	CUL2	-			
2752	33.88	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
2753	33.87	kd	CGS001-5004	ORM1	Lipocalins			
2754	33.86	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
2755	33.82	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
2756	33.8	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
2757	33.8	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
2758	33.8	kd	CGS001-23344	ESYT1	Synaptotagmins			
2759	33.79	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2760	33.79	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
2761	33.77	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
2762	33.76	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
2763	33.73	kd	CGS001-6258	RXRG	Retinoid X receptors			
2764	33.72	kd	CGS001-337867	UBAC2	-			
2765	33.69	oe	ccsbBroad304_04891	TMEM174	-			
2766	33.67	kd	CGS001-6342	SCP2	-			
2767	33.67	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
2768	33.62	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
2769	33.62	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
2770	33.61	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
2771	33.56	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2772	33.56	kd	CGS001-27034	ACAD8	-			
2773	33.52	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
2774	33.45	oe	ccsbBroad304_00034	AES	-			
2775	33.41	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
2776	33.25	kd	CGS001-59286	UBL5	-			
2777	33.24	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2778	33.21	oe	ccsbBroad304_00865	ILF2	-			
2779	33.2	oe	ccsbBroad304_00665	GOT1	-			
2780	33.2	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
2781	33.18	oe	ccsbBroad304_02002	RNMT	-			
2782	33.13	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
2783	33.08	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
2784	33.02	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
2785	33.01	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
2786	32.99	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
2787	32.96	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2788	32.93	kd	CGS001-9531	BAG3	-			
2789	32.85	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
2790	32.83	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
2791	32.83	kd	CGS001-4303	FOXO4	Forkhead boxes			
2792	32.81	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
2793	32.75	kd	CGS001-624	BDKRB2	Bradykinin receptors			
2794	32.74	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
2795	32.71	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2796	32.69	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
2797	32.66	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2798	32.66	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
2799	32.62	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
2800	32.6	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
2801	32.59	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
2802	32.57	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
2803	32.56	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
2804	32.55	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
2805	32.5	oe	ccsbBroad304_01392	TRIM27	-			
2806	32.47	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
2807	32.46	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
2808	32.45	kd	CGS001-55214	LEPREL1	-			
2809	32.44	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
2810	32.42	kd	CGS001-114785	MBD6	-			
2811	32.38	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
2812	32.38	kd	CGS001-4151	MB	-			
2813	32.37	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2814	32.35	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
2815	32.35	oe	ccsbBroad304_00183	C1S	Complement system			
2816	32.34	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
2817	32.32	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
2818	32.31	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2819	32.25	kd	CGS001-3638	INSIG1	-			
2820	32.21	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
2821	32.2	oe	ccsbBroad304_01675	TK1	-			
2822	32.17	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
2823	32.08	kd	CGS001-10046	MAMLD1	-			
2824	32.03	oe	ccsbBroad304_12008	NLK	nmo subfamily			
2825	32.03	kd	CGS001-185	AGTR1	Angiotensin receptors			
2826	32.02	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
2827	32.01	kd	CGS001-4194	MDM4	-			
2828	31.94	oe	ccsbBroad304_02506	EBP	-			
2829	31.89	oe	ccsbBroad304_02306	PQBP1	-			
2830	31.89	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
2831	31.76	kd	CGS001-896	CCND3	-			
2832	31.73	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
2833	31.7	kd	CGS001-9447	AIM2	-			
2834	31.68	kd	CGS001-3800	KIF5C	Kinesins			
2835	31.68	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2836	31.62	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
2837	31.6	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
2838	31.58	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
2839	31.58	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
2840	31.55	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
2841	31.5	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
2842	31.5	kd	CGS001-2335	FN1	Endogenous ligands			
2843	31.47	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
2844	31.44	oe	ccsbBroad304_04655	TRIM9	-			
2845	31.39	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
2846	31.39	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
2847	31.39	kd	CGS001-5105	PCK1	-			
2848	31.34	kd	CGS001-23647	ARFIP2	-			
2849	31.33	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2850	31.33	kd	CGS001-29982	NRBF2	-			
2851	31.24	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
2852	31.24	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
2853	31.22	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
2854	31.2	oe	ccsbBroad304_05135	PARP15	-			
2855	31.1	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
2856	31.05	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
2857	31.03	kd	CGS001-6469	SHH	-			
2858	31.02	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2859	30.94	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
2860	30.92	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
2861	30.92	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
2862	30.92	kd	CGS001-1756	DMD	-			
2863	30.91	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
2864	30.9	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
2865	30.88	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
2866	30.87	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2867	30.86	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
2868	30.83	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
2869	30.82	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
2870	30.8	oe	ccsbBroad304_05981	CDO1	-			
2871	30.78	kd	CGS001-5883	RAD9A	-			
2872	30.73	oe	ccsbBroad304_08694	TBX20	T-boxes			
2873	30.73	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2874	30.72	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
2875	30.65	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
2876	30.62	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
2877	30.6	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
2878	30.6	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
2879	30.59	kd	CGS001-5202	PFDN2	-			
2880	30.57	kd	CGS001-4299	AFF1	-			
2881	30.56	kd	CGS001-64094	SMOC2	EF-hand domain containing			
2882	30.53	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
2883	30.51	kd	CGS001-2295	FOXF2	Forkhead boxes			
2884	30.44	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
2885	30.43	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
2886	30.41	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
2887	30.36	kd	CGS001-9128	PRPF4	WD repeat domain containing			
2888	30.35	oe	ccsbBroad304_00225	CAT	-			
2889	30.35	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
2890	30.35	kd	CGS001-8428	STK24	YSK subfamily			
2891	30.34	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
2892	30.26	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
2893	30.26	kd	CGS001-4547	MTTP	-			
2894	30.22	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
2895	30.19	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
2896	30.18	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
2897	30.16	oe	ccsbBroad304_03934	LEPRE1	-			
2898	30.16	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
2899	30.16	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
2900	30.15	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
2901	30.14	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
2902	30.14	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
2903	30.09	oe	ccsbBroad304_06549	SMAD3	SMADs			
2904	30.07	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
2905	30.05	kd	CGS001-6461	SHB	SH2 domain containing			
2906	30.04	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
2907	30.01	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
2908	29.99	kd	CGS001-116519	APOA5	Apolipoproteins			
2909	29.98	kd	CGS001-9200	PTPLA	-			
2910	29.97	kd	CGS001-4016	LOXL1	-			
2911	29.94	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2912	29.91	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
2913	29.9	kd	CGS001-3663	IRF5	-			
2914	29.9	kd	CGS001-29083	GTPBP8	-			
2915	29.9	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
2916	29.83	kd	CGS001-861	RUNX1	-			
2917	29.79	kd	CGS001-7374	UNG	-			
2918	29.67	kd	CGS001-1737	DLAT	-			
2919	29.63	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
2920	29.59	kd	CGS001-2010	EMD	-			
2921	29.57	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
2922	29.53	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
2923	29.51	cc		Serotonin receptor antagonist	-			
2924	29.5	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
2925	29.45	oe	ccsbBroad304_00098	ARG1	Arginase			
2926	29.39	kd	CGS001-55968	NSFL1C	UBX domain containing			
2927	29.38	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2928	29.36	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
2929	29.34	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
2930	29.34	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
2931	29.33	oe	ccsbBroad304_00725	HADHA	-			
2932	29.32	kd	CGS001-5909	RAP1GAP	-			
2933	29.31	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
2934	29.3	kd	CGS001-57157	PHTF2	-			
2935	29.25	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
2936	29.24	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
2937	29.22	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
2938	29.21	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
2939	29.19	kd	CGS001-11340	EXOSC8	-			
2940	29.18	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
2941	29.04	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2942	29.02	kd	CGS001-10657	KHDRBS1	-			
2943	29.01	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
2944	29	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
2945	28.98	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
2946	28.98	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
2947	28.98	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
2948	28.85	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
2949	28.83	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
2950	28.8	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
2951	28.76	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
2952	28.75	oe	ccsbBroad304_04194	ELL3	-			
2953	28.75	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
2954	28.67	kd	CGS001-1154	CISH	SH2 domain containing			
2955	28.61	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2956	28.5	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
2957	28.5	oe	ccsbBroad304_06420	ICAM3	CD molecules			
2958	28.48	kd	CGS001-2550	GABBR1	GABA receptors			
2959	28.43	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
2960	28.42	kd	CGS001-26128	KIAA1279	-			
2961	28.39	kd	CGS001-283450	C12ORF51	-			
2962	28.36	kd	CGS001-1534	CYB561	Cytochrome b genes			
2963	28.35	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
2964	28.34	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
2965	28.32	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
2966	28.32	kd	CGS001-116931	MED12L	-			
2967	28.31	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
2968	28.3	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
2969	28.26	kd	CGS001-55577	NAGK	-			
2970	28.2	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
2971	28.1	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
2972	28.08	oe	ccsbBroad304_04490	RSPH1	-			
2973	28.04	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
2974	28.04	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
2975	28.02	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
2976	28.01	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
2977	27.98	cc		DNA synthesis inhibitor	-			
2978	27.82	kd	CGS001-286380	FOXD4L3	-			
2979	27.81	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
2980	27.75	kd	CGS001-10253	SPRY2	-			
2981	27.72	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
2982	27.71	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2983	27.67	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
2984	27.61	kd	CGS001-57819	LSM2	-			
2985	27.51	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
2986	27.49	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
2987	27.48	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
2988	27.45	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
2989	27.45	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
2990	27.44	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
2991	27.4	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
2992	27.4	kd	CGS001-5708	PSMD2	Proteasome subunits			
2993	27.39	kd	CGS001-661	POLR3D	RNA polymerase subunits			
2994	27.36	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
2995	27.33	kd	CGS001-8467	SMARCA5	-			
2996	27.31	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2997	27.31	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
2998	27.3	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
2999	27.3	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
3000	27.23	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
3001	27.23	kd	CGS001-5684	PSMA3	Proteasome subunits			
3002	27.21	kd	CGS001-4925	NUCB2	EF-hand domain containing			
3003	27.17	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
3004	27.17	kd	CGS001-8731	RNMT	-			
3005	27.13	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
3006	27.13	kd	CGS001-7471	WNT1	Endogenous ligands			
3007	27.12	kd	CGS001-64428	NARFL	-			
3008	27.11	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
3009	27.09	kd	CGS001-29116	MYLIP	-			
3010	27.06	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
3011	27.05	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
3012	27.05	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
3013	27.04	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
3014	26.95	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
3015	26.77	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
3016	26.68	kd	CGS001-57147	SCYL3	-			
3017	26.67	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3018	26.61	kd	CGS001-10923	SUB1	-			
3019	26.6	kd	CGS001-9655	SOCS5	SH2 domain containing			
3020	26.57	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
3021	26.51	oe	ccsbBroad304_02133	CD83	CD molecules			
3022	26.5	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
3023	26.5	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
3024	26.46	kd	CGS001-7360	UGP2	-			
3025	26.46	kd	CGS001-3988	LIPA	-			
3026	26.42	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3027	26.38	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
3028	26.37	cc		Bacterial DNA gyrase inhibitor	-			
3029	26.36	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
3030	26.33	oe	ccsbBroad304_01152	PCNA	-			
3031	26.33	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
3032	26.31	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3033	26.31	kd	CGS001-4179	CD46	CD molecules			
3034	26.22	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
3035	26.16	kd	CGS001-8801	SUCLG2	-			
3036	26.11	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
3037	26.1	kd	CGS001-10312	TCIRG1	ATPases / V-type			
3038	26.09	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
3039	26.07	cc		Reverse transcriptase inhibitor	-			
3040	26.01	oe	ccsbBroad304_13880	IDH3G	-			
3041	26	kd	CGS001-7917	BAG6	-			
3042	25.96	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
3043	25.87	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
3044	25.87	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
3045	25.86	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
3046	25.86	kd	CGS001-22930	RAB3GAP1	-			
3047	25.82	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
3048	25.8	kd	CGS001-8841	HDAC3	Histone deacetylases			
3049	25.77	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
3050	25.75	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
3051	25.68	kd	CGS001-58528	RRAGD	-			
3052	25.64	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
3053	25.64	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
3054	25.64	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
3055	25.6	kd	CGS001-823	CAPN1	EF-hand domain containing			
3056	25.57	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
3057	25.51	kd	CGS001-4507	MTAP	-			
3058	25.47	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3059	25.46	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
3060	25.45	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
3061	25.38	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
3062	25.36	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
3063	25.28	oe	ccsbBroad304_00811	ICAM1	CD molecules			
3064	25.21	kd	CGS001-27097	TAF5L	WD repeat domain containing			
3065	25.19	kd	CGS001-1950	EGF	-			
3066	25.13	kd	CGS001-55206	SBNO1	-			
3067	25.07	oe	ccsbBroad304_06836	RAD23B	-			
3068	25.02	cc		Akt Signaling LOF	-			
3069	24.94	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
3070	24.92	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
3071	24.89	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
3072	24.83	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3073	24.8	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
3074	24.78	oe	ccsbBroad304_03182	GLOD4	-			
3075	24.76	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
3076	24.75	kd	CGS001-6714	SRC	Src family			
3077	24.73	oe	ccsbBroad304_07528	DMTF1	-			
3078	24.6	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3079	24.4	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
3080	24.37	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
3081	24.36	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
3082	24.32	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
3083	24.31	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
3084	24.28	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
3085	24.23	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
3086	24.15	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
3087	24.08	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
3088	24.04	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
3089	24.03	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
3090	23.99	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
3091	23.89	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
3092	23.69	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
3093	23.61	oe	ccsbBroad304_03119	C16ORF5	-			
3094	23.57	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
3095	23.57	oe	ccsbBroad304_06862	RGS3	-			
3096	23.57	kd	CGS001-5355	PLP2	-			
3097	23.53	oe	ccsbBroad304_07761	CORO1A	Coronins			
3098	23.4	kd	CGS001-5894	RAF1	RAF family			
3099	23.39	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
3100	23.37	kd	CGS001-2919	CXCL1	Endogenous ligands			
3101	23.33	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
3102	23.28	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
3103	23.26	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3104	23.19	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
3105	23.18	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
3106	23.1	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
3107	23.07	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
3108	23.07	kd	CGS001-55379	LRRC59	-			
3109	23.04	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
3110	23	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
3111	22.99	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
3112	22.98	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
3113	22.86	kd	CGS001-182	JAG1	CD molecules			
3114	22.82	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
3115	22.6	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
3116	22.54	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3117	22.52	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
3118	22.49	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
3119	22.48	kd	CGS001-6201	RPS7	S ribosomal proteins			
3120	22.45	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
3121	22.41	kd	CGS001-2864	FFAR1	Fatty acid receptors			
3122	22.32	kd	CGS001-7078	TIMP3	-			
3123	22.23	kd	CGS001-5621	PRNP	CD molecules			
3124	22.22	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
3125	22.22	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
3126	22.21	oe	ccsbBroad304_02416	TUBB4B	-			
3127	22.17	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
3128	22.17	kd	CGS001-271	AMPD2	-			
3129	22.1	kd	CGS001-6050	RNH1	-			
3130	22	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
3131	21.96	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
3132	21.89	kd	CGS001-5613	PRKX	Protein kinase A			
3133	21.82	kd	CGS001-4436	MSH2	-			
3134	21.8	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
3135	21.75	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3136	21.73	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
3137	21.71	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
3138	21.68	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
3139	21.65	cc		Ubiquitin-specific peptidases LOF	-			
3140	21.63	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3141	21.54	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
3142	21.36	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
3143	21.28	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
3144	21.18	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
3145	21.11	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
3146	21.02	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
3147	20.72	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
3148	20.67	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
3149	20.54	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
3150	20.38	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
3151	20.28	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
3152	20.2	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
3153	19.77	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
3154	19.75	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
3155	19.65	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
3156	19.53	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
3157	19.52	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
3158	19.39	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
3159	19.37	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3160	19.32	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
3161	19.17	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
3162	18.9	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
3163	18.85	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
3164	18.6	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
3165	18.33	kd	CGS001-4976	OPA1	-			
3166	18.25	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
3167	18.17	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
3168	18.15	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3169	18.13	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
3170	18.12	cc		Tubulin inhibitor	-			
3171	18.1	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
3172	17.92	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3173	17.6	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
3174	17.56	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
3175	17.35	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3176	17.33	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
3177	17.25	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
3178	17.16	oe	ccsbBroad304_02452	NXF1	-			
3179	17.04	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
3180	16.99	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
3181	16.91	kd	CGS001-6774	STAT3	SH2 domain containing			
3182	16.84	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
3183	16.74	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
3184	16.69	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
3185	16.37	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
3186	16.2	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
3187	16.14	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
3188	15.93	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
3189	15.85	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
3190	15.66	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
3191	15.57	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
3192	15.46	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
3193	15.41	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
3194	15.32	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
3195	15.12	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
3196	15	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
3197	14.87	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3198	14.56	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3199	14.47	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
3200	14.37	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
3201	14.3	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
3202	14.25	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
3203	14.24	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
3204	14.17	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
3205	14.06	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
3206	13.86	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3207	13.71	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
3208	13.62	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
3209	13.48	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
3210	13.27	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
3211	13.27	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
3212	13.16	kd	CGS001-3479	IGF1	Endogenous ligands			
3213	12.8	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
3214	12.62	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
3215	12.35	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
3216	12.15	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
3217	11.88	cc		Angiotensin receptor antagonist	-			
3218	11.45	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
3219	11.36	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
3220	11.07	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
3221	10.83	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
3222	10.76	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
3223	10.34	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
3224	10.29	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3225	10.24	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
3226	10.01	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3227	9.94	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
3228	9.1	cc		Mediator complex LOF	-			
3229	8.96	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
3230	8.81	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
3231	7.61	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
3232	7.42	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3233	6.74	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3234	5.88	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
3235	-7.33	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
3236	-7.55	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
3237	-8.4	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3238	-8.65	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
3239	-8.88	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
3240	-9.36	cc		SRY LOF	-			
3241	-9.4	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
3242	-9.44	cc		Progesterone receptor antagonist	-			
3243	-9.64	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
3244	-9.8	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
3245	-10.07	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3246	-10.11	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
3247	-10.6	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
3248	-11.38	cc		BMP Signaling LOF	-			
3249	-11.46	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
3250	-11.78	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
3251	-12.23	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
3252	-12.53	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
3253	-12.77	cc		Wnt family GOF	-			
3254	-12.85	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
3255	-12.88	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
3256	-12.91	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
3257	-13.09	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
3258	-13.09	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
3259	-13.54	kd	CGS001-50808	AK3	-			
3260	-13.66	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
3261	-13.68	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
3262	-13.72	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
3263	-13.72	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
3264	-13.92	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
3265	-14.07	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
3266	-14.13	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
3267	-14.43	kd	CGS001-1633	DCK	-			
3268	-14.48	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
3269	-14.66	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
3270	-14.83	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
3271	-15.26	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
3272	-15.41	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
3273	-15.42	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
3274	-15.62	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
3275	-15.67	kd	CGS001-5979	RET	Type XIV RTKs: RET			
