Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	99.99	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
2	99.98	oe	ccsbBroad304_00964	SMAD7	SMADs			
3	99.98	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
4	99.98	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
5	99.98	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
6	99.98	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
7	99.98	oe	ccsbBroad304_03308	YTHDF2	-			
8	99.98	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
9	99.98	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
10	99.98	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
11	99.98	oe	ccsbBroad304_02058	PLOD3	-			
12	99.98	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
13	99.98	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
14	99.98	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
15	99.98	oe	ccsbBroad304_00975	MAT2A	-			
16	99.98	oe	ccsbBroad304_08840	KIF9	Kinesins			
17	99.98	oe	ccsbBroad304_06458	IRF3	-			
18	99.98	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
19	99.98	oe	ccsbBroad304_00795	HSF2	-			
20	99.98	oe	ccsbBroad304_00644	GCLC	-			
21	99.98	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
22	99.98	oe	ccsbBroad304_00532	F11	Chymotrypsin			
23	99.98	oe	ccsbBroad304_02143	CNOT8	-			
24	99.98	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
25	99.98	oe	ccsbBroad304_02292	BCL2L11	-			
26	99.98	oe	ccsbBroad304_00146	BAD	-			
27	99.98	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
28	99.98	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
29	99.98	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
30	99.98	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
31	99.98	cp	BRD-K44353683	nateglinide	Insulin secretagogue		ABCC8, KCNJ11, CYP3A4, INS, KCNJ10, PPARG	Insulin secretagogue
32	99.98	cp	BRD-A49172652	lansoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4, CYP3A5	ATPase inhibitor
33	99.98	cp	BRD-K11630072	carmofur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
34	99.98	cp	BRD-K85925969	zalcitabine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
35	99.98	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
36	99.98	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
37	99.98	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
38	99.98	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
39	99.98	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
40	99.98	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
41	99.98	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
42	99.98	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
43	99.98	kd	CGS001-6469	SHH	-			
44	99.98	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
45	99.98	kd	CGS001-83694	RPS6KL1	RSKL family			
46	99.98	kd	CGS001-79170	PRR15L	-			
47	99.98	kd	CGS001-85315	PAQR8	-			
48	99.98	kd	CGS001-4841	NONO	RNA binding motif (RRM) containing			
49	99.98	kd	CGS001-28512	NKIRAS1	-			
50	99.98	kd	CGS001-64863	METTL4	-			
51	99.98	kd	CGS001-84539	MCHR2	GPCR / Class A : MCH receptors			
52	99.98	kd	CGS001-3176	HNMT	-			
53	99.98	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
54	99.98	kd	CGS001-2937	GSS	-			
55	99.98	kd	CGS001-57459	GATAD2B	GATA zinc finger domain containing			
56	99.98	kd	CGS001-23401	FRAT2	-			
57	99.98	kd	CGS001-1305	COL13A1	Collagens			
58	99.98	kd	CGS001-55536	CDCA7L	-			
59	99.98	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
60	99.98	kd	CGS001-85027	C5ORF62	-			
61	99.96	cc		Targets of VEGFR inhibitors GOF	-			
62	99.96	cc		Protein phosphatase catalytic subunits LOF	-			
63	99.96	cc		Sodium channel blocker	-			
64	99.96	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
65	99.96	oe	ccsbBroad304_04153	PHF17	-			
66	99.96	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
67	99.96	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
68	99.96	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
69	99.96	oe	ccsbBroad304_03023	CRCP	-			
70	99.96	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
71	99.96	cp	BRD-K01649396	indatraline	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine transporter inhibitor
72	99.96	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
73	99.96	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
74	99.96	kd	CGS001-57761	TRIB3	Trbl family			
75	99.96	kd	CGS001-6895	TARBP2	-			
76	99.96	kd	CGS001-8435	SOAT2	-			
77	99.96	kd	CGS001-57154	SMURF1	-			
78	99.96	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
79	99.96	kd	CGS001-10928	RALBP1	-			
80	99.96	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
81	99.96	kd	CGS001-10957	PNRC1	-			
82	99.96	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
83	99.96	kd	CGS001-54815	GATAD2A	GATA zinc finger domain containing			
84	99.95	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
85	99.95	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
86	99.95	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
87	99.95	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
88	99.95	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
89	99.95	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
90	99.95	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
91	99.95	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
92	99.95	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
93	99.95	kd	CGS001-27336	HTATSF1	RNA binding motif (RRM) containing			
94	99.95	kd	CGS001-51022	GLRX2	-			
95	99.95	kd	CGS001-2243	FGA	Endogenous ligands			
96	99.95	kd	CGS001-694	BTG1	-			
97	99.94	oe	ccsbBroad304_01651	TCF7L2	-			
98	99.94	oe	ccsbBroad304_04064	PRR15L	-			
99	99.94	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
100	99.94	oe	ccsbBroad304_00418	CD55	CD molecules			
101	99.94	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
102	99.94	kd	CGS001-6658	SOX3	SRY (sex determining region Y)-boxes			
103	99.94	kd	CGS001-9767	PHF16	-			
104	99.94	kd	CGS001-29982	NRBF2	-			
105	99.94	kd	CGS001-7025	NR2F1	COUP-TF-like receptors			
106	99.94	kd	CGS001-3930	LBR	Tudor domain containing			
107	99.94	kd	CGS001-55608	ANKRD10	Ankyrin repeat domain containing			
108	99.93	oe	ccsbBroad304_07128	VHL	-			
109	99.93	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
110	99.93	oe	ccsbBroad304_02686	COPZ1	-			
111	99.93	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
112	99.93	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
113	99.93	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
114	99.93	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
115	99.93	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
116	99.93	kd	CGS001-3225	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
117	99.93	kd	CGS001-405	ARNT	Basic helix-loop-helix proteins			
118	99.91	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
119	99.91	oe	ccsbBroad304_00009	ACLY	-			
120	99.91	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
121	99.91	kd	CGS001-5066	PAM	-			
122	99.9	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
123	99.9	oe	ccsbBroad304_01519	SET	-			
124	99.9	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
125	99.9	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
126	99.9	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
127	99.9	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
128	99.9	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
129	99.9	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
130	99.9	kd	CGS001-6821	SUOX	-			
131	99.9	kd	CGS001-3162	HMOX1	Haem oxygenase			
132	99.89	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
133	99.89	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
134	99.89	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
135	99.89	kd	CGS001-23378	RRP8	-			
136	99.89	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
137	99.89	kd	CGS001-218	ALDH3A1	Aldehyde dehydrogenases			
138	99.88	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
139	99.88	cp	BRD-K22009844	phenprobamate	Muscle relaxant			Muscle relaxant
140	99.88	kd	CGS001-51588	PIAS4	Zinc fingers, MIZ-type			
141	99.88	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
142	99.88	kd	CGS001-23139	MAST2	MAST family			
143	99.88	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
144	99.88	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
145	99.88	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
146	99.87	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
147	99.87	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
148	99.87	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
149	99.87	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
150	99.87	kd	CGS001-10721	POLQ	DNA polymerases			
151	99.85	kd	CGS001-171017	ZNF384	Zinc fingers, C2H2-type			
152	99.85	kd	CGS001-2072	ERCC4	-			
153	99.84	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
154	99.84	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
155	99.84	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
156	99.84	kd	CGS001-6519	SLC3A1	SLC3 family			
157	99.83	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
158	99.83	kd	CGS001-5445	PON2	Paraoxonases			
159	99.83	kd	CGS001-53836	GPR87	GPCR / Class A : Orphans			
160	99.82	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
161	99.82	cp	BRD-K34508425	KUC103898N	-666			-666
162	99.82	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
163	99.82	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
164	99.82	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
165	99.82	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
166	99.82	kd	CGS001-118442	GPR62	GPCR / Class A : Orphans			
167	99.82	kd	CGS001-1843	DUSP1	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
168	99.82	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
169	99.81	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
170	99.81	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
171	99.81	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
172	99.81	kd	CGS001-6118	RPA2	-			
173	99.79	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
174	99.79	oe	ccsbBroad304_02737	JMJD6	-			
175	99.79	kd	CGS001-10451	VAV3	Rho guanine nucleotide exchange factors			
176	99.79	kd	CGS001-7004	TEAD4	-			
177	99.79	kd	CGS001-6720	SREBF1	Basic helix-loop-helix proteins			
178	99.79	kd	CGS001-7905	REEP5	Receptor accessory proteins			
179	99.79	kd	CGS001-5091	PC	Carboxylases			
180	99.79	kd	CGS001-835	CASP2	Caspases			
181	99.79	kd	CGS001-25966	C2CD2	-			
182	99.78	oe	ccsbBroad304_02845	PRPF6	-			
183	99.78	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
184	99.78	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
185	99.78	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
186	99.78	kd	CGS001-124583	CANT1	-			
187	99.78	kd	CGS001-2683	B4GALT1	Beta 4-glycosyltransferases			
188	99.78	kd	CGS001-87	ACTN1	EF-hand domain containing			
189	99.77	oe	ccsbBroad304_04891	TMEM174	-			
190	99.77	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
191	99.77	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
192	99.76	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
193	99.76	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
194	99.76	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
195	99.76	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
196	99.76	kd	CGS001-2261	FGFR3	Type V RTKs: FGF (fibroblast growth factor) receptor family			
197	99.74	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
198	99.74	kd	CGS001-4282	MIF	-			
199	99.74	kd	CGS001-1763	DNA2	-			
200	99.73	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
201	99.73	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
202	99.73	cp	BRD-A52282606	lacidipine	Calcium channel blocker		CACNA1C	Calcium channel blocker
203	99.73	cp	BRD-K82143716	flucytosine	Antifungal		DNMT1	Antifungal
204	99.73	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
205	99.73	kd	CGS001-10308	ZNF267	Zinc fingers, C2H2-type			
206	99.73	kd	CGS001-55312	RFK	-			
207	99.73	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
208	99.73	kd	CGS001-1201	CLN3	-			
209	99.72	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
210	99.72	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
211	99.72	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
212	99.72	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
213	99.72	kd	CGS001-6887	TAL2	Basic helix-loop-helix proteins			
214	99.72	kd	CGS001-4707	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
215	99.72	kd	CGS001-9290	GPR55	GPCR / Class A : Orphans			
216	99.72	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
217	99.71	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
218	99.71	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
219	99.71	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
220	99.71	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
221	99.71	kd	CGS001-6257	RXRB	Retinoid X receptors			
222	99.7	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
223	99.7	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
224	99.7	kd	CGS001-3131	HLF	-			
225	99.69	oe	ccsbBroad304_01605	SSX2	-			
226	99.69	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
227	99.68	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
228	99.68	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
229	99.68	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
230	99.68	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
231	99.68	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
232	99.68	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
233	99.68	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
234	99.67	oe	ccsbBroad304_07280	LAMTOR3	-			
235	99.67	kd	CGS001-1677	DFFB	-			
236	99.66	cp	BRD-K49404994	levetiracetam	Calcium channel blocker		SV2A, CACNA1B, SCN1A	Calcium channel blocker
237	99.66	kd	CGS001-2048	EPHB2	Type XIII RTKs: Ephrin receptor family			
238	99.66	kd	CGS001-51027	BOLA1	-			
239	99.64	cc		FGFR inhibitor	-			
240	99.64	kd	CGS001-7750	ZMYM2	Zinc fingers, MYM type			
241	99.63	cp	BRD-K85090592	pilocarpine	Acetylcholine receptor agonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor agonist
242	99.63	kd	CGS001-134187	POU5F2	Homeoboxes / POU class			
243	99.62	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
244	99.62	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
245	99.61	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
246	99.61	kd	CGS001-8148	TAF15	RNA binding motif (RRM) containing			
247	99.6	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
248	99.6	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
249	99.6	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
250	99.6	kd	CGS001-51271	UBAP1	-			
251	99.6	kd	CGS001-2876	GPX1	-			
252	99.59	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
253	99.58	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
254	99.57	kd	CGS001-5428	POLG	DNA polymerases			
255	99.57	kd	CGS001-3665	IRF7	-			
256	99.57	kd	CGS001-2130	EWSR1	RNA binding motif (RRM) containing			
257	99.57	kd	CGS001-148327	CREB3L4	basic leucine zipper proteins			
258	99.56	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
259	99.56	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
260	99.56	kd	CGS001-10135	NAMPT	-			
261	99.55	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
262	99.55	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
263	99.54	oe	ccsbBroad304_01038	MSRA	-			
264	99.54	oe	ccsbBroad304_03357	RASD1	-			
265	99.54	oe	ccsbBroad304_00063	AMPD2	-			
266	99.54	cp	BRD-K56450366	NSC-94258	Antineoplastic		AKR1B1, CYP19A1, HSD17B1	Antineoplastic
267	99.53	cp	BRD-A56892734	esomeprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
268	99.53	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
269	99.52	kd	CGS001-3995	FADS3	Fatty acid desaturases			
270	99.5	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
271	99.48	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
272	99.48	kd	CGS001-5352	PLOD2	-			
273	99.47	oe	ccsbBroad304_06695	PCK2	-			
274	99.47	kd	CGS001-26959	HBP1	-			
275	99.46	oe	ccsbBroad304_03934	LEPRE1	-			
276	99.45	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
277	99.45	kd	CGS001-7150	TOP1	DNA Topoisomerases			
278	99.45	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
279	99.44	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
280	99.43	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
281	99.43	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
282	99.42	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
283	99.42	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
284	99.42	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
285	99.41	cc		Nucleoside reverse transcriptase inhibitor	-			
286	99.4	oe	ccsbBroad304_01617	STX4	-			
287	99.4	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
288	99.39	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
289	99.38	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
290	99.38	oe	ccsbBroad304_00226	CAV1	-			
291	99.37	oe	ccsbBroad304_06642	NIT1	-			
292	99.36	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
293	99.36	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
294	99.36	kd	CGS001-126208	ZNF787	Zinc fingers, C2H2-type			
295	99.35	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
296	99.34	oe	ccsbBroad304_09225	BUD13	-			
297	99.34	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
298	99.34	kd	CGS001-3373	HYAL1	-			
299	99.32	kd	CGS001-6472	SHMT2	-			
300	99.32	kd	CGS001-55226	NAT10	-			
301	99.32	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
302	99.31	kd	CGS001-6196	RPS6KA2	RSK subfamily			
303	99.3	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
304	99.28	kd	CGS001-930	CD19	CD molecules			
305	99.27	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
306	99.27	oe	ccsbBroad304_02047	AP1S2	-			
307	99.26	oe	ccsbBroad304_07363	AIFM1	-			
308	99.26	oe	ccsbBroad304_07478	CCP110	-			
309	99.26	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
310	99.26	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
311	99.26	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
312	99.26	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
313	99.25	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
314	99.25	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
315	99.25	kd	CGS001-23530	NNT	-			
316	99.25	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
317	99.23	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
318	99.22	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
319	99.21	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
320	99.2	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
321	99.19	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
322	99.19	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
323	99.17	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
324	99.17	kd	CGS001-84365	MKI67IP	-			
325	99.15	kd	CGS001-3939	LDHA	-			
326	99.14	oe	ccsbBroad304_07349	MAP7	-			
327	99.14	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
328	99.14	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
329	99.13	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
330	99.13	kd	CGS001-5992	RFX4	-			
331	99.12	oe	ccsbBroad304_07704	SUB1	-			
332	99.12	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
333	99.12	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
334	99.11	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
335	99.11	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
336	99.1	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
337	99.08	cp	BRD-K50938287	sumatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1A, HTR1F, HTR1E, HTR5A, HTR6, HTR7	Serotonin receptor agonist
338	99.08	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
339	99.08	kd	CGS001-84759	PCGF1	Polycomb group ring fingers			
340	99.08	kd	CGS001-65123	INTS3	-			
341	99.08	kd	CGS001-54805	CNNM2	-			
342	99.07	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
343	99.07	kd	CGS001-5019	OXCT1	-			
344	99.06	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
345	99.06	kd	CGS001-23647	ARFIP2	-			
346	99.02	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
347	99.02	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
348	99.02	kd	CGS001-4012	LNPEP	Aminopeptidase N			
349	99.01	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
350	99	oe	ccsbBroad304_01662	TFDP2	-			
351	99	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
352	99	oe	ccsbBroad304_03047	BZW2	-			
353	99	kd	CGS001-4668	NAGA	-			
354	98.94	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
355	98.94	oe	ccsbBroad304_06852	RBP4	Lipocalins			
356	98.94	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
357	98.94	kd	CGS001-1719	DHFR	Oxidoreductases			
358	98.93	kd	CGS001-26292	MYCBP	-			
359	98.92	kd	CGS001-624	BDKRB2	Bradykinin receptors			
360	98.91	kd	CGS001-8767	RIPK2	Receptor interacting protein kinase (RIPK) family			
361	98.9	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
362	98.89	oe	ccsbBroad304_01102	NMT1	-			
363	98.89	kd	CGS001-8522	GAS7	-			
364	98.88	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
365	98.88	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
366	98.87	oe	ccsbBroad304_00650	GNA11	-			
367	98.87	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
368	98.87	kd	CGS001-6241	RRM2	Ribonucleoside-diphosphate reductases			
369	98.87	kd	CGS001-3385	ICAM3	CD molecules			
370	98.86	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
371	98.86	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
372	98.86	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
373	98.86	kd	CGS001-9318	COPS2	-			
374	98.84	oe	ccsbBroad304_02157	MED21	-			
375	98.83	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
376	98.83	cp	BRD-A37052580	physostigmine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Cholinesterase inhibitor
377	98.82	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
378	98.82	cp	BRD-K84566043	fenpiverinium	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
379	98.78	kd	CGS001-2565	GABRG1	GABA receptors			
380	98.77	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
381	98.77	kd	CGS001-8531	CSDA	-			
382	98.76	kd	CGS001-5194	PEX13	-			
383	98.74	oe	ccsbBroad304_00106	ARRB1	-			
384	98.74	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
385	98.74	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
386	98.73	kd	CGS001-7298	TYMS	Methyltransferases			
387	98.73	kd	CGS001-4782	NFIC	-			
388	98.73	kd	CGS001-84811	BUD13	-			
389	98.73	oe	ccsbBroad304_08217	SCCPDH	-			
390	98.72	kd	CGS001-5928	RBBP4	WD repeat domain containing			
391	98.71	kd	CGS001-10477	UBE2E3	Ubiquitin-conjugating enzymes E2			
392	98.71	kd	CGS001-2161	F12	Chymotrypsin			
393	98.7	oe	ccsbBroad304_09006	RPF1	-			
394	98.7	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
395	98.68	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
396	98.65	kd	CGS001-5584	PRKCI	Iota subfamily			
397	98.63	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
398	98.63	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
399	98.62	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
400	98.62	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
401	98.62	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
402	98.61	kd	CGS001-203	AK1	Adenylate kinases			
403	98.59	oe	ccsbBroad304_09054	EGFL8	-			
404	98.59	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
405	98.59	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
406	98.58	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
407	98.57	kd	CGS001-1154	CISH	SH2 domain containing			
408	98.55	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
409	98.53	kd	CGS001-3755	KCNG1	Voltage-gated potassium channels			
410	98.51	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
411	98.51	kd	CGS001-58533	SNX6	Sorting nexins			
412	98.51	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
413	98.5	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
414	98.5	kd	CGS001-54807	ZNF586	Zinc fingers, C2H2-type			
415	98.5	kd	CGS001-30	ACAA1	-			
416	98.49	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
417	98.48	kd	CGS001-9961	MVP	-			
418	98.48	kd	CGS001-2071	ERCC3	General transcription factors			
419	98.48	kd	CGS001-8573	CASK	CASK family			
420	98.47	kd	CGS001-6117	RPA1	-			
421	98.46	oe	ccsbBroad304_06998	SRPK1	SRPK family			
422	98.45	kd	CGS001-29937	NENF	-			
423	98.45	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
424	98.4	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
425	98.4	kd	CGS001-3030	HADHA	-			
426	98.37	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
427	98.36	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
428	98.36	cp	BRD-K99447003	enalaprilat	ACE inhibitor		ACE	ACE inhibitor
429	98.35	oe	ccsbBroad304_00550	FDXR	-			
430	98.34	cp	BRD-K29113274	ketoconazole	Sterol demethylase inhibitor		AR, CYP19A1, CYP21A2, CYP2C19, CYP3A5, CYP3A7, KCNA10	Sterol demethylase inhibitor
431	98.33	kd	CGS001-7108	TM7SF2	-			
432	98.32	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
433	98.32	kd	CGS001-462	SERPINC1	Serine (or cysteine) peptidase inhibitors			
434	98.32	kd	CGS001-1500	CTNND1	Catenins			
435	98.31	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
436	98.31	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
437	98.3	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
438	98.3	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
439	98.29	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
440	98.29	oe	ccsbBroad304_06671	OPA1	-			
441	98.28	kd	CGS001-6309	SC5DL	-			
442	98.27	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
443	98.26	oe	ccsbBroad304_02738	RRS1	-			
444	98.23	oe	ccsbBroad304_00420	DAP	-			
445	98.22	kd	CGS001-185	AGTR1	Angiotensin receptors			
446	98.2	oe	ccsbBroad304_06174	ERCC1	-			
447	98.2	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
448	98.17	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
449	98.14	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
450	98.13	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
451	98.12	kd	CGS001-8727	CTNNAL1	Catenins			
452	98.11	oe	ccsbBroad304_00392	CTLA4	CD molecules			
453	98.1	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
454	98.09	cp	BRD-K33483813	actarit	Interleukin receptor agonist			Interleukin receptor agonist
455	98.09	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
456	98.09	kd	CGS001-3017	HIST1H2BD	Histones / Replication-dependent			
457	98.08	cp	BRD-K41903098	diphenoxylate	Opioid receptor agonist		OPRM1, OPRD1	Opioid receptor agonist
458	98.07	oe	ccsbBroad304_07531	TANK	-			
459	98.07	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
460	98.06	oe	ccsbBroad304_00390	CTGF	-			
461	98.05	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
462	98.05	oe	ccsbBroad304_03739	NRIP3	-			
463	98.04	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
464	98.02	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
465	98.02	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
466	98.02	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
467	98.02	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
468	98	cp	BRD-A48261811	argatroban	Thrombin inhibitor		F2, CYP3A5	Thrombin inhibitor
469	97.99	cc		Wnt family LOF	-			
470	97.96	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
471	97.96	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
472	97.95	oe	ccsbBroad304_00962	SMAD4	SMADs			
473	97.95	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
474	97.95	kd	CGS001-2168	FABP1	Fatty acid-binding proteins			
475	97.94	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
476	97.92	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
477	97.92	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
478	97.91	kd	CGS001-10657	KHDRBS1	-			
479	97.91	kd	CGS001-81533	ITFG1	-			
480	97.9	kd	CGS001-718	C3	Endogenous ligands			
481	97.89	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
482	97.88	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
483	97.85	kd	CGS001-83440	ADPGK	-			
484	97.84	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
485	97.84	kd	CGS001-8635	RNASET2	-			
486	97.83	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
487	97.81	kd	CGS001-337867	UBAC2	-			
488	97.8	kd	CGS001-2098	ESD	-			
489	97.79	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
490	97.79	oe	ccsbBroad304_08605	PBK	TOPK family			
491	97.78	kd	CGS001-51719	CAB39	-			
492	97.74	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
493	97.74	kd	CGS001-79001	VKORC1	Oxidoreductases			
494	97.73	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
495	97.7	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
496	97.7	kd	CGS001-7082	TJP1	-			
497	97.69	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
498	97.69	kd	CGS001-573	BAG1	-			
499	97.68	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
