Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
2	99.99	kd	CGS001-1786	DNMT1	Methyltransferases			
3	99.97	cc		Ubiquitin-specific peptidases LOF	-			
4	99.97	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
5	99.97	oe	ccsbBroad304_07097	TRAF1	-			
6	99.97	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
7	99.97	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
8	99.97	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
9	99.97	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
10	99.97	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
11	99.97	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
12	99.97	oe	ccsbBroad304_07561	YAF2	-			
13	99.97	oe	ccsbBroad304_08116	TBK1	IKK family			
14	99.97	oe	ccsbBroad304_07238	STK24	YSK subfamily			
15	99.97	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
16	99.97	oe	ccsbBroad304_12106	PXK	Slob family			
17	99.97	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
18	99.97	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
19	99.97	oe	ccsbBroad304_06665	OAT	-			
20	99.97	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
21	99.97	oe	ccsbBroad304_03848	METTL14	-			
22	99.97	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
23	99.97	oe	ccsbBroad304_00644	GCLC	-			
24	99.97	oe	ccsbBroad304_00469	DUT	-			
25	99.97	oe	ccsbBroad304_08346	COQ3	-			
26	99.97	oe	ccsbBroad304_02686	COPZ1	-			
27	99.97	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
28	99.97	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
29	99.97	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
30	99.97	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
31	99.97	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
32	99.97	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
33	99.97	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
34	99.97	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
35	99.97	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
36	99.97	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
37	99.97	kd	CGS001-6282	S100A11	EF-hand domain containing			
38	99.97	kd	CGS001-6204	RPS10	S ribosomal proteins			
39	99.97	kd	CGS001-4781	NFIB	-			
40	99.97	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
41	99.97	kd	CGS001-3566	IL4R	IL-2 receptor family			
42	99.97	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
43	99.97	kd	CGS001-3033	HADH	-			
44	99.97	kd	CGS001-9638	FEZ1	-			
45	99.97	kd	CGS001-55556	ENOSF1	-			
46	99.97	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
47	99.97	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
48	99.97	kd	CGS001-7917	BAG6	-			
49	99.97	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
50	99.96	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
51	99.96	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
52	99.96	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
53	99.96	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
54	99.96	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
55	99.96	kd	CGS001-2023	ENO1	-			
56	99.96	kd	CGS001-11129	CLASRP	-			
57	99.94	oe	ccsbBroad304_02045	BUD31	-			
58	99.94	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
59	99.94	oe	ccsbBroad304_02057	P4HA2	-			
60	99.94	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
61	99.94	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
62	99.94	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
63	99.94	kd	CGS001-6857	SYT1	Synaptotagmins			
64	99.94	kd	CGS001-8576	STK16	NAK family			
65	99.94	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
66	99.94	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
67	99.94	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
68	99.94	oe	ccsbBroad304_06739	PLOD1	-			
69	99.93	cc		Beta-adrenergic receptor agonist	-			
70	99.93	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
71	99.93	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
72	99.93	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
73	99.93	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
74	99.93	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
75	99.93	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
76	99.93	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
77	99.93	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
78	99.93	kd	CGS001-24140	FTSJ1	-			
79	99.93	kd	CGS001-10289	EIF1B	-			
80	99.93	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
81	99.93	kd	CGS001-32	ACACB	Carboxylases			
82	99.92	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
83	99.91	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
84	99.91	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
85	99.91	oe	ccsbBroad304_03565	ADI1	-			
86	99.91	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
87	99.91	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
88	99.91	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
89	99.9	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
90	99.9	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
91	99.9	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
92	99.9	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
93	99.9	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
94	99.9	kd	CGS001-5236	PGM1	-			
95	99.9	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
96	99.9	kd	CGS001-100	ADA	Adenosine turnover			
97	99.88	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
98	99.88	kd	CGS001-3925	STMN1	-			
99	99.88	kd	CGS001-23536	ADAT1	-			
100	99.87	cc		IL4 Pathway LOF	-			
101	99.87	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
102	99.87	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
103	99.87	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
104	99.87	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
105	99.87	kd	CGS001-7298	TYMS	Methyltransferases			
106	99.87	kd	CGS001-10613	ERLIN1	-			
107	99.87	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
108	99.86	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
109	99.85	oe	ccsbBroad304_09281	TPD52L3	-			
110	99.85	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
111	99.85	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
112	99.85	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
113	99.85	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
114	99.85	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
115	99.85	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
116	99.85	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
117	99.84	oe	ccsbBroad304_00836	IGF2	-			
118	99.84	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
119	99.82	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
120	99.82	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
121	99.82	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
122	99.82	kd	CGS001-5590	PRKCZ	Iota subfamily			
123	99.82	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
124	99.81	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
125	99.81	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
126	99.81	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
127	99.79	oe	ccsbBroad304_00359	CPT1A	-			
128	99.79	kd	CGS001-10474	TADA3	-			
129	99.79	kd	CGS001-4668	NAGA	-			
130	99.79	kd	CGS001-3980	LIG3	-			
131	99.78	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
132	99.78	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
133	99.78	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
134	99.76	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
135	99.76	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
136	99.75	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
137	99.75	oe	ccsbBroad304_00509	EPHX1	-			
138	99.75	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
139	99.75	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
140	99.75	kd	CGS001-4946	OAZ1	-			
141	99.75	kd	CGS001-115	ADCY9	Adenylyl cyclases			
142	99.73	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
143	99.73	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
144	99.73	kd	CGS001-10972	TMED10	-			
145	99.73	kd	CGS001-2770	GNAI1	-			
146	99.72	kd	CGS001-10617	STAMBP	-			
147	99.71	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
148	99.69	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
149	99.69	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
150	99.68	kd	CGS001-51441	YTHDF2	-			
151	99.66	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
152	99.66	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
153	99.66	kd	CGS001-51001	MTERFD1	-			
154	99.66	oe	ccsbBroad304_07017	SUOX	-			
155	99.65	oe	ccsbBroad304_07920	NUP62	-			
156	99.65	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
157	99.64	kd	CGS001-23142	DCUN1D4	-			
158	99.63	oe	ccsbBroad304_00833	IFNG	Interferons			
159	99.63	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
160	99.63	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
161	99.63	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
162	99.62	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
163	99.62	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
164	99.61	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
165	99.6	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
166	99.59	oe	ccsbBroad304_08266	PIPOX	-			
167	99.59	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
168	99.59	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
169	99.59	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
170	99.58	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
171	99.58	kd	CGS001-2961	GTF2E2	General transcription factors			
172	99.57	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
173	99.56	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
174	99.54	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
175	99.54	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
176	99.54	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
177	99.54	kd	CGS001-7525	YES1	Src family			
178	99.53	oe	ccsbBroad304_06013	CLPTM1	-			
179	99.53	oe	ccsbBroad304_05756	ACAA1	-			
180	99.53	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
181	99.53	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
182	99.52	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
183	99.52	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
184	99.51	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
185	99.51	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
186	99.51	kd	CGS001-54915	YTHDF1	-			
187	99.51	kd	CGS001-5306	PITPNA	-			
188	99.51	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
189	99.51	kd	CGS001-3676	ITGA4	Integrins			
190	99.5	kd	CGS001-23678	SGK3	SGK family			
191	99.48	oe	ccsbBroad304_03372	CAB39	-			
192	99.48	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
193	99.48	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
194	99.48	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
195	99.48	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
196	99.48	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
197	99.48	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
198	99.47	oe	ccsbBroad304_01139	PA2G4	-			
199	99.47	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
200	99.47	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
201	99.47	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
202	99.47	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
203	99.45	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
204	99.44	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
205	99.42	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
206	99.4	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
207	99.38	oe	ccsbBroad304_00001	NAT1	-			
208	99.38	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
209	99.38	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
210	99.36	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
211	99.35	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
212	99.35	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
213	99.35	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
214	99.34	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
215	99.32	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
216	99.32	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
217	99.3	kd	CGS001-1763	DNA2	-			
218	99.29	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
219	99.29	kd	CGS001-2115	ETV1	ETS Transcription Factors			
220	99.28	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
221	99.28	kd	CGS001-185	AGTR1	Angiotensin receptors			
222	99.26	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
223	99.26	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
224	99.23	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
225	99.23	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
226	99.23	kd	CGS001-717	C2	Complement system			
227	99.22	oe	ccsbBroad304_08093	DCPS	-			
228	99.2	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
229	99.2	kd	CGS001-8720	MBTPS1	Subtilisin			
230	99.19	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
231	99.18	kd	CGS001-4193	MDM2	-			
232	99.18	kd	CGS001-55715	DOK4	Pleckstrin homology (PH) domain containing			
233	99.18	kd	CGS001-25874	BRP44	-			
234	99.17	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
235	99.17	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
236	99.17	oe	ccsbBroad304_06172	EPS8	-			
237	99.16	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
238	99.16	kd	CGS001-8692	HYAL2	-			
239	99.15	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
240	99.15	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
241	99.14	cc		IGF-1 inhibitor	-			
242	99.14	kd	CGS001-3251	HPRT1	-			
243	99.13	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
244	99.13	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
245	99.1	oe	ccsbBroad304_00424	DBI	-			
246	99.08	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
247	99.07	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
248	99.06	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
249	99.03	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
250	99.03	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
251	99.01	kd	CGS001-6513	SLC2A1	Solute carriers			
252	99.01	kd	CGS001-1356	CP	-			
253	99	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
254	98.98	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
255	98.95	oe	ccsbBroad304_01674	TIMP4	-			
256	98.94	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
257	98.94	oe	ccsbBroad304_01186	PHB	-			
258	98.94	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
259	98.94	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
260	98.92	cc		Homeobox Gene GOF	-			
261	98.92	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
262	98.92	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
263	98.91	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
264	98.91	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
265	98.89	oe	ccsbBroad304_07053	TFPI	-			
266	98.87	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
267	98.86	oe	ccsbBroad304_03878	SENP2	-			
268	98.86	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
269	98.82	kd	CGS001-587	BCAT2	-			
270	98.79	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
271	98.79	oe	ccsbBroad304_05823	ANXA2	Annexins			
272	98.78	oe	ccsbBroad304_00459	DPYD	-			
273	98.76	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
274	98.76	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
275	98.75	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
276	98.73	kd	CGS001-378	ARF4	ADP-ribosylation factors			
277	98.72	oe	ccsbBroad304_00003	ABAT	GABA turnover			
278	98.72	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
279	98.72	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
280	98.71	kd	CGS001-84433	CARD11	-			
281	98.71	kd	CGS001-8896	BUD31	-			
282	98.7	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
283	98.69	oe	ccsbBroad304_06695	PCK2	-			
284	98.69	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
285	98.67	kd	CGS001-9943	OXSR1	FRAY subfamily			
286	98.66	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
287	98.66	kd	CGS001-5359	PLSCR1	-			
288	98.66	kd	CGS001-5091	PC	Carboxylases			
289	98.66	kd	CGS001-56675	NRIP3	-			
290	98.66	kd	CGS001-5927	KDM5A	Histone demethylases			
291	98.66	kd	CGS001-55612	FERMT1	Fermitins			
292	98.66	kd	CGS001-2184	FAH	-			
293	98.65	oe	ccsbBroad304_01880	LAGE3	-			
294	98.64	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
295	98.64	kd	CGS001-9967	THRAP3	-			
296	98.63	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
297	98.63	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
298	98.58	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
299	98.58	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
300	98.58	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
301	98.57	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
302	98.54	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
303	98.53	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
304	98.52	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
305	98.51	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
306	98.47	kd	CGS001-51002	TPRKB	-			
307	98.46	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
308	98.45	oe	ccsbBroad304_08386	SMOX	-			
309	98.45	kd	CGS001-79006	METRN	-			
310	98.44	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
311	98.4	oe	ccsbBroad304_01374	RAP1A	-			
312	98.38	oe	ccsbBroad304_03853	LSM2	-			
313	98.38	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
314	98.38	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
315	98.36	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
316	98.36	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
317	98.34	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
318	98.32	kd	CGS001-10973	ASCC3	-			
319	98.31	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
320	98.3	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
321	98.29	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
322	98.29	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
323	98.28	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
324	98.28	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
325	98.28	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
326	98.27	kd	CGS001-665	BNIP3L	-			
327	98.26	oe	ccsbBroad304_07851	FAM120A	-			
328	98.22	cc		Estrogen receptor antagonist	-			
329	98.22	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
330	98.2	oe	ccsbBroad304_01234	POLB	DNA polymerases			
331	98.2	kd	CGS001-5446	PON3	Paraoxonases			
332	98.19	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
333	98.19	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
334	98.17	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
335	98.17	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
336	98.16	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
337	98.14	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
338	98.13	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
339	98.12	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
340	98.1	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
341	98.09	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
342	98.08	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
343	98.08	kd	CGS001-4817	NIT1	-			
344	98.08	kd	CGS001-9404	LPXN	-			
345	98.08	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
346	98.07	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
347	98.05	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
348	98.04	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
349	98.04	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
350	98.04	kd	CGS001-5562	PRKAA1	AMPK subfamily			
351	98.03	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
352	98.03	kd	CGS001-10221	TRIB1	Trbl family			
353	98.02	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
354	98.02	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
355	98.01	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
356	98.01	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
357	98.01	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
358	98.01	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
359	97.95	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
360	97.94	kd	CGS001-23530	NNT	-			
361	97.92	kd	CGS001-10284	SAP18	-			
362	97.9	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
363	97.9	kd	CGS001-9158	FIBP	-			
364	97.88	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
365	97.85	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
366	97.85	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
367	97.84	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
368	97.83	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
369	97.83	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
370	97.83	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
371	97.83	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
372	97.83	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
373	97.82	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
374	97.82	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
375	97.82	kd	CGS001-9833	MELK	MELK subfamily			
376	97.8	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
377	97.78	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
378	97.78	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
379	97.77	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
380	97.76	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
381	97.75	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
382	97.74	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
383	97.74	kd	CGS001-79947	DHDDS	-			
384	97.71	kd	CGS001-873	CBR1	Prostaglandin synthases			
385	97.7	oe	ccsbBroad304_03308	YTHDF2	-			
386	97.69	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
387	97.68	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
388	97.67	oe	ccsbBroad304_03910	CCDC90A	-			
389	97.67	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
390	97.67	kd	CGS001-1955	MEGF9	-			
391	97.63	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
392	97.63	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
393	97.62	oe	ccsbBroad304_07768	NISCH	-			
394	97.62	oe	ccsbBroad304_01623	SUPT4H1	-			
395	97.56	oe	ccsbBroad304_03097	CNOT7	-			
396	97.49	kd	CGS001-22954	TRIM32	-			
397	97.47	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
398	97.46	oe	ccsbBroad304_00552	FEN1	-			
399	97.46	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
400	97.45	cc		NFkB pathway inhibitor	-			
401	97.45	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
402	97.43	oe	ccsbBroad304_06458	IRF3	-			
403	97.43	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
404	97.41	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
405	97.41	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
406	97.4	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
407	97.37	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
408	97.36	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
409	97.33	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
410	97.33	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
411	97.31	kd	CGS001-6598	SMARCB1	-			
412	97.29	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
413	97.27	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
414	97.26	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
415	97.26	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
416	97.24	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
417	97.23	oe	ccsbBroad304_06294	GNAZ	-			
418	97.23	kd	CGS001-10423	CDIPT	-			
419	97.22	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
420	97.21	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
421	97.21	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
422	97.19	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
423	97.17	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
424	97.16	kd	CGS001-1509	CTSD	Cathepsins			
425	97.15	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
426	97.13	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
427	97.13	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
428	97.12	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
429	97.09	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
430	97.08	oe	ccsbBroad304_02052	KYNU	-			
431	97.08	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
432	97.03	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
433	97.02	kd	CGS001-545	ATR	ATR subfamily			
434	96.97	cc		Cyclooxygenase inhibitor	-			
435	96.96	oe	ccsbBroad304_02425	CDIPT	-			
436	96.96	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
437	96.96	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
438	96.92	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
439	96.91	kd	CGS001-51564	HDAC7	Histone deacetylases			
440	96.9	kd	CGS001-9443	MED7	-			
441	96.86	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
442	96.82	kd	CGS001-23223	RRP12	-			
443	96.81	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
444	96.8	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
445	96.78	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
446	96.76	oe	ccsbBroad304_03268	GMPR2	-			
447	96.72	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
448	96.71	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
449	96.71	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
450	96.7	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
451	96.69	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
452	96.69	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
453	96.69	kd	CGS001-255877	BCL6B	BTB/POZ domain containing			
454	96.64	oe	ccsbBroad304_01203	PIM1	PIM family			
455	96.61	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
456	96.6	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
457	96.58	kd	CGS001-1105	CHD1	-			
458	96.56	kd	CGS001-89882	TPD52L3	-			
459	96.54	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
460	96.54	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
461	96.52	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
462	96.49	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
463	96.48	kd	CGS001-391013	PLA2G2C	-			
464	96.42	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
465	96.4	oe	ccsbBroad304_07102	TSG101	-			
466	96.4	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
467	96.37	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
468	96.33	oe	ccsbBroad304_07511	KIF14	Kinesins			
469	96.33	oe	ccsbBroad304_06159	CTTN	-			
470	96.33	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
471	96.3	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
472	96.27	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
473	96.27	kd	CGS001-4299	AFF1	-			
474	96.25	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
475	96.25	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
476	96.25	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
477	96.24	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
478	96.23	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
479	96.22	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
480	96.2	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
481	96.18	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
482	96.18	oe	ccsbBroad304_01605	SSX2	-			
483	96.12	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
484	96.08	oe	ccsbBroad304_00164	BLMH	-			
485	96.08	kd	CGS001-1951	CELSR3	Cadherins / Major cadherins			
486	96.06	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
487	96.05	oe	ccsbBroad304_08825	LHPP	-			
488	96.05	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
489	96.03	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
490	96.01	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
491	96.01	kd	CGS001-23344	ESYT1	Synaptotagmins			
492	95.98	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
493	95.95	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
494	95.92	kd	CGS001-2108	ETFA	-			
495	95.9	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
496	95.86	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
497	95.8	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
498	95.75	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
499	95.72	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
500	95.68	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
501	95.68	oe	ccsbBroad304_14242	MCCC2	-			
502	95.55	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
503	95.5	oe	ccsbBroad304_03232	VPS28	-			
504	95.5	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
505	95.5	kd	CGS001-9180	OSMR	IL-6 receptor family			
506	95.45	oe	ccsbBroad304_02834	GABARAPL1	-			
507	95.44	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
508	95.42	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
509	95.41	oe	ccsbBroad304_02565	RALBP1	-			
510	95.37	oe	ccsbBroad304_01845	RDBP	-			
511	95.35	oe	ccsbBroad304_01651	TCF7L2	-			
512	95.35	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
513	95.35	kd	CGS001-2592	GALT	-			
514	95.29	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
515	95.29	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
516	95.26	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
517	95.24	oe	ccsbBroad304_03640	CEP72	-			
518	95.23	kd	CGS001-2745	GLRX	-			
519	95.23	kd	CGS001-29940	DSE	-			
520	95.21	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
521	95.17	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
522	95.17	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
523	95.17	kd	CGS001-1659	DHX8	DEAH-boxes			
524	95.14	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
525	95.12	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
526	95.08	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
527	95.05	oe	ccsbBroad304_00063	AMPD2	-			
528	95.05	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
529	95.05	kd	CGS001-7423	VEGFB	-			
530	95.01	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
531	94.99	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
532	94.94	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
533	94.94	kd	CGS001-22908	SACM1L	-			
534	94.92	kd	CGS001-10452	TOMM40	-			
535	94.91	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
536	94.91	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
537	94.88	kd	CGS001-23464	GCAT	-			
538	94.88	oe	ccsbBroad304_06998	SRPK1	SRPK family			
539	94.84	kd	CGS001-57804	POLD4	DNA polymerases			
540	94.82	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
541	94.82	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
542	94.77	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
543	94.75	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
544	94.72	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
545	94.72	kd	CGS001-3169	FOXA1	Forkhead boxes			
546	94.7	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
547	94.62	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
548	94.59	oe	ccsbBroad304_02837	BHMT2	-			
549	94.54	kd	CGS001-27297	CRCP	-			
550	94.51	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
551	94.5	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
552	94.47	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
553	94.47	kd	CGS001-1120	CHKB	-			
554	94.39	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
555	94.38	kd	CGS001-1837	DTNA	-			
556	94.37	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
557	94.37	kd	CGS001-1026	CDKN1A	-			
558	94.36	kd	CGS001-6652	SORD	-			
559	94.32	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
560	94.3	oe	ccsbBroad304_02737	JMJD6	-			
561	94.26	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
562	94.21	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
563	94.18	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
564	94.13	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
565	94.07	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
566	94.01	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
567	94.01	kd	CGS001-57819	LSM2	-			
568	94	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
569	93.91	kd	CGS001-83440	ADPGK	-			
570	93.89	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
571	93.81	kd	CGS001-6727	SRP14	-			
572	93.78	kd	CGS001-4610	MYCL1	-			
573	93.77	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
574	93.77	oe	ccsbBroad304_03113	DSE	-			
575	93.75	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
576	93.75	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
577	93.74	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
578	93.69	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
579	93.67	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
580	93.65	kd	CGS001-116832	RPL39L	L ribosomal proteins			
581	93.5	cc		PI3K inhibitor	-			
582	93.5	kd	CGS001-5653	KLK6	Chymotrypsin			
583	93.49	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
584	93.46	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
585	93.4	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
586	93.38	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
587	93.34	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
588	93.33	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
589	93.29	kd	CGS001-10398	MYL9	EF-hand domain containing			
590	93.28	kd	CGS001-7029	TFDP2	-			
591	93.27	oe	ccsbBroad304_05547	TMEM110	-			
592	93.26	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
593	93.25	oe	ccsbBroad304_00392	CTLA4	CD molecules			
594	93.25	oe	ccsbBroad304_06098	DHCR24	-			
595	93.25	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
596	93.25	kd	CGS001-57680	CHD8	-			
597	93.21	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
598	93.21	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
599	93.17	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
600	93.13	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
601	93.13	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
602	93.1	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
603	93.09	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
604	93.05	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
605	93.04	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
606	93	kd	CGS001-3029	HAGH	-			
607	92.95	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
608	92.91	oe	ccsbBroad304_08662	MCCC1	-			
609	92.88	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
610	92.86	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
611	92.85	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
612	92.85	oe	ccsbBroad304_01613	STK11	LKB subfamily			
613	92.83	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
614	92.83	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
615	92.81	cc		Tubulin inhibitor	-			
616	92.8	oe	ccsbBroad304_03933	CARD9	-			
617	92.79	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
618	92.75	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
619	92.69	oe	ccsbBroad304_01485	SC5DL	-			
620	92.66	kd	CGS001-3800	KIF5C	Kinesins			
621	92.66	oe	ccsbBroad304_03080	C16ORF80	-			
622	92.65	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
623	92.64	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
624	92.52	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
625	92.49	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
626	92.49	kd	CGS001-727	C5	Endogenous ligands			
627	92.46	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
628	92.41	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
629	92.39	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
630	92.3	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
631	92.28	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
632	92.26	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
633	92.25	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
634	92.25	kd	CGS001-5831	PYCR1	-			
635	92.23	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
636	92.22	kd	CGS001-11212	PROSC	-			
637	92.2	oe	ccsbBroad304_04170	PANK2	-			
638	92.2	oe	ccsbBroad304_03415	GFOD1	-			
639	92.19	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
640	92.14	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
641	92.13	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
642	92.08	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
643	92.05	oe	ccsbBroad304_06889	RPN2	-			
644	91.99	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
645	91.98	kd	CGS001-11124	FAF1	UBX domain containing			
646	91.96	kd	CGS001-89910	UBE3B	-			
647	91.94	cc		C2 domain containing LOF	-			
648	91.93	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
649	91.8	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
650	91.76	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
651	91.72	oe	ccsbBroad304_06089	DDIT3	-			
652	91.72	kd	CGS001-55176	SEC61A2	-			
653	91.7	kd	CGS001-6714	SRC	Src family			
654	91.69	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
655	91.66	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
656	91.65	kd	CGS001-29763	PACSIN3	-			
657	91.64	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
658	91.64	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
659	91.56	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
660	91.53	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
661	91.51	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
662	91.47	kd	CGS001-572	BAD	-			
663	91.43	oe	ccsbBroad304_04655	TRIM9	-			
664	91.4	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
665	91.31	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
666	91.29	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
667	91.29	kd	CGS001-11182	SLC2A6	Solute carriers			
668	91.29	kd	CGS001-3034	HAL	-			
669	91.26	oe	ccsbBroad304_06255	LRRC32	-			
670	91.22	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
671	91.17	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
672	91.16	kd	CGS001-9709	HERPUD1	-			
673	91.15	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
674	91.13	oe	ccsbBroad304_09615	LACC1	-			
675	91.13	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
676	91.11	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
677	91.08	oe	ccsbBroad304_06720	PHYH	-			
678	91.07	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
679	91.07	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
680	91.04	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
681	91.02	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
682	90.9	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
683	90.89	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
684	90.88	kd	CGS001-5092	PCBD1	-			
685	90.84	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
686	90.83	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
687	90.77	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
688	90.76	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
689	90.6	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
690	90.57	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
691	90.57	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
692	90.49	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
693	90.41	oe	ccsbBroad304_03951	NARFL	-			
694	90.41	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
695	90.39	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
696	90.38	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
697	90.37	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
698	90.34	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
699	90.31	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
700	90.27	kd	CGS001-1376	CPT2	-			
701	90.24	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
702	90.2	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
703	90.19	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
704	90.19	kd	CGS001-8050	PDHX	-			
705	90.12	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
706	90.04	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
707	90.03	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
708	90.01	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
709	90	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
710	89.97	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
711	89.97	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
712	89.93	kd	CGS001-2538	G6PC	-			
713	89.92	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
714	89.83	kd	CGS001-4976	OPA1	-			
715	89.82	oe	ccsbBroad304_10437	STMN1	-			
716	89.79	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
717	89.78	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
718	89.76	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
719	89.76	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
720	89.76	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
721	89.75	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
722	89.74	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
723	89.67	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
724	89.67	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
725	89.65	cc		Targets of VEGFR inhibitors GOF	-			
726	89.63	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
727	89.61	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
728	89.6	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
729	89.58	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
730	89.56	kd	CGS001-6778	STAT6	SH2 domain containing			
731	89.54	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
732	89.53	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
733	89.5	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
734	89.48	oe	ccsbBroad304_02708	TRIM32	-			
735	89.42	oe	ccsbBroad304_01787	YES1	Src family			
736	89.42	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
737	89.37	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
738	89.32	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
739	89.29	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
740	89.26	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
741	89.23	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
742	89.21	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
743	89.21	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
744	89.21	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
745	89.14	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
746	89.11	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
747	89.09	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
748	89.06	kd	CGS001-7405	UVRAG	-			
749	88.95	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
750	88.92	oe	ccsbBroad304_06382	HMGCL	-			
751	88.91	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
752	88.88	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
753	88.81	kd	CGS001-4292	MLH1	-			
754	88.76	oe	ccsbBroad304_00116	ASS1	-			
755	88.74	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
756	88.73	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
757	88.72	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
758	88.71	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
759	88.7	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
760	88.67	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
761	88.61	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
762	88.59	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
763	88.59	kd	CGS001-3608	ILF2	-			
764	88.58	kd	CGS001-10928	RALBP1	-			
765	88.56	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
766	88.55	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
767	88.52	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
768	88.46	kd	CGS001-23014	FBXO21	F-boxes / other			
769	88.46	kd	CGS001-25966	C2CD2	-			
770	88.45	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
771	88.44	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
772	88.44	kd	CGS001-1840	DTX1	-			
773	88.42	kd	CGS001-6603	SMARCD2	-			
774	88.39	cc		IKK inhibitor	-			
775	88.37	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
776	88.36	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
777	88.36	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
778	88.35	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
779	88.34	kd	CGS001-161	AP2A2	-			
780	88.3	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
781	88.29	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
782	88.29	kd	CGS001-8435	SOAT2	-			
783	88.28	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
784	88.28	oe	ccsbBroad304_06574	MDH2	-			
785	88.24	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
786	88.21	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
787	88.2	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
788	88.18	oe	ccsbBroad304_06562	MAT1A	-			
789	88.13	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
790	88.11	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
791	88.09	kd	CGS001-5073	PARN	-			
792	88.08	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
793	88.07	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
794	88.07	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
795	87.99	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
796	87.92	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
797	87.85	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
798	87.84	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
799	87.82	kd	CGS001-10670	RRAGA	-			
800	87.8	kd	CGS001-8826	IQGAP1	-			
801	87.8	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
802	87.78	oe	ccsbBroad304_03129	ERO1L	-			
803	87.77	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
804	87.74	oe	ccsbBroad304_00532	F11	Chymotrypsin			
805	87.7	kd	CGS001-30836	DNTTIP2	-			
806	87.69	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
807	87.69	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
808	87.63	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
809	87.61	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
810	87.61	kd	CGS001-2353	FOS	basic leucine zipper proteins			
811	87.52	kd	CGS001-4312	MMP1	Matrix metallopeptidase			
812	87.47	oe	ccsbBroad304_03405	CHRAC1	-			
813	87.47	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
814	87.43	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
815	87.3	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
816	87.23	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
817	87.23	kd	CGS001-2113	ETS1	ETS Transcription Factors			
818	87.21	oe	ccsbBroad304_03357	RASD1	-			
819	87.18	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
820	87.13	kd	CGS001-389421	LIN28B	-			
821	87.12	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
822	87.09	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
823	87.07	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
824	87.05	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
825	87	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
826	86.99	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
827	86.94	kd	CGS001-10682	EBP	-			
828	86.93	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
829	86.87	oe	ccsbBroad304_00570	FIGF	-			
830	86.86	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
831	86.85	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
832	86.82	kd	CGS001-230	ALDOC	-			
833	86.8	kd	CGS001-3420	IDH3B	-			
834	86.75	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
835	86.69	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
836	86.69	kd	CGS001-8295	TRRAP	TRRAP subfamily			
837	86.66	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
838	86.66	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
839	86.6	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
840	86.54	kd	CGS001-3630	INS	-			
841	86.54	kd	CGS001-3479	IGF1	Endogenous ligands			
842	86.53	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
843	86.5	kd	CGS001-10434	LYPLA1	-			
844	86.49	kd	CGS001-2057	EPOR	Prolactin receptor family			
845	86.49	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
846	86.48	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
847	86.43	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
848	86.41	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
849	86.39	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
850	86.38	kd	CGS001-2773	GNAI3	-			
851	86.38	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
852	86.37	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
853	86.36	kd	CGS001-51292	GMPR2	-			
854	86.32	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
855	86.31	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
856	86.26	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
857	86.25	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
858	86.24	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
859	86.18	oe	ccsbBroad304_02756	RRP8	-			
860	86.18	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
861	86.16	oe	ccsbBroad304_01247	POU2AF1	-			
862	86.15	kd	CGS001-2244	FGB	Endogenous ligands			
863	86.11	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
864	86.11	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
865	86.11	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
866	86.03	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
867	86.01	kd	CGS001-55082	ARGLU1	-			
868	85.99	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
869	85.93	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
870	85.92	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
871	85.91	kd	CGS001-1725	DHPS	-			
872	85.89	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
873	85.81	kd	CGS001-2079	ERH	-			
874	85.81	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
875	85.8	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
876	85.7	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
877	85.68	oe	ccsbBroad304_08775	SQRDL	-			
878	85.67	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
879	85.66	kd	CGS001-5966	REL	NFkappaB transcription factor family			
880	85.6	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
881	85.59	kd	CGS001-150094	SIK1	QIK subfamily			
882	85.56	oe	ccsbBroad304_02361	MFSD10	-			
883	85.46	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
884	85.46	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
885	85.42	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
886	85.4	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
887	85.39	kd	CGS001-9231	DLG5	-			
888	85.38	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
889	85.37	oe	ccsbBroad304_04202	MED28	-			
890	85.37	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
891	85.32	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