3276	-16.07	cc		Bacterial cell wall synthesis inhibitor	-			
3277	-16.12	kd	CGS001-169436	C9ORF96	-			
3278	-16.17	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
3279	-16.18	kd	CGS001-6776	STAT5A	SH2 domain containing			
3280	-16.23	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
3281	-16.68	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
3282	-17.11	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
3283	-17.19	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
3284	-17.2	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
3285	-17.29	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
3286	-17.38	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
3287	-17.38	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
3288	-17.41	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
3289	-17.43	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
3290	-17.45	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3291	-17.51	kd	CGS001-7965	AIMP2	-			
3292	-17.61	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
3293	-17.65	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
3294	-17.66	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
3295	-17.71	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
3296	-17.77	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
3297	-17.99	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
3298	-18.17	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
3299	-18.18	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
3300	-18.33	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
3301	-18.4	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
3302	-18.45	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
3303	-18.8	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
3304	-18.85	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
3305	-18.94	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
3306	-19.19	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
3307	-19.29	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
3308	-19.3	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
3309	-19.34	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
3310	-19.42	kd	CGS001-4697	NDUFA4	-			
3311	-19.48	kd	CGS001-4439	MSH5	-			
3312	-19.55	kd	CGS001-1111	CHEK1	CHK1 subfamily			
3313	-19.66	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
3314	-19.8	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3315	-19.82	oe	ccsbBroad304_01485	SC5DL	-			
3316	-19.82	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
3317	-19.86	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
3318	-19.86	kd	CGS001-54805	CNNM2	-			
3319	-19.9	oe	ccsbBroad304_05745	CD24	CD molecules			
3320	-19.9	kd	CGS001-51586	MED15	-			
3321	-19.93	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
3322	-20.03	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
3323	-20.09	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
3324	-20.12	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
3325	-20.12	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3326	-20.14	kd	CGS001-10314	LANCL1	-			
3327	-20.21	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
3328	-20.32	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3329	-20.32	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
3330	-20.36	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
3331	-20.5	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
3332	-20.5	oe	ccsbBroad304_06140	EEF1D	-			
3333	-20.52	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
3334	-20.56	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
3335	-20.62	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
3336	-20.69	kd	CGS001-54861	SNRK	SNRK subfamily			
3337	-20.73	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
3338	-20.77	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
3339	-20.79	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
3340	-20.85	oe	ccsbBroad304_10846	GGT1	CD molecules			
3341	-20.94	kd	CGS001-7187	TRAF3	-			
3342	-20.95	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
3343	-20.96	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
3344	-20.97	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3345	-21.09	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
3346	-21.12	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
3347	-21.17	kd	CGS001-9232	PTTG1	-			
3348	-21.18	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3349	-21.21	oe	ccsbBroad304_05907	BUB1B	Bub family			
3350	-21.21	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
3351	-21.21	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
3352	-21.24	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
3353	-21.26	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
3354	-21.36	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
3355	-21.42	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
3356	-21.44	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
3357	-21.47	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
3358	-21.51	kd	CGS001-4069	LYZ	-			
3359	-21.51	kd	CGS001-2203	FBP1	-			
3360	-21.62	oe	ccsbBroad304_02278	THRAP3	-			
3361	-21.7	kd	CGS001-6871	TADA2A	-			
3362	-21.79	kd	CGS001-2782	GNB1	WD repeat domain containing			
3363	-21.84	kd	CGS001-55038	CDCA4	-			
3364	-21.88	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
3365	-21.95	cc		Histone deacetylases LOF	-			
3366	-21.98	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
3367	-22	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
3368	-22.03	cc		Purinergic receptors P2Y GOF	-			
3369	-22.05	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
3370	-22.07	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
3371	-22.07	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
3372	-22.09	kd	CGS001-513	ATP5D	ATPases / F-type			
3373	-22.15	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
3374	-22.16	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
3375	-22.19	oe	ccsbBroad304_06040	CRY1	-			
3376	-22.2	kd	CGS001-83933	HDAC10	Histone deacetylases			
3377	-22.22	kd	CGS001-83440	ADPGK	-			
3378	-22.25	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
3379	-22.3	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
3380	-22.36	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
3381	-22.45	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
3382	-22.49	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
3383	-22.49	kd	CGS001-5727	PTCH1	-			
3384	-22.5	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3385	-22.52	oe	ccsbBroad304_01605	SSX2	-			
3386	-22.54	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
3387	-22.6	kd	CGS001-2592	GALT	-			
3388	-22.66	oe	ccsbBroad304_06671	OPA1	-			
3389	-22.75	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3390	-22.8	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
3391	-22.83	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
3392	-22.85	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
3393	-22.86	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
3394	-22.87	oe	ccsbBroad304_01483	SAT1	-			
3395	-22.88	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
3396	-22.91	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
3397	-22.91	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
3398	-22.92	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
3399	-22.96	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
3400	-22.97	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
3401	-22.98	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
3402	-22.98	kd	CGS001-84515	MCM8	-			
3403	-22.99	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
3404	-22.99	kd	CGS001-2588	GALNS	Arylsulfatase family			
3405	-23.02	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
3406	-23.05	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
3407	-23.07	oe	ccsbBroad304_09578	PASD1	-			
3408	-23.1	oe	ccsbBroad304_00085	APRT	-			
3409	-23.13	kd	CGS001-54407	SLC38A2	System A-like transporters			
3410	-23.19	oe	ccsbBroad304_00501	EMD	-			
3411	-23.24	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
3412	-23.24	kd	CGS001-2760	GM2A	-			
3413	-23.32	kd	CGS001-475	ATOX1	-			
3414	-23.33	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
3415	-23.36	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
3416	-23.36	kd	CGS001-317705	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
3417	-23.42	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
3418	-23.42	kd	CGS001-11232	POLG2	DNA polymerases			
3419	-23.53	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
3420	-23.53	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
3421	-23.55	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
3422	-23.57	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
3423	-23.66	kd	CGS001-6643	SNX2	Sorting nexins			
3424	-23.73	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
3425	-23.73	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
3426	-23.76	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
3427	-23.79	oe	ccsbBroad304_00070	ANXA5	Annexins			
3428	-23.92	cp	BRD-K10065684	dantron	Laxative			Laxative
3429	-23.97	kd	CGS001-29888	STRN4	WD repeat domain containing			
3430	-24	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
3431	-24.01	kd	CGS001-9637	FEZ2	-			
3432	-24.04	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
3433	-24.04	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
3434	-24.05	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
3435	-24.06	oe	ccsbBroad304_00226	CAV1	-			
3436	-24.34	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
3437	-24.34	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
3438	-24.36	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
3439	-24.37	kd	CGS001-10497	UNC13B	-			
3440	-24.38	oe	ccsbBroad304_07887	GCAT	-			
3441	-24.44	kd	CGS001-6217	RPS16	S ribosomal proteins			
3442	-24.47	kd	CGS001-7020	TFAP2A	-			
3443	-24.48	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
3444	-24.57	oe	ccsbBroad304_07088	TP53	-			
3445	-24.58	oe	ccsbBroad304_02318	KIF20A	Kinesins			
3446	-24.6	kd	CGS001-55536	CDCA7L	-			
3447	-24.62	kd	CGS001-1827	RCAN1	-			
3448	-24.67	oe	ccsbBroad304_04649	ADC	-			
3449	-24.68	oe	ccsbBroad304_07094	TPMT	-			
3450	-24.68	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3451	-24.69	kd	CGS001-9354	UBE4A	U-box domain containing			
3452	-24.75	kd	CGS001-23509	POFUT1	Fucosyltransferases			
3453	-24.78	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
3454	-24.8	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
3455	-24.81	oe	ccsbBroad304_06180	ESD	-			
3456	-24.84	kd	CGS001-1284	COL4A2	Collagens			
3457	-24.85	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
3458	-24.85	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
3459	-24.87	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
3460	-24.87	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
3461	-24.89	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
3462	-24.92	kd	CGS001-11007	CCDC85B	-			
3463	-24.95	kd	CGS001-5688	PSMA7	Proteasome subunits			
3464	-24.96	oe	ccsbBroad304_07320	SQSTM1	-			
3465	-24.99	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
3466	-25.02	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
3467	-25.07	cc		P38 MAPK inhibitor	-			
3468	-25.1	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
3469	-25.15	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
3470	-25.16	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
3471	-25.19	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
3472	-25.19	kd	CGS001-23588	KLHDC2	-			
3473	-25.2	oe	ccsbBroad304_00651	GNAI3	-			
3474	-25.25	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
3475	-25.27	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
3476	-25.28	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
3477	-25.29	oe	ccsbBroad304_03773	CIAPIN1	-			
3478	-25.31	kd	CGS001-5934	RBL2	-			
3479	-25.35	kd	CGS001-35	ACADS	-			
3480	-25.39	oe	ccsbBroad304_02086	PDLIM1	-			
3481	-25.43	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
3482	-25.44	kd	CGS001-2597	GAPDH	-			
3483	-25.45	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
3484	-25.46	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
3485	-25.49	oe	ccsbBroad304_05192	SPRED2	-			
3486	-25.5	kd	CGS001-634	CEACAM1	CD molecules			
3487	-25.51	kd	CGS001-87	ACTN1	EF-hand domain containing			
3488	-25.56	kd	CGS001-58533	SNX6	Sorting nexins			
3489	-25.56	kd	CGS001-5565	PRKAB2	AMPK subfamily			
3490	-25.59	oe	ccsbBroad304_03235	TUBD1	Tubulins			
3491	-25.59	kd	CGS001-5562	PRKAA1	AMPK subfamily			
3492	-25.61	kd	CGS001-7296	TXNRD1	-			
3493	-25.66	oe	ccsbBroad304_00883	ISG20	-			
3494	-25.67	oe	ccsbBroad304_02399	TNIP1	-			
3495	-25.69	kd	CGS001-122618	PLD4	-			
3496	-25.77	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
3497	-25.8	oe	ccsbBroad304_06126	TSC22D3	-			
3498	-25.81	kd	CGS001-5257	PHKB	-			
3499	-25.81	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
3500	-25.81	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
3501	-25.82	kd	CGS001-4245	MGAT1	-			
3502	-25.82	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
3503	-25.85	oe	ccsbBroad304_04257	SPRY4	-			
3504	-25.87	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
3505	-25.88	kd	CGS001-204851	HIPK1	HIPK subfamily			
3506	-25.89	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
3507	-25.91	oe	ccsbBroad304_02919	KIAA1279	-			
3508	-25.93	oe	ccsbBroad304_06525	LIPA	-			
3509	-25.97	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
3510	-25.97	kd	CGS001-1070	CETN3	EF-hand domain containing			
3511	-25.97	kd	CGS001-183	AGT	Endogenous ligands			
3512	-25.99	oe	ccsbBroad304_07045	TEAD4	-			
3513	-26	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3514	-26.05	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
3515	-26.08	oe	ccsbBroad304_04399	PGBD1	-			
3516	-26.08	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
3517	-26.09	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
3518	-26.11	kd	CGS001-3956	LGALS1	Endogenous ligands			
3519	-26.12	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
3520	-26.13	oe	ccsbBroad304_01724	TTR	-			
3521	-26.15	oe	ccsbBroad304_00645	GCLM	-			
3522	-26.15	kd	CGS001-7358	UGDH	-			
3523	-26.18	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
3524	-26.2	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
3525	-26.26	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3526	-26.31	oe	ccsbBroad304_08480	PNPO	-			
3527	-26.31	kd	CGS001-6793	STK10	SLK subfamily			
3528	-26.33	kd	CGS001-31	ACACA	Carboxylases			
3529	-26.34	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3530	-26.39	kd	CGS001-2072	ERCC4	-			
3531	-26.41	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3532	-26.41	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
3533	-26.42	kd	CGS001-3821	KLRC1	CD molecules			
3534	-26.44	cc		GPCR Subset GOF	-			
3535	-26.45	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
3536	-26.53	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
3537	-26.53	kd	CGS001-8575	PRKRA	-			
3538	-26.54	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
3539	-26.55	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
3540	-26.59	kd	CGS001-55437	STRADB	STLK subfamily			
3541	-26.6	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
3542	-26.61	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3543	-26.62	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
3544	-26.64	oe	ccsbBroad304_07490	SCRN1	-			
3545	-26.65	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
3546	-26.66	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
3547	-26.66	kd	CGS001-4087	SMAD2	SMADs			
3548	-26.67	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
3549	-26.68	kd	CGS001-6446	SGK1	SGK family			
3550	-26.69	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
3551	-26.69	kd	CGS001-65263	PYCRL	-			
3552	-26.71	kd	CGS001-7088	TLE1	WD repeat domain containing			
3553	-26.71	kd	CGS001-24148	PRPF6	-			
3554	-26.78	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
3555	-26.78	oe	ccsbBroad304_07688	FAM114A2	-			
3556	-26.79	oe	ccsbBroad304_03767	TOMM22	-			
3557	-26.79	oe	ccsbBroad304_00881	IRF5	-			
3558	-26.81	oe	ccsbBroad304_02671	ECD	-			
3559	-26.84	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
3560	-26.87	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
3561	-26.87	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
3562	-26.87	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
3563	-26.88	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
3564	-26.88	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
3565	-26.94	kd	CGS001-1999	ELF3	ETS Transcription Factors			
3566	-26.96	oe	ccsbBroad304_03533	CDCA8	-			
3567	-26.98	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
3568	-26.99	oe	ccsbBroad304_01985	EIF3H	-			
3569	-26.99	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
3570	-26.99	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
3571	-27.02	kd	CGS001-1981	EIF4G1	Parkinson disease			
3572	-27.05	kd	CGS001-8804	CREG1	-			
3573	-27.09	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
3574	-27.11	kd	CGS001-3456	IFNB1	Interferons			
3575	-27.11	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
3576	-27.13	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
3577	-27.16	kd	CGS001-8833	GMPS	-			
3578	-27.16	kd	CGS001-8772	FADD	-			
3579	-27.2	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
3580	-27.22	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
3581	-27.23	kd	CGS001-2161	F12	Chymotrypsin			
3582	-27.24	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
3583	-27.25	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
3584	-27.26	oe	ccsbBroad304_00113	ASNS	-			
3585	-27.32	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
3586	-27.34	oe	ccsbBroad304_05890	BHMT	-			
3587	-27.36	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
3588	-27.37	kd	CGS001-308	ANXA5	Annexins			
3589	-27.37	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
3590	-27.38	kd	CGS001-9688	NUP93	-			
3591	-27.39	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
3592	-27.4	oe	ccsbBroad304_02285	MED6	-			
3593	-27.41	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
3594	-27.42	cc		Nucleophosmin inhibitor	-			
3595	-27.42	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
3596	-27.42	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
3597	-27.43	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
3598	-27.43	oe	ccsbBroad304_03155	DHH	-			
3599	-27.43	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
3600	-27.43	kd	CGS001-11267	SNF8	-			
3601	-27.43	kd	CGS001-51293	CD320	CD molecules			
3602	-27.44	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
3603	-27.44	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
3604	-27.48	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
3605	-27.51	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
3606	-27.54	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
3607	-27.57	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
3608	-27.61	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
3609	-27.62	cc		Wnt family LOF	-			
3610	-27.64	kd	CGS001-23650	TRIM29	-			
3611	-27.65	kd	CGS001-5378	PMS1	-			
3612	-27.65	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
3613	-27.67	oe	ccsbBroad304_08993	DHDDS	-			
3614	-27.68	kd	CGS001-10587	TXNRD2	-			
3615	-27.69	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
3616	-27.7	kd	CGS001-29105	C16ORF80	-			
3617	-27.74	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
3618	-27.74	kd	CGS001-382	ARF6	ADP-ribosylation factors			
3619	-27.79	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
3620	-27.8	oe	ccsbBroad304_05821	ANXA1	Annexins			
3621	-27.81	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
3622	-27.82	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
3623	-27.84	oe	ccsbBroad304_01640	TAF12	-			
3624	-27.84	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
3625	-27.85	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
3626	-27.85	kd	CGS001-6491	STIL	-			
3627	-27.87	oe	ccsbBroad304_03186	GMNN	-			
3628	-27.89	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
3629	-27.9	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
3630	-27.91	oe	ccsbBroad304_06651	NOV	-			
3631	-27.92	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
3632	-27.92	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
3633	-27.94	kd	CGS001-3832	KIF11	Kinesins			
3634	-27.95	oe	ccsbBroad304_01519	SET	-			
3635	-27.95	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
3636	-27.96	kd	CGS001-1948	EFNB2	Ephrins			
3637	-27.96	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
3638	-27.99	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
3639	-27.99	kd	CGS001-4086	SMAD1	SMADs			
3640	-28.01	kd	CGS001-11198	SUPT16H	-			
3641	-28.02	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
3642	-28.03	kd	CGS001-10198	MPHOSPH9	-			
3643	-28.05	kd	CGS001-1490	CTGF	-			
3644	-28.07	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
3645	-28.07	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
3646	-28.08	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
3647	-28.09	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
3648	-28.1	kd	CGS001-5160	PDHA1	-			
3649	-28.12	kd	CGS001-3269	HRH1	Histamine receptors			
3650	-28.14	oe	ccsbBroad304_02357	SSX3	-			
3651	-28.14	kd	CGS001-64750	SMURF2	-			
3652	-28.18	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
3653	-28.19	kd	CGS001-83729	INHBE	-			
3654	-28.23	cc		Progesterone receptor agonist	-			
3655	-28.25	kd	CGS001-1066	CES1	Carboxylesterases			
3656	-28.26	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
3657	-28.31	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
3658	-28.38	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
3659	-28.38	kd	CGS001-9791	PTDSS1	-			
3660	-28.38	kd	CGS001-4864	NPC1	-			
3661	-28.38	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3662	-28.39	oe	ccsbBroad304_01142	PAFAH1B2	-			
3663	-28.39	kd	CGS001-51447	IP6K2	-			
3664	-28.4	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
3665	-28.42	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
3666	-28.45	oe	ccsbBroad304_04534	HN1L	-			
3667	-28.45	kd	CGS001-283	ANG	Ribonucleases, RNase A			
3668	-28.47	oe	ccsbBroad304_02173	ATG5	-			
3669	-28.47	kd	CGS001-7477	WNT7B	Endogenous ligands			
3670	-28.47	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
3671	-28.48	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
3672	-28.51	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
3673	-28.51	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
3674	-28.53	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
3675	-28.6	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
3676	-28.64	kd	CGS001-2878	GPX3	-			
3677	-28.69	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
3678	-28.71	kd	CGS001-6827	SUPT4H1	-			
3679	-28.75	kd	CGS001-51160	VPS28	-			
3680	-28.76	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
3681	-28.78	oe	ccsbBroad304_02831	SGK3	SGK family			
3682	-28.79	kd	CGS001-80349	WDR61	WD repeat domain containing			
3683	-28.79	kd	CGS001-9797	TATDN2	-			
3684	-28.8	oe	ccsbBroad304_02702	MSRB2	-			
3685	-28.8	kd	CGS001-51805	COQ3	-			
3686	-28.82	kd	CGS001-10105	PPIF	-			
3687	-28.82	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
3688	-28.82	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
3689	-28.84	cc		Topoisomerase inhibitor	-			
3690	-28.84	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
3691	-28.91	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
3692	-28.94	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
3693	-28.97	kd	CGS001-6189	RPS3A	S ribosomal proteins			
3694	-28.99	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
3695	-29	oe	ccsbBroad304_00876	INSIG1	-			
3696	-29.01	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
3697	-29.07	kd	CGS001-5387	PMS2P3	-			
3698	-29.11	kd	CGS001-3176	HNMT	-			
3699	-29.11	kd	CGS001-351	APP	Endogenous ligands			
3700	-29.16	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
3701	-29.17	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
3702	-29.21	oe	ccsbBroad304_07178	ZFP112	-			
3703	-29.21	kd	CGS001-2212	FCGR2A	CD molecules			
3704	-29.22	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
3705	-29.22	kd	CGS001-1955	MEGF9	-			
3706	-29.23	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
3707	-29.23	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
3708	-29.24	oe	ccsbBroad304_08898	TRAK2	-			
3709	-29.24	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
3710	-29.24	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
3711	-29.24	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
3712	-29.25	kd	CGS001-7298	TYMS	Methyltransferases			
3713	-29.26	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
3714	-29.3	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
3715	-29.35	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
3716	-29.36	oe	ccsbBroad304_06562	MAT1A	-			
3717	-29.39	oe	ccsbBroad304_02497	YKT6	-			
3718	-29.4	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
3719	-29.46	cc		Tricyclic antidepressant	-			
3720	-29.49	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
3721	-29.5	kd	CGS001-149428	BNIPL	-			
3722	-29.51	oe	ccsbBroad304_00430	GADD45A	-			
3723	-29.51	kd	CGS001-57149	LYRM1	LYR motif containing			
3724	-29.53	oe	ccsbBroad304_09095	PUS7L	-			
3725	-29.54	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
3726	-29.55	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
3727	-29.57	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
3728	-29.6	oe	ccsbBroad304_06565	MB	-			
3729	-29.64	kd	CGS001-54438	GFOD1	-			
3730	-29.66	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
3731	-29.67	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
3732	-29.67	kd	CGS001-5660	PSAP	Endogenous ligands			
3733	-29.69	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
3734	-29.69	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
3735	-29.71	kd	CGS001-9380	GRHPR	-			
3736	-29.72	kd	CGS001-5618	PRLR	Prolactin receptor family			
3737	-29.73	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
3738	-29.73	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
3739	-29.81	kd	CGS001-10250	SRRM1	-			
3740	-29.82	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
3741	-29.85	kd	CGS001-1128	CHRM1	Cholinergic receptors			
3742	-29.87	kd	CGS001-4782	NFIC	-			
3743	-29.88	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
3744	-29.89	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
3745	-29.9	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
3746	-29.91	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
3747	-29.93	kd	CGS001-84365	MKI67IP	-			
3748	-29.94	oe	ccsbBroad304_08137	HOOK2	-			
3749	-29.98	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
3750	-30	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
3751	-30.02	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
3752	-30.02	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
3753	-30.04	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
3754	-30.05	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
3755	-30.1	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
3756	-30.14	kd	CGS001-54205	CYCS	-			
3757	-30.15	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
3758	-30.16	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
3759	-30.18	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
3760	-30.19	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
3761	-30.19	kd	CGS001-23102	TBC1D2B	-			
3762	-30.22	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
3763	-30.26	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
3764	-30.26	kd	CGS001-80212	CCDC92	-			
3765	-30.28	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
3766	-30.32	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
3767	-30.32	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
3768	-30.34	kd	CGS001-10013	HDAC6	Histone deacetylases			
3769	-30.35	cc		HRH1 antagonist	-			
3770	-30.36	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
3771	-30.39	kd	CGS001-3682	ITGAE	Integrins			
3772	-30.41	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
3773	-30.42	oe	ccsbBroad304_07827	STK38L	NDR family			
3774	-30.44	kd	CGS001-56675	NRIP3	-			
3775	-30.45	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
3776	-30.45	kd	CGS001-27244	SESN1	-			
3777	-30.46	kd	CGS001-5170	PDPK1	PDK1 family			
3778	-30.46	kd	CGS001-84669	USP32	EF-hand domain containing			
3779	-30.47	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
3780	-30.48	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
3781	-30.48	kd	CGS001-26993	AKAP8L	-			
3782	-30.53	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
3783	-30.53	kd	CGS001-776	CACNA1D	Calcium channel subunits			
3784	-30.54	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
3785	-30.56	kd	CGS001-10494	STK25	YSK subfamily			
3786	-30.57	kd	CGS001-7105	TSPAN6	Tetraspanins			
3787	-30.57	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
3788	-30.61	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
3789	-30.62	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
3790	-30.62	kd	CGS001-6223	RPS19	S ribosomal proteins			
3791	-30.63	oe	ccsbBroad304_03072	GTPBP8	-			
3792	-30.63	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3793	-30.64	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
3794	-30.65	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
3795	-30.65	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
3796	-30.68	oe	ccsbBroad304_06523	LIG1	-			
3797	-30.7	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
3798	-30.71	kd	CGS001-8681	JMJD7-PLA2G4B	-			
3799	-30.78	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
3800	-30.79	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
3801	-30.84	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
3802	-30.84	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
3803	-30.85	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
3804	-30.88	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
3805	-30.91	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
3806	-30.93	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
3807	-30.97	kd	CGS001-5188	PET112	-			
3808	-30.97	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
3809	-31.01	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
3810	-31.03	oe	ccsbBroad304_00102	RND3	-			
3811	-31.06	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
3812	-31.07	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
3813	-31.08	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
3814	-31.09	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