500	97.67	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
501	97.67	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
502	97.64	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
503	97.64	kd	CGS001-9891	NUAK1	NuaK subfamily			
504	97.61	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
505	97.61	kd	CGS001-10608	MXD4	Basic helix-loop-helix proteins			
506	97.6	kd	CGS001-7965	AIMP2	-			
507	97.59	oe	ccsbBroad304_00954	LYN	Src family			
508	97.59	kd	CGS001-3663	IRF5	-			
509	97.58	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
510	97.56	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
511	97.54	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
512	97.54	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
513	97.54	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
514	97.52	oe	ccsbBroad304_07688	FAM114A2	-			
515	97.51	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
516	97.5	oe	ccsbBroad304_02203	MAD2L1BP	-			
517	97.48	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
518	97.48	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
519	97.48	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
520	97.48	kd	CGS001-8804	CREG1	-			
521	97.47	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
522	97.46	cc		Bacterial DNA gyrase inhibitor	-			
523	97.46	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
524	97.46	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
525	97.41	kd	CGS001-3689	ITGB2	Integrins			
526	97.4	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
527	97.4	kd	CGS001-467	ATF3	basic leucine zipper proteins			
528	97.39	kd	CGS001-6541	SLC7A1	SLC7 family			
529	97.37	oe	ccsbBroad304_03604	ENOSF1	-			
530	97.34	kd	CGS001-427	ASAH1	Acid ceramidase			
531	97.33	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
532	97.32	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
533	97.31	kd	CGS001-23224	SYNE2	-			
534	97.29	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
535	97.29	kd	CGS001-638	BIK	-			
536	97.28	kd	CGS001-3799	KIF5B	Kinesins			
537	97.27	kd	CGS001-51776	ZAK	MLK subfamily			
538	97.21	oe	ccsbBroad304_01401	RIT1	-			
539	97.2	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
540	97.14	kd	CGS001-9459	ARHGEF6	Rho guanine nucleotide exchange factors			
541	97.13	kd	CGS001-10491	CRTAP	-			
542	97.12	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
543	97.12	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
544	97.09	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
545	97.09	oe	ccsbBroad304_07088	TP53	-			
546	97.08	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
547	97.07	cp	BRD-K32311154	nifekalant	Potassium channel blocker			Potassium channel blocker
548	97.06	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
549	97.02	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
550	97	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
551	97	kd	CGS001-80762	NDFIP1	-			
552	96.99	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
553	96.98	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
554	96.95	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
555	96.95	cp	BRD-K51730347	diphencyprone	Immunostimulant			Immunostimulant
556	96.94	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
557	96.93	kd	CGS001-147179	WIPF2	-			
558	96.93	kd	CGS001-89882	TPD52L3	-			
559	96.9	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
560	96.9	kd	CGS001-8548	BLZF1	-			
561	96.88	oe	ccsbBroad304_06494	KLRC1	CD molecules			
562	96.86	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
563	96.83	kd	CGS001-55437	STRADB	STLK subfamily			
564	96.8	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
565	96.79	kd	CGS001-79006	METRN	-			
566	96.76	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
567	96.72	kd	CGS001-4942	OAT	-			
568	96.71	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
569	96.71	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
570	96.67	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
571	96.67	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
572	96.65	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
573	96.64	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
574	96.63	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
575	96.62	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
576	96.6	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
577	96.6	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
578	96.57	oe	ccsbBroad304_06278	GK	Glycerol kinases			
579	96.56	kd	CGS001-9415	FADS2	Fatty acid desaturases			
580	96.55	kd	CGS001-5699	PSMB10	Proteasome (prosome, macropain) subunits			
581	96.55	kd	CGS001-995	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
582	96.53	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
583	96.52	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
584	96.51	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
585	96.48	kd	CGS001-840	CASP7	Caspases			
586	96.4	kd	CGS001-256364	EML3	WD repeat domain containing			
587	96.37	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
588	96.33	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
589	96.33	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
590	96.33	kd	CGS001-7727	ZNF174	Zinc fingers, C2H2-type			
591	96.32	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
592	96.29	cp	BRD-A42423104	benproperine	Antitussive			Antitussive
593	96.29	kd	CGS001-9261	MAPKAPK2	MAPKAPK subfamily			
594	96.27	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
595	96.23	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
596	96.21	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
597	96.15	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
598	96.14	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
599	96.13	oe	ccsbBroad304_06420	ICAM3	CD molecules			
600	96.12	oe	ccsbBroad304_02361	MFSD10	-			
601	96.12	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
602	96.12	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
603	96.1	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
604	96.08	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
605	96.06	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
606	96.05	kd	CGS001-9759	HDAC4	Histone deacetylases			
607	96.01	kd	CGS001-3909	LAMA3	Laminins			
608	95.99	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
609	95.96	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
610	95.93	kd	CGS001-2356	FPGS	-			
611	95.91	cp	BRD-K44094599	tacrolimus	Calcineurin inhibitor		FKBP1A, CYP3A5, CYP3A7	Calcineurin inhibitor
612	95.9	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
613	95.9	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
614	95.9	kd	CGS001-1635	DCTD	-			
615	95.83	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
616	95.81	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
617	95.81	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
618	95.81	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
619	95.79	kd	CGS001-10198	MPHOSPH9	-			
620	95.78	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
621	95.76	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
622	95.75	kd	CGS001-23013	SPEN	RNA binding motif (RRM) containing			
623	95.74	kd	CGS001-10810	WASF3	-			
624	95.73	cc		Sterol demethylase inhibitor	-			
625	95.73	oe	ccsbBroad304_02367	CALCOCO2	-			
626	95.73	kd	CGS001-1028	CDKN1C	-			
627	95.72	kd	CGS001-333929	SNAI3	Snail homologs			
628	95.7	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
629	95.69	oe	ccsbBroad304_02964	TIMM9	-			
630	95.69	cp	BRD-K96740444	itopride	Dopamine receptor antagonist		DRD2, ACHE, CHRM3	Dopamine receptor antagonist
631	95.64	kd	CGS001-2159	F10	Chymotrypsin			
632	95.63	kd	CGS001-3651	PDX1	Homeoboxes / ANTP class : HOXL subclass			
633	95.62	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
634	95.62	oe	ccsbBroad304_00811	ICAM1	CD molecules			
635	95.6	oe	ccsbBroad304_06291	GNAI1	-			
636	95.58	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
637	95.53	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
638	95.5	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
639	95.5	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
640	95.48	oe	ccsbBroad304_02741	PDS5A	-			
641	95.48	kd	CGS001-900	CCNG1	-			
642	95.48	kd	CGS001-538	ATP7A	ATPases / P-type			
643	95.47	cc		Akt Signaling GOF	-			
644	95.47	kd	CGS001-7424	VEGFC	-			
645	95.46	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
646	95.44	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
647	95.43	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
648	95.4	oe	ccsbBroad304_01371	RALA	-			
649	95.4	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
650	95.4	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
651	95.4	kd	CGS001-2976	GTF3C2	General transcription factors			
652	95.39	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
653	95.36	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
654	95.35	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
655	95.29	oe	ccsbBroad304_00171	BNIP3L	-			
656	95.27	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
657	95.26	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
658	95.23	kd	CGS001-5446	PON3	Paraoxonases			
659	95.21	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
660	95.2	oe	ccsbBroad304_06098	DHCR24	-			
661	95.17	oe	ccsbBroad304_02576	MLLT11	-			
662	95.17	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
663	95.13	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
664	95.13	kd	CGS001-9943	OXSR1	FRAY subfamily			
665	95.12	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
666	95.07	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
667	95.04	cc		TGF beta receptor inhibitor	-			
668	95.04	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
669	95.03	oe	ccsbBroad304_02501	DCTN6	-			
670	95.03	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
671	95.03	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
672	95.02	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
673	95.01	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
674	95	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
675	94.99	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
676	94.97	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
677	94.96	oe	ccsbBroad304_00995	MECP2	-			
678	94.96	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
679	94.93	cc		HIV protease inhibitor	-			
680	94.9	oe	ccsbBroad304_02759	DICER1	-			
681	94.86	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
682	94.84	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
683	94.8	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
684	94.78	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
685	94.76	kd	CGS001-4125	MAN2B1	-			
686	94.74	kd	CGS001-84328	LZIC	-			
687	94.71	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
688	94.7	kd	CGS001-253430	IPMK	-			
689	94.7	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
690	94.69	kd	CGS001-7982	ST7	-			
691	94.66	oe	ccsbBroad304_03415	GFOD1	-			
692	94.63	kd	CGS001-4700	NDUFA6	LYR motif containing			
693	94.62	oe	ccsbBroad304_02580	TMED10	-			
694	94.62	kd	CGS001-1736	DKC1	-			
695	94.6	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
696	94.6	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
697	94.59	kd	CGS001-10493	VAT1	-			
698	94.59	kd	CGS001-60528	ELAC2	-			
699	94.58	oe	ccsbBroad304_01257	PPOX	-			
700	94.56	cp	BRD-A79903587	tegafur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
701	94.53	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
702	94.53	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
703	94.48	oe	ccsbBroad304_06226	FTL	-			
704	94.46	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
705	94.46	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
706	94.45	oe	ccsbBroad304_02195	SPAG7	-			
707	94.45	kd	CGS001-58508	MLL3	-			
708	94.41	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
709	94.37	kd	CGS001-5328	PLAU	Chymotrypsin			
710	94.37	kd	CGS001-51335	NGRN	-			
711	94.34	kd	CGS001-55937	APOM	Apolipoproteins			
712	94.32	oe	ccsbBroad304_01372	RALB	-			
713	94.32	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
714	94.3	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
715	94.26	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
716	94.26	kd	CGS001-8801	SUCLG2	-			
717	94.25	oe	ccsbBroad304_08386	SMOX	-			
718	94.22	kd	CGS001-1810	DR1	-			
719	94.21	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
720	94.18	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
721	94.16	oe	ccsbBroad304_01247	POU2AF1	-			
722	94.16	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
723	94.15	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
724	94.11	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
725	94.11	cp	BRD-K06878038	deferiprone	Chelating agent		CYP4F2	Chelating agent
726	94.08	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
727	94.08	kd	CGS001-3203	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
728	94.05	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
729	94.02	kd	CGS001-2730	GCLM	-			
730	93.99	kd	CGS001-10237	SLC35B1	SLC35 family of nucleotide sugar transporters			
731	93.97	kd	CGS001-3046	HBE1	-			
732	93.95	oe	ccsbBroad304_08322	UFM1	-			
733	93.95	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
734	93.93	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
735	93.91	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
736	93.89	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
737	93.86	kd	CGS001-1389	CREBL2	basic leucine zipper proteins			
738	93.84	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
739	93.83	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
740	93.82	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
741	93.8	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
742	93.79	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
743	93.77	kd	CGS001-117581	TWIST2	Basic helix-loop-helix proteins			
744	93.76	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
745	93.73	kd	CGS001-286530	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
746	93.73	kd	CGS001-8022	LHX3	Homeoboxes / LIM class			
747	93.71	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
748	93.67	kd	CGS001-6775	STAT4	SH2 domain containing			
749	93.59	kd	CGS001-84433	CARD11	-			
750	93.58	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
751	93.57	kd	CGS001-84923	FAM104A	-			
752	93.56	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
753	93.55	kd	CGS001-29940	DSE	-			
754	93.54	cp	BRD-K33226500	indinavir	HIV protease inhibitor		CYP3A5	HIV protease inhibitor
755	93.52	kd	CGS001-2264	FGFR4	Type V RTKs: FGF (fibroblast growth factor) receptor family			
756	93.49	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
757	93.46	kd	CGS001-890	CCNA2	-			
758	93.43	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
759	93.41	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
760	93.39	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
761	93.36	kd	CGS001-10538	BATF	basic leucine zipper proteins			
762	93.35	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
763	93.32	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
764	93.32	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
765	93.31	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
766	93.27	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
767	93.24	kd	CGS001-1284	COL4A2	Collagens			
768	93.19	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
769	93.16	kd	CGS001-10587	TXNRD2	-			
770	93.15	kd	CGS001-1384	CRAT	-			
771	93.13	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
772	93.11	kd	CGS001-5327	PLAT	Chymotrypsin			
773	93.02	oe	ccsbBroad304_00394	CTSD	Cathepsins			
774	93	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
775	92.99	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
776	92.98	kd	CGS001-25898	RCHY1	RING-type (C3HC4) zinc fingers			
777	92.95	oe	ccsbBroad304_00564	FGR	Src family			
778	92.95	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
779	92.92	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
780	92.9	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
781	92.9	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
782	92.89	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
783	92.89	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
784	92.88	kd	CGS001-11319	ECD	-			
785	92.87	kd	CGS001-5048	PAFAH1B1	WD repeat domain containing			
786	92.86	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
787	92.85	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
788	92.84	oe	ccsbBroad304_00464	DTNA	-			
789	92.84	oe	ccsbBroad304_01576	SOAT1	-			
790	92.8	kd	CGS001-8720	MBTPS1	Subtilisin			
791	92.78	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
792	92.73	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
793	92.73	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
794	92.68	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
795	92.64	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
796	92.63	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
797	92.62	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
798	92.62	kd	CGS001-51547	SIRT7	Histone deacetylases (HDACs)			
799	92.6	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
800	92.6	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
801	92.6	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
802	92.6	kd	CGS001-4771	NF2	A-kinase anchor proteins			
803	92.58	oe	ccsbBroad304_01304	PSEN1	Presenilin			
804	92.54	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
805	92.5	kd	CGS001-114904	C1QTNF6	-			
806	92.49	kd	CGS001-8669	EIF3J	-			
807	92.44	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
808	92.42	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
809	92.37	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
810	92.36	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
811	92.35	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
812	92.35	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
813	92.3	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
814	92.26	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
815	92.25	kd	CGS001-6676	SPAG4	-			
816	92.25	kd	CGS001-4712	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
817	92.24	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
818	92.22	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
819	92.21	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
820	92.18	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
821	92.18	oe	ccsbBroad304_03386	SPA17	-			
822	92.14	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
823	92.08	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
824	92.08	kd	CGS001-3297	HSF1	-			
825	92.07	oe	ccsbBroad304_04471	C5ORF62	-			
826	92.06	kd	CGS001-5563	PRKAA2	AMPK subfamily			
827	92.06	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
828	92.01	kd	CGS001-6453	ITSN1	Rho guanine nucleotide exchange factors			
829	91.95	oe	ccsbBroad304_07528	DMTF1	-			
830	91.92	cc		CCK receptor antagonist	-			
831	91.91	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
832	91.91	kd	CGS001-9183	ZW10	-			
833	91.85	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
834	91.83	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
835	91.8	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
836	91.76	oe	ccsbBroad304_00223	CASP9	Caspases			
837	91.69	kd	CGS001-2237	FEN1	-			
838	91.67	oe	ccsbBroad304_01699	TPD52L2	-			
839	91.67	kd	CGS001-5223	PGAM1	-			
840	91.62	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
841	91.61	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
842	91.58	oe	ccsbBroad304_13939	MOK	RCK family			
843	91.56	oe	ccsbBroad304_02110	VAPB	-			
844	91.53	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
845	91.5	kd	CGS001-84722	PSRC1	-			
846	91.48	kd	CGS001-8061	FOSL1	basic leucine zipper proteins			
847	91.44	kd	CGS001-8692	HYAL2	-			
848	91.41	cc		Bile acid	-			
849	91.4	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
850	91.35	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
851	91.35	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
852	91.34	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
853	91.34	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
854	91.34	kd	CGS001-286380	FOXD4L3	-			
855	91.32	oe	ccsbBroad304_01114	NUP88	-			
856	91.32	kd	CGS001-81539	SLC38A1	System A-like transporters			
857	91.3	kd	CGS001-7528	YY1	INO80 complex subunits			
858	91.29	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
859	91.29	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
860	91.26	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
861	91.25	kd	CGS001-64087	MCCC2	-			
862	91.25	kd	CGS001-79071	ELOVL6	-			
863	91.24	oe	ccsbBroad304_01532	SIAH1	-			
864	91.23	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
865	91.22	kd	CGS001-23534	TNPO3	Importins			
866	91.21	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
867	91.19	kd	CGS001-8480	RAE1	WD repeat domain containing			
868	91.14	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
869	91.11	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
870	91.07	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
871	91.07	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
872	91.05	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
873	91.04	oe	ccsbBroad304_02052	KYNU	-			
874	91.04	oe	ccsbBroad304_10758	CTBP2	-			
875	90.93	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
876	90.92	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
877	90.91	kd	CGS001-716	C1S	Complement system			
878	90.86	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
879	90.83	kd	CGS001-375	ARF1	ADP-ribosylation factors			
880	90.81	cp	BRD-K96134740	kitasamycin	Protein synthesis inhibitor			Protein synthesis inhibitor
881	90.8	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
882	90.8	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
883	90.78	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
884	90.78	kd	CGS001-3688	ITGB1	Integrins			
885	90.76	kd	CGS001-9189	ZBED1	Pseudoautosomal regions / PAR1			
886	90.74	kd	CGS001-3170	FOXA2	Forkhead boxes			
887	90.72	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
888	90.71	oe	ccsbBroad304_05758	ACADSB	-			
889	90.6	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
890	90.59	oe	ccsbBroad304_02026	NRP1	CD molecules			
891	90.59	kd	CGS001-7504	XK	Blood group antigens			
892	90.57	oe	ccsbBroad304_00469	DUT	-			
893	90.57	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
894	90.55	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
895	90.52	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
896	90.46	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
897	90.43	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
898	90.39	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
899	90.38	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
900	90.34	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
901	90.33	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
902	90.32	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
903	90.32	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
904	90.29	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
905	90.27	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
906	90.25	kd	CGS001-55214	LEPREL1	-			
907	90.23	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
908	90.23	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
909	90.2	oe	ccsbBroad304_01203	PIM1	PIM family			
910	90.19	oe	ccsbBroad304_01211	PKM2	-			
911	90.12	kd	CGS001-151742	PPM1L	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
912	90.12	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
913	90.05	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
914	89.98	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
915	89.92	kd	CGS001-367	AR	Nuclear hormone receptors			
916	89.91	kd	CGS001-7866	IFRD2	-			
917	89.86	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
918	89.82	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
919	89.77	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
920	89.74	kd	CGS001-55662	HIF1AN	-			
921	89.73	oe	ccsbBroad304_03591	ETNK1	-			
922	89.72	kd	CGS001-24140	FTSJ1	-			
923	89.7	oe	ccsbBroad304_03573	BRF2	-			
924	89.61	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
925	89.59	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
926	89.48	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
927	89.43	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
928	89.4	kd	CGS001-516	ATP5G1	ATPases / F-type			
929	89.39	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
930	89.3	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
931	89.3	kd	CGS001-10400	PEMT	-			
932	89.29	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
933	89.28	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
934	89.19	kd	CGS001-1468	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
935	89.18	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
936	89.17	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
937	89.12	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
938	89.08	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
939	88.99	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
940	88.97	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
941	88.96	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
942	88.94	kd	CGS001-8428	STK24	YSK subfamily			
943	88.93	kd	CGS001-10617	STAMBP	-			
944	88.92	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
945	88.89	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
946	88.86	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
947	88.85	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
948	88.83	kd	CGS001-6884	TAF13	-			
949	88.79	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
950	88.78	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
951	88.78	kd	CGS001-9128	PRPF4	WD repeat domain containing			
952	88.76	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
953	88.74	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
954	88.72	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
955	88.72	kd	CGS001-83933	HDAC10	Histone deacetylases			
956	88.72	kd	CGS001-9854	C2CD2L	-			
957	88.72	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
958	88.64	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
959	88.64	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
960	88.63	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
961	88.62	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
962	88.6	kd	CGS001-64175	LEPRE1	-			
963	88.58	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
964	88.58	kd	CGS001-4856	NOV	-			
965	88.49	kd	CGS001-26039	SS18L1	-			
966	88.45	kd	CGS001-57026	PDXP	-			
967	88.44	kd	CGS001-55206	SBNO1	-			
968	88.33	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
969	88.24	kd	CGS001-894	CCND2	-			
970	88.21	kd	CGS001-1387	CREBBP	Chromatin-modifying enzymes / K-acetyltransferases			
971	88.19	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
972	88.19	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
973	88.17	cp	BRD-A62890442	3-methyl-GABA	GABA aminotransferase activator			GABA aminotransferase activator
974	88.15	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
975	88.07	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
976	88.02	kd	CGS001-6709	SPTAN1	EF-hand domain containing			
977	87.99	cp	BRD-A09495397	bicuculline	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, KCNN1	GABA receptor antagonist
978	87.98	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
979	87.91	oe	ccsbBroad304_01832	PAX8	Paired boxes			
980	87.91	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
981	87.91	kd	CGS001-4779	NFE2L1	basic leucine zipper proteins			
982	87.85	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
983	87.8	oe	ccsbBroad304_13952	SHMT2	-			
984	87.79	kd	CGS001-8985	PLOD3	-			
985	87.78	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
986	87.78	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
987	87.74	kd	CGS001-79722	ANKRD55	Ankyrin repeat domain containing			
988	87.73	kd	CGS001-2495	FTH1	-			
989	87.63	oe	ccsbBroad304_07140	XPC	-			
990	87.58	kd	CGS001-23621	BACE1	Pepsin			
991	87.57	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
992	87.54	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
993	87.52	oe	ccsbBroad304_01674	TIMP4	-			
994	87.48	kd	CGS001-285267	ZNF619	Zinc fingers, C2H2-type			
995	87.48	kd	CGS001-2534	FYN	Src family			
996	87.47	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
997	87.46	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
998	87.45	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