892	85.3	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
893	85.3	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
894	85.3	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
895	85.27	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
896	85.27	kd	CGS001-8535	CBX4	-			
897	85.24	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
898	85.21	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
899	85.17	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
900	85.16	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
901	85.14	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
902	85.12	kd	CGS001-25819	CCRN4L	-			
903	85.06	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
904	85.03	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
905	85	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
906	85	kd	CGS001-3725	JUN	basic leucine zipper proteins			
907	84.97	oe	ccsbBroad304_02551	CPSF4	-			
908	84.93	oe	ccsbBroad304_01013	MIF	-			
909	84.92	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
910	84.91	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
911	84.89	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
912	84.88	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
913	84.83	cc		MTOR inhibitor	-			
914	84.8	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
915	84.79	kd	CGS001-51727	CMPK1	-			
916	84.73	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
917	84.72	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
918	84.71	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
919	84.69	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
920	84.67	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
921	84.61	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
922	84.61	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
923	84.58	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
924	84.56	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
925	84.51	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
926	84.51	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
927	84.5	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
928	84.46	kd	CGS001-2475	MTOR	FRAP subfamily			
929	84.44	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
930	84.44	kd	CGS001-29105	C16ORF80	-			
931	84.42	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
932	84.23	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
933	84.19	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
934	84.17	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
935	84.13	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
936	84.12	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
937	84.04	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
938	84.02	kd	CGS001-1314	COPA	Endogenous ligands			
939	84	oe	ccsbBroad304_02772	ICMT	-			
940	83.96	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
941	83.91	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
942	83.88	oe	ccsbBroad304_01163	PDHA1	-			
943	83.87	oe	ccsbBroad304_01066	NDUFA4	-			
944	83.86	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
945	83.86	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
946	83.82	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
947	83.82	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
948	83.82	kd	CGS001-1604	CD55	CD molecules			
949	83.8	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
950	83.8	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
951	83.8	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
952	83.79	kd	CGS001-133690	CAPSL	EF-hand domain containing			
953	83.73	kd	CGS001-54861	SNRK	SNRK subfamily			
954	83.72	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
955	83.71	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
956	83.7	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
957	83.69	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
958	83.69	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
959	83.68	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
960	83.65	kd	CGS001-10247	HRSP12	-			
961	83.64	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
962	83.63	kd	CGS001-2247	FGF2	Endogenous ligands			
963	83.6	cc		FOS transcription factor family GOF	-			
964	83.56	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
965	83.53	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
966	83.53	oe	ccsbBroad304_01974	RNASET2	-			
967	83.52	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
968	83.52	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
969	83.5	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
970	83.48	oe	ccsbBroad304_06048	CRYZ	-			
971	83.45	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
972	83.43	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
973	83.42	oe	ccsbBroad304_01208	PITPNA	-			
974	83.41	oe	ccsbBroad304_03772	CCNL1	-			
975	83.38	kd	CGS001-6223	RPS19	S ribosomal proteins			
976	83.36	kd	CGS001-7295	TXN	-			
977	83.35	kd	CGS001-10904	BLCAP	-			
978	83.34	kd	CGS001-103	ADAR	-			
979	83.3	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
980	83.27	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
981	83.23	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
982	83.23	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
983	83.2	kd	CGS001-3682	ITGAE	Integrins			
984	83.19	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
985	83.17	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
986	83.13	oe	ccsbBroad304_02048	BCL10	-			
987	83.11	oe	ccsbBroad304_03023	CRCP	-			
988	83.03	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
989	83.03	kd	CGS001-4170	MCL1	-			
990	83	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
991	83	kd	CGS001-10657	KHDRBS1	-			
992	82.99	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
993	82.96	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
994	82.95	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
995	82.95	oe	ccsbBroad304_00961	SMAD2	SMADs			
996	82.95	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
997	82.9	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
998	82.86	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
999	82.71	oe	ccsbBroad304_03164	MTERFD1	-			
1000	82.68	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
1001	82.63	oe	ccsbBroad304_00060	AMBP	Lipocalins			
1002	82.6	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
1003	82.57	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
1004	82.53	kd	CGS001-5992	RFX4	-			
1005	82.49	kd	CGS001-25793	FBXO7	F-boxes / other			
1006	82.38	oe	ccsbBroad304_01215	PLAUR	CD molecules			
1007	82.37	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
1008	82.36	oe	ccsbBroad304_00034	AES	-			
1009	82.35	kd	CGS001-9847	KIAA0528	-			
1010	82.35	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
1011	82.34	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
1012	82.33	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
1013	82.31	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
1014	82.18	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
1015	82.13	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
1016	82.05	kd	CGS001-253260	RICTOR	-			
1017	82.04	kd	CGS001-64094	SMOC2	EF-hand domain containing			
1018	82.03	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
1019	82.02	kd	CGS001-51070	NOSIP	-			
1020	82	kd	CGS001-10465	PPIH	-			
1021	81.98	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
1022	81.98	kd	CGS001-79581	GPR172A	-			
1023	81.96	kd	CGS001-4122	MAN2A2	-			
1024	81.94	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
1025	81.9	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1026	81.87	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
1027	81.77	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
1028	81.77	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
1029	81.69	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1030	81.67	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
1031	81.65	oe	ccsbBroad304_02249	KIAA0494	-			
1032	81.63	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
1033	81.62	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1034	81.58	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
1035	81.58	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
1036	81.42	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
1037	81.39	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
1038	81.35	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1039	81.33	kd	CGS001-60528	ELAC2	-			
1040	81.31	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
1041	81.29	kd	CGS001-10400	PEMT	-			
1042	81.24	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
1043	81.24	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
1044	81.24	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
1045	81.22	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
1046	81.2	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
1047	81.2	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
1048	81.12	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
1049	81.12	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
1050	81	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
1051	80.99	kd	CGS001-7187	TRAF3	-			
1052	80.92	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
1053	80.9	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
1054	80.85	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
1055	80.77	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
1056	80.76	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
1057	80.74	kd	CGS001-4190	MDH1	-			
1058	80.7	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
1059	80.64	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
1060	80.62	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
1061	80.56	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
1062	80.54	oe	ccsbBroad304_00462	DR1	-			
1063	80.52	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1064	80.51	oe	ccsbBroad304_00650	GNA11	-			
1065	80.47	oe	ccsbBroad304_07834	GGA2	-			
1066	80.45	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
1067	80.42	kd	CGS001-644	BLVRA	-			
1068	80.38	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
1069	80.35	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
1070	80.35	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
1071	80.33	oe	ccsbBroad304_02110	VAPB	-			
1072	80.31	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
1073	80.26	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
1074	80.24	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1075	80.19	cc		ATP synthase inhibitor	-			
1076	80.18	cc		PKC inhibitor	-			
1077	80.11	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
1078	80.08	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
1079	80.06	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
1080	80.03	oe	ccsbBroad304_05763	ACTB	-			
1081	80.02	cc		SRC inhibitor	-			
1082	79.99	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
1083	79.87	kd	CGS001-26277	TINF2	-			
1084	79.82	cc		Mediator complex LOF	-			
1085	79.8	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
1086	79.79	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
1087	79.77	cc		NFKB Activation GOF	-			
1088	79.75	oe	ccsbBroad304_01661	TFCP2	-			
1089	79.71	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
1090	79.7	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
1091	79.68	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
1092	79.65	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
1093	79.63	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
1094	79.59	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
1095	79.57	oe	ccsbBroad304_07018	SUPT5H	-			
1096	79.54	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
1097	79.54	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
1098	79.54	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
1099	79.47	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
1100	79.45	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
1101	79.45	kd	CGS001-10190	TXNDC9	-			
1102	79.4	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
1103	79.39	kd	CGS001-3560	IL2RB	IL-2 receptor family			
1104	79.34	kd	CGS001-3131	HLF	-			
1105	79.29	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
1106	79.27	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1107	79.26	kd	CGS001-523	ATP6V1A	ATPases / V-type			
1108	79.23	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
1109	79.18	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1110	79.16	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
1111	79.08	kd	CGS001-578	BAK1	-			
1112	79.07	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
1113	79.06	kd	CGS001-10096	ACTR3	-			
1114	79.04	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
1115	78.95	kd	CGS001-9788	MTSS1	-			
1116	78.91	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
1117	78.88	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
1118	78.84	oe	ccsbBroad304_04786	CANT1	-			
1119	78.65	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
1120	78.65	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
1121	78.59	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
1122	78.47	oe	ccsbBroad304_01373	RAN	-			
1123	78.44	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
1124	78.42	oe	ccsbBroad304_05758	ACADSB	-			
1125	78.36	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
1126	78.36	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
1127	78.3	oe	ccsbBroad304_10431	HADHB	-			
1128	78.14	kd	CGS001-57721	METTL14	-			
1129	78.1	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
1130	78.1	kd	CGS001-6757	SSX2	-			
1131	78.03	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
1132	78.02	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
1133	78.02	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
1134	77.97	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
1135	77.92	oe	ccsbBroad304_02287	GNPDA1	-			
1136	77.92	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
1137	77.78	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
1138	77.75	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
1139	77.72	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
1140	77.69	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
1141	77.67	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
1142	77.65	kd	CGS001-801	CALM1	EF-hand domain containing			
1143	77.63	kd	CGS001-4616	GADD45B	-			
1144	77.6	kd	CGS001-23670	TMEM2	-			
1145	77.53	kd	CGS001-10513	APPBP2	-			
1146	77.5	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
1147	77.5	kd	CGS001-6050	RNH1	-			
1148	77.45	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
1149	77.44	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
1150	77.43	oe	ccsbBroad304_06523	LIG1	-			
1151	77.38	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
1152	77.38	kd	CGS001-4194	MDM4	-			
1153	77.34	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1154	77.31	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
1155	77.31	kd	CGS001-435	ASL	-			
1156	77.24	oe	ccsbBroad304_00072	ANXA7	Annexins			
1157	77.24	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
1158	77.13	kd	CGS001-4121	MAN1A1	-			
1159	77.13	kd	CGS001-3689	ITGB2	Integrins			
1160	77.11	cc		JAK inhibitor	-			
1161	77.03	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
1162	77.02	kd	CGS001-571	BACH1	BTB/POZ domain containing			
1163	77.01	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
1164	76.93	oe	ccsbBroad304_06852	RBP4	Lipocalins			
1165	76.73	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
1166	76.71	oe	ccsbBroad304_03450	TMED9	-			
1167	76.63	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
1168	76.62	oe	ccsbBroad304_06237	GAA	Glycosidases			
1169	76.62	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
1170	76.54	oe	ccsbBroad304_00783	HPRT1	-			
1171	76.51	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
1172	76.5	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
1173	76.49	kd	CGS001-54957	TXNL4B	-			
1174	76.42	oe	ccsbBroad304_06349	HAGH	-			
1175	76.37	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
1176	76.29	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
1177	76.29	kd	CGS001-91433	RCCD1	-			
1178	76.24	kd	CGS001-5428	POLG	DNA polymerases			
1179	76.23	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
1180	76.21	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
1181	76.17	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
1182	76.13	kd	CGS001-9541	CIR1	-			
1183	76.12	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
1184	76.09	kd	CGS001-10475	TRIM38	-			
1185	76.08	kd	CGS001-26993	AKAP8L	-			
1186	76.06	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
1187	76.05	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
1188	76.05	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
1189	76.03	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
1190	75.96	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
1191	75.92	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
1192	75.91	kd	CGS001-6185	RPN2	-			
1193	75.8	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
1194	75.78	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
1195	75.67	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
1196	75.65	kd	CGS001-4700	NDUFA6	LYR motif containing			
1197	75.64	oe	ccsbBroad304_06282	GLDC	-			
1198	75.63	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
1199	75.58	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
1200	75.56	oe	ccsbBroad304_01061	NAB2	-			
1201	75.54	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
1202	75.53	kd	CGS001-5018	OXA1L	-			
1203	75.51	kd	CGS001-7919	DDX39B	DEAD-boxes			
1204	75.5	oe	ccsbBroad304_02229	TRAM2	-			
1205	75.48	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
1206	75.47	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
1207	75.43	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
1208	75.42	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1209	75.41	kd	CGS001-340371	NRBP2	NRBP family			
1210	75.37	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
1211	75.34	oe	ccsbBroad304_00370	CS	-			
1212	75.3	oe	ccsbBroad304_02298	DNM1L	-			
1213	75.29	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
1214	75.23	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
1215	75.23	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
1216	75.19	kd	CGS001-388650	FAM69A	-			
1217	75.18	kd	CGS001-5579	PRKCB	Alpha subfamily			
1218	75.11	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1219	75.07	oe	ccsbBroad304_01576	SOAT1	-			
1220	75.04	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1221	74.89	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
1222	74.89	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
1223	74.83	oe	ccsbBroad304_06975	SMARCC2	-			
1224	74.83	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
1225	74.78	kd	CGS001-79109	MAPKAP1	-			
1226	74.73	kd	CGS001-57057	TBX20	T-boxes			
1227	74.68	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
1228	74.66	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
1229	74.56	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
1230	74.49	oe	ccsbBroad304_06670	OGG1	-			
1231	74.36	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
1232	74.3	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
1233	74.22	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
1234	74.19	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
1235	74.15	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
1236	74.14	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
1237	74.12	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
1238	74	kd	CGS001-2768	GNA12	-			
1239	73.99	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
1240	73.95	kd	CGS001-3659	IRF1	-			
1241	73.94	oe	ccsbBroad304_00237	CCND3	-			
1242	73.9	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
1243	73.9	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
1244	73.89	oe	ccsbBroad304_06718	PFN2	-			
1245	73.81	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
1246	73.81	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
1247	73.78	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
1248	73.68	kd	CGS001-51071	DERA	-			
1249	73.66	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
1250	73.66	kd	CGS001-4255	MGMT	-			
1251	73.65	oe	ccsbBroad304_02857	BAMBI	-			
1252	73.6	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
1253	73.56	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
1254	73.52	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
1255	73.49	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1256	73.48	oe	ccsbBroad304_01271	PPT1	-			
1257	73.43	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
1258	73.42	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
1259	73.24	kd	CGS001-3176	HNMT	-			
1260	73.23	cp	BRD-A71009679	KUC103420N	-666			-666
1261	73.22	oe	ccsbBroad304_00515	ERH	-			
1262	73.19	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
1263	73.19	oe	ccsbBroad304_03652	EXOC2	-			
1264	73.12	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
1265	73.1	kd	CGS001-1495	CTNNA1	Catenins			
1266	73.08	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
1267	73.08	oe	ccsbBroad304_07326	EIF2B2	-			
1268	73.06	kd	CGS001-4605	MYBL2	-			
1269	73.03	oe	ccsbBroad304_02157	MED21	-			
1270	73.01	oe	ccsbBroad304_00728	HBE1	-			
1271	72.99	kd	CGS001-351	APP	Endogenous ligands			
1272	72.92	kd	CGS001-253430	IPMK	-			
1273	72.91	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
1274	72.85	oe	ccsbBroad304_01054	GADD45B	-			
1275	72.77	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
1276	72.69	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1277	72.67	oe	ccsbBroad304_03506	AURKAIP1	-			
1278	72.66	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
1279	72.65	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
1280	72.65	kd	CGS001-1211	CLTA	-			
1281	72.61	kd	CGS001-818	CAMK2G	CAMK2 family			
1282	72.6	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
1283	72.58	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
1284	72.5	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
1285	72.44	kd	CGS001-53340	SPA17	-			
1286	72.43	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
1287	72.37	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
1288	72.33	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
1289	72.32	kd	CGS001-7248	TSC1	-			
1290	72.28	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
1291	72.25	kd	CGS001-8829	NRP1	CD molecules			
1292	72.2	oe	ccsbBroad304_02589	COPS5	-			
1293	72.2	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
1294	72.12	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
1295	72.12	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
1296	72.11	kd	CGS001-6647	SOD1	-			
1297	72.03	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
1298	72	oe	ccsbBroad304_08536	PARL	-			
1299	71.99	oe	ccsbBroad304_01008	KITLG	-			
1300	71.96	oe	ccsbBroad304_04038	ELOVL6	-			
1301	71.96	kd	CGS001-6461	SHB	SH2 domain containing			
1302	71.95	oe	ccsbBroad304_07890	CBX7	-			
1303	71.88	kd	CGS001-9170	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1304	71.85	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1305	71.83	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
1306	71.76	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
1307	71.76	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
1308	71.74	kd	CGS001-64943	NT5DC2	-			
1309	71.64	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1310	71.64	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
1311	71.6	oe	ccsbBroad304_02220	MTFR1	-			
1312	71.57	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1313	71.53	oe	ccsbBroad304_06291	GNAI1	-			
1314	71.53	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
1315	71.47	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
1316	71.45	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
1317	71.44	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
1318	71.41	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
1319	71.32	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
1320	71.3	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
1321	71.29	cc		Vesicular Transport LOF	-			
1322	71.18	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
1323	71.12	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
1324	71.11	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
1325	71.1	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
1326	71.04	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
1327	70.88	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
1328	70.83	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
1329	70.82	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
1330	70.77	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
1331	70.73	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
1332	70.72	oe	ccsbBroad304_06538	LSP1	-			
1333	70.71	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
1334	70.66	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
1335	70.62	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
1336	70.62	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
1337	70.59	oe	ccsbBroad304_08684	CXCR7	-			
1338	70.54	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
1339	70.53	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1340	70.5	oe	ccsbBroad304_01872	DGCR14	-			
1341	70.49	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
1342	70.39	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1343	70.36	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
1344	70.36	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
1345	70.27	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
1346	70.25	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
1347	70.2	oe	ccsbBroad304_07478	CCP110	-			
1348	70.19	kd	CGS001-955	ENTPD6	-			
1349	70.12	kd	CGS001-10018	BCL2L11	-			
1350	70.1	kd	CGS001-25913	POT1	-			
1351	70.04	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
1352	70	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
1353	69.98	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
1354	69.91	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
1355	69.9	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
1356	69.83	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
1357	69.81	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
1358	69.81	kd	CGS001-10493	VAT1	-			
1359	69.72	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
1360	69.67	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
1361	69.65	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
1362	69.64	kd	CGS001-10969	EBNA1BP2	-			
1363	69.59	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
1364	69.54	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
1365	69.49	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
1366	69.39	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
1367	69.37	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
1368	69.32	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
1369	69.27	oe	ccsbBroad304_00492	EIF5A	-			
1370	69.25	kd	CGS001-7849	PAX8	Paired boxes			
1371	69.17	oe	ccsbBroad304_02002	RNMT	-			
1372	69.17	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
1373	69.12	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
1374	68.97	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
1375	68.94	cc		Tumor necrosis factor superfamily LOF	-			
1376	68.94	kd	CGS001-3927	LASP1	-			
1377	68.9	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
1378	68.88	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
1379	68.84	oe	ccsbBroad304_01002	METTL1	-			
1380	68.84	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
1381	68.83	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
1382	68.82	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
1383	68.79	oe	ccsbBroad304_01618	STXBP1	-			
1384	68.75	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
1385	68.74	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
1386	68.72	cc		Supressors of cytokine signaling GOF	-			
1387	68.71	kd	CGS001-4734	NEDD4	-			
1388	68.68	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
1389	68.67	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
1390	68.66	kd	CGS001-4144	MAT2A	-			
1391	68.64	oe	ccsbBroad304_03625	HIF1AN	-			
1392	68.58	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
1393	68.58	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
1394	68.56	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
1395	68.53	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
1396	68.49	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
1397	68.47	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
1398	68.46	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
1399	68.35	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
1400	68.34	kd	CGS001-6387	CXCL12	Endogenous ligands			
1401	68.32	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
1402	68.29	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
1403	68.29	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
1404	68.2	kd	CGS001-56889	TM9SF3	-			
1405	68.16	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
1406	68.15	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
1407	68.1	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
1408	68.06	cc		MDM inhibitor	-			
1409	68	kd	CGS001-51097	SCCPDH	-			
1410	67.95	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
1411	67.92	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
1412	67.86	kd	CGS001-2931	GSK3A	GSK subfamily			
1413	67.84	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
1414	67.78	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
1415	67.73	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
1416	67.66	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
1417	67.65	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
1418	67.63	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
1419	67.56	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
1420	67.55	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
1421	67.52	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1422	67.51	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
1423	67.46	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
1424	67.43	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
1425	67.38	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
1426	67.34	oe	ccsbBroad304_00036	AFP	-			
1427	67.34	kd	CGS001-3418	IDH2	-			
1428	67.26	kd	CGS001-4088	SMAD3	SMADs			
1429	67.23	oe	ccsbBroad304_02862	CCRN4L	-			
1430	67.21	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
1431	67.2	oe	ccsbBroad304_00150	BAX	-			
1432	67.19	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
1433	67.19	kd	CGS001-23212	RRS1	-			
1434	67.18	cc		RAF inhibitor	-			
1435	67.16	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
1436	67.16	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
1437	67.14	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
1438	67.13	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
1439	67.12	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
1440	67.12	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
1441	67.04	kd	CGS001-255738	PCSK9	Subtilisin			
1442	67.02	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
1443	67.01	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
1444	66.98	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
1445	66.94	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
1446	66.93	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
1447	66.9	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
1448	66.86	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
1449	66.86	oe	ccsbBroad304_00626	GDI1	-			
1450	66.82	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1451	66.69	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
1452	66.68	cc		VEGFR inhibitor	-			
1453	66.65	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
1454	66.62	kd	CGS001-6723	SRM	-			
1455	66.6	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
1456	66.44	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1457	66.41	oe	ccsbBroad304_01933	TEAD2	-			
1458	66.34	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
1459	66.31	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1460	66.24	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
1461	66.2	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
1462	66.19	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
1463	66.07	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1464	66.04	oe	ccsbBroad304_12226	NAGK	-			
1465	66.02	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
1466	66.01	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
1467	65.97	kd	CGS001-26298	EHF	-			
1468	65.94	oe	ccsbBroad304_02026	NRP1	CD molecules			
1469	65.94	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1470	65.89	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
1471	65.89	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
1472	65.85	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
1473	65.82	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
1474	65.72	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
1475	65.67	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
1476	65.64	oe	ccsbBroad304_07616	ZNF238	-			
1477	65.62	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
1478	65.61	oe	ccsbBroad304_01035	MSH5	-			
1479	65.58	kd	CGS001-5223	PGAM1	-			
1480	65.58	kd	CGS001-2896	GRN	-			
1481	65.53	oe	ccsbBroad304_07662	NPRL2	-			
1482	65.51	cc		FLT3 inhibitor	-			
1483	65.51	kd	CGS001-1643	DDB2	WD repeat domain containing			
1484	65.48	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
1485	65.48	kd	CGS001-2067	ERCC1	-			
1486	65.45	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
1487	65.42	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
1488	65.4	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
1489	65.37	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
1490	65.36	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
1491	65.34	kd	CGS001-5050	PAFAH1B3	-			
1492	65.33	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
1493	65.3	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
1494	65.29	oe	ccsbBroad304_02890	SYF2	-			
1495	65.28	kd	CGS001-22889	KIAA0907	-			
1496	65.27	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
1497	65.23	oe	ccsbBroad304_00710	GUSB	-			
1498	65.19	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
1499	65.15	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
1500	65.13	kd	CGS001-7353	UFD1L	-			
1501	65.05	kd	CGS001-57787	MARK4	MARK subfamily			
1502	65.03	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
1503	65.01	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
1504	64.96	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
1505	64.89	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
1506	64.88	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
1507	64.87	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
1508	64.86	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
1509	64.83	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
1510	64.73	kd	CGS001-8974	P4HA2	-			
1511	64.72	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
1512	64.7	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1513	64.7	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
1514	64.69	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
1515	64.63	oe	ccsbBroad304_05098	MAGEB6	-			
1516	64.54	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
1517	64.51	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
1518	64.49	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
1519	64.47	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
1520	64.46	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
1521	64.4	kd	CGS001-10253	SPRY2	-			
1522	64.38	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
1523	64.35	kd	CGS001-23077	MYCBP2	-			
1524	64.35	kd	CGS001-30	ACAA1	-			
1525	64.3	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
1526	64.3	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
1527	64.22	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
1528	64.22	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
1529	64.2	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
1530	64.18	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
1531	64.15	kd	CGS001-7157	TP53	-			
1532	64.08	kd	CGS001-4522	MTHFD1	-			
1533	63.96	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
1534	63.96	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
1535	63.95	oe	ccsbBroad304_13998	PDXK	-			
1536	63.95	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
1537	63.94	oe	ccsbBroad304_07704	SUB1	-			
1538	63.94	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
1539	63.91	kd	CGS001-4221	MEN1	-			
1540	63.88	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
1541	63.84	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
1542	63.84	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1543	63.83	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
1544	63.82	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
1545	63.8	kd	CGS001-8802	SUCLG1	-			
1546	63.77	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
1547	63.77	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
1548	63.75	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
1549	63.68	oe	ccsbBroad304_01560	SNAPC1	-			
1550	63.58	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
1551	63.48	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
1552	63.48	kd	CGS001-7097	TLR2	Toll-like receptor family			
1553	63.47	kd	CGS001-27034	ACAD8	-			
1554	63.29	kd	CGS001-84890	ADO	-			
1555	63.27	oe	ccsbBroad304_02592	KIF2C	Kinesins			
1556	63.27	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
1557	63.15	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
1558	63.14	oe	ccsbBroad304_06642	NIT1	-			
1559	63.14	kd	CGS001-64343	AZI2	-			
1560	63.08	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
1561	63.08	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
1562	63.04	oe	ccsbBroad304_07766	RASSF1	-			
1563	63.04	kd	CGS001-6256	RXRA	Retinoid X receptors			
1564	63.01	kd	CGS001-367	AR	Nuclear hormone receptors			
1565	62.99	cc		GATA Zinc finger domain containing LOF	-			
1566	62.99	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
1567	62.99	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1568	62.87	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
1569	62.87	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
1570	62.86	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
1571	62.85	oe	ccsbBroad304_06820	PTS	-			
1572	62.79	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
1573	62.77	kd	CGS001-9500	MAGED1	-			
1574	62.76	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
1575	62.75	oe	ccsbBroad304_02843	FTSJ1	-			
1576	62.72	kd	CGS001-111	ADCY5	Adenylate cyclases			
1577	62.71	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
1578	62.67	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
1579	62.66	kd	CGS001-306	ANXA3	Annexins			
1580	62.63	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
1581	62.63	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
1582	62.63	kd	CGS001-58528	RRAGD	-			
1583	62.57	oe	ccsbBroad304_07808	RAB11FIP2	-			
1584	62.54	kd	CGS001-823	CAPN1	EF-hand domain containing			
1585	62.47	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
1586	62.41	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
1587	62.4	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
1588	62.39	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
1589	62.28	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
1590	62.25	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
1591	62.23	oe	ccsbBroad304_02884	POT1	-			
1592	62.23	kd	CGS001-1676	DFFA	-			
1593	62.21	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
1594	62.18	kd	CGS001-3066	HDAC2	Histone deacetylases			
1595	62.13	oe	ccsbBroad304_01164	PDHB	-			
1596	62.1	kd	CGS001-328	APEX1	-			
1597	62.09	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
1598	62.08	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
1599	62.08	kd	CGS001-84617	TUBB6	Tubulins			
1600	62.07	oe	ccsbBroad304_03191	NOSIP	-			
1601	62.07	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
1602	62.04	cc		Lysine acetyltransferases LOF	-			
1603	62	kd	CGS001-3660	IRF2	-			
1604	61.99	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
1605	61.94	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
1606	61.92	oe	ccsbBroad304_02115	PTTG1	-			
1607	61.92	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
1608	61.91	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1609	61.91	kd	CGS001-10007	GNPDA1	-			
1610	61.85	kd	CGS001-216	ALDH1A1	Aldehyde dehydrogenases			
1611	61.84	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
1612	61.82	cc		Aromatase inhibitor	-			
1613	61.8	oe	ccsbBroad304_04404	TUBB6	Tubulins			
1614	61.79	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
1615	61.78	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
1616	61.76	oe	ccsbBroad304_07320	SQSTM1	-			
1617	61.69	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
1618	61.64	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
1619	61.55	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
1620	61.48	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
1621	61.46	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
1622	61.45	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1623	61.44	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
1624	61.39	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
1625	61.26	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
1626	61.26	kd	CGS001-10914	PAPOLA	-			
1627	61.22	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
1628	61.21	oe	ccsbBroad304_00957	M6PR	-			
1629	61.18	kd	CGS001-53632	PRKAG3	AMPK subfamily			
1630	61.15	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
1631	61.11	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1632	61.01	oe	ccsbBroad304_08452	PIH1D1	-			
1633	61.01	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
1634	60.99	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
1635	60.98	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
1636	60.96	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
1637	60.91	kd	CGS001-5891	MOK	RCK family			
1638	60.81	oe	ccsbBroad304_03047	BZW2	-			
1639	60.8	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
1640	60.76	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
1641	60.76	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
1642	60.73	oe	ccsbBroad304_00658	GNG5	-			
1643	60.71	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
1644	60.69	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
1645	60.65	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
1646	60.57	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
1647	60.54	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
1648	60.53	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
1649	60.48	oe	ccsbBroad304_03237	LEF1	-			
1650	60.48	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
1651	60.45	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
1652	60.42	kd	CGS001-624	BDKRB2	Bradykinin receptors			
1653	60.4	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
1654	60.31	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
1655	60.3	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
1656	60.3	kd	CGS001-26511	CHIC2	-			
1657	60.27	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
1658	60.27	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
1659	60.26	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
1660	60.25	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
1661	60.24	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
1662	60.23	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1663	60.22	oe	ccsbBroad304_03266	ERGIC2	-			
1664	60.2	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1665	60.16	kd	CGS001-64080	RBKS	-			
1666	60.11	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1667	60.1	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
1668	60.06	kd	CGS001-64223	MLST8	WD repeat domain containing			
1669	60.04	kd	CGS001-4172	MCM3	-			
1670	60	cc		Bacterial 30S ribosomal subunit inhibitor	-			
1671	59.97	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
1672	59.91	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
1673	59.9	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
1674	59.85	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
1675	59.83	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
1676	59.82	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
1677	59.81	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
1678	59.79	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
1679	59.76	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
1680	59.71	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
1681	59.7	cc		Akt Signaling LOF	-			
1682	59.63	oe	ccsbBroad304_01673	TIMP3	-			
1683	59.62	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
1684	59.59	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
1685	59.56	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
1686	59.56	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
1687	59.49	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
1688	59.48	oe	ccsbBroad304_01091	NFIB	-			
1689	59.43	kd	CGS001-3248	HPGD	Prostaglandin synthases			
1690	59.36	kd	CGS001-65243	ZNF643	-			
1691	59.32	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
1692	59.27	kd	CGS001-2639	GCDH	-			
1693	59.24	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
1694	59.22	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
1695	59.21	kd	CGS001-661	POLR3D	RNA polymerase subunits			
1696	59.11	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
1697	59.02	oe	ccsbBroad304_06462	ITGAE	Integrins			
1698	59	oe	ccsbBroad304_05590	NOTCH2NL	-			
1699	59	kd	CGS001-80274	SCUBE1	-			
1700	58.93	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
1701	58.88	cc		Lipocalins GOF	-			
1702	58.88	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
1703	58.79	cc		PDGFR/KIT inhibitor	-			
1704	58.76	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
1705	58.73	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
1706	58.71	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
1707	58.71	kd	CGS001-3098	HK1	-			
1708	58.69	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
1709	58.64	kd	CGS001-10078	TSSC4	-			
1710	58.62	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
1711	58.59	kd	CGS001-8220	DGCR14	-			
1712	58.56	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
1713	58.52	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
1714	58.46	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
1715	58.43	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
1716	58.4	kd	CGS001-8453	CUL2	-			
1717	58.38	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
1718	58.33	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
1719	58.33	kd	CGS001-6520	SLC3A2	SLC3 family			
1720	58.32	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
1721	58.32	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
1722	58.32	kd	CGS001-11151	CORO1A	Coronins			
1723	58.31	kd	CGS001-4836	NMT1	-			
1724	58.18	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
1725	58.16	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
1726	58.16	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
1727	58.08	oe	ccsbBroad304_04387	MKI67IP	-			
1728	58.08	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
1729	58.06	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
1730	58	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
1731	57.99	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
1732	57.99	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
1733	57.9	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
1734	57.89	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
1735	57.89	kd	CGS001-55179	FAIM	-			
1736	57.84	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
1737	57.82	kd	CGS001-51290	ERGIC2	-			
1738	57.82	kd	CGS001-55837	EAPP	-			
1739	57.8	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
1740	57.79	kd	CGS001-1384	CRAT	-			
1741	57.76	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
1742	57.76	kd	CGS001-51380	CSAD	-			
1743	57.75	oe	ccsbBroad304_06264	GBP2	-			
1744	57.7	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
1745	57.69	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1746	57.68	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
1747	57.65	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
1748	57.6	kd	CGS001-7374	UNG	-			
1749	57.58	kd	CGS001-7099	TLR4	Toll-like receptor family			
1750	57.57	kd	CGS001-1655	DDX5	DEAD-boxes			
1751	57.54	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
1752	57.5	kd	CGS001-5167	ENPP1	-			
1753	57.48	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1754	57.46	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
1755	57.4	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
1756	57.4	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
1757	57.35	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
1758	57.32	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
1759	57.3	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
1760	57.22	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
1761	57.19	kd	CGS001-1949	EFNB3	Ephrins			
1762	57.16	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
1763	57.14	kd	CGS001-182	JAG1	CD molecules			
1764	57.12	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
1765	57.06	oe	ccsbBroad304_06292	GNAI2	-			
1766	57.06	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1767	56.97	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1768	56.94	kd	CGS001-3035	HARS	Aminoacyl tRNA synthetases / Class II			
1769	56.93	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
1770	56.89	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
1771	56.88	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
1772	56.88	kd	CGS001-116519	APOA5	Apolipoproteins			
1773	56.87	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