3815	-31.13	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
3816	-31.13	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
3817	-31.15	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
3818	-31.15	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
3819	-31.18	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
3820	-31.2	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
3821	-31.25	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
3822	-31.25	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
3823	-31.26	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
3824	-31.26	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
3825	-31.27	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
3826	-31.32	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
3827	-31.33	kd	CGS001-2197	FAU	S ribosomal proteins			
3828	-31.35	kd	CGS001-9695	EDEM1	-			
3829	-31.36	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
3830	-31.36	oe	ccsbBroad304_00222	CASP6	Caspases			
3831	-31.39	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
3832	-31.4	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
3833	-31.4	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
3834	-31.4	kd	CGS001-3421	IDH3G	-			
3835	-31.42	cc		Glucocorticoid receptor agonist	-			
3836	-31.49	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
3837	-31.54	kd	CGS001-2852	GPER	-			
3838	-31.56	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
3839	-31.58	kd	CGS001-826	CAPNS1	EF-hand domain containing			
3840	-31.62	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
3841	-31.62	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
3842	-31.63	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
3843	-31.64	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
3844	-31.66	kd	CGS001-53632	PRKAG3	AMPK subfamily			
3845	-31.67	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
3846	-31.68	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
3847	-31.69	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
3848	-31.7	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
3849	-31.74	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
3850	-31.75	kd	CGS001-2288	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
3851	-31.76	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
3852	-31.78	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
3853	-31.79	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3854	-31.8	cc		Aminoacyl tRNA synthetases class II LOF	-			
3855	-31.84	oe	ccsbBroad304_08461	CDCA4	-			
3856	-31.88	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
3857	-31.88	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
3858	-31.88	kd	CGS001-1120	CHKB	-			
3859	-31.9	kd	CGS001-9124	PDLIM1	-			
3860	-31.93	kd	CGS001-11319	ECD	-			
3861	-31.96	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3862	-32.01	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
3863	-32.01	kd	CGS001-3590	IL11RA	IL-6 receptor family			
3864	-32.02	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
3865	-32.04	oe	ccsbBroad304_06711	PFAS	-			
3866	-32.06	kd	CGS001-7165	TPD52L2	-			
3867	-32.09	oe	ccsbBroad304_02109	XPR1	-			
3868	-32.11	kd	CGS001-5427	POLE2	DNA polymerases			
3869	-32.12	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
3870	-32.15	oe	ccsbBroad304_03269	CD320	CD molecules			
3871	-32.21	kd	CGS001-23118	TAB2	-			
3872	-32.23	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
3873	-32.23	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
3874	-32.26	kd	CGS001-2783	GNB2	WD repeat domain containing			
3875	-32.27	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3876	-32.29	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
3877	-32.33	kd	CGS001-11179	ZNF277	-			
3878	-32.34	oe	ccsbBroad304_14011	PAPSS1	-			
3879	-32.36	cc		IL4 Pathway LOF	-			
3880	-32.37	oe	ccsbBroad304_01019	MLH1	-			
3881	-32.37	kd	CGS001-5581	PRKCE	Eta subfamily			
3882	-32.38	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
3883	-32.41	kd	CGS001-10513	APPBP2	-			
3884	-32.43	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
3885	-32.44	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
3886	-32.46	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
3887	-32.5	kd	CGS001-5073	PARN	-			
3888	-32.51	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
3889	-32.55	kd	CGS001-275	AMT	-			
3890	-32.58	kd	CGS001-50846	DHH	-			
3891	-32.59	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3892	-32.59	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
3893	-32.59	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3894	-32.62	kd	CGS001-27125	AFF4	-			
3895	-32.63	cc		GABA receptor antagonist	-			
3896	-32.7	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
3897	-32.73	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
3898	-32.74	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
3899	-32.82	oe	ccsbBroad304_00446	DKC1	-			
3900	-32.85	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
3901	-32.86	kd	CGS001-63892	THADA	-			
3902	-32.86	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
3903	-32.86	kd	CGS001-930	CD19	CD molecules			
3904	-32.87	oe	ccsbBroad304_00552	FEN1	-			
3905	-32.87	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
3906	-32.88	kd	CGS001-57057	TBX20	T-boxes			
3907	-32.92	cc		Cannabinoid receptor agonist	-			
3908	-32.92	kd	CGS001-57721	METTL14	-			
3909	-32.93	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
3910	-32.93	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
3911	-32.94	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
3912	-32.94	kd	CGS001-2664	GDI1	-			
3913	-32.94	kd	CGS001-1962	EHHADH	-			
3914	-32.94	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
3915	-32.94	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
3916	-32.96	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
3917	-32.96	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
3918	-32.99	oe	ccsbBroad304_03591	ETNK1	-			
3919	-33.01	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
3920	-33.02	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
3921	-33.02	oe	ccsbBroad304_09833	SENP5	-			
3922	-33.02	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
3923	-33.02	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
3924	-33.03	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
3925	-33.03	oe	ccsbBroad304_07017	SUOX	-			
3926	-33.06	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
3927	-33.07	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
3928	-33.12	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
3929	-33.17	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
3930	-33.23	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
3931	-33.23	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
3932	-33.24	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
3933	-33.31	cc		G2 M Checkpoint LOF	-			
3934	-33.35	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
3935	-33.36	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
3936	-33.37	kd	CGS001-350	APOH	Apolipoproteins			
3937	-33.39	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
3938	-33.39	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
3939	-33.4	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
3940	-33.42	cc		Calmodulin antagonist	-			
3941	-33.42	kd	CGS001-9218	VAPA	-			
3942	-33.44	kd	CGS001-1131	CHRM3	Cholinergic receptors			
3943	-33.46	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
3944	-33.47	kd	CGS001-5045	FURIN	Subtilisin			
3945	-33.48	oe	ccsbBroad304_02217	FEZ1	-			
3946	-33.5	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
3947	-33.52	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
3948	-33.54	kd	CGS001-8313	AXIN2	-			
3949	-33.57	oe	ccsbBroad304_03310	LCMT1	-			
3950	-33.58	kd	CGS001-9221	NOLC1	-			
3951	-33.61	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
3952	-33.61	kd	CGS001-819	CAMLG	-			
3953	-33.62	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
3954	-33.62	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3955	-33.62	oe	ccsbBroad304_07220	CDC45	-			
3956	-33.65	oe	ccsbBroad304_02367	CALCOCO2	-			
3957	-33.65	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
3958	-33.65	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
3959	-33.68	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
3960	-33.69	oe	ccsbBroad304_02990	LYPD3	-			
3961	-33.7	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
3962	-33.74	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
3963	-33.75	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
3964	-33.77	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
3965	-33.77	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3966	-33.78	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
3967	-33.81	oe	ccsbBroad304_02018	SUCLA2	-			
3968	-33.85	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
3969	-33.85	kd	CGS001-283150	FOXR1	Forkhead boxes			
3970	-33.86	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3971	-33.88	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
3972	-33.93	oe	ccsbBroad304_02092	SYNGR3	-			
3973	-33.94	oe	ccsbBroad304_08452	PIH1D1	-			
3974	-33.94	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
3975	-33.97	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
3976	-33.99	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3977	-33.99	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
3978	-34.03	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
3979	-34.04	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
3980	-34.05	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
3981	-34.05	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
3982	-34.05	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
3983	-34.07	cc		GATA Zinc finger domain containing LOF	-			
3984	-34.07	kd	CGS001-6185	RPN2	-			
3985	-34.08	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
3986	-34.1	kd	CGS001-9871	SEC24D	-			
3987	-34.13	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
3988	-34.14	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
3989	-34.16	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
3990	-34.16	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
3991	-34.16	kd	CGS001-161	AP2A2	-			
3992	-34.18	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
3993	-34.22	oe	ccsbBroad304_06916	SCP2	-			
3994	-34.25	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
3995	-34.26	oe	ccsbBroad304_02708	TRIM32	-			
3996	-34.27	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
3997	-34.28	kd	CGS001-23636	NUP62	-			
3998	-34.29	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
3999	-34.34	oe	ccsbBroad304_03479	YTHDF1	-			
4000	-34.34	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
4001	-34.34	kd	CGS001-1069	CETN2	EF-hand domain containing			
4002	-34.35	oe	ccsbBroad304_00329	CLTA	-			
4003	-34.35	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
4004	-34.36	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
4005	-34.37	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
4006	-34.42	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
4007	-34.43	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
4008	-34.46	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4009	-34.46	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
4010	-34.47	oe	ccsbBroad304_06462	ITGAE	Integrins			
4011	-34.48	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
4012	-34.49	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
4013	-34.52	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
4014	-34.54	kd	CGS001-6778	STAT6	SH2 domain containing			
4015	-34.55	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
4016	-34.57	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
4017	-34.57	kd	CGS001-29911	HOOK2	-			
4018	-34.58	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
4019	-34.59	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
4020	-34.59	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
4021	-34.59	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
4022	-34.59	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
4023	-34.59	oe	ccsbBroad304_00003	ABAT	GABA turnover			
4024	-34.59	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4025	-34.6	oe	ccsbBroad304_01174	PEX13	-			
4026	-34.61	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
4027	-34.63	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
4028	-34.63	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
4029	-34.7	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
4030	-34.7	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
4031	-34.71	kd	CGS001-6477	SIAH1	-			
4032	-34.73	oe	ccsbBroad304_00212	CAMLG	-			
4033	-34.74	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
4034	-34.79	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
4035	-34.8	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
4036	-34.8	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
4037	-34.81	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
4038	-34.81	kd	CGS001-545	ATR	ATR subfamily			
4039	-34.82	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
4040	-34.83	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
4041	-34.84	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
4042	-34.84	kd	CGS001-26227	PHGDH	-			
4043	-34.88	oe	ccsbBroad304_04616	ORMDL3	-			
4044	-34.88	oe	ccsbBroad304_06004	CKB	-			
4045	-34.88	kd	CGS001-25987	TSKU	-			
4046	-34.9	kd	CGS001-55176	SEC61A2	-			
4047	-34.93	kd	CGS001-670	BPHL	-			
4048	-34.94	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
4049	-34.95	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
4050	-34.96	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
4051	-34.97	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
4052	-34.98	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
4053	-34.99	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
4054	-35.01	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
4055	-35.01	kd	CGS001-6599	SMARCC1	-			
4056	-35.02	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
4057	-35.04	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
4058	-35.08	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
4059	-35.1	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
4060	-35.1	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
4061	-35.12	kd	CGS001-9738	CCP110	-			
4062	-35.13	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
4063	-35.14	kd	CGS001-1736	DKC1	-			
4064	-35.15	oe	ccsbBroad304_01832	PAX8	Paired boxes			
4065	-35.16	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
4066	-35.17	oe	ccsbBroad304_05038	HORMAD2	-			
4067	-35.18	kd	CGS001-7486	WRN	-			
4068	-35.18	kd	CGS001-8669	EIF3J	-			
4069	-35.19	kd	CGS001-4175	MCM6	-			
4070	-35.22	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
4071	-35.23	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
4072	-35.24	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
4073	-35.25	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
4074	-35.25	kd	CGS001-22908	SACM1L	-			
4075	-35.26	kd	CGS001-4946	OAZ1	-			
4076	-35.27	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
4077	-35.27	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
4078	-35.33	oe	ccsbBroad304_02686	COPZ1	-			
4079	-35.33	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
4080	-35.34	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
4081	-35.34	kd	CGS001-1604	CD55	CD molecules			
4082	-35.36	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4083	-35.39	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
4084	-35.4	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
4085	-35.42	kd	CGS001-2113	ETS1	ETS Transcription Factors			
4086	-35.43	kd	CGS001-2030	SLC29A1	SLC29 family			
4087	-35.46	kd	CGS001-23658	LSM5	-			
4088	-35.49	oe	ccsbBroad304_00101	RHOC	-			
4089	-35.53	kd	CGS001-4665	NAB2	-			
4090	-35.59	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4091	-35.61	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
4092	-35.61	kd	CGS001-56647	BCCIP	-			
4093	-35.62	kd	CGS001-5230	PGK1	-			
4094	-35.64	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
4095	-35.65	oe	ccsbBroad304_01641	TAF13	-			
4096	-35.66	oe	ccsbBroad304_08217	SCCPDH	-			
4097	-35.68	kd	CGS001-63933	CCDC90A	-			
4098	-35.73	kd	CGS001-708	C1QBP	-			
4099	-35.74	kd	CGS001-9759	HDAC4	Histone deacetylases			
4100	-35.75	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
4101	-35.79	oe	ccsbBroad304_01930	CUL2	-			
4102	-35.81	oe	ccsbBroad304_02458	STK25	YSK subfamily			
4103	-35.81	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
4104	-35.82	oe	ccsbBroad304_02862	CCRN4L	-			
4105	-35.83	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
4106	-35.85	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
4107	-35.87	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
4108	-35.91	kd	CGS001-3827	KNG1	Endogenous ligands			
4109	-35.96	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
4110	-35.97	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
4111	-35.98	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
4112	-35.99	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
4113	-36	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
4114	-36.01	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
4115	-36.01	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
4116	-36.01	kd	CGS001-1196	CLK2	CDC-like kinases			
4117	-36.02	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
4118	-36.06	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
4119	-36.14	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
4120	-36.18	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
4121	-36.18	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
4122	-36.2	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
4123	-36.21	oe	ccsbBroad304_03311	EVL	-			
4124	-36.22	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
4125	-36.22	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
4126	-36.25	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
4127	-36.27	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
4128	-36.31	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
4129	-36.34	kd	CGS001-23210	JMJD6	-			
4130	-36.36	kd	CGS001-51466	EVL	-			
4131	-36.38	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
4132	-36.39	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
4133	-36.4	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
4134	-36.41	oe	ccsbBroad304_09821	TMEM154	-			
4135	-36.41	oe	ccsbBroad304_07889	QPRT	-			
4136	-36.41	oe	ccsbBroad304_03118	NRBP1	NRBP family			
4137	-36.43	kd	CGS001-7013	TERF1	-			
4138	-36.45	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
4139	-36.46	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
4140	-36.47	oe	ccsbBroad304_00009	ACLY	-			
4141	-36.48	oe	ccsbBroad304_02197	VPS26A	-			
4142	-36.5	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
4143	-36.53	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
4144	-36.55	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
4145	-36.59	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
4146	-36.6	kd	CGS001-7270	TTF1	-			
4147	-36.62	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
4148	-36.62	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
4149	-36.7	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
4150	-36.72	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
4151	-36.73	oe	ccsbBroad304_08839	IFIH1	-			
4152	-36.76	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
4153	-36.85	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
4154	-36.85	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
4155	-36.85	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
4156	-36.87	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
4157	-36.87	kd	CGS001-4833	NME4	-			
4158	-36.94	kd	CGS001-79139	DERL1	-			
4159	-36.96	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
4160	-36.98	kd	CGS001-255877	BCL6B	BTB/POZ domain containing			
4161	-37	cc		TGF beta receptor inhibitor	-			
4162	-37.02	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4163	-37.03	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
4164	-37.03	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
4165	-37.07	oe	ccsbBroad304_00392	CTLA4	CD molecules			
4166	-37.08	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
4167	-37.12	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
4168	-37.13	cc		S100 calcium binding proteins LOF	-			
4169	-37.13	oe	ccsbBroad304_03164	MTERFD1	-			
4170	-37.13	kd	CGS001-3131	HLF	-			
4171	-37.15	oe	ccsbBroad304_06569	MCM5	-			
4172	-37.16	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
4173	-37.19	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
4174	-37.19	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
4175	-37.19	kd	CGS001-7913	DEK	-			
4176	-37.21	kd	CGS001-7431	VIM	Intermediate filaments type III			
4177	-37.22	oe	ccsbBroad304_01527	SGK1	SGK family			
4178	-37.23	oe	ccsbBroad304_00931	LCN2	Lipocalins			
4179	-37.25	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
4180	-37.26	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
4181	-37.26	oe	ccsbBroad304_09225	BUD13	-			
4182	-37.27	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
4183	-37.29	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
4184	-37.3	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
4185	-37.31	kd	CGS001-54512	EXOSC4	-			
4186	-37.34	kd	CGS001-890	CCNA2	-			
4187	-37.39	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
4188	-37.4	oe	ccsbBroad304_07598	PEMT	-			
4189	-37.45	oe	ccsbBroad304_07217	AXIN2	-			
4190	-37.46	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
4191	-37.49	kd	CGS001-5019	OXCT1	-			
4192	-37.49	kd	CGS001-2115	ETV1	ETS Transcription Factors			
4193	-37.59	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
4194	-37.6	oe	ccsbBroad304_07923	LSM5	-			
4195	-37.68	oe	ccsbBroad304_00099	ARG2	Arginase			
4196	-37.69	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
4197	-37.7	kd	CGS001-53343	NUDT9	Nudix motif containing			
4198	-37.71	kd	CGS001-4836	NMT1	-			
4199	-37.71	kd	CGS001-3460	IFNGR2	Interferon receptor family			
4200	-37.72	oe	ccsbBroad304_11405	UBE3C	-			
4201	-37.72	oe	ccsbBroad304_03023	CRCP	-			
4202	-37.73	kd	CGS001-4232	MEST	-			
4203	-37.73	kd	CGS001-4176	MCM7	-			
4204	-37.74	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
4205	-37.75	oe	ccsbBroad304_01769	VEGFB	-			
4206	-37.76	oe	ccsbBroad304_02446	TADA3	-			
4207	-37.76	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4208	-37.79	kd	CGS001-1499	CTNNB1	Catenins			
4209	-37.83	kd	CGS001-7276	TTR	-			
4210	-37.89	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
4211	-37.9	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
4212	-37.91	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
4213	-37.92	kd	CGS001-4267	CD99	CD molecules			
4214	-37.95	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
4215	-38	oe	ccsbBroad304_07754	FGFR1OP	-			
4216	-38.01	kd	CGS001-1841	DTYMK	-			
4217	-38.04	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
4218	-38.07	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
4219	-38.1	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
4220	-38.11	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
4221	-38.12	kd	CGS001-8996	NOL3	-			
4222	-38.13	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
4223	-38.16	kd	CGS001-8050	PDHX	-			
4224	-38.18	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
4225	-38.21	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4226	-38.23	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
4227	-38.24	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
4228	-38.25	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
4229	-38.29	kd	CGS001-4170	MCL1	-			
4230	-38.32	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
4231	-38.34	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
4232	-38.35	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
4233	-38.35	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
4234	-38.42	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
4235	-38.43	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
4236	-38.46	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
4237	-38.56	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
4238	-38.59	oe	ccsbBroad304_07814	SACM1L	-			
4239	-38.59	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
4240	-38.64	oe	ccsbBroad304_01624	SUPV3L1	-			
4241	-38.68	kd	CGS001-23386	NUDCD3	-			
4242	-38.7	oe	ccsbBroad304_06159	CTTN	-			
4243	-38.71	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
4244	-38.74	oe	ccsbBroad304_07843	FCHO1	-			
4245	-38.82	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
4246	-38.85	kd	CGS001-1398	CRK	SH2 domain containing			
4247	-38.89	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
4248	-38.9	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
4249	-38.9	kd	CGS001-6857	SYT1	Synaptotagmins			
4250	-38.91	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
4251	-38.93	kd	CGS001-353	APRT	-			
4252	-38.96	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
4253	-39.02	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
4254	-39.06	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4255	-39.06	kd	CGS001-8667	EIF3H	-			
4256	-39.07	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
4257	-39.1	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
4258	-39.1	kd	CGS001-56889	TM9SF3	-			
4259	-39.1	kd	CGS001-4795	NFKBIL1	-			
4260	-39.12	oe	ccsbBroad304_07053	TFPI	-			
4261	-39.13	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
4262	-39.14	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
4263	-39.15	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
4264	-39.2	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
4265	-39.22	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
4266	-39.24	kd	CGS001-3030	HADHA	-			
4267	-39.24	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
4268	-39.25	oe	ccsbBroad304_01061	NAB2	-			
4269	-39.29	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
4270	-39.31	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
4271	-39.35	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
4272	-39.37	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4273	-39.37	kd	CGS001-23139	MAST2	MAST family			
4274	-39.39	oe	ccsbBroad304_06350	HAL	-			
4275	-39.39	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
4276	-39.39	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
4277	-39.4	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
4278	-39.4	oe	ccsbBroad304_07531	TANK	-			
4279	-39.42	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
4280	-39.45	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
4281	-39.51	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
4282	-39.53	kd	CGS001-7077	TIMP2	-			
4283	-39.54	oe	ccsbBroad304_01661	TFCP2	-			
4284	-39.54	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
4285	-39.54	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
4286	-39.56	kd	CGS001-1997	ELF1	ETS Transcription Factors			
4287	-39.56	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
4288	-39.58	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4289	-39.63	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
4290	-39.64	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
4291	-39.65	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
4292	-39.65	kd	CGS001-433	ASGR2	C-type lectin domain containing			
4293	-39.67	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
4294	-39.69	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
4295	-39.72	oe	ccsbBroad304_03089	PACSIN3	-			
4296	-39.76	kd	CGS001-55802	DCP1A	-			
4297	-39.77	kd	CGS001-10298	PAK4	PAKB subfamily			
4298	-39.78	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
4299	-39.81	oe	ccsbBroad304_09281	TPD52L3	-			
4300	-39.82	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
4301	-39.83	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
4302	-39.85	oe	ccsbBroad304_00262	CD59	CD molecules			
4303	-39.86	kd	CGS001-1643	DDB2	WD repeat domain containing			
4304	-39.88	kd	CGS001-2230	FDX1	-			
4305	-39.92	kd	CGS001-10810	WASF3	-			
4306	-39.94	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
4307	-39.99	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
4308	-39.99	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
4309	-40.01	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
4310	-40.02	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
4311	-40.02	kd	CGS001-7982	ST7	-			
4312	-40.03	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
4313	-40.03	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
4314	-40.04	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
4315	-40.05	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
4316	-40.06	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
4317	-40.08	kd	CGS001-55644	OSGEP	-			
4318	-40.09	kd	CGS001-3265	HRAS	RAS subfamily			
4319	-40.11	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
4320	-40.11	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
4321	-40.14	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
4322	-40.14	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
4323	-40.21	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
4324	-40.23	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
4325	-40.27	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
4326	-40.27	kd	CGS001-9467	SH3BP5	-			
4327	-40.29	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
4328	-40.3	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
4329	-40.41	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4330	-40.43	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
4331	-40.45	oe	ccsbBroad304_02218	IKBKE	IKK family			
4332	-40.48	oe	ccsbBroad304_02361	MFSD10	-			
4333	-40.52	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
4334	-40.55	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
4335	-40.55	kd	CGS001-11200	CHEK2	CHK1 subfamily			
4336	-40.62	kd	CGS001-2313	FLI1	ETS Transcription Factors			
4337	-40.63	oe	ccsbBroad304_00161	BID	Endogenous ligands			
4338	-40.63	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
4339	-40.65	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
4340	-40.68	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
4341	-40.73	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
4342	-40.74	oe	ccsbBroad304_07119	UGP2	-			
4343	-40.75	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
4344	-40.77	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
4345	-40.79	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
4346	-40.79	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