999	87.41	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
1000	87.37	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1001	87.34	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
1002	87.29	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
1003	87.28	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
1004	87.27	kd	CGS001-6713	SQLE	Lanosterol biosynthesis pathway			
1005	87.24	cc		C2 domain containing LOF	-			
1006	87.23	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
1007	87.21	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
1008	87.18	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
1009	87.16	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
1010	87.13	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1011	87.08	kd	CGS001-80135	RPF1	-			
1012	87.07	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
1013	87.06	oe	ccsbBroad304_00225	CAT	-			
1014	87.03	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
1015	87.02	oe	ccsbBroad304_10207	ERLIN1	-			
1016	87.02	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
1017	87.02	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
1018	87.02	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
1019	87	kd	CGS001-1984	EIF5A	-			
1020	86.97	kd	CGS001-7917	BAG6	-			
1021	86.96	kd	CGS001-6277	S100A6	EF-hand domain containing			
1022	86.94	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
1023	86.94	kd	CGS001-2618	GART	Ribosyl transferases			
1024	86.92	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
1025	86.85	kd	CGS001-5982	RFC2	ATPases / AAA-type			
1026	86.84	oe	ccsbBroad304_07561	YAF2	-			
1027	86.83	kd	CGS001-10991	SLC38A3	System N-like transporters			
1028	86.82	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
1029	86.82	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
1030	86.75	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
1031	86.72	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1032	86.7	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
1033	86.7	kd	CGS001-113878	DTX2	RING-type (C3HC4) zinc fingers			
1034	86.69	kd	CGS001-7389	UROD	-			
1035	86.67	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
1036	86.65	kd	CGS001-11343	MGLL	Endocannabinoid turnover			
1037	86.6	oe	ccsbBroad304_09821	TMEM154	-			
1038	86.59	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
1039	86.56	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
1040	86.54	kd	CGS001-29959	NRBP1	NRBP family			
1041	86.43	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
1042	86.39	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1043	86.38	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
1044	86.37	cp	BRD-K51485625	ritonavir	HIV protease inhibitor		CYP3A4, CYP1A2, CYP2B6, CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
1045	86.37	kd	CGS001-84527	ZNF559	Zinc fingers, C2H2-type			
1046	86.37	kd	CGS001-1120	CHKB	-			
1047	86.36	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
1048	86.33	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
1049	86.27	oe	ccsbBroad304_09708	PNLDC1	-			
1050	86.19	oe	ccsbBroad304_05756	ACAA1	-			
1051	86.16	kd	CGS001-9616	RNF7	RING-type (C3HC4) zinc fingers			
1052	86.15	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1053	86.12	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
1054	86.11	kd	CGS001-58472	SQRDL	-			
1055	86.06	kd	CGS001-2731	GLDC	-			
1056	86.05	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
1057	86.01	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
1058	86	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
1059	85.91	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
1060	85.9	kd	CGS001-3516	RBPJ	-			
1061	85.87	kd	CGS001-1910	EDNRB	Endothelin receptors			
1062	85.81	cc		Histone deacetylases LOF	-			
1063	85.81	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
1064	85.76	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
1065	85.71	oe	ccsbBroad304_08660	SMARCAD1	-			
1066	85.7	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
1067	85.7	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
1068	85.69	kd	CGS001-7035	TFPI	-			
1069	85.67	kd	CGS001-10481	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
1070	85.66	kd	CGS001-1647	GADD45A	-			
1071	85.56	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
1072	85.56	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
1073	85.52	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
1074	85.5	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
1075	85.48	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
1076	85.42	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
1077	85.42	kd	CGS001-1837	DTNA	-			
1078	85.41	cp	BRD-K40758068	efavirenz	HIV protease inhibitor		CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5	HIV protease inhibitor
1079	85.41	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
1080	85.39	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1081	85.39	kd	CGS001-10059	DNM1L	-			
1082	85.35	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
1083	85.35	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
1084	85.32	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
1085	85.31	kd	CGS001-54884	RETSAT	-			
1086	85.29	kd	CGS001-1460	CSNK2B	Casein kinase 2 (CK2) family			
1087	85.26	cp	BRD-K37516142	idebenone	Calcium channel modulator			Calcium channel modulator
1088	85.2	oe	ccsbBroad304_06645	NQO2	-			
1089	85.15	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
1090	85.11	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
1091	85.11	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
1092	85.1	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
1093	85.04	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
1094	85.03	kd	CGS001-8463	TEAD2	-			
1095	85.01	kd	CGS001-10058	ABCB6	ATP binding cassette transporters / subfamily B			
1096	84.94	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
1097	84.94	kd	CGS001-51655	RASD1	-			
1098	84.93	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
1099	84.9	cp	BRD-K81916719	triclabendazole	Microtubule inhibitor		DNMT1	Microtubule inhibitor
1100	84.85	oe	ccsbBroad304_13633	PI4KAP2	-			
1101	84.8	oe	ccsbBroad304_02446	TADA3	-			
1102	84.79	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
1103	84.77	kd	CGS001-4830	NME1	-			
1104	84.66	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
1105	84.66	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
1106	84.66	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
1107	84.65	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1108	84.65	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
1109	84.63	kd	CGS001-114112	TXNRD3	-			
1110	84.63	kd	CGS001-390	RND3	-			
1111	84.61	kd	CGS001-3586	IL10	Interleukins and interleukin receptors			
1112	84.58	kd	CGS001-3419	IDH3A	-			
1113	84.55	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
1114	84.52	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
1115	84.51	cc		MDM inhibitor	-			
1116	84.5	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
1117	84.38	kd	CGS001-25861	DFNB31	-			
1118	84.37	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
1119	84.35	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
1120	84.31	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
1121	84.28	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
1122	84.27	oe	ccsbBroad304_00268	CD81	CD molecules			
1123	84.15	kd	CGS001-147837	ZNF563	Zinc fingers, C2H2-type			
1124	84.12	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
1125	84.06	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
1126	84.03	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
1127	84.02	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
1128	84.01	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
1129	83.97	kd	CGS001-1429	CRYZ	-			
1130	83.94	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1131	83.94	kd	CGS001-323	APBB2	-			
1132	83.93	oe	ccsbBroad304_03191	NOSIP	-			
1133	83.9	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
1134	83.89	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
1135	83.87	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
1136	83.87	kd	CGS001-1642	DDB1	-			
1137	83.86	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
1138	83.81	kd	CGS001-6198	RPS6KB1	p70 subfamily			
1139	83.71	cc		Retinoid receptor agonist	-			
1140	83.67	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
1141	83.64	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
1142	83.62	kd	CGS001-6478	SIAH2	-			
1143	83.56	oe	ccsbBroad304_02386	EIF1B	-			
1144	83.56	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
1145	83.49	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
1146	83.49	kd	CGS001-899	CCNF	F-boxes / other			
1147	83.48	kd	CGS001-629	CFB	Complement system			
1148	83.47	kd	CGS001-23	ABCF1	ATP binding cassette transporters / subfamily F			
1149	83.44	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
1150	83.43	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
1151	83.41	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
1152	83.4	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
1153	83.38	kd	CGS001-23710	GABARAPL1	-			
1154	83.37	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
1155	83.36	kd	CGS001-55193	PBRM1	Non-enzymatic BRD containing proteins			
1156	83.35	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1157	83.33	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1158	83.33	kd	CGS001-6455	SH3GL1	-			
1159	83.25	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
1160	83.16	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1161	83.12	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
1162	83.12	kd	CGS001-30001	ERO1L	-			
1163	83.09	cc		GPCR Subset GOF	-			
1164	83.08	kd	CGS001-54107	POLE3	DNA polymerases			
1165	83.06	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
1166	83.04	cc		Potassium channel activator	-			
1167	82.99	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
1168	82.97	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
1169	82.94	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
1170	82.93	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
1171	82.89	cc		Integrin subunits beta LOF	-			
1172	82.84	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
1173	82.84	cp	BRD-K70883034	nimetazepam	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA receptor agonist
1174	82.75	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
1175	82.75	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
1176	82.74	kd	CGS001-58497	PRUNE	-			
1177	82.72	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
1178	82.68	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
1179	82.67	kd	CGS001-8566	PDXK	-			
1180	82.65	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
1181	82.59	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
1182	82.56	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
1183	82.55	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
1184	82.49	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
1185	82.49	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
1186	82.47	kd	CGS001-51564	HDAC7	Histone deacetylases			
1187	82.45	kd	CGS001-8535	CBX4	-			
1188	82.42	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
1189	82.41	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
1190	82.39	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
1191	82.39	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
1192	82.36	kd	CGS001-9587	MAD2L1BP	-			
1193	82.35	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
1194	82.32	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
1195	82.28	kd	CGS001-4688	NCF2	Tetratricopeptide (TTC) repeat domain containing			
1196	82.26	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
1197	82.25	oe	ccsbBroad304_01066	NDUFA4	-			
1198	82.24	oe	ccsbBroad304_02579	YWHAQ	-			
1199	82.21	kd	CGS001-5583	PRKCH	Eta subfamily			
1200	82.18	cp	BRD-K99063460	didanosine	Nucleoside reverse transcriptase inhibitor		PNP	Nucleoside reverse transcriptase inhibitor
1201	82.18	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1202	82.16	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
1203	82.15	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
1204	82.09	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
1205	82	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
1206	82	kd	CGS001-843	CASP10	Caspases			
1207	81.99	oe	ccsbBroad304_06349	HAGH	-			
1208	81.78	cp	BRD-K16336526	capsaicin	TRPV agonist		TRPV1, CFTR, ENOX2	TRPV agonist
1209	81.77	kd	CGS001-468	ATF4	basic leucine zipper proteins			
1210	81.72	kd	CGS001-5450	POU2AF1	-			
1211	81.7	kd	CGS001-3912	LAMB1	Laminins			
1212	81.69	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
1213	81.68	kd	CGS001-80274	SCUBE1	-			
1214	81.67	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
1215	81.66	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
1216	81.65	kd	CGS001-6608	SMO	GPCR / Class F : Frizzled receptors			
1217	81.65	kd	CGS001-135	ADORA2A	GPCR / Class A : Adenosine receptors			
1218	81.61	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
1219	81.6	kd	CGS001-1045	CDX2	Homeoboxes / ANTP class : HOXL subclass			
1220	81.58	kd	CGS001-7248	TSC1	-			
1221	81.55	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
1222	81.5	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
1223	81.5	kd	CGS001-10161	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1224	81.49	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
1225	81.35	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
1226	81.35	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
1227	81.33	kd	CGS001-7486	WRN	-			
1228	81.3	kd	CGS001-4016	LOXL1	-			
1229	81.27	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
1230	81.21	kd	CGS001-3589	IL11	Endogenous ligands			
1231	81.18	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
1232	81.16	kd	CGS001-1029	CDKN2A	-			
1233	81.12	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
1234	81.11	kd	CGS001-51447	IP6K2	-			
1235	81.09	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
1236	81.07	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
1237	81.07	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1238	81.05	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
1239	81.05	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
1240	81.04	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
1241	81.01	oe	ccsbBroad304_02922	TES	-			
1242	80.94	kd	CGS001-7099	TLR4	Toll-like receptor family			
1243	80.91	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
1244	80.84	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
1245	80.82	kd	CGS001-5052	PRDX1	-			
1246	80.81	oe	ccsbBroad304_01527	SGK1	SGK family			
1247	80.78	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
1248	80.78	kd	CGS001-57661	PHRF1	Zinc fingers, PHD-type			
1249	80.6	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
1250	80.53	kd	CGS001-5979	RET	Type XIV RTKs: RET			
1251	80.5	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
1252	80.46	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
1253	80.46	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
1254	80.45	kd	CGS001-100133941	CD24	CD molecules			
1255	80.41	kd	CGS001-6813	STXBP2	-			
1256	80.4	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
1257	80.36	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
1258	80.36	kd	CGS001-51128	SAR1B	-			
1259	80.32	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
1260	80.3	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
1261	80.3	kd	CGS001-9181	ARHGEF2	Rho guanine nucleotide exchange factors			
1262	80.24	kd	CGS001-3717	JAK2	Janus kinase (JakA) family			
1263	80.22	kd	CGS001-9231	DLG5	-			
1264	80.16	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1265	80.16	kd	CGS001-9788	MTSS1	-			
1266	80.16	kd	CGS001-1390	CREM	basic leucine zipper proteins			
1267	80.15	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
1268	80.15	kd	CGS001-1069	CETN2	EF-hand domain containing			
1269	80.1	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
1270	80.1	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
1271	79.96	kd	CGS001-6499	SKIV2L	-			
1272	79.94	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
1273	79.89	oe	ccsbBroad304_03089	PACSIN3	-			
1274	79.89	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
1275	79.88	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
1276	79.79	kd	CGS001-3177	SLC29A2	SLC29 family			
1277	79.74	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
1278	79.66	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
1279	79.6	cc		DNA Replication LOF	-			
1280	79.6	kd	CGS001-823	CAPN1	EF-hand domain containing			
1281	79.58	kd	CGS001-1786	DNMT1	Methyltransferases			
1282	79.58	oe	ccsbBroad304_02487	TXNIP	-			
1283	79.56	kd	CGS001-116535	MRGPRF	GPCR / Class A : Orphans			
1284	79.54	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
1285	79.51	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1286	79.51	kd	CGS001-4303	FOXO4	Forkhead boxes			
1287	79.5	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
1288	79.48	kd	CGS001-7852	CXCR4	Chemokine receptors			
1289	79.33	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
1290	79.32	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
1291	79.31	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
1292	79.28	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
1293	79.27	kd	CGS001-5277	PIGA	Glycosyltransferase group 1 domain containing			
1294	79.21	oe	ccsbBroad304_07362	NMI	-			
1295	79.2	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
1296	79.18	kd	CGS001-3417	IDH1	-			
1297	79.09	kd	CGS001-5300	PIN1	-			
1298	79.09	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
1299	79.09	kd	CGS001-4849	CNOT3	-			
1300	79.06	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
1301	79.03	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
1302	79.03	kd	CGS001-4798	NFRKB	INO80 complex subunits			
1303	79.02	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
1304	78.93	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
1305	78.89	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
1306	78.82	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
1307	78.81	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
1308	78.79	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
1309	78.79	kd	CGS001-55577	NAGK	-			
1310	78.75	kd	CGS001-10180	RBM6	G patch domain containing			
1311	78.74	oe	ccsbBroad304_07238	STK24	YSK subfamily			
1312	78.74	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
1313	78.7	kd	CGS001-837	CASP4	Caspases			
1314	78.67	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
1315	78.59	kd	CGS001-10252	SPRY1	-			
1316	78.58	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
1317	78.57	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
1318	78.57	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
1319	78.43	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
1320	78.4	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
1321	78.4	kd	CGS001-23274	CLEC16A	C-type lectin domain containing			
1322	78.26	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
1323	78.17	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
1324	78.17	kd	CGS001-2523	FUT1	Fucosyltransferases			
1325	78.11	kd	CGS001-2004	ELK3	ETS Transcription Factors			
1326	78.1	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
1327	78.08	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
1328	78.03	kd	CGS001-3339	HSPG2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1329	78	oe	ccsbBroad304_00316	CKS1B	-			
1330	77.91	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
1331	77.81	kd	CGS001-56993	TOMM22	-			
1332	77.81	kd	CGS001-139135	PASD1	-			
1333	77.75	kd	CGS001-10681	GNB5	WD repeat domain containing			
1334	77.72	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
1335	77.72	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
1336	77.66	kd	CGS001-9868	TOMM70A	Tetratricopeptide (TTC) repeat domain containing			
1337	77.61	kd	CGS001-4352	MPL	Prolactin receptor family			
1338	77.57	kd	CGS001-7001	PRDX2	-			
1339	77.55	cp	BRD-K31491153	1-phenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
1340	77.54	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
1341	77.49	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
1342	77.47	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
1343	77.46	kd	CGS001-150962	PUS10	-			
1344	77.41	oe	ccsbBroad304_03040	NKIRAS2	-			
1345	77.35	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
1346	77.31	cp	BRD-K34437622	BRD-K34437622	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
1347	77.3	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
1348	77.23	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
1349	77.22	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
1350	77.19	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
1351	77.18	kd	CGS001-2118	ETV4	ETS Transcription Factors			
1352	77.17	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
1353	77.16	kd	CGS001-471	ATIC	-			
1354	77.11	cc		Wnt family GOF	-			
1355	77.09	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
1356	77.09	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
1357	77.03	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
1358	77	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
1359	76.96	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
1360	76.94	kd	CGS001-286075	ZNF707	Zinc fingers, C2H2-type			
1361	76.91	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
1362	76.81	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
1363	76.78	oe	ccsbBroad304_08825	LHPP	-			
1364	76.75	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
1365	76.74	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
1366	76.71	kd	CGS001-6727	SRP14	-			
1367	76.69	oe	ccsbBroad304_05947	CCNC	-			
1368	76.61	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
1369	76.6	oe	ccsbBroad304_02416	TUBB4B	-			
1370	76.57	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1371	76.54	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
1372	76.54	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
1373	76.53	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
1374	76.51	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
1375	76.48	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
1376	76.45	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
1377	76.45	kd	CGS001-11116	FGFR1OP	-			
1378	76.41	oe	ccsbBroad304_02500	RRAGA	-			
1379	76.39	kd	CGS001-3482	IGF2R	CD molecules			
1380	76.38	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
1381	76.38	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
1382	76.37	kd	CGS001-1622	DBI	-			
1383	76.3	kd	CGS001-11004	KIF2C	Kinesins			
1384	76.28	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
1385	76.26	kd	CGS001-10476	ATP5H	ATPases / F-type			
1386	76.21	kd	CGS001-481	ATP1B1	ATPases / P-type			
1387	76.18	oe	ccsbBroad304_01186	PHB	-			
1388	76.17	oe	ccsbBroad304_07851	FAM120A	-			
1389	76.15	kd	CGS001-54677	CROT	-			
1390	76.1	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
1391	76.1	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
1392	76.1	kd	CGS001-10971	YWHAQ	-			
1393	76.09	kd	CGS001-571	BACH1	BTB/POZ domain containing			
1394	75.99	kd	CGS001-5910	RAP1GDS1	Armadillo repeat containing			
1395	75.96	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
1396	75.95	oe	ccsbBroad304_03910	CCDC90A	-			
1397	75.86	kd	CGS001-124535	HSF5	-			
1398	75.71	kd	CGS001-4781	NFIB	-			
1399	75.68	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
1400	75.68	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1401	75.68	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
1402	75.65	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1403	75.63	cp	BRD-A24191444	ifenprodil	Adrenergic receptor antagonist		GRIN1, GRIN2B	Adrenergic receptor antagonist, Glutamate receptor antagonist
1404	75.59	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
1405	75.48	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
1406	75.46	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
1407	75.37	kd	CGS001-54472	TOLLIP	-			
1408	75.36	kd	CGS001-664	BNIP3	-			
1409	75.34	kd	CGS001-2817	GPC1	Proteoglycans / Cell Surface : Glypicans			
1410	75.34	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1411	75.32	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
1412	75.3	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
1413	75.3	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
1414	75.29	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
1415	75.24	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
1416	75.21	kd	CGS001-29965	C16ORF5	-			
1417	75.2	oe	ccsbBroad304_01787	YES1	Src family			
1418	75.2	kd	CGS001-1891	ECH1	-			
1419	75.19	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
1420	75.16	kd	CGS001-285676	ZNF454	Zinc fingers, C2H2-type			
1421	75.13	kd	CGS001-4795	NFKBIL1	-			
1422	75.1	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
1423	75.1	kd	CGS001-23030	KDM4B	Histone demethylases			
1424	75.04	oe	ccsbBroad304_02349	MPHOSPH9	-			
1425	75.02	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
1426	75.01	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
1427	74.93	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
1428	74.85	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
1429	74.83	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
1430	74.79	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
1431	74.77	kd	CGS001-1030	CDKN2B	-			
1432	74.68	kd	CGS001-3065	HDAC1	Histone deacetylases			
1433	74.58	kd	CGS001-192669	EIF2C3	-			
1434	74.57	kd	CGS001-3315	HSPB1	Heat shock proteins / HSPB			
1435	74.54	oe	ccsbBroad304_04399	PGBD1	-			
1436	74.53	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
1437	74.51	oe	ccsbBroad304_01091	NFIB	-			
1438	74.46	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
1439	74.36	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
1440	74.22	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
1441	74.22	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
1442	74.17	kd	CGS001-5915	RARB	Retinoic acid receptors			
1443	74.1	kd	CGS001-53834	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
1444	74.07	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
1445	74.06	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
1446	74.05	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
1447	74.03	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
1448	73.96	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
1449	73.89	kd	CGS001-23131	GPATCH8	G patch domain containing			
1450	73.88	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
1451	73.84	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
1452	73.84	cp	BRD-K32398298	alprazolam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, CYP3A5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
1453	73.75	oe	ccsbBroad304_06889	RPN2	-			
1454	73.73	kd	CGS001-801	CALM1	EF-hand domain containing			
1455	73.71	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
1456	73.62	kd	CGS001-2615	LRRC32	-			
1457	73.55	kd	CGS001-861	RUNX1	-			
1458	73.48	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
1459	73.47	oe	ccsbBroad304_00529	F3	CD molecules			
1460	73.46	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
1461	73.44	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
1462	73.39	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
1463	73.37	kd	CGS001-54505	DHX29	DEAH-boxes			
1464	73.35	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
1465	73.33	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
1466	73.32	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
1467	73.28	cc		Toll like receptors LOF	-			
1468	73.28	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
1469	73.25	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
1470	73.17	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
1471	73.17	oe	ccsbBroad304_07605	LYPLA1	-			
1472	73.16	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1473	73.16	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
1474	73.15	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
1475	73.14	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
1476	73.14	kd	CGS001-8508	NIPSNAP1	-			
1477	73.11	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
1478	73.1	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
1479	73.09	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
1480	73.08	kd	CGS001-55038	CDCA4	-			
1481	73.07	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
1482	73.04	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
1483	73.04	cp	BRD-K86003836	flubendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