1774	56.87	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
1775	56.87	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
1776	56.87	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
1777	56.85	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
1778	56.82	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
1779	56.77	oe	ccsbBroad304_04775	NTAN1	-			
1780	56.75	oe	ccsbBroad304_06301	GOT2	-			
1781	56.74	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
1782	56.71	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
1783	56.64	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
1784	56.59	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
1785	56.55	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
1786	56.53	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
1787	56.42	oe	ccsbBroad304_02163	MED7	-			
1788	56.41	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
1789	56.41	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
1790	56.38	kd	CGS001-5373	PMM2	-			
1791	56.24	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1792	56.22	cc		Toll like receptors LOF	-			
1793	56.22	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
1794	56.17	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
1795	56.15	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
1796	56.15	kd	CGS001-1465	CSRP1	-			
1797	56.11	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
1798	56.09	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
1799	56.02	kd	CGS001-1119	CHKA	-			
1800	55.99	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
1801	55.99	kd	CGS001-944	TNFSF8	CD molecules			
1802	55.98	kd	CGS001-9276	COPB2	WD repeat domain containing			
1803	55.96	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
1804	55.87	oe	ccsbBroad304_07569	TRIB1	Trbl family			
1805	55.87	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
1806	55.86	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
1807	55.83	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
1808	55.79	kd	CGS001-80135	RPF1	-			
1809	55.72	kd	CGS001-2771	GNAI2	-			
1810	55.68	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
1811	55.67	cc		Sigma receptor antagonist	-			
1812	55.65	cc		Adenosine receptor agonist	-			
1813	55.61	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
1814	55.58	kd	CGS001-663	BNIP2	-			
1815	55.55	kd	CGS001-55604	LRRC16A	-			
1816	55.49	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1817	55.47	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
1818	55.42	oe	ccsbBroad304_07411	LPXN	-			
1819	55.4	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
1820	55.39	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
1821	55.37	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
1822	55.2	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
1823	55.19	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
1824	55.16	oe	ccsbBroad304_03604	ENOSF1	-			
1825	55.12	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
1826	55.08	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
1827	55.08	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
1828	55.03	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
1829	55	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
1830	54.97	kd	CGS001-4665	NAB2	-			
1831	54.87	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
1832	54.86	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
1833	54.85	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
1834	54.85	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
1835	54.83	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
1836	54.79	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
1837	54.79	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
1838	54.78	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
1839	54.77	kd	CGS001-5898	RALA	-			
1840	54.76	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
1841	54.75	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
1842	54.75	kd	CGS001-10325	RRAGB	-			
1843	54.74	cc		BCL inhibitor	-			
1844	54.69	kd	CGS001-64750	SMURF2	-			
1845	54.66	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
1846	54.65	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
1847	54.65	kd	CGS001-169841	ZNF169	Zinc fingers, C2H2-type			
1848	54.57	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
1849	54.54	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1850	54.45	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
1851	54.41	kd	CGS001-57222	ERGIC1	-			
1852	54.4	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
1853	54.38	kd	CGS001-2731	GLDC	-			
1854	54.37	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
1855	54.35	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
1856	54.32	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
1857	54.27	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
1858	54.26	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
1859	54.24	kd	CGS001-10174	SORBS3	-			
1860	54.2	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
1861	54.16	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
1862	54.16	kd	CGS001-64077	LHPP	-			
1863	54.13	kd	CGS001-161725	OTUD7A	OTU domain containing			
1864	54.11	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
1865	54.05	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
1866	53.97	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
1867	53.96	kd	CGS001-79094	CHAC1	-			
1868	53.95	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1869	53.91	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
1870	53.9	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
1871	53.82	oe	ccsbBroad304_00101	RHOC	-			
1872	53.77	kd	CGS001-308	ANXA5	Annexins			
1873	53.71	oe	ccsbBroad304_02964	TIMM9	-			
1874	53.71	oe	ccsbBroad304_04788	OVCA2	-			
1875	53.66	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
1876	53.63	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
1877	53.57	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
1878	53.56	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
1879	53.53	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
1880	53.53	kd	CGS001-8914	TIMELESS	-			
1881	53.51	kd	CGS001-59343	SENP2	-			
1882	53.5	oe	ccsbBroad304_12008	NLK	nmo subfamily			
1883	53.41	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
1884	53.38	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
1885	53.37	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
1886	53.36	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
1887	53.35	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
1888	53.35	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
1889	53.3	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
1890	53.3	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1891	53.27	kd	CGS001-4282	MIF	-			
1892	53.26	kd	CGS001-2295	FOXF2	Forkhead boxes			
1893	53.25	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
1894	53.24	oe	ccsbBroad304_09035	COASY	-			
1895	53.21	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1896	53.17	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
1897	53.06	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
1898	53.06	kd	CGS001-5366	PMAIP1	-			
1899	53.06	kd	CGS001-64863	METTL4	-			
1900	53.03	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
1901	52.95	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
1902	52.94	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
1903	52.92	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
1904	52.89	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
1905	52.86	kd	CGS001-27241	BBS9	-			
1906	52.82	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
1907	52.82	kd	CGS001-5743	PTGS2	Cyclooxygenase			
1908	52.78	oe	ccsbBroad304_09708	PNLDC1	-			
1909	52.77	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
1910	52.77	kd	CGS001-399664	MEX3D	Mex-3 homologs			
1911	52.75	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
1912	52.65	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
1913	52.64	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
1914	52.62	kd	CGS001-4016	LOXL1	-			
1915	52.61	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
1916	52.55	kd	CGS001-8639	AOC3	Oxidoreductases			
1917	52.52	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1918	52.51	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
1919	52.51	kd	CGS001-81848	SPRY4	-			
1920	52.49	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
1921	52.47	oe	ccsbBroad304_01105	PNP	-			
1922	52.43	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
1923	52.41	kd	CGS001-8667	EIF3H	-			
1924	52.32	kd	CGS001-4232	MEST	-			
1925	52.25	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
1926	52.25	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1927	52.2	kd	CGS001-5062	PAK2	PAKA subfamily			
1928	52.18	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
1929	52.15	oe	ccsbBroad304_06549	SMAD3	SMADs			
1930	52.12	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
1931	52.12	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
1932	52.02	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1933	52.01	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1934	52	oe	ccsbBroad304_00226	CAV1	-			
1935	51.94	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
1936	51.91	oe	ccsbBroad304_09195	MCM8	-			
1937	51.91	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
1938	51.87	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
1939	51.85	oe	ccsbBroad304_06278	GK	Glycerol kinases			
1940	51.83	oe	ccsbBroad304_07875	SPECC1L	-			
1941	51.79	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
1942	51.71	kd	CGS001-83448	PUS7L	-			
1943	51.7	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
1944	51.66	oe	ccsbBroad304_03544	FAIM	-			
1945	51.6	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1946	51.51	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
1947	51.51	oe	ccsbBroad304_05887	CFB	Complement system			
1948	51.5	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
1949	51.46	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
1950	51.44	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
1951	51.43	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
1952	51.39	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
1953	51.38	cc		Sterol demethylase inhibitor	-			
1954	51.37	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
1955	51.36	kd	CGS001-1892	ECHS1	-			
1956	51.26	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
1957	51.25	oe	ccsbBroad304_02741	PDS5A	-			
1958	51.25	oe	ccsbBroad304_02402	TMEM5	-			
1959	51.21	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
1960	51.19	kd	CGS001-4846	NOS3	Nitric oxide synthases			
1961	51.17	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
1962	51.14	kd	CGS001-3032	HADHB	-			
1963	51.1	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1964	51.04	kd	CGS001-2717	GLA	-			
1965	51.02	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
1966	51.02	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
1967	51.02	kd	CGS001-900	CCNG1	-			
1968	50.94	oe	ccsbBroad304_00221	CASP3	Caspases			
1969	50.94	oe	ccsbBroad304_02367	CALCOCO2	-			
1970	50.94	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
1971	50.86	kd	CGS001-55111	PLEKHJ1	Pleckstrin homology (PH) domain containing			
1972	50.81	kd	CGS001-8864	PER2	-			
1973	50.8	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
1974	50.72	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
1975	50.72	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
1976	50.7	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
1977	50.7	kd	CGS001-8089	YEATS4	-			
1978	50.69	kd	CGS001-23658	LSM5	-			
1979	50.68	kd	CGS001-7083	TK1	-			
1980	50.66	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
1981	50.66	kd	CGS001-8313	AXIN2	-			
1982	50.6	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
1983	50.58	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
1984	50.53	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
1985	50.5	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
1986	50.42	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
1987	50.39	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
1988	50.37	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
1989	50.34	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
1990	50.3	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
1991	50.3	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
1992	50.23	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
1993	50.22	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
1994	50.17	kd	CGS001-8835	SOCS2	SH2 domain containing			
1995	50.13	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
1996	50.06	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
1997	49.95	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
1998	49.87	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
1999	49.84	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
2000	49.83	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
2001	49.73	kd	CGS001-6347	CCL2	Chemokine ligands			
2002	49.72	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
2003	49.52	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
2004	49.5	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
2005	49.5	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
2006	49.49	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
2007	49.49	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
2008	49.4	kd	CGS001-9447	AIM2	-			
2009	49.39	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
2010	49.37	oe	ccsbBroad304_04626	EGLN3	-			
2011	49.36	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
2012	49.36	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
2013	49.3	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
2014	49.29	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
2015	49.29	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
2016	49.27	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
2017	49.27	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
2018	49.26	oe	ccsbBroad304_13939	MOK	RCK family			
2019	49.26	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
2020	49.14	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
2021	49.13	oe	ccsbBroad304_02443	HAX1	-			
2022	49.12	oe	ccsbBroad304_02386	EIF1B	-			
2023	49.1	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
2024	49.07	oe	ccsbBroad304_02496	MTX2	-			
2025	49.06	kd	CGS001-5257	PHKB	-			
2026	49.02	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
2027	48.94	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
2028	48.92	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
2029	48.87	kd	CGS001-481	ATP1B1	ATPases / P-type			
2030	48.84	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
2031	48.83	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
2032	48.77	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
2033	48.77	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
2034	48.74	kd	CGS001-901	CCNG2	-			
2035	48.69	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
2036	48.69	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
2037	48.68	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2038	48.62	kd	CGS001-50813	COPS7A	-			
2039	48.61	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
2040	48.51	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
2041	48.51	kd	CGS001-54821	ERCC6L	-			
2042	48.5	kd	CGS001-5900	RALGDS	-			
2043	48.47	oe	ccsbBroad304_02484	PAICS	-			
2044	48.46	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
2045	48.37	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
2046	48.37	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
2047	48.37	kd	CGS001-8678	BECN1	-			
2048	48.35	kd	CGS001-813	CALU	EF-hand domain containing			
2049	48.32	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
2050	48.32	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
2051	48.17	kd	CGS001-4837	NNMT	-			
2052	48.14	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
2053	48.11	oe	ccsbBroad304_13633	PI4KAP2	-			
2054	48.08	kd	CGS001-10810	WASF3	-			
2055	48.08	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
2056	48.07	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
2057	48.05	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
2058	48.03	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
2059	47.99	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2060	47.99	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
2061	47.89	oe	ccsbBroad304_01101	NME1	-			
2062	47.89	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
2063	47.86	kd	CGS001-22978	NT5C2	Adenosine turnover			
2064	47.76	kd	CGS001-348	APOE	Apolipoproteins			
2065	47.76	oe	ccsbBroad304_08045	NOX1	-			
2066	47.74	kd	CGS001-9124	PDLIM1	-			
2067	47.72	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
2068	47.68	oe	ccsbBroad304_06133	TOR1A	-			
2069	47.64	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
2070	47.63	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
2071	47.62	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
2072	47.61	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
2073	47.6	kd	CGS001-2550	GABBR1	GABA receptors			
2074	47.5	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2075	47.5	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
2076	47.47	oe	ccsbBroad304_06654	NPM1	-			
2077	47.37	kd	CGS001-79600	TCTN1	Tectonic proteins			
2078	47.36	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
2079	47.36	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
2080	47.34	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
2081	47.34	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
2082	47.33	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
2083	47.27	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
2084	47.24	oe	ccsbBroad304_07491	IP6K1	-			
2085	47.22	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
2086	47.21	oe	ccsbBroad304_07217	AXIN2	-			
2087	47.19	kd	CGS001-9474	ATG5	-			
2088	47.17	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
2089	47.1	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
2090	47.09	oe	ccsbBroad304_04294	ATG10	-			
2091	47.06	oe	ccsbBroad304_04619	GNG8	-			
2092	46.99	kd	CGS001-10671	DCTN6	-			
2093	46.98	oe	ccsbBroad304_02956	EHF	-			
2094	46.98	kd	CGS001-2017	CTTN	-			
2095	46.97	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
2096	46.96	oe	ccsbBroad304_02239	RASSF2	-			
2097	46.96	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
2098	46.95	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
2099	46.92	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
2100	46.91	kd	CGS001-51128	SAR1B	-			
2101	46.9	oe	ccsbBroad304_02203	MAD2L1BP	-			
2102	46.86	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
2103	46.81	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
2104	46.7	kd	CGS001-6850	SYK	Syk family			
2105	46.68	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
2106	46.65	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
2107	46.65	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
2108	46.61	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
2109	46.5	oe	ccsbBroad304_01699	TPD52L2	-			
2110	46.5	kd	CGS001-51268	PIPOX	-			
2111	46.47	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
2112	46.46	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
2113	46.45	kd	CGS001-8569	MKNK1	MKN subfamily			
2114	46.44	cc		Vitamin D receptor agonist	-			
2115	46.37	kd	CGS001-11168	PSIP1	-			
2116	46.36	oe	ccsbBroad304_02502	GNA13	-			
2117	46.36	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
2118	46.35	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
2119	46.33	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
2120	46.32	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
2121	46.31	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
2122	46.3	kd	CGS001-84923	FAM104A	-			
2123	46.3	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
2124	46.29	oe	ccsbBroad304_00418	CD55	CD molecules			
2125	46.27	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
2126	46.25	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
2127	46.24	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
2128	46.22	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
2129	46.12	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
2130	46.09	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
2131	46.08	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
2132	46.07	oe	ccsbBroad304_00568	FHL2	-			
2133	46.04	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
2134	46.01	kd	CGS001-1606	DGKA	EF-hand domain containing			
2135	45.9	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
2136	45.89	oe	ccsbBroad304_06711	PFAS	-			
2137	45.88	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
2138	45.86	kd	CGS001-29984	RHOD	-			
2139	45.84	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
2140	45.83	kd	CGS001-80347	COASY	-			
2141	45.82	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
2142	45.8	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
2143	45.72	oe	ccsbBroad304_02058	PLOD3	-			
2144	45.71	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
2145	45.7	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
2146	45.69	kd	CGS001-7728	ZNF175	Zinc fingers, C2H2-type			
2147	45.62	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
2148	45.6	cp	BRD-A02189320	met-leu-phe	-666			-666
2149	45.57	oe	ccsbBroad304_08167	DNTTIP2	-			
2150	45.53	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
2151	45.49	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2152	45.46	oe	ccsbBroad304_00161	BID	Endogenous ligands			
2153	45.46	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
2154	45.45	kd	CGS001-58478	ENOPH1	-			
2155	45.43	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2156	45.41	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
2157	45.36	oe	ccsbBroad304_04153	PHF17	-			
2158	45.33	oe	ccsbBroad304_00725	HADHA	-			
2159	45.32	kd	CGS001-10691	GMEB1	-			
2160	45.28	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
2161	45.24	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
2162	45.22	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
2163	45.19	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
2164	45.14	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
2165	45.11	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
2166	45.1	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
2167	45.1	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
2168	45.09	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
2169	44.97	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
2170	44.95	kd	CGS001-29978	UBQLN2	Ubiquilin family			
2171	44.91	oe	ccsbBroad304_00155	CCND1	-			
2172	44.91	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
2173	44.9	kd	CGS001-2882	GPX7	-			
2174	44.9	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
2175	44.86	oe	ccsbBroad304_02534	UTP14A	-			
2176	44.85	oe	ccsbBroad304_00032	ADSL	-			
2177	44.84	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
2178	44.82	kd	CGS001-10084	PQBP1	-			
2179	44.73	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
2180	44.73	kd	CGS001-8431	NR0B2	DAX-like receptors			
2181	44.7	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
2182	44.7	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
2183	44.66	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
2184	44.65	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
2185	44.61	oe	ccsbBroad304_07531	TANK	-			
2186	44.59	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
2187	44.57	oe	ccsbBroad304_02231	USP6NL	-			
2188	44.57	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
2189	44.54	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
2190	44.51	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
2191	44.51	kd	CGS001-2159	F10	Chymotrypsin			
2192	44.5	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
2193	44.48	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
2194	44.38	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
2195	44.35	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
2196	44.35	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
2197	44.33	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
2198	44.3	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
2199	44.28	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
2200	44.26	oe	ccsbBroad304_00963	SMAD5	SMADs			
2201	44.24	oe	ccsbBroad304_06569	MCM5	-			
2202	44.23	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
2203	44.19	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
2204	44.15	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
2205	44.09	oe	ccsbBroad304_01148	PCBD1	-			
2206	44.05	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
2207	44.02	oe	ccsbBroad304_02416	TUBB4B	-			
2208	43.99	kd	CGS001-18	ABAT	GABA turnover			
2209	43.97	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
2210	43.92	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
2211	43.91	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
2212	43.89	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
2213	43.89	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2214	43.88	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
2215	43.86	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
2216	43.84	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
2217	43.8	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
2218	43.79	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
2219	43.78	kd	CGS001-36	ACADSB	-			
2220	43.76	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
2221	43.75	kd	CGS001-11284	PNKP	-			
2222	43.69	oe	ccsbBroad304_10491	PFKL	-			
2223	43.61	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
2224	43.6	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
2225	43.59	oe	ccsbBroad304_07605	LYPLA1	-			
2226	43.58	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
2227	43.54	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
2228	43.47	kd	CGS001-5538	PPT1	-			
2229	43.38	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
2230	43.37	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
2231	43.36	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
2232	43.32	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
2233	43.27	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
2234	43.24	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
2235	43.23	oe	ccsbBroad304_07094	TPMT	-			
2236	43.23	kd	CGS001-11116	FGFR1OP	-			
2237	43.19	oe	ccsbBroad304_00464	DTNA	-			
2238	43.19	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
2239	43.13	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
2240	43.09	kd	CGS001-3978	LIG1	-			
2241	43.03	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
2242	42.93	kd	CGS001-55379	LRRC59	-			
2243	42.89	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
2244	42.87	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
2245	42.85	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
2246	42.83	kd	CGS001-4303	FOXO4	Forkhead boxes			
2247	42.82	oe	ccsbBroad304_03773	CIAPIN1	-			
2248	42.75	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
2249	42.74	kd	CGS001-1198	CLK3	CDC-like kinases			
2250	42.7	kd	CGS001-23636	NUP62	-			
2251	42.69	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
2252	42.65	cc		DNA synthesis inhibitor	-			
2253	42.62	oe	ccsbBroad304_08511	RFK	-			
2254	42.62	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
2255	42.62	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
2256	42.61	oe	ccsbBroad304_00179	BTG1	-			
2257	42.53	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
2258	42.48	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
2259	42.45	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
2260	42.42	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
2261	42.41	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
2262	42.24	kd	CGS001-9870	KIAA0317	-			
2263	42.21	oe	ccsbBroad304_02572	SERINC3	-			
2264	42.21	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
2265	42.2	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
2266	42.19	oe	ccsbBroad304_06008	AP2M1	-			
2267	42.17	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
2268	42.16	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
2269	42.11	oe	ccsbBroad304_07280	LAMTOR3	-			
2270	42.1	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
2271	42.08	kd	CGS001-7105	TSPAN6	Tetraspanins			
2272	42.07	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
2273	42.07	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
2274	42.05	oe	ccsbBroad304_02501	DCTN6	-			
2275	42.02	kd	CGS001-2963	GTF2F2	General transcription factors			
2276	41.97	cc		Protein phosphatase catalytic subunits LOF	-			
2277	41.88	oe	ccsbBroad304_03112	NENF	-			
2278	41.86	oe	ccsbBroad304_00542	FBP1	-			
2279	41.85	oe	ccsbBroad304_02195	SPAG7	-			
2280	41.79	oe	ccsbBroad304_02604	B3GNT1	-			
2281	41.78	kd	CGS001-2010	EMD	-			
2282	41.76	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
2283	41.72	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
2284	41.69	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
2285	41.69	kd	CGS001-1997	ELF1	ETS Transcription Factors			
2286	41.67	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
2287	41.67	kd	CGS001-6285	S100B	EF-hand domain containing			
2288	41.65	kd	CGS001-5163	PDK1	-			
2289	41.64	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
2290	41.61	kd	CGS001-93594	WDR67	-			
2291	41.59	cc		IMPDH inhibitor	-			
2292	41.53	oe	ccsbBroad304_03874	UBL5	-			
2293	41.52	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
2294	41.48	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
2295	41.44	kd	CGS001-4482	MSRA	-			
2296	41.42	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
2297	41.42	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
2298	41.34	kd	CGS001-6499	SKIV2L	-			
2299	41.33	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
2300	41.33	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
2301	41.33	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
2302	41.32	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
2303	41.3	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
2304	41.28	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
2305	41.26	oe	ccsbBroad304_04064	PRR15L	-			
2306	41.26	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
2307	41.25	kd	CGS001-5883	RAD9A	-			
2308	41.22	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
2309	41.16	oe	ccsbBroad304_01413	RPA2	-			
2310	41.14	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
2311	41.09	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
2312	41.07	cc		PI3K Signaling LOF	-			
2313	41.04	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
2314	41.01	kd	CGS001-5045	FURIN	Subtilisin			
2315	40.99	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
2316	40.99	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
2317	40.93	kd	CGS001-527	ATP6V0C	ATPases / V-type			
2318	40.92	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
2319	40.89	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
2320	40.88	kd	CGS001-11180	WDR6	WD repeat domain containing			
2321	40.87	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
2322	40.75	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
2323	40.73	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
2324	40.71	oe	ccsbBroad304_03767	TOMM22	-			
2325	40.67	kd	CGS001-1512	CTSH	Cathepsins			
2326	40.58	kd	CGS001-23710	GABARAPL1	-			
2327	40.56	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
2328	40.55	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
2329	40.53	oe	ccsbBroad304_03179	BOLA1	-			
2330	40.52	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
2331	40.48	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
2332	40.48	kd	CGS001-55437	STRADB	STLK subfamily			
2333	40.44	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
2334	40.42	oe	ccsbBroad304_00738	HINT1	-			
2335	40.37	oe	ccsbBroad304_00614	GAMT	-			
2336	40.35	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
2337	40.33	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
2338	40.32	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
2339	40.31	kd	CGS001-9797	TATDN2	-			
2340	40.29	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
2341	40.28	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
2342	40.27	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
2343	40.27	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
2344	40.25	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
2345	40.22	kd	CGS001-65123	INTS3	-			
2346	40.2	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
2347	40.2	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
2348	40.14	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
2349	40.14	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
2350	40.11	kd	CGS001-23585	TMEM50A	-			
2351	40.1	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
2352	40.08	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
2353	40.07	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
2354	40.06	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
2355	40.06	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
2356	40.04	kd	CGS001-10645	CAMKK2	Meta subfamily			
2357	39.97	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
2358	39.94	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
2359	39.93	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
2360	39.93	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
2361	39.9	kd	CGS001-6722	SRF	-			
2362	39.88	kd	CGS001-1605	DAG1	-			
2363	39.83	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
2364	39.83	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
2365	39.8	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
2366	39.8	kd	CGS001-23131	GPATCH8	G patch domain containing			
2367	39.77	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
2368	39.7	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
2369	39.68	kd	CGS001-388	RHOB	-			
2370	39.67	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
2371	39.64	oe	ccsbBroad304_00572	FKBP3	-			
2372	39.59	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
2373	39.58	kd	CGS001-701	BUB1B	Bub family			
2374	39.55	oe	ccsbBroad304_00960	SMAD1	SMADs			
2375	39.54	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
2376	39.53	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
2377	39.51	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
2378	39.5	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
2379	39.48	kd	CGS001-593	BCKDHA	-			
2380	39.46	kd	CGS001-2956	MSH6	-			
2381	39.45	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
2382	39.43	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
2383	39.43	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
2384	39.37	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
2385	39.36	oe	ccsbBroad304_01962	STK16	NAK family			
2386	39.35	kd	CGS001-1440	CSF3	Endogenous ligands			
2387	39.34	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
2388	39.31	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
2389	39.28	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
2390	39.24	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
2391	39.23	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
2392	39.16	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
2393	39.14	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2394	39.09	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
2395	39.07	kd	CGS001-2230	FDX1	-			
2396	39.04	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
2397	39.03	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
2398	39	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
2399	38.96	kd	CGS001-4048	LTA4H	Hydrolases			
2400	38.95	oe	ccsbBroad304_02674	STK38	NDR family			
2401	38.94	kd	CGS001-7251	TSG101	-			
2402	38.91	kd	CGS001-23378	RRP8	-			
2403	38.9	kd	CGS001-6732	SRPK1	SRPK family			
2404	38.85	oe	ccsbBroad304_06290	GNA15	-			
2405	38.85	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
2406	38.85	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
2407	38.83	kd	CGS001-6884	TAF13	-			
2408	38.79	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
2409	38.79	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
2410	38.75	oe	ccsbBroad304_00933	LDHB	-			
2411	38.73	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
2412	38.71	oe	ccsbBroad304_04257	SPRY4	-			
2413	38.62	kd	CGS001-7311	UBA52	L ribosomal proteins			
2414	38.58	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
2415	38.55	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
2416	38.55	kd	CGS001-57147	SCYL3	-			
2417	38.52	oe	ccsbBroad304_02759	DICER1	-			
2418	38.44	oe	ccsbBroad304_00954	LYN	Src family			
2419	38.44	oe	ccsbBroad304_01930	CUL2	-			
2420	38.33	oe	ccsbBroad304_13880	IDH3G	-			
2421	38.31	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
2422	38.3	oe	ccsbBroad304_03798	PHTF2	-			
2423	38.28	kd	CGS001-9111	NMI	-			
2424	38.27	kd	CGS001-965	CD58	CD molecules			
2425	38.23	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
2426	38.2	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
2427	38.2	oe	ccsbBroad304_00054	ALDOC	-			
2428	38.16	oe	ccsbBroad304_07140	XPC	-			
2429	38.14	cc		LIM class homeoboxes GOF	-			
2430	38.14	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
2431	38.13	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
2432	38.1	oe	ccsbBroad304_02922	TES	-			
2433	38.1	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
2434	38.06	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
2435	38.04	oe	ccsbBroad304_01150	PCCB	Carboxylases			
2436	38.04	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
2437	38.02	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
2438	37.99	kd	CGS001-55968	NSFL1C	UBX domain containing			
2439	37.99	kd	CGS001-4795	NFKBIL1	-			
2440	37.97	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2441	37.96	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
2442	37.95	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
2443	37.94	oe	ccsbBroad304_01723	TTK	TTK family			
2444	37.93	oe	ccsbBroad304_06318	GPER	-			
2445	37.88	kd	CGS001-2212	FCGR2A	CD molecules			
2446	37.87	kd	CGS001-25942	SIN3A	-			
2447	37.84	kd	CGS001-3669	ISG20	-			
2448	37.84	kd	CGS001-1497	CTNS	-			
2449	37.84	kd	CGS001-56647	BCCIP	-			
2450	37.81	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
2451	37.78	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
2452	37.77	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
2453	37.76	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2454	37.73	oe	ccsbBroad304_09225	BUD13	-			
2455	37.72	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
2456	37.72	kd	CGS001-57026	PDXP	-			
2457	37.71	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
2458	37.71	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
2459	37.71	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
2460	37.7	kd	CGS001-513	ATP5D	ATPases / F-type			
2461	37.66	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
2462	37.66	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2463	37.66	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
2464	37.65	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
2465	37.59	kd	CGS001-8464	SUPT3H	-			
2466	37.57	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
2467	37.57	kd	CGS001-6477	SIAH1	-			
2468	37.51	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
2469	37.5	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
2470	37.49	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
2471	37.45	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
2472	37.45	kd	CGS001-1374	CPT1A	-			
2473	37.44	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
2474	37.43	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
2475	37.42	kd	CGS001-399694	SHC4	SH2 domain containing			
2476	37.37	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
2477	37.36	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
2478	37.34	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
2479	37.32	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
2480	37.28	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
2481	37.23	oe	ccsbBroad304_01624	SUPV3L1	-			
2482	37.22	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2483	37.2	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
2484	37.14	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
2485	37.12	oe	ccsbBroad304_00268	CD81	CD molecules			
2486	37.1	kd	CGS001-2078	ERG	ETS Transcription Factors			
2487	37.09	oe	ccsbBroad304_06435	RBPJ	-			
2488	37.07	kd	CGS001-6443	SGCB	-			
2489	37.05	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
2490	37.05	oe	ccsbBroad304_01841	BAG6	-			
2491	37.04	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
2492	37.01	kd	CGS001-3481	IGF2	-			
2493	36.96	kd	CGS001-55802	DCP1A	-			
2494	36.95	oe	ccsbBroad304_02553	BLCAP	-			
2495	36.94	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
2496	36.93	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
2497	36.9	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
2498	36.86	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
2499	36.82	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
2500	36.81	kd	CGS001-5411	PNN	-			
2501	36.8	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
2502	36.79	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
2503	36.75	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
2504	36.61	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
2505	36.6	kd	CGS001-387	RHOA	-			
2506	36.55	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
2507	36.54	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
2508	36.53	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
2509	36.48	oe	ccsbBroad304_03433	DDIT4	-			
2510	36.46	oe	ccsbBroad304_02012	FADD	-			
2511	36.45	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2512	36.39	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
2513	36.37	oe	ccsbBroad304_07124	UROD	-			
2514	36.35	cp	BRD-K65910366	KUC103904N	-666			-666
2515	36.33	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
2516	36.33	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
2517	36.3	cc		Cell Cycle Inhibition GOF	-			
2518	36.29	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
2519	36.28	kd	CGS001-58472	SQRDL	-			
2520	36.25	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
2521	36.25	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
2522	36.24	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
2523	36.22	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2524	36.21	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2525	36.2	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
2526	36.18	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
2527	36.17	oe	ccsbBroad304_05194	LIPH	-			
2528	36.17	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
2529	36.11	oe	ccsbBroad304_02566	MORF4L1	-			
2530	36.1	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
2531	36.07	kd	CGS001-22794	CASC3	-			
2532	36.05	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
2533	36.03	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
2534	35.94	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
2535	35.91	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
2536	35.86	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
2537	35.84	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
2538	35.81	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
2539	35.8	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
2540	35.78	kd	CGS001-2524	FUT2	Fucosyltransferases			
2541	35.75	oe	ccsbBroad304_03118	NRBP1	NRBP family			
2542	35.74	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
2543	35.71	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
2544	35.71	kd	CGS001-4801	NFYB	-			
2545	35.68	cc		PKC activator	-			
2546	35.68	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
2547	35.67	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
2548	35.67	oe	ccsbBroad304_00471	E2F6	-			
2549	35.66	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
2550	35.65	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
2551	35.58	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
2552	35.57	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
2553	35.52	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
2554	35.51	kd	CGS001-337867	UBAC2	-			
2555	35.5	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
2556	35.5	kd	CGS001-11319	ECD	-			
2557	35.47	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
2558	35.47	kd	CGS001-3664	IRF6	-			
2559	35.43	oe	ccsbBroad304_07557	NAMPT	-			
2560	35.43	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
2561	35.43	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
2562	35.41	kd	CGS001-597	BCL2A1	-			
2563	35.39	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2564	35.38	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
2565	35.31	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
2566	35.29	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
2567	35.25	oe	ccsbBroad304_02500	RRAGA	-			
2568	35.23	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
2569	35.23	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
2570	35.17	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
2571	35.16	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
2572	35.09	oe	ccsbBroad304_10230	STK19	G11 family			
2573	34.96	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
2574	34.92	kd	CGS001-7389	UROD	-			
2575	34.84	oe	ccsbBroad304_00661	GNGT2	-			
2576	34.81	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
2577	34.74	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
2578	34.71	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
2579	34.69	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
2580	34.68	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2581	34.64	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
2582	34.64	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
2583	34.56	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
2584	34.54	kd	CGS001-835	CASP2	Caspases			
2585	34.53	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
2586	34.52	oe	ccsbBroad304_05985	CFL1	-			
2587	34.51	oe	ccsbBroad304_02716	NMNAT2	-			
2588	34.51	oe	ccsbBroad304_02804	KLHDC2	-			
2589	34.49	oe	ccsbBroad304_00147	BAG1	-			
2590	34.49	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
2591	34.48	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
2592	34.47	oe	ccsbBroad304_06350	HAL	-			
2593	34.45	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
2594	34.45	kd	CGS001-1788	DNMT3A	Methyltransferases			
2595	34.43	kd	CGS001-5427	POLE2	DNA polymerases			
2596	34.4	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
2597	34.36	oe	ccsbBroad304_00747	HLF	-			
2598	34.35	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
2599	34.29	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
2600	34.29	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
2601	34.26	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
2602	34.24	oe	ccsbBroad304_00549	FDX1	-			
2603	34.2	kd	CGS001-11164	NUDT5	Nudix motif containing			
2604	34.17	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2605	34.16	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
2606	34.11	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
2607	34.09	kd	CGS001-708	C1QBP	-			
2608	34.01	kd	CGS001-23647	ARFIP2	-			
2609	34	kd	CGS001-10390	CEPT1	-			
2610	33.98	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
2611	33.98	kd	CGS001-54899	PXK	Slob family			
2612	33.94	oe	ccsbBroad304_04053	DERL1	-			
2613	33.92	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
2614	33.86	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
2615	33.83	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
2616	33.78	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
2617	33.75	kd	CGS001-6632	SNRPD1	-			
2618	33.74	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
2619	33.73	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
2620	33.73	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
2621	33.7	kd	CGS001-9787	DLGAP5	-			
2622	33.61	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
2623	33.6	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
2624	33.55	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
2625	33.51	kd	CGS001-1195	CLK1	CDC-like kinases			
2626	33.5	kd	CGS001-29775	CARD10	-			
2627	33.48	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
2628	33.44	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
2629	33.43	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
2630	33.42	oe	ccsbBroad304_06090	DDOST	-			
2631	33.39	oe	ccsbBroad304_03732	NPDC1	-			
2632	33.37	oe	ccsbBroad304_02205	WTAP	-			
2633	33.37	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
2634	33.35	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
2635	33.31	kd	CGS001-1737	DLAT	-			
2636	33.26	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
2637	33.23	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
2638	33.21	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
2639	33.14	oe	ccsbBroad304_05135	PARP15	-			
2640	33.12	kd	CGS001-5645	PRSS2	Serine peptidases			
2641	33.12	kd	CGS001-55486	PARL	-			
2642	33.05	kd	CGS001-54805	CNNM2	-			
2643	33.03	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
2644	33.01	kd	CGS001-170463	SSBP4	-			
2645	32.99	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
2646	32.93	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
2647	32.92	kd	CGS001-56922	MCCC1	-			
2648	32.9	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
2649	32.89	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
2650	32.87	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
2651	32.8	cp	BRD-K34508425	KUC103898N	-666			-666
2652	32.8	kd	CGS001-5037	PEBP1	-			
2653	32.79	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2654	32.77	kd	CGS001-10544	PROCR	CD molecules			
2655	32.74	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
2656	32.73	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
2657	32.69	oe	ccsbBroad304_03269	CD320	CD molecules			
2658	32.68	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
2659	32.67	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