4347	-40.8	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
4348	-40.88	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
4349	-40.89	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
4350	-40.92	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
4351	-40.93	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
4352	-40.96	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
4353	-41.06	kd	CGS001-2966	GTF2H2	General transcription factors			
4354	-41.07	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
4355	-41.07	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4356	-41.1	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
4357	-41.1	kd	CGS001-10841	FTCD	-			
4358	-41.13	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
4359	-41.14	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
4360	-41.2	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4361	-41.22	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
4362	-41.24	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
4363	-41.29	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
4364	-41.29	kd	CGS001-59343	SENP2	-			
4365	-41.32	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
4366	-41.35	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
4367	-41.39	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
4368	-41.41	kd	CGS001-65243	ZNF643	-			
4369	-41.43	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
4370	-41.44	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
4371	-41.46	oe	ccsbBroad304_02501	DCTN6	-			
4372	-41.47	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
4373	-41.49	cc		Aurora kinase inhibitor	-			
4374	-41.49	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
4375	-41.49	kd	CGS001-4837	NNMT	-			
4376	-41.55	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
4377	-41.59	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
4378	-41.6	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
4379	-41.64	kd	CGS001-25842	ASF1A	-			
4380	-41.65	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
4381	-41.66	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
4382	-41.67	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
4383	-41.69	kd	CGS001-2100	ESR2	Estrogen receptors			
4384	-41.73	kd	CGS001-1201	CLN3	-			
4385	-41.75	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
4386	-41.76	oe	ccsbBroad304_06639	NFYB	-			
4387	-41.85	oe	ccsbBroad304_00956	LYZ	-			
4388	-41.85	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
4389	-41.86	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
4390	-41.87	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
4391	-41.87	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
4392	-41.92	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
4393	-41.94	kd	CGS001-5479	PPIB	-			
4394	-41.94	oe	ccsbBroad304_06464	ITGB2	Integrins			
4395	-41.99	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
4396	-41.99	kd	CGS001-54884	RETSAT	-			
4397	-42	oe	ccsbBroad304_02017	PEX11A	-			
4398	-42.01	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
4399	-42.03	oe	ccsbBroad304_00239	CCNG1	-			
4400	-42.05	oe	ccsbBroad304_02032	TSC22D1	-			
4401	-42.06	oe	ccsbBroad304_00841	IKBKB	IKK family			
4402	-42.06	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
4403	-42.07	kd	CGS001-2079	ERH	-			
4404	-42.08	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
4405	-42.09	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
4406	-42.1	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4407	-42.1	kd	CGS001-4758	NEU1	-			
4408	-42.1	kd	CGS001-2004	ELK3	ETS Transcription Factors			
4409	-42.13	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
4410	-42.2	oe	ccsbBroad304_01394	RFX4	-			
4411	-42.21	oe	ccsbBroad304_03933	CARD9	-			
4412	-42.23	kd	CGS001-6788	STK3	MST subfamily			
4413	-42.25	kd	CGS001-472	ATM	Other PIKK family kinases			
4414	-42.26	oe	ccsbBroad304_03565	ADI1	-			
4415	-42.27	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
4416	-42.29	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
4417	-42.3	kd	CGS001-50943	FOXP3	Forkhead boxes			
4418	-42.31	kd	CGS001-335	APOA1	Apolipoproteins			
4419	-42.32	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
4420	-42.32	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
4421	-42.37	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
4422	-42.37	kd	CGS001-9140	ATG12	-			
4423	-42.4	oe	ccsbBroad304_02271	LPGAT1	-			
4424	-42.4	kd	CGS001-113451	ADC	-			
4425	-42.41	oe	ccsbBroad304_02425	CDIPT	-			
4426	-42.43	kd	CGS001-10775	POP4	-			
4427	-42.44	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
4428	-42.46	oe	ccsbBroad304_02815	SSBP2	-			
4429	-42.46	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
4430	-42.51	kd	CGS001-6944	VPS72	-			
4431	-42.53	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
4432	-42.59	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
4433	-42.63	oe	ccsbBroad304_00313	TBCB	-			
4434	-42.63	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
4435	-42.66	kd	CGS001-538	ATP7A	ATPases / P-type			
4436	-42.67	oe	ccsbBroad304_01923	UXT	-			
4437	-42.73	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4438	-42.75	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
4439	-42.8	oe	ccsbBroad304_03696	C19ORF10	-			
4440	-42.89	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
4441	-42.9	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
4442	-42.93	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
4443	-42.93	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
4444	-42.98	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
4445	-42.99	oe	ccsbBroad304_13998	PDXK	-			
4446	-43	oe	ccsbBroad304_01674	TIMP4	-			
4447	-43	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
4448	-43.02	oe	ccsbBroad304_02596	KDELR3	-			
4449	-43.02	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4450	-43.03	kd	CGS001-8295	TRRAP	TRRAP subfamily			
4451	-43.05	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
4452	-43.05	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
4453	-43.06	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
4454	-43.09	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
4455	-43.12	kd	CGS001-10247	HRSP12	-			
4456	-43.13	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
4457	-43.13	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4458	-43.14	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
4459	-43.17	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
4460	-43.19	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
4461	-43.21	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
4462	-43.23	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
4463	-43.24	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
4464	-43.27	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4465	-43.29	cc		Toll like receptors LOF	-			
4466	-43.29	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
4467	-43.34	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
4468	-43.36	kd	CGS001-85480	TSLP	-			
4469	-43.39	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
4470	-43.39	oe	ccsbBroad304_00985	MCL1	-			
4471	-43.41	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4472	-43.42	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
4473	-43.47	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
4474	-43.49	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
4475	-43.5	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
4476	-43.54	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
4477	-43.56	oe	ccsbBroad304_13633	PI4KAP2	-			
4478	-43.58	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
4479	-43.6	oe	ccsbBroad304_06134	ECH1	-			
4480	-43.6	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
4481	-43.63	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
4482	-43.64	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
4483	-43.65	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
4484	-43.68	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
4485	-43.7	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
4486	-43.73	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
4487	-43.76	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
4488	-43.79	kd	CGS001-9541	CIR1	-			
4489	-43.81	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
4490	-43.83	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
4491	-43.83	kd	CGS001-11336	EXOC3	-			
4492	-43.87	oe	ccsbBroad304_08596	EAPP	-			
4493	-43.89	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
4494	-43.94	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
4495	-43.96	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
4496	-43.97	kd	CGS001-1028	CDKN1C	-			
4497	-43.99	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
4498	-43.99	kd	CGS001-151126	ZNF385B	-			
4499	-44.02	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4500	-44.03	oe	ccsbBroad304_07401	TXNL1	-			
4501	-44.07	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
4502	-44.11	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
4503	-44.13	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
4504	-44.14	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
4505	-44.18	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
4506	-44.18	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
4507	-44.18	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
4508	-44.21	kd	CGS001-3660	IRF2	-			
4509	-44.22	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
4510	-44.24	kd	CGS001-3566	IL4R	IL-2 receptor family			
4511	-44.26	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
4512	-44.29	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
4513	-44.29	oe	ccsbBroad304_01186	PHB	-			
4514	-44.31	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
4515	-44.32	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
4516	-44.36	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
4517	-44.37	kd	CGS001-2155	F7	Chymotrypsin			
4518	-44.42	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
4519	-44.44	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
4520	-44.46	oe	ccsbBroad304_07605	LYPLA1	-			
4521	-44.47	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
4522	-44.49	kd	CGS001-3725	JUN	basic leucine zipper proteins			
4523	-44.56	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
4524	-44.6	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4525	-44.69	kd	CGS001-8780	RIOK3	RIO3 subfamily			
4526	-44.74	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
4527	-44.75	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
4528	-44.75	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
4529	-44.82	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
4530	-44.85	oe	ccsbBroad304_01658	PRDX2	-			
4531	-44.85	kd	CGS001-10180	RBM6	G patch domain containing			
4532	-44.86	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
4533	-44.87	cc		Protein phosphatase catalytic subunits LOF	-			
4534	-44.88	oe	ccsbBroad304_02822	ARFIP2	-			
4535	-44.9	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
4536	-44.92	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
4537	-44.97	kd	CGS001-58477	SRPRB	-			
4538	-45	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
4539	-45.03	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4540	-45.03	oe	ccsbBroad304_01960	CASK	CASK family			
4541	-45.06	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
4542	-45.07	oe	ccsbBroad304_02592	KIF2C	Kinesins			
4543	-45.07	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
4544	-45.07	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4545	-45.08	kd	CGS001-6118	RPA2	-			
4546	-45.09	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
4547	-45.12	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
4548	-45.12	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
4549	-45.12	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4550	-45.13	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
4551	-45.17	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
4552	-45.18	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
4553	-45.18	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
4554	-45.19	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4555	-45.21	kd	CGS001-6397	SEC14L1	-			
4556	-45.22	oe	ccsbBroad304_06290	GNA15	-			
4557	-45.23	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
4558	-45.24	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
4559	-45.27	kd	CGS001-11168	PSIP1	-			
4560	-45.32	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
4561	-45.34	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
4562	-45.39	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
4563	-45.39	kd	CGS001-23196	FAM120A	-			
4564	-45.42	oe	ccsbBroad304_07820	SNW1	-			
4565	-45.42	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
4566	-45.42	oe	ccsbBroad304_02026	NRP1	CD molecules			
4567	-45.44	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4568	-45.44	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
4569	-45.46	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
4570	-45.47	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
4571	-45.57	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
4572	-45.59	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
4573	-45.71	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
4574	-45.78	kd	CGS001-174	AFP	-			
4575	-45.81	oe	ccsbBroad304_02484	PAICS	-			
4576	-45.81	kd	CGS001-9552	SPAG7	-			
4577	-45.84	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
4578	-45.84	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
4579	-45.85	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
4580	-45.87	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
4581	-45.88	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
4582	-45.9	oe	ccsbBroad304_02229	TRAM2	-			
4583	-45.93	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
4584	-45.95	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
4585	-45.99	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4586	-46	kd	CGS001-6727	SRP14	-			
4587	-46.01	oe	ccsbBroad304_07374	PTPLA	-			
4588	-46.01	kd	CGS001-64786	TBC1D15	-			
4589	-46.02	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
4590	-46.03	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
4591	-46.03	kd	CGS001-7100	TLR5	Toll-like receptor family			
4592	-46.04	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
4593	-46.05	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
4594	-46.06	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
4595	-46.11	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
4596	-46.12	oe	ccsbBroad304_01091	NFIB	-			
4597	-46.12	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4598	-46.12	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
4599	-46.13	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
4600	-46.14	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
4601	-46.17	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
4602	-46.2	oe	ccsbBroad304_03415	GFOD1	-			
4603	-46.21	kd	CGS001-22921	MSRB2	-			
4604	-46.34	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
4605	-46.35	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
4606	-46.37	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
4607	-46.37	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
4608	-46.39	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
4609	-46.42	oe	ccsbBroad304_09503	KLHDC9	-			
4610	-46.42	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
4611	-46.45	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
4612	-46.53	oe	ccsbBroad304_03728	DIABLO	-			
4613	-46.55	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
4614	-46.56	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4615	-46.61	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
4616	-46.63	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
4617	-46.64	oe	ccsbBroad304_06234	G6PC	-			
4618	-46.64	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
4619	-46.64	kd	CGS001-10606	PAICS	-			
4620	-46.65	oe	ccsbBroad304_02534	UTP14A	-			
4621	-46.67	oe	ccsbBroad304_04752	IKBIP	-			
4622	-46.67	oe	ccsbBroad304_10207	ERLIN1	-			
4623	-46.68	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
4624	-46.68	kd	CGS001-4830	NME1	-			
4625	-46.73	kd	CGS001-25797	QPCT	Aminopeptidase Y			
4626	-46.76	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
4627	-46.83	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4628	-46.83	kd	CGS001-10827	FAM114A2	-			
4629	-46.85	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
4630	-46.85	kd	CGS001-6282	S100A11	EF-hand domain containing			
4631	-46.88	oe	ccsbBroad304_06178	ERCC5	-			
4632	-46.89	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
4633	-46.96	oe	ccsbBroad304_02313	ACTR3	-			
4634	-46.99	kd	CGS001-2099	ESR1	Estrogen receptors			
4635	-47.01	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
4636	-47.01	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
4637	-47.07	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
4638	-47.07	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
4639	-47.07	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
4640	-47.11	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
4641	-47.13	kd	CGS001-23378	RRP8	-			
4642	-47.23	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
4643	-47.3	oe	ccsbBroad304_00492	EIF5A	-			
4644	-47.4	cc		Dihydrofolate reductase inhibitor	-			
4645	-47.45	oe	ccsbBroad304_07411	LPXN	-			
4646	-47.45	kd	CGS001-1854	DUT	-			
4647	-47.49	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
4648	-47.56	oe	ccsbBroad304_06574	MDH2	-			
4649	-47.57	oe	ccsbBroad304_03047	BZW2	-			
4650	-47.59	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
4651	-47.61	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
4652	-47.62	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4653	-47.63	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
4654	-47.66	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
4655	-47.66	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
4656	-47.72	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4657	-47.73	kd	CGS001-2747	GLUD2	-			
4658	-47.76	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4659	-47.84	kd	CGS001-637	BID	Endogenous ligands			
4660	-47.89	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
4661	-47.89	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
4662	-47.9	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
4663	-47.92	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
4664	-47.93	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
4665	-47.97	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
4666	-48.04	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
4667	-48.06	kd	CGS001-5110	PCMT1	-			
4668	-48.09	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
4669	-48.09	kd	CGS001-718	C3	Endogenous ligands			
4670	-48.15	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
4671	-48.19	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
4672	-48.21	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
4673	-48.21	kd	CGS001-80274	SCUBE1	-			
4674	-48.24	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
4675	-48.26	oe	ccsbBroad304_01701	TPI1	-			
4676	-48.28	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
4677	-48.29	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
4678	-48.3	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
4679	-48.3	kd	CGS001-1155	TBCB	-			
4680	-48.32	cc		HMGCR inhibitor	-			
4681	-48.33	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
4682	-48.33	kd	CGS001-7086	TKT	-			
4683	-48.36	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
4684	-48.45	oe	ccsbBroad304_02801	CASP14	Caspases			
4685	-48.47	oe	ccsbBroad304_02205	WTAP	-			
4686	-48.48	oe	ccsbBroad304_06136	ECHS1	-			
4687	-48.51	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
4688	-48.52	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
4689	-48.58	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
4690	-48.66	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
4691	-48.7	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4692	-48.72	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
4693	-48.73	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
4694	-48.74	kd	CGS001-4199	ME1	-			
4695	-48.86	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
4696	-48.87	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
4697	-48.9	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
4698	-48.92	oe	ccsbBroad304_01147	PC	Carboxylases			
4699	-48.92	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
4700	-48.96	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
4701	-49	oe	ccsbBroad304_02345	TXNDC9	-			
4702	-49	kd	CGS001-2957	GTF2A1	General transcription factors			
4703	-49.01	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
4704	-49.01	kd	CGS001-2697	GJA1	Ion channels / Gap junction proteins (connexins)			
4705	-49.03	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
4706	-49.08	kd	CGS001-10001	MED6	-			
4707	-49.13	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
4708	-49.14	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4709	-49.17	cc		Imidazoline ligand	-			
4710	-49.22	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
4711	-49.29	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
4712	-49.38	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
4713	-49.42	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
4714	-49.58	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
4715	-49.63	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
4716	-49.64	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
4717	-49.69	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
4718	-49.69	oe	ccsbBroad304_06225	FTH1	-			
4719	-49.69	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
4720	-49.71	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
4721	-49.74	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
4722	-49.75	oe	ccsbBroad304_01754	UCK2	-			
4723	-49.78	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
4724	-49.79	kd	CGS001-158	ADSL	-			
4725	-49.82	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
4726	-49.84	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
4727	-49.85	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
4728	-49.86	oe	ccsbBroad304_03961	SMURF2	-			
4729	-49.87	oe	ccsbBroad304_08645	BCCIP	-			
4730	-49.89	oe	ccsbBroad304_10230	STK19	G11 family			
4731	-49.89	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
4732	-49.9	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
4733	-49.94	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
4734	-49.98	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
4735	-50.04	kd	CGS001-2000	ELF4	ETS Transcription Factors			
4736	-50.05	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
4737	-50.12	kd	CGS001-7018	TF	-			
4738	-50.13	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
4739	-50.19	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
4740	-50.2	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
4741	-50.21	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
4742	-50.22	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
4743	-50.25	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
4744	-50.25	kd	CGS001-23581	CASP14	Caspases			
4745	-50.31	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
4746	-50.31	kd	CGS001-4931	NVL	ATPases / AAA-type			
4747	-50.4	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
4748	-50.42	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
4749	-50.42	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
4750	-50.44	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
4751	-50.45	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
4752	-50.45	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
4753	-50.5	kd	CGS001-6119	RPA3	-			
4754	-50.52	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4755	-50.57	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
4756	-50.59	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
4757	-50.65	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
4758	-50.67	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
4759	-50.69	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
4760	-50.77	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
4761	-50.78	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
4762	-50.82	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
4763	-50.83	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
4764	-50.84	cc		PRD class homeoboxes and psudogenes LOF	-			
4765	-50.84	oe	ccsbBroad304_05439	O3FAR1	-			
4766	-50.85	oe	ccsbBroad304_07632	PROCR	CD molecules			
4767	-50.87	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
4768	-50.87	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
4769	-50.87	kd	CGS001-10174	SORBS3	-			
4770	-50.88	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
4771	-50.89	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
4772	-50.89	oe	ccsbBroad304_00491	EIF4EBP2	-			
4773	-50.89	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
4774	-50.9	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
4775	-50.91	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
4776	-50.93	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
4777	-50.98	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4778	-51.01	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
4779	-51.03	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
4780	-51.03	oe	ccsbBroad304_02589	COPS5	-			
4781	-51.04	oe	ccsbBroad304_00394	CTSD	Cathepsins			
4782	-51.05	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4783	-51.1	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
4784	-51.16	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
4785	-51.16	kd	CGS001-5824	PEX19	-			
4786	-51.17	kd	CGS001-6443	SGCB	-			
4787	-51.18	oe	ccsbBroad304_00960	SMAD1	SMADs			
4788	-51.25	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
4789	-51.27	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
4790	-51.28	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
4791	-51.29	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
4792	-51.33	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
4793	-51.35	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
4794	-51.37	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
4795	-51.41	kd	CGS001-47	ACLY	-			
4796	-51.43	oe	ccsbBroad304_02163	MED7	-			
4797	-51.43	kd	CGS001-10645	CAMKK2	Meta subfamily			
4798	-51.45	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
4799	-51.45	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
4800	-51.46	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
4801	-51.55	oe	ccsbBroad304_00817	IDH2	-			
4802	-51.63	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
4803	-51.63	kd	CGS001-23076	RRP1B	-			
4804	-51.64	kd	CGS001-5338	PLD2	Hydrolases			
4805	-51.66	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
4806	-51.67	oe	ccsbBroad304_01672	TIMP2	-			
4807	-51.7	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
4808	-51.78	oe	ccsbBroad304_04292	INHBE	-			
4809	-51.78	kd	CGS001-10904	BLCAP	-			
4810	-51.81	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4811	-51.97	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
4812	-52	oe	ccsbBroad304_00162	BIK	-			
4813	-52.02	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
4814	-52.03	oe	ccsbBroad304_00854	IL8	-			
4815	-52.04	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
4816	-52.05	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
4817	-52.17	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
4818	-52.22	kd	CGS001-439	ASNA1	-			
4819	-52.28	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4820	-52.28	kd	CGS001-23192	ATG4B	Aut2 peptidase			
4821	-52.3	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
4822	-52.31	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
4823	-52.32	oe	ccsbBroad304_08802	ELAC2	-			
4824	-52.33	cc		Bacterial 30S ribosomal subunit inhibitor	-			
4825	-52.37	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
4826	-52.4	kd	CGS001-79073	TMEM109	-			
4827	-52.46	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
4828	-52.49	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
4829	-52.49	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
4830	-52.5	kd	CGS001-5361	PLXNA1	Plexins			
4831	-52.51	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
4832	-52.51	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
4833	-52.55	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
4834	-52.58	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
4835	-52.59	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
4836	-52.59	kd	CGS001-4893	NRAS	RAS subfamily			
4837	-52.61	oe	ccsbBroad304_00447	DLD	-			
4838	-52.61	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
4839	-52.63	kd	CGS001-5245	PHB	-			
4840	-52.69	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
4841	-52.7	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
4842	-52.71	kd	CGS001-6622	SNCA	Parkinson disease			
4843	-52.73	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
4844	-52.74	kd	CGS001-79902	NUP85	-			
4845	-52.75	kd	CGS001-1514	CTSL1	-			
4846	-52.78	kd	CGS001-10482	NXF1	-			
4847	-52.85	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
4848	-52.86	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
4849	-52.86	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
4850	-52.87	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
4851	-52.87	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
4852	-52.88	kd	CGS001-162699	TCEB3C	-			
4853	-52.89	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
4854	-52.91	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
4855	-52.93	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
4856	-53.01	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
4857	-53.02	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
4858	-53.03	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
4859	-53.04	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
4860	-53.05	kd	CGS001-6210	RPS15A	S ribosomal proteins			
4861	-53.07	kd	CGS001-375133	PI4KAP2	-			
4862	-53.08	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
4863	-53.09	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
4864	-53.1	oe	ccsbBroad304_14143	NUSAP1	-			
4865	-53.12	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
4866	-53.13	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
4867	-53.15	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
4868	-53.21	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
4869	-53.28	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
4870	-53.31	oe	ccsbBroad304_08426	TEX10	-			