1484	73	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
1485	73	oe	ccsbBroad304_03179	BOLA1	-			
1486	72.93	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
1487	72.91	oe	ccsbBroad304_02566	MORF4L1	-			
1488	72.9	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
1489	72.87	kd	CGS001-23588	KLHDC2	-			
1490	72.85	oe	ccsbBroad304_06382	HMGCL	-			
1491	72.84	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
1492	72.82	oe	ccsbBroad304_00624	GCK	Hexokinases			
1493	72.8	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
1494	72.79	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
1495	72.78	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
1496	72.72	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
1497	72.7	oe	ccsbBroad304_06089	DDIT3	-			
1498	72.7	kd	CGS001-4232	MEST	-			
1499	72.69	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
1500	72.67	kd	CGS001-221393	GPR115	Adhesion Class GPCRs			
1501	72.65	cp	BRD-K59456551	methotrexate	Dihydrofolate reductase inhibitor		DHFR, AOX1, FOLR1, TYMS	Dihydrofolate reductase inhibitor
1502	72.62	kd	CGS001-3776	KCNK2	Two-P potassium channels			
1503	72.42	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
1504	72.39	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
1505	72.37	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
1506	72.33	kd	CGS001-10553	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
1507	72.32	kd	CGS001-58492	ZNF77	Zinc fingers, C2H2-type			
1508	72.29	kd	CGS001-80758	PRR7	-			
1509	72.28	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1510	72.18	kd	CGS001-2963	GTF2F2	General transcription factors			
1511	72.16	cc		Tachykinin antagonist	-			
1512	72.12	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
1513	72.1	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
1514	72.07	oe	ccsbBroad304_00164	BLMH	-			
1515	72.03	kd	CGS001-9441	MED26	-			
1516	72.01	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
1517	71.97	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
1518	71.9	cc		Na-K-Cl transporter inhibitor	-			
1519	71.9	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
1520	71.85	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
1521	71.83	kd	CGS001-8409	UXT	-			
1522	71.75	kd	CGS001-8193	DPF1	Zinc fingers, PHD-type			
1523	71.74	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
1524	71.73	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
1525	71.73	kd	CGS001-4724	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
1526	71.66	oe	ccsbBroad304_01139	PA2G4	-			
1527	71.56	cp	BRD-K93618743	ipriflavone	Bone resorption inhibitor			Bone resorption inhibitor
1528	71.56	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
1529	71.54	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
1530	71.54	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
1531	71.45	kd	CGS001-26523	EIF2C1	-			
1532	71.43	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
1533	71.38	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1534	71.26	kd	CGS001-8495	PPFIBP2	Sterile alpha motif (SAM) domain containing			
1535	71.25	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1536	71.19	oe	ccsbBroad304_00658	GNG5	-			
1537	71.18	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
1538	71.14	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
1539	71.14	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
1540	71.02	kd	CGS001-9500	MAGED1	-			
1541	71.01	kd	CGS001-6927	HNF1A	Homeoboxes / HNF class			
1542	70.96	oe	ccsbBroad304_07884	RYBP	-			
1543	70.96	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
1544	70.96	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
1545	70.96	kd	CGS001-84875	PARP10	Poly (ADP-ribose) polymerases			
1546	70.96	kd	CGS001-2181	ACSL3	Acyl-CoA synthetase family			
1547	70.88	kd	CGS001-5257	PHKB	-			
1548	70.87	oe	ccsbBroad304_01019	MLH1	-			
1549	70.84	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
1550	70.8	kd	CGS001-121599	SPIC	ETS Transcription Factors			
1551	70.77	kd	CGS001-7337	UBE3A	-			
1552	70.68	oe	ccsbBroad304_03420	TOLLIP	-			
1553	70.64	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
1554	70.63	kd	CGS001-975	CD81	CD molecules			
1555	70.58	oe	ccsbBroad304_03450	TMED9	-			
1556	70.46	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
1557	70.45	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
1558	70.42	kd	CGS001-5108	PCM1	-			
1559	70.42	kd	CGS001-335	APOA1	Apolipoproteins			
1560	70.41	oe	ccsbBroad304_08339	CMPK1	-			
1561	70.4	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
1562	70.37	kd	CGS001-25793	FBXO7	F-boxes / other			
1563	70.36	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
1564	70.34	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
1565	70.33	kd	CGS001-5654	HTRA1	Serine peptidases / Serine peptidases			
1566	70.31	oe	ccsbBroad304_06367	HK1	-			
1567	70.31	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
1568	70.24	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
1569	70.22	cc		X linked mental retardation group 1 LOF	-			
1570	70.21	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
1571	70.2	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
1572	70.2	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
1573	70.19	oe	ccsbBroad304_01469	RSU1	-			
1574	70.18	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
1575	70.18	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1576	70.16	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
1577	70.14	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
1578	70.02	kd	CGS001-54881	TEX10	-			
1579	70	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
1580	69.93	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
1581	69.86	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
1582	69.86	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
1583	69.81	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
1584	69.75	oe	ccsbBroad304_06282	GLDC	-			
1585	69.73	kd	CGS001-10641	NPRL2	-			
1586	69.73	kd	CGS001-57121	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1587	69.72	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
1588	69.64	kd	CGS001-55311	ZNF444	Zinc fingers, C2H2-type			
1589	69.62	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
1590	69.52	kd	CGS001-27109	ATP5S	-			
1591	69.45	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
1592	69.44	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
1593	69.41	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
1594	69.4	oe	ccsbBroad304_06992	SRC	Src family			
1595	69.33	kd	CGS001-2562	GABRB3	GABA receptors			
1596	69.3	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
1597	69.29	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
1598	69.28	oe	ccsbBroad304_07097	TRAF1	-			
1599	69.27	oe	ccsbBroad304_02345	TXNDC9	-			
1600	69.26	kd	CGS001-3416	IDE	Pitrilysin			
1601	69.25	kd	CGS001-2101	ESRRA	Estrogen-related receptors			
1602	69.17	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
1603	69.17	kd	CGS001-6678	SPARC	-			
1604	69.16	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
1605	69.09	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
1606	68.89	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
1607	68.84	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
1608	68.84	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
1609	68.73	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
1610	68.65	kd	CGS001-11129	CLASRP	-			
1611	68.63	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
1612	68.62	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
1613	68.61	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
1614	68.59	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
1615	68.57	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
1616	68.56	oe	ccsbBroad304_09254	PAQR8	-			
1617	68.5	kd	CGS001-3098	HK1	-			
1618	68.44	oe	ccsbBroad304_02485	STAMBP	-			
1619	68.42	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1620	68.4	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
1621	68.28	kd	CGS001-4176	MCM7	-			
1622	68.26	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
1623	68.24	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
1624	68.24	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
1625	68.23	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
1626	68.2	oe	ccsbBroad304_02708	TRIM32	-			
1627	68.12	kd	CGS001-593	BCKDHA	-			
1628	67.97	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
1629	67.91	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
1630	67.9	kd	CGS001-23212	RRS1	-			
1631	67.8	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
1632	67.77	cp	BRD-A23637604	oxymetholone	Androgen receptor agonist		AR	Androgen receptor agonist
1633	67.74	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
1634	67.7	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
1635	67.67	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
1636	67.65	kd	CGS001-10987	COPS5	-			
1637	67.64	kd	CGS001-5906	RAP1A	-			
1638	67.63	kd	CGS001-3596	IL13	Interleukins and interleukin receptors			
1639	67.58	oe	ccsbBroad304_06294	GNAZ	-			
1640	67.57	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
1641	67.52	kd	CGS001-51001	MTERFD1	-			
1642	67.49	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
1643	67.41	kd	CGS001-2152	F3	CD molecules			
1644	67.37	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
1645	67.32	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
1646	67.31	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
1647	67.22	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1648	67.13	kd	CGS001-170591	S100Z	EF-hand domain containing			
1649	67.1	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
1650	67.06	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
1651	67.06	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
1652	67.03	kd	CGS001-4548	MTR	-			
1653	67	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
1654	66.85	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
1655	66.84	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
1656	66.81	kd	CGS001-1534	CYB561	Cytochrome b genes			
1657	66.79	cc		PKC activator	-			
1658	66.79	kd	CGS001-55191	NADSYN1	-			
1659	66.7	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
1660	66.62	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
1661	66.6	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
1662	66.58	kd	CGS001-23344	ESYT1	Synaptotagmins			
1663	66.56	oe	ccsbBroad304_02509	GMEB1	-			
1664	66.55	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
1665	66.53	oe	ccsbBroad304_07761	CORO1A	Coronins			
1666	66.5	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
1667	66.49	oe	ccsbBroad304_07275	PSMG1	-			
1668	66.48	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
1669	66.46	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
1670	66.43	kd	CGS001-819	CAMLG	-			
1671	66.4	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
1672	66.4	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1673	66.36	oe	ccsbBroad304_06654	NPM1	-			
1674	66.34	oe	ccsbBroad304_02220	MTFR1	-			
1675	66.33	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
1676	66.33	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
1677	66.33	kd	CGS001-4331	MNAT1	RING-type (C3HC4) zinc fingers			
1678	66.24	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
1679	66.21	kd	CGS001-6883	TAF12	-			
1680	66.2	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
1681	66.14	oe	ccsbBroad304_07017	SUOX	-			
1682	66.12	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
1683	66.02	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
1684	66.01	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1685	65.98	kd	CGS001-122809	SOCS4	SH2 domain containing			
1686	65.93	kd	CGS001-6304	SATB1	Homeoboxes / CUT class			
1687	65.87	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
1688	65.85	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
1689	65.84	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
1690	65.8	kd	CGS001-2119	ETV5	ETS Transcription Factors			
1691	65.79	cc		GABA receptor antagonist	-			
1692	65.79	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
1693	65.73	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
1694	65.56	oe	ccsbBroad304_06745	PNN	-			
1695	65.54	kd	CGS001-55278	QRSL1	-			
1696	65.52	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
1697	65.5	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
1698	65.45	kd	CGS001-55723	ASF1B	-			
1699	65.44	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
1700	65.43	kd	CGS001-54407	SLC38A2	System A-like transporters			
1701	65.39	oe	ccsbBroad304_05135	PARP15	-			
1702	65.39	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
1703	65.32	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
1704	65.18	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
1705	65.14	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
1706	65.13	cp	BRD-M47937986	cefatrizine	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1707	65.13	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
1708	65.13	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
1709	65.09	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
1710	65.08	kd	CGS001-2017	CTTN	-			
1711	65.07	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
1712	65.07	kd	CGS001-439	ASNA1	-			
1713	65.06	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
1714	65.02	kd	CGS001-163688	CALML6	EF-hand domain containing			
1715	64.93	kd	CGS001-5645	PRSS2	Serine peptidases			
1716	64.9	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
1717	64.68	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
1718	64.66	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
1719	64.63	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
1720	64.56	kd	CGS001-5162	PDHB	-			
1721	64.4	kd	CGS001-9898	UBAP2L	-			
1722	64.33	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
1723	64.32	cc		Dihydrofolate reductase inhibitor	-			
1724	64.27	oe	ccsbBroad304_06048	CRYZ	-			
1725	64.24	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1726	64.21	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
1727	64.18	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
1728	64.17	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
1729	64.16	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
1730	64.14	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
1731	64.12	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
1732	64.05	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
1733	64.04	kd	CGS001-3691	ITGB4	Integrins			
1734	63.9	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
1735	63.9	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
1736	63.77	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
1737	63.76	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
1738	63.76	kd	CGS001-22889	KIAA0907	-			
1739	63.66	kd	CGS001-4194	MDM4	-			
1740	63.65	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
1741	63.65	cp	BRD-K85503079	perospirone	Dopamine receptor antagonist		DRD2, HTR2A, DRD3, DRD4, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
1742	63.63	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
1743	63.56	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
1744	63.55	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
1745	63.53	kd	CGS001-25925	ZNF521	Zinc fingers, C2H2-type			
1746	63.51	oe	ccsbBroad304_07592	CEPT1	-			
1747	63.5	oe	ccsbBroad304_09396	TIRAP	-			
1748	63.5	kd	CGS001-2770	GNAI1	-			
1749	63.42	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
1750	63.42	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
1751	63.4	kd	CGS001-6601	SMARCC2	-			
1752	63.4	kd	CGS001-5053	PAH	Amino acid hydroxylases			
1753	63.36	kd	CGS001-5578	PRKCA	Delta subfamily			
1754	63.3	kd	CGS001-2308	FOXO1	Forkhead boxes			
1755	63.28	kd	CGS001-342926	ZNF677	Zinc fingers, C2H2-type			
1756	63.12	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
1757	63.07	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
1758	63.02	oe	ccsbBroad304_00221	CASP3	Caspases			
1759	62.94	oe	ccsbBroad304_02217	FEZ1	-			
1760	62.91	oe	ccsbBroad304_08553	STAP2	-			
1761	62.87	kd	CGS001-284	ANGPT1	Fibrinogen C domain containing			
1762	62.86	kd	CGS001-9140	ATG12	-			
1763	62.81	kd	CGS001-3958	LGALS3	Endogenous ligands			
1764	62.72	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
1765	62.64	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
1766	62.53	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
1767	62.49	oe	ccsbBroad304_03164	MTERFD1	-			
1768	62.49	kd	CGS001-23585	TMEM50A	-			
1769	62.47	kd	CGS001-7056	THBD	CD molecules			
1770	62.43	oe	ccsbBroad304_06237	GAA	Glycosidases			
1771	62.43	cp	BRD-K52080565	rilmenidine	Imidazoline receptor agonist		NISCH	Imidazoline receptor agonist
1772	62.2	cp	BRD-A07395371	esmolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
1773	62.19	kd	CGS001-1111	CHEK1	CHK1 subfamily			
1774	62.17	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
1775	62.08	kd	CGS001-10412	NSA2	-			
1776	62	oe	ccsbBroad304_02340	SORBS3	-			
1777	61.97	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
1778	61.96	kd	CGS001-8974	P4HA2	-			
1779	61.89	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
1780	61.88	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
1781	61.86	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1782	61.84	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1783	61.83	kd	CGS001-478	ATP1A3	ATPases / P-type			
1784	61.81	oe	ccsbBroad304_03121	NRBF2	-			
1785	61.81	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
1786	61.73	kd	CGS001-115727	RASGRP4	EF-hand domain containing			
1787	61.72	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
1788	61.7	kd	CGS001-10444	ZER1	ZYG11 cell cycle regulator family			
1789	61.7	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
1790	61.66	oe	ccsbBroad304_02318	KIF20A	Kinesins			
1791	61.62	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
1792	61.61	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
1793	61.59	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
1794	61.56	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
1795	61.55	oe	ccsbBroad304_03658	DCP1A	-			
1796	61.5	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
1797	61.49	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
1798	61.44	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
1799	61.43	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
1800	61.42	oe	ccsbBroad304_02017	PEX11A	-			
1801	61.36	kd	CGS001-5106	PCK2	-			
1802	61.34	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
1803	61.32	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
1804	61.31	kd	CGS001-11340	EXOSC8	-			
1805	61.17	kd	CGS001-29116	MYLIP	-			
1806	61.15	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
1807	61.14	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
1808	61.11	kd	CGS001-55958	KLHL9	BTB/POZ domain containing			
1809	61.02	kd	CGS001-27241	BBS9	-			
1810	60.97	kd	CGS001-9870	KIAA0317	-			
1811	60.83	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
1812	60.82	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
1813	60.78	kd	CGS001-466	ATF1	basic leucine zipper proteins			
1814	60.76	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
1815	60.72	kd	CGS001-2149	F2R	Protease activated receptors			
1816	60.7	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
1817	60.7	kd	CGS001-10269	ZMPSTE24	-			
1818	60.69	kd	CGS001-79902	NUP85	-			
1819	60.53	oe	ccsbBroad304_02197	VPS26A	-			
1820	60.5	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
1821	60.45	kd	CGS001-8905	AP1S2	-			
1822	60.39	kd	CGS001-2580	GAK	Heat shock proteins / DNAJ (HSP40)			
1823	60.33	kd	CGS001-650	BMP2	Bone morphogenetic proteins			
1824	60.23	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
1825	60.18	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
1826	60.11	kd	CGS001-6778	STAT6	SH2 domain containing			
1827	60.07	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
1828	59.98	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
1829	59.95	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
1830	59.9	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
1831	59.89	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
1832	59.84	oe	ccsbBroad304_00738	HINT1	-			
1833	59.84	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
1834	59.84	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
1835	59.72	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1836	59.66	oe	ccsbBroad304_03155	DHH	-			
1837	59.65	kd	CGS001-701	BUB1B	Bub family			
1838	59.64	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
1839	59.62	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
1840	59.61	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
1841	59.59	kd	CGS001-57657	HCN3	Cyclic nucleotide-regulated channels			
1842	59.56	oe	ccsbBroad304_00471	E2F6	-			
1843	59.55	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
1844	59.48	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
1845	59.47	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
1846	59.45	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
1847	59.35	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
1848	59.26	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
1849	59.26	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
1850	59.22	kd	CGS001-22891	ZNF365	Zinc fingers, C2H2-type			
1851	59.15	oe	ccsbBroad304_06383	HMMR	CD molecules			
1852	59.14	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
1853	59.14	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
1854	59.12	oe	ccsbBroad304_01215	PLAUR	CD molecules			
1855	59.1	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
1856	59.1	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
1857	59.07	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
1858	59.06	oe	ccsbBroad304_01208	PITPNA	-			
1859	58.96	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
1860	58.95	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
1861	58.94	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
1862	58.93	oe	ccsbBroad304_02569	BTG3	-			
1863	58.82	kd	CGS001-10312	TCIRG1	ATPases / V-type			
1864	58.74	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
1865	58.71	kd	CGS001-10007	GNPDA1	-			
1866	58.66	oe	ccsbBroad304_03874	UBL5	-			
1867	58.55	kd	CGS001-4205	MEF2A	Myocyte enhancer factors			
1868	58.52	oe	ccsbBroad304_03433	DDIT4	-			
1869	58.49	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
1870	58.47	kd	CGS001-10010	TANK	-			
1871	58.41	kd	CGS001-6804	STX1A	-			
1872	58.37	oe	ccsbBroad304_06013	CLPTM1	-			
1873	58.35	cp	BRD-K18895904	olanzapine	Dopamine receptor antagonist		DRD2, HTR2A, HTR2C, DRD1, DRD3, DRD4, HRH1, HTR1A, HTR1B, HTR1D, HTR1E, HTR6, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C8, DRD5, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH2, HRH4, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
1874	58.33	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
1875	58.32	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
1876	58.32	kd	CGS001-3486	IGFBP3	insulin-like growth factor (IGF) binding proteins			
1877	58.32	kd	CGS001-10023	FRAT1	-			
1878	58.3	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
1879	58.29	oe	ccsbBroad304_00617	GBA	-			
1880	58.25	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
1881	58.21	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
1882	58.19	kd	CGS001-539	ATP5O	ATPases / F-type			
1883	58.15	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
1884	58.14	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
1885	58.13	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1886	58.08	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
1887	58.02	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1888	58	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
1889	57.93	kd	CGS001-4088	SMAD3	SMADs			
1890	57.92	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
1891	57.91	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
1892	57.82	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
1893	57.8	kd	CGS001-4069	LYZ	-			
1894	57.79	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
1895	57.75	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
1896	57.74	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
1897	57.7	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1898	57.66	kd	CGS001-3455	IFNAR2	Interferon receptor family			
1899	57.6	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
1900	57.57	kd	CGS001-4173	MCM4	-			
1901	57.56	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
1902	57.56	kd	CGS001-1066	CES1	Carboxylesterases			
1903	57.48	oe	ccsbBroad304_04626	EGLN3	-			
1904	57.44	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
1905	57.43	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
1906	57.4	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1907	57.39	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
1908	57.37	oe	ccsbBroad304_01143	PAFAH1B3	-			
1909	57.33	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
1910	57.32	kd	CGS001-83439	TCF7L1	-			
1911	57.32	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
1912	57.3	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
1913	57.13	kd	CGS001-4292	MLH1	-			
1914	57.1	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
1915	57.06	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
1916	57.05	kd	CGS001-9146	HGS	Zinc fingers, FYVE domain containing			
1917	57.03	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
1918	56.95	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
1919	56.87	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1920	56.83	kd	CGS001-51495	PTPLAD1	-			
1921	56.8	cc		HMGCR inhibitor	-			
1922	56.77	kd	CGS001-152	ADRA2C	GPCR / Class A : Adrenoceptors : alpha			
1923	56.71	oe	ccsbBroad304_09954	PTRF	-			
1924	56.71	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
1925	56.67	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
1926	56.66	oe	ccsbBroad304_06711	PFAS	-			
1927	56.61	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1928	56.61	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
1929	56.56	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
1930	56.54	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
1931	56.52	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
1932	56.49	kd	CGS001-213	ALB	-			
1933	56.43	oe	ccsbBroad304_02230	HERPUD1	-			
1934	56.43	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
1935	56.43	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
1936	56.4	kd	CGS001-2859	GPR35	GPCR / Class A : Orphans			
1937	56.37	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
1938	56.23	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
1939	56.17	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
1940	56.15	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
1941	56.14	kd	CGS001-23523	CABIN1	-			
1942	56.13	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
1943	56.13	kd	CGS001-435	ASL	-			
1944	56.1	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
1945	56.1	kd	CGS001-51135	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
1946	56.04	oe	ccsbBroad304_05590	NOTCH2NL	-			
1947	55.95	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
1948	55.94	kd	CGS001-509	ATP5C1	ATPases / F-type			
1949	55.93	kd	CGS001-11140	CDC37	-			
1950	55.92	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
1951	55.88	kd	CGS001-2155	F7	Chymotrypsin			
1952	55.86	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
1953	55.86	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
1954	55.79	kd	CGS001-79733	E2F8	-			
1955	55.63	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
1956	55.61	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
1957	55.59	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
1958	55.59	kd	CGS001-1050	CEBPA	basic leucine zipper proteins			
1959	55.41	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
1960	55.32	kd	CGS001-4552	MTRR	-			
1961	55.3	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
1962	55.28	kd	CGS001-328	APEX1	-			
1963	55.24	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
1964	55.24	kd	CGS001-5378	PMS1	-			
1965	55.23	kd	CGS001-3705	ITPK1	-			
1966	55.17	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
1967	55.15	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
1968	55.13	kd	CGS001-168374	ZNF92	Zinc fingers, C2H2-type			
1969	55.1	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
1970	55.01	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
1971	55	cp	BRD-K63265447	docetaxel	Tubulin inhibitor		TUBB, BCL2, MAP2, MAP4, MAPT, NR1I2, TUBB1	Tubulin inhibitor