2660	32.67	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
2661	32.65	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
2662	32.62	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
2663	32.62	kd	CGS001-345	APOC3	Apolipoproteins			
2664	32.6	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
2665	32.58	oe	ccsbBroad304_06136	ECHS1	-			
2666	32.56	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
2667	32.53	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
2668	32.5	kd	CGS001-8837	CFLAR	Endogenous ligands			
2669	32.49	kd	CGS001-55893	ZNF395	Zinc fingers, C2H2-type			
2670	32.43	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2671	32.43	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
2672	32.43	kd	CGS001-54205	CYCS	-			
2673	32.41	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
2674	32.37	cc		Serine proteases GOF	-			
2675	32.31	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
2676	32.29	oe	ccsbBroad304_09354	IGSF8	CD molecules			
2677	32.29	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
2678	32.27	kd	CGS001-9807	IP6K1	-			
2679	32.23	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2680	32.22	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
2681	32.21	oe	ccsbBroad304_07362	NMI	-			
2682	32.13	oe	ccsbBroad304_00120	ATOX1	-			
2683	32.12	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
2684	32.12	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
2685	32.1	kd	CGS001-64135	IFIH1	-			
2686	32.08	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
2687	32.04	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
2688	31.97	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
2689	31.96	oe	ccsbBroad304_06383	HMMR	CD molecules			
2690	31.94	kd	CGS001-6210	RPS15A	S ribosomal proteins			
2691	31.94	kd	CGS001-7852	CXCR4	Chemokine receptors			
2692	31.92	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
2693	31.89	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
2694	31.88	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
2695	31.86	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
2696	31.84	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
2697	31.83	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
2698	31.82	oe	ccsbBroad304_07798	EXOC3	-			
2699	31.75	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
2700	31.71	oe	ccsbBroad304_09006	RPF1	-			
2701	31.68	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
2702	31.66	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
2703	31.59	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
2704	31.59	kd	CGS001-1128	CHRM1	Cholinergic receptors			
2705	31.57	kd	CGS001-6776	STAT5A	SH2 domain containing			
2706	31.57	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
2707	31.57	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
2708	31.48	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
2709	31.31	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
2710	31.25	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
2711	31.21	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2712	31.18	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
2713	31.15	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
2714	31.1	kd	CGS001-9128	PRPF4	WD repeat domain containing			
2715	31.09	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
2716	31.08	kd	CGS001-80349	WDR61	WD repeat domain containing			
2717	31	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
2718	30.99	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
2719	30.85	oe	ccsbBroad304_00212	CAMLG	-			
2720	30.83	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
2721	30.82	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
2722	30.72	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
2723	30.68	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
2724	30.67	kd	CGS001-9412	MED21	-			
2725	30.66	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
2726	30.65	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
2727	30.65	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
2728	30.65	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
2729	30.62	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
2730	30.62	kd	CGS001-23102	TBC1D2B	-			
2731	30.61	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
2732	30.61	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
2733	30.58	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
2734	30.52	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
2735	30.49	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
2736	30.48	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
2737	30.44	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
2738	30.44	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
2739	30.44	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
2740	30.43	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
2741	30.41	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
2742	30.4	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
2743	30.39	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
2744	30.38	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
2745	30.33	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
2746	30.3	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
2747	30.29	oe	ccsbBroad304_07071	TKT	-			
2748	30.26	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2749	30.26	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
2750	30.26	kd	CGS001-345611	IRGM	-			
2751	30.25	kd	CGS001-56616	DIABLO	-			
2752	30.16	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
2753	30.15	oe	ccsbBroad304_05980	CDKN1B	-			
2754	30.07	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
2755	30.05	kd	CGS001-3988	LIPA	-			
2756	30.03	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
2757	30.01	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
2758	29.92	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
2759	29.88	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
2760	29.88	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
2761	29.85	kd	CGS001-861	RUNX1	-			
2762	29.83	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2763	29.79	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
2764	29.76	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
2765	29.63	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
2766	29.61	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
2767	29.59	kd	CGS001-24148	PRPF6	-			
2768	29.58	cc		DNA dependent protein kinase inhibitor	-			
2769	29.57	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
2770	29.52	kd	CGS001-94234	FOXQ1	Forkhead boxes			
2771	29.44	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
2772	29.43	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
2773	29.43	kd	CGS001-771	CA12	Carbonic anhydrases			
2774	29.41	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
2775	29.4	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2776	29.38	kd	CGS001-8801	SUCLG2	-			
2777	29.36	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
2778	29.35	oe	ccsbBroad304_10212	GRHL3	-			
2779	29.35	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
2780	29.32	kd	CGS001-7471	WNT1	Endogenous ligands			
2781	29.28	kd	CGS001-23139	MAST2	MAST family			
2782	29.27	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
2783	29.25	kd	CGS001-9552	SPAG7	-			
2784	29.23	oe	ccsbBroad304_04399	PGBD1	-			
2785	29.19	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
2786	29.19	kd	CGS001-498	ATP5A1	ATPases / F-type			
2787	29.11	kd	CGS001-5209	PFKFB3	-			
2788	29.1	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
2789	29.1	kd	CGS001-5144	PDE4D	Phosphodiesterases			
2790	29.08	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
2791	29.08	kd	CGS001-7035	TFPI	-			
2792	29.07	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
2793	29.04	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
2794	29.02	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
2795	28.95	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
2796	28.94	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
2797	28.94	kd	CGS001-3269	HRH1	Histamine receptors			
2798	28.86	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
2799	28.82	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
2800	28.75	oe	ccsbBroad304_06828	PYCR1	-			
2801	28.75	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
2802	28.74	kd	CGS001-2335	FN1	Endogenous ligands			
2803	28.72	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
2804	28.71	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
2805	28.65	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
2806	28.64	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
2807	28.58	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
2808	28.51	oe	ccsbBroad304_02446	TADA3	-			
2809	28.41	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
2810	28.35	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2811	28.31	kd	CGS001-178	AGL	-			
2812	28.3	oe	ccsbBroad304_04649	ADC	-			
2813	28.3	kd	CGS001-55191	NADSYN1	-			
2814	28.29	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
2815	28.29	kd	CGS001-4683	NBN	-			
2816	28.28	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
2817	28.24	oe	ccsbBroad304_01222	PLP2	-			
2818	28.22	kd	CGS001-2752	GLUL	-			
2819	28.17	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
2820	28.16	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
2821	28.14	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
2822	28.1	kd	CGS001-2242	FES	Fer family			
2823	28.06	kd	CGS001-3416	IDE	Pitrilysin			
2824	28.05	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
2825	28.02	kd	CGS001-29116	MYLIP	-			
2826	27.93	kd	CGS001-3909	LAMA3	Laminins			
2827	27.93	kd	CGS001-11340	EXOSC8	-			
2828	27.88	cc		Cyclin dependent kinases LOF	-			
2829	27.84	oe	ccsbBroad304_04194	ELL3	-			
2830	27.84	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
2831	27.77	kd	CGS001-54442	KCTD5	-			
2832	27.72	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
2833	27.68	kd	CGS001-9670	IPO13	Importins			
2834	27.67	kd	CGS001-51466	EVL	-			
2835	27.66	oe	ccsbBroad304_05038	HORMAD2	-			
2836	27.62	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
2837	27.58	oe	ccsbBroad304_08461	CDCA4	-			
2838	27.56	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
2839	27.55	kd	CGS001-350	APOH	Apolipoproteins			
2840	27.52	kd	CGS001-5378	PMS1	-			
2841	27.51	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
2842	27.5	oe	ccsbBroad304_04457	TOX2	-			
2843	27.48	kd	CGS001-283	ANG	Ribonucleases, RNase A			
2844	27.45	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
2845	27.43	kd	CGS001-439	ASNA1	-			
2846	27.4	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
2847	27.38	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
2848	27.35	kd	CGS001-5690	PSMB2	Proteasome subunits			
2849	27.35	kd	CGS001-283450	C12ORF51	-			
2850	27.15	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
2851	27.14	oe	ccsbBroad304_00100	RHOA	-			
2852	27.13	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
2853	27.13	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
2854	27.09	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
2855	27.06	kd	CGS001-2782	GNB1	WD repeat domain containing			
2856	26.95	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
2857	26.92	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
2858	26.87	kd	CGS001-4931	NVL	ATPases / AAA-type			
2859	26.86	kd	CGS001-8467	SMARCA5	-			
2860	26.86	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
2861	26.84	oe	ccsbBroad304_06976	SMARCE1	-			
2862	26.76	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
2863	26.65	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
2864	26.63	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
2865	26.63	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
2866	26.55	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2867	26.53	oe	ccsbBroad304_04616	ORMDL3	-			
2868	26.5	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
2869	26.49	kd	CGS001-1111	CHEK1	CHK1 subfamily			
2870	26.49	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
2871	26.45	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
2872	26.42	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
2873	26.41	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2874	26.41	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
2875	26.39	kd	CGS001-595	CCND1	-			
2876	26.38	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2877	26.37	cc		EGFR inhibitor	-			
2878	26.35	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
2879	26.34	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
2880	26.3	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
2881	26.25	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
2882	26.24	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2883	26.19	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
2884	26.19	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
2885	26.18	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
2886	26.18	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
2887	26.17	oe	ccsbBroad304_07045	TEAD4	-			
2888	26.16	kd	CGS001-27035	NOX1	-			
2889	26.14	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
2890	26.05	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
2891	26.02	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
2892	25.99	oe	ccsbBroad304_02357	SSX3	-			
2893	25.85	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
2894	25.85	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
2895	25.77	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2896	25.67	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
2897	25.64	oe	ccsbBroad304_02243	DLGAP5	-			
2898	25.6	kd	CGS001-1072	CFL1	-			
2899	25.53	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
2900	25.44	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2901	25.36	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
2902	25.32	kd	CGS001-6829	SUPT5H	-			
2903	25.29	cc		HRH1 antagonist	-			
2904	25.28	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
2905	25.14	cc		MEK inhibitor	-			
2906	25.14	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
2907	25.06	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
2908	25.06	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
2909	25.02	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
2910	24.98	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
2911	24.96	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
2912	24.95	kd	CGS001-29083	GTPBP8	-			
2913	24.93	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2914	24.91	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
2915	24.87	oe	ccsbBroad304_09821	TMEM154	-			
2916	24.87	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
2917	24.83	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
2918	24.83	kd	CGS001-8669	EIF3J	-			
2919	24.82	kd	CGS001-23030	KDM4B	Histone demethylases			
2920	24.78	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
2921	24.76	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
2922	24.75	oe	ccsbBroad304_07887	GCAT	-			
2923	24.75	kd	CGS001-5894	RAF1	RAF family			
2924	24.73	kd	CGS001-10105	PPIF	-			
2925	24.6	cc		HOXL subclass homeoboxes LOF	-			
2926	24.55	kd	CGS001-4245	MGAT1	-			
2927	24.47	oe	ccsbBroad304_00865	ILF2	-			
2928	24.47	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2929	24.39	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
2930	24.38	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
2931	24.29	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
2932	24.26	kd	CGS001-4860	PNP	-			
2933	24.16	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
2934	24.14	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
2935	24.11	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
2936	24.05	oe	ccsbBroad304_06367	HK1	-			
2937	24.02	kd	CGS001-1429	CRYZ	-			
2938	24.01	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
2939	24	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
2940	23.99	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
2941	23.92	kd	CGS001-1029	CDKN2A	-			
2942	23.9	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
2943	23.89	oe	ccsbBroad304_02175	MAGED1	-			
2944	23.83	kd	CGS001-154197	PNLDC1	-			
2945	23.8	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
2946	23.77	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
2947	23.71	kd	CGS001-9612	NCOR2	-			
2948	23.7	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
2949	23.64	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
2950	23.41	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
2951	23.36	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
2952	23.33	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
2953	23.28	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
2954	23.27	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
2955	23.22	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
2956	23.19	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
2957	23.1	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2958	23.07	kd	CGS001-317705	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
2959	23.07	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
2960	23	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
2961	22.99	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
2962	22.89	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
2963	22.88	kd	CGS001-11198	SUPT16H	-			
2964	22.88	kd	CGS001-5663	PSEN1	Presenilin			
2965	22.88	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2966	22.87	cc		PKA inhibitor	-			
2967	22.86	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
2968	22.85	oe	ccsbBroad304_02086	PDLIM1	-			
2969	22.77	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
2970	22.76	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
2971	22.64	kd	CGS001-1036	CDO1	-			
2972	22.58	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
2973	22.54	oe	ccsbBroad304_07374	PTPLA	-			
2974	22.48	kd	CGS001-2932	GSK3B	GSK subfamily			
2975	22.46	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
2976	22.41	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
2977	22.41	oe	ccsbBroad304_03618	OSGEP	-			
2978	22.41	oe	ccsbBroad304_00239	CCNG1	-			
2979	22.35	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
2980	22.35	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
2981	22.3	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
2982	22.19	cc		BMP Signaling LOF	-			
2983	22.16	kd	CGS001-6871	TADA2A	-			
2984	22.15	kd	CGS001-23509	POFUT1	Fucosyltransferases			
2985	22.11	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
2986	22.07	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
2987	22	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
2988	21.88	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
2989	21.86	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
2990	21.67	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
2991	21.54	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
2992	21.5	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
2993	21.48	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
2994	21.43	kd	CGS001-27125	AFF4	-			
2995	21.38	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2996	21.37	kd	CGS001-9232	PTTG1	-			
2997	21.26	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
2998	21.2	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
2999	20.96	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
3000	20.51	cc		Reverse transcriptase inhibitor	-			
3001	20.47	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
3002	20.03	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
3003	19.85	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
3004	19.8	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
3005	19.66	cc		General transcription factors group 2 LOF	-			
3006	19.61	oe	ccsbBroad304_03444	PAF1	-			
3007	19.61	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
3008	19.52	oe	ccsbBroad304_00817	IDH2	-			
3009	19.29	kd	CGS001-1736	DKC1	-			
3010	19.27	kd	CGS001-2203	FBP1	-			
3011	19.24	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
3012	19.04	oe	ccsbBroad304_00690	GRN	-			
3013	19	cc		CDK inhibitor	-			
3014	18.95	kd	CGS001-662	BNIP1	-			
3015	18.93	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
3016	18.74	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
3017	18.6	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
3018	18.56	kd	CGS001-57521	RPTOR	WD repeat domain containing			
3019	18.53	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
3020	18.47	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
3021	18.1	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
3022	18	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
3023	17.97	cc		Thymidylate synthase inhibitor	-			
3024	17.86	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
3025	17.77	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3026	17.75	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
3027	17.69	kd	CGS001-1499	CTNNB1	Catenins			
3028	17.63	kd	CGS001-205	AK4	Adenylate kinases			
3029	17.6	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
3030	17.39	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
3031	17.25	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
3032	17.14	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
3033	16.79	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
3034	16.75	oe	ccsbBroad304_01372	RALB	-			
3035	16.75	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3036	16.75	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
3037	16.64	kd	CGS001-2957	GTF2A1	General transcription factors			
3038	16.59	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
3039	16.56	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3040	16.5	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
3041	16.43	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
3042	16.39	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
3043	16.33	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
3044	16.28	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
3045	16.24	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
3046	16.04	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
3047	16.01	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
3048	15.89	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
3049	15.82	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
3050	15.76	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3051	15.71	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
3052	15.6	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
3053	15.52	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
3054	15.49	cc		Apolipoproteins LOF	-			
3055	15.44	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
3056	15.32	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
3057	15.12	kd	CGS001-966	CD59	CD molecules			
3058	15	cp	BRD-K10065684	dantron	Laxative			Laxative
3059	14.95	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3060	14.93	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
3061	14.89	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
3062	14.74	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
3063	14.66	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
3064	14.49	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
3065	14.35	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
3066	14.31	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
3067	14.28	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3068	14.23	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
3069	13.77	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3070	13.53	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
3071	13.5	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
3072	13.38	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
3073	13.07	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
3074	13.05	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
3075	12.94	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
3076	12.88	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3077	12.84	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
3078	12.75	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
3079	12.66	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
3080	12.52	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
3081	12.47	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
3082	12.46	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
3083	12.45	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3084	12.36	cc		Cyclins LOF	-			
3085	12.29	kd	CGS001-6622	SNCA	Parkinson disease			
3086	11.85	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
3087	11.54	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
3088	10.64	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
3089	10.51	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
3090	10.47	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
3091	10.01	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
3092	9.87	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
3093	9.64	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
3094	9.24	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
3095	8.8	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
3096	8.64	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
3097	7.43	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3098	7.38	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
3099	7.12	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
3100	-5.59	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
3101	-7	kd	CGS001-2288	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
3102	-7.67	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
3103	-7.68	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
3104	-8.27	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
3105	-8.58	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
3106	-8.68	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3107	-8.72	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3108	-8.99	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
3109	-9.55	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
3110	-9.67	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
3111	-9.72	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
3112	-9.94	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
3113	-10.17	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
3114	-10.18	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
3115	-10.23	kd	CGS001-50808	AK3	-			
3116	-10.26	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
3117	-10.35	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3118	-10.67	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
3119	-10.88	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
3120	-11.23	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
3121	-11.25	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
3122	-11.25	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
3123	-11.39	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
3124	-11.56	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
3125	-11.71	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
3126	-11.91	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
3127	-12.26	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
3128	-12.49	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3129	-12.51	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
3130	-12.67	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
3131	-12.79	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
3132	-12.94	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
3133	-12.94	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
3134	-13.39	kd	CGS001-65263	PYCRL	-			
3135	-13.56	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
3136	-13.57	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
3137	-13.73	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
3138	-13.87	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
3139	-14.45	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
3140	-14.53	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
3141	-14.63	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
3142	-14.64	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3143	-14.68	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
3144	-14.7	kd	CGS001-11040	PIM2	PIM family			
3145	-15.02	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
3146	-15.03	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
3147	-15.05	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
3148	-15.12	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
3149	-15.22	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
3150	-15.23	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
3151	-15.4	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
3152	-15.41	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
3153	-15.52	kd	CGS001-5933	RBL1	-			
3154	-15.54	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
3155	-15.54	kd	CGS001-2277	FIGF	-			
3156	-15.64	oe	ccsbBroad304_00231	CBFB	-			
3157	-15.65	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
3158	-16	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
3159	-16.11	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
3160	-16.25	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
3161	-16.52	oe	ccsbBroad304_01084	NEU1	-			
3162	-16.57	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
3163	-16.67	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
3164	-16.67	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
3165	-16.71	kd	CGS001-84669	USP32	EF-hand domain containing			
3166	-16.79	kd	CGS001-11344	TWF2	Twinfilin subfamily			
3167	-16.8	cc		ATPase inhibitor	-			
3168	-16.98	kd	CGS001-7965	AIMP2	-			
3169	-17.08	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
3170	-17.17	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
3171	-17.25	oe	ccsbBroad304_01327	PSPH	-			
3172	-17.31	kd	CGS001-112858	TP53RK	Bud32 family			
3173	-17.41	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
3174	-17.42	oe	ccsbBroad304_02497	YKT6	-			
3175	-17.43	oe	ccsbBroad304_00162	BIK	-			
3176	-17.57	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
3177	-17.57	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
3178	-17.69	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
3179	-17.71	cc		Phospholipases LOF	-			
3180	-17.98	kd	CGS001-8536	CAMK1	CAMK1 family			
3181	-17.99	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
3182	-18.02	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
3183	-18.03	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
3184	-18.29	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
3185	-18.32	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
3186	-18.37	kd	CGS001-6197	RPS6KA3	RSK subfamily			
3187	-18.46	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
3188	-18.5	oe	ccsbBroad304_04292	INHBE	-			
3189	-18.51	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
3190	-18.66	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
3191	-18.69	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
3192	-18.73	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
3193	-18.79	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
3194	-18.91	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
3195	-18.93	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
3196	-18.99	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
3197	-19.12	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
3198	-19.13	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
3199	-19.13	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
3200	-19.14	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
3201	-19.31	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
3202	-19.31	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
3203	-19.33	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
3204	-19.38	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
3205	-19.4	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
3206	-19.45	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
3207	-19.47	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
3208	-19.48	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
3209	-19.54	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
3210	-19.55	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
3211	-19.76	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
3212	-19.8	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
3213	-19.83	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
3214	-19.93	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
3215	-19.96	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
3216	-19.97	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
3217	-20.08	kd	CGS001-7013	TERF1	-			
3218	-20.14	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
3219	-20.16	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
3220	-20.17	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
3221	-20.18	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3222	-20.22	kd	CGS001-4151	MB	-			
3223	-20.29	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
3224	-20.29	kd	CGS001-4067	LYN	Src family			
3225	-20.35	kd	CGS001-5962	RDX	-			
3226	-20.39	kd	CGS001-7057	THBS1	-			
3227	-20.39	kd	CGS001-10797	MTHFD2	-			
3228	-20.45	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3229	-20.45	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
3230	-20.54	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
3231	-20.59	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
3232	-20.73	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
3233	-20.76	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
3234	-20.8	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
3235	-20.85	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
3236	-20.87	kd	CGS001-347736	NME9	-			
3237	-20.94	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
3238	-20.99	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
3239	-20.99	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
3240	-21	kd	CGS001-51586	MED15	-			
3241	-21.09	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
3242	-21.19	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
3243	-21.19	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
3244	-21.2	oe	ccsbBroad304_06234	G6PC	-			
3245	-21.29	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
3246	-21.33	kd	CGS001-5688	PSMA7	Proteasome subunits			
3247	-21.33	kd	CGS001-23510	KCTD2	-			
3248	-21.38	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
3249	-21.38	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
3250	-21.4	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
3251	-21.43	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
3252	-21.45	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
3253	-21.46	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
3254	-21.46	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
3255	-21.56	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
3256	-21.61	cc		Progesterone receptor antagonist	-			
3257	-21.68	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
3258	-21.7	oe	ccsbBroad304_04534	HN1L	-			
3259	-21.7	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
3260	-21.76	kd	CGS001-2615	LRRC32	-			
3261	-21.8	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
3262	-21.8	kd	CGS001-9318	COPS2	-			
3263	-21.91	cc		Proteasome inhibitor	-			
3264	-21.92	oe	ccsbBroad304_02509	GMEB1	-			
3265	-21.92	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
3266	-21.92	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
3267	-22.01	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
3268	-22.01	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
3269	-22.03	kd	CGS001-4436	MSH2	-			
3270	-22.07	kd	CGS001-8192	CLPP	ATPases / AAA-type			
3271	-22.11	kd	CGS001-4637	MYL6	EF-hand domain containing			
3272	-22.15	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
3273	-22.2	kd	CGS001-5613	PRKX	Protein kinase A			
3274	-22.21	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3275	-22.29	oe	ccsbBroad304_00985	MCL1	-			
3276	-22.29	kd	CGS001-117154	DACH2	-			
3277	-22.3	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
3278	-22.3	oe	ccsbBroad304_02452	NXF1	-			
3279	-22.32	oe	ccsbBroad304_07598	PEMT	-			
3280	-22.32	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
3281	-22.36	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
3282	-22.36	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
3283	-22.37	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
3284	-22.38	kd	CGS001-7477	WNT7B	Endogenous ligands			
3285	-22.4	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
3286	-22.41	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
3287	-22.42	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
3288	-22.44	kd	CGS001-5245	PHB	-			
3289	-22.46	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
3290	-22.46	kd	CGS001-2877	GPX2	-			
3291	-22.48	oe	ccsbBroad304_02487	TXNIP	-			
3292	-22.51	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
3293	-22.56	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
3294	-22.56	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
3295	-22.58	oe	ccsbBroad304_00645	GCLM	-			
3296	-22.64	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
3297	-22.67	kd	CGS001-10329	TMEM5	-			
3298	-22.71	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
3299	-22.75	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
3300	-22.77	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
3301	-22.87	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
3302	-22.87	kd	CGS001-2588	GALNS	Arylsulfatase family			
3303	-22.93	kd	CGS001-4664	NAB1	-			
3304	-22.94	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
3305	-22.96	kd	CGS001-271	AMPD2	-			
3306	-23.07	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
3307	-23.07	kd	CGS001-54407	SLC38A2	System A-like transporters			
3308	-23.08	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
3309	-23.09	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
3310	-23.1	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
3311	-23.11	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
3312	-23.12	kd	CGS001-4069	LYZ	-			
3313	-23.22	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
3314	-23.23	kd	CGS001-213	ALB	-			
3315	-23.25	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
3316	-23.26	kd	CGS001-10001	MED6	-			
3317	-23.26	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
3318	-23.27	oe	ccsbBroad304_00969	MAGEA10	-			
3319	-23.29	kd	CGS001-25885	POLR1A	RNA polymerase subunits			
3320	-23.39	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3321	-23.51	kd	CGS001-7088	TLE1	WD repeat domain containing			
3322	-23.55	oe	ccsbBroad304_07012	STK3	MST subfamily			
3323	-23.57	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
3324	-23.6	oe	ccsbBroad304_08325	LIPT1	-			
3325	-23.61	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
3326	-23.62	oe	ccsbBroad304_06837	RAF1	RAF family			
3327	-23.67	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3328	-23.73	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
3329	-23.81	kd	CGS001-6788	STK3	MST subfamily			
3330	-23.85	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
3331	-23.91	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3332	-23.98	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
3333	-24.01	oe	ccsbBroad304_07754	FGFR1OP	-			
3334	-24.01	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
3335	-24.07	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
3336	-24.08	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
3337	-24.1	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
3338	-24.17	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
3339	-24.19	kd	CGS001-2309	FOXO3	Forkhead boxes			
3340	-24.22	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
3341	-24.23	oe	ccsbBroad304_05947	CCNC	-			
3342	-24.28	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
3343	-24.29	kd	CGS001-9926	LPGAT1	-			
3344	-24.31	kd	CGS001-6193	RPS5	S ribosomal proteins			
3345	-24.31	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
3346	-24.32	kd	CGS001-23588	KLHDC2	-			
3347	-24.36	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
3348	-24.41	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
3349	-24.42	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
3350	-24.46	oe	ccsbBroad304_01392	TRIM27	-			
3351	-24.47	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
3352	-24.48	kd	CGS001-10314	LANCL1	-			
3353	-24.49	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
3354	-24.53	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
3355	-24.56	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
3356	-24.56	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
3357	-24.57	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
3358	-24.57	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
3359	-24.58	cc		Interleukin receptors LOF	-			
3360	-24.66	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
3361	-24.66	kd	CGS001-4547	MTTP	-			
3362	-24.68	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
3363	-24.69	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
3364	-24.72	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
3365	-24.72	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
3366	-24.73	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
3367	-24.73	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
3368	-24.76	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3369	-24.78	oe	ccsbBroad304_06648	CNOT3	-			
3370	-24.79	kd	CGS001-5110	PCMT1	-			
3371	-24.81	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
3372	-24.81	kd	CGS001-310	ANXA7	Annexins			
3373	-24.81	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
3374	-24.82	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
3375	-24.87	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
3376	-24.88	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
3377	-24.94	kd	CGS001-5979	RET	Type XIV RTKs: RET			
3378	-24.94	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
3379	-24.95	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
3380	-24.96	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
3381	-24.97	oe	ccsbBroad304_06140	EEF1D	-			
3382	-24.98	kd	CGS001-8870	IER3	-			
3383	-25.01	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
3384	-25.03	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
3385	-25.03	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3386	-25.11	kd	CGS001-2697	GJA1	Ion channels / Gap junction proteins (connexins)			
3387	-25.12	kd	CGS001-5355	PLP2	-			
3388	-25.21	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
3389	-25.23	cc		Sodium channel blocker	-			
3390	-25.25	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
3391	-25.29	kd	CGS001-11136	SLC7A9	SLC7 family			
3392	-25.29	kd	CGS001-4179	CD46	CD molecules			
3393	-25.37	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
3394	-25.39	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
3395	-25.43	kd	CGS001-6895	TARBP2	-			
3396	-25.47	oe	ccsbBroad304_09881	RFX6	-			
3397	-25.5	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
3398	-25.52	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
3399	-25.53	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
3400	-25.54	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
3401	-25.57	kd	CGS001-80314	EPC1	-			
3402	-25.6	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
3403	-25.62	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
3404	-25.62	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
3405	-25.64	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
3406	-25.66	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
3407	-25.67	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
3408	-25.69	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
3409	-25.7	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
3410	-25.88	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
3411	-25.89	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
3412	-25.93	kd	CGS001-5194	PEX13	-			
3413	-25.96	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
3414	-25.97	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
3415	-25.98	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
3416	-25.99	kd	CGS001-1950	EGF	-			
3417	-26.02	kd	CGS001-149233	IL23R	IL-12 receptor family			
3418	-26.03	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
3419	-26.06	kd	CGS001-9275	BCL7B	-			
3420	-26.08	kd	CGS001-3383	ICAM1	CD molecules			
3421	-26.13	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
3422	-26.13	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
3423	-26.14	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
3424	-26.16	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
3425	-26.2	cc		Non Homologous End Joining LOF	-			
3426	-26.2	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
3427	-26.21	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
3428	-26.24	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
3429	-26.3	kd	CGS001-9322	TRIP10	-			
3430	-26.31	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
3431	-26.32	kd	CGS001-5253	PHF2	Histone demethylases			
3432	-26.36	kd	CGS001-9159	PCSK7	Subtilisin			
3433	-26.37	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
3434	-26.38	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
3435	-26.42	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
3436	-26.43	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
3437	-26.45	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
3438	-26.48	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
3439	-26.51	oe	ccsbBroad304_02533	NOXA1	-			
3440	-26.53	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
3441	-26.55	kd	CGS001-10652	YKT6	-			
3442	-26.55	kd	CGS001-4173	MCM4	-			
3443	-26.57	kd	CGS001-1503	CTPS	-			
3444	-26.59	oe	ccsbBroad304_02109	XPR1	-			
3445	-26.62	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
3446	-26.63	oe	ccsbBroad304_03186	GMNN	-			
3447	-26.63	kd	CGS001-6201	RPS7	S ribosomal proteins			
3448	-26.64	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
3449	-26.67	kd	CGS001-174	AFP	-			
3450	-26.68	oe	ccsbBroad304_02838	SDF2L1	-			
3451	-26.68	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
3452	-26.68	oe	ccsbBroad304_00053	ALDOA	-			
3453	-26.68	kd	CGS001-144811	LACC1	-			
3454	-26.69	oe	ccsbBroad304_02919	KIAA1279	-			
3455	-26.71	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
3456	-26.71	oe	ccsbBroad304_07466	VGLL4	-			
3457	-26.71	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
3458	-26.74	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
3459	-26.76	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
3460	-26.77	oe	ccsbBroad304_07197	PDHX	-			
3461	-26.87	oe	ccsbBroad304_00222	CASP6	Caspases			
3462	-26.87	kd	CGS001-1948	EFNB2	Ephrins			
3463	-26.9	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
3464	-26.9	kd	CGS001-10614	HEXIM1	-			
3465	-26.9	kd	CGS001-2000	ELF4	ETS Transcription Factors			
3466	-26.93	kd	CGS001-8800	PEX11A	-			
3467	-27.02	kd	CGS001-3242	HPD	Oxidoreductases			
3468	-27.04	kd	CGS001-10755	GIPC1	-			
3469	-27.05	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
3470	-27.05	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
3471	-27.08	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
3472	-27.1	kd	CGS001-25824	PRDX5	-			
3473	-27.14	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
3474	-27.14	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
3475	-27.14	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
3476	-27.15	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
3477	-27.25	kd	CGS001-3572	IL6ST	IL-6 receptor family			
3478	-27.26	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
3479	-27.28	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
3480	-27.34	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
3481	-27.34	oe	ccsbBroad304_03728	DIABLO	-			
3482	-27.35	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
3483	-27.35	kd	CGS001-122402	TDRD9	Tudor domain containing			
3484	-27.35	kd	CGS001-23192	ATG4B	Aut2 peptidase			
3485	-27.36	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
3486	-27.37	kd	CGS001-23369	PUM2	-			
3487	-27.37	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
3488	-27.39	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
3489	-27.4	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
3490	-27.4	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
3491	-27.4	kd	CGS001-3161	HMMR	CD molecules			
3492	-27.5	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
3493	-27.5	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
3494	-27.51	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
3495	-27.51	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
3496	-27.51	oe	ccsbBroad304_06765	PRCC	-			
3497	-27.57	oe	ccsbBroad304_07528	DMTF1	-			
3498	-27.57	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
3499	-27.59	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
3500	-27.59	kd	CGS001-1528	CYB5A	Cytochrome b genes			
3501	-27.61	oe	ccsbBroad304_00491	EIF4EBP2	-			
3502	-27.61	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
3503	-27.66	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
3504	-27.66	kd	CGS001-26292	MYCBP	-			
3505	-27.73	oe	ccsbBroad304_06144	EFNB3	Ephrins			
3506	-27.73	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
3507	-27.75	oe	ccsbBroad304_02373	SPRY2	-			
3508	-27.77	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
3509	-27.77	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
3510	-27.83	oe	ccsbBroad304_09954	PTRF	-			
3511	-27.85	kd	CGS001-3421	IDH3G	-			
3512	-27.86	cc		Serpin peptidase inhibitors LOF	-			
3513	-27.86	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
3514	-27.87	cc		Topoisomerase inhibitor	-			
3515	-27.89	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
3516	-27.9	oe	ccsbBroad304_03555	PANK4	-			
3517	-27.92	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
3518	-27.97	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
3519	-28	kd	CGS001-4046	LSP1	-			