4871	-53.32	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
4872	-53.35	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
4873	-53.37	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
4874	-53.39	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
4875	-53.41	oe	ccsbBroad304_00550	FDXR	-			
4876	-53.41	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
4877	-53.43	oe	ccsbBroad304_03554	NAT10	-			
4878	-53.45	kd	CGS001-23075	SWAP70	EF-hand domain containing			
4879	-53.46	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
4880	-53.5	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4881	-53.51	kd	CGS001-117154	DACH2	-			
4882	-53.52	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
4883	-53.53	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
4884	-53.54	kd	CGS001-64223	MLST8	WD repeat domain containing			
4885	-53.63	kd	CGS001-10755	GIPC1	-			
4886	-53.67	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
4887	-53.69	cc		FOS transcription factor family GOF	-			
4888	-53.76	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
4889	-53.76	oe	ccsbBroad304_03950	ATG3	-			
4890	-53.77	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
4891	-53.78	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
4892	-53.79	kd	CGS001-2932	GSK3B	GSK subfamily			
4893	-53.79	kd	CGS001-2057	EPOR	Prolactin receptor family			
4894	-53.86	kd	CGS001-8914	TIMELESS	-			
4895	-53.9	kd	CGS001-8569	MKNK1	MKN subfamily			
4896	-53.92	kd	CGS001-10607	TBL3	WD repeat domain containing			
4897	-53.95	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
4898	-53.96	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
4899	-54.03	kd	CGS001-10252	SPRY1	-			
4900	-54.12	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
4901	-54.13	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
4902	-54.16	kd	CGS001-388	RHOB	-			
4903	-54.17	kd	CGS001-80314	EPC1	-			
4904	-54.18	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
4905	-54.2	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
4906	-54.21	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
4907	-54.27	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
4908	-54.31	oe	ccsbBroad304_01560	SNAPC1	-			
4909	-54.32	kd	CGS001-54681	P4HTM	-			
4910	-54.34	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
4911	-54.35	oe	ccsbBroad304_05823	ANXA2	Annexins			
4912	-54.37	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
4913	-54.39	oe	ccsbBroad304_02738	RRS1	-			
4914	-54.4	cc		Estrogen receptor antagonist	-			
4915	-54.42	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
4916	-54.43	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
4917	-54.45	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
4918	-54.47	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
4919	-54.54	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4920	-54.56	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
4921	-54.63	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
4922	-54.67	oe	ccsbBroad304_02373	SPRY2	-			
4923	-54.68	kd	CGS001-3575	IL7R	IL-2 receptor family			
4924	-54.7	kd	CGS001-1738	DLD	-			
4925	-54.75	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
4926	-54.76	kd	CGS001-7158	TP53BP1	-			
4927	-54.8	kd	CGS001-9180	OSMR	IL-6 receptor family			
4928	-54.82	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
4929	-54.83	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4930	-54.87	oe	ccsbBroad304_07875	SPECC1L	-			
4931	-54.93	oe	ccsbBroad304_06852	RBP4	Lipocalins			
4932	-54.95	cc		DNA Replication LOF	-			
4933	-54.99	oe	ccsbBroad304_05931	CAPG	-			
4934	-55	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
4935	-55.01	kd	CGS001-5686	PSMA5	Proteasome subunits			
4936	-55.04	kd	CGS001-51593	SRRT	-			
4937	-55.05	oe	ccsbBroad304_01654	TCTA	-			
4938	-55.05	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4939	-55.05	kd	CGS001-81533	ITFG1	-			
4940	-55.06	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
4941	-55.08	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
4942	-55.12	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
4943	-55.16	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4944	-55.17	kd	CGS001-5108	PCM1	-			
4945	-55.36	oe	ccsbBroad304_09035	COASY	-			
4946	-55.37	kd	CGS001-375	ARF1	ADP-ribosylation factors			
4947	-55.44	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
4948	-55.49	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
4949	-55.51	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
4950	-55.53	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
4951	-55.54	oe	ccsbBroad304_03191	NOSIP	-			
4952	-55.6	kd	CGS001-3998	LMAN1	-			
4953	-55.62	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4954	-55.67	oe	ccsbBroad304_00106	ARRB1	-			
4955	-55.71	kd	CGS001-55662	HIF1AN	-			
4956	-55.72	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
4957	-55.72	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
4958	-55.76	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
4959	-55.77	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
4960	-55.8	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
4961	-55.84	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
4962	-55.95	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
4963	-55.96	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
4964	-55.97	kd	CGS001-4074	M6PR	-			
4965	-56.08	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
4966	-56.15	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
4967	-56.16	oe	ccsbBroad304_06535	LPL	-			
4968	-56.16	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
4969	-56.2	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
4970	-56.23	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
4971	-56.32	kd	CGS001-3672	ITGA1	Integrins			
4972	-56.33	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
4973	-56.36	kd	CGS001-222546	RFX6	-			
4974	-56.37	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
4975	-56.4	kd	CGS001-2767	GNA11	-			
4976	-56.43	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
4977	-56.47	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
4978	-56.53	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4979	-56.54	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
4980	-56.61	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
4981	-56.63	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
4982	-56.66	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
4983	-56.67	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
4984	-56.73	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
4985	-56.75	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
4986	-56.76	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
4987	-56.82	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
4988	-56.82	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
4989	-56.9	kd	CGS001-5933	RBL1	-			
4990	-56.92	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
4991	-56.99	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
4992	-57.04	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
4993	-57.04	kd	CGS001-1105	CHD1	-			
4994	-57.05	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
4995	-57.06	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
4996	-57.06	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
4997	-57.14	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
4998	-57.17	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
4999	-57.18	oe	ccsbBroad304_06952	SKP1	-			
5000	-57.28	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
5001	-57.28	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
5002	-57.34	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
5003	-57.37	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
5004	-57.37	kd	CGS001-5411	PNN	-			
5005	-57.41	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
5006	-57.43	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
5007	-57.48	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
5008	-57.49	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
5009	-57.51	oe	ccsbBroad304_10758	CTBP2	-			
5010	-57.52	oe	ccsbBroad304_00250	CD19	CD molecules			
5011	-57.54	oe	ccsbBroad304_07561	YAF2	-			
5012	-57.54	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5013	-57.55	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
5014	-57.58	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
5015	-57.66	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
5016	-57.67	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
5017	-57.69	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
5018	-57.69	kd	CGS001-642	BLMH	-			
5019	-57.7	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
5020	-57.72	oe	ccsbBroad304_13891	LCK	Src family			
5021	-57.73	kd	CGS001-1493	CTLA4	CD molecules			
5022	-57.78	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
5023	-57.79	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
5024	-57.8	oe	ccsbBroad304_02243	DLGAP5	-			
5025	-57.82	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
5026	-57.9	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
5027	-57.92	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
5028	-57.97	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
5029	-57.97	kd	CGS001-403	ARL3	ADP-ribosylation factors			
5030	-58.02	kd	CGS001-6016	RIT1	-			
5031	-58.02	kd	CGS001-2879	GPX4	-			
5032	-58.03	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
5033	-58.04	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
5034	-58.07	oe	ccsbBroad304_00657	GNG4	-			
5035	-58.12	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
5036	-58.13	oe	ccsbBroad304_04294	ATG10	-			
5037	-58.13	kd	CGS001-1062	CENPE	Kinesins			
5038	-58.14	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
5039	-58.16	kd	CGS001-2534	FYN	Src family			
5040	-58.2	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
5041	-58.21	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
5042	-58.27	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
5043	-58.29	kd	CGS001-11116	FGFR1OP	-			
5044	-58.32	kd	CGS001-51172	NAGPA	-			
5045	-58.33	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
5046	-58.36	kd	CGS001-10641	NPRL2	-			
5047	-58.46	kd	CGS001-9183	ZW10	-			
5048	-58.48	cc		FGFR inhibitor	-			
5049	-58.5	kd	CGS001-8870	IER3	-			
5050	-58.52	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
5051	-58.57	kd	CGS001-9805	SCRN1	-			
5052	-58.59	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
5053	-58.61	oe	ccsbBroad304_01577	SOD1	-			
5054	-58.65	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
5055	-58.72	kd	CGS001-4200	ME2	-			
5056	-58.74	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
5057	-58.74	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5058	-58.75	kd	CGS001-8826	IQGAP1	-			
5059	-58.76	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
5060	-58.78	oe	ccsbBroad304_01183	PGD	-			
5061	-58.81	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
5062	-58.83	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
5063	-58.85	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
5064	-58.86	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
5065	-58.88	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
5066	-58.91	kd	CGS001-11284	PNKP	-			
5067	-58.93	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
5068	-58.93	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
5069	-59.03	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
5070	-59.1	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
5071	-59.15	oe	ccsbBroad304_00054	ALDOC	-			
5072	-59.17	cc		Nucleoporin LOF	-			
5073	-59.24	kd	CGS001-55793	FAM63A	-			
5074	-59.25	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
5075	-59.25	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
5076	-59.25	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
5077	-59.3	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
5078	-59.31	oe	ccsbBroad304_01102	NMT1	-			
5079	-59.37	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
5080	-59.43	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
5081	-59.46	kd	CGS001-2961	GTF2E2	General transcription factors			
5082	-59.55	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
5083	-59.56	kd	CGS001-11315	PARK7	Parkinson disease			
5084	-59.59	oe	ccsbBroad304_03179	BOLA1	-			
5085	-59.62	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
5086	-59.62	kd	CGS001-144811	LACC1	-			
5087	-59.64	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
5088	-59.65	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5089	-59.67	oe	ccsbBroad304_03625	HIF1AN	-			
5090	-59.68	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
5091	-59.68	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
5092	-59.82	kd	CGS001-89766	UMODL1	-			
5093	-59.86	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
5094	-59.89	oe	ccsbBroad304_07884	RYBP	-			
5095	-59.92	kd	CGS001-23492	CBX7	-			
5096	-59.94	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
5097	-59.98	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
5098	-60	cc		Non Homologous End Joining LOF	-			
5099	-60.02	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
5100	-60.07	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
5101	-60.07	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
5102	-60.15	kd	CGS001-7099	TLR4	Toll-like receptor family			
5103	-60.15	kd	CGS001-55620	STAP2	-			
5104	-60.18	kd	CGS001-8508	NIPSNAP1	-			
5105	-60.26	kd	CGS001-840	CASP7	Caspases			
5106	-60.28	kd	CGS001-836	CASP3	Caspases			
5107	-60.32	kd	CGS001-54499	TMCO1	-			
5108	-60.35	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
5109	-60.37	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
5110	-60.39	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
5111	-60.45	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
5112	-60.46	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5113	-60.5	oe	ccsbBroad304_00509	EPHX1	-			
5114	-60.52	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5115	-60.53	kd	CGS001-4616	GADD45B	-			
5116	-60.54	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
5117	-60.59	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
5118	-60.62	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
5119	-60.66	oe	ccsbBroad304_03544	FAIM	-			
5120	-60.68	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
5121	-60.79	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
5122	-60.83	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
5123	-60.94	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5124	-60.97	kd	CGS001-527	ATP6V0C	ATPases / V-type			
5125	-60.98	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
5126	-61.01	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
5127	-61.08	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
5128	-61.08	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
5129	-61.1	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
5130	-61.13	oe	ccsbBroad304_02626	PKIG	-			
5131	-61.21	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
5132	-61.21	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
5133	-61.22	kd	CGS001-4683	NBN	-			
5134	-61.22	kd	CGS001-6500	SKP1	-			
5135	-61.23	kd	CGS001-54541	DDIT4	-			
5136	-61.25	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
5137	-61.27	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
5138	-61.28	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
5139	-61.32	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
5140	-61.34	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
5141	-61.35	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
5142	-61.37	oe	ccsbBroad304_00600	FYN	Src family			
5143	-61.41	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5144	-61.44	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
5145	-61.51	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
5146	-61.53	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
5147	-61.55	kd	CGS001-9159	PCSK7	Subtilisin			
5148	-61.83	oe	ccsbBroad304_05936	CASP2	Caspases			
5149	-61.85	kd	CGS001-9322	TRIP10	-			
5150	-61.91	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
5151	-61.93	kd	CGS001-54899	PXK	Slob family			
5152	-61.95	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
5153	-61.96	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
5154	-61.96	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
5155	-62	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
5156	-62.03	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
5157	-62.06	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
5158	-62.08	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
5159	-62.11	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
5160	-62.18	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
5161	-62.19	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
5162	-62.23	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
5163	-62.23	kd	CGS001-5480	PPIC	-			
5164	-62.25	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
5165	-62.28	kd	CGS001-2673	GFPT1	-			
5166	-62.29	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
5167	-62.32	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
5168	-62.33	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
5169	-62.47	oe	ccsbBroad304_02964	TIMM9	-			
5170	-62.48	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
5171	-62.7	oe	ccsbBroad304_01184	PGK1	-			
5172	-62.77	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
5173	-62.77	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
5174	-62.78	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
5175	-62.8	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
5176	-62.8	kd	CGS001-5997	RGS2	Endogenous ligands			
5177	-62.83	kd	CGS001-3845	KRAS	RAS subfamily			
5178	-62.88	oe	ccsbBroad304_06845	RARRES3	-			
5179	-62.94	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
5180	-62.97	oe	ccsbBroad304_06889	RPN2	-			
5181	-62.97	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
5182	-63.02	cc		Structural maintenance of chromosomes proteins LOF	-			
5183	-63.09	kd	CGS001-22889	KIAA0907	-			
5184	-63.1	kd	CGS001-55191	NADSYN1	-			
5185	-63.21	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
5186	-63.26	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5187	-63.29	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
5188	-63.35	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
5189	-63.35	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
5190	-63.37	oe	ccsbBroad304_01379	RBBP6	-			
5191	-63.39	oe	ccsbBroad304_00624	GCK	Hexokinases			
5192	-63.42	kd	CGS001-6233	RPS27A	S ribosomal proteins			
5193	-63.43	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
5194	-63.47	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
5195	-63.5	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
5196	-63.5	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
5197	-63.55	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
5198	-63.59	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5199	-63.62	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
5200	-63.63	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
5201	-63.63	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
5202	-63.67	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
5203	-63.68	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
5204	-63.71	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
5205	-63.75	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
5206	-63.76	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
5207	-63.82	oe	ccsbBroad304_06975	SMARCC2	-			
5208	-63.83	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
5209	-63.83	kd	CGS001-302	ANXA2	Annexins			
5210	-63.84	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
5211	-63.85	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
5212	-63.87	kd	CGS001-6611	SMS	-			
5213	-63.88	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
5214	-63.89	kd	CGS001-7185	TRAF1	-			
5215	-63.99	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
5216	-64	oe	ccsbBroad304_03433	DDIT4	-			
5217	-64.05	oe	ccsbBroad304_01114	NUP88	-			
5218	-64.12	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
5219	-64.15	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5220	-64.19	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
5221	-64.22	oe	ccsbBroad304_02415	TUBB3	Tubulins			
5222	-64.24	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
5223	-64.25	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
5224	-64.31	oe	ccsbBroad304_06301	GOT2	-			
5225	-64.33	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
5226	-64.35	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
5227	-64.38	kd	CGS001-7485	WRB	-			
5228	-64.41	kd	CGS001-11136	SLC7A9	SLC7 family			
5229	-64.48	cc		Serotonin receptor agonist	-			
5230	-64.57	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
5231	-64.58	kd	CGS001-5359	PLSCR1	-			
5232	-64.6	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
5233	-64.65	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
5234	-64.69	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
5235	-64.76	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
5236	-64.76	kd	CGS001-2232	FDXR	-			
5237	-64.82	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
5238	-64.86	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
5239	-64.96	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
5240	-64.97	oe	ccsbBroad304_00112	ASNA1	-			
5241	-64.98	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
5242	-65	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
5243	-65.05	cc		Leucine rich repeat kinase inhibitor	-			
5244	-65.21	oe	ccsbBroad304_01327	PSPH	-			
5245	-65.22	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
5246	-65.22	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
5247	-65.29	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
5248	-65.31	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
5249	-65.33	kd	CGS001-2781	GNAZ	-			
5250	-65.39	oe	ccsbBroad304_06324	GPX7	-			
5251	-65.39	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
5252	-65.41	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
5253	-65.43	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
5254	-65.45	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
5255	-65.51	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
5256	-65.55	oe	ccsbBroad304_01398	RHEB	-			
5257	-65.56	kd	CGS001-7389	UROD	-			
5258	-65.62	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
5259	-65.68	oe	ccsbBroad304_02340	SORBS3	-			
5260	-65.69	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
5261	-65.71	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
5262	-65.73	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
5263	-65.73	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
5264	-65.74	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
5265	-65.75	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
5266	-65.78	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
5267	-65.78	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
5268	-65.88	kd	CGS001-8226	HDHD1	-			
5269	-66.01	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
5270	-66.04	kd	CGS001-2885	GRB2	SH2 domain containing			
5271	-66.14	oe	ccsbBroad304_05757	ACADS	-			
5272	-66.14	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
5273	-66.17	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
5274	-66.2	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
5275	-66.2	kd	CGS001-5167	ENPP1	-			
5276	-66.29	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
5277	-66.32	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
5278	-66.35	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
5279	-66.36	kd	CGS001-56005	C19ORF10	-			
5280	-66.38	kd	CGS001-5162	PDHB	-			
5281	-66.38	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
5282	-66.42	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
5283	-66.45	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
5284	-66.55	oe	ccsbBroad304_03122	RHOD	-			
5285	-66.56	oe	ccsbBroad304_02175	MAGED1	-			
5286	-66.56	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
5287	-66.57	kd	CGS001-5050	PAFAH1B3	-			
5288	-66.65	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
5289	-66.65	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
5290	-66.7	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
5291	-66.72	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
5292	-66.78	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
5293	-66.79	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
5294	-66.86	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
5295	-66.87	kd	CGS001-125965	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
5296	-66.96	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5297	-67.02	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
5298	-67.08	kd	CGS001-7035	TFPI	-			
5299	-67.09	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
5300	-67.09	oe	ccsbBroad304_04190	CCDC92	-			
5301	-67.11	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
5302	-67.11	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
5303	-67.12	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
5304	-67.26	cc		SRC inhibitor	-			
5305	-67.39	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
5306	-67.39	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
5307	-67.44	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
5308	-67.44	kd	CGS001-2309	FOXO3	Forkhead boxes			
5309	-67.45	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5310	-67.49	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
5311	-67.5	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
5312	-67.54	oe	ccsbBroad304_09284	UBE3B	-			
5313	-67.55	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
5314	-67.58	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
5315	-67.61	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
5316	-67.62	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
5317	-67.66	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
5318	-67.68	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
5319	-67.73	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
5320	-67.75	kd	CGS001-7056	THBD	CD molecules			
5321	-67.8	oe	ccsbBroad304_04406	PLA2G12B	-			
5322	-67.8	kd	CGS001-25824	PRDX5	-			
5323	-67.81	oe	ccsbBroad304_00880	IRF2	-			
5324	-67.82	kd	CGS001-2053	EPHX2	-			
5325	-67.84	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
5326	-67.84	kd	CGS001-2729	GCLC	-			
5327	-67.85	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
5328	-67.87	kd	CGS001-399694	SHC4	SH2 domain containing			
5329	-67.9	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
5330	-67.91	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
5331	-67.94	kd	CGS001-533	ATP6V0B	ATPases / V-type			
5332	-68	oe	ccsbBroad304_09254	PAQR8	-			
5333	-68.12	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
5334	-68.15	oe	ccsbBroad304_02864	PRDX5	-			
5335	-68.16	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
5336	-68.17	oe	ccsbBroad304_07491	IP6K1	-			
5337	-68.24	kd	CGS001-3420	IDH3B	-			
5338	-68.3	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
5339	-68.32	kd	CGS001-23244	PDS5A	-			
5340	-68.35	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
5341	-68.36	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
5342	-68.36	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
5343	-68.4	oe	ccsbBroad304_07651	HEXIM1	-			
5344	-68.46	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
5345	-68.47	kd	CGS001-3685	ITGAV	Integrins			
5346	-68.52	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
5347	-68.54	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
5348	-68.54	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
5349	-68.6	kd	CGS001-388650	FAM69A	-			
5350	-68.62	kd	CGS001-7016	TESK1	TESK subfamily			
5351	-68.67	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
5352	-68.67	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
5353	-68.68	kd	CGS001-1312	COMT	Catecholamine turnover			
5354	-68.71	kd	CGS001-6696	SPP1	Endogenous ligands			
5355	-68.71	kd	CGS001-3992	FADS1	Fatty acid desaturases			
5356	-68.77	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
5357	-68.79	cc		Proteasome Pathway LOF	-			
5358	-68.81	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
5359	-68.82	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
5360	-68.82	kd	CGS001-5362	PLXNA2	Plexins			
5361	-68.84	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
5362	-68.85	oe	ccsbBroad304_13952	SHMT2	-			
5363	-68.86	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
5364	-68.9	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
5365	-68.91	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
5366	-68.94	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
5367	-68.94	kd	CGS001-3560	IL2RB	IL-2 receptor family			
5368	-68.98	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
5369	-68.99	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
5370	-69.03	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
5371	-69.05	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
5372	-69.08	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
5373	-69.2	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
5374	-69.2	kd	CGS001-5743	PTGS2	Cyclooxygenase			
5375	-69.21	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
5376	-69.22	kd	CGS001-83999	KREMEN1	-			
5377	-69.23	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
5378	-69.23	kd	CGS001-5914	RARA	Retinoic acid receptors			
5379	-69.24	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
5380	-69.32	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
5381	-69.34	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
5382	-69.37	kd	CGS001-9451	EIF2AK3	PEK subfamily			
5383	-69.39	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
5384	-69.39	kd	CGS001-7003	TEAD1	-			
5385	-69.4	cc		V type ATPases LOF	-			
5386	-69.42	kd	CGS001-51022	GLRX2	-			
5387	-69.5	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
5388	-69.55	oe	ccsbBroad304_01632	SYPL1	-			
5389	-69.59	kd	CGS001-9612	NCOR2	-			
5390	-69.62	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
5391	-69.65	kd	CGS001-8535	CBX4	-			
5392	-69.67	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
5393	-69.69	oe	ccsbBroad304_00789	HSBP1	-			
5394	-69.71	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
5395	-69.73	kd	CGS001-27035	NOX1	-			
5396	-69.75	kd	CGS001-1611	DAP	-			
5397	-69.79	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
5398	-69.79	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
5399	-69.8	kd	CGS001-9788	MTSS1	-			
5400	-69.8	kd	CGS001-6364	CCL20	Chemokine ligands			
5401	-69.82	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