1972	54.99	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1973	54.84	oe	ccsbBroad304_01962	STK16	NAK family			
1974	54.84	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
1975	54.82	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
1976	54.8	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
1977	54.79	oe	ccsbBroad304_04257	SPRY4	-			
1978	54.78	oe	ccsbBroad304_00155	CCND1	-			
1979	54.73	kd	CGS001-10250	SRRM1	-			
1980	54.7	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
1981	54.58	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
1982	54.54	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
1983	54.5	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
1984	54.31	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
1985	54.29	kd	CGS001-4763	NF1	-			
1986	54.28	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
1987	54.27	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
1988	54.25	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
1989	54.24	oe	ccsbBroad304_03186	GMNN	-			
1990	54.21	kd	CGS001-2592	GALT	-			
1991	54.21	oe	ccsbBroad304_02002	RNMT	-			
1992	54.2	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
1993	54.16	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
1994	54.15	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
1995	54.13	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
1996	54.08	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
1997	54.06	kd	CGS001-978	CDA	-			
1998	54.05	cp	BRD-K37814297	acepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
1999	54.01	cc		Lipocalins GOF	-			
2000	53.96	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
2001	53.95	kd	CGS001-7936	RDBP	-			
2002	53.83	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
2003	53.8	kd	CGS001-221391	OPN5	GPCR / Class A : Opsin receptors			
2004	53.78	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
2005	53.76	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2006	53.75	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
2007	53.74	kd	CGS001-3783	KCNN4	Calcium-activated potassium channels			
2008	53.73	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
2009	53.72	kd	CGS001-374291	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
2010	53.58	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2011	53.55	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
2012	53.41	kd	CGS001-4204	MECP2	-			
2013	53.29	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
2014	53.13	kd	CGS001-10202	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2015	53.03	kd	CGS001-9263	STK17A	Death-associated kinase (DAPK) family			
2016	53.03	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
2017	53.02	kd	CGS001-9738	CCP110	-			
2018	53	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
2019	52.99	oe	ccsbBroad304_08993	DHDDS	-			
2020	52.98	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
2021	52.98	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
2022	52.97	kd	CGS001-4905	NSF	ATPases / AAA-type			
2023	52.9	kd	CGS001-5887	RAD23B	-			
2024	52.88	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
2025	52.87	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
2026	52.85	kd	CGS001-122402	TDRD9	Tudor domain containing			
2027	52.82	kd	CGS001-1493	CTLA4	CD molecules			
2028	52.81	kd	CGS001-7846	TUBA1A	Tubulins			
2029	52.74	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
2030	52.74	kd	CGS001-1356	CP	-			
2031	52.71	kd	CGS001-9475	ROCK2	Pleckstrin homology (PH) domain containing			
2032	52.7	kd	CGS001-5618	PRLR	Prolactin receptor family			
2033	52.69	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
2034	52.66	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
2035	52.64	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
2036	52.61	kd	CGS001-4043	LRPAP1	-			
2037	52.6	cc		Serotonin receptor agonist	-			
2038	52.6	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
2039	52.58	oe	ccsbBroad304_08167	DNTTIP2	-			
2040	52.57	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
2041	52.55	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
2042	52.53	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
2043	52.49	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
2044	52.48	kd	CGS001-8878	SQSTM1	-			
2045	52.36	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
2046	52.35	oe	ccsbBroad304_03372	CAB39	-			
2047	52.31	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
2048	52.29	kd	CGS001-4916	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
2049	52.24	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
2050	52.23	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
2051	52.1	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
2052	52.03	oe	ccsbBroad304_08952	E2F8	-			
2053	52.02	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
2054	51.94	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
2055	51.89	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
2056	51.84	kd	CGS001-2313	FLI1	ETS Transcription Factors			
2057	51.83	cp	BRD-K04196797	oxcarbazepine	Sodium channel blocker		CYP2C19, CYP3A4, CYP3A5, SCN1A, SCN3A, SCN5A	Sodium channel blocker
2058	51.81	kd	CGS001-25987	TSKU	-			
2059	51.81	kd	CGS001-10887	PROKR1	GPCR / Class A : Prokineticin receptors			
2060	51.79	kd	CGS001-717	C2	Complement system			
2061	51.77	oe	ccsbBroad304_05745	CD24	CD molecules			
2062	51.75	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
2063	51.73	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
2064	51.66	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
2065	51.61	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
2066	51.56	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
2067	51.49	kd	CGS001-10513	APPBP2	-			
2068	51.46	kd	CGS001-1738	DLD	-			
2069	51.44	oe	ccsbBroad304_00632	GGCX	Carboxylases			
2070	51.4	kd	CGS001-5590	PRKCZ	Iota subfamily			
2071	51.39	kd	CGS001-10078	TSSC4	-			
2072	51.37	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
2073	51.36	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
2074	51.36	kd	CGS001-865	CBFB	-			
2075	51.28	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
2076	51.27	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
2077	51.21	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
2078	51.17	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
2079	51.16	oe	ccsbBroad304_07118	UGDH	-			
2080	51.15	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
2081	51.13	kd	CGS001-9900	SV2A	Major facilitator superfamily (MFS) of transporters			
2082	51.13	kd	CGS001-2010	EMD	-			
2083	51.02	oe	ccsbBroad304_07798	EXOC3	-			
2084	50.96	kd	CGS001-11232	POLG2	DNA polymerases			
2085	50.91	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
2086	50.87	oe	ccsbBroad304_03848	METTL14	-			
2087	50.84	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
2088	50.83	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
2089	50.77	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
2090	50.73	kd	CGS001-27347	STK39	FRAY subfamily			
2091	50.65	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
2092	50.56	kd	CGS001-3690	ITGB3	Integrins			
2093	50.5	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
2094	50.48	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
2095	50.42	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
2096	50.39	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
2097	50.39	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
2098	50.36	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
2099	50.32	cc		EMSY complex LOF	-			
2100	50.24	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
2101	50.17	kd	CGS001-51684	SUFU	-			
2102	50.1	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
2103	50.1	oe	ccsbBroad304_06140	EEF1D	-			
2104	50.03	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
2105	50	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
2106	49.94	kd	CGS001-4316	MMP7	Matrix metallopeptidase			
2107	49.9	kd	CGS001-1407	CRY1	-			
2108	49.88	kd	CGS001-79796	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
2109	49.8	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
2110	49.77	kd	CGS001-7405	UVRAG	-			
2111	49.75	kd	CGS001-4170	MCL1	-			
2112	49.73	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
2113	49.68	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
2114	49.67	kd	CGS001-27113	BBC3	-			
2115	49.59	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
2116	49.59	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
2117	49.57	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
2118	49.56	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
2119	49.56	kd	CGS001-10482	NXF1	-			
2120	49.49	kd	CGS001-2810	SFN	-			
2121	49.48	kd	CGS001-2793	GNGT2	-			
2122	49.47	cp	BRD-K62858456	lomerizine	Calcium channel blocker		ABCB1, CACNA1B, SCN5A	Calcium channel blocker
2123	49.45	cp	BRD-K66206289	lobeline	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist
2124	49.44	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
2125	49.43	kd	CGS001-5546	PRCC	-			
2126	49.38	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
2127	49.34	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
2128	49.12	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
2129	49.08	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
2130	49.06	kd	CGS001-391013	PLA2G2C	-			
2131	48.97	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
2132	48.92	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
2133	48.88	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
2134	48.87	oe	ccsbBroad304_08694	TBX20	T-boxes			
2135	48.86	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
2136	48.85	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
2137	48.74	kd	CGS001-23635	SSBP2	-			
2138	48.71	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
2139	48.69	kd	CGS001-1363	CPE	Carboxypeptidase A			
2140	48.68	kd	CGS001-118738	ZNF488	Zinc fingers, C2H2-type			
2141	48.66	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
2142	48.63	oe	ccsbBroad304_04619	GNG8	-			
2143	48.61	kd	CGS001-1211	CLTA	-			
2144	48.53	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
2145	48.4	kd	CGS001-4507	MTAP	-			
2146	48.39	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
2147	48.36	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
2148	48.34	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
2149	48.33	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
2150	48.28	kd	CGS001-64319	FBRS	-			
2151	48.25	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
2152	48.2	kd	CGS001-10401	PIAS3	Zinc fingers, MIZ-type			
2153	48.16	oe	ccsbBroad304_02133	CD83	CD molecules			
2154	48.14	kd	CGS001-81848	SPRY4	-			
2155	48.12	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
2156	48.11	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
2157	48.04	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
2158	48.04	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
2159	48.03	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
2160	48.01	cp	BRD-A24543851	nornicotine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2161	48	oe	ccsbBroad304_00665	GOT1	-			
2162	47.98	kd	CGS001-3976	LIF	-			
2163	47.95	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
2164	47.94	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
2165	47.92	kd	CGS001-10765	KDM5B	Histone demethylases			
2166	47.9	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
2167	47.87	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
2168	47.83	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
2169	47.81	oe	ccsbBroad304_03118	NRBP1	NRBP family			
2170	47.7	kd	CGS001-80349	WDR61	WD repeat domain containing			
2171	47.68	kd	CGS001-6827	SUPT4H1	-			
2172	47.64	cp	BRD-A80928489	1-monopalmitin	P-glycoprotein inhibitor		ABCB1	P-glycoprotein inhibitor
2173	47.56	oe	ccsbBroad304_01008	KITLG	-			
2174	47.55	oe	ccsbBroad304_05823	ANXA2	Annexins			
2175	47.45	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
2176	47.45	kd	CGS001-833	CARS	Aminoacyl tRNA synthetases / Class I			
2177	47.44	kd	CGS001-1509	CTSD	Cathepsins			
2178	47.38	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
2179	47.33	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
2180	47.31	kd	CGS001-64943	NT5DC2	-			
2181	47.28	kd	CGS001-89765	RSPH1	-			
2182	47.25	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
2183	47.25	oe	ccsbBroad304_03405	CHRAC1	-			
2184	47.18	oe	ccsbBroad304_08104	MED4	-			
2185	47.16	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
2186	47.16	kd	CGS001-6347	CCL2	Chemokine ligands			
2187	47.13	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
2188	47.13	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
2189	47.09	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
2190	47.07	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
2191	47.02	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
2192	46.98	kd	CGS001-5966	REL	NFkappaB transcription factor family			
2193	46.98	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
2194	46.95	kd	CGS001-4179	CD46	CD molecules			
2195	46.94	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
2196	46.87	oe	ccsbBroad304_06518	LDHA	-			
2197	46.81	kd	CGS001-10906	TRAFD1	-			
2198	46.8	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
2199	46.79	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
2200	46.77	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
2201	46.75	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
2202	46.73	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
2203	46.69	oe	ccsbBroad304_07808	RAB11FIP2	-			
2204	46.67	kd	CGS001-3094	HINT1	-			
2205	46.63	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
2206	46.58	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
2207	46.54	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
2208	46.53	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
2209	46.49	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
2210	46.37	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
2211	46.35	kd	CGS001-8777	MPDZ	-			
2212	46.27	oe	ccsbBroad304_02668	PNKP	-			
2213	46.26	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
2214	46.02	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
2215	46.01	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
2216	46	oe	ccsbBroad304_01985	EIF3H	-			
2217	45.99	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
2218	45.93	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
2219	45.92	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
2220	45.89	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
2221	45.82	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
2222	45.81	kd	CGS001-7572	ZNF24	Zinc fingers, C2H2-type			
2223	45.69	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
2224	45.69	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
2225	45.68	cc		Nucleophosmin inhibitor	-			
2226	45.67	kd	CGS001-154197	PNLDC1	-			
2227	45.61	kd	CGS001-5164	PDK2	PDHK family			
2228	45.59	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
2229	45.57	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
2230	45.53	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
2231	45.51	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
2232	45.42	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
2233	45.38	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
2234	45.37	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
2235	45.35	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
2236	45.29	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
2237	45.26	kd	CGS001-26036	ZNF451	Zinc fingers, C2H2-type			
2238	45.23	kd	CGS001-10795	ZNF268	Zinc fingers, C2H2-type			
2239	45.16	kd	CGS001-23161	SNX13	Sorting nexins			
2240	45.15	cp	BRD-K29653726	topiramate	Carbonic anhydrase inhibitor		CA2, CA4, GRIK1, CA1, CA12, CA7, CYP2C19, CYP3A4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA1, SCN1A, SCN5A	Carbonic anhydrase inhibitor, Glutamate receptor antagonist, Kainate receptor antagonist
2241	45.11	kd	CGS001-23408	SIRT5	Histone deacetylases			
2242	45.09	oe	ccsbBroad304_02048	BCL10	-			
2243	45.06	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
2244	45.04	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
2245	45.01	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
2246	44.96	kd	CGS001-21	ABCA3	ATP binding cassette transporters / subfamily A			
2247	44.84	oe	ccsbBroad304_05757	ACADS	-			
2248	44.83	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2249	44.81	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
2250	44.8	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
2251	44.74	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
2252	44.74	kd	CGS001-23429	RYBP	-			
2253	44.72	kd	CGS001-9847	KIAA0528	-			
2254	44.68	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
2255	44.68	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
2256	44.66	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
2257	44.59	oe	ccsbBroad304_03858	SRPRB	-			
2258	44.59	kd	CGS001-776	CACNA1D	Calcium channel subunits			
2259	44.58	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
2260	44.57	kd	CGS001-10475	TRIM38	-			
2261	44.54	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
2262	44.54	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
2263	44.51	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
2264	44.5	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
2265	44.46	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
2266	44.46	kd	CGS001-9380	GRHPR	-			
2267	44.45	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
2268	44.33	kd	CGS001-6810	STX4	-			
2269	44.32	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
2270	44.32	kd	CGS001-93487	MAPK1IP1L	-			
2271	44.31	oe	ccsbBroad304_00883	ISG20	-			
2272	44.28	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2273	44.26	kd	CGS001-4773	NFATC2	Nuclear factor of activated T-cells			
2274	44.17	cp	BRD-A87125127	3-matida	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2275	44.15	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
2276	44.09	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
2277	44.07	kd	CGS001-9455	HOMER2	-			
2278	43.99	kd	CGS001-83729	INHBE	-			
2279	43.97	oe	ccsbBroad304_01013	MIF	-			
2280	43.85	kd	CGS001-23142	DCUN1D4	-			
2281	43.82	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
2282	43.73	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
2283	43.69	kd	CGS001-9632	SEC24C	-			
2284	43.68	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
2285	43.66	oe	ccsbBroad304_06837	RAF1	RAF family			
2286	43.63	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
2287	43.63	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
2288	43.55	kd	CGS001-84333	PCGF5	Polycomb group ring fingers			
2289	43.55	kd	CGS001-599	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2290	43.52	oe	ccsbBroad304_02313	ACTR3	-			
2291	43.51	kd	CGS001-9791	PTDSS1	-			
2292	43.51	kd	CGS001-26086	GPSM1	Tetratricopeptide (TTC) repeat domain containing			
2293	43.42	cc		Thromboxane receptor antagonist	-			
2294	43.39	kd	CGS001-10048	RANBP9	-			
2295	43.37	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
2296	43.32	cc		MEK inhibitor	-			
2297	43.29	kd	CGS001-390212	GPR152	GPCR / Class A : Orphans			
2298	43.28	oe	ccsbBroad304_02554	TRAFD1	-			
2299	43.27	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2300	43.21	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
2301	43.2	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2302	43.16	kd	CGS001-5049	PAFAH1B2	-			
2303	43.12	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
2304	43.09	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
2305	43.05	kd	CGS001-23405	DICER1	-			
2306	42.98	kd	CGS001-8892	EIF2B2	-			
2307	42.97	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
2308	42.96	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
2309	42.95	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
2310	42.78	kd	CGS001-51002	TPRKB	-			
2311	42.78	kd	CGS001-9955	HS3ST3A1	Sulfotransferases, membrane-bound			
2312	42.77	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
2313	42.73	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
2314	42.72	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
2315	42.72	kd	CGS001-4121	MAN1A1	-			
2316	42.71	kd	CGS001-23223	RRP12	-			
2317	42.67	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
2318	42.64	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
2319	42.61	kd	CGS001-55837	EAPP	-			
2320	42.6	kd	CGS001-23043	TNIK	MSN subfamily			
2321	42.56	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
2322	42.53	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
2323	42.51	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
2324	42.45	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
2325	42.38	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
2326	42.36	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
2327	42.36	kd	CGS001-51727	CMPK1	-			
2328	42.34	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
2329	42.33	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
2330	42.29	kd	CGS001-4836	NMT1	-			
2331	42.28	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
2332	42.26	oe	ccsbBroad304_05547	TMEM110	-			
2333	42.22	cc		KCNJ11 modulator	-			
2334	42.22	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
2335	42.2	kd	CGS001-79960	PHF17	-			
2336	42.13	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
2337	42.11	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
2338	42.11	kd	CGS001-64077	LHPP	-			
2339	42.08	oe	ccsbBroad304_07217	AXIN2	-			
2340	41.92	kd	CGS001-4904	YBX1	-			
2341	41.91	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
2342	41.86	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
2343	41.85	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
2344	41.84	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2345	41.84	kd	CGS001-5817	PVR	Immunoglobulin superfamily / C2-set domain containing			
2346	41.81	oe	ccsbBroad304_01701	TPI1	-			
2347	41.81	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
2348	41.8	kd	CGS001-150094	SIK1	QIK subfamily			
2349	41.79	kd	CGS001-5469	MED1	-			
2350	41.76	kd	CGS001-9131	AIFM1	-			
2351	41.75	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
2352	41.73	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
2353	41.71	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
2354	41.69	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
2355	41.66	oe	ccsbBroad304_02012	FADD	-			
2356	41.66	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
2357	41.66	kd	CGS001-6233	RPS27A	S ribosomal proteins			
2358	41.65	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
2359	41.61	kd	CGS001-790	CAD	-			
2360	41.6	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
2361	41.59	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
2362	41.59	kd	CGS001-4711	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
2363	41.58	cc		DNA synthesis inhibitor	-			
2364	41.58	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
2365	41.53	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
2366	41.43	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
2367	41.43	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
2368	41.42	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
2369	41.41	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
2370	41.4	oe	ccsbBroad304_07616	ZNF238	-			
2371	41.38	kd	CGS001-811	CALR	-			
2372	41.36	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
2373	41.35	kd	CGS001-1112	FOXN3	Forkhead boxes			
2374	41.35	kd	CGS001-8894	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2375	41.32	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
2376	41.32	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
2377	41.3	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
2378	41.27	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
2379	41.24	kd	CGS001-5004	ORM1	Lipocalins			
2380	41.22	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
2381	41.18	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
2382	41.18	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
2383	41.18	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
2384	41.05	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
2385	41	oe	ccsbBroad304_09756	PAQR7	-			
2386	41	kd	CGS001-4190	MDH1	-			
2387	40.99	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
2388	40.99	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
2389	40.98	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
2390	40.98	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
2391	40.96	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
2392	40.95	kd	CGS001-103	ADAR	-			
2393	40.93	kd	CGS001-2184	FAH	-			
2394	40.9	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
2395	40.89	oe	ccsbBroad304_13499	KSR2	RAF family			
2396	40.86	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
2397	40.83	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
2398	40.82	kd	CGS001-7079	TIMP4	-			
2399	40.79	kd	CGS001-2767	GNA11	-			
2400	40.75	kd	CGS001-5898	RALA	-			
2401	40.73	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
2402	40.69	kd	CGS001-382	ARF6	ADP-ribosylation factors			
2403	40.68	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
2404	40.63	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
2405	40.61	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
2406	40.61	kd	CGS001-23670	TMEM2	-			
2407	40.61	kd	CGS001-727	C5	Endogenous ligands			
2408	40.6	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
2409	40.54	oe	ccsbBroad304_02414	IRF9	-			
2410	40.54	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
2411	40.54	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
2412	40.51	kd	CGS001-10165	SLC25A13	Mitochondrial amino acid transporter subfamily			
2413	40.47	kd	CGS001-6434	TRA2B	RNA binding motif (RRM) containing			
2414	40.46	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
2415	40.45	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
2416	40.43	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
2417	40.42	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
2418	40.39	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
2419	40.37	cc		Sigma receptor antagonist	-			
2420	40.35	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
2421	40.35	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
2422	40.31	oe	ccsbBroad304_07557	NAMPT	-			
2423	40.25	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
2424	40.24	oe	ccsbBroad304_04170	PANK2	-			
2425	40.24	kd	CGS001-3566	IL4R	IL-2 receptor family			
2426	40.23	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
2427	40.23	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
2428	40.23	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
2429	40.19	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
2430	40.19	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
2431	40.08	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
2432	40.06	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
2433	40.05	kd	CGS001-4175	MCM6	-			
2434	40.04	kd	CGS001-8895	CPNE3	-			
2435	40.03	kd	CGS001-5581	PRKCE	Eta subfamily			
2436	40.02	oe	ccsbBroad304_02243	DLGAP5	-			
2437	40.01	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
2438	39.97	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
2439	39.96	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
2440	39.93	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
2441	39.91	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
2442	39.88	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
2443	39.83	kd	CGS001-2617	GARS	Aminoacyl tRNA synthetases / Class II			
2444	39.79	oe	ccsbBroad304_02057	P4HA2	-			
2445	39.73	kd	CGS001-5359	PLSCR1	-			
2446	39.71	kd	CGS001-211	ALAS1	-			
2447	39.69	kd	CGS001-23576	DDAH1	Dimethylarginine dimethylaminohydrolases			
2448	39.65	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
2449	39.64	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
2450	39.62	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
2451	39.6	oe	ccsbBroad304_03266	ERGIC2	-			
2452	39.54	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
2453	39.49	kd	CGS001-8089	YEATS4	-			
2454	39.36	oe	ccsbBroad304_10846	GGT1	CD molecules			
2455	39.36	kd	CGS001-634	CEACAM1	CD molecules			
2456	39.35	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
2457	39.32	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
2458	39.31	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
2459	39.31	oe	ccsbBroad304_00424	DBI	-			
2460	39.31	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
2461	39.28	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
2462	39.28	oe	ccsbBroad304_05907	BUB1B	Bub family			
2463	39.21	kd	CGS001-205564	SENP5	-			