3520	-28.02	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
3521	-28.02	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
3522	-28.06	kd	CGS001-4998	ORC1	ATPases / AAA-type			
3523	-28.07	oe	ccsbBroad304_03121	NRBF2	-			
3524	-28.07	kd	CGS001-5105	PCK1	-			
3525	-28.12	oe	ccsbBroad304_00519	ETFB	-			
3526	-28.15	kd	CGS001-7090	TLE3	WD repeat domain containing			
3527	-28.16	kd	CGS001-10214	SSX3	-			
3528	-28.16	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
3529	-28.2	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
3530	-28.2	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
3531	-28.23	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
3532	-28.23	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
3533	-28.25	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
3534	-28.31	kd	CGS001-54681	P4HTM	-			
3535	-28.33	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
3536	-28.35	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
3537	-28.35	oe	ccsbBroad304_01862	YEATS4	-			
3538	-28.38	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
3539	-28.44	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
3540	-28.45	kd	CGS001-23075	SWAP70	EF-hand domain containing			
3541	-28.54	cc		Wnt family LOF	-			
3542	-28.54	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3543	-28.56	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
3544	-28.57	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
3545	-28.58	kd	CGS001-3663	IRF5	-			
3546	-28.59	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
3547	-28.61	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
3548	-28.65	kd	CGS001-2114	ETS2	ETS Transcription Factors			
3549	-28.66	oe	ccsbBroad304_06174	ERCC1	-			
3550	-28.71	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
3551	-28.72	kd	CGS001-11336	EXOC3	-			
3552	-28.73	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
3553	-28.73	oe	ccsbBroad304_00648	GLRX	-			
3554	-28.74	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
3555	-28.74	kd	CGS001-63892	THADA	-			
3556	-28.75	oe	ccsbBroad304_02875	BRP44	-			
3557	-28.78	cc		Kruppel like transcription factors LOF	-			
3558	-28.78	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
3559	-28.79	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
3560	-28.79	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
3561	-28.9	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
3562	-28.94	kd	CGS001-57018	CCNL1	-			
3563	-29.01	kd	CGS001-9641	IKBKE	IKK family			
3564	-29.02	oe	ccsbBroad304_02869	ASF1A	-			
3565	-29.03	kd	CGS001-1647	GADD45A	-			
3566	-29.08	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
3567	-29.08	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
3568	-29.1	kd	CGS001-57149	LYRM1	LYR motif containing			
3569	-29.11	oe	ccsbBroad304_08426	TEX10	-			
3570	-29.11	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3571	-29.11	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
3572	-29.13	kd	CGS001-56654	NPDC1	-			
3573	-29.15	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
3574	-29.16	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
3575	-29.17	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
3576	-29.18	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
3577	-29.2	kd	CGS001-5004	ORM1	Lipocalins			
3578	-29.25	kd	CGS001-7270	TTF1	-			
3579	-29.26	kd	CGS001-3590	IL11RA	IL-6 receptor family			
3580	-29.27	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
3581	-29.27	kd	CGS001-4833	NME4	-			
3582	-29.3	oe	ccsbBroad304_00389	CTBP1	-			
3583	-29.33	kd	CGS001-375133	PI4KAP2	-			
3584	-29.34	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
3585	-29.37	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
3586	-29.37	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
3587	-29.38	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
3588	-29.39	kd	CGS001-5292	PIM1	PIM family			
3589	-29.42	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
3590	-29.42	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
3591	-29.43	oe	ccsbBroad304_03040	NKIRAS2	-			
3592	-29.48	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
3593	-29.48	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
3594	-29.5	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
3595	-29.52	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
3596	-29.52	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
3597	-29.55	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3598	-29.57	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
3599	-29.58	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
3600	-29.61	oe	ccsbBroad304_06040	CRY1	-			
3601	-29.67	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
3602	-29.75	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3603	-29.76	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
3604	-29.79	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
3605	-29.8	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
3606	-29.82	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
3607	-29.84	kd	CGS001-11142	PKIG	-			
3608	-29.85	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
3609	-29.88	oe	ccsbBroad304_00510	EPHX2	-			
3610	-29.92	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
3611	-29.92	kd	CGS001-1514	CTSL1	-			
3612	-29.93	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
3613	-29.95	kd	CGS001-29915	HCFC2	-			
3614	-29.96	kd	CGS001-2534	FYN	Src family			
3615	-29.99	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
3616	-30	kd	CGS001-7292	TNFSF4	CD molecules			
3617	-30	kd	CGS001-122809	SOCS4	SH2 domain containing			
3618	-30	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
3619	-30.01	oe	ccsbBroad304_01001	MEST	-			
3620	-30.03	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
3621	-30.12	oe	ccsbBroad304_02133	CD83	CD molecules			
3622	-30.14	cc		Bacterial DNA gyrase inhibitor	-			
3623	-30.16	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
3624	-30.19	oe	ccsbBroad304_02605	PAPD7	-			
3625	-30.2	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
3626	-30.2	kd	CGS001-169436	C9ORF96	-			
3627	-30.22	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
3628	-30.24	kd	CGS001-10476	ATP5H	ATPases / F-type			
3629	-30.28	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3630	-30.34	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
3631	-30.34	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
3632	-30.35	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
3633	-30.35	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
3634	-30.39	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
3635	-30.44	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
3636	-30.45	oe	ccsbBroad304_01034	MSH2	-			
3637	-30.47	kd	CGS001-9270	ITGB1BP1	-			
3638	-30.48	kd	CGS001-1196	CLK2	CDC-like kinases			
3639	-30.49	oe	ccsbBroad304_06134	ECH1	-			
3640	-30.49	kd	CGS001-5573	PRKAR1A	Protein kinase A			
3641	-30.5	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
3642	-30.5	kd	CGS001-5575	PRKAR1B	Protein kinase A			
3643	-30.52	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
3644	-30.52	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
3645	-30.55	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
3646	-30.55	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3647	-30.56	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
3648	-30.56	kd	CGS001-7832	BTG2	-			
3649	-30.61	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
3650	-30.65	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
3651	-30.67	oe	ccsbBroad304_01351	PEX19	-			
3652	-30.68	kd	CGS001-6258	RXRG	Retinoid X receptors			
3653	-30.69	kd	CGS001-629	CFB	Complement system			
3654	-30.7	oe	ccsbBroad304_10207	ERLIN1	-			
3655	-30.72	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
3656	-30.81	kd	CGS001-55620	STAP2	-			
3657	-30.82	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
3658	-30.83	oe	ccsbBroad304_00949	LRPAP1	-			
3659	-30.83	oe	ccsbBroad304_07592	CEPT1	-			
3660	-30.83	kd	CGS001-29110	TBK1	IKK family			
3661	-30.84	kd	CGS001-149428	BNIPL	-			
3662	-30.85	oe	ccsbBroad304_01131	OXCT1	-			
3663	-30.87	kd	CGS001-93185	IGSF8	CD molecules			
3664	-30.87	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
3665	-31	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
3666	-31	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
3667	-31.02	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
3668	-31.09	kd	CGS001-54541	DDIT4	-			
3669	-31.11	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
3670	-31.12	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
3671	-31.13	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
3672	-31.14	oe	ccsbBroad304_02318	KIF20A	Kinesins			
3673	-31.14	oe	ccsbBroad304_00282	CDKN1A	-			
3674	-31.16	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
3675	-31.18	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
3676	-31.19	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
3677	-31.22	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
3678	-31.23	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
3679	-31.27	oe	ccsbBroad304_13813	ARAF	RAF family			
3680	-31.3	kd	CGS001-10250	SRRM1	-			
3681	-31.31	oe	ccsbBroad304_05439	O3FAR1	-			
3682	-31.31	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
3683	-31.39	kd	CGS001-4086	SMAD1	SMADs			
3684	-31.5	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
3685	-31.5	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
3686	-31.5	oe	ccsbBroad304_00183	C1S	Complement system			
3687	-31.53	cc		Trace amine receptors LOF	-			
3688	-31.56	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
3689	-31.57	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
3690	-31.63	oe	ccsbBroad304_03696	C19ORF10	-			
3691	-31.64	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
3692	-31.65	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
3693	-31.65	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
3694	-31.67	kd	CGS001-6195	RPS6KA1	RSK subfamily			
3695	-31.68	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
3696	-31.68	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
3697	-31.68	kd	CGS001-56731	SLC2A4RG	-			
3698	-31.69	kd	CGS001-5997	RGS2	Endogenous ligands			
3699	-31.69	kd	CGS001-8841	HDAC3	Histone deacetylases			
3700	-31.69	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
3701	-31.71	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
3702	-31.73	oe	ccsbBroad304_07814	SACM1L	-			
3703	-31.73	kd	CGS001-26227	PHGDH	-			
3704	-31.74	oe	ccsbBroad304_00652	GNAS	-			
3705	-31.77	oe	ccsbBroad304_00397	CTSK	Cathepsins			
3706	-31.78	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
3707	-31.78	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
3708	-31.78	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
3709	-31.78	kd	CGS001-1488	CTBP2	-			
3710	-31.81	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
3711	-31.82	kd	CGS001-200734	SPRED2	-			
3712	-31.84	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
3713	-31.85	oe	ccsbBroad304_07029	TADA2A	-			
3714	-31.85	kd	CGS001-6009	RHEB	-			
3715	-31.86	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
3716	-31.87	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
3717	-31.88	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
3718	-31.88	oe	ccsbBroad304_01143	PAFAH1B3	-			
3719	-31.88	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
3720	-31.97	oe	ccsbBroad304_01976	EIF4EBP3	-			
3721	-32	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
3722	-32.02	kd	CGS001-3171	FOXA3	Forkhead boxes			
3723	-32.09	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
3724	-32.09	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3725	-32.12	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
3726	-32.13	oe	ccsbBroad304_10846	GGT1	CD molecules			
3727	-32.22	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
3728	-32.23	oe	ccsbBroad304_10758	CTBP2	-			
3729	-32.23	kd	CGS001-1534	CYB561	Cytochrome b genes			
3730	-32.24	oe	ccsbBroad304_05937	CASP7	Caspases			
3731	-32.26	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
3732	-32.27	kd	CGS001-4287	ATXN3	Ataxins			
3733	-32.28	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
3734	-32.3	oe	ccsbBroad304_00709	GUK1	-			
3735	-32.31	kd	CGS001-7020	TFAP2A	-			
3736	-32.34	oe	ccsbBroad304_03934	LEPRE1	-			
3737	-32.34	kd	CGS001-7504	XK	Blood group antigens			
3738	-32.34	kd	CGS001-10013	HDAC6	Histone deacetylases			
3739	-32.36	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
3740	-32.36	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
3741	-32.4	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3742	-32.41	oe	ccsbBroad304_14143	NUSAP1	-			
3743	-32.42	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
3744	-32.42	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
3745	-32.43	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
3746	-32.43	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
3747	-32.44	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
3748	-32.45	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
3749	-32.47	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3750	-32.49	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
3751	-32.51	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
3752	-32.52	kd	CGS001-2523	FUT1	Fucosyltransferases			
3753	-32.55	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
3754	-32.59	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
3755	-32.65	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
3756	-32.72	oe	ccsbBroad304_07843	FCHO1	-			
3757	-32.72	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
3758	-32.74	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
3759	-32.78	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
3760	-32.79	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
3761	-32.8	kd	CGS001-353	APRT	-			
3762	-32.86	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
3763	-32.9	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
3764	-32.91	kd	CGS001-2053	EPHX2	-			
3765	-32.93	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
3766	-32.97	cc		FXR antagonist	-			
3767	-32.97	oe	ccsbBroad304_04675	ATG4A	-			
3768	-33.06	oe	ccsbBroad304_07888	CBX6	-			
3769	-33.07	kd	CGS001-4171	MCM2	-			
3770	-33.08	oe	ccsbBroad304_07401	TXNL1	-			
3771	-33.12	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
3772	-33.12	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
3773	-33.17	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
3774	-33.17	kd	CGS001-8895	CPNE3	-			
3775	-33.23	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
3776	-33.24	oe	ccsbBroad304_06420	ICAM3	CD molecules			
3777	-33.25	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
3778	-33.31	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
3779	-33.33	oe	ccsbBroad304_01114	NUP88	-			
3780	-33.35	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
3781	-33.36	oe	ccsbBroad304_06178	ERCC5	-			
3782	-33.39	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
3783	-33.39	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
3784	-33.4	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
3785	-33.41	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
3786	-33.42	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
3787	-33.42	kd	CGS001-283150	FOXR1	Forkhead boxes			
3788	-33.42	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
3789	-33.43	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
3790	-33.45	oe	ccsbBroad304_04891	TMEM174	-			
3791	-33.45	kd	CGS001-9375	TM9SF2	-			
3792	-33.45	kd	CGS001-4200	ME2	-			
3793	-33.48	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
3794	-33.5	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
3795	-33.5	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
3796	-33.51	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
3797	-33.51	kd	CGS001-5621	PRNP	CD molecules			
3798	-33.52	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
3799	-33.52	kd	CGS001-54499	TMCO1	-			
3800	-33.52	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
3801	-33.55	oe	ccsbBroad304_14291	GDPD5	-			
3802	-33.56	kd	CGS001-7263	TST	-			
3803	-33.59	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
3804	-33.62	kd	CGS001-4267	CD99	CD molecules			
3805	-33.65	oe	ccsbBroad304_00941	LIG3	-			
3806	-33.65	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
3807	-33.68	kd	CGS001-11179	ZNF277	-			
3808	-33.7	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
3809	-33.72	kd	CGS001-10198	MPHOSPH9	-			
3810	-33.75	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
3811	-33.79	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
3812	-33.82	oe	ccsbBroad304_00262	CD59	CD molecules			
3813	-33.82	kd	CGS001-8525	DGKZ	-			
3814	-33.83	kd	CGS001-5887	RAD23B	-			
3815	-33.84	oe	ccsbBroad304_00249	CD14	CD molecules			
3816	-33.85	kd	CGS001-83593	RASSF5	-			
3817	-33.86	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
3818	-33.86	kd	CGS001-1062	CENPE	Kinesins			
3819	-33.92	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
3820	-33.95	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
3821	-33.97	oe	ccsbBroad304_03386	SPA17	-			
3822	-33.98	kd	CGS001-25987	TSKU	-			
3823	-34.03	kd	CGS001-7016	TESK1	TESK subfamily			
3824	-34.04	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
3825	-34.05	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
3826	-34.11	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
3827	-34.16	kd	CGS001-11329	STK38	NDR family			
3828	-34.17	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
3829	-34.18	kd	CGS001-28511	NKIRAS2	-			
3830	-34.21	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
3831	-34.23	kd	CGS001-64428	NARFL	-			
3832	-34.24	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
3833	-34.25	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
3834	-34.26	kd	CGS001-2548	GAA	Glycosidases			
3835	-34.32	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
3836	-34.32	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
3837	-34.35	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
3838	-34.37	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
3839	-34.42	oe	ccsbBroad304_02345	TXNDC9	-			
3840	-34.44	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
3841	-34.49	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
3842	-34.51	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
3843	-34.51	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
3844	-34.54	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
3845	-34.56	oe	ccsbBroad304_00876	INSIG1	-			
3846	-34.56	kd	CGS001-29883	CNOT7	-			
3847	-34.57	kd	CGS001-5763	PTMS	-			
3848	-34.57	kd	CGS001-427	ASAH1	Acid ceramidase			
3849	-34.59	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
3850	-34.59	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3851	-34.6	kd	CGS001-10111	RAD50	-			
3852	-34.61	oe	ccsbBroad304_01166	PDK2	PDHK family			
3853	-34.61	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
3854	-34.65	kd	CGS001-80212	CCDC92	-			
3855	-34.68	kd	CGS001-3845	KRAS	RAS subfamily			
3856	-34.68	kd	CGS001-2987	GUK1	-			
3857	-34.69	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
3858	-34.69	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
3859	-34.69	kd	CGS001-54108	CHRAC1	-			
3860	-34.71	kd	CGS001-51593	SRRT	-			
3861	-34.73	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
3862	-34.74	cc		C2 domain containing protein kinases LOF	-			
3863	-34.77	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
3864	-34.77	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
3865	-34.79	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
3866	-34.82	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
3867	-34.82	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
3868	-34.83	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
3869	-34.88	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
3870	-34.91	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
3871	-34.93	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3872	-34.95	kd	CGS001-2098	ESD	-			
3873	-34.98	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
3874	-34.99	kd	CGS001-1869	E2F1	-			
3875	-35	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
3876	-35	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
3877	-35.01	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
3878	-35.02	oe	ccsbBroad304_08553	STAP2	-			
3879	-35.02	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
3880	-35.08	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
3881	-35.08	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
3882	-35.08	kd	CGS001-5588	PRKCQ	Delta subfamily			
3883	-35.1	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
3884	-35.1	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
3885	-35.12	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
3886	-35.13	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3887	-35.14	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
3888	-35.17	oe	ccsbBroad304_03072	GTPBP8	-			
3889	-35.17	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
3890	-35.19	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
3891	-35.2	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
3892	-35.2	kd	CGS001-50846	DHH	-			
3893	-35.22	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
3894	-35.22	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
3895	-35.22	kd	CGS001-5480	PPIC	-			
3896	-35.29	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
3897	-35.32	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
3898	-35.32	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
3899	-35.33	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
3900	-35.38	oe	ccsbBroad304_02047	AP1S2	-			
3901	-35.39	oe	ccsbBroad304_06952	SKP1	-			
3902	-35.4	oe	ccsbBroad304_06855	RDX	-			
3903	-35.44	oe	ccsbBroad304_08839	IFIH1	-			
3904	-35.44	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
3905	-35.48	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
3906	-35.48	kd	CGS001-55038	CDCA4	-			
3907	-35.49	kd	CGS001-5906	RAP1A	-			
3908	-35.51	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
3909	-35.52	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
3910	-35.53	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
3911	-35.57	oe	ccsbBroad304_01184	PGK1	-			
3912	-35.58	oe	ccsbBroad304_03850	TRIB3	Trbl family			
3913	-35.58	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
3914	-35.6	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
3915	-35.61	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
3916	-35.62	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3917	-35.62	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
3918	-35.65	kd	CGS001-6514	SLC2A2	Solute carriers			
3919	-35.65	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
3920	-35.67	oe	ccsbBroad304_05152	SSBP4	-			
3921	-35.67	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
3922	-35.69	kd	CGS001-55214	LEPREL1	-			
3923	-35.7	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
3924	-35.7	kd	CGS001-29102	DROSHA	-			
3925	-35.74	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
3926	-35.75	oe	ccsbBroad304_01617	STX4	-			
3927	-35.75	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
3928	-35.76	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
3929	-35.76	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
3930	-35.77	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
3931	-35.78	oe	ccsbBroad304_06862	RGS3	-			
3932	-35.78	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
3933	-35.86	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
3934	-35.87	kd	CGS001-9140	ATG12	-			
3935	-35.88	oe	ccsbBroad304_07922	TRIM29	-			
3936	-35.9	kd	CGS001-2645	GCK	Hexokinases			
3937	-35.92	kd	CGS001-1611	DAP	-			
3938	-35.95	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
3939	-35.95	kd	CGS001-3992	FADS1	Fatty acid desaturases			
3940	-35.96	oe	ccsbBroad304_02633	LSM6	-			
3941	-35.96	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
3942	-35.98	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
3943	-36	kd	CGS001-670	BPHL	-			
3944	-36.04	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
3945	-36.05	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
3946	-36.05	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
3947	-36.07	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
3948	-36.07	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
3949	-36.08	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
3950	-36.09	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
3951	-36.1	cc		Canonical high mobility group proteins LOF	-			
3952	-36.12	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
3953	-36.12	kd	CGS001-10841	FTCD	-			
3954	-36.14	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
3955	-36.14	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
3956	-36.16	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
3957	-36.16	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
3958	-36.16	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
3959	-36.17	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
3960	-36.19	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
3961	-36.19	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
3962	-36.2	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
3963	-36.22	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3964	-36.23	kd	CGS001-8807	IL18RAP	CD molecules			
3965	-36.23	oe	ccsbBroad304_05821	ANXA1	Annexins			
3966	-36.24	kd	CGS001-8805	TRIM24	TIF1 family			
3967	-36.26	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
3968	-36.26	kd	CGS001-91304	C19ORF6	-			
3969	-36.27	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
3970	-36.27	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3971	-36.32	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
3972	-36.35	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
3973	-36.4	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
3974	-36.43	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
3975	-36.44	kd	CGS001-896	CCND3	-			
3976	-36.51	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
3977	-36.53	oe	ccsbBroad304_00665	GOT1	-			
3978	-36.55	kd	CGS001-8833	GMPS	-			
3979	-36.59	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
3980	-36.61	kd	CGS001-10672	GNA13	-			
3981	-36.62	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
3982	-36.62	kd	CGS001-790	CAD	-			
3983	-36.63	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
3984	-36.66	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
3985	-36.67	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
3986	-36.68	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
3987	-36.72	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
3988	-36.78	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3989	-36.81	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
3990	-36.82	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
3991	-36.82	kd	CGS001-384	ARG2	Arginase			
3992	-36.86	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
3993	-36.87	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
3994	-36.88	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
3995	-36.88	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3996	-36.91	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
3997	-36.92	oe	ccsbBroad304_04379	LZIC	-			
3998	-36.92	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
3999	-36.94	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
4000	-36.97	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
4001	-37.06	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
4002	-37.07	oe	ccsbBroad304_01754	UCK2	-			
4003	-37.08	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
4004	-37.08	oe	ccsbBroad304_00551	FECH	-			
4005	-37.11	oe	ccsbBroad304_08217	SCCPDH	-			
4006	-37.11	kd	CGS001-1154	CISH	SH2 domain containing			
4007	-37.14	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
4008	-37.15	kd	CGS001-7185	TRAF1	-			
4009	-37.17	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
4010	-37.18	oe	ccsbBroad304_02668	PNKP	-			
4011	-37.2	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
4012	-37.21	kd	CGS001-1854	DUT	-			
4013	-37.25	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
4014	-37.25	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
4015	-37.26	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
4016	-37.26	kd	CGS001-338	APOB	Apolipoproteins			
4017	-37.27	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
4018	-37.28	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
4019	-37.29	kd	CGS001-3046	HBE1	-			
4020	-37.32	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
4021	-37.33	oe	ccsbBroad304_01654	TCTA	-			
4022	-37.33	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
4023	-37.33	kd	CGS001-8531	CSDA	-			
4024	-37.34	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
4025	-37.37	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
4026	-37.4	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
4027	-37.42	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
4028	-37.43	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
4029	-37.45	oe	ccsbBroad304_00809	HUS1	-			
4030	-37.48	oe	ccsbBroad304_07080	TM7SF2	-			
4031	-37.52	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4032	-37.52	kd	CGS001-2077	ERF	ETS Transcription Factors			
4033	-37.53	oe	ccsbBroad304_00854	IL8	-			
4034	-37.53	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
4035	-37.55	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
4036	-37.55	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
4037	-37.57	kd	CGS001-4811	NID1	-			
4038	-37.58	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
4039	-37.58	kd	CGS001-3065	HDAC1	Histone deacetylases			
4040	-37.59	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
4041	-37.63	oe	ccsbBroad304_02218	IKBKE	IKK family			
4042	-37.64	oe	ccsbBroad304_00795	HSF2	-			
4043	-37.65	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
4044	-37.68	kd	CGS001-3995	FADS3	Fatty acid desaturases			
4045	-37.68	oe	ccsbBroad304_13903	MTAP	-			
4046	-37.69	kd	CGS001-6119	RPA3	-			
4047	-37.7	cc		DNA Replication LOF	-			
4048	-37.71	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
4049	-37.71	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
4050	-37.75	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
4051	-37.75	kd	CGS001-25836	NIPBL	-			
4052	-37.76	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4053	-37.78	kd	CGS001-4594	MUT	-			
4054	-37.79	kd	CGS001-64781	CERK	Ceramide kinase			
4055	-37.84	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
4056	-37.84	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
4057	-37.87	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
4058	-37.87	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
4059	-37.88	oe	ccsbBroad304_02415	TUBB3	Tubulins			
4060	-37.88	kd	CGS001-29982	NRBF2	-			
4061	-37.9	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
4062	-37.93	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
4063	-37.96	kd	CGS001-9813	KIAA0494	-			
4064	-37.99	kd	CGS001-2109	ETFB	-			
4065	-38.02	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
4066	-38.05	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
4067	-38.05	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
4068	-38.09	oe	ccsbBroad304_00376	CSK	Csk family			
4069	-38.1	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
4070	-38.13	kd	CGS001-6364	CCL20	Chemokine ligands			
4071	-38.15	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
4072	-38.16	kd	CGS001-7001	PRDX2	-			
4073	-38.18	kd	CGS001-5170	PDPK1	PDK1 family			
4074	-38.19	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
4075	-38.21	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
4076	-38.21	kd	CGS001-6832	SUPV3L1	-			
4077	-38.24	kd	CGS001-8624	PSMG1	-			
4078	-38.28	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
4079	-38.29	oe	ccsbBroad304_01662	TFDP2	-			
4080	-38.36	kd	CGS001-4830	NME1	-			
4081	-38.37	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
4082	-38.39	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
4083	-38.4	kd	CGS001-822	CAPG	-			
4084	-38.41	oe	ccsbBroad304_06424	IFI16	-			
4085	-38.41	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
4086	-38.44	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
4087	-38.46	kd	CGS001-55644	OSGEP	-			
4088	-38.46	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
4089	-38.47	oe	ccsbBroad304_02485	STAMBP	-			
4090	-38.51	cc		Calmodulin antagonist	-			
4091	-38.51	oe	ccsbBroad304_02285	MED6	-			
4092	-38.56	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
4093	-38.58	kd	CGS001-3456	IFNB1	Interferons			
4094	-38.6	kd	CGS001-3895	KTN1	-			
4095	-38.64	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4096	-38.64	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
4097	-38.65	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
4098	-38.66	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
4099	-38.68	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
4100	-38.69	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
4101	-38.74	oe	ccsbBroad304_02349	MPHOSPH9	-			
4102	-38.76	kd	CGS001-637	BID	Endogenous ligands			
4103	-38.79	kd	CGS001-5914	RARA	Retinoic acid receptors			
4104	-38.79	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
4105	-38.82	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
4106	-38.82	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
4107	-38.82	oe	ccsbBroad304_02955	MYCBP	-			
4108	-38.83	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4109	-38.85	kd	CGS001-5934	RBL2	-			
4110	-38.88	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
4111	-38.89	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4112	-38.9	oe	ccsbBroad304_02432	IFI30	-			
4113	-38.9	oe	ccsbBroad304_03089	PACSIN3	-			
4114	-38.91	kd	CGS001-56993	TOMM22	-			
4115	-38.93	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
4116	-38.95	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
4117	-38.97	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
4118	-38.99	oe	ccsbBroad304_01257	PPOX	-			
4119	-38.99	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
4120	-39	oe	ccsbBroad304_05948	CCND2	-			
4121	-39.04	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
4122	-39.05	cc		Potassium channel activator	-			
4123	-39.07	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
4124	-39.13	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
4125	-39.14	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
4126	-39.14	kd	CGS001-10491	CRTAP	-			
4127	-39.15	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
4128	-39.15	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
4129	-39.18	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
4130	-39.25	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
4131	-39.26	oe	ccsbBroad304_06235	G6PD	-			
4132	-39.26	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
4133	-39.28	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
4134	-39.3	kd	CGS001-3939	LDHA	-			
4135	-39.31	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
4136	-39.31	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
4137	-39.33	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
4138	-39.35	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
4139	-39.4	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
4140	-39.4	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
4141	-39.42	kd	CGS001-84722	PSRC1	-			
4142	-39.43	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
4143	-39.43	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
4144	-39.45	oe	ccsbBroad304_03573	BRF2	-			
4145	-39.45	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
4146	-39.45	kd	CGS001-6774	STAT3	SH2 domain containing			
4147	-39.45	kd	CGS001-124583	CANT1	-			
4148	-39.46	kd	CGS001-10298	PAK4	PAKB subfamily			
4149	-39.48	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
4150	-39.48	kd	CGS001-59286	UBL5	-			
4151	-39.49	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
4152	-39.49	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
4153	-39.52	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
4154	-39.55	oe	ccsbBroad304_02579	YWHAQ	-			
4155	-39.56	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
4156	-39.58	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
4157	-39.59	oe	ccsbBroad304_01395	RFX5	-			
4158	-39.59	kd	CGS001-2002	ELK1	ETS Transcription Factors			
4159	-39.6	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
4160	-39.61	oe	ccsbBroad304_06449	ILF3	-			
4161	-39.61	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
4162	-39.62	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4163	-39.63	kd	CGS001-55810	FOXJ2	Forkhead boxes			
4164	-39.66	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4165	-39.66	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
4166	-39.7	oe	ccsbBroad304_00115	ASPH	-			
4167	-39.7	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4168	-39.71	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
4169	-39.72	oe	ccsbBroad304_00550	FDXR	-			
4170	-39.72	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
4171	-39.72	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
4172	-39.74	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
4173	-39.75	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
4174	-39.77	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
4175	-39.79	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
4176	-39.81	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
4177	-39.83	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
4178	-39.86	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
4179	-39.87	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
4180	-39.87	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4181	-39.92	kd	CGS001-5164	PDK2	PDHK family			
4182	-39.94	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
4183	-39.97	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
4184	-39.97	oe	ccsbBroad304_08888	ACD	-			
4185	-39.97	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
4186	-39.97	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
4187	-40.03	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
4188	-40.03	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
4189	-40.04	kd	CGS001-3155	HMGCL	-			
4190	-40.05	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
4191	-40.06	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
4192	-40.12	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
4193	-40.15	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
4194	-40.18	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
4195	-40.19	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
4196	-40.25	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
4197	-40.27	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4198	-40.27	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
4199	-40.28	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
4200	-40.29	oe	ccsbBroad304_02845	PRPF6	-			
4201	-40.29	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
4202	-40.3	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
4203	-40.4	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
4204	-40.45	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
4205	-40.45	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
4206	-40.46	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
4207	-40.48	oe	ccsbBroad304_06745	PNN	-			
4208	-40.48	kd	CGS001-23196	FAM120A	-			
4209	-40.52	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
4210	-40.55	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
4211	-40.57	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
4212	-40.61	oe	ccsbBroad304_02414	IRF9	-			
4213	-40.61	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
4214	-40.62	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
4215	-40.63	kd	CGS001-3690	ITGB3	Integrins			
4216	-40.66	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
4217	-40.73	cc		Glycogen synthase kinase inhibitor	-			
4218	-40.73	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
4219	-40.76	kd	CGS001-6469	SHH	-			
4220	-40.78	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
4221	-40.78	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
4222	-40.81	oe	ccsbBroad304_04406	PLA2G12B	-			
4223	-40.84	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
4224	-40.92	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
4225	-40.97	kd	CGS001-6519	SLC3A1	SLC3 family			
4226	-40.97	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
4227	-40.99	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
4228	-41	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
4229	-41.01	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
4230	-41.04	kd	CGS001-55206	SBNO1	-			
4231	-41.14	kd	CGS001-2155	F7	Chymotrypsin			
4232	-41.15	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
4233	-41.16	oe	ccsbBroad304_00238	CCNE1	-			
4234	-41.2	oe	ccsbBroad304_02143	CNOT8	-			
4235	-41.22	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
4236	-41.3	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
4237	-41.36	kd	CGS001-11004	KIF2C	Kinesins			
4238	-41.39	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
4239	-41.4	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
4240	-41.45	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4241	-41.46	cc		HSP inhibitor	-			
4242	-41.47	oe	ccsbBroad304_08605	PBK	TOPK family			
4243	-41.47	kd	CGS001-114609	TIRAP	-			
4244	-41.48	kd	CGS001-23047	PDS5B	-			
4245	-41.49	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
4246	-41.5	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
4247	-41.52	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
4248	-41.55	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4249	-41.56	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
4250	-41.56	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
4251	-41.57	cc		Dihydrofolate reductase inhibitor	-			
4252	-41.65	kd	CGS001-6601	SMARCC2	-			
4253	-41.67	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
4254	-41.76	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
4255	-41.77	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
4256	-41.78	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
4257	-41.79	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
4258	-41.83	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
4259	-41.85	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
4260	-41.85	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
4261	-41.86	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
4262	-41.9	oe	ccsbBroad304_07548	TSSC4	-			
4263	-41.9	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
4264	-41.95	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
4265	-41.95	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
4266	-41.97	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
4267	-42.01	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
4268	-42.02	oe	ccsbBroad304_08660	SMARCAD1	-			
4269	-42.02	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
4270	-42.04	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
4271	-42.06	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
4272	-42.09	oe	ccsbBroad304_08709	SCYL3	-			
4273	-42.09	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
4274	-42.1	oe	ccsbBroad304_06226	FTL	-			
4275	-42.15	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
4276	-42.33	kd	CGS001-7086	TKT	-			
4277	-42.35	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
4278	-42.37	kd	CGS001-64333	ARHGAP9	Rho GTPase activating proteins			
4279	-42.38	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
4280	-42.38	kd	CGS001-8649	LAMTOR3	-			
4281	-42.39	kd	CGS001-6599	SMARCC1	-			
4282	-42.4	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
4283	-42.41	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
4284	-42.41	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
4285	-42.41	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
4286	-42.43	oe	ccsbBroad304_07923	LSM5	-			
4287	-42.46	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
4288	-42.49	oe	ccsbBroad304_09833	SENP5	-			
4289	-42.52	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
4290	-42.53	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
4291	-42.54	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
4292	-42.55	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
4293	-42.58	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
4294	-42.59	kd	CGS001-3569	IL6	Interferons			
4295	-42.63	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4296	-42.64	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
4297	-42.65	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
4298	-42.69	cc		AHSP Pathway LOF	-			
4299	-42.7	oe	ccsbBroad304_03746	CDC42SE1	-			
4300	-42.7	kd	CGS001-64786	TBC1D15	-			
4301	-42.71	oe	ccsbBroad304_02831	SGK3	SGK family			
4302	-42.71	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
4303	-42.72	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
4304	-42.76	kd	CGS001-11315	PARK7	Parkinson disease			
4305	-42.79	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
4306	-42.8	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
4307	-42.81	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
4308	-42.81	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
4309	-42.82	oe	ccsbBroad304_01659	TERF1	-			
4310	-42.87	oe	ccsbBroad304_06645	NQO2	-			
4311	-42.88	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
4312	-42.88	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
4313	-42.9	kd	CGS001-54498	SMOX	-			
4314	-42.95	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4315	-42.97	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
4316	-42.97	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
4317	-43.01	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
4318	-43.04	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
4319	-43.05	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
4320	-43.05	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
4321	-43.06	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
4322	-43.09	cc		Mitogen activated protein kinases LOF	-			
4323	-43.1	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
4324	-43.11	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
4325	-43.12	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
4326	-43.13	oe	ccsbBroad304_01146	PARN	-			
4327	-43.17	kd	CGS001-58533	SNX6	Sorting nexins			
4328	-43.19	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
4329	-43.2	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4330	-43.24	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
4331	-43.25	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
4332	-43.25	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
4333	-43.25	kd	CGS001-29888	STRN4	WD repeat domain containing			
4334	-43.26	kd	CGS001-8772	FADD	-			
4335	-43.29	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
4336	-43.29	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
4337	-43.32	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
4338	-43.38	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
4339	-43.39	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
4340	-43.39	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
4341	-43.4	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
4342	-43.43	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
4343	-43.52	kd	CGS001-840	CASP7	Caspases			
4344	-43.53	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
4345	-43.53	kd	CGS001-9791	PTDSS1	-			
4346	-43.55	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
4347	-43.55	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
4348	-43.78	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
4349	-43.83	oe	ccsbBroad304_03917	RBKS	-			
4350	-43.87	oe	ccsbBroad304_02653	PRAF2	-			
4351	-43.91	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
4352	-43.93	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
4353	-43.95	kd	CGS001-23463	ICMT	-			
4354	-43.99	kd	CGS001-9415	FADS2	Fatty acid desaturases			
4355	-44	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
4356	-44.01	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
4357	-44.03	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
4358	-44.08	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
4359	-44.08	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
4360	-44.12	oe	ccsbBroad304_00615	GAPDH	-			
4361	-44.14	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4362	-44.16	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4363	-44.18	kd	CGS001-83933	HDAC10	Histone deacetylases			
4364	-44.19	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
4365	-44.24	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
4366	-44.29	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
4367	-44.31	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
4368	-44.45	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
4369	-44.46	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
4370	-44.46	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4371	-44.47	oe	ccsbBroad304_02738	RRS1	-			
4372	-44.52	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
4373	-44.52	kd	CGS001-9218	VAPA	-			
4374	-44.53	cc		Tricyclic antidepressant	-			
4375	-44.53	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
4376	-44.53	kd	CGS001-10827	FAM114A2	-			
4377	-44.6	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
4378	-44.62	oe	ccsbBroad304_00170	BNIP1	-			
4379	-44.63	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
4380	-44.64	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
4381	-44.64	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
4382	-44.67	oe	ccsbBroad304_02306	PQBP1	-			
4383	-44.67	oe	ccsbBroad304_09254	PAQR8	-			
4384	-44.67	kd	CGS001-8985	PLOD3	-			
4385	-44.71	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
4386	-44.71	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
4387	-44.71	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
4388	-44.75	kd	CGS001-1212	CLTB	-			
4389	-44.76	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
4390	-44.79	oe	ccsbBroad304_01855	NCOA4	-			