5402	-69.85	oe	ccsbBroad304_02292	BCL2L11	-			
5403	-69.85	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
5404	-69.86	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
5405	-69.89	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5406	-69.91	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
5407	-69.92	oe	ccsbBroad304_07832	XPO7	Exportins			
5408	-69.93	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
5409	-69.94	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
5410	-69.99	kd	CGS001-3608	ILF2	-			
5411	-70.05	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5412	-70.05	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
5413	-70.08	kd	CGS001-22794	CASC3	-			
5414	-70.11	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
5415	-70.16	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
5416	-70.19	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
5417	-70.2	kd	CGS001-11124	FAF1	UBX domain containing			
5418	-70.43	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
5419	-70.44	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
5420	-70.44	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
5421	-70.54	oe	ccsbBroad304_02349	MPHOSPH9	-			
5422	-70.59	oe	ccsbBroad304_03056	MCTS1	-			
5423	-70.59	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
5424	-70.61	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
5425	-70.61	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
5426	-70.65	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
5427	-70.65	kd	CGS001-6519	SLC3A1	SLC3 family			
5428	-70.66	kd	CGS001-10681	GNB5	WD repeat domain containing			
5429	-70.7	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
5430	-70.72	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
5431	-70.72	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
5432	-70.73	oe	ccsbBroad304_06278	GK	Glycerol kinases			
5433	-70.73	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
5434	-70.76	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
5435	-70.78	oe	ccsbBroad304_00038	AGL	-			
5436	-70.81	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
5437	-70.84	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
5438	-70.88	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
5439	-70.9	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
5440	-70.94	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
5441	-70.94	kd	CGS001-2274	FHL2	-			
5442	-71	oe	ccsbBroad304_06008	AP2M1	-			
5443	-71.02	oe	ccsbBroad304_03618	OSGEP	-			
5444	-71.04	kd	CGS001-11014	KDELR2	-			
5445	-71.16	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
5446	-71.2	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
5447	-71.22	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
5448	-71.28	kd	CGS001-23149	FCHO1	-			
5449	-71.29	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
5450	-71.32	oe	ccsbBroad304_07600	NSA2	-			
5451	-71.33	kd	CGS001-6277	S100A6	EF-hand domain containing			
5452	-71.34	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
5453	-71.4	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
5454	-71.41	kd	CGS001-2548	GAA	Glycosidases			
5455	-71.46	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
5456	-71.47	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
5457	-71.51	oe	ccsbBroad304_05947	CCNC	-			
5458	-71.52	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
5459	-71.53	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
5460	-71.61	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
5461	-71.62	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
5462	-71.7	oe	ccsbBroad304_01084	NEU1	-			
5463	-71.73	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
5464	-71.73	kd	CGS001-5357	PLS1	EF-hand domain containing			
5465	-71.75	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
5466	-71.82	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
5467	-71.88	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
5468	-71.96	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
5469	-72.02	oe	ccsbBroad304_03746	CDC42SE1	-			
5470	-72.02	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5471	-72.02	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
5472	-72.03	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
5473	-72.05	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
5474	-72.06	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5475	-72.1	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
5476	-72.11	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
5477	-72.14	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
5478	-72.14	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5479	-72.21	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
5480	-72.24	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
5481	-72.25	kd	CGS001-727	C5	Endogenous ligands			
5482	-72.26	oe	ccsbBroad304_05590	NOTCH2NL	-			
5483	-72.31	kd	CGS001-85442	KNDC1	-			
5484	-72.32	oe	ccsbBroad304_09756	PAQR7	-			
5485	-72.33	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
5486	-72.33	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
5487	-72.37	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
5488	-72.37	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
5489	-72.4	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
5490	-72.41	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5491	-72.41	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
5492	-72.42	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
5493	-72.43	kd	CGS001-1287	COL4A5	Collagens			
5494	-72.47	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
5495	-72.5	oe	ccsbBroad304_02094	FIBP	-			
5496	-72.55	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
5497	-72.58	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
5498	-72.58	oe	ccsbBroad304_03812	PBXIP1	-			
5499	-72.6	kd	CGS001-9441	MED26	-			
5500	-72.61	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
5501	-72.64	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
5502	-72.66	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
5503	-72.76	oe	ccsbBroad304_03658	DCP1A	-			
5504	-72.79	oe	ccsbBroad304_01001	MEST	-			
5505	-72.8	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
5506	-72.82	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
5507	-72.9	cc		ATPase inhibitor	-			
5508	-73.03	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
5509	-73.05	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
5510	-73.1	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
5511	-73.19	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
5512	-73.19	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
5513	-73.33	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
5514	-73.35	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
5515	-73.36	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
5516	-73.36	kd	CGS001-8192	CLPP	ATPases / AAA-type			
5517	-73.39	kd	CGS001-6646	SOAT1	-			
5518	-73.4	oe	ccsbBroad304_10491	PFKL	-			
5519	-73.41	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
5520	-73.42	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5521	-73.46	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
5522	-73.47	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
5523	-73.49	kd	CGS001-3569	IL6	Interferons			
5524	-73.57	kd	CGS001-2147	F2	Endogenous ligands			
5525	-73.58	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
5526	-73.65	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
5527	-73.66	oe	ccsbBroad304_02533	NOXA1	-			
5528	-73.68	oe	ccsbBroad304_00389	CTBP1	-			
5529	-73.7	kd	CGS001-10873	ME3	-			
5530	-73.72	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
5531	-73.76	kd	CGS001-10617	STAMBP	-			
5532	-73.77	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
5533	-73.8	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
5534	-73.87	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
5535	-74.03	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
5536	-74.05	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
5537	-74.08	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
5538	-74.13	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
5539	-74.27	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
5540	-74.29	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
5541	-74.3	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
5542	-74.35	kd	CGS001-4144	MAT2A	-			
5543	-74.37	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
5544	-74.41	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
5545	-74.46	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
5546	-74.55	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
5547	-74.55	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
5548	-74.58	oe	ccsbBroad304_00152	BCAT2	-			
5549	-74.65	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
5550	-74.66	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5551	-74.68	kd	CGS001-638	BIK	-			
5552	-74.7	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
5553	-74.74	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
5554	-74.76	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
5555	-74.76	kd	CGS001-4122	MAN2A2	-			
5556	-74.77	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
5557	-74.8	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
5558	-74.81	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
5559	-74.82	oe	ccsbBroad304_03121	NRBF2	-			
5560	-74.84	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
5561	-74.87	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
5562	-74.89	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
5563	-74.9	kd	CGS001-6856	SYPL1	-			
5564	-74.91	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
5565	-74.97	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
5566	-75.04	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
5567	-75.15	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
5568	-75.16	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
5569	-75.24	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
5570	-75.39	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
5571	-75.45	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
5572	-75.48	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
5573	-75.5	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
5574	-75.58	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
5575	-75.6	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
5576	-75.63	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
5577	-75.64	kd	CGS001-25	ABL1	Abl family			
5578	-75.71	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
5579	-75.77	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
5580	-75.77	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5581	-75.81	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
5582	-75.87	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
5583	-75.9	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
5584	-75.92	kd	CGS001-54498	SMOX	-			
5585	-75.93	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
5586	-75.96	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
5587	-75.99	oe	ccsbBroad304_06386	HNMT	-			
5588	-76.03	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
5589	-76.04	oe	ccsbBroad304_03570	QRSL1	-			
5590	-76.05	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
5591	-76.09	oe	ccsbBroad304_01948	GAS7	-			
5592	-76.1	kd	CGS001-11344	TWF2	Twinfilin subfamily			
5593	-76.13	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
5594	-76.17	kd	CGS001-51741	WWOX	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5595	-76.19	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
5596	-76.19	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
5597	-76.21	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
5598	-76.27	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
5599	-76.31	oe	ccsbBroad304_02580	TMED10	-			
5600	-76.4	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
5601	-76.52	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
5602	-76.53	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
5603	-76.56	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
5604	-76.58	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
5605	-76.59	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
5606	-76.6	kd	CGS001-7128	TNFAIP3	OTU domain containing			
5607	-76.62	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
5608	-76.62	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
5609	-76.64	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
5610	-76.67	oe	ccsbBroad304_02677	PDAP1	-			
5611	-76.67	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
5612	-76.79	kd	CGS001-10898	CPSF4	-			
5613	-76.81	kd	CGS001-3939	LDHA	-			
5614	-76.94	oe	ccsbBroad304_00888	ITPK1	-			
5615	-76.94	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
5616	-76.95	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
5617	-77.05	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5618	-77.05	kd	CGS001-3163	HMOX2	Haem oxygenase			
5619	-77.07	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
5620	-77.11	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
5621	-77.16	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
5622	-77.17	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
5623	-77.24	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
5624	-77.28	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
5625	-77.35	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
5626	-77.38	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
5627	-77.39	kd	CGS001-2967	GTF2H3	General transcription factors			
5628	-77.42	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
5629	-77.46	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
5630	-77.51	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
5631	-77.56	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
5632	-77.64	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
5633	-77.67	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
5634	-77.75	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
5635	-77.77	oe	ccsbBroad304_02834	GABARAPL1	-			
5636	-77.81	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5637	-77.84	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
5638	-77.85	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
5639	-77.88	kd	CGS001-6195	RPS6KA1	RSK subfamily			
5640	-77.9	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
5641	-77.91	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
5642	-77.92	kd	CGS001-2810	SFN	-			
5643	-77.95	oe	ccsbBroad304_06777	PRNP	CD molecules			
5644	-77.95	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
5645	-78.01	kd	CGS001-3930	LBR	Tudor domain containing			
5646	-78.02	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
5647	-78.04	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
5648	-78.12	oe	ccsbBroad304_00954	LYN	Src family			
5649	-78.27	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
5650	-78.28	kd	CGS001-90861	HN1L	-			
5651	-78.3	kd	CGS001-857	CAV1	-			
5652	-78.34	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
5653	-78.38	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
5654	-78.46	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5655	-78.48	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
5656	-78.5	oe	ccsbBroad304_06820	PTS	-			
5657	-78.52	kd	CGS001-29978	UBQLN2	Ubiquilin family			
5658	-78.54	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
5659	-78.56	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
5660	-78.57	oe	ccsbBroad304_07012	STK3	MST subfamily			
5661	-78.59	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
5662	-78.66	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
5663	-78.68	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
5664	-78.69	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5665	-78.7	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
5666	-78.86	kd	CGS001-4637	MYL6	EF-hand domain containing			
5667	-78.87	oe	ccsbBroad304_03420	TOLLIP	-			
5668	-78.89	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
5669	-78.93	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5670	-79	oe	ccsbBroad304_06144	EFNB3	Ephrins			
5671	-79.01	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
5672	-79.02	kd	CGS001-122809	SOCS4	SH2 domain containing			
5673	-79.03	kd	CGS001-400	ARL1	ADP-ribosylation factors			
5674	-79.04	oe	ccsbBroad304_00462	DR1	-			
5675	-79.06	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
5676	-79.06	kd	CGS001-1632	ECI1	-			
5677	-79.09	oe	ccsbBroad304_06318	GPER	-			
5678	-79.11	kd	CGS001-51053	GMNN	-			
5679	-79.17	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
5680	-79.18	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
5681	-79.21	cc		Interleukin receptors LOF	-			
5682	-79.21	kd	CGS001-5887	RAD23B	-			
5683	-79.28	kd	CGS001-29102	DROSHA	-			
5684	-79.29	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
5685	-79.29	kd	CGS001-5763	PTMS	-			
5686	-79.35	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
5687	-79.4	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
5688	-79.48	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
5689	-79.49	cc		Phospholipases GOF	-			
5690	-79.49	oe	ccsbBroad304_00223	CASP9	Caspases			
5691	-79.53	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
5692	-79.55	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
5693	-79.57	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
5694	-79.61	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
5695	-79.65	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
5696	-79.66	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
5697	-79.69	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
5698	-79.7	kd	CGS001-5827	PXMP2	-			
5699	-79.71	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
5700	-79.76	oe	ccsbBroad304_00184	C2	Complement system			
5701	-79.77	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
5702	-79.8	oe	ccsbBroad304_07118	UGDH	-			
5703	-79.82	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
5704	-79.82	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
5705	-79.82	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
5706	-79.87	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
5707	-79.88	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
5708	-79.91	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5709	-79.95	kd	CGS001-4849	CNOT3	-			
5710	-79.99	oe	ccsbBroad304_01976	EIF4EBP3	-			
5711	-80.02	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
5712	-80.02	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
5713	-80.03	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
5714	-80.03	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
5715	-80.12	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
5716	-80.17	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
5717	-80.2	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
5718	-80.2	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
5719	-80.22	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
5720	-80.23	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
5721	-80.28	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
5722	-80.28	kd	CGS001-150280	HORMAD2	-			
5723	-80.3	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
5724	-80.31	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
5725	-80.31	oe	ccsbBroad304_10212	GRHL3	-			
5726	-80.32	kd	CGS001-4594	MUT	-			
5727	-80.35	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
5728	-80.36	kd	CGS001-4351	MPI	-			
5729	-80.37	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
5730	-80.37	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
5731	-80.38	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
5732	-80.39	kd	CGS001-10972	TMED10	-			
5733	-80.4	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
5734	-80.43	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
5735	-80.45	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5736	-80.49	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
5737	-80.5	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
5738	-80.55	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
5739	-80.56	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
5740	-80.58	oe	ccsbBroad304_02298	DNM1L	-			
5741	-80.63	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
5742	-80.65	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
5743	-80.68	oe	ccsbBroad304_00510	EPHX2	-			
5744	-80.68	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
5745	-80.68	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
5746	-80.69	oe	ccsbBroad304_01663	TFF2	-			
5747	-80.71	kd	CGS001-5690	PSMB2	Proteasome subunits			
5748	-80.73	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
5749	-80.74	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
5750	-80.84	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
5751	-80.85	oe	ccsbBroad304_01257	PPOX	-			
5752	-80.85	kd	CGS001-54386	TERF2IP	-			
5753	-80.88	kd	CGS001-29946	SERTAD3	-			
5754	-80.91	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
5755	-80.92	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
5756	-80.94	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
5757	-80.95	kd	CGS001-10452	TOMM40	-			
5758	-80.97	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
5759	-80.98	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
5760	-80.98	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
5761	-80.99	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
5762	-81	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
5763	-81.04	cc		Adenosine receptor agonist	-			
5764	-81.1	oe	ccsbBroad304_01222	PLP2	-			
5765	-81.16	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
5766	-81.2	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
5767	-81.21	kd	CGS001-1840	DTX1	-			
5768	-81.22	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
5769	-81.25	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
5770	-81.25	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
5771	-81.25	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
5772	-81.27	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
5773	-81.31	oe	ccsbBroad304_02676	PHB2	-			
5774	-81.33	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
5775	-81.34	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
5776	-81.36	oe	ccsbBroad304_00710	GUSB	-			
5777	-81.39	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
5778	-81.42	oe	ccsbBroad304_02405	TFG	-			
5779	-81.42	oe	ccsbBroad304_02012	FADD	-			
5780	-81.44	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
5781	-81.51	oe	ccsbBroad304_01617	STX4	-			
5782	-81.55	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
5783	-81.56	oe	ccsbBroad304_07337	TAF1B	-			
5784	-81.58	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5785	-81.65	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
5786	-81.68	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
5787	-81.68	kd	CGS001-1528	CYB5A	Cytochrome b genes			
5788	-81.75	kd	CGS001-9111	NMI	-			
5789	-81.77	oe	ccsbBroad304_02048	BCL10	-			
5790	-81.78	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
5791	-81.84	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
5792	-81.88	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
5793	-81.89	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
5794	-81.94	kd	CGS001-1831	TSC22D3	-			
5795	-81.94	kd	CGS001-9784	SNX17	Sorting nexins			
5796	-81.95	oe	ccsbBroad304_02884	POT1	-			
5797	-81.95	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
5798	-81.96	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
5799	-81.96	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
5800	-82	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
5801	-82	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
5802	-82.07	oe	ccsbBroad304_04457	TOX2	-			
5803	-82.09	oe	ccsbBroad304_06133	TOR1A	-			
5804	-82.11	kd	CGS001-388677	NOTCH2NL	-			
5805	-82.12	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
5806	-82.15	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
5807	-82.15	oe	ccsbBroad304_05963	CD44	CD molecules			
5808	-82.19	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
5809	-82.21	cc		Phospholipases LOF	-			
5810	-82.22	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
5811	-82.23	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
5812	-82.3	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
5813	-82.38	oe	ccsbBroad304_06996	SRM	-			
5814	-82.42	oe	ccsbBroad304_10487	BPHL	-			
5815	-82.43	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5816	-82.46	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
5817	-82.53	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
5818	-82.57	kd	CGS001-673	BRAF	RAF family			
5819	-82.6	kd	CGS001-664	BNIP3	-			
5820	-82.62	oe	ccsbBroad304_00472	EBF1	-			
5821	-82.63	kd	CGS001-84619	ZGPAT	G patch domain containing			
5822	-82.65	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
5823	-82.66	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
5824	-82.82	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
5825	-82.86	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
5826	-82.88	kd	CGS001-5920	RARRES3	-			
5827	-82.89	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
5828	-82.91	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
5829	-82.95	kd	CGS001-11329	STK38	NDR family			
5830	-82.98	kd	CGS001-4121	MAN1A1	-			
5831	-83	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
5832	-83.06	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
5833	-83.14	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
5834	-83.19	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
5835	-83.2	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
5836	-83.2	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5837	-83.22	kd	CGS001-3932	LCK	Src family			
5838	-83.25	oe	ccsbBroad304_00626	GDI1	-			
5839	-83.25	kd	CGS001-5498	PPOX	-			
5840	-83.35	kd	CGS001-5932	RBBP8	-			
5841	-83.38	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
5842	-83.39	kd	CGS001-7040	TGFB1	Endogenous ligands			
5843	-83.4	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
5844	-83.41	kd	CGS001-9270	ITGB1BP1	-			
5845	-83.43	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
5846	-83.49	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
5847	-83.52	oe	ccsbBroad304_06745	PNN	-			
5848	-83.56	oe	ccsbBroad304_02143	CNOT8	-			
5849	-83.57	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
5850	-83.58	cc		MEK inhibitor	-			
5851	-83.63	kd	CGS001-57521	RPTOR	WD repeat domain containing			
5852	-83.66	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
5853	-83.67	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
5854	-83.67	kd	CGS001-226	ALDOA	-			
5855	-83.76	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
5856	-83.78	kd	CGS001-5255	PHKA1	-			
5857	-83.8	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
5858	-83.81	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
5859	-83.81	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
5860	-83.84	cc		BCL inhibitor	-			
5861	-83.88	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5862	-83.9	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
5863	-83.93	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
5864	-83.93	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
5865	-83.95	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
5866	-83.98	oe	ccsbBroad304_01748	UFD1L	-			
5867	-84.01	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
5868	-84.06	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
5869	-84.09	oe	ccsbBroad304_01038	MSRA	-			
5870	-84.11	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
5871	-84.14	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5872	-84.15	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
5873	-84.19	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
5874	-84.19	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
5875	-84.23	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
5876	-84.25	kd	CGS001-327	APEH	Prolyl oligopeptidase			
5877	-84.3	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
5878	-84.41	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
5879	-84.42	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
5880	-84.42	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
5881	-84.42	kd	CGS001-6850	SYK	Syk family			
5882	-84.46	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
5883	-84.51	oe	ccsbBroad304_07102	TSG101	-			
5884	-84.51	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
5885	-84.51	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
5886	-84.53	oe	ccsbBroad304_02414	IRF9	-			
5887	-84.54	kd	CGS001-22933	SIRT2	Histone deacetylases			
5888	-84.55	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
5889	-84.56	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
5890	-84.61	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
5891	-84.63	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
5892	-84.66	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
5893	-84.67	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
5894	-84.69	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
5895	-84.71	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
5896	-84.72	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
5897	-84.72	kd	CGS001-57019	CIAPIN1	-			
5898	-84.73	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
5899	-84.81	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
5900	-84.83	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
5901	-84.86	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
5902	-84.9	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
5903	-84.91	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
5904	-84.93	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
5905	-84.96	kd	CGS001-5106	PCK2	-			
5906	-84.97	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
5907	-85.02	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
5908	-85.05	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
5909	-85.08	kd	CGS001-6184	RPN1	-			
5910	-85.15	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
5911	-85.16	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
5912	-85.17	oe	ccsbBroad304_03928	RRAGC	-			
5913	-85.17	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
5914	-85.17	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
5915	-85.23	kd	CGS001-6810	STX4	-			
5916	-85.23	kd	CGS001-3281	HSBP1	-			
5917	-85.27	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
5918	-85.28	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
5919	-85.28	kd	CGS001-966	CD59	CD molecules			
5920	-85.29	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