2464	39.2	oe	ccsbBroad304_05981	CDO1	-			
2465	39.2	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
2466	39.19	kd	CGS001-8800	PEX11A	-			
2467	39.16	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
2468	39.14	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
2469	39.13	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
2470	39.13	kd	CGS001-7625	ZNF74	Zinc fingers, C2H2-type			
2471	39.07	oe	ccsbBroad304_00184	C2	Complement system			
2472	39.07	kd	CGS001-51268	PIPOX	-			
2473	39.03	kd	CGS001-3251	HPRT1	-			
2474	39.01	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
2475	38.99	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
2476	38.95	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
2477	38.94	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
2478	38.92	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
2479	38.91	oe	ccsbBroad304_03533	CDCA8	-			
2480	38.91	kd	CGS001-170463	SSBP4	-			
2481	38.9	kd	CGS001-3053	SERPIND1	Serine (or cysteine) peptidase inhibitors			
2482	38.88	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
2483	38.85	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
2484	38.84	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
2485	38.81	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
2486	38.76	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
2487	38.75	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
2488	38.73	oe	ccsbBroad304_00783	HPRT1	-			
2489	38.69	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
2490	38.69	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
2491	38.64	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
2492	38.62	kd	CGS001-444	ASPH	-			
2493	38.6	oe	ccsbBroad304_03746	CDC42SE1	-			
2494	38.57	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
2495	38.56	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
2496	38.48	kd	CGS001-604	BCL6	BTB/POZ domain containing			
2497	38.47	oe	ccsbBroad304_06286	GLUL	-			
2498	38.45	oe	ccsbBroad304_07598	PEMT	-			
2499	38.42	kd	CGS001-10745	PHTF1	-			
2500	38.38	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
2501	38.37	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
2502	38.32	cp	BRD-A68589262	troxipide	Glucosamine synthetase stimulant			Glucosamine synthetase stimulant
2503	38.21	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
2504	38.19	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2505	38.19	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
2506	38.18	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
2507	38.12	kd	CGS001-7511	XPNPEP1	Methionyl aminopeptidase			
2508	38.09	oe	ccsbBroad304_02239	RASSF2	-			
2509	38.09	kd	CGS001-2878	GPX3	-			
2510	38.03	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
2511	38.02	kd	CGS001-91949	COG7	Components of oligomeric golgi complex			
2512	37.91	cc		Poly ADP ribose polymerases LOF	-			
2513	37.91	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
2514	37.89	kd	CGS001-8836	GGH	Gamma-glutamyl hydrolase			
2515	37.86	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
2516	37.81	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
2517	37.78	kd	CGS001-10381	TUBB3	Tubulins			
2518	37.75	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
2519	37.75	kd	CGS001-64786	TBC1D15	-			
2520	37.74	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
2521	37.71	kd	CGS001-7693	ZNF134	Zinc fingers, C2H2-type			
2522	37.69	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
2523	37.68	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
2524	37.58	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
2525	37.55	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
2526	37.53	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
2527	37.51	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
2528	37.51	kd	CGS001-6098	ROS1	Type XVII RTKs: ROS receptors			
2529	37.46	kd	CGS001-55324	ABCF3	ATP binding cassette transporters / subfamily F			
2530	37.45	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
2531	37.44	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
2532	37.44	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
2533	37.42	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
2534	37.38	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2535	37.37	kd	CGS001-51601	LIPT1	-			
2536	37.24	kd	CGS001-23509	POFUT1	Fucosyltransferases			
2537	37.23	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
2538	37.22	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
2539	37.09	kd	CGS001-84109	QRFPR	GPCR / Class A : RF amide peptide receptors			
2540	37.08	kd	CGS001-283450	C12ORF51	-			
2541	37.04	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
2542	37.01	kd	CGS001-55722	CEP72	-			
2543	37	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
2544	36.97	kd	CGS001-11007	CCDC85B	-			
2545	36.88	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
2546	36.83	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
2547	36.83	kd	CGS001-9637	FEZ2	-			
2548	36.79	oe	ccsbBroad304_00725	HADHA	-			
2549	36.74	oe	ccsbBroad304_04404	TUBB6	Tubulins			
2550	36.72	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
2551	36.71	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
2552	36.71	kd	CGS001-2260	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
2553	36.7	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
2554	36.7	kd	CGS001-11198	SUPT16H	-			
2555	36.69	oe	ccsbBroad304_02653	PRAF2	-			
2556	36.67	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
2557	36.67	kd	CGS001-55509	BATF3	basic leucine zipper proteins			
2558	36.65	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
2559	36.65	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
2560	36.61	oe	ccsbBroad304_05192	SPRED2	-			
2561	36.59	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
2562	36.55	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
2563	36.54	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
2564	36.52	oe	ccsbBroad304_00710	GUSB	-			
2565	36.51	kd	CGS001-58528	RRAGD	-			
2566	36.42	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
2567	36.42	kd	CGS001-29110	TBK1	IKK family			
2568	36.38	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
2569	36.37	oe	ccsbBroad304_07875	SPECC1L	-			
2570	36.37	kd	CGS001-5467	PPARD	Nuclear hormone receptors			
2571	36.35	kd	CGS001-808	CALM3	EF-hand domain containing			
2572	36.35	kd	CGS001-60	ACTB	-			
2573	36.3	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2574	36.3	kd	CGS001-8996	NOL3	-			
2575	36.28	kd	CGS001-22841	RAB11FIP2	-			
2576	36.27	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
2577	36.27	kd	CGS001-375318	AQP12A	Ion channels / Aquaporins			
2578	36.25	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
2579	36.19	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
2580	36.18	kd	CGS001-8204	NRIP1	-			
2581	36.13	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
2582	36.08	kd	CGS001-11113	CIT	Other DMPK family kinases			
2583	36.04	oe	ccsbBroad304_03072	GTPBP8	-			
2584	36.04	kd	CGS001-1594	CYP27B1	Cytochrome P450s			
2585	36.01	kd	CGS001-29911	HOOK2	-			
2586	36	kd	CGS001-8050	PDHX	-			
2587	35.99	kd	CGS001-8805	TRIM24	TIF1 family			
2588	35.98	kd	CGS001-5710	PSMD4	Proteasome (prosome, macropain) subunits			
2589	35.96	cp	BRD-K82357231	desloratadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2590	35.9	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
2591	35.9	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
2592	35.89	cp	BRD-K60690191	MPEP	Glutamate receptor antagonist		GRM5, GRM1, GRM4	Glutamate receptor antagonist
2593	35.89	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
2594	35.87	kd	CGS001-1955	MEGF9	-			
2595	35.85	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
2596	35.85	oe	ccsbBroad304_01923	UXT	-			
2597	35.75	cp	BRD-K43236057	piceid	ICAM1 inhibitor		GAA, XDH	ICAM1 inhibitor
2598	35.75	kd	CGS001-3827	KNG1	Endogenous ligands			
2599	35.71	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
2600	35.7	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
2601	35.68	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
2602	35.67	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
2603	35.64	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
2604	35.62	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
2605	35.59	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
2606	35.58	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
2607	35.57	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
2608	35.57	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
2609	35.56	cp	BRD-K06817181	BRD-K06817181	JAK inhibitor		JAK2	JAK inhibitor
2610	35.53	kd	CGS001-6774	STAT3	SH2 domain containing			
2611	35.5	oe	ccsbBroad304_02372	SPRY1	-			
2612	35.5	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
2613	35.47	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
2614	35.43	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
2615	35.39	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
2616	35.37	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
2617	35.34	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
2618	35.33	oe	ccsbBroad304_00747	HLF	-			
2619	35.32	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
2620	35.27	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
2621	35.26	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
2622	35.25	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2623	35.24	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
2624	35.13	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
2625	35.12	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
2626	35.11	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
2627	35.1	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
2628	35.09	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
2629	35.08	kd	CGS001-4547	MTTP	-			
2630	35.07	kd	CGS001-4122	MAN2A2	-			
2631	35.06	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
2632	35.02	kd	CGS001-10392	NOD1	Nucleotide-binding domain and leucine rich repeat containing			
2633	35.02	kd	CGS001-3127	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
2634	34.97	oe	ccsbBroad304_00120	ATOX1	-			
2635	34.96	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
2636	34.93	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
2637	34.93	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
2638	34.92	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
2639	34.92	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
2640	34.89	oe	ccsbBroad304_08797	FASTKD5	-			
2641	34.88	cc		PKC inhibitor	-			
2642	34.86	oe	ccsbBroad304_06720	PHYH	-			
2643	34.86	kd	CGS001-3032	HADHB	-			
2644	34.85	kd	CGS001-19	ABCA1	ATP binding cassette transporters / subfamily A			
2645	34.79	kd	CGS001-6603	SMARCD2	-			
2646	34.78	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
2647	34.7	kd	CGS001-5933	RBL1	-			
2648	34.68	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
2649	34.64	kd	CGS001-5894	RAF1	RAF family			
2650	34.63	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
2651	34.63	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
2652	34.57	oe	ccsbBroad304_06462	ITGAE	Integrins			
2653	34.54	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
2654	34.52	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
2655	34.52	kd	CGS001-3169	FOXA1	Forkhead boxes			
2656	34.5	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
2657	34.48	kd	CGS001-9344	TAOK2	TAO subfamily			
2658	34.42	kd	CGS001-2212	FCGR2A	CD molecules			
2659	34.38	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
2660	34.32	kd	CGS001-9817	KEAP1	Kelch-like proteins			
2661	34.3	kd	CGS001-7342	UBP1	-			
2662	34.27	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
2663	34.22	oe	ccsbBroad304_00370	CS	-			
2664	34.22	cp	BRD-K27184429	levocetirizine	Histamine receptor antagonist		HRH1, CXCL8	Histamine receptor antagonist
2665	34.2	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
2666	34.18	cc		Cyclins LOF	-			
2667	34.18	oe	ccsbBroad304_00709	GUK1	-			
2668	34.16	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
2669	34.14	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
2670	34.1	oe	ccsbBroad304_00519	ETFB	-			
2671	34.09	kd	CGS001-10489	LRRC41	-			
2672	34.08	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
2673	34.03	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
2674	34	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
2675	34	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
2676	33.93	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
2677	33.92	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
2678	33.91	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
2679	33.91	oe	ccsbBroad304_04406	PLA2G12B	-			
2680	33.91	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
2681	33.9	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
2682	33.89	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
2683	33.85	oe	ccsbBroad304_03773	CIAPIN1	-			
2684	33.76	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
2685	33.72	kd	CGS001-65975	STK33	CAMK-unique family			
2686	33.71	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
2687	33.64	kd	CGS001-23038	WDTC1	DDB1 and CUL4 associated factors			
2688	33.57	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
2689	33.56	oe	ccsbBroad304_06862	RGS3	-			
2690	33.55	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
2691	33.52	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
2692	33.51	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
2693	33.49	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
2694	33.49	kd	CGS001-5479	PPIB	-			
2695	33.48	oe	ccsbBroad304_05038	HORMAD2	-			
2696	33.47	oe	ccsbBroad304_06235	G6PD	-			
2697	33.46	kd	CGS001-25874	BRP44	-			
2698	33.43	oe	ccsbBroad304_01174	PEX13	-			
2699	33.42	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
2700	33.41	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
2701	33.37	kd	CGS001-1643	DDB2	WD repeat domain containing			
2702	33.31	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
2703	33.26	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
2704	33.25	cc		S100 calcium binding proteins LOF	-			
2705	33.25	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
2706	33.25	kd	CGS001-6885	MAP3K7	MAPKKK:TAK1 subfamily			
2707	33.17	kd	CGS001-3376	IARS	Aminoacyl tRNA synthetases / Class I			
2708	33.14	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
2709	33.12	oe	ccsbBroad304_01664	TGFA	-			
2710	33.12	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
2711	33.12	kd	CGS001-11168	PSIP1	-			
2712	33.1	kd	CGS001-283455	KSR2	RAF family			
2713	33.09	kd	CGS001-22930	RAB3GAP1	-			
2714	33.06	oe	ccsbBroad304_00459	DPYD	-			
2715	33.05	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
2716	33.03	kd	CGS001-51071	DERA	-			
2717	32.98	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
2718	32.97	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
2719	32.95	kd	CGS001-26277	TINF2	-			
2720	32.94	kd	CGS001-2920	CXCL2	Endogenous ligands			
2721	32.92	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
2722	32.87	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
2723	32.87	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
2724	32.86	kd	CGS001-9221	NOLC1	-			
2725	32.84	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
2726	32.82	kd	CGS001-200734	SPRED2	-			
2727	32.8	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
2728	32.77	kd	CGS001-5167	ENPP1	-			
2729	32.75	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
2730	32.75	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
2731	32.74	oe	ccsbBroad304_09358	MAPK1IP1L	-			
2732	32.71	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
2733	32.67	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
2734	32.67	kd	CGS001-6925	TCF4	Basic helix-loop-helix proteins			
2735	32.62	oe	ccsbBroad304_03641	ASF1B	-			
2736	32.61	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
2737	32.6	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2738	32.57	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
2739	32.57	kd	CGS001-2052	EPHX1	-			
2740	32.56	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
2741	32.55	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
2742	32.53	kd	CGS001-6046	BRD2	Bromodomain kinase (BRDK) family			
2743	32.5	kd	CGS001-3880	KRT19	Intermediate filaments type I, keratins (acidic)			
2744	32.45	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
2745	32.44	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
2746	32.43	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
2747	32.42	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
2748	32.42	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
2749	32.4	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
2750	32.4	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
2751	32.4	kd	CGS001-8467	SMARCA5	-			
2752	32.39	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
2753	32.37	kd	CGS001-6251	RSU1	-			
2754	32.37	kd	CGS001-116443	GRIN3A	Glutamate receptors			
2755	32.36	cc		Aminoacyl tRNA synthetases class II LOF	-			
2756	32.36	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
2757	32.35	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2758	32.34	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
2759	32.34	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
2760	32.3	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
2761	32.28	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
2762	32.28	kd	CGS001-161725	OTUD7A	OTU domain containing			
2763	32.25	kd	CGS001-2786	GNG4	-			
2764	32.24	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
2765	32.24	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
2766	32.24	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
2767	32.23	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
2768	32.22	kd	CGS001-5577	PRKAR2B	Protein kinase A			
2769	32.18	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2770	32.15	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
2771	32.14	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2772	32.14	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
2773	32.08	oe	ccsbBroad304_00486	EFNB2	Ephrins			
2774	32.08	kd	CGS001-22933	SIRT2	Histone deacetylases			
2775	32.03	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
2776	31.94	kd	CGS001-6715	SRD5A1	-			
2777	31.92	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
2778	31.91	oe	ccsbBroad304_01716	TSN	-			
2779	31.91	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
2780	31.84	kd	CGS001-8743	TNFSF10	CD molecules			
2781	31.81	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
2782	31.79	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
2783	31.75	kd	CGS001-3418	IDH2	-			
2784	31.65	cp	BRD-A96107863	nisoldipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNB2, CYP3A5	Calcium channel blocker
2785	31.65	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
2786	31.65	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
2787	31.64	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
2788	31.63	oe	ccsbBroad304_01641	TAF13	-			
2789	31.58	oe	ccsbBroad304_01613	STK11	LKB subfamily			
2790	31.53	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
2791	31.51	cc		PARP inhibitor	-			
2792	31.51	kd	CGS001-22944	KIN	-			
2793	31.5	kd	CGS001-5649	RELN	-			
2794	31.49	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
2795	31.48	kd	CGS001-7175	TPR	-			
2796	31.47	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
2797	31.45	kd	CGS001-56848	SPHK2	Sphingosine kinase			
2798	31.44	oe	ccsbBroad304_05948	CCND2	-			
2799	31.43	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
2800	31.39	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
2801	31.35	oe	ccsbBroad304_01392	TRIM27	-			
2802	31.33	kd	CGS001-976	CD97	Adhesion Class GPCRs			
2803	31.32	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
2804	31.3	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2805	31.28	oe	ccsbBroad304_00509	EPHX1	-			
2806	31.28	kd	CGS001-55234	SMU1	WD repeat domain containing			
2807	31.28	kd	CGS001-2138	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2808	31.28	kd	CGS001-901	CCNG2	-			
2809	31.21	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2810	31.19	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
2811	31.17	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
2812	31.14	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
2813	31.12	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
2814	31.12	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
2815	31.09	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
2816	31.08	kd	CGS001-9709	HERPUD1	-			
2817	31.07	kd	CGS001-109	ADCY3	Adenylyl cyclases			
2818	31.04	kd	CGS001-183	AGT	Endogenous ligands			
2819	31.01	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2820	31	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
2821	30.97	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
2822	30.96	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
2823	30.95	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
2824	30.87	kd	CGS001-4717	NDUFC1	Mitochondrial respiratory chain complex / Complex I			
2825	30.85	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
2826	30.85	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
2827	30.81	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
2828	30.81	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
2829	30.79	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
2830	30.75	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
2831	30.74	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
2832	30.72	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
2833	30.69	kd	CGS001-8802	SUCLG1	-			
2834	30.68	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
2835	30.68	kd	CGS001-5899	RALB	-			
2836	30.67	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
2837	30.66	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
2838	30.66	kd	CGS001-1497	CTNS	-			
2839	30.65	kd	CGS001-1440	CSF3	Endogenous ligands			
2840	30.63	kd	CGS001-29984	RHOD	-			
2841	30.61	kd	CGS001-93185	IGSF8	CD molecules			
2842	30.54	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
2843	30.53	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
2844	30.51	kd	CGS001-3364	HUS1	-			
2845	30.46	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
2846	30.46	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
2847	30.45	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
2848	30.44	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
2849	30.42	oe	ccsbBroad304_00931	LCN2	Lipocalins			
2850	30.41	cp	BRD-A35519318	benidipine	Calcium channel blocker		CACNA1C, CACNA1G, CYP3A5	Calcium channel blocker
2851	30.39	oe	ccsbBroad304_03269	CD320	CD molecules			
2852	30.36	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
2853	30.33	oe	ccsbBroad304_02496	MTX2	-			
2854	30.31	oe	ccsbBroad304_03950	ATG3	-			
2855	30.31	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
2856	30.31	kd	CGS001-81577	GFOD2	-			
2857	30.3	kd	CGS001-7029	TFDP2	-			
2858	30.29	kd	CGS001-79090	TRAPPC6A	Trafficking protein particle complex			
2859	30.25	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
2860	30.23	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
2861	30.23	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
2862	30.21	kd	CGS001-1649	DDIT3	-			
2863	30.19	kd	CGS001-2	A2M	-			
2864	30.17	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
2865	30.15	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2866	30.15	kd	CGS001-9352	TXNL1	-			
2867	30.14	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
2868	30.08	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
2869	30.08	kd	CGS001-57787	MARK4	MARK subfamily			
2870	30.03	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
2871	30.01	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
2872	30	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
2873	29.98	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
2874	29.95	cp	BRD-K56614220	clofazimine	GK0582 inhibitor			GK0582 inhibitor
2875	29.94	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
2876	29.91	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
2877	29.88	oe	ccsbBroad304_06085	DCK	-			
2878	29.88	oe	ccsbBroad304_03268	GMPR2	-			
2879	29.85	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
2880	29.85	kd	CGS001-7158	TP53BP1	-			
2881	29.83	kd	CGS001-2295	FOXF2	Forkhead boxes			
2882	29.81	kd	CGS001-3927	LASP1	-			
2883	29.8	kd	CGS001-27035	NOX1	-			
2884	29.7	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
2885	29.67	kd	CGS001-11014	KDELR2	-			
2886	29.63	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
2887	29.62	oe	ccsbBroad304_07768	NISCH	-			
2888	29.61	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
2889	29.59	oe	ccsbBroad304_06783	LGMN	Legumain			
2890	29.59	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
2891	29.56	oe	ccsbBroad304_08116	TBK1	IKK family			
2892	29.56	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
2893	29.51	kd	CGS001-51160	VPS28	-			
2894	29.46	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
2895	29.45	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
2896	29.45	kd	CGS001-4091	SMAD6	SMADs			
2897	29.35	oe	ccsbBroad304_08709	SCYL3	-			
2898	29.34	kd	CGS001-36	ACADSB	-			
2899	29.33	kd	CGS001-5594	MAPK1	MAPK:ERK subfamily			
2900	29.3	oe	ccsbBroad304_06789	PSEN2	Presenilin			
2901	29.28	oe	ccsbBroad304_01672	TIMP2	-			
2902	29.28	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
2903	29.28	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
2904	29.27	kd	CGS001-54901	CDKAL1	-			
2905	29.26	kd	CGS001-10554	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
2906	29.24	kd	CGS001-5888	RAD51	-			
2907	29.23	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
2908	29.2	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
2909	29.2	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
2910	29.18	kd	CGS001-8864	PER2	-			
2911	29.17	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
2912	29.17	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
2913	29.16	kd	CGS001-10628	TXNIP	-			
2914	29.11	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
2915	29.11	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
2916	29.04	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
2917	29.02	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
2918	29	kd	CGS001-7010	TEK	Type XII RTKs: TIE family of angiopoietin receptors			
2919	28.99	kd	CGS001-23386	NUDCD3	-			
2920	28.98	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
2921	28.94	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
2922	28.92	oe	ccsbBroad304_02534	UTP14A	-			
2923	28.88	kd	CGS001-5535	PPP3R2	EF-hand domain containing			
2924	28.86	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
2925	28.85	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
2926	28.82	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
2927	28.8	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
2928	28.79	kd	CGS001-5624	PROC	Endogenous ligands			
2929	28.77	oe	ccsbBroad304_00183	C1S	Complement system			
2930	28.73	kd	CGS001-9134	CCNE2	-			
2931	28.7	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
2932	28.7	kd	CGS001-9	NAT1	-			
2933	28.7	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
2934	28.69	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
2935	28.69	oe	ccsbBroad304_00212	CAMLG	-			
2936	28.66	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
2937	28.64	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
2938	28.63	kd	CGS001-8780	RIOK3	RIO3 subfamily			
2939	28.62	oe	ccsbBroad304_07219	CDC7	CDC7 family			
2940	28.62	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
2941	28.61	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
2942	28.6	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
2943	28.6	kd	CGS001-51347	TAOK3	TAO subfamily			
2944	28.59	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2945	28.58	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
2946	28.57	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
2947	28.56	kd	CGS001-595	CCND1	-			
2948	28.52	oe	ccsbBroad304_04194	ELL3	-			
2949	28.51	kd	CGS001-2000	ELF4	ETS Transcription Factors			
2950	28.48	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
2951	28.41	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
2952	28.4	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
2953	28.36	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2954	28.36	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
2955	28.36	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
2956	28.35	kd	CGS001-4947	OAZ2	-			