4391	-44.81	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
4392	-44.84	kd	CGS001-4176	MCM7	-			
4393	-44.86	oe	ccsbBroad304_07349	MAP7	-			
4394	-44.86	kd	CGS001-23650	TRIM29	-			
4395	-44.88	kd	CGS001-116931	MED12L	-			
4396	-44.92	kd	CGS001-2099	ESR1	Estrogen receptors			
4397	-44.98	kd	CGS001-23492	CBX7	-			
4398	-45.01	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4399	-45.01	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4400	-45.02	oe	ccsbBroad304_02399	TNIP1	-			
4401	-45.02	oe	ccsbBroad304_01923	UXT	-			
4402	-45.04	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
4403	-45.08	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
4404	-45.14	oe	ccsbBroad304_03739	NRIP3	-			
4405	-45.15	oe	ccsbBroad304_04544	RCCD1	-			
4406	-45.17	kd	CGS001-1632	ECI1	-			
4407	-45.18	oe	ccsbBroad304_00964	SMAD7	SMADs			
4408	-45.19	kd	CGS001-7982	ST7	-			
4409	-45.19	kd	CGS001-25797	QPCT	Aminopeptidase Y			
4410	-45.25	kd	CGS001-7039	TGFA	-			
4411	-45.25	kd	CGS001-23242	COBL	-			
4412	-45.4	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
4413	-45.4	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
4414	-45.41	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
4415	-45.44	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
4416	-45.44	kd	CGS001-6944	VPS72	-			
4417	-45.45	oe	ccsbBroad304_03173	TMED7	-			
4418	-45.45	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
4419	-45.47	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
4420	-45.49	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
4421	-45.5	oe	ccsbBroad304_02822	ARFIP2	-			
4422	-45.51	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
4423	-45.54	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
4424	-45.55	oe	ccsbBroad304_00420	DAP	-			
4425	-45.6	oe	ccsbBroad304_05745	CD24	CD molecules			
4426	-45.61	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
4427	-45.62	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
4428	-45.63	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4429	-45.63	kd	CGS001-375449	MAST4	MAST family			
4430	-45.7	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
4431	-45.72	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
4432	-45.72	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
4433	-45.75	oe	ccsbBroad304_07252	DGKZ	-			
4434	-45.78	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
4435	-45.78	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
4436	-45.85	oe	ccsbBroad304_08878	METTL4	-			
4437	-45.85	kd	CGS001-51720	UIMC1	-			
4438	-45.86	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
4439	-45.87	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
4440	-45.89	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
4441	-45.92	kd	CGS001-11325	DDX42	DEAD-boxes			
4442	-45.98	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
4443	-45.99	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
4444	-45.99	kd	CGS001-47	ACLY	-			
4445	-46	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
4446	-46.03	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
4447	-46.04	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
4448	-46.07	kd	CGS001-5188	PET112	-			
4449	-46.08	kd	CGS001-4849	CNOT3	-			
4450	-46.09	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
4451	-46.11	kd	CGS001-4758	NEU1	-			
4452	-46.15	oe	ccsbBroad304_02278	THRAP3	-			
4453	-46.17	oe	ccsbBroad304_06287	GM2A	-			
4454	-46.19	oe	ccsbBroad304_06535	LPL	-			
4455	-46.2	cc		Aminoacyl tRNA synthetases class II LOF	-			
4456	-46.24	oe	ccsbBroad304_00472	EBF1	-			
4457	-46.24	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
4458	-46.24	kd	CGS001-10468	FST	-			
4459	-46.26	kd	CGS001-6194	RPS6	S ribosomal proteins			
4460	-46.27	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
4461	-46.28	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
4462	-46.28	kd	CGS001-694	BTG1	-			
4463	-46.29	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
4464	-46.3	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
4465	-46.32	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
4466	-46.33	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
4467	-46.35	oe	ccsbBroad304_09358	MAPK1IP1L	-			
4468	-46.35	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
4469	-46.37	oe	ccsbBroad304_13891	LCK	Src family			
4470	-46.38	oe	ccsbBroad304_06870	RNH1	-			
4471	-46.42	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
4472	-46.44	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
4473	-46.46	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
4474	-46.49	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4475	-46.52	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
4476	-46.53	kd	CGS001-85480	TSLP	-			
4477	-46.6	oe	ccsbBroad304_02092	SYNGR3	-			
4478	-46.6	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
4479	-46.63	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
4480	-46.65	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
4481	-46.66	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
4482	-46.67	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
4483	-46.71	oe	ccsbBroad304_02554	TRAFD1	-			
4484	-46.73	oe	ccsbBroad304_00975	MAT2A	-			
4485	-46.74	oe	ccsbBroad304_08365	CYCS	-			
4486	-46.75	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
4487	-46.78	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
4488	-46.8	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
4489	-46.85	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
4490	-46.93	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
4491	-46.95	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
4492	-46.95	kd	CGS001-949	SCARB1	-			
4493	-46.95	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
4494	-46.99	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4495	-47.02	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
4496	-47.15	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
4497	-47.16	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
4498	-47.17	kd	CGS001-63948	DMRTB1	-			
4499	-47.18	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
4500	-47.21	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
4501	-47.24	cc		Protein synthesis inhibitor	-			
4502	-47.25	oe	ccsbBroad304_05907	BUB1B	Bub family			
4503	-47.26	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
4504	-47.37	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
4505	-47.37	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
4506	-47.38	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
4507	-47.4	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
4508	-47.5	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
4509	-47.5	kd	CGS001-2073	ERCC5	-			
4510	-47.54	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
4511	-47.54	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
4512	-47.54	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
4513	-47.59	cc		Bromodomain Inhibitor	-			
4514	-47.61	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
4515	-47.63	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
4516	-47.72	kd	CGS001-1962	EHHADH	-			
4517	-47.72	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
4518	-47.74	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
4519	-47.75	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
4520	-47.76	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
4521	-47.76	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
4522	-47.79	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
4523	-47.8	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
4524	-47.8	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
4525	-47.81	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
4526	-47.87	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
4527	-47.88	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
4528	-47.91	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
4529	-47.98	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
4530	-47.99	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
4531	-47.99	kd	CGS001-4300	MLLT3	-			
4532	-48.05	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
4533	-48.05	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
4534	-48.06	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
4535	-48.06	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
4536	-48.08	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
4537	-48.12	kd	CGS001-5565	PRKAB2	AMPK subfamily			
4538	-48.14	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
4539	-48.16	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
4540	-48.17	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
4541	-48.24	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
4542	-48.25	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
4543	-48.25	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
4544	-48.26	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
4545	-48.35	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
4546	-48.35	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
4547	-48.36	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
4548	-48.38	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
4549	-48.41	oe	ccsbBroad304_00987	MCM3	-			
4550	-48.42	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4551	-48.44	oe	ccsbBroad304_03812	PBXIP1	-			
4552	-48.47	oe	ccsbBroad304_07337	TAF1B	-			
4553	-48.47	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
4554	-48.53	kd	CGS001-6643	SNX2	Sorting nexins			
4555	-48.55	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
4556	-48.57	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
4557	-48.6	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
4558	-48.61	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
4559	-48.64	kd	CGS001-30001	ERO1L	-			
4560	-48.67	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
4561	-48.74	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
4562	-48.78	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
4563	-48.79	oe	ccsbBroad304_05902	BNIP3	-			
4564	-48.84	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
4565	-48.85	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
4566	-48.86	kd	CGS001-7771	ZFP112	-			
4567	-48.91	kd	CGS001-64170	CARD9	-			
4568	-48.92	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
4569	-49.01	kd	CGS001-55278	QRSL1	-			
4570	-49.04	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
4571	-49.07	kd	CGS001-60493	FASTKD5	-			
4572	-49.08	kd	CGS001-9374	PPT2	-			
4573	-49.12	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
4574	-49.16	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
4575	-49.17	cc		PRD class homeoboxes and psudogenes LOF	-			
4576	-49.17	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
4577	-49.2	oe	ccsbBroad304_02438	FAM3C	-			
4578	-49.22	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
4579	-49.22	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
4580	-49.25	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
4581	-49.27	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
4582	-49.27	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
4583	-49.28	kd	CGS001-22921	MSRB2	-			
4584	-49.33	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
4585	-49.33	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
4586	-49.35	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
4587	-49.38	cc		Histone deacetylases LOF	-			
4588	-49.39	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4589	-49.44	kd	CGS001-5362	PLXNA2	Plexins			
4590	-49.49	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
4591	-49.52	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
4592	-49.53	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
4593	-49.54	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
4594	-49.57	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
4595	-49.6	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4596	-49.6	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
4597	-49.62	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
4598	-49.62	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
4599	-49.64	cc		T-type calcium channel blocker	-			
4600	-49.69	cc		G2 M Checkpoint LOF	-			
4601	-49.7	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
4602	-49.71	kd	CGS001-23451	SF3B1	-			
4603	-49.79	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
4604	-49.82	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
4605	-49.82	oe	ccsbBroad304_01641	TAF13	-			
4606	-49.83	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
4607	-49.83	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
4608	-49.84	kd	CGS001-8872	CDC123	-			
4609	-49.88	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
4610	-49.97	cc		Phospholipases GOF	-			
4611	-49.98	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
4612	-50.07	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
4613	-50.11	kd	CGS001-3685	ITGAV	Integrins			
4614	-50.14	kd	CGS001-55634	ZNF673	-			
4615	-50.14	kd	CGS001-472	ATM	Other PIKK family kinases			
4616	-50.23	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
4617	-50.26	oe	ccsbBroad304_03311	EVL	-			
4618	-50.26	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
4619	-50.26	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
4620	-50.27	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
4621	-50.3	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
4622	-50.31	oe	ccsbBroad304_04490	RSPH1	-			
4623	-50.43	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
4624	-50.5	kd	CGS001-11014	KDELR2	-			
4625	-50.51	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4626	-50.54	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
4627	-50.57	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
4628	-50.58	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
4629	-50.61	kd	CGS001-5338	PLD2	Hydrolases			
4630	-50.62	oe	ccsbBroad304_00818	IDH3A	-			
4631	-50.68	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
4632	-50.7	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
4633	-50.71	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
4634	-50.74	kd	CGS001-1493	CTLA4	CD molecules			
4635	-50.76	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
4636	-50.87	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
4637	-50.87	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
4638	-50.98	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
4639	-51	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
4640	-51.03	cc		Wnt family GOF	-			
4641	-51.11	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
4642	-51.12	kd	CGS001-53343	NUDT9	Nudix motif containing			
4643	-51.13	cc		KCNJ11 modulator	-			
4644	-51.16	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
4645	-51.18	oe	ccsbBroad304_05528	TICAM2	-			
4646	-51.18	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
4647	-51.21	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
4648	-51.24	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
4649	-51.26	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
4650	-51.3	kd	CGS001-5682	PSMA1	Proteasome subunits			
4651	-51.31	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
4652	-51.34	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
4653	-51.44	kd	CGS001-4125	MAN2B1	-			
4654	-51.45	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
4655	-51.47	kd	CGS001-63933	CCDC90A	-			
4656	-51.51	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
4657	-51.55	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
4658	-51.57	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
4659	-51.58	kd	CGS001-6233	RPS27A	S ribosomal proteins			
4660	-51.59	oe	ccsbBroad304_08339	CMPK1	-			
4661	-51.6	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
4662	-51.64	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
4663	-51.7	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
4664	-51.8	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4665	-51.8	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
4666	-51.84	oe	ccsbBroad304_07277	RTCD1	-			
4667	-51.87	oe	ccsbBroad304_00223	CASP9	Caspases			
4668	-51.89	oe	ccsbBroad304_07024	SYK	Syk family			
4669	-51.89	kd	CGS001-2072	ERCC4	-			
4670	-51.92	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
4671	-51.92	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4672	-51.97	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
4673	-52.13	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
4674	-52.14	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
4675	-52.21	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
4676	-52.21	oe	ccsbBroad304_00529	F3	CD molecules			
4677	-52.21	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
4678	-52.22	kd	CGS001-28960	DCPS	-			
4679	-52.26	kd	CGS001-3281	HSBP1	-			
4680	-52.27	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
4681	-52.28	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
4682	-52.28	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
4683	-52.29	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
4684	-52.3	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
4685	-52.34	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
4686	-52.38	kd	CGS001-51741	WWOX	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4687	-52.39	oe	ccsbBroad304_01483	SAT1	-			
4688	-52.41	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
4689	-52.43	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
4690	-52.45	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
4691	-52.45	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
4692	-52.45	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
4693	-52.52	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
4694	-52.53	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
4695	-52.53	kd	CGS001-8634	RTCD1	-			
4696	-52.54	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4697	-52.56	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
4698	-52.6	kd	CGS001-7316	UBC	-			
4699	-52.62	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
4700	-52.64	kd	CGS001-11157	LSM6	-			
4701	-52.65	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
4702	-52.72	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
4703	-52.75	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
4704	-52.75	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4705	-52.76	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
4706	-52.78	oe	ccsbBroad304_06783	LGMN	Legumain			
4707	-52.82	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4708	-52.89	oe	ccsbBroad304_00394	CTSD	Cathepsins			
4709	-52.89	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
4710	-52.93	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
4711	-52.97	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
4712	-52.98	oe	ccsbBroad304_08993	DHDDS	-			
4713	-53.01	kd	CGS001-3579	CXCR2	Chemokine receptors			
4714	-53.06	oe	ccsbBroad304_00009	ACLY	-			
4715	-53.07	kd	CGS001-10494	STK25	YSK subfamily			
4716	-53.09	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
4717	-53.11	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
4718	-53.16	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
4719	-53.16	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
4720	-53.17	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
4721	-53.26	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
4722	-53.27	kd	CGS001-5982	RFC2	ATPases / AAA-type			
4723	-53.31	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
4724	-53.35	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
4725	-53.37	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
4726	-53.45	oe	ccsbBroad304_14020	SH3BP5	-			
4727	-53.46	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
4728	-53.46	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
4729	-53.47	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
4730	-53.48	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
4731	-53.49	kd	CGS001-116443	GRIN3A	Glutamate receptors			
4732	-53.52	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
4733	-53.52	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
4734	-53.58	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
4735	-53.58	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
4736	-53.59	kd	CGS001-6118	RPA2	-			
4737	-53.6	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
4738	-53.6	kd	CGS001-2783	GNB2	WD repeat domain containing			
4739	-53.69	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
4740	-53.71	kd	CGS001-26128	KIAA1279	-			
4741	-53.71	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
4742	-53.72	kd	CGS001-5202	PFDN2	-			
4743	-53.82	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
4744	-53.86	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
4745	-53.87	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
4746	-53.98	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
4747	-53.98	kd	CGS001-6464	SHC1	SH2 domain containing			
4748	-53.99	cc		HMGCR inhibitor	-			
4749	-54.06	oe	ccsbBroad304_02398	LANCL1	-			
4750	-54.08	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
4751	-54.08	kd	CGS001-87	ACTN1	EF-hand domain containing			
4752	-54.11	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
4753	-54.14	kd	CGS001-3956	LGALS1	Endogenous ligands			
4754	-54.18	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
4755	-54.2	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
4756	-54.22	oe	ccsbBroad304_01205	PIN1	-			
4757	-54.22	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
4758	-54.26	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
4759	-54.26	kd	CGS001-29916	SNX11	Sorting nexins			
4760	-54.29	kd	CGS001-7913	DEK	-			
4761	-54.33	kd	CGS001-4864	NPC1	-			
4762	-54.43	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
4763	-54.51	kd	CGS001-51271	UBAP1	-			
4764	-54.52	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
4765	-54.55	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
4766	-54.58	kd	CGS001-7466	WFS1	-			
4767	-54.62	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
4768	-54.75	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
4769	-54.75	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
4770	-54.78	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
4771	-54.81	oe	ccsbBroad304_14047	TACC3	-			
4772	-54.83	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
4773	-54.84	oe	ccsbBroad304_08104	MED4	-			
4774	-54.84	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
4775	-54.84	kd	CGS001-7840	ALMS1	-			
4776	-54.86	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
4777	-54.91	oe	ccsbBroad304_02864	PRDX5	-			
4778	-54.91	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
4779	-54.91	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
4780	-54.94	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
4781	-54.97	oe	ccsbBroad304_07861	COBL	-			
4782	-55.01	kd	CGS001-23118	TAB2	-			
4783	-55.03	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
4784	-55.05	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
4785	-55.08	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4786	-55.09	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
4787	-55.1	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
4788	-55.14	oe	ccsbBroad304_05936	CASP2	Caspases			
4789	-55.16	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
4790	-55.18	kd	CGS001-5827	PXMP2	-			
4791	-55.19	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
4792	-55.24	kd	CGS001-10607	TBL3	WD repeat domain containing			
4793	-55.26	kd	CGS001-2621	GAS6	-			
4794	-55.27	kd	CGS001-1879	EBF1	-			
4795	-55.3	kd	CGS001-9441	MED26	-			
4796	-55.36	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
4797	-55.37	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
4798	-55.37	kd	CGS001-10943	MSL3	-			
4799	-55.48	oe	ccsbBroad304_07287	HYAL2	-			
4800	-55.49	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
4801	-55.71	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4802	-55.73	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
4803	-55.77	oe	ccsbBroad304_07178	ZFP112	-			
4804	-55.78	oe	ccsbBroad304_01183	PGD	-			
4805	-55.79	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
4806	-55.83	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
4807	-55.9	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
4808	-55.91	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
4809	-55.93	oe	ccsbBroad304_03808	ERGIC1	-			
4810	-55.95	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
4811	-55.95	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
4812	-55.97	oe	ccsbBroad304_06888	RPN1	-			
4813	-55.99	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
4814	-56.03	kd	CGS001-2356	FPGS	-			
4815	-56.04	oe	ccsbBroad304_01948	GAS7	-			
4816	-56.05	kd	CGS001-29937	NENF	-			
4817	-56.06	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
4818	-56.08	oe	ccsbBroad304_09396	TIRAP	-			
4819	-56.13	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
4820	-56.14	kd	CGS001-9156	EXO1	-			
4821	-56.15	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
4822	-56.15	kd	CGS001-8804	CREG1	-			
4823	-56.18	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
4824	-56.25	kd	CGS001-11243	PMF1	-			
4825	-56.29	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
4826	-56.3	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4827	-56.33	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
4828	-56.34	kd	CGS001-190	NR0B1	DAX-like receptors			
4829	-56.35	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
4830	-56.36	oe	ccsbBroad304_04752	IKBIP	-			
4831	-56.39	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
4832	-56.42	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
4833	-56.43	kd	CGS001-23743	BHMT2	-			
4834	-56.45	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
4835	-56.5	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
4836	-56.51	cc		TGF beta receptor inhibitor	-			
4837	-56.57	kd	CGS001-433	ASGR2	C-type lectin domain containing			
4838	-56.62	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
4839	-56.64	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
4840	-56.67	kd	CGS001-10412	NSA2	-			
4841	-56.68	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
4842	-56.7	oe	ccsbBroad304_08055	ATP5S	-			
4843	-56.7	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
4844	-56.73	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
4845	-56.78	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
4846	-56.79	kd	CGS001-7018	TF	-			
4847	-56.82	kd	CGS001-403	ARL3	ADP-ribosylation factors			
4848	-56.87	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4849	-56.88	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
4850	-56.88	kd	CGS001-388677	NOTCH2NL	-			
4851	-56.89	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
4852	-56.89	kd	CGS001-9817	KEAP1	Kelch-like proteins			
4853	-56.94	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
4854	-56.95	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
4855	-56.97	kd	CGS001-7158	TP53BP1	-			
4856	-57.01	oe	ccsbBroad304_06180	ESD	-			
4857	-57.07	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4858	-57.09	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
4859	-57.12	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
4860	-57.13	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
4861	-57.14	kd	CGS001-10312	TCIRG1	ATPases / V-type			
4862	-57.19	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
4863	-57.19	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
4864	-57.19	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
4865	-57.19	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
4866	-57.19	kd	CGS001-9455	HOMER2	-			
4867	-57.2	oe	ccsbBroad304_00398	CTSL2	-			
4868	-57.2	kd	CGS001-84515	MCM8	-			
4869	-57.22	kd	CGS001-7078	TIMP3	-			
4870	-57.25	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
4871	-57.26	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
4872	-57.3	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
4873	-57.32	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
4874	-57.33	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
4875	-57.43	oe	ccsbBroad304_08879	CASD1	-			
4876	-57.45	kd	CGS001-6500	SKP1	-			
4877	-57.46	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
4878	-57.48	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
4879	-57.49	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
4880	-57.57	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
4881	-57.58	oe	ccsbBroad304_03950	ATG3	-			
4882	-57.63	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
4883	-57.65	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
4884	-57.69	kd	CGS001-2235	FECH	-			
4885	-57.77	oe	ccsbBroad304_07515	GFPT2	-			
4886	-57.79	kd	CGS001-10318	TNIP1	-			
4887	-57.84	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4888	-57.85	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
4889	-57.91	kd	CGS001-3460	IFNGR2	Interferon receptor family			
4890	-57.92	oe	ccsbBroad304_00171	BNIP3L	-			
4891	-57.93	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
4892	-57.94	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
4893	-57.95	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
4894	-57.98	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
4895	-57.99	kd	CGS001-5479	PPIB	-			
4896	-58.03	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
4897	-58.04	oe	ccsbBroad304_02219	MORF4L2	-			
4898	-58.07	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
4899	-58.1	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4900	-58.19	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
4901	-58.19	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
4902	-58.23	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
4903	-58.23	kd	CGS001-9988	DMTF1	-			
4904	-58.24	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
4905	-58.24	kd	CGS001-4439	MSH5	-			
4906	-58.25	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
4907	-58.26	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
4908	-58.3	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
4909	-58.33	oe	ccsbBroad304_03122	RHOD	-			
4910	-58.34	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
4911	-58.34	kd	CGS001-664	BNIP3	-			
4912	-58.4	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
4913	-58.41	kd	CGS001-1490	CTGF	-			
4914	-58.44	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
4915	-58.48	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
4916	-58.5	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
4917	-58.55	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
4918	-58.58	oe	ccsbBroad304_01663	TFF2	-			
4919	-58.6	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
4920	-58.62	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
4921	-58.64	oe	ccsbBroad304_06565	MB	-			
4922	-58.69	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
4923	-58.77	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
4924	-58.77	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
4925	-58.77	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4926	-58.77	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4927	-58.8	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
4928	-58.82	kd	CGS001-3476	IGBP1	-			
4929	-58.83	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
4930	-58.85	kd	CGS001-29911	HOOK2	-			
4931	-58.88	cc		SRY LOF	-			
4932	-58.9	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
4933	-58.91	kd	CGS001-4507	MTAP	-			
4934	-58.91	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
4935	-58.92	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
4936	-58.92	kd	CGS001-150280	HORMAD2	-			
4937	-58.93	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
4938	-58.97	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
4939	-58.99	oe	ccsbBroad304_00210	CALR	-			
4940	-58.99	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
4941	-59.01	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
4942	-59.02	kd	CGS001-85004	RERG	-			
4943	-59.11	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
4944	-59.15	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4945	-59.21	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
4946	-59.25	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
4947	-59.26	kd	CGS001-2821	GPI	-			
4948	-59.33	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
4949	-59.47	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
4950	-59.5	oe	ccsbBroad304_03428	EXOSC4	-			
4951	-59.57	oe	ccsbBroad304_00794	HSF1	-			
4952	-59.58	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
4953	-59.59	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
4954	-59.63	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
4955	-59.67	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
4956	-59.7	kd	CGS001-11044	PAPD7	-			
4957	-59.71	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
4958	-59.72	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
4959	-59.74	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
4960	-59.74	kd	CGS001-5498	PPOX	-			
4961	-59.75	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4962	-59.78	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
4963	-59.84	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
4964	-59.84	kd	CGS001-475	ATOX1	-			
4965	-59.9	cc		Norepinephrine reuptake inhibitor	-			
4966	-59.91	kd	CGS001-7360	UGP2	-			
4967	-59.97	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
4968	-59.99	cc		Retinoid receptor agonist	-			
4969	-59.99	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
4970	-59.99	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
4971	-60.01	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
4972	-60.04	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
4973	-60.04	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
4974	-60.09	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
4975	-60.2	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
4976	-60.23	kd	CGS001-114785	MBD6	-			
4977	-60.23	kd	CGS001-55165	CEP55	-			
4978	-60.28	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
4979	-60.31	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
4980	-60.37	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
4981	-60.38	kd	CGS001-147179	WIPF2	-			
4982	-60.42	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
4983	-60.51	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
4984	-60.56	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
4985	-60.7	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
4986	-60.72	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
4987	-60.76	kd	CGS001-5198	PFAS	-			
4988	-60.8	oe	ccsbBroad304_04465	RERG	-			
4989	-60.83	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
4990	-60.95	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
4991	-61.01	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
4992	-61.05	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
4993	-61.07	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
4994	-61.1	kd	CGS001-1155	TBCB	-			
4995	-61.11	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
4996	-61.12	cc		Akt Signaling GOF	-			
4997	-61.17	kd	CGS001-54555	DDX49	DEAD-boxes			
4998	-61.19	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4999	-61.27	oe	ccsbBroad304_00174	BRAF	RAF family			
5000	-61.28	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
5001	-61.31	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5002	-61.33	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
5003	-61.35	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
5004	-61.44	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
5005	-61.45	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
5006	-61.47	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
5007	-61.57	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
5008	-61.57	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
5009	-61.59	kd	CGS001-83729	INHBE	-			
5010	-61.63	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
5011	-61.69	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
5012	-61.71	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
5013	-61.74	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
5014	-61.74	oe	ccsbBroad304_01985	EIF3H	-			
5015	-61.74	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
5016	-61.75	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
5017	-61.76	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
5018	-61.76	kd	CGS001-5264	PHYH	-			
5019	-61.78	oe	ccsbBroad304_01519	SET	-			
5020	-61.84	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
5021	-61.89	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
5022	-61.93	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
5023	-61.93	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
5024	-61.94	cc		HIF activator	-			
5025	-62.03	oe	ccsbBroad304_14174	CDKAL1	-			
5026	-62.04	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
5027	-62.08	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
5028	-62.16	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
5029	-62.23	oe	ccsbBroad304_04471	C5ORF62	-			
5030	-62.24	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
5031	-62.26	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
5032	-62.27	oe	ccsbBroad304_08480	PNPO	-			
5033	-62.27	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
5034	-62.29	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
5035	-62.29	kd	CGS001-836	CASP3	Caspases			
5036	-62.3	oe	ccsbBroad304_08322	UFM1	-			
5037	-62.31	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
5038	-62.36	kd	CGS001-4077	NBR1	-			
5039	-62.43	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
5040	-62.46	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
5041	-62.47	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
5042	-62.48	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
5043	-62.5	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
5044	-62.52	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
5045	-62.58	kd	CGS001-1999	ELF3	ETS Transcription Factors			
5046	-62.65	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5047	-62.66	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
5048	-62.66	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
5049	-62.72	kd	CGS001-2287	FKBP3	-			
5050	-62.74	kd	CGS001-55577	NAGK	-			
5051	-62.79	oe	ccsbBroad304_00225	CAT	-			
5052	-62.81	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
5053	-62.85	cp	BRD-K53220666	trimetozine	Sedative			Sedative
5054	-62.85	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
5055	-62.89	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
5056	-62.92	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
5057	-62.97	oe	ccsbBroad304_00489	EHHADH	-			
5058	-62.98	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
5059	-63.03	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5060	-63.09	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5061	-63.13	kd	CGS001-10497	UNC13B	-			
5062	-63.22	oe	ccsbBroad304_00624	GCK	Hexokinases			
5063	-63.26	oe	ccsbBroad304_08802	ELAC2	-			
5064	-63.28	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
5065	-63.29	oe	ccsbBroad304_07727	LIAS	-			
5066	-63.32	oe	ccsbBroad304_00564	FGR	Src family			
5067	-63.37	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
5068	-63.37	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
5069	-63.4	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
5070	-63.46	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
5071	-63.56	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
5072	-63.58	kd	CGS001-382	ARF6	ADP-ribosylation factors			
5073	-63.59	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
5074	-63.59	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
5075	-63.61	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
5076	-63.65	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
5077	-63.67	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
5078	-63.74	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5079	-63.74	kd	CGS001-857	CAV1	-			
5080	-63.76	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
5081	-63.8	oe	ccsbBroad304_00501	EMD	-			
5082	-63.86	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
5083	-63.89	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
5084	-63.9	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
5085	-63.9	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
5086	-63.92	kd	CGS001-2673	GFPT1	-			
5087	-64.04	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
5088	-64.04	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
5089	-64.06	kd	CGS001-538	ATP7A	ATPases / P-type			
5090	-64.06	oe	ccsbBroad304_07219	CDC7	CDC7 family			
5091	-64.15	oe	ccsbBroad304_06996	SRM	-			
5092	-64.16	oe	ccsbBroad304_08952	E2F8	-			
5093	-64.23	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
5094	-64.29	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
5095	-64.31	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
5096	-64.35	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
5097	-64.38	kd	CGS001-51014	TMED7	-			
5098	-64.38	kd	CGS001-1362	CPD	Carboxypeptidase A			
5099	-64.39	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
5100	-64.39	kd	CGS001-6196	RPS6KA2	RSK subfamily			
5101	-64.42	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
5102	-64.45	oe	ccsbBroad304_07884	RYBP	-			
5103	-64.56	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
5104	-64.61	oe	ccsbBroad304_02526	POP4	-			
5105	-64.64	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
5106	-64.65	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
5107	-64.7	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5108	-64.75	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
5109	-64.8	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
5110	-64.82	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
5111	-64.85	kd	CGS001-4905	NSF	ATPases / AAA-type			
5112	-64.92	kd	CGS001-84619	ZGPAT	G patch domain containing			
5113	-64.94	kd	CGS001-776	CACNA1D	Calcium channel subunits			
5114	-64.98	kd	CGS001-7431	VIM	Intermediate filaments type III			
5115	-65.02	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
5116	-65.02	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
5117	-65.05	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
5118	-65.17	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
5119	-65.17	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
5120	-65.18	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5121	-65.24	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
5122	-65.26	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
5123	-65.27	cc		Cannabinoid receptor agonist	-			
5124	-65.28	oe	ccsbBroad304_10487	BPHL	-			
5125	-65.28	oe	ccsbBroad304_06324	GPX7	-			
5126	-65.35	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
5127	-65.4	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
5128	-65.44	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
5129	-65.46	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
5130	-65.48	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
5131	-65.49	kd	CGS001-6217	RPS16	S ribosomal proteins			
5132	-65.49	kd	CGS001-2852	GPER	-			
5133	-65.5	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
5134	-65.52	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
5135	-65.56	oe	ccsbBroad304_03980	DCLRE1B	-			
5136	-65.58	kd	CGS001-8480	RAE1	WD repeat domain containing			
5137	-65.64	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
5138	-65.68	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5139	-65.7	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
5140	-65.79	oe	ccsbBroad304_07827	STK38L	NDR family			
5141	-65.8	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
5142	-65.8	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
5143	-65.8	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
5144	-65.82	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
5145	-65.83	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
5146	-65.93	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
5147	-66.03	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
5148	-66.06	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
5149	-66.08	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
5150	-66.11	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
5151	-66.23	kd	CGS001-5053	PAH	Amino acid hydroxylases			
5152	-66.23	kd	CGS001-2152	F3	CD molecules			
5153	-66.25	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
5154	-66.27	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
5155	-66.28	oe	ccsbBroad304_06386	HNMT	-			
5156	-66.31	kd	CGS001-400	ARL1	ADP-ribosylation factors			
5157	-66.4	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
5158	-66.41	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
5159	-66.47	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
5160	-66.48	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
5161	-66.53	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
5162	-66.54	kd	CGS001-6117	RPA1	-			
5163	-66.54	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
5164	-66.56	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
5165	-66.65	kd	CGS001-718	C3	Endogenous ligands			
5166	-66.66	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
5167	-66.7	oe	ccsbBroad304_02368	TIMM17B	-			
5168	-66.72	oe	ccsbBroad304_01152	PCNA	-			
5169	-66.73	oe	ccsbBroad304_02580	TMED10	-			
5170	-66.73	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
5171	-66.86	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
5172	-66.87	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
5173	-66.88	oe	ccsbBroad304_00966	MAFG	-			
5174	-66.88	oe	ccsbBroad304_00832	IFNB1	Interferons			
5175	-66.89	kd	CGS001-6275	S100A4	EF-hand domain containing			
5176	-66.91	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
5177	-66.92	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
5178	-66.95	cc		CCK receptor antagonist	-			
5179	-66.97	oe	ccsbBroad304_00098	ARG1	Arginase			
5180	-66.97	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
5181	-67.04	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
5182	-67.2	oe	ccsbBroad304_01180	PFKFB3	-			
5183	-67.23	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
5184	-67.25	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
5185	-67.31	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
5186	-67.34	oe	ccsbBroad304_03533	CDCA8	-			
5187	-67.35	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
5188	-67.35	kd	CGS001-1662	DDX10	DEAD-boxes			
5189	-67.43	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5190	-67.47	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
5191	-67.51	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
5192	-67.53	kd	CGS001-84971	ATG4D	-			
5193	-67.54	kd	CGS001-23499	MACF1	EF-hand domain containing			
5194	-67.55	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
5195	-67.64	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
5196	-67.64	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
5197	-67.69	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
5198	-67.7	oe	ccsbBroad304_00789	HSBP1	-			
5199	-67.72	oe	ccsbBroad304_01211	PKM2	-			
5200	-67.73	kd	CGS001-9688	NUP93	-			
5201	-67.76	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
5202	-67.76	kd	CGS001-6342	SCP2	-			
5203	-67.77	oe	ccsbBroad304_09578	PASD1	-			
5204	-67.82	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
5205	-67.83	kd	CGS001-8731	RNMT	-			
5206	-67.94	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5207	-67.97	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
5208	-68.02	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
5209	-68.07	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
5210	-68.11	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
5211	-68.15	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5212	-68.16	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
5213	-68.16	kd	CGS001-9695	EDEM1	-			
5214	-68.22	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
5215	-68.23	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
5216	-68.25	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
5217	-68.34	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
5218	-68.35	kd	CGS001-54884	RETSAT	-			
5219	-68.39	kd	CGS001-11200	CHEK2	CHK1 subfamily			
5220	-68.42	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
5221	-68.44	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
5222	-68.47	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
5223	-68.48	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
5224	-68.48	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
5225	-68.48	oe	ccsbBroad304_13952	SHMT2	-			
5226	-68.5	oe	ccsbBroad304_07889	QPRT	-			
5227	-68.5	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
5228	-68.52	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
5229	-68.53	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
5230	-68.53	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
5231	-68.55	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
5232	-68.57	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
5233	-68.57	kd	CGS001-3163	HMOX2	Haem oxygenase			
5234	-68.58	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
5235	-68.61	oe	ccsbBroad304_01632	SYPL1	-			
5236	-68.61	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
5237	-68.62	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
5238	-68.67	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
5239	-68.68	kd	CGS001-6188	RPS3	S ribosomal proteins			
5240	-68.69	oe	ccsbBroad304_01951	BLZF1	-			
5241	-68.7	kd	CGS001-51015	ISOC1	-			
5242	-68.8	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
5243	-68.82	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5244	-68.87	kd	CGS001-4947	OAZ2	-			
5245	-68.88	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
5246	-68.98	kd	CGS001-226	ALDOA	-			
5247	-69	kd	CGS001-64858	DCLRE1B	-			
5248	-69.01	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
5249	-69.12	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
5250	-69.15	kd	CGS001-9354	UBE4A	U-box domain containing			
5251	-69.16	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5252	-69.24	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
5253	-69.25	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