5921	-85.31	kd	CGS001-23670	TMEM2	-			
5922	-85.33	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
5923	-85.35	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
5924	-85.35	kd	CGS001-1504	CTRB1	-			
5925	-85.36	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
5926	-85.38	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
5927	-85.4	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
5928	-85.51	oe	ccsbBroad304_13499	KSR2	RAF family			
5929	-85.56	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
5930	-85.56	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
5931	-85.64	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
5932	-85.66	kd	CGS001-5538	PPT1	-			
5933	-85.7	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
5934	-85.7	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
5935	-85.75	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5936	-85.8	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5937	-85.84	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
5938	-85.84	kd	CGS001-3242	HPD	Oxidoreductases			
5939	-85.85	cc		Canonical high mobility group proteins LOF	-			
5940	-85.9	kd	CGS001-2287	FKBP3	-			
5941	-85.91	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5942	-85.96	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
5943	-85.98	oe	ccsbBroad304_00174	BRAF	RAF family			
5944	-86.04	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
5945	-86.04	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
5946	-86.06	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
5947	-86.1	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
5948	-86.17	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
5949	-86.2	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
5950	-86.21	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
5951	-86.22	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
5952	-86.25	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
5953	-86.28	kd	CGS001-4998	ORC1	ATPases / AAA-type			
5954	-86.31	kd	CGS001-843	CASP10	Caspases			
5955	-86.35	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
5956	-86.44	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
5957	-86.45	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
5958	-86.46	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
5959	-86.48	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
5960	-86.48	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
5961	-86.52	kd	CGS001-122402	TDRD9	Tudor domain containing			
5962	-86.52	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
5963	-86.54	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
5964	-86.58	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
5965	-86.61	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
5966	-86.61	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
5967	-86.65	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
5968	-86.7	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
5969	-86.74	kd	CGS001-124535	HSF5	-			
5970	-86.75	oe	ccsbBroad304_08797	FASTKD5	-			
5971	-86.76	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
5972	-86.8	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
5973	-86.82	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
5974	-86.88	oe	ccsbBroad304_01951	BLZF1	-			
5975	-86.89	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
5976	-86.9	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
5977	-86.91	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
5978	-86.93	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
5979	-86.98	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
5980	-86.99	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
5981	-87.02	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5982	-87.02	kd	CGS001-8807	IL18RAP	CD molecules			
5983	-87.03	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
5984	-87.07	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
5985	-87.08	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
5986	-87.08	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
5987	-87.1	kd	CGS001-4860	PNP	-			
5988	-87.12	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
5989	-87.15	oe	ccsbBroad304_01372	RALB	-			
5990	-87.15	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5991	-87.16	cc		Homeobox Gene GOF	-			
5992	-87.19	cc		Dopamine receptor antagonist	-			
5993	-87.19	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
5994	-87.22	cc		PDGFR/KIT inhibitor	-			
5995	-87.22	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
5996	-87.22	kd	CGS001-54881	TEX10	-			
5997	-87.24	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
5998	-87.26	kd	CGS001-54106	TLR9	Toll-like receptor family			
5999	-87.29	kd	CGS001-11041	B3GNT1	-			
6000	-87.36	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
6001	-87.37	oe	ccsbBroad304_06103	DMD	-			
6002	-87.38	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
6003	-87.38	kd	CGS001-384	ARG2	Arginase			
6004	-87.42	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
6005	-87.47	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
6006	-87.47	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
6007	-87.53	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
6008	-87.53	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
6009	-87.55	oe	ccsbBroad304_02789	ADAT1	-			
6010	-87.55	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
6011	-87.56	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
6012	-87.59	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
6013	-87.66	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
6014	-87.67	oe	ccsbBroad304_02419	NDRG1	-			
6015	-87.68	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
6016	-87.69	cc		PKA inhibitor	-			
6017	-87.69	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
6018	-87.7	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6019	-87.73	kd	CGS001-5829	PXN	-			
6020	-87.77	cc		Glycogen synthase kinase inhibitor	-			
6021	-87.77	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
6022	-87.78	kd	CGS001-6275	S100A4	EF-hand domain containing			
6023	-87.78	kd	CGS001-10914	PAPOLA	-			
6024	-87.84	kd	CGS001-4172	MCM3	-			
6025	-87.86	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
6026	-87.86	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6027	-87.88	kd	CGS001-65123	INTS3	-			
6028	-87.94	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
6029	-88.03	cc		Vesicular Transport LOF	-			
6030	-88.03	kd	CGS001-190	NR0B1	DAX-like receptors			
6031	-88.03	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
6032	-88.03	oe	ccsbBroad304_02605	PAPD7	-			
6033	-88.09	kd	CGS001-11140	CDC37	-			
6034	-88.11	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
6035	-88.11	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
6036	-88.11	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
6037	-88.2	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
6038	-88.24	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
6039	-88.24	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
6040	-88.28	cc		MCM family LOF	-			
6041	-88.35	oe	ccsbBroad304_01584	SPARC	-			
6042	-88.35	kd	CGS001-55278	QRSL1	-			
6043	-88.35	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
6044	-88.35	kd	CGS001-595	CCND1	-			
6045	-88.38	oe	ccsbBroad304_08152	PSAT1	-			
6046	-88.38	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
6047	-88.39	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
6048	-88.4	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6049	-88.42	oe	ccsbBroad304_01052	MYB	-			
6050	-88.42	kd	CGS001-2109	ETFB	-			
6051	-88.46	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
6052	-88.53	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
6053	-88.54	kd	CGS001-9275	BCL7B	-			
6054	-88.57	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
6055	-88.57	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
6056	-88.61	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
6057	-88.62	kd	CGS001-5423	POLB	DNA polymerases			
6058	-88.63	kd	CGS001-10412	NSA2	-			
6059	-88.67	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
6060	-88.67	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
6061	-88.68	kd	CGS001-149233	IL23R	IL-12 receptor family			
6062	-88.7	oe	ccsbBroad304_08292	IP6K2	-			
6063	-88.78	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
6064	-88.79	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
6065	-88.81	oe	ccsbBroad304_06188	F10	Chymotrypsin			
6066	-88.87	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6067	-88.91	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
6068	-88.91	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6069	-88.95	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
6070	-88.98	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
6071	-89	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
6072	-89	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
6073	-89.03	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
6074	-89.05	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
6075	-89.1	kd	CGS001-8800	PEX11A	-			
6076	-89.1	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
6077	-89.11	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
6078	-89.12	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
6079	-89.22	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
6080	-89.25	oe	ccsbBroad304_02759	DICER1	-			
6081	-89.32	kd	CGS001-1163	CKS1B	-			
6082	-89.34	kd	CGS001-9	NAT1	-			
6083	-89.37	kd	CGS001-2235	FECH	-			
6084	-89.39	kd	CGS001-4817	NIT1	-			
6085	-89.46	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
6086	-89.49	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
6087	-89.52	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6088	-89.55	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
6089	-89.57	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
6090	-89.62	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
6091	-89.67	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
6092	-89.67	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
6093	-89.68	oe	ccsbBroad304_06837	RAF1	RAF family			
6094	-89.68	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
6095	-89.74	kd	CGS001-10285	SMNDC1	Tudor domain containing			
6096	-89.75	kd	CGS001-112858	TP53RK	Bud32 family			
6097	-89.77	oe	ccsbBroad304_00032	ADSL	-			
6098	-89.78	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
6099	-89.84	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
6100	-89.85	cc		CCK receptor antagonist	-			
6101	-89.85	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
6102	-89.86	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6103	-89.87	kd	CGS001-4089	SMAD4	SMADs			
6104	-89.89	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
6105	-89.91	cc		RAF inhibitor	-			
6106	-89.92	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
6107	-89.94	kd	CGS001-55634	ZNF673	-			
6108	-89.95	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
6109	-89.96	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
6110	-89.97	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6111	-90.02	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
6112	-90.03	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
6113	-90.07	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
6114	-90.1	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
6115	-90.1	kd	CGS001-3046	HBE1	-			
6116	-90.12	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
6117	-90.13	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
6118	-90.19	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
6119	-90.22	cc		Potassium channel activator	-			
6120	-90.24	kd	CGS001-7082	TJP1	-			
6121	-90.32	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
6122	-90.33	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
6123	-90.38	oe	ccsbBroad304_07724	KDELR2	-			
6124	-90.45	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
6125	-90.45	kd	CGS001-8480	RAE1	WD repeat domain containing			
6126	-90.48	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
6127	-90.49	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
6128	-90.53	kd	CGS001-6464	SHC1	SH2 domain containing			
6129	-90.58	oe	ccsbBroad304_01211	PKM2	-			
6130	-90.58	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
6131	-90.6	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
6132	-90.65	kd	CGS001-2067	ERCC1	-			
6133	-90.68	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
6134	-90.69	oe	ccsbBroad304_08339	CMPK1	-			
6135	-90.74	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
6136	-90.75	cc		NFKB Activation GOF	-			
6137	-90.78	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
6138	-90.86	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
6139	-90.93	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
6140	-90.95	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
6141	-91.06	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
6142	-91.07	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
6143	-91.09	kd	CGS001-8900	CCNA1	-			
6144	-91.1	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
6145	-91.13	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
6146	-91.18	cp	BRD-K53220666	trimetozine	Sedative			Sedative
6147	-91.18	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
6148	-91.18	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
6149	-91.19	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
6150	-91.19	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
6151	-91.23	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
6152	-91.25	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
6153	-91.26	kd	CGS001-56993	TOMM22	-			
6154	-91.26	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
6155	-91.27	cc		VEGFR inhibitor	-			
6156	-91.27	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
6157	-91.35	kd	CGS001-213	ALB	-			
6158	-91.38	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
6159	-91.4	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
6160	-91.42	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
6161	-91.43	oe	ccsbBroad304_07208	NRIP1	-			
6162	-91.49	kd	CGS001-10020	GNE	-			
6163	-91.51	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6164	-91.53	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
6165	-91.54	oe	ccsbBroad304_01304	PSEN1	Presenilin			
6166	-91.55	oe	ccsbBroad304_08660	SMARCAD1	-			
6167	-91.56	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
6168	-91.56	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
6169	-91.58	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
6170	-91.58	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
6171	-91.59	oe	ccsbBroad304_00489	EHHADH	-			
6172	-91.61	oe	ccsbBroad304_08952	E2F8	-			
6173	-91.62	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6174	-91.65	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
6175	-91.69	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
6176	-91.73	oe	ccsbBroad304_07101	TSC2	-			
6177	-91.73	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
6178	-91.74	kd	CGS001-10128	LRPPRC	-			
6179	-91.76	oe	ccsbBroad304_06783	LGMN	Legumain			
6180	-91.78	cc		IGF-1 inhibitor	-			
6181	-91.79	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
6182	-91.79	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
6183	-91.81	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
6184	-91.81	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
6185	-91.82	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
6186	-91.82	kd	CGS001-5881	RAC3	Endogenous ligands			
6187	-91.83	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
6188	-91.84	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
6189	-91.85	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
6190	-91.9	kd	CGS001-5663	PSEN1	Presenilin			
6191	-91.92	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
6192	-92	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6193	-92.03	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
6194	-92.03	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6195	-92.08	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
6196	-92.1	oe	ccsbBroad304_05183	TXLNA	-			
6197	-92.13	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
6198	-92.15	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
6199	-92.15	kd	CGS001-1029	CDKN2A	-			
6200	-92.16	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
6201	-92.18	oe	ccsbBroad304_00518	ETFA	-			
6202	-92.18	kd	CGS001-10765	KDM5B	Histone demethylases			
6203	-92.23	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6204	-92.23	kd	CGS001-6723	SRM	-			
6205	-92.24	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
6206	-92.26	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6207	-92.26	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
6208	-92.26	kd	CGS001-2581	GALC	-			
6209	-92.27	oe	ccsbBroad304_07326	EIF2B2	-			
6210	-92.27	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
6211	-92.27	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
6212	-92.28	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
6213	-92.29	kd	CGS001-23499	MACF1	EF-hand domain containing			
6214	-92.31	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
6215	-92.31	kd	CGS001-644	BLVRA	-			
6216	-92.39	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
6217	-92.43	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
6218	-92.43	kd	CGS001-11044	PAPD7	-			
6219	-92.44	cc		Lipocalins GOF	-			
6220	-92.47	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
6221	-92.47	kd	CGS001-3985	LIMK2	LIMK subfamily			
6222	-92.49	oe	ccsbBroad304_02398	LANCL1	-			
6223	-92.49	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
6224	-92.5	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
6225	-92.52	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
6226	-92.55	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
6227	-92.55	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6228	-92.61	kd	CGS001-11243	PMF1	-			
6229	-92.65	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
6230	-92.65	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
6231	-92.65	kd	CGS001-7316	UBC	-			
6232	-92.68	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6233	-92.68	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
6234	-92.73	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
6235	-92.76	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
6236	-92.77	cc		Cyclins LOF	-			
6237	-92.8	oe	ccsbBroad304_07592	CEPT1	-			
6238	-92.8	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
6239	-92.82	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
6240	-92.85	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
6241	-92.87	cc		CDK inhibitor	-			
6242	-92.9	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
6243	-92.94	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
6244	-92.95	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
6245	-92.95	kd	CGS001-498	ATP5A1	ATPases / F-type			
6246	-92.99	cc		Ribosomal 40s Subunit LOF	-			
6247	-93.03	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
6248	-93.06	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
6249	-93.06	kd	CGS001-2077	ERF	ETS Transcription Factors			
6250	-93.09	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
6251	-93.1	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
6252	-93.1	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
6253	-93.11	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
6254	-93.12	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
6255	-93.13	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
6256	-93.18	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
6257	-93.22	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
6258	-93.22	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
6259	-93.23	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
6260	-93.24	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
6261	-93.26	cc		FLT3 inhibitor	-			
6262	-93.26	kd	CGS001-4664	NAB1	-			
6263	-93.35	cc		SMAD family LOF	-			
6264	-93.35	kd	CGS001-2645	GCK	Hexokinases			
6265	-93.36	kd	CGS001-4046	LSP1	-			
6266	-93.39	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
6267	-93.4	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
6268	-93.41	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
6269	-93.42	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
6270	-93.46	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
6271	-93.5	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6272	-93.51	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
6273	-93.55	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
6274	-93.58	cc		HOXL subclass homeoboxes LOF	-			
6275	-93.58	kd	CGS001-64858	DCLRE1B	-			
6276	-93.62	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
6277	-93.66	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
6278	-93.67	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
6279	-93.74	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
6280	-93.78	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6281	-93.82	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
6282	-93.82	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
6283	-93.83	oe	ccsbBroad304_00238	CCNE1	-			
6284	-93.87	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
6285	-93.88	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
6286	-93.9	kd	CGS001-55165	CEP55	-			
6287	-93.91	oe	ccsbBroad304_06992	SRC	Src family			
6288	-93.93	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
6289	-93.94	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
6290	-94	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
6291	-94.06	oe	ccsbBroad304_02579	YWHAQ	-			
6292	-94.06	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
6293	-94.06	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
6294	-94.07	cc		Serpin peptidase inhibitors LOF	-			
6295	-94.09	oe	ccsbBroad304_06538	LSP1	-			
6296	-94.12	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
6297	-94.16	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
6298	-94.17	oe	ccsbBroad304_06095	DFFB	-			
6299	-94.18	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
6300	-94.2	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6301	-94.2	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
6302	-94.2	kd	CGS001-3029	HAGH	-			
6303	-94.21	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
6304	-94.22	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
6305	-94.23	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
6306	-94.29	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
6307	-94.31	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
6308	-94.33	kd	CGS001-383	ARG1	Arginase			
6309	-94.35	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
6310	-94.38	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6311	-94.38	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
6312	-94.39	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
6313	-94.41	oe	ccsbBroad304_05528	TICAM2	-			
6314	-94.42	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
6315	-94.43	kd	CGS001-375449	MAST4	MAST family			
6316	-94.46	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
6317	-94.46	kd	CGS001-2160	F11	Chymotrypsin			
6318	-94.47	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
6319	-94.49	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
6320	-94.51	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
6321	-94.59	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
6322	-94.66	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
6323	-94.67	oe	ccsbBroad304_07275	PSMG1	-			
6324	-94.69	oe	ccsbBroad304_00398	CTSL2	-			
6325	-94.7	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
6326	-94.73	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
6327	-94.75	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
6328	-94.81	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
6329	-94.88	oe	ccsbBroad304_13813	ARAF	RAF family			
6330	-94.92	cc		HDAC inhibitor	-			
6331	-94.94	oe	ccsbBroad304_06494	KLRC1	CD molecules			
6332	-94.97	kd	CGS001-9375	TM9SF2	-			
6333	-94.98	kd	CGS001-27161	EIF2C2	-			
6334	-94.99	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
6335	-95	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
6336	-95	kd	CGS001-6514	SLC2A2	Solute carriers			
6337	-95.02	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
6338	-95.03	oe	ccsbBroad304_07861	COBL	-			
6339	-95.03	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
6340	-95.05	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
6341	-95.08	oe	ccsbBroad304_02402	TMEM5	-			
6342	-95.09	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
6343	-95.1	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
6344	-95.11	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
6345	-95.12	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
6346	-95.13	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
6347	-95.15	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
6348	-95.17	kd	CGS001-1429	CRYZ	-			
6349	-95.18	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
6350	-95.2	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
6351	-95.22	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6352	-95.23	cc		JAK inhibitor	-			
6353	-95.26	oe	ccsbBroad304_00690	GRN	-			
6354	-95.27	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
6355	-95.27	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
6356	-95.28	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
6357	-95.29	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
6358	-95.29	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
6359	-95.31	kd	CGS001-29915	HCFC2	-			
6360	-95.35	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
6361	-95.37	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
6362	-95.39	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
6363	-95.4	cc		Thromboxane receptor antagonist	-			
6364	-95.41	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
6365	-95.42	kd	CGS001-216	ALDH1A1	Aldehyde dehydrogenases			
6366	-95.49	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
6367	-95.52	cc		Trace amine receptors LOF	-			
6368	-95.54	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
6369	-95.57	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
6370	-95.58	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
6371	-95.59	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
6372	-95.6	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
6373	-95.62	oe	ccsbBroad304_00632	GGCX	Carboxylases			
6374	-95.64	kd	CGS001-51720	UIMC1	-			
6375	-95.65	oe	ccsbBroad304_01673	TIMP3	-			
6376	-95.65	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
6377	-95.65	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
6378	-95.66	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
6379	-95.67	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
6380	-95.7	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
6381	-95.72	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
6382	-95.73	oe	ccsbBroad304_07050	TFAP2A	-			
6383	-95.73	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
6384	-95.77	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
6385	-95.79	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
6386	-95.8	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
6387	-95.83	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
6388	-95.91	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
6389	-95.93	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
6390	-95.93	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
6391	-95.94	oe	ccsbBroad304_07071	TKT	-			
6392	-95.94	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
6393	-95.96	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
6394	-96.02	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
6395	-96.04	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
6396	-96.05	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6397	-96.06	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
6398	-96.12	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
6399	-96.18	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6400	-96.21	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
6401	-96.21	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
6402	-96.22	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
6403	-96.23	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
6404	-96.24	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
6405	-96.27	kd	CGS001-4067	LYN	Src family			
6406	-96.27	kd	CGS001-23242	COBL	-			
6407	-96.29	oe	ccsbBroad304_00975	MAT2A	-			
6408	-96.29	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
6409	-96.3	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
6410	-96.3	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
6411	-96.3	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
6412	-96.3	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
6413	-96.3	kd	CGS001-18	ABAT	GABA turnover			
6414	-96.32	cc		PI3K inhibitor	-			
6415	-96.33	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
6416	-96.33	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
6417	-96.33	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
6418	-96.34	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
6419	-96.37	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
6420	-96.39	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6421	-96.4	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
6422	-96.43	oe	ccsbBroad304_03850	TRIB3	Trbl family			
6423	-96.43	kd	CGS001-4221	MEN1	-			
6424	-96.44	oe	ccsbBroad304_09396	TIRAP	-			
6425	-96.45	cc		PKC inhibitor	-			
6426	-96.48	cc		EGFR inhibitor	-			
6427	-96.48	kd	CGS001-9710	KIAA0355	-			
6428	-96.49	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
6429	-96.49	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
6430	-96.5	oe	ccsbBroad304_05152	SSBP4	-			
6431	-96.52	kd	CGS001-121599	SPIC	ETS Transcription Factors			
6432	-96.52	kd	CGS001-85004	RERG	-			
6433	-96.54	kd	CGS001-5900	RALGDS	-			
6434	-96.58	kd	CGS001-3383	ICAM1	CD molecules			
6435	-96.59	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
6436	-96.59	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
6437	-96.61	kd	CGS001-10472	ZNF238	-			
6438	-96.61	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
6439	-96.63	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
6440	-96.68	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6441	-96.69	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6442	-96.69	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
6443	-96.72	cc		Proteasome inhibitor	-			
6444	-96.72	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6445	-96.72	oe	ccsbBroad304_08709	SCYL3	-			