2957	28.34	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
2958	28.33	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
2959	28.29	oe	ccsbBroad304_03878	SENP2	-			
2960	28.25	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
2961	28.24	oe	ccsbBroad304_03859	ENOPH1	-			
2962	28.24	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
2963	28.2	oe	ccsbBroad304_08392	EXOC6	-			
2964	28.18	kd	CGS001-5925	RB1	Endogenous ligands			
2965	28.16	kd	CGS001-23012	STK38L	NDR family			
2966	28.15	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
2967	28.14	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
2968	28.14	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
2969	28.08	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
2970	28.05	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
2971	28.05	kd	CGS001-4833	NME4	-			
2972	28.02	oe	ccsbBroad304_01398	RHEB	-			
2973	28	kd	CGS001-7100	TLR5	Toll-like receptor family			
2974	27.96	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
2975	27.87	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
2976	27.8	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
2977	27.79	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2978	27.76	kd	CGS001-55423	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
2979	27.75	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
2980	27.73	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2981	27.73	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
2982	27.73	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
2983	27.7	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2984	27.68	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
2985	27.66	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
2986	27.62	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
2987	27.61	oe	ccsbBroad304_02553	BLCAP	-			
2988	27.59	oe	ccsbBroad304_06845	RARRES3	-			
2989	27.58	oe	ccsbBroad304_00060	AMBP	Lipocalins			
2990	27.51	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
2991	27.51	kd	CGS001-4323	MMP14	Matrix metallopeptidase			
2992	27.5	oe	ccsbBroad304_06318	GPER	-			
2993	27.49	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
2994	27.48	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
2995	27.44	oe	ccsbBroad304_09195	MCM8	-			
2996	27.43	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2997	27.37	kd	CGS001-114609	TIRAP	-			
2998	27.36	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
2999	27.36	kd	CGS001-80351	TNKS2	Ankyrin repeat domain containing			
3000	27.34	oe	ccsbBroad304_02589	COPS5	-			
3001	27.33	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
3002	27.32	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
3003	27.28	kd	CGS001-4482	MSRA	-			
3004	27.26	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
3005	27.2	kd	CGS001-5987	TRIM27	-			
3006	27.19	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
3007	27.18	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
3008	27.16	kd	CGS001-308	ANXA5	Annexins			
3009	27.14	cp	BRD-K50384076	7,4'-dihydroxyflavone	Opioid receptor antagonist		CYP19A1	Opioid receptor antagonist
3010	27.14	kd	CGS001-22921	MSRB2	-			
3011	27.09	kd	CGS001-10670	RRAGA	-			
3012	27.09	kd	CGS001-10097	ACTR2	-			
3013	27.08	kd	CGS001-2059	EPS8	-			
3014	27.06	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
3015	26.97	kd	CGS001-2857	GPR34	GPCR / Class A : Orphans			
3016	26.91	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
3017	26.91	kd	CGS001-408	ARRB1	-			
3018	26.85	kd	CGS001-7343	UBTF	-			
3019	26.82	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
3020	26.81	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
3021	26.81	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
3022	26.79	kd	CGS001-5985	RFC5	ATPases / AAA-type			
3023	26.72	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
3024	26.72	kd	CGS001-182	JAG1	CD molecules			
3025	26.71	kd	CGS001-5920	RARRES3	-			
3026	26.7	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
3027	26.63	oe	ccsbBroad304_02526	POP4	-			
3028	26.61	oe	ccsbBroad304_08645	BCCIP	-			
3029	26.61	kd	CGS001-2853	GPR31	GPCR / Class A : Orphans			
3030	26.6	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
3031	26.59	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
3032	26.55	kd	CGS001-326	AIRE	Zinc fingers, PHD-type			
3033	26.51	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
3034	26.48	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
3035	26.44	oe	ccsbBroad304_02399	TNIP1	-			
3036	26.42	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
3037	26.39	oe	ccsbBroad304_00956	LYZ	-			
3038	26.39	kd	CGS001-5813	PURA	-			
3039	26.37	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
3040	26.18	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
3041	26.14	kd	CGS001-384	ARG2	Arginase			
3042	26.12	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
3043	26.1	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3044	26.07	kd	CGS001-9360	PPIG	-			
3045	26.04	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
3046	25.99	kd	CGS001-6146	RPL22	L ribosomal proteins			
3047	25.97	kd	CGS001-271	AMPD2	-			
3048	25.94	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
3049	25.94	oe	ccsbBroad304_01131	OXCT1	-			
3050	25.93	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
3051	25.89	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
3052	25.88	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
3053	25.85	kd	CGS001-29978	UBQLN2	Ubiquilin family			
3054	25.83	kd	CGS001-338557	O3FAR1	-			
3055	25.83	kd	CGS001-1345	COX6C	Mitochondrial respiratory chain complex			
3056	25.8	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
3057	25.75	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
3058	25.69	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
3059	25.66	kd	CGS001-2073	ERCC5	-			
3060	25.65	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
3061	25.65	kd	CGS001-51720	UIMC1	-			
3062	25.65	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
3063	25.65	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
3064	25.62	oe	ccsbBroad304_02843	FTSJ1	-			
3065	25.55	cc		Sirtuins GOF	-			
3066	25.54	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
3067	25.53	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
3068	25.48	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
3069	25.42	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
3070	25.42	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
3071	25.37	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
3072	25.35	oe	ccsbBroad304_08461	CDCA4	-			
3073	25.26	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
3074	25.22	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
3075	25.22	kd	CGS001-5727	PTCH1	-			
3076	25.22	kd	CGS001-4846	NOS3	Nitric oxide synthases			
3077	25.18	oe	ccsbBroad304_12226	NAGK	-			
3078	25.15	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
3079	25.12	kd	CGS001-10014	HDAC5	Histone deacetylases			
3080	25.05	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
3081	25.05	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
3082	25.02	kd	CGS001-4046	LSP1	-			
3083	24.98	kd	CGS001-23057	NMNAT2	-			
3084	24.92	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
3085	24.89	cc		PI3K Signaling LOF	-			
3086	24.85	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
3087	24.84	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
3088	24.84	kd	CGS001-9258	MFHAS1	-			
3089	24.83	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
3090	24.82	kd	CGS001-4299	AFF1	-			
3091	24.81	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
3092	24.8	oe	ccsbBroad304_02533	NOXA1	-			
3093	24.78	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
3094	24.73	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
3095	24.65	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
3096	24.63	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
3097	24.62	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
3098	24.58	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
3099	24.54	oe	ccsbBroad304_00966	MAFG	-			
3100	24.53	kd	CGS001-57720	GPR107	GPCR / Unclassified : 7TM orphan receptors			
3101	24.52	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
3102	24.46	kd	CGS001-23536	ADAT1	-			
3103	24.43	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
3104	24.33	oe	ccsbBroad304_02990	LYPD3	-			
3105	24.29	kd	CGS001-23649	POLA2	DNA polymerases			
3106	24.26	kd	CGS001-10094	ARPC3	Actin related protein 2/3 complex subunits			
3107	24.19	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
3108	24.17	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
3109	24.15	kd	CGS001-563	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
3110	24.14	kd	CGS001-1827	RCAN1	-			
3111	24.12	kd	CGS001-10329	TMEM5	-			
3112	24.1	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
3113	24.09	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
3114	24.06	oe	ccsbBroad304_09354	IGSF8	CD molecules			
3115	23.99	kd	CGS001-5432	POLR2C	RNA polymerase subunits			
3116	23.99	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
3117	23.97	kd	CGS001-3654	IRAK1	Interleukin-1 receptor-associated kinase (IRAK) family			
3118	23.87	kd	CGS001-3718	JAK3	Janus kinase (JakA) family			
3119	23.79	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
3120	23.63	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
3121	23.61	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
3122	23.59	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
3123	23.58	kd	CGS001-51451	LCMT1	-			
3124	23.57	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
3125	23.43	oe	ccsbBroad304_03951	NARFL	-			
3126	23.4	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
3127	23.33	kd	CGS001-23492	CBX7	-			
3128	23.32	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
3129	23.3	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
3130	23.28	kd	CGS001-5338	PLD2	Hydrolases			
3131	23.25	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
3132	23.23	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3133	23.21	kd	CGS001-397	ARHGDIB	Endogenous ligands			
3134	23.2	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
3135	23.19	cc		Beta-adrenergic receptor agonist	-			
3136	23.19	kd	CGS001-7280	TUBB2A	Tubulins			
3137	23.18	kd	CGS001-54658	UGT1A1	UDP glucuronosyltransferases			
3138	23.17	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
3139	23.14	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
3140	23.05	kd	CGS001-7181	NR2C1	Testicular receptors			
3141	23.02	kd	CGS001-6199	RPS6KB2	p70 subfamily			
3142	23.01	kd	CGS001-55869	HDAC8	Histone deacetylases			
3143	22.99	kd	CGS001-56675	NRIP3	-			
3144	22.97	kd	CGS001-190	NR0B1	DAX-like receptors			
3145	22.97	kd	CGS001-1856	DVL2	Dishevelled homologs			
3146	22.89	kd	CGS001-6932	TCF7	-			
3147	22.88	kd	CGS001-336	APOA2	Apolipoproteins			
3148	22.84	kd	CGS001-23464	GCAT	-			
3149	22.75	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
3150	22.73	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
3151	22.73	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
3152	22.69	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
3153	22.64	kd	CGS001-134288	TMEM174	-			
3154	22.62	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
3155	22.62	kd	CGS001-1605	DAG1	-			
3156	22.6	kd	CGS001-1644	DDC	Catecholamine turnover			
3157	22.51	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
3158	22.51	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
3159	22.47	kd	CGS001-84775	ZNF607	Zinc fingers, C2H2-type			
3160	22.46	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
3161	22.39	oe	ccsbBroad304_00032	ADSL	-			
3162	22.39	kd	CGS001-546	ATRX	-			
3163	22.38	kd	CGS001-11112	HIBADH	-			
3164	22.32	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3165	22.12	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3166	22.07	kd	CGS001-2717	GLA	-			
3167	21.88	kd	CGS001-9700	ESPL1	-			
3168	21.84	kd	CGS001-2335	FN1	Endogenous ligands			
3169	21.84	kd	CGS001-116519	APOA5	Apolipoproteins			
3170	21.82	kd	CGS001-2581	GALC	-			
3171	21.81	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
3172	21.78	kd	CGS001-7086	TKT	-			
3173	21.78	kd	CGS001-5292	PIM1	PIM family			
3174	21.77	oe	ccsbBroad304_00880	IRF2	-			
3175	21.74	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
3176	21.7	kd	CGS001-28985	MCTS1	-			
3177	21.68	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
3178	21.68	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
3179	21.62	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
3180	21.61	kd	CGS001-10841	FTCD	-			
3181	21.59	kd	CGS001-1287	COL4A5	Collagens			
3182	21.51	kd	CGS001-3029	HAGH	-			
3183	21.48	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
3184	21.46	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
3185	21.45	kd	CGS001-51520	LARS	Aminoacyl tRNA synthetases / Class I			
3186	21.44	kd	CGS001-3956	LGALS1	Endogenous ligands			
3187	21.35	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
3188	21.35	kd	CGS001-11041	B3GNT1	-			
3189	21.32	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
3190	21.29	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
3191	21.14	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
3192	21.12	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
3193	21.07	kd	CGS001-148103	ZNF599	Zinc fingers, C2H2-type			
3194	21.06	kd	CGS001-9978	RBX1	RING-type (C3HC4) zinc fingers			
3195	21	oe	ccsbBroad304_07766	RASSF1	-			
3196	20.98	kd	CGS001-2194	FASN	Short chain dehydrogenase/reductase superfamily / Atypical members			
3197	20.97	kd	CGS001-6787	NEK4	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3198	20.96	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3199	20.95	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
3200	20.93	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
3201	20.92	oe	ccsbBroad304_01675	TK1	-			
3202	20.9	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
3203	20.75	kd	CGS001-8527	DGKD	Pleckstrin homology (PH) domain containing			
3204	20.74	kd	CGS001-129685	TAF8	-			
3205	20.68	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
3206	20.65	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
3207	20.63	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
3208	20.54	kd	CGS001-4791	NFKB2	NFkappaB transcription factor family			
3209	20.51	kd	CGS001-5591	PRKDC	Other PIKK family kinases			
3210	20.47	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
3211	20.44	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
3212	20.34	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
3213	20.24	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
3214	20.22	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
3215	20.2	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
3216	20.2	kd	CGS001-10196	PRMT3	Protein arginine N-methyltransferases			
3217	20.11	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3218	20.1	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
3219	20.04	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
3220	20.03	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
3221	19.97	kd	CGS001-4072	EPCAM	CD molecules			
3222	19.9	oe	ccsbBroad304_01485	SC5DL	-			
3223	19.89	kd	CGS001-56139	PCDHA10	Cadherins / Protocadherins : Clustered			
3224	19.86	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
3225	19.86	kd	CGS001-817	CAMK2D	CAMK2 family			
3226	19.77	kd	CGS001-3579	CXCR2	Chemokine receptors			
3227	19.76	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
3228	19.75	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
3229	19.72	kd	CGS001-10474	TADA3	-			
3230	19.69	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
3231	19.68	kd	CGS001-51222	ZNF219	Zinc fingers, C2H2-type			
3232	19.67	kd	CGS001-81611	ANP32E	ANP32 acidic nuclear phosphoproteins			
3233	19.66	kd	CGS001-64710	NUCKS1	-			
3234	19.64	kd	CGS001-1445	CSK	Csk family			
3235	19.63	kd	CGS001-5653	KLK6	Chymotrypsin			
3236	19.55	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
3237	19.55	kd	CGS001-5660	PSAP	Endogenous ligands			
3238	19.52	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
3239	19.49	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
3240	19.47	kd	CGS001-23066	CAND2	-			
3241	19.45	oe	ccsbBroad304_00489	EHHADH	-			
3242	19.44	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
3243	19.36	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
3244	19.28	kd	CGS001-56922	MCCC1	-			
3245	19.25	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
3246	19.22	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
3247	19.19	kd	CGS001-4094	MAF	-			
3248	19.14	cc		PRD class homeoboxes and psudogenes LOF	-			
3249	19.14	kd	CGS001-841	CASP8	Caspases			
3250	19.05	kd	CGS001-23743	BHMT2	-			
3251	18.9	kd	CGS001-2266	FGG	Endogenous ligands			
3252	18.85	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
3253	18.81	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
3254	18.78	oe	ccsbBroad304_06095	DFFB	-			
3255	18.74	kd	CGS001-22949	PTGR1	-			
3256	18.7	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
3257	18.69	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
3258	18.65	kd	CGS001-29968	PSAT1	-			
3259	18.62	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
3260	18.59	oe	ccsbBroad304_01872	DGCR14	-			
3261	18.57	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
3262	18.41	kd	CGS001-4594	MUT	-			
3263	18.28	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3264	17.93	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
3265	17.89	kd	CGS001-123803	NTAN1	-			
3266	17.87	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
3267	17.86	kd	CGS001-3460	IFNGR2	Interferon receptor family			
3268	17.81	cc		Estrogen receptor antagonist	-			
3269	17.7	oe	ccsbBroad304_01142	PAFAH1B2	-			
3270	17.61	kd	CGS001-5950	RBP4	Lipocalins			
3271	17.61	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
3272	17.59	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
3273	17.53	kd	CGS001-54498	SMOX	-			
3274	17.52	kd	CGS001-10472	ZNF238	-			
3275	17.51	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
3276	17.45	kd	CGS001-7187	TRAF3	-			
3277	17.35	kd	CGS001-2834	PRLHR	GPCR / Class A : RF amide peptide receptors			
3278	17.28	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
3279	17.19	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
3280	17.18	kd	CGS001-3458	IFNG	Interferons			
3281	17.15	kd	CGS001-4171	MCM2	-			
3282	17.14	kd	CGS001-5163	PDK1	-			
3283	17.09	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
3284	17.05	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
3285	16.99	kd	CGS001-2990	GUSB	-			
3286	16.9	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
3287	16.72	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
3288	16.71	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
3289	16.71	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
3290	16.69	kd	CGS001-10138	YAF2	-			
3291	16.68	oe	ccsbBroad304_04457	TOX2	-			
3292	16.54	kd	CGS001-403	ARL3	ADP-ribosylation factors			
3293	16.47	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
3294	16.44	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3295	16.29	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
3296	16.25	kd	CGS001-125919	ZNF543	Zinc fingers, C2H2-type			
3297	16.22	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
3298	16.21	kd	CGS001-51079	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
3299	16.17	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
3300	16.12	oe	ccsbBroad304_05749	A2M	-			
3301	16.1	oe	ccsbBroad304_02633	LSM6	-			
3302	16.08	kd	CGS001-506	ATP5B	ATPases / F-type			
3303	16	oe	ccsbBroad304_13903	MTAP	-			
3304	15.96	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
3305	15.96	kd	CGS001-4208	MEF2C	Myocyte enhancer factors			
3306	15.93	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
3307	15.87	kd	CGS001-10873	ME3	-			
3308	15.86	kd	CGS001-256281	NUDT14	Nudix motif containing			
3309	15.83	oe	ccsbBroad304_00161	BID	Endogenous ligands			
3310	15.76	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
3311	15.64	oe	ccsbBroad304_01374	RAP1A	-			
3312	15.62	kd	CGS001-10933	MORF4L1	-			
3313	15.58	oe	ccsbBroad304_02094	FIBP	-			
3314	15.52	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
3315	15.4	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
3316	15.33	kd	CGS001-1906	EDN1	Endogenous ligands			
3317	15.3	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
3318	15.3	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
3319	15.29	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
3320	15.19	cc		ATPase inhibitor	-			
3321	15.11	kd	CGS001-3155	HMGCL	-			
3322	15.06	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
3323	14.96	kd	CGS001-94235	GNG8	-			
3324	14.88	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
3325	14.64	oe	ccsbBroad304_01724	TTR	-			
3326	14.5	oe	ccsbBroad304_00034	AES	-			
3327	14.41	oe	ccsbBroad304_00865	ILF2	-			
3328	14.4	kd	CGS001-23192	ATG4B	Aut2 peptidase			
3329	14.34	kd	CGS001-488	ATP2A2	Calcium-ATPases			
3330	14.33	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
3331	14	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
3332	13.9	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
3333	13.68	cc		Mitogen activated protein kinases LOF	-			
3334	13.4	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
3335	13.36	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
3336	13.04	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
3337	13	kd	CGS001-57521	RPTOR	WD repeat domain containing			
3338	12.9	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
3339	12.83	cc		Phospholipases GOF	-			
3340	12.82	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
3341	12.77	kd	CGS001-5883	RAD9A	-			
3342	12.76	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
3343	12.22	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
3344	12.2	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
3345	12.18	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
3346	11.91	oe	ccsbBroad304_03056	MCTS1	-			
3347	11.72	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
3348	11.59	cc		IMPDH inhibitor	-			
3349	11.56	oe	ccsbBroad304_05963	CD44	CD molecules			
3350	11.51	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
3351	11.49	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
3352	11.13	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3353	10.97	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
3354	10.95	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
3355	10.43	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
3356	10.31	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
3357	9.72	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
3358	9.66	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
3359	9.65	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
3360	9.55	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
3361	9.53	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
3362	9.44	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
3363	9.36	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
3364	9.13	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
3365	8.9	kd	CGS001-2931	GSK3A	GSK subfamily			
3366	8.84	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
3367	8.59	oe	ccsbBroad304_06424	IFI16	-			
3368	8.36	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
3369	8.04	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
3370	7.93	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
3371	7.48	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
3372	7.21	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
3373	7.2	cc		Rho GTPase activating proteins LOF	-			
3374	7.15	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
3375	7.13	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
3376	7.01	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
3377	6.29	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
3378	6.25	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
3379	6.1	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
3380	6.08	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
3381	5.97	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
3382	5.07	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
3383	3.73	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
3384	-3.4	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
3385	-4.92	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
3386	-5.62	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
3387	-5.96	kd	CGS001-8536	CAMK1	CAMK1 family			
3388	-6.52	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
3389	-6.66	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
3390	-6.92	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3391	-7.1	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
3392	-7.3	oe	ccsbBroad304_05937	CASP7	Caspases			
3393	-7.58	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
3394	-7.6	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
3395	-7.96	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
3396	-8.03	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
3397	-8.12	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
3398	-8.32	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
3399	-8.58	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
3400	-8.76	kd	CGS001-9156	EXO1	-			
3401	-9.05	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
3402	-9.43	kd	CGS001-8505	PARG	-			
3403	-9.51	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
3404	-9.51	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3405	-9.64	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
3406	-9.65	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
3407	-9.84	kd	CGS001-3675	ITGA3	Integrins			
3408	-9.86	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
3409	-9.88	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
3410	-9.9	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
3411	-9.93	kd	CGS001-5573	PRKAR1A	Protein kinase A			
3412	-10.02	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
3413	-10.1	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3414	-10.23	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
3415	-10.43	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
3416	-10.5	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3417	-10.63	kd	CGS001-3932	LCK	Src family			
3418	-10.93	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
3419	-11	kd	CGS001-10390	CEPT1	-			
3420	-11	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
3421	-11.11	oe	ccsbBroad304_04294	ATG10	-			
3422	-11.34	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
3423	-11.4	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
3424	-11.49	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
3425	-11.58	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
3426	-11.59	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3427	-11.82	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
3428	-11.93	oe	ccsbBroad304_07012	STK3	MST subfamily			
3429	-11.98	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
3430	-12.06	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
3431	-12.23	cc		BCL inhibitor	-			
3432	-12.48	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
3433	-12.6	kd	CGS001-3163	HMOX2	Haem oxygenase			
3434	-12.61	kd	CGS001-6776	STAT5A	SH2 domain containing			
3435	-12.64	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
3436	-12.72	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
3437	-12.83	oe	ccsbBroad304_13880	IDH3G	-			
3438	-12.84	kd	CGS001-4929	NR4A2	Nerve growth factor IB-like receptors			
3439	-12.97	oe	ccsbBroad304_00447	DLD	-			
3440	-13.02	kd	CGS001-83737	ITCH	-			
3441	-13.07	kd	CGS001-6464	SHC1	SH2 domain containing			
3442	-13.11	kd	CGS001-10632	ATP5L	ATPases / F-type			
3443	-13.23	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
3444	-13.25	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
3445	-13.26	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
3446	-13.47	kd	CGS001-32	ACACB	Carboxylases			
3447	-13.51	oe	ccsbBroad304_06180	ESD	-			
3448	-13.57	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
3449	-13.59	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
3450	-13.6	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
3451	-13.65	kd	CGS001-1495	CTNNA1	Catenins			
3452	-13.66	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
3453	-13.68	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
3454	-13.77	cc		Purinergic receptors P2Y GOF	-			
3455	-13.77	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
3456	-13.78	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
3457	-13.8	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