5254	-69.26	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
5255	-69.27	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
5256	-69.28	cc		Gamma secretase inhibitor	-			
5257	-69.29	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
5258	-69.37	kd	CGS001-11232	POLG2	DNA polymerases			
5259	-69.37	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
5260	-69.39	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
5261	-69.4	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
5262	-69.41	kd	CGS001-2313	FLI1	ETS Transcription Factors			
5263	-69.45	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
5264	-69.47	kd	CGS001-1028	CDKN1C	-			
5265	-69.47	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
5266	-69.5	kd	CGS001-1727	CYB5R3	-			
5267	-69.52	cc		Na-K-Cl transporter inhibitor	-			
5268	-69.53	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
5269	-69.55	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
5270	-69.59	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5271	-69.63	oe	ccsbBroad304_00816	IDE	Pitrilysin			
5272	-69.65	oe	ccsbBroad304_01577	SOD1	-			
5273	-69.67	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
5274	-69.67	kd	CGS001-5624	PROC	Endogenous ligands			
5275	-69.7	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
5276	-69.74	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
5277	-69.87	oe	ccsbBroad304_00447	DLD	-			
5278	-69.9	kd	CGS001-7056	THBD	CD molecules			
5279	-69.93	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
5280	-69.93	kd	CGS001-27244	SESN1	-			
5281	-69.98	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
5282	-70.01	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
5283	-70.01	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
5284	-70.03	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
5285	-70.08	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
5286	-70.09	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
5287	-70.11	kd	CGS001-6772	STAT1	SH2 domain containing			
5288	-70.12	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
5289	-70.23	kd	CGS001-1287	COL4A5	Collagens			
5290	-70.26	oe	ccsbBroad304_06671	OPA1	-			
5291	-70.3	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
5292	-70.32	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5293	-70.33	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
5294	-70.44	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
5295	-70.44	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
5296	-70.52	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
5297	-70.55	oe	ccsbBroad304_01019	MLH1	-			
5298	-70.55	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
5299	-70.57	cc		Leucine rich repeat kinase inhibitor	-			
5300	-70.61	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
5301	-70.61	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
5302	-70.65	kd	CGS001-10587	TXNRD2	-			
5303	-70.69	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
5304	-70.7	kd	CGS001-54881	TEX10	-			
5305	-70.7	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
5306	-70.74	oe	ccsbBroad304_00316	CKS1B	-			
5307	-70.79	oe	ccsbBroad304_07128	VHL	-			
5308	-70.79	kd	CGS001-8428	STK24	YSK subfamily			
5309	-70.79	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
5310	-70.86	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
5311	-70.86	oe	ccsbBroad304_06225	FTH1	-			
5312	-70.87	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
5313	-70.88	oe	ccsbBroad304_00490	EIF4EBP1	-			
5314	-70.9	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
5315	-70.92	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
5316	-71	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
5317	-71	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
5318	-71.02	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
5319	-71.02	kd	CGS001-7358	UGDH	-			
5320	-71.02	kd	CGS001-9759	HDAC4	Histone deacetylases			
5321	-71.04	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
5322	-71.07	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
5323	-71.09	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
5324	-71.1	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
5325	-71.2	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
5326	-71.25	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
5327	-71.43	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
5328	-71.43	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
5329	-71.47	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
5330	-71.47	kd	CGS001-35	ACADS	-			
5331	-71.55	kd	CGS001-1070	CETN3	EF-hand domain containing			
5332	-71.57	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
5333	-71.6	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
5334	-71.64	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
5335	-71.69	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
5336	-71.71	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
5337	-71.74	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
5338	-71.78	kd	CGS001-54386	TERF2IP	-			
5339	-71.84	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
5340	-71.89	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
5341	-71.99	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
5342	-72	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
5343	-72.01	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
5344	-72.05	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
5345	-72.06	oe	ccsbBroad304_03182	GLOD4	-			
5346	-72.1	kd	CGS001-1738	DLD	-			
5347	-72.11	oe	ccsbBroad304_07800	EXOSC8	-			
5348	-72.11	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
5349	-72.11	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
5350	-72.11	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
5351	-72.11	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
5352	-72.2	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
5353	-72.23	cc		Zinc fingers RanBP2 type LOF	-			
5354	-72.24	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
5355	-72.24	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
5356	-72.29	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
5357	-72.31	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
5358	-72.35	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
5359	-72.39	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
5360	-72.4	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
5361	-72.42	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
5362	-72.43	oe	ccsbBroad304_02671	ECD	-			
5363	-72.44	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
5364	-72.45	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
5365	-72.47	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
5366	-72.49	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
5367	-72.51	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
5368	-72.58	oe	ccsbBroad304_06464	ITGB2	Integrins			
5369	-72.61	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
5370	-72.62	kd	CGS001-8848	TSC22D1	-			
5371	-72.63	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
5372	-72.64	kd	CGS001-121599	SPIC	ETS Transcription Factors			
5373	-72.75	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
5374	-72.78	oe	ccsbBroad304_08898	TRAK2	-			
5375	-72.82	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
5376	-72.85	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
5377	-72.88	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
5378	-72.95	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
5379	-72.95	kd	CGS001-5664	PSEN2	Presenilin			
5380	-73.01	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
5381	-73.02	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
5382	-73.02	kd	CGS001-1399	CRKL	SH2 domain containing			
5383	-73.08	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
5384	-73.08	kd	CGS001-57157	PHTF2	-			
5385	-73.08	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
5386	-73.1	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
5387	-73.1	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
5388	-73.15	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
5389	-73.17	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
5390	-73.32	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
5391	-73.34	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
5392	-73.4	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
5393	-73.42	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
5394	-73.42	kd	CGS001-10673	TNFSF13B	CD molecules			
5395	-73.43	cc		Aurora kinase inhibitor	-			
5396	-73.44	oe	ccsbBroad304_00099	ARG2	Arginase			
5397	-73.46	kd	CGS001-56882	CDC42SE1	-			
5398	-73.51	kd	CGS001-6446	SGK1	SGK family			
5399	-73.54	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
5400	-73.57	kd	CGS001-11267	SNF8	-			
5401	-73.58	kd	CGS001-2885	GRB2	SH2 domain containing			
5402	-73.61	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
5403	-73.67	kd	CGS001-10447	FAM3C	-			
5404	-73.7	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
5405	-73.7	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
5406	-73.71	oe	ccsbBroad304_06085	DCK	-			
5407	-73.72	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
5408	-73.73	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
5409	-73.81	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
5410	-73.83	cc		Serotonin receptor agonist	-			
5411	-73.89	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
5412	-73.97	kd	CGS001-2729	GCLC	-			
5413	-73.98	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
5414	-73.99	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
5415	-74	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
5416	-74.01	cc		Imidazoline ligand	-			
5417	-74.03	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
5418	-74.03	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
5419	-74.09	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
5420	-74.14	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5421	-74.16	oe	ccsbBroad304_00038	AGL	-			
5422	-74.18	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
5423	-74.24	oe	ccsbBroad304_06518	LDHA	-			
5424	-74.33	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
5425	-74.36	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
5426	-74.38	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5427	-74.4	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
5428	-74.4	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
5429	-74.41	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
5430	-74.48	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
5431	-74.55	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
5432	-74.58	oe	ccsbBroad304_00986	MCM2	-			
5433	-74.63	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
5434	-74.64	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
5435	-74.74	oe	ccsbBroad304_01371	RALA	-			
5436	-74.75	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
5437	-74.75	kd	CGS001-256281	NUDT14	Nudix motif containing			
5438	-74.8	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
5439	-74.84	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
5440	-74.87	oe	ccsbBroad304_03119	C16ORF5	-			
5441	-74.93	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
5442	-74.94	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
5443	-74.94	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
5444	-75.01	oe	ccsbBroad304_08137	HOOK2	-			
5445	-75.01	kd	CGS001-54584	GNB1L	WD repeat domain containing			
5446	-75.03	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
5447	-75.03	kd	CGS001-9697	TRAM2	-			
5448	-75.06	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
5449	-75.08	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5450	-75.13	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
5451	-75.15	cc		Angiotensin receptor antagonist	-			
5452	-75.15	oe	ccsbBroad304_03479	YTHDF1	-			
5453	-75.29	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
5454	-75.34	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
5455	-75.36	kd	CGS001-183	AGT	Endogenous ligands			
5456	-75.41	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
5457	-75.43	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
5458	-75.48	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
5459	-75.49	kd	CGS001-6016	RIT1	-			
5460	-75.55	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
5461	-75.55	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
5462	-75.56	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5463	-75.58	kd	CGS001-89766	UMODL1	-			
5464	-75.75	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
5465	-75.76	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
5466	-75.86	oe	ccsbBroad304_03155	DHH	-			
5467	-75.92	oe	ccsbBroad304_01532	SIAH1	-			
5468	-75.93	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
5469	-75.94	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
5470	-75.97	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
5471	-75.98	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
5472	-76.04	oe	ccsbBroad304_02596	KDELR3	-			
5473	-76.1	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
5474	-76.18	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
5475	-76.2	oe	ccsbBroad304_05183	TXLNA	-			
5476	-76.23	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
5477	-76.32	kd	CGS001-1633	DCK	-			
5478	-76.35	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
5479	-76.38	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
5480	-76.38	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
5481	-76.4	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
5482	-76.4	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5483	-76.41	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
5484	-76.42	kd	CGS001-9380	GRHPR	-			
5485	-76.46	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
5486	-76.48	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
5487	-76.49	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
5488	-76.51	kd	CGS001-6856	SYPL1	-			
5489	-76.54	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
5490	-76.59	kd	CGS001-6397	SEC14L1	-			
5491	-76.59	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
5492	-76.63	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
5493	-76.7	oe	ccsbBroad304_00600	FYN	Src family			
5494	-76.71	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
5495	-76.71	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
5496	-76.79	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
5497	-76.84	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
5498	-76.86	oe	ccsbBroad304_02578	EBNA1BP2	-			
5499	-76.91	oe	ccsbBroad304_00841	IKBKB	IKK family			
5500	-76.91	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
5501	-76.92	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
5502	-76.92	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
5503	-76.95	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
5504	-76.97	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
5505	-77.01	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
5506	-77.02	kd	CGS001-2030	SLC29A1	SLC29 family			
5507	-77.07	oe	ccsbBroad304_02094	FIBP	-			
5508	-77.07	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
5509	-77.1	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
5510	-77.17	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
5511	-77.18	oe	ccsbBroad304_01724	TTR	-			
5512	-77.2	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
5513	-77.21	kd	CGS001-54623	PAF1	-			
5514	-77.25	kd	CGS001-5160	PDHA1	-			
5515	-77.28	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
5516	-77.3	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
5517	-77.35	oe	ccsbBroad304_00962	SMAD4	SMADs			
5518	-77.37	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
5519	-77.49	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
5520	-77.52	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
5521	-77.57	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
5522	-77.62	oe	ccsbBroad304_03310	LCMT1	-			
5523	-77.66	oe	ccsbBroad304_02789	ADAT1	-			
5524	-77.72	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
5525	-77.76	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
5526	-77.77	kd	CGS001-1069	CETN2	EF-hand domain containing			
5527	-77.78	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
5528	-77.85	kd	CGS001-1981	EIF4G1	Parkinson disease			
5529	-77.99	oe	ccsbBroad304_02032	TSC22D1	-			
5530	-77.99	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
5531	-78.03	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5532	-78.1	oe	ccsbBroad304_00874	INS	-			
5533	-78.22	oe	ccsbBroad304_02136	COPS2	-			
5534	-78.24	kd	CGS001-2878	GPX3	-			
5535	-78.32	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
5536	-78.33	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
5537	-78.35	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5538	-78.38	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
5539	-78.39	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
5540	-78.39	kd	CGS001-11041	B3GNT1	-			
5541	-78.45	oe	ccsbBroad304_05192	SPRED2	-			
5542	-78.47	oe	ccsbBroad304_00077	APEX1	-			
5543	-78.49	oe	ccsbBroad304_08292	IP6K2	-			
5544	-78.54	oe	ccsbBroad304_07119	UGP2	-			
5545	-78.56	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
5546	-78.57	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
5547	-78.61	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
5548	-78.62	cc		Minor histocompatibility antigens LOF	-			
5549	-78.7	oe	ccsbBroad304_00931	LCN2	Lipocalins			
5550	-78.71	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
5551	-78.78	kd	CGS001-31	ACACA	Carboxylases			
5552	-78.8	oe	ccsbBroad304_13598	NRBP2	NRBP family			
5553	-78.94	kd	CGS001-7040	TGFB1	Endogenous ligands			
5554	-78.94	kd	CGS001-2664	GDI1	-			
5555	-78.97	kd	CGS001-11230	PRAF2	-			
5556	-79.02	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
5557	-79.06	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
5558	-79.07	kd	CGS001-7128	TNFAIP3	OTU domain containing			
5559	-79.08	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
5560	-79.09	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
5561	-79.1	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
5562	-79.1	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
5563	-79.11	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
5564	-79.18	kd	CGS001-2037	EPB41L2	-			
5565	-79.21	oe	ccsbBroad304_03858	SRPRB	-			
5566	-79.22	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
5567	-79.22	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
5568	-79.23	oe	ccsbBroad304_01832	PAX8	Paired boxes			
5569	-79.23	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
5570	-79.28	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
5571	-79.28	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5572	-79.35	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
5573	-79.36	oe	ccsbBroad304_03615	ZNF673	-			
5574	-79.37	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
5575	-79.39	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
5576	-79.42	kd	CGS001-5684	PSMA3	Proteasome subunits			
5577	-79.43	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
5578	-79.44	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
5579	-79.52	oe	ccsbBroad304_01701	TPI1	-			
5580	-79.54	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
5581	-79.54	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5582	-79.54	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
5583	-79.61	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
5584	-79.62	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
5585	-79.65	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
5586	-79.66	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
5587	-79.7	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
5588	-79.76	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
5589	-79.76	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
5590	-79.76	kd	CGS001-2966	GTF2H2	General transcription factors			
5591	-79.78	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
5592	-79.78	kd	CGS001-9131	AIFM1	-			
5593	-79.79	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
5594	-79.79	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
5595	-79.86	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
5596	-79.89	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
5597	-79.9	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
5598	-79.96	cc		Sirtuins GOF	-			
5599	-80.01	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5600	-80.03	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
5601	-80.07	kd	CGS001-23621	BACE1	Pepsin			
5602	-80.17	cc		Serotonin receptor antagonist	-			
5603	-80.24	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
5604	-80.34	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
5605	-80.37	kd	CGS001-6696	SPP1	Endogenous ligands			
5606	-80.39	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
5607	-80.42	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
5608	-80.43	kd	CGS001-84647	PLA2G12B	-			
5609	-80.47	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
5610	-80.5	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
5611	-80.51	kd	CGS001-51734	SEPX1	-			
5612	-80.54	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
5613	-80.55	oe	ccsbBroad304_06126	TSC22D3	-			
5614	-80.6	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
5615	-80.62	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
5616	-80.63	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
5617	-80.66	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
5618	-80.68	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
5619	-80.71	kd	CGS001-847	CAT	-			
5620	-80.73	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
5621	-80.75	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
5622	-80.75	kd	CGS001-4087	SMAD2	SMADs			
5623	-80.76	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
5624	-80.8	kd	CGS001-3265	HRAS	RAS subfamily			
5625	-80.81	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
5626	-80.81	kd	CGS001-7486	WRN	-			
5627	-80.82	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
5628	-80.84	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
5629	-80.88	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
5630	-80.94	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
5631	-80.95	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
5632	-81.03	kd	CGS001-51805	COQ3	-			
5633	-81.07	kd	CGS001-51160	VPS28	-			
5634	-81.08	kd	CGS001-4602	MYB	-			
5635	-81.09	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
5636	-81.11	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
5637	-81.19	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
5638	-81.21	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
5639	-81.22	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
5640	-81.24	oe	ccsbBroad304_02276	MVP	-			
5641	-81.34	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
5642	-81.36	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
5643	-81.36	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
5644	-81.37	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
5645	-81.42	oe	ccsbBroad304_03658	DCP1A	-			
5646	-81.48	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
5647	-81.49	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
5648	-81.5	kd	CGS001-7296	TXNRD1	-			
5649	-81.55	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
5650	-81.56	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5651	-81.56	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
5652	-81.59	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5653	-81.6	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
5654	-81.6	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
5655	-81.6	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
5656	-81.62	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5657	-81.63	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
5658	-81.64	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
5659	-81.65	kd	CGS001-302	ANXA2	Annexins			
5660	-81.68	oe	ccsbBroad304_02702	MSRB2	-			
5661	-81.73	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
5662	-81.74	oe	ccsbBroad304_06004	CKB	-			
5663	-81.81	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
5664	-81.85	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
5665	-81.86	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
5666	-81.88	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
5667	-81.9	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
5668	-81.9	kd	CGS001-3827	KNG1	Endogenous ligands			
5669	-81.9	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
5670	-81.91	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
5671	-81.94	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
5672	-82.12	kd	CGS001-5033	P4HA1	-			
5673	-82.14	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
5674	-82.16	kd	CGS001-55793	FAM63A	-			
5675	-82.17	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
5676	-82.18	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
5677	-82.2	kd	CGS001-9512	PMPCB	-			
5678	-82.22	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
5679	-82.22	kd	CGS001-22887	FOXJ3	Forkhead boxes			
5680	-82.23	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
5681	-82.23	kd	CGS001-6611	SMS	-			
5682	-82.24	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
5683	-82.32	oe	ccsbBroad304_06094	DFFA	-			
5684	-82.33	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
5685	-82.33	kd	CGS001-58477	SRPRB	-			
5686	-82.33	kd	CGS001-2004	ELK3	ETS Transcription Factors			
5687	-82.34	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
5688	-82.41	oe	ccsbBroad304_00070	ANXA5	Annexins			
5689	-82.42	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
5690	-82.44	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
5691	-82.47	oe	ccsbBroad304_02217	FEZ1	-			
5692	-82.48	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
5693	-82.58	oe	ccsbBroad304_06525	LIPA	-			
5694	-82.58	kd	CGS001-23475	QPRT	-			
5695	-82.62	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
5696	-82.63	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
5697	-82.65	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
5698	-82.65	kd	CGS001-839	CASP6	Caspases			
5699	-82.66	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
5700	-82.66	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
5701	-82.76	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
5702	-82.77	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
5703	-82.8	cc		Tachykinin antagonist	-			
5704	-82.8	kd	CGS001-5909	RAP1GAP	-			
5705	-82.84	kd	CGS001-10252	SPRY1	-			
5706	-82.86	cc		Purinergic receptors P2Y GOF	-			
5707	-82.86	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
5708	-82.87	kd	CGS001-64422	ATG3	-			
5709	-82.9	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
5710	-82.9	kd	CGS001-2161	F12	Chymotrypsin			
5711	-82.92	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
5712	-82.95	oe	ccsbBroad304_06683	FURIN	Subtilisin			
5713	-82.97	kd	CGS001-634	CEACAM1	CD molecules			
5714	-83.07	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
5715	-83.08	oe	ccsbBroad304_06494	KLRC1	CD molecules			
5716	-83.08	kd	CGS001-4174	MCM5	-			
5717	-83.09	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
5718	-83.11	oe	ccsbBroad304_07267	PDLIM4	-			
5719	-83.12	cc		Progesterone receptor agonist	-			
5720	-83.13	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
5721	-83.13	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
5722	-83.17	oe	ccsbBroad304_06188	F10	Chymotrypsin			
5723	-83.28	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
5724	-83.29	kd	CGS001-23210	JMJD6	-			
5725	-83.32	cc		Dopamine receptor antagonist	-			
5726	-83.34	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
5727	-83.34	kd	CGS001-3821	KLRC1	CD molecules			
5728	-83.35	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
5729	-83.35	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
5730	-83.36	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
5731	-83.37	oe	ccsbBroad304_00651	GNAI3	-			
5732	-83.38	kd	CGS001-10538	BATF	basic leucine zipper proteins			
5733	-83.4	cc		RNA Polymerase Enzymes LOF	-			
5734	-83.41	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
5735	-83.42	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
5736	-83.44	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
5737	-83.45	oe	ccsbBroad304_00880	IRF2	-			
5738	-83.47	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
5739	-83.5	kd	CGS001-162699	TCEB3C	-			
5740	-83.52	kd	CGS001-3998	LMAN1	-			
5741	-83.54	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
5742	-83.55	oe	ccsbBroad304_02372	SPRY1	-			
5743	-83.55	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
5744	-83.58	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
5745	-83.6	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
5746	-83.63	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
5747	-83.68	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
5748	-83.7	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
5749	-83.71	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
5750	-83.74	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
5751	-83.76	kd	CGS001-151126	ZNF385B	-			
5752	-83.77	kd	CGS001-6827	SUPT4H1	-			
5753	-83.81	kd	CGS001-7003	TEAD1	-			
5754	-83.86	oe	ccsbBroad304_00006	ACADM	-			
5755	-83.95	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
5756	-83.98	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5757	-84.02	kd	CGS001-10606	PAICS	-			
5758	-84.06	oe	ccsbBroad304_05757	ACADS	-			
5759	-84.07	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
5760	-84.1	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
5761	-84.11	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
5762	-84.17	kd	CGS001-2747	GLUD2	-			
5763	-84.22	oe	ccsbBroad304_00888	ITPK1	-			
5764	-84.26	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
5765	-84.29	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
5766	-84.29	oe	ccsbBroad304_00620	GCDH	-			
5767	-84.32	kd	CGS001-23753	SDF2L1	-			
5768	-84.32	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
5769	-84.33	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5770	-84.36	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
5771	-84.38	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
5772	-84.38	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
5773	-84.41	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
5774	-84.42	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
5775	-84.46	kd	CGS001-2100	ESR2	Estrogen receptors			
5776	-84.61	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
5777	-84.61	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
5778	-84.64	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
5779	-84.64	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
5780	-84.64	kd	CGS001-3516	RBPJ	-			
5781	-84.65	kd	CGS001-9767	PHF16	-			
5782	-84.7	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
5783	-84.72	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
5784	-84.74	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
5785	-84.76	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
5786	-84.81	oe	ccsbBroad304_01658	PRDX2	-			
5787	-84.82	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
5788	-84.83	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
5789	-84.88	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
5790	-84.89	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
5791	-84.93	oe	ccsbBroad304_01640	TAF12	-			
5792	-84.94	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
5793	-84.95	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5794	-85	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
5795	-85.01	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5796	-85.04	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
5797	-85.04	kd	CGS001-1445	CSK	Csk family			
5798	-85.07	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
5799	-85.2	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
5800	-85.24	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
5801	-85.26	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
5802	-85.28	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
5803	-85.32	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
5804	-85.33	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5805	-85.35	kd	CGS001-85442	KNDC1	-			
5806	-85.36	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
5807	-85.36	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
5808	-85.4	oe	ccsbBroad304_00390	CTGF	-			
5809	-85.41	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
5810	-85.43	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
5811	-85.47	oe	ccsbBroad304_02138	TRIP10	-			
5812	-85.5	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
5813	-85.5	kd	CGS001-257397	TAB3	-			
5814	-85.5	kd	CGS001-3638	INSIG1	-			
5815	-85.53	oe	ccsbBroad304_02197	VPS26A	-			
5816	-85.53	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
5817	-85.59	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
5818	-85.6	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
5819	-85.62	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
5820	-85.65	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
5821	-85.66	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
5822	-85.66	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
5823	-85.68	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
5824	-85.7	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5825	-85.71	kd	CGS001-8780	RIOK3	RIO3 subfamily			
5826	-85.74	cc		GPCR Subset GOF	-			
5827	-85.77	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
5828	-85.78	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
5829	-85.81	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
5830	-85.81	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
5831	-85.81	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
5832	-85.82	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
5833	-85.86	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
5834	-85.88	kd	CGS001-2597	GAPDH	-			
5835	-85.92	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
5836	-85.93	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
5837	-85.99	kd	CGS001-51655	RASD1	-			
5838	-86.01	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
5839	-86.01	kd	CGS001-930	CD19	CD molecules			
5840	-86.15	oe	ccsbBroad304_02569	BTG3	-			
5841	-86.15	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
5842	-86.18	oe	ccsbBroad304_07761	CORO1A	Coronins			
5843	-86.18	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
5844	-86.25	oe	ccsbBroad304_00995	MECP2	-			
5845	-86.25	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
5846	-86.32	kd	CGS001-1398	CRK	SH2 domain containing			
5847	-86.34	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
5848	-86.35	kd	CGS001-9531	BAG3	-			
5849	-86.35	kd	CGS001-397	ARHGDIB	Endogenous ligands			
5850	-86.37	cp	BRD-K15842202	eudesmic-acid	-666			-666
5851	-86.43	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5852	-86.43	kd	CGS001-11007	CCDC85B	-			
5853	-86.72	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
5854	-86.76	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
5855	-86.77	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
5856	-86.79	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
5857	-86.8	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
5858	-86.84	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
5859	-86.85	oe	ccsbBroad304_03037	TMEM97	-			
5860	-86.91	kd	CGS001-4925	NUCB2	EF-hand domain containing			
5861	-86.97	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
5862	-87.01	kd	CGS001-7077	TIMP2	-			
5863	-87.01	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
5864	-87.03	oe	ccsbBroad304_06286	GLUL	-			
5865	-87.05	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
5866	-87.05	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
5867	-87.1	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
5868	-87.1	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5869	-87.13	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
5870	-87.15	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
5871	-87.16	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
5872	-87.16	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5873	-87.2	kd	CGS001-2266	FGG	Endogenous ligands			
5874	-87.22	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
5875	-87.23	oe	ccsbBroad304_08481	CEP55	-			
5876	-87.23	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
5877	-87.26	oe	ccsbBroad304_01142	PAFAH1B2	-			
5878	-87.26	kd	CGS001-10923	SUB1	-			
5879	-87.28	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
5880	-87.28	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
5881	-87.28	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
5882	-87.28	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
5883	-87.31	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
5884	-87.35	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
5885	-87.35	kd	CGS001-5618	PRLR	Prolactin receptor family			
5886	-87.37	kd	CGS001-10482	NXF1	-			
5887	-87.38	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
5888	-87.41	cc		Rho associated kinase inhibitor	-			
5889	-87.41	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
5890	-87.43	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
5891	-87.43	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
5892	-87.44	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
5893	-87.47	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
5894	-87.48	cc		HDAC inhibitor	-			
5895	-87.48	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
5896	-87.48	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
5897	-87.48	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
5898	-87.48	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
5899	-87.5	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
5900	-87.52	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
5901	-87.55	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
5902	-87.62	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
5903	-87.65	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
5904	-87.66	oe	ccsbBroad304_03859	ENOPH1	-			
5905	-87.67	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
5906	-87.68	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
5907	-87.69	oe	ccsbBroad304_02018	SUCLA2	-			
5908	-87.69	kd	CGS001-29946	SERTAD3	-			
5909	-87.69	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
5910	-87.69	kd	CGS001-10046	MAMLD1	-			
5911	-87.77	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
5912	-87.78	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
5913	-87.8	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
5914	-87.84	kd	CGS001-10775	POP4	-			
5915	-87.84	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
5916	-87.85	kd	CGS001-1284	COL4A2	Collagens			
5917	-87.88	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
5918	-87.94	kd	CGS001-8996	NOL3	-			
5919	-87.94	kd	CGS001-383	ARG1	Arginase			
5920	-87.95	oe	ccsbBroad304_01174	PEX13	-			
5921	-87.95	kd	CGS001-51293	CD320	CD molecules			
5922	-87.97	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
5923	-87.97	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
5924	-88	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
5925	-88	oe	ccsbBroad304_07632	PROCR	CD molecules			
5926	-88.01	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
5927	-88.04	kd	CGS001-3985	LIMK2	LIMK subfamily			
5928	-88.04	kd	CGS001-50943	FOXP3	Forkhead boxes			
5929	-88.05	oe	ccsbBroad304_11405	UBE3C	-			
5930	-88.05	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
5931	-88.05	kd	CGS001-22938	SNW1	-			
5932	-88.05	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
5933	-88.06	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
5934	-88.06	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
5935	-88.06	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
5936	-88.09	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
5937	-88.1	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
5938	-88.15	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
5939	-88.19	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5940	-88.23	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5941	-88.26	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
5942	-88.32	oe	ccsbBroad304_02270	FAM20B	-			
5943	-88.32	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
5944	-88.35	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
5945	-88.37	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
5946	-88.38	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
5947	-88.38	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5948	-88.4	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
5949	-88.41	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5950	-88.43	cc		Glucocorticoid receptor agonist	-			
5951	-88.44	kd	CGS001-51022	GLRX2	-			
5952	-88.6	oe	ccsbBroad304_02676	PHB2	-			
5953	-88.62	kd	CGS001-8900	CCNA1	-			
5954	-88.63	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
5955	-88.64	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
5956	-88.67	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
5957	-88.67	kd	CGS001-1201	CLN3	-			
5958	-88.68	oe	ccsbBroad304_06103	DMD	-			
5959	-88.69	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
5960	-88.71	kd	CGS001-2581	GALC	-			
5961	-88.75	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
5962	-88.76	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
5963	-88.84	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5964	-88.84	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
5965	-88.87	kd	CGS001-10020	GNE	-			
5966	-88.98	oe	ccsbBroad304_03420	TOLLIP	-			
5967	-88.99	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
5968	-89.05	oe	ccsbBroad304_07118	UGDH	-			
5969	-89.07	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
5970	-89.08	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
5971	-89.09	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
5972	-89.14	oe	ccsbBroad304_10240	CROT	-			
5973	-89.14	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
5974	-89.15	cc		Ribosomal 40s Subunit LOF	-			
5975	-89.15	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
5976	-89.15	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
5977	-89.16	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
5978	-89.21	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
5979	-89.21	kd	CGS001-22930	RAB3GAP1	-			
5980	-89.22	kd	CGS001-126823	KLHDC9	-			
5981	-89.24	kd	CGS001-27113	BBC3	-			
5982	-89.27	oe	ccsbBroad304_02419	NDRG1	-			
5983	-89.28	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
5984	-89.3	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
5985	-89.33	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5986	-89.33	kd	CGS001-5106	PCK2	-			
5987	-89.35	kd	CGS001-5357	PLS1	EF-hand domain containing			
5988	-89.37	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
5989	-89.39	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
5990	-89.39	kd	CGS001-2678	GGT1	CD molecules			
5991	-89.44	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
5992	-89.49	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
5993	-89.49	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
5994	-89.54	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
5995	-89.54	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
5996	-89.55	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
5997	-89.56	kd	CGS001-3575	IL7R	IL-2 receptor family			
5998	-89.6	oe	ccsbBroad304_07101	TSC2	-			
5999	-89.61	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
6000	-89.66	kd	CGS001-3551	IKBKB	IKK family			
6001	-89.69	kd	CGS001-54505	DHX29	DEAH-boxes			
6002	-89.7	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
6003	-89.73	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
6004	-89.73	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
6005	-89.74	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6006	-89.74	oe	ccsbBroad304_07724	KDELR2	-			
6007	-89.74	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
6008	-89.76	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
6009	-89.78	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
6010	-89.79	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
6011	-89.82	cc		V type ATPases LOF	-			
6012	-89.83	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6013	-89.88	kd	CGS001-139135	PASD1	-			
6014	-89.89	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
6015	-89.9	kd	CGS001-23081	KDM4C	Histone demethylases			
6016	-89.93	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
6017	-89.99	kd	CGS001-2810	SFN	-			
6018	-90.01	oe	ccsbBroad304_00991	MDH1	-			
6019	-90.02	oe	ccsbBroad304_01584	SPARC	-			
6020	-90.09	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
6021	-90.13	oe	ccsbBroad304_06992	SRC	Src family			
6022	-90.14	cc		Nucleophosmin inhibitor	-			
6023	-90.15	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
6024	-90.16	oe	ccsbBroad304_06985	SORD	-			
6025	-90.18	oe	ccsbBroad304_07490	SCRN1	-			
6026	-90.19	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
6027	-90.19	oe	ccsbBroad304_01304	PSEN1	Presenilin			
6028	-90.19	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
6029	-90.2	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
6030	-90.2	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
6031	-90.24	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
6032	-90.26	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
6033	-90.31	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
6034	-90.34	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
6035	-90.36	cc		Androgen receptor modulator	-			
6036	-90.4	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
6037	-90.41	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
6038	-90.43	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
6039	-90.49	kd	CGS001-8508	NIPSNAP1	-			
6040	-90.52	oe	ccsbBroad304_09095	PUS7L	-			
6041	-90.56	oe	ccsbBroad304_07220	CDC45	-			
6042	-90.58	kd	CGS001-5300	PIN1	-			
6043	-90.6	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6044	-90.69	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6045	-90.71	kd	CGS001-5019	OXCT1	-			
6046	-90.73	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
6047	-90.76	oe	ccsbBroad304_00430	GADD45A	-			
6048	-90.78	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
6049	-90.82	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
6050	-90.85	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
6051	-90.85	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
6052	-90.93	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
6053	-90.94	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
6054	-90.98	oe	ccsbBroad304_05931	CAPG	-			
6055	-91	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
6056	-91.05	kd	CGS001-1131	CHRM3	Cholinergic receptors			
6057	-91.08	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
6058	-91.08	kd	CGS001-151306	GPBAR1	Bile acid receptor			
6059	-91.1	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
6060	-91.14	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
6061	-91.15	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
6062	-91.15	kd	CGS001-533	ATP6V0B	ATPases / V-type			
6063	-91.18	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
6064	-91.2	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
6065	-91.22	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
6066	-91.24	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
6067	-91.28	kd	CGS001-5361	PLXNA1	Plexins			
6068	-91.41	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
6069	-91.42	kd	CGS001-9710	KIAA0355	-			
6070	-91.44	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
6071	-91.46	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
6072	-91.5	kd	CGS001-54106	TLR9	Toll-like receptor family			
6073	-91.52	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
6074	-91.54	oe	ccsbBroad304_08645	BCCIP	-			
6075	-91.54	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
6076	-91.56	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
6077	-91.57	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
6078	-91.58	oe	ccsbBroad304_07651	HEXIM1	-			
6079	-91.6	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
6080	-91.61	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
6081	-91.64	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
6082	-91.69	oe	ccsbBroad304_06836	RAD23B	-			
6083	-91.72	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
6084	-91.72	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
6085	-91.75	oe	ccsbBroad304_00993	MDM4	-			
6086	-91.76	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
6087	-91.81	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
6088	-91.84	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
6089	-91.86	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
6090	-91.88	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
6091	-91.92	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
6092	-91.92	kd	CGS001-819	CAMLG	-			
6093	-91.94	kd	CGS001-5708	PSMD2	Proteasome subunits			
6094	-91.96	oe	ccsbBroad304_02626	PKIG	-			
6095	-91.97	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
6096	-91.97	kd	CGS001-84547	PGBD1	-			
6097	-91.98	oe	ccsbBroad304_00184	C2	Complement system			
6098	-91.98	kd	CGS001-842	CASP9	Caspases			
6099	-92	kd	CGS001-10681	GNB5	WD repeat domain containing			
6100	-92.04	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
6101	-92.07	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
6102	-92.07	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
6103	-92.07	kd	CGS001-51447	IP6K2	-			
6104	-92.09	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
6105	-92.09	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
6106	-92.15	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
6107	-92.16	oe	ccsbBroad304_02458	STK25	YSK subfamily			
6108	-92.16	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
6109	-92.17	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
6110	-92.17	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
6111	-92.18	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