6446	-96.73	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
6447	-96.74	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6448	-96.74	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
6449	-96.74	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
6450	-96.76	oe	ccsbBroad304_00962	SMAD4	SMADs			
6451	-96.77	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6452	-96.78	kd	CGS001-51014	TMED7	-			
6453	-96.79	oe	ccsbBroad304_02276	MVP	-			
6454	-96.8	kd	CGS001-5580	PRKCD	Delta subfamily			
6455	-96.82	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
6456	-96.82	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6457	-96.82	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
6458	-96.82	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6459	-96.83	kd	CGS001-8536	CAMK1	CAMK1 family			
6460	-96.84	cc		HIF activator	-			
6461	-96.84	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
6462	-96.84	kd	CGS001-26511	CHIC2	-			
6463	-96.84	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
6464	-96.86	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
6465	-96.88	cc		Bromodomain Inhibitor	-			
6466	-96.9	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
6467	-96.92	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
6468	-96.92	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
6469	-96.92	kd	CGS001-4905	NSF	ATPases / AAA-type			
6470	-96.92	kd	CGS001-10491	CRTAP	-			
6471	-96.93	kd	CGS001-55486	PARL	-			
6472	-96.94	cc		PARP inhibitor	-			
6473	-96.99	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
6474	-97.02	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
6475	-97.07	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
6476	-97.09	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
6477	-97.09	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
6478	-97.1	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
6479	-97.1	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
6480	-97.12	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
6481	-97.12	kd	CGS001-4090	SMAD5	SMADs			
6482	-97.13	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
6483	-97.14	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
6484	-97.17	oe	ccsbBroad304_00268	CD81	CD molecules			
6485	-97.17	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
6486	-97.18	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
6487	-97.2	oe	ccsbBroad304_01180	PFKFB3	-			
6488	-97.2	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
6489	-97.21	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
6490	-97.21	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
6491	-97.23	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
6492	-97.23	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
6493	-97.24	kd	CGS001-3572	IL6ST	IL-6 receptor family			
6494	-97.26	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
6495	-97.28	kd	CGS001-8837	CFLAR	Endogenous ligands			
6496	-97.29	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
6497	-97.31	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
6498	-97.33	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
6499	-97.33	kd	CGS001-11180	WDR6	WD repeat domain containing			
6500	-97.35	oe	ccsbBroad304_00282	CDKN1A	-			
6501	-97.37	oe	ccsbBroad304_00728	HBE1	-			
6502	-97.4	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
6503	-97.41	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
6504	-97.42	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
6505	-97.46	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
6506	-97.48	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
6507	-97.49	cc		Minor histocompatibility antigens LOF	-			
6508	-97.49	oe	ccsbBroad304_03264	UBAP1	-			
6509	-97.5	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
6510	-97.52	cc		MTOR inhibitor	-			
6511	-97.53	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6512	-97.53	kd	CGS001-23369	PUM2	-			
6513	-97.53	kd	CGS001-2615	LRRC32	-			
6514	-97.56	kd	CGS001-6772	STAT1	SH2 domain containing			
6515	-97.56	kd	CGS001-1879	EBF1	-			
6516	-97.58	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
6517	-97.6	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
6518	-97.61	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
6519	-97.64	oe	ccsbBroad304_00376	CSK	Csk family			
6520	-97.64	oe	ccsbBroad304_01351	PEX19	-			
6521	-97.65	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
6522	-97.65	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
6523	-97.67	kd	CGS001-51290	ERGIC2	-			
6524	-97.69	oe	ccsbBroad304_01662	TFDP2	-			
6525	-97.7	kd	CGS001-10544	PROCR	CD molecules			
6526	-97.75	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
6527	-97.76	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
6528	-97.78	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6529	-97.79	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
6530	-97.81	oe	ccsbBroad304_02569	BTG3	-			
6531	-97.82	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6532	-97.82	kd	CGS001-55526	DHTKD1	-			
6533	-97.83	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
6534	-97.85	oe	ccsbBroad304_03177	FIS1	-			
6535	-97.88	kd	CGS001-3481	IGF2	-			
6536	-97.89	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
6537	-97.9	oe	ccsbBroad304_04786	CANT1	-			
6538	-97.9	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
6539	-97.9	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
6540	-97.92	oe	ccsbBroad304_04038	ELOVL6	-			
6541	-97.94	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
6542	-97.94	kd	CGS001-4907	NT5E	Adenosine turnover			
6543	-97.96	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
6544	-97.97	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
6545	-97.97	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
6546	-97.97	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
6547	-98	oe	ccsbBroad304_00490	EIF4EBP1	-			
6548	-98	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
6549	-98.01	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
6550	-98.01	oe	ccsbBroad304_03444	PAF1	-			
6551	-98.01	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
6552	-98.02	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
6553	-98.03	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
6554	-98.06	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
6555	-98.07	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
6556	-98.08	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
6557	-98.1	oe	ccsbBroad304_02890	SYF2	-			
6558	-98.1	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
6559	-98.1	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
6560	-98.1	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
6561	-98.1	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
6562	-98.13	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
6563	-98.13	kd	CGS001-10943	MSL3	-			
6564	-98.15	kd	CGS001-84722	PSRC1	-			
6565	-98.17	oe	ccsbBroad304_00617	GBA	-			
6566	-98.17	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
6567	-98.17	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
6568	-98.17	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
6569	-98.18	cc		PKC activator	-			
6570	-98.19	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
6571	-98.2	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
6572	-98.21	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
6573	-98.21	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
6574	-98.21	kd	CGS001-6208	RPS14	S ribosomal proteins			
6575	-98.23	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
6576	-98.23	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
6577	-98.23	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
6578	-98.24	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6579	-98.24	kd	CGS001-284119	PTRF	-			
6580	-98.26	kd	CGS001-6387	CXCL12	Endogenous ligands			
6581	-98.27	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
6582	-98.28	oe	ccsbBroad304_01862	YEATS4	-			
6583	-98.29	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
6584	-98.3	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
6585	-98.31	kd	CGS001-23475	QPRT	-			
6586	-98.32	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6587	-98.32	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
6588	-98.33	kd	CGS001-9512	PMPCB	-			
6589	-98.34	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6590	-98.36	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
6591	-98.36	kd	CGS001-54555	DDX49	DEAD-boxes			
6592	-98.37	oe	ccsbBroad304_01664	TGFA	-			
6593	-98.39	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
6594	-98.4	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
6595	-98.4	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
6596	-98.42	oe	ccsbBroad304_14291	GDPD5	-			
6597	-98.42	kd	CGS001-7832	BTG2	-			
6598	-98.43	kd	CGS001-9455	HOMER2	-			
6599	-98.47	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
6600	-98.48	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
6601	-98.49	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
6602	-98.5	kd	CGS001-1497	CTNS	-			
6603	-98.5	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
6604	-98.51	kd	CGS001-10652	YKT6	-			
6605	-98.52	oe	ccsbBroad304_06976	SMARCE1	-			
6606	-98.52	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
6607	-98.52	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
6608	-98.53	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
6609	-98.54	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
6610	-98.55	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
6611	-98.56	kd	CGS001-10427	SEC24B	-			
6612	-98.57	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
6613	-98.58	oe	ccsbBroad304_08878	METTL4	-			
6614	-98.63	kd	CGS001-6193	RPS5	S ribosomal proteins			
6615	-98.64	oe	ccsbBroad304_02840	PISD	Decarboxylases			
6616	-98.67	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
6617	-98.67	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
6618	-98.7	oe	ccsbBroad304_01556	SMARCB1	-			
6619	-98.7	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
6620	-98.72	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6621	-98.73	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
6622	-98.73	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
6623	-98.75	cc		Cell Cycle Inhibition GOF	-			
6624	-98.76	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6625	-98.76	oe	ccsbBroad304_03615	ZNF673	-			
6626	-98.76	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
6627	-98.79	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
6628	-98.79	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
6629	-98.81	kd	CGS001-771	CA12	Carbonic anhydrases			
6630	-98.82	cc		IMPDH inhibitor	-			
6631	-98.82	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
6632	-98.83	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
6633	-98.84	kd	CGS001-5292	PIM1	PIM family			
6634	-98.85	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
6635	-98.86	oe	ccsbBroad304_00519	ETFB	-			
6636	-98.86	oe	ccsbBroad304_07466	VGLL4	-			
6637	-98.87	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
6638	-98.88	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
6639	-98.91	kd	CGS001-23753	SDF2L1	-			
6640	-98.94	oe	ccsbBroad304_00832	IFNB1	Interferons			
6641	-98.94	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
6642	-98.94	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
6643	-98.95	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
6644	-98.96	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
6645	-98.96	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
6646	-98.97	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
6647	-98.98	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
6648	-98.98	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
6649	-98.99	oe	ccsbBroad304_09054	EGFL8	-			
6650	-99.01	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
6651	-99.04	kd	CGS001-5194	PEX13	-			
6652	-99.06	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
6653	-99.06	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
6654	-99.06	kd	CGS001-84890	ADO	-			
6655	-99.07	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
6656	-99.07	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
6657	-99.07	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
6658	-99.08	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6659	-99.09	oe	ccsbBroad304_01469	RSU1	-			
6660	-99.09	oe	ccsbBroad304_06094	DFFA	-			
6661	-99.09	kd	CGS001-345611	IRGM	-			
6662	-99.11	cc		AHSP Pathway LOF	-			
6663	-99.11	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
6664	-99.11	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
6665	-99.12	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
6666	-99.13	oe	ccsbBroad304_03450	TMED9	-			
6667	-99.13	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
6668	-99.13	kd	CGS001-64343	AZI2	-			
6669	-99.15	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
6670	-99.15	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
6671	-99.17	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
6672	-99.18	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
6673	-99.18	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
6674	-99.18	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
6675	-99.18	kd	CGS001-1662	DDX10	DEAD-boxes			
6676	-99.19	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
6677	-99.2	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
6678	-99.2	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
6679	-99.2	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
6680	-99.21	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
6681	-99.22	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
6682	-99.22	kd	CGS001-84547	PGBD1	-			
6683	-99.23	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
6684	-99.23	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
6685	-99.23	kd	CGS001-5209	PFKFB3	-			
6686	-99.25	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
6687	-99.25	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
6688	-99.25	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
6689	-99.25	kd	CGS001-3516	RBPJ	-			
6690	-99.25	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
6691	-99.26	kd	CGS001-55746	NUP133	-			
6692	-99.26	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
6693	-99.26	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
6694	-99.28	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6695	-99.29	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
6696	-99.29	kd	CGS001-29940	DSE	-			
6697	-99.31	kd	CGS001-28960	DCPS	-			
6698	-99.32	cc		T-type calcium channel blocker	-			
6699	-99.32	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
6700	-99.33	kd	CGS001-1152	CKB	-			
6701	-99.34	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
6702	-99.34	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
6703	-99.34	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
6704	-99.35	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
6705	-99.35	oe	ccsbBroad304_07197	PDHX	-			
6706	-99.35	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6707	-99.36	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
6708	-99.37	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
6709	-99.37	oe	ccsbBroad304_00966	MAFG	-			
6710	-99.37	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
6711	-99.37	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
6712	-99.39	kd	CGS001-7840	ALMS1	-			
6713	-99.4	cc		Sterol demethylase inhibitor	-			
6714	-99.4	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
6715	-99.4	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
6716	-99.41	cc		Ribonucleotide reductase inhibitor	-			
6717	-99.41	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
6718	-99.41	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
6719	-99.41	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6720	-99.41	kd	CGS001-23081	KDM4C	Histone demethylases			
6721	-99.43	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6722	-99.43	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
6723	-99.45	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
6724	-99.45	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
6725	-99.47	cc		Cyclin dependent kinases LOF	-			
6726	-99.47	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
6727	-99.47	oe	ccsbBroad304_05980	CDKN1B	-			
6728	-99.47	kd	CGS001-9276	COPB2	WD repeat domain containing			
6729	-99.48	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
6730	-99.48	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
6731	-99.48	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
6732	-99.48	kd	CGS001-5264	PHYH	-			
6733	-99.5	oe	ccsbBroad304_02230	HERPUD1	-			
6734	-99.5	oe	ccsbBroad304_05894	BLVRA	-			
6735	-99.52	kd	CGS001-10538	BATF	basic leucine zipper proteins			
6736	-99.53	cc		Protein synthesis inhibitor	-			
6737	-99.53	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
6738	-99.53	kd	CGS001-1503	CTPS	-			
6739	-99.54	oe	ccsbBroad304_07277	RTCD1	-			
6740	-99.54	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
6741	-99.54	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
6742	-99.54	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
6743	-99.56	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
6744	-99.56	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
6745	-99.56	kd	CGS001-10673	TNFSF13B	CD molecules			
6746	-99.57	cc		General transcription factors group 2 LOF	-			
6747	-99.57	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
6748	-99.57	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
6749	-99.57	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
6750	-99.57	kd	CGS001-30001	ERO1L	-			
6751	-99.57	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6752	-99.58	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
6753	-99.59	cc		Sirtuins GOF	-			
6754	-99.59	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
6755	-99.59	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
6756	-99.59	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
6757	-99.59	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
6758	-99.59	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
6759	-99.59	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
6760	-99.6	oe	ccsbBroad304_07145	ZFP161	-			
6761	-99.6	oe	ccsbBroad304_06888	RPN1	-			
6762	-99.6	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
6763	-99.6	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
6764	-99.6	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
6765	-99.6	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
6766	-99.62	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
6767	-99.62	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
6768	-99.62	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
6769	-99.62	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
6770	-99.63	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
6771	-99.63	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
6772	-99.63	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6773	-99.63	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
6774	-99.63	kd	CGS001-847	CAT	-			
6775	-99.65	cc		DNA polymerase inhibitor	-			
6776	-99.65	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
6777	-99.65	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
6778	-99.65	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
6779	-99.65	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
6780	-99.65	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
6781	-99.65	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
6782	-99.65	kd	CGS001-1072	CFL1	-			
6783	-99.66	oe	ccsbBroad304_02136	COPS2	-			
6784	-99.66	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
6785	-99.66	kd	CGS001-64121	RRAGC	-			
6786	-99.66	kd	CGS001-6194	RPS6	S ribosomal proteins			
6787	-99.66	kd	CGS001-178	AGL	-			
6788	-99.67	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
6789	-99.68	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
6790	-99.68	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
6791	-99.68	kd	CGS001-11040	PIM2	PIM family			
6792	-99.69	oe	ccsbBroad304_01401	RIT1	-			
6793	-99.69	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
6794	-99.69	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
6795	-99.69	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
6796	-99.69	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6797	-99.69	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
6798	-99.69	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
6799	-99.69	kd	CGS001-51750	RTEL1	-			
6800	-99.7	oe	ccsbBroad304_07128	VHL	-			
6801	-99.71	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
6802	-99.71	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
6803	-99.71	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
6804	-99.71	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
6805	-99.72	oe	ccsbBroad304_00146	BAD	-			
6806	-99.72	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
6807	-99.72	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
6808	-99.73	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
6809	-99.73	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
6810	-99.73	oe	ccsbBroad304_00316	CKS1B	-			
6811	-99.73	kd	CGS001-3920	LAMP2	CD molecules			
6812	-99.73	kd	CGS001-9641	IKBKE	IKK family			
6813	-99.75	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
6814	-99.75	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
6815	-99.75	oe	ccsbBroad304_02788	PRAME	-			
6816	-99.75	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
6817	-99.75	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
6818	-99.75	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
6819	-99.76	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
6820	-99.76	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
6821	-99.76	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
6822	-99.77	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6823	-99.78	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
6824	-99.78	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
6825	-99.78	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
6826	-99.78	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
6827	-99.78	kd	CGS001-11230	PRAF2	-			
6828	-99.78	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6829	-99.79	oe	ccsbBroad304_07506	UBAP2L	-			
6830	-99.79	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
6831	-99.79	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
6832	-99.79	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
6833	-99.79	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
6834	-99.8	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
6835	-99.81	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
6836	-99.81	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
6837	-99.81	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
6838	-99.81	kd	CGS001-5573	PRKAR1A	Protein kinase A			
6839	-99.81	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
6840	-99.81	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
6841	-99.81	kd	CGS001-11212	PROSC	-			
6842	-99.82	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
6843	-99.82	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
6844	-99.82	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
6845	-99.82	kd	CGS001-7054	TH	Amino acid hydroxylases			
6846	-99.84	oe	ccsbBroad304_02509	GMEB1	-			
6847	-99.84	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
6848	-99.85	cc		IKK inhibitor	-			
6849	-99.85	oe	ccsbBroad304_01165	PDK1	-			
6850	-99.85	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
6851	-99.85	kd	CGS001-10523	CHERP	G patch domain containing			
6852	-99.86	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
6853	-99.87	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
6854	-99.87	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
6855	-99.87	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
6856	-99.87	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6857	-99.87	kd	CGS001-126823	KLHDC9	-			
6858	-99.87	kd	CGS001-8727	CTNNAL1	Catenins			
6859	-99.88	cc		DNA dependent protein kinase inhibitor	-			
6860	-99.88	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
6861	-99.88	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
6862	-99.88	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
6863	-99.88	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
6864	-99.88	kd	CGS001-81539	SLC38A1	System A-like transporters			
6865	-99.88	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
6866	-99.89	kd	CGS001-56882	CDC42SE1	-			
6867	-99.9	oe	ccsbBroad304_07124	UROD	-			
6868	-99.9	oe	ccsbBroad304_06789	PSEN2	Presenilin			
6869	-99.9	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
6870	-99.9	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
6871	-99.91	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
6872	-99.91	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
6873	-99.91	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
6874	-99.91	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
6875	-99.91	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
6876	-99.91	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
6877	-99.91	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
6878	-99.91	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
6879	-99.91	kd	CGS001-25885	POLR1A	RNA polymerase subunits			
6880	-99.93	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
6881	-99.93	oe	ccsbBroad304_08392	EXOC6	-			
6882	-99.93	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
6883	-99.93	oe	ccsbBroad304_00118	ATIC	-			
6884	-99.93	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
6885	-99.93	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
6886	-99.93	kd	CGS001-6188	RPS3	S ribosomal proteins			
6887	-99.93	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
6888	-99.93	kd	CGS001-256281	NUDT14	Nudix motif containing			
6889	-99.93	kd	CGS001-10682	EBP	-			
6890	-99.93	kd	CGS001-64170	CARD9	-			
6891	-99.93	oe	ccsbBroad304_00551	FECH	-			
6892	-99.94	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
6893	-99.94	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6894	-99.94	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
6895	-99.94	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6896	-99.94	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
6897	-99.94	kd	CGS001-10797	MTHFD2	-			
6898	-99.95	kd	CGS001-10318	TNIP1	-			
6899	-99.96	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
6900	-99.96	oe	ccsbBroad304_03798	PHTF2	-			
6901	-99.96	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
6902	-99.96	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
6903	-99.96	oe	ccsbBroad304_00529	F3	CD molecules			
6904	-99.96	oe	ccsbBroad304_10240	CROT	-			
6905	-99.96	oe	ccsbBroad304_00077	APEX1	-			
6906	-99.96	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
6907	-99.96	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
6908	-99.96	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
6909	-99.96	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
6910	-99.96	kd	CGS001-3476	IGBP1	-			
6911	-99.96	kd	CGS001-7089	TLE2	WD repeat domain containing			
6912	-99.96	kd	CGS001-6197	RPS6KA3	RSK subfamily			
6913	-99.96	kd	CGS001-2963	GTF2F2	General transcription factors			
6914	-99.96	kd	CGS001-2266	FGG	Endogenous ligands			
6915	-99.96	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
6916	-99.97	oe	ccsbBroad304_02487	TXNIP	-			
6917	-99.97	oe	ccsbBroad304_07363	AIFM1	-			
6918	-99.97	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
6919	-99.97	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
6920	-99.97	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
6921	-99.97	oe	ccsbBroad304_06993	SRD5A1	-			
6922	-99.97	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
6923	-99.97	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
6924	-99.97	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
6925	-99.97	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
6926	-99.97	oe	ccsbBroad304_06828	PYCR1	-			
6927	-99.97	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
6928	-99.97	oe	ccsbBroad304_01034	MSH2	-			
6929	-99.97	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
6930	-99.97	oe	ccsbBroad304_08840	KIF9	Kinesins			
6931	-99.97	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
6932	-99.97	oe	ccsbBroad304_00794	HSF1	-			
6933	-99.97	oe	ccsbBroad304_02370	HRSP12	-			
6934	-99.97	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
6935	-99.97	oe	ccsbBroad304_06286	GLUL	-			
6936	-99.97	oe	ccsbBroad304_00420	DAP	-			
6937	-99.97	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
6938	-99.97	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
6939	-99.97	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
6940	-99.97	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
6941	-99.97	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
6942	-99.97	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
6943	-99.97	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
6944	-99.97	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6945	-99.97	kd	CGS001-8741	TNFSF13	CD molecules			
6946	-99.97	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
6947	-99.97	kd	CGS001-347736	NME9	-			
6948	-99.97	kd	CGS001-4174	MCM5	-			
6949	-99.97	kd	CGS001-11019	LIAS	-			
6950	-99.97	kd	CGS001-23510	KCTD2	-			
6951	-99.97	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
6952	-99.97	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
6953	-99.97	kd	CGS001-2821	GPI	-			
6954	-99.97	kd	CGS001-2277	FIGF	-			
6955	-99.97	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
6956	-99.97	kd	CGS001-79071	ELOVL6	-			
6957	-99.97	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
6958	-99.97	kd	CGS001-1399	CRKL	SH2 domain containing			
6959	-99.97	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
6960	-99.97	kd	CGS001-9133	CCNB2	-			
6961	-99.97	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
6962	-99.97	kd	CGS001-842	CASP9	Caspases			
6963	-99.97	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
6964	-99.97	kd	CGS001-310	ANXA7	Annexins			
6965	-99.97	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
6966	-99.97	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
6967	-99.97	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
6968	-99.97	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
6969	-99.97	oe	ccsbBroad304_03732	NPDC1	-			
6970	-100	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
6971	-100	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
6972	-100	kd	CGS001-5033	P4HA1	-			