6112	-92.18	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
6113	-92.21	oe	ccsbBroad304_07050	TFAP2A	-			
6114	-92.23	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
6115	-92.24	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
6116	-92.26	kd	CGS001-638	BIK	-			
6117	-92.27	cc		MCM family LOF	-			
6118	-92.27	cc		Ribonucleotide reductase inhibitor	-			
6119	-92.3	oe	ccsbBroad304_00883	ISG20	-			
6120	-92.3	kd	CGS001-23244	PDS5A	-			
6121	-92.32	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
6122	-92.37	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
6123	-92.45	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
6124	-92.46	oe	ccsbBroad304_00112	ASNA1	-			
6125	-92.49	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
6126	-92.5	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
6127	-92.51	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
6128	-92.56	kd	CGS001-8727	CTNNAL1	Catenins			
6129	-92.65	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
6130	-92.66	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
6131	-92.7	oe	ccsbBroad304_00118	ATIC	-			
6132	-92.73	oe	ccsbBroad304_03928	RRAGC	-			
6133	-92.73	oe	ccsbBroad304_00810	HYAL1	-			
6134	-92.73	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
6135	-92.74	oe	ccsbBroad304_03177	FIS1	-			
6136	-92.78	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
6137	-92.79	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6138	-92.79	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
6139	-92.83	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
6140	-92.86	oe	ccsbBroad304_05894	BLVRA	-			
6141	-92.91	kd	CGS001-9655	SOCS5	SH2 domain containing			
6142	-92.92	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
6143	-92.92	kd	CGS001-55526	DHTKD1	-			
6144	-92.93	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
6145	-92.95	kd	CGS001-9805	SCRN1	-			
6146	-93.01	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
6147	-93.02	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
6148	-93.03	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
6149	-93.09	oe	ccsbBroad304_00881	IRF5	-			
6150	-93.1	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
6151	-93.13	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
6152	-93.18	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
6153	-93.2	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
6154	-93.2	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
6155	-93.21	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
6156	-93.21	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
6157	-93.22	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6158	-93.24	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
6159	-93.25	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
6160	-93.28	kd	CGS001-5423	POLB	DNA polymerases			
6161	-93.3	kd	CGS001-10472	ZNF238	-			
6162	-93.32	oe	ccsbBroad304_08392	EXOC6	-			
6163	-93.32	kd	CGS001-6810	STX4	-			
6164	-93.36	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
6165	-93.38	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6166	-93.38	kd	CGS001-7079	TIMP4	-			
6167	-93.38	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
6168	-93.38	kd	CGS001-90861	HN1L	-			
6169	-93.4	kd	CGS001-673	BRAF	RAF family			
6170	-93.4	kd	CGS001-506	ATP5B	ATPases / F-type			
6171	-93.42	kd	CGS001-1312	COMT	Catecholamine turnover			
6172	-93.44	oe	ccsbBroad304_00102	RND3	-			
6173	-93.45	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
6174	-93.46	oe	ccsbBroad304_02506	EBP	-			
6175	-93.47	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
6176	-93.5	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
6177	-93.51	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
6178	-93.53	oe	ccsbBroad304_08694	TBX20	T-boxes			
6179	-93.58	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
6180	-93.63	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
6181	-93.65	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
6182	-93.65	kd	CGS001-64121	RRAGC	-			
6183	-93.66	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6184	-93.66	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
6185	-93.68	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
6186	-93.75	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
6187	-93.76	oe	ccsbBroad304_01664	TGFA	-			
6188	-93.76	oe	ccsbBroad304_09503	KLHDC9	-			
6189	-93.78	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6190	-93.79	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
6191	-93.8	kd	CGS001-5566	PRKACA	Protein kinase A			
6192	-93.81	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
6193	-93.83	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
6194	-93.83	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
6195	-93.84	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
6196	-93.85	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
6197	-93.85	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
6198	-93.87	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
6199	-93.88	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
6200	-93.89	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
6201	-93.9	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
6202	-93.9	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
6203	-93.91	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
6204	-93.92	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
6205	-93.92	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
6206	-93.92	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
6207	-93.98	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
6208	-93.99	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
6209	-94.05	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
6210	-94.05	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
6211	-94.06	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
6212	-94.09	kd	CGS001-5727	PTCH1	-			
6213	-94.1	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
6214	-94.14	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
6215	-94.15	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
6216	-94.16	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
6217	-94.17	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
6218	-94.17	kd	CGS001-843	CASP10	Caspases			
6219	-94.18	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
6220	-94.2	oe	ccsbBroad304_01960	CASK	CASK family			
6221	-94.21	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
6222	-94.28	kd	CGS001-2919	CXCL1	Endogenous ligands			
6223	-94.31	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
6224	-94.34	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
6225	-94.36	oe	ccsbBroad304_02292	BCL2L11	-			
6226	-94.37	kd	CGS001-284119	PTRF	-			
6227	-94.38	cc		Potassium channel blocker	-			
6228	-94.4	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
6229	-94.41	kd	CGS001-9183	ZW10	-			
6230	-94.43	oe	ccsbBroad304_03641	ASF1B	-			
6231	-94.44	kd	CGS001-5932	RBBP8	-			
6232	-94.45	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
6233	-94.46	kd	CGS001-4697	NDUFA4	-			
6234	-94.49	kd	CGS001-4199	ME1	-			
6235	-94.5	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
6236	-94.51	cc		DNA polymerase inhibitor	-			
6237	-94.52	cc		X linked mental retardation group 2 LOF	-			
6238	-94.52	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
6239	-94.55	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
6240	-94.58	oe	ccsbBroad304_02370	HRSP12	-			
6241	-94.59	oe	ccsbBroad304_06651	NOV	-			
6242	-94.62	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
6243	-94.63	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
6244	-94.64	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
6245	-94.66	oe	ccsbBroad304_02173	ATG5	-			
6246	-94.66	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
6247	-94.68	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
6248	-94.69	kd	CGS001-5387	PMS2P3	-			
6249	-94.71	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
6250	-94.73	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
6251	-94.75	oe	ccsbBroad304_00033	ADSS	-			
6252	-94.77	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
6253	-94.78	oe	ccsbBroad304_07506	UBAP2L	-			
6254	-94.78	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
6255	-94.78	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
6256	-94.81	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
6257	-94.81	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
6258	-94.82	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
6259	-94.85	oe	ccsbBroad304_02677	PDAP1	-			
6260	-94.85	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
6261	-94.86	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
6262	-94.89	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
6263	-94.89	kd	CGS001-3482	IGF2R	CD molecules			
6264	-94.9	cc		PPAR receptor agonist	-			
6265	-94.95	kd	CGS001-3932	LCK	Src family			
6266	-94.95	kd	CGS001-57019	CIAPIN1	-			
6267	-94.99	kd	CGS001-55746	NUP133	-			
6268	-95.02	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
6269	-95.02	kd	CGS001-1756	DMD	-			
6270	-95.06	kd	CGS001-642	BLMH	-			
6271	-95.08	kd	CGS001-826	CAPNS1	EF-hand domain containing			
6272	-95.11	kd	CGS001-7165	TPD52L2	-			
6273	-95.11	kd	CGS001-6189	RPS3A	S ribosomal proteins			
6274	-95.12	kd	CGS001-4175	MCM6	-			
6275	-95.13	oe	ccsbBroad304_00956	LYZ	-			
6276	-95.14	oe	ccsbBroad304_05981	CDO1	-			
6277	-95.15	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
6278	-95.17	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
6279	-95.21	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
6280	-95.22	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
6281	-95.23	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
6282	-95.26	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
6283	-95.27	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
6284	-95.28	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
6285	-95.29	oe	ccsbBroad304_00250	CD19	CD molecules			
6286	-95.29	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
6287	-95.3	kd	CGS001-275	AMT	-			
6288	-95.37	oe	ccsbBroad304_02576	MLLT11	-			
6289	-95.38	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
6290	-95.39	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
6291	-95.39	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
6292	-95.4	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
6293	-95.41	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
6294	-95.42	oe	ccsbBroad304_02230	HERPUD1	-			
6295	-95.43	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
6296	-95.43	oe	ccsbBroad304_09284	UBE3B	-			
6297	-95.44	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
6298	-95.44	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
6299	-95.46	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
6300	-95.47	kd	CGS001-4907	NT5E	Adenosine turnover			
6301	-95.48	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
6302	-95.5	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
6303	-95.5	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6304	-95.51	kd	CGS001-55163	PNPO	-			
6305	-95.52	oe	ccsbBroad304_08797	FASTKD5	-			
6306	-95.54	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
6307	-95.56	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
6308	-95.58	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
6309	-95.58	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
6310	-95.6	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
6311	-95.61	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
6312	-95.65	kd	CGS001-23028	KDM1A	Histone demethylase			
6313	-95.7	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
6314	-95.7	kd	CGS001-55536	CDCA7L	-			
6315	-95.73	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
6316	-95.73	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
6317	-95.74	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
6318	-95.75	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
6319	-95.76	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
6320	-95.78	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
6321	-95.79	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
6322	-95.79	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
6323	-95.85	kd	CGS001-10641	NPRL2	-			
6324	-95.86	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6325	-95.87	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
6326	-95.88	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
6327	-95.91	oe	ccsbBroad304_03264	UBAP1	-			
6328	-95.94	oe	ccsbBroad304_06066	CTSL1	-			
6329	-95.94	kd	CGS001-2781	GNAZ	-			
6330	-95.95	kd	CGS001-79071	ELOVL6	-			
6331	-95.96	oe	ccsbBroad304_00146	BAD	-			
6332	-95.98	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
6333	-96.01	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
6334	-96.03	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
6335	-96.09	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
6336	-96.14	kd	CGS001-8741	TNFSF13	CD molecules			
6337	-96.15	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
6338	-96.15	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
6339	-96.15	oe	ccsbBroad304_07832	XPO7	Exportins			
6340	-96.16	oe	ccsbBroad304_00329	CLTA	-			
6341	-96.17	oe	ccsbBroad304_00819	IDH3B	-			
6342	-96.18	oe	ccsbBroad304_02801	CASP14	Caspases			
6343	-96.18	oe	ccsbBroad304_01469	RSU1	-			
6344	-96.19	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
6345	-96.2	kd	CGS001-5829	PXN	-			
6346	-96.21	kd	CGS001-79073	TMEM109	-			
6347	-96.22	kd	CGS001-6208	RPS14	S ribosomal proteins			
6348	-96.22	kd	CGS001-5162	PDHB	-			
6349	-96.23	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
6350	-96.24	kd	CGS001-2232	FDXR	-			
6351	-96.26	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
6352	-96.28	oe	ccsbBroad304_06639	NFYB	-			
6353	-96.28	oe	ccsbBroad304_02313	ACTR3	-			
6354	-96.28	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
6355	-96.29	kd	CGS001-9221	NOLC1	-			
6356	-96.32	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
6357	-96.32	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
6358	-96.34	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
6359	-96.34	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
6360	-96.34	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
6361	-96.36	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
6362	-96.39	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
6363	-96.39	kd	CGS001-9687	GREB1	-			
6364	-96.39	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6365	-96.41	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
6366	-96.42	oe	ccsbBroad304_02788	PRAME	-			
6367	-96.43	oe	ccsbBroad304_01038	MSRA	-			
6368	-96.45	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
6369	-96.48	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
6370	-96.49	kd	CGS001-3920	LAMP2	CD molecules			
6371	-96.51	oe	ccsbBroad304_02840	PISD	Decarboxylases			
6372	-96.53	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
6373	-96.59	kd	CGS001-6491	STIL	-			
6374	-96.6	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
6375	-96.61	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
6376	-96.64	oe	ccsbBroad304_01716	TSN	-			
6377	-96.64	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
6378	-96.65	oe	ccsbBroad304_01527	SGK1	SGK family			
6379	-96.66	oe	ccsbBroad304_08152	PSAT1	-			
6380	-96.66	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
6381	-96.7	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
6382	-96.71	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
6383	-96.71	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
6384	-96.73	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
6385	-96.74	oe	ccsbBroad304_01347	RAD1	-			
6386	-96.77	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
6387	-96.79	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
6388	-96.81	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
6389	-96.82	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
6390	-96.84	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
6391	-96.85	cc		Nucleoporin LOF	-			
6392	-96.85	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
6393	-96.85	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
6394	-96.87	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
6395	-96.89	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
6396	-96.89	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
6397	-96.89	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
6398	-96.89	kd	CGS001-51053	GMNN	-			
6399	-96.9	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
6400	-96.9	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
6401	-96.91	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
6402	-96.91	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
6403	-96.94	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
6404	-96.97	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
6405	-96.98	oe	ccsbBroad304_00486	EFNB2	Ephrins			
6406	-96.98	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6407	-96.99	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
6408	-97	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
6409	-97.04	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6410	-97.04	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
6411	-97.07	oe	ccsbBroad304_00657	GNG4	-			
6412	-97.08	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
6413	-97.08	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
6414	-97.08	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6415	-97.09	kd	CGS001-10873	ME3	-			
6416	-97.1	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
6417	-97.1	kd	CGS001-83999	KREMEN1	-			
6418	-97.12	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
6419	-97.13	kd	CGS001-27097	TAF5L	WD repeat domain containing			
6420	-97.13	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
6421	-97.14	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
6422	-97.14	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
6423	-97.15	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
6424	-97.15	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
6425	-97.16	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
6426	-97.16	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
6427	-97.16	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
6428	-97.17	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
6429	-97.18	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6430	-97.18	kd	CGS001-6793	STK10	SLK subfamily			
6431	-97.2	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
6432	-97.23	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6433	-97.25	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
6434	-97.26	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
6435	-97.26	kd	CGS001-335	APOA1	Apolipoproteins			
6436	-97.28	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
6437	-97.29	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6438	-97.32	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
6439	-97.32	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
6440	-97.33	kd	CGS001-2274	FHL2	-			
6441	-97.34	cc		Structural maintenance of chromosomes proteins LOF	-			
6442	-97.34	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6443	-97.35	kd	CGS001-5925	RB1	Endogenous ligands			
6444	-97.39	oe	ccsbBroad304_07145	ZFP161	-			
6445	-97.39	kd	CGS001-23161	SNX13	Sorting nexins			
6446	-97.39	kd	CGS001-4089	SMAD4	SMADs			
6447	-97.41	oe	ccsbBroad304_01593	SRP14	-			
6448	-97.41	kd	CGS001-8743	TNFSF10	CD molecules			
6449	-97.41	kd	CGS001-6184	RPN1	-			
6450	-97.42	kd	CGS001-84365	MKI67IP	-			
6451	-97.43	kd	CGS001-2864	FFAR1	Fatty acid receptors			
6452	-97.45	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
6453	-97.46	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
6454	-97.48	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
6455	-97.48	oe	ccsbBroad304_02340	SORBS3	-			
6456	-97.49	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
6457	-97.51	oe	ccsbBroad304_02017	PEX11A	-			
6458	-97.52	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
6459	-97.53	oe	ccsbBroad304_06253	GALT	-			
6460	-97.54	cc		P38 MAPK inhibitor	-			
6461	-97.55	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
6462	-97.57	cc		Estrogen receptor agonist	-			
6463	-97.57	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
6464	-97.57	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
6465	-97.59	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
6466	-97.61	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
6467	-97.62	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
6468	-97.64	oe	ccsbBroad304_01748	UFD1L	-			
6469	-97.65	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
6470	-97.66	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
6471	-97.66	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
6472	-97.7	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
6473	-97.72	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
6474	-97.72	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
6475	-97.72	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
6476	-97.73	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
6477	-97.75	cc		Proteasome Pathway LOF	-			
6478	-97.75	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
6479	-97.76	cc		SMAD family LOF	-			
6480	-97.76	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
6481	-97.77	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
6482	-97.8	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
6483	-97.8	kd	CGS001-8681	JMJD7-PLA2G4B	-			
6484	-97.81	cc		Bile acid	-			
6485	-97.82	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
6486	-97.83	kd	CGS001-11019	LIAS	-			
6487	-97.84	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
6488	-97.85	oe	ccsbBroad304_00446	DKC1	-			
6489	-97.85	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
6490	-97.86	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
6491	-97.9	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
6492	-97.91	kd	CGS001-222546	RFX6	-			
6493	-97.93	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
6494	-97.93	kd	CGS001-5920	RARRES3	-			
6495	-97.94	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
6496	-97.94	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
6497	-97.94	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
6498	-97.94	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
6499	-97.97	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
6500	-97.97	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
6501	-97.97	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
6502	-97.97	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
6503	-97.97	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
6504	-97.98	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
6505	-98.01	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
6506	-98.02	kd	CGS001-122618	PLD4	-			
6507	-98.04	oe	ccsbBroad304_06095	DFFB	-			
6508	-98.05	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
6509	-98.06	kd	CGS001-4090	SMAD5	SMADs			
6510	-98.07	kd	CGS001-4074	M6PR	-			
6511	-98.09	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
6512	-98.09	oe	ccsbBroad304_00811	ICAM1	CD molecules			
6513	-98.1	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
6514	-98.13	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
6515	-98.13	kd	CGS001-5108	PCM1	-			
6516	-98.15	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
6517	-98.15	kd	CGS001-7089	TLE2	WD repeat domain containing			
6518	-98.17	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
6519	-98.17	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
6520	-98.17	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
6521	-98.17	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
6522	-98.18	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
6523	-98.18	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
6524	-98.19	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
6525	-98.2	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
6526	-98.21	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
6527	-98.21	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
6528	-98.22	oe	ccsbBroad304_03591	ETNK1	-			
6529	-98.23	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
6530	-98.23	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
6531	-98.28	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
6532	-98.28	oe	ccsbBroad304_05963	CD44	CD molecules			
6533	-98.29	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
6534	-98.3	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
6535	-98.3	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
6536	-98.3	kd	CGS001-113451	ADC	-			
6537	-98.31	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6538	-98.32	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
6539	-98.32	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
6540	-98.33	oe	ccsbBroad304_09054	EGFL8	-			
6541	-98.35	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
6542	-98.36	oe	ccsbBroad304_06663	OAS1	-			
6543	-98.36	kd	CGS001-1841	DTYMK	-			
6544	-98.38	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
6545	-98.39	oe	ccsbBroad304_00423	DAXX	-			
6546	-98.39	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
6547	-98.39	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
6548	-98.4	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
6549	-98.41	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
6550	-98.42	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
6551	-98.42	kd	CGS001-5881	RAC3	Endogenous ligands			
6552	-98.44	oe	ccsbBroad304_01165	PDK1	-			
6553	-98.44	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
6554	-98.44	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
6555	-98.45	kd	CGS001-10898	CPSF4	-			
6556	-98.45	kd	CGS001-890	CCNA2	-			
6557	-98.46	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6558	-98.46	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
6559	-98.48	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
6560	-98.48	kd	CGS001-55662	HIF1AN	-			
6561	-98.49	kd	CGS001-9133	CCNB2	-			
6562	-98.5	oe	ccsbBroad304_06777	PRNP	CD molecules			
6563	-98.5	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
6564	-98.5	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
6565	-98.5	oe	ccsbBroad304_03554	NAT10	-			
6566	-98.51	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6567	-98.51	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
6568	-98.54	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
6569	-98.54	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
6570	-98.55	kd	CGS001-2879	GPX4	-			
6571	-98.56	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
6572	-98.57	oe	ccsbBroad304_08840	KIF9	Kinesins			
6573	-98.58	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
6574	-98.58	kd	CGS001-56005	C19ORF10	-			
6575	-98.59	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
6576	-98.6	kd	CGS001-204851	HIPK1	HIPK subfamily			
6577	-98.63	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
6578	-98.63	kd	CGS001-5660	PSAP	Endogenous ligands			
6579	-98.64	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
6580	-98.64	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6581	-98.65	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
6582	-98.66	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
6583	-98.66	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
6584	-98.66	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
6585	-98.67	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
6586	-98.69	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
6587	-98.69	kd	CGS001-10180	RBM6	G patch domain containing			
6588	-98.7	kd	CGS001-23076	RRP1B	-			
6589	-98.7	kd	CGS001-27161	EIF2C2	-			
6590	-98.71	kd	CGS001-327	APEH	Prolyl oligopeptidase			
6591	-98.72	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
6592	-98.74	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
6593	-98.75	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
6594	-98.75	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
6595	-98.76	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
6596	-98.76	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
6597	-98.76	kd	CGS001-1066	CES1	Carboxylesterases			
6598	-98.77	oe	ccsbBroad304_01398	RHEB	-			
6599	-98.79	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
6600	-98.81	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
6601	-98.81	oe	ccsbBroad304_13499	KSR2	RAF family			
6602	-98.81	kd	CGS001-9784	SNX17	Sorting nexins			
6603	-98.82	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
6604	-98.83	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
6605	-98.83	kd	CGS001-10765	KDM5B	Histone demethylases			
6606	-98.86	oe	ccsbBroad304_00632	GGCX	Carboxylases			
6607	-98.86	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
6608	-98.88	oe	ccsbBroad304_07275	PSMG1	-			
6609	-98.89	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6610	-98.92	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
6611	-98.93	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
6612	-98.93	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
6613	-98.94	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
6614	-98.94	kd	CGS001-23581	CASP14	Caspases			
6615	-98.95	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
6616	-98.95	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
6617	-98.95	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
6618	-98.99	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
6619	-99	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
6620	-99.01	oe	ccsbBroad304_00113	ASNS	-			
6621	-99.01	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
6622	-99.01	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
6623	-99.02	oe	ccsbBroad304_02990	LYPD3	-			
6624	-99.03	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6625	-99.03	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
6626	-99.04	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6627	-99.05	oe	ccsbBroad304_03961	SMURF2	-			
6628	-99.06	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
6629	-99.07	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
6630	-99.07	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
6631	-99.07	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
6632	-99.09	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
6633	-99.1	oe	ccsbBroad304_03235	TUBD1	Tubulins			
6634	-99.1	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
6635	-99.1	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
6636	-99.12	oe	ccsbBroad304_01147	PC	Carboxylases			
6637	-99.13	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
6638	-99.13	kd	CGS001-79902	NUP85	-			
6639	-99.15	kd	CGS001-22933	SIRT2	Histone deacetylases			
6640	-99.15	oe	ccsbBroad304_03497	TXNL4B	-			
6641	-99.15	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
6642	-99.16	cc		FGFR inhibitor	-			
6643	-99.16	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
6644	-99.16	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
6645	-99.16	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6646	-99.17	kd	CGS001-2197	FAU	S ribosomal proteins			
6647	-99.18	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6648	-99.19	kd	CGS001-54512	EXOSC4	-			
6649	-99.2	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6650	-99.22	kd	CGS001-25	ABL1	Abl family			
6651	-99.23	oe	ccsbBroad304_07600	NSA2	-			
6652	-99.23	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
6653	-99.23	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
6654	-99.23	kd	CGS001-9	NAT1	-			
6655	-99.26	oe	ccsbBroad304_06993	SRD5A1	-			
6656	-99.26	kd	CGS001-51750	RTEL1	-			
6657	-99.27	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
6658	-99.28	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
6659	-99.29	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
6660	-99.29	kd	CGS001-10285	SMNDC1	Tudor domain containing			
6661	-99.29	kd	CGS001-56916	SMARCAD1	-			
6662	-99.3	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
6663	-99.32	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
6664	-99.32	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
6665	-99.32	kd	CGS001-124535	HSF5	-			
6666	-99.32	kd	CGS001-2160	F11	Chymotrypsin			
6667	-99.33	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
6668	-99.34	cc		Interleukins GOF	-			
6669	-99.34	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
6670	-99.34	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6671	-99.34	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
6672	-99.35	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
6673	-99.35	kd	CGS001-51172	NAGPA	-			
6674	-99.37	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
6675	-99.37	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
6676	-99.37	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
6677	-99.38	cc		PARP inhibitor	-			
6678	-99.38	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
6679	-99.38	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
6680	-99.38	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
6681	-99.4	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
6682	-99.41	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
6683	-99.41	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
6684	-99.43	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
6685	-99.43	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
6686	-99.44	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
6687	-99.45	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
6688	-99.45	kd	CGS001-5255	PHKA1	-			
6689	-99.47	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6690	-99.47	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
6691	-99.47	kd	CGS001-7054	TH	Amino acid hydroxylases			
6692	-99.47	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
6693	-99.47	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
6694	-99.47	kd	CGS001-11140	CDC37	-			
6695	-99.48	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
6696	-99.48	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
6697	-99.48	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
6698	-99.48	kd	CGS001-5686	PSMA5	Proteasome subunits			
6699	-99.48	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
6700	-99.49	kd	CGS001-1827	RCAN1	-			
6701	-99.5	cc		GABA receptor antagonist	-			
6702	-99.5	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
6703	-99.5	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
6704	-99.51	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
6705	-99.51	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
6706	-99.51	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
6707	-99.51	oe	ccsbBroad304_01394	RFX4	-			
6708	-99.53	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
6709	-99.53	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
6710	-99.53	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
6711	-99.54	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
6712	-99.54	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
6713	-99.56	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
6714	-99.57	oe	ccsbBroad304_01052	MYB	-			
6715	-99.57	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6716	-99.57	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6717	-99.57	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
6718	-99.59	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
6719	-99.59	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
6720	-99.59	kd	CGS001-9637	FEZ2	-			
6721	-99.6	oe	ccsbBroad304_04190	CCDC92	-			
6722	-99.6	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6723	-99.6	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
6724	-99.6	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
6725	-99.6	kd	CGS001-1831	TSC22D3	-			
6726	-99.6	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
6727	-99.6	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6728	-99.61	oe	ccsbBroad304_14011	PAPSS1	-			
6729	-99.62	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
6730	-99.62	oe	ccsbBroad304_00518	ETFA	-			
6731	-99.62	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6732	-99.62	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
6733	-99.62	kd	CGS001-8226	HDHD1	-			
6734	-99.63	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
6735	-99.64	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
6736	-99.65	oe	ccsbBroad304_00020	ACY1	-			
6737	-99.65	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
6738	-99.65	kd	CGS001-10523	CHERP	G patch domain containing			
6739	-99.66	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
6740	-99.66	oe	ccsbBroad304_07363	AIFM1	-			
6741	-99.66	oe	ccsbBroad304_05749	A2M	-			
6742	-99.66	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
6743	-99.66	kd	CGS001-57048	PLSCR3	-			
6744	-99.67	kd	CGS001-81539	SLC38A1	System A-like transporters			
6745	-99.67	kd	CGS001-2967	GTF2H3	General transcription factors			
6746	-99.68	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
6747	-99.68	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
6748	-99.68	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
6749	-99.69	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6750	-99.69	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
6751	-99.69	oe	ccsbBroad304_01401	RIT1	-			
6752	-99.69	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
6753	-99.69	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
6754	-99.69	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
6755	-99.69	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
6756	-99.69	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
6757	-99.69	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
6758	-99.7	oe	ccsbBroad304_07088	TP53	-			
6759	-99.71	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
6760	-99.71	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
6761	-99.71	kd	CGS001-7276	TTR	-			
6762	-99.72	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
6763	-99.72	kd	CGS001-7100	TLR5	Toll-like receptor family			
6764	-99.73	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
6765	-99.73	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
6766	-99.73	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
6767	-99.73	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
6768	-99.73	kd	CGS001-5581	PRKCE	Eta subfamily			
6769	-99.73	kd	CGS001-5580	PRKCD	Delta subfamily			
6770	-99.73	kd	CGS001-23386	NUDCD3	-			
6771	-99.73	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
6772	-99.75	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
6773	-99.75	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
6774	-99.75	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
6775	-99.75	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
6776	-99.75	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
6777	-99.75	kd	CGS001-1152	CKB	-			
6778	-99.75	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
6779	-99.76	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
6780	-99.76	oe	ccsbBroad304_06789	PSEN2	Presenilin			
6781	-99.76	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
6782	-99.76	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
6783	-99.76	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
6784	-99.76	kd	CGS001-6646	SOAT1	-			
6785	-99.76	kd	CGS001-10427	SEC24B	-			
6786	-99.76	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6787	-99.76	kd	CGS001-3030	HADHA	-			
6788	-99.76	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
6789	-99.77	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
6790	-99.78	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
6791	-99.78	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6792	-99.78	kd	CGS001-79139	DERL1	-			
6793	-99.79	oe	ccsbBroad304_01556	SMARCB1	-			
6794	-99.79	oe	ccsbBroad304_08023	EIF2C1	-			
6795	-99.79	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
6796	-99.79	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6797	-99.79	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
6798	-99.79	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
6799	-99.81	cc		S100 calcium binding proteins LOF	-			
6800	-99.81	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
6801	-99.81	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
6802	-99.81	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6803	-99.81	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
6804	-99.82	oe	ccsbBroad304_00313	TBCB	-			
6805	-99.82	oe	ccsbBroad304_00152	BCAT2	-			
6806	-99.82	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
6807	-99.82	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
6808	-99.82	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
6809	-99.84	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
6810	-99.84	oe	ccsbBroad304_00085	APRT	-			
6811	-99.84	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
6812	-99.84	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
6813	-99.85	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
6814	-99.85	kd	CGS001-8575	PRKRA	-			
6815	-99.87	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
6816	-99.87	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
6817	-99.87	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
6818	-99.87	kd	CGS001-286380	FOXD4L3	-			
6819	-99.87	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
6820	-99.87	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
6821	-99.87	kd	CGS001-3832	KIF11	Kinesins			
6822	-99.88	oe	ccsbBroad304_01102	NMT1	-			
6823	-99.88	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
6824	-99.88	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
6825	-99.88	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
6826	-99.88	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
6827	-99.88	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
6828	-99.88	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6829	-99.88	kd	CGS001-7082	TJP1	-			
6830	-99.88	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
6831	-99.88	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
6832	-99.88	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
6833	-99.89	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
6834	-99.9	oe	ccsbBroad304_06916	SCP2	-			
6835	-99.9	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
6836	-99.9	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
6837	-99.9	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
6838	-99.9	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
6839	-99.9	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
6840	-99.9	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
6841	-99.9	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
6842	-99.9	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
6843	-99.9	kd	CGS001-2760	GM2A	-			
6844	-99.9	kd	CGS001-23149	FCHO1	-			
6845	-99.9	kd	CGS001-2147	F2	Endogenous ligands			
6846	-99.9	kd	CGS001-79733	E2F8	-			
6847	-99.9	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
6848	-99.91	oe	ccsbBroad304_02581	ASCC3	-			
6849	-99.91	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
6850	-99.91	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
6851	-99.91	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
6852	-99.91	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
6853	-99.91	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
6854	-99.91	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
6855	-99.91	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
6856	-99.91	kd	CGS001-25842	ASF1A	-			
6857	-99.91	oe	ccsbBroad304_07688	FAM114A2	-			
6858	-99.92	oe	ccsbBroad304_02405	TFG	-			
6859	-99.93	oe	ccsbBroad304_01769	VEGFB	-			
6860	-99.93	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
6861	-99.93	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
6862	-99.93	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
6863	-99.93	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
6864	-99.93	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
6865	-99.93	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
6866	-99.93	kd	CGS001-9451	EIF2AK3	PEK subfamily			
6867	-99.94	oe	ccsbBroad304_00617	GBA	-			
6868	-99.94	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
6869	-99.94	oe	ccsbBroad304_01675	TK1	-			
6870	-99.94	oe	ccsbBroad304_03056	MCTS1	-			
6871	-99.94	oe	ccsbBroad304_02271	LPGAT1	-			
6872	-99.94	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6873	-99.94	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6874	-99.94	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
6875	-99.94	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
6876	-99.94	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6877	-99.94	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
6878	-99.94	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
6879	-99.94	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
6880	-99.94	kd	CGS001-10128	LRPPRC	-			
6881	-99.94	kd	CGS001-81533	ITFG1	-			
6882	-99.94	kd	CGS001-54438	GFOD1	-			
6883	-99.95	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
6884	-99.96	cc		Bacterial cell wall synthesis inhibitor	-			
6885	-99.96	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
6886	-99.96	oe	ccsbBroad304_02815	SSBP2	-			
6887	-99.96	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
6888	-99.96	oe	ccsbBroad304_05890	BHMT	-			
6889	-99.96	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
6890	-99.96	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
6891	-99.96	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
6892	-99.96	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
6893	-99.96	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
6894	-99.96	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6895	-99.96	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
6896	-99.96	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
6897	-99.96	kd	CGS001-9200	PTPLA	-			
6898	-99.96	kd	CGS001-3930	LBR	Tudor domain containing			
6899	-99.96	kd	CGS001-2767	GNA11	-			
6900	-99.96	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6901	-99.96	kd	CGS001-1163	CKS1B	-			
6902	-99.96	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
6903	-99.97	cc		HIV protease inhibitor	-			
6904	-99.97	oe	ccsbBroad304_07820	SNW1	-			
6905	-99.97	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
6906	-99.97	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
6907	-99.97	oe	ccsbBroad304_01672	TIMP2	-			
6908	-99.97	oe	ccsbBroad304_01379	RBBP6	-			
6909	-99.97	oe	ccsbBroad304_06845	RARRES3	-			
6910	-99.97	oe	ccsbBroad304_03570	QRSL1	-			
6911	-99.97	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
6912	-99.97	oe	ccsbBroad304_09756	PAQR7	-			
6913	-99.97	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
6914	-99.97	oe	ccsbBroad304_07208	NRIP1	-			
6915	-99.97	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
6916	-99.97	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
6917	-99.97	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
6918	-99.97	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6919	-99.97	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
6920	-99.97	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
6921	-99.97	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
6922	-99.97	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
6923	-99.97	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
6924	-99.97	oe	ccsbBroad304_08596	EAPP	-			
6925	-99.97	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
6926	-99.97	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
6927	-99.97	oe	ccsbBroad304_00106	ARRB1	-			
6928	-99.97	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
6929	-99.97	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
6930	-99.97	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
6931	-99.97	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
6932	-99.97	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
6933	-99.97	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
6934	-99.97	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6935	-99.97	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
6936	-99.97	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
6937	-99.97	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
6938	-99.97	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
6939	-99.97	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
6940	-99.97	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
6941	-99.97	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
6942	-99.97	kd	CGS001-7485	WRB	-			
6943	-99.97	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
6944	-99.97	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
6945	-99.97	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
6946	-99.97	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
6947	-99.97	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
6948	-99.97	kd	CGS001-9467	SH3BP5	-			
6949	-99.97	kd	CGS001-9871	SEC24D	-			
6950	-99.97	kd	CGS001-6277	S100A6	EF-hand domain containing			
6951	-99.97	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
6952	-99.97	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
6953	-99.97	kd	CGS001-5230	PGK1	-			
6954	-99.97	kd	CGS001-5824	PEX19	-			
6955	-99.97	kd	CGS001-4893	NRAS	RAS subfamily			
6956	-99.97	kd	CGS001-4782	NFIC	-			
6957	-99.97	kd	CGS001-4351	MPI	-			
6958	-99.97	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
6959	-99.97	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
6960	-99.97	kd	CGS001-3672	ITGA1	Integrins			
6961	-99.97	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
6962	-99.97	kd	CGS001-1504	CTRB1	-			
6963	-99.97	kd	CGS001-125965	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
6964	-99.97	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6965	-99.97	kd	CGS001-9738	CCP110	-			
6966	-99.97	kd	CGS001-375	ARF1	ADP-ribosylation factors			
6967	-99.97	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
6968	-99.97	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
6969	-99.97	kd	CGS001-158	ADSL	-			
6970	-99.97	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
6971	-99.97	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
6972	-100	cc		Thromboxane receptor antagonist	-			