3458	-13.86	oe	ccsbBroad304_00794	HSF1	-			
3459	-13.88	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
3460	-13.91	oe	ccsbBroad304_03853	LSM2	-			
3461	-13.91	oe	ccsbBroad304_00876	INSIG1	-			
3462	-13.91	kd	CGS001-1036	CDO1	-			
3463	-14.08	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
3464	-14.1	kd	CGS001-25801	GCA	EF-hand domain containing			
3465	-14.15	kd	CGS001-55802	DCP1A	-			
3466	-14.22	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
3467	-14.28	kd	CGS001-64425	POLR1E	RNA polymerase subunits			
3468	-14.29	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
3469	-14.29	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3470	-14.42	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
3471	-14.53	kd	CGS001-6009	RHEB	-			
3472	-14.55	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
3473	-14.63	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
3474	-14.74	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
3475	-14.8	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
3476	-14.84	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
3477	-14.87	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
3478	-14.97	kd	CGS001-2710	GK	Glycerol kinases			
3479	-15.01	kd	CGS001-64376	IKZF5	IKAROS zinc fingers			
3480	-15.1	oe	ccsbBroad304_02092	SYNGR3	-			
3481	-15.16	kd	CGS001-10725	NFAT5	Nuclear factor of activated T-cells			
3482	-15.17	kd	CGS001-2869	GRK5	GRK1/3 subfamily			
3483	-15.2	kd	CGS001-222894	FERD3L	Basic helix-loop-helix proteins			
3484	-15.22	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3485	-15.23	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
3486	-15.23	kd	CGS001-200879	LIPH	-			
3487	-15.25	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
3488	-15.27	kd	CGS001-1879	EBF1	-			
3489	-15.27	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
3490	-15.29	kd	CGS001-9541	CIR1	-			
3491	-15.3	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
3492	-15.32	kd	CGS001-126823	KLHDC9	-			
3493	-15.33	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
3494	-15.37	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
3495	-15.41	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
3496	-15.44	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
3497	-15.44	kd	CGS001-3269	HRH1	Histamine receptors			
3498	-15.46	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
3499	-15.55	kd	CGS001-2645	GCK	Hexokinases			
3500	-15.58	kd	CGS001-6598	SMARCB1	-			
3501	-15.6	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
3502	-15.75	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3503	-15.76	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
3504	-15.76	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
3505	-15.82	kd	CGS001-353	APRT	-			
3506	-15.87	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3507	-15.88	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
3508	-15.9	kd	CGS001-25913	POT1	-			
3509	-15.92	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
3510	-15.93	kd	CGS001-4287	ATXN3	Ataxins			
3511	-16.09	kd	CGS001-91975	ZNF300	Zinc fingers, C2H2-type			
3512	-16.14	kd	CGS001-7249	TSC2	-			
3513	-16.18	oe	ccsbBroad304_00329	CLTA	-			
3514	-16.21	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
3515	-16.24	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
3516	-16.25	oe	ccsbBroad304_08802	ELAC2	-			
3517	-16.27	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
3518	-16.3	kd	CGS001-771	CA12	Carbonic anhydrases			
3519	-16.37	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
3520	-16.38	kd	CGS001-4255	MGMT	-			
3521	-16.4	kd	CGS001-10289	EIF1B	-			
3522	-16.42	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
3523	-16.44	kd	CGS001-64147	KIF9	Kinesins			
3524	-16.54	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
3525	-16.54	kd	CGS001-79139	DERL1	-			
3526	-16.55	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
3527	-16.58	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
3528	-16.58	oe	ccsbBroad304_08511	RFK	-			
3529	-16.58	kd	CGS001-662	BNIP1	-			
3530	-16.59	kd	CGS001-133522	PPARGC1B	RNA binding motif (RRM) containing			
3531	-16.6	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
3532	-16.6	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
3533	-16.63	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
3534	-16.63	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
3535	-16.63	kd	CGS001-2987	GUK1	-			
3536	-16.64	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
3537	-16.64	kd	CGS001-2242	FES	Fer family			
3538	-16.68	kd	CGS001-2147	F2	Endogenous ligands			
3539	-16.77	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3540	-16.79	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
3541	-16.8	kd	CGS001-1841	DTYMK	-			
3542	-16.81	kd	CGS001-8681	JMJD7-PLA2G4B	-			
3543	-16.85	kd	CGS001-10128	LRPPRC	-			
3544	-16.87	oe	ccsbBroad304_02136	COPS2	-			
3545	-16.91	oe	ccsbBroad304_08481	CEP55	-			
3546	-16.93	kd	CGS001-80314	EPC1	-			
3547	-17.01	kd	CGS001-10413	YAP1	Hippo Signaling			
3548	-17.02	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
3549	-17.08	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
3550	-17.08	kd	CGS001-3565	IL4	Interleukins and interleukin receptors			
3551	-17.08	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
3552	-17.1	cc		Aurora kinase inhibitor	-			
3553	-17.12	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
3554	-17.29	kd	CGS001-836	CASP3	Caspases			
3555	-17.34	kd	CGS001-79618	HMBOX1	Homeoboxes / HNF class			
3556	-17.36	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
3557	-17.4	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
3558	-17.43	kd	CGS001-1184	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
3559	-17.44	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
3560	-17.44	kd	CGS001-8226	HDHD1	-			
3561	-17.44	kd	CGS001-10955	SERINC3	-			
3562	-17.48	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
3563	-17.48	kd	CGS001-10891	PPARGC1A	RNA binding motif (RRM) containing			
3564	-17.5	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
3565	-17.5	kd	CGS001-10096	ACTR3	-			
3566	-17.51	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
3567	-17.52	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
3568	-17.54	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
3569	-17.54	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
3570	-17.57	kd	CGS001-10398	MYL9	EF-hand domain containing			
3571	-17.59	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
3572	-17.73	kd	CGS001-892	CCNC	-			
3573	-17.75	kd	CGS001-57665	RDH14	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3574	-17.83	kd	CGS001-7423	VEGFB	-			
3575	-17.84	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3576	-17.85	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
3577	-17.88	kd	CGS001-151126	ZNF385B	-			
3578	-17.89	kd	CGS001-6286	S100P	EF-hand domain containing			
3579	-17.91	oe	ccsbBroad304_00993	MDM4	-			
3580	-17.92	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
3581	-17.94	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
3582	-17.99	oe	ccsbBroad304_07277	RTCD1	-			
3583	-17.99	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
3584	-18.06	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
3585	-18.11	kd	CGS001-9655	SOCS5	SH2 domain containing			
3586	-18.11	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
3587	-18.12	kd	CGS001-57157	PHTF2	-			
3588	-18.17	kd	CGS001-166793	ZBTB49	BTB/POZ domain containing			
3589	-18.2	kd	CGS001-93349	SP140L	Zinc fingers, PHD-type			
3590	-18.21	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
3591	-18.21	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
3592	-18.22	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
3593	-18.27	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
3594	-18.27	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
3595	-18.29	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
3596	-18.31	kd	CGS001-2289	FKBP5	Tetratricopeptide (TTC) repeat domain containing			
3597	-18.33	cp	BRD-K47780086	penciclovir	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor
3598	-18.34	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
3599	-18.34	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
3600	-18.36	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
3601	-18.4	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
3602	-18.43	kd	CGS001-1869	E2F1	-			
3603	-18.45	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
3604	-18.46	oe	ccsbBroad304_04190	CCDC92	-			
3605	-18.48	cp	BRD-A16444946	acarbose	Glucosidase inhibitor		GAA, MGAM, AMY2A, SI	Glucosidase inhibitor
3606	-18.48	kd	CGS001-2056	EPO	Endogenous ligands			
3607	-18.5	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
3608	-18.51	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
3609	-18.52	kd	CGS001-2932	GSK3B	GSK subfamily			
3610	-18.55	kd	CGS001-822	CAPG	-			
3611	-18.56	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
3612	-18.58	kd	CGS001-55810	FOXJ2	Forkhead boxes			
3613	-18.59	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
3614	-18.6	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
3615	-18.61	kd	CGS001-5881	RAC3	Endogenous ligands			
3616	-18.64	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
3617	-18.64	kd	CGS001-4893	NRAS	RAS subfamily			
3618	-18.65	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
3619	-18.74	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
3620	-18.76	kd	CGS001-9111	NMI	-			
3621	-18.77	kd	CGS001-221895	JAZF1	Zinc fingers, C2H2-type			
3622	-18.82	kd	CGS001-7525	YES1	Src family			
3623	-18.85	kd	CGS001-4300	MLLT3	-			
3624	-18.87	kd	CGS001-22978	NT5C2	Adenosine turnover			
3625	-18.88	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
3626	-18.88	kd	CGS001-4143	MAT1A	-			
3627	-18.99	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
3628	-18.99	kd	CGS001-79885	HDAC11	Histone deacetylases			
3629	-19	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
3630	-19.02	oe	ccsbBroad304_04649	ADC	-			
3631	-19.02	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
3632	-19.02	kd	CGS001-4023	LPL	-			
3633	-19.05	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
3634	-19.12	kd	CGS001-6757	SSX2	-			
3635	-19.13	oe	ccsbBroad304_12106	PXK	Slob family			
3636	-19.16	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
3637	-19.2	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
3638	-19.22	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
3639	-19.24	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
3640	-19.24	kd	CGS001-637	BID	Endogenous ligands			
3641	-19.25	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
3642	-19.27	oe	ccsbBroad304_06916	SCP2	-			
3643	-19.28	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
3644	-19.31	kd	CGS001-54106	TLR9	Toll-like receptor family			
3645	-19.32	kd	CGS001-7078	TIMP3	-			
3646	-19.33	kd	CGS001-23314	SATB2	Homeoboxes / CUT class			
3647	-19.37	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
3648	-19.38	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
3649	-19.4	oe	ccsbBroad304_01035	MSH5	-			
3650	-19.4	oe	ccsbBroad304_07050	TFAP2A	-			
3651	-19.41	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
3652	-19.41	kd	CGS001-1606	DGKA	EF-hand domain containing			
3653	-19.42	kd	CGS001-7031	TFF1	-			
3654	-19.43	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
3655	-19.43	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
3656	-19.49	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
3657	-19.49	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
3658	-19.52	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
3659	-19.54	oe	ccsbBroad304_00102	RND3	-			
3660	-19.54	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
3661	-19.55	cc		Progesterone receptor agonist	-			
3662	-19.56	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
3663	-19.58	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
3664	-19.58	oe	ccsbBroad304_01351	PEX19	-			
3665	-19.61	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
3666	-19.61	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
3667	-19.64	kd	CGS001-64783	RBM15	RNA binding motif (RRM) containing			
3668	-19.64	kd	CGS001-1374	CPT1A	-			
3669	-19.75	kd	CGS001-158	ADSL	-			
3670	-19.76	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
3671	-19.76	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
3672	-19.77	cc		MCM family LOF	-			
3673	-19.78	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
3674	-19.82	kd	CGS001-2232	FDXR	-			
3675	-19.86	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
3676	-19.89	kd	CGS001-7353	UFD1L	-			
3677	-19.9	kd	CGS001-7159	TP53BP2	Ankyrin repeat domain containing			
3678	-19.94	kd	CGS001-7374	UNG	-			
3679	-19.95	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
3680	-19.96	kd	CGS001-3428	IFI16	-			
3681	-19.97	kd	CGS001-5134	PDCD2	Zinc fingers, MYND-type			
3682	-19.98	kd	CGS001-839	CASP6	Caspases			
3683	-20	oe	ccsbBroad304_00054	ALDOC	-			
3684	-20	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
3685	-20.04	kd	CGS001-9122	SLC16A4	SLC16 family of monocarboxylate transporters			
3686	-20.08	kd	CGS001-6652	SORD	-			
3687	-20.1	oe	ccsbBroad304_00282	CDKN1A	-			
3688	-20.12	kd	CGS001-6514	SLC2A2	Solute carriers			
3689	-20.13	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
3690	-20.14	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
3691	-20.14	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
3692	-20.16	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3693	-20.16	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
3694	-20.18	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3695	-20.18	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
3696	-20.2	kd	CGS001-22934	RPIA	-			
3697	-20.21	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
3698	-20.23	oe	ccsbBroad304_06290	GNA15	-			
3699	-20.24	kd	CGS001-3895	KTN1	-			
3700	-20.25	kd	CGS001-84878	ZBTB45	BTB/POZ domain containing			
3701	-20.28	oe	ccsbBroad304_08878	METTL4	-			
3702	-20.29	kd	CGS001-5111	PCNA	-			
3703	-20.29	kd	CGS001-9774	BCLAF1	-			
3704	-20.29	kd	CGS001-581	BAX	-			
3705	-20.3	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
3706	-20.32	kd	CGS001-51014	TMED7	-			
3707	-20.33	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
3708	-20.38	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
3709	-20.4	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
3710	-20.48	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
3711	-20.49	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
3712	-20.49	kd	CGS001-27297	CRCP	-			
3713	-20.5	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
3714	-20.5	kd	CGS001-4946	OAZ1	-			
3715	-20.52	kd	CGS001-5471	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
3716	-20.52	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
3717	-20.52	kd	CGS001-9687	GREB1	-			
3718	-20.61	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
3719	-20.63	oe	ccsbBroad304_01347	RAD1	-			
3720	-20.64	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
3721	-20.67	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
3722	-20.68	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
3723	-20.68	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
3724	-20.68	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
3725	-20.7	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
3726	-20.7	kd	CGS001-5160	PDHA1	-			
3727	-20.73	kd	CGS001-2550	GABBR1	GABA receptors			
3728	-20.74	kd	CGS001-167826	OLIG3	Basic helix-loop-helix proteins			
3729	-20.75	kd	CGS001-5427	POLE2	DNA polymerases			
3730	-20.76	kd	CGS001-5062	PAK2	PAKA subfamily			
3731	-20.79	kd	CGS001-10421	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3732	-20.82	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
3733	-20.83	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
3734	-20.84	cc		FLT3 inhibitor	-			
3735	-20.84	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
3736	-20.85	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
3737	-20.86	kd	CGS001-58477	SRPRB	-			
3738	-20.87	kd	CGS001-7083	TK1	-			
3739	-20.89	kd	CGS001-7471	WNT1	Endogenous ligands			
3740	-20.91	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
3741	-20.92	kd	CGS001-826	CAPNS1	EF-hand domain containing			
3742	-20.94	kd	CGS001-55907	CMAS	-			
3743	-20.96	kd	CGS001-3676	ITGA4	Integrins			
3744	-21	kd	CGS001-5934	RBL2	-			
3745	-21.03	oe	ccsbBroad304_06993	SRD5A1	-			
3746	-21.03	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
3747	-21.05	cp	BRD-K25310650	ormetoprim	Bacterial antifolate			Bacterial antifolate
3748	-21.06	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
3749	-21.07	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
3750	-21.07	kd	CGS001-3559	IL2RA	IL-2 receptor family			
3751	-21.18	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
3752	-21.2	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
3753	-21.24	kd	CGS001-7039	TGFA	-			
3754	-21.25	oe	ccsbBroad304_03173	TMED7	-			
3755	-21.29	kd	CGS001-5860	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
3756	-21.3	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
3757	-21.34	kd	CGS001-84971	ATG4D	-			
3758	-21.35	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
3759	-21.35	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
3760	-21.36	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
3761	-21.36	kd	CGS001-140612	ZFP28	Zinc fingers, C2H2-type			
3762	-21.37	kd	CGS001-140690	CTCFL	Zinc fingers, C2H2-type			
3763	-21.39	kd	CGS001-6722	SRF	-			
3764	-21.44	kd	CGS001-8408	ULK1	Unc-51-like kinase (ULK) family			
3765	-21.46	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
3766	-21.48	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
3767	-21.49	oe	ccsbBroad304_03544	FAIM	-			
3768	-21.54	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
3769	-21.56	kd	CGS001-3298	HSF2	-			
3770	-21.58	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
3771	-21.6	kd	CGS001-7360	UGP2	-			
3772	-21.66	oe	ccsbBroad304_06975	SMARCC2	-			
3773	-21.73	oe	ccsbBroad304_03444	PAF1	-			
3774	-21.74	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
3775	-21.78	oe	ccsbBroad304_00949	LRPAP1	-			
3776	-21.81	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
3777	-21.84	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
3778	-21.84	kd	CGS001-23355	VPS8	-			
3779	-21.91	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
3780	-21.92	kd	CGS001-1198	CLK3	CDC-like kinases			
3781	-21.94	cp	BRD-A15914070	4-hydroxy-2-nonenal	Cytotoxic lipid peroxidation product		IKBKB	Cytotoxic lipid peroxidation product
3782	-21.94	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
3783	-21.95	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
3784	-21.97	kd	CGS001-27148	STK36	Unc-51-like kinase (ULK) family			
3785	-21.98	kd	CGS001-210	ALAD	-			
3786	-22.02	kd	CGS001-4680	CEACAM6	CD molecules			
3787	-22.05	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3788	-22.05	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
3789	-22.07	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3790	-22.12	kd	CGS001-5092	PCBD1	-			
3791	-22.13	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
3792	-22.14	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
3793	-22.14	kd	CGS001-81894	SLC25A28	Miscellaneous SLC25 mitochondrial transporters			
3794	-22.15	kd	CGS001-965	CD58	CD molecules			
3795	-22.19	kd	CGS001-2593	GAMT	-			
3796	-22.24	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
3797	-22.26	kd	CGS001-6917	TCEA1	General transcription factors			
3798	-22.28	oe	ccsbBroad304_00077	APEX1	-			
3799	-22.29	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
3800	-22.3	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
3801	-22.31	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
3802	-22.33	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
3803	-22.34	oe	ccsbBroad304_01148	PCBD1	-			
3804	-22.37	kd	CGS001-90655	TGIF2LY	Homeoboxes / TALE class			
3805	-22.4	cc		V type ATPases LOF	-			
3806	-22.4	kd	CGS001-11162	NUDT6	Nudix motif containing			
3807	-22.41	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
3808	-22.44	kd	CGS001-5264	PHYH	-			
3809	-22.48	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
3810	-22.48	kd	CGS001-2254	FGF9	Endogenous ligands			
3811	-22.5	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
3812	-22.52	kd	CGS001-7484	WNT9B	Wingless-type MMTV integration sites			
3813	-22.53	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
3814	-22.55	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
3815	-22.6	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
3816	-22.63	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
3817	-22.64	kd	CGS001-149233	IL23R	IL-12 receptor family			
3818	-22.64	kd	CGS001-1999	ELF3	ETS Transcription Factors			
3819	-22.65	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
3820	-22.66	kd	CGS001-2002	ELK1	ETS Transcription Factors			
3821	-22.67	kd	CGS001-10247	HRSP12	-			
3822	-22.68	oe	ccsbBroad304_03177	FIS1	-			
3823	-22.68	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
3824	-22.68	kd	CGS001-9213	XPR1	-			
3825	-22.68	kd	CGS001-9252	RPS6KA5	MSK subfamily			
3826	-22.69	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
3827	-22.71	kd	CGS001-6195	RPS6KA1	RSK subfamily			
3828	-22.72	kd	CGS001-10923	SUB1	-			
3829	-22.73	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3830	-22.75	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
3831	-22.76	kd	CGS001-5357	PLS1	EF-hand domain containing			
3832	-22.77	kd	CGS001-4267	CD99	CD molecules			
3833	-22.78	kd	CGS001-151306	GPBAR1	Bile acid receptor			
3834	-22.8	kd	CGS001-10888	GPR83	GPCR / Class A : Orphans			
3835	-22.81	oe	ccsbBroad304_01184	PGK1	-			
3836	-22.82	oe	ccsbBroad304_07080	TM7SF2	-			
3837	-22.83	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
3838	-22.86	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
3839	-22.86	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
3840	-22.86	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
3841	-22.87	kd	CGS001-9412	MED21	-			
3842	-22.89	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
3843	-22.9	cc		Vitamin D receptor agonist	-			
3844	-22.92	kd	CGS001-4602	MYB	-			
3845	-22.95	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
3846	-22.96	cc		Androgen receptor modulator	-			
3847	-22.97	kd	CGS001-3682	ITGAE	Integrins			
3848	-22.98	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3849	-23	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
3850	-23.03	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3851	-23.05	kd	CGS001-10682	EBP	-			
3852	-23.06	oe	ccsbBroad304_03917	RBKS	-			
3853	-23.06	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
3854	-23.07	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
3855	-23.09	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3856	-23.11	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
3857	-23.12	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
3858	-23.13	kd	CGS001-5918	RARRES1	-			
3859	-23.13	kd	CGS001-392	ARHGAP1	Rho GTPase activating proteins			
3860	-23.14	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
3861	-23.16	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
3862	-23.2	kd	CGS001-6832	SUPV3L1	-			
3863	-23.26	kd	CGS001-578	BAK1	-			
3864	-23.27	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
3865	-23.27	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
3866	-23.28	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
3867	-23.29	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
3868	-23.34	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
3869	-23.37	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
3870	-23.4	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
3871	-23.43	kd	CGS001-10379	IRF9	-			
3872	-23.45	kd	CGS001-6605	SMARCE1	-			
3873	-23.46	cc		Thymidylate synthase inhibitor	-			
3874	-23.48	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
3875	-23.48	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
3876	-23.49	kd	CGS001-2263	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
3877	-23.49	kd	CGS001-80347	COASY	-			
3878	-23.5	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
3879	-23.51	oe	ccsbBroad304_04675	ATG4A	-			
3880	-23.51	kd	CGS001-3661	IRF3	-			
3881	-23.51	kd	CGS001-1718	DHCR24	-			
3882	-23.54	oe	ccsbBroad304_01974	RNASET2	-			
3883	-23.56	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
3884	-23.6	kd	CGS001-2864	FFAR1	Fatty acid receptors			
3885	-23.61	kd	CGS001-9375	TM9SF2	-			
3886	-23.62	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
3887	-23.62	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
3888	-23.63	kd	CGS001-3456	IFNB1	Interferons			
3889	-23.63	kd	CGS001-1349	COX7B	Mitochondrial respiratory chain complex			
3890	-23.65	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
3891	-23.68	kd	CGS001-3856	KRT8	Intermediate filaments type II, keratins (basic)			
3892	-23.69	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
3893	-23.69	kd	CGS001-114785	MBD6	-			
3894	-23.69	kd	CGS001-1820	ARID3A	-			
3895	-23.75	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
3896	-23.75	kd	CGS001-7247	TSN	-			
3897	-23.76	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3898	-23.77	kd	CGS001-55143	CDCA8	-			
3899	-23.78	kd	CGS001-5198	PFAS	-			
3900	-23.79	kd	CGS001-23512	SUZ12	Zinc fingers, C2H2-type			
3901	-23.79	kd	CGS001-4329	ALDH6A1	Aldehyde dehydrogenases			
3902	-23.8	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
3903	-23.81	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
3904	-23.81	kd	CGS001-6203	RPS9	S ribosomal proteins			
3905	-23.81	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
3906	-23.83	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
3907	-23.84	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
3908	-23.84	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
3909	-23.89	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
3910	-23.93	kd	CGS001-7533	YWHAH	-			
3911	-23.94	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
3912	-23.97	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
3913	-23.99	kd	CGS001-2348	FOLR1	-			
3914	-24	cp	BRD-A79314293	cephalosporanic-acid	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3915	-24.01	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
3916	-24.02	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
3917	-24.02	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
3918	-24.02	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
3919	-24.02	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
3920	-24.04	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
3921	-24.06	kd	CGS001-85480	TSLP	-			
3922	-24.11	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
3923	-24.11	oe	ccsbBroad304_01560	SNAPC1	-			
3924	-24.12	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
3925	-24.12	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
3926	-24.15	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
3927	-24.17	cp	BRD-K57930253	nitrazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, SCN1A	Benzodiazepine receptor agonist
3928	-24.17	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
3929	-24.19	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
3930	-24.21	cc		SRC inhibitor	-			
3931	-24.21	kd	CGS001-29946	SERTAD3	-			
3932	-24.22	cc		IGF-1 inhibitor	-			
3933	-24.22	cp	BRD-A94543220	bifonazole	Sterol demethylase inhibitor		CYP2B6	Sterol demethylase inhibitor
3934	-24.24	oe	ccsbBroad304_06648	CNOT3	-			
3935	-24.26	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
3936	-24.27	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
3937	-24.28	kd	CGS001-55634	ZNF673	-			
3938	-24.28	kd	CGS001-54490	UGT2B28	UDP glucuronosyltransferases			
3939	-24.32	kd	CGS001-3054	HCFC1	-			
3940	-24.32	kd	CGS001-1632	ECI1	-			
3941	-24.33	kd	CGS001-2639	GCDH	-			
3942	-24.37	kd	CGS001-1675	CFD	Complement system			
3943	-24.38	cp	BRD-K05350981	oligomycin-c	ATPase inhibitor		ATP5A1	ATPase inhibitor, ATP synthase inhibitor
3944	-24.41	kd	CGS001-22937	SCAP	WD repeat domain containing			
3945	-24.41	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
3946	-24.44	kd	CGS001-9612	NCOR2	-			
3947	-24.45	kd	CGS001-345	APOC3	Apolipoproteins			
3948	-24.46	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
3949	-24.46	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
3950	-24.46	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
3951	-24.46	kd	CGS001-883	CCBL1	Hydrogen sulphide synthesis			
3952	-24.47	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3953	-24.47	kd	CGS001-4172	MCM3	-			
3954	-24.48	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
3955	-24.48	kd	CGS001-399694	SHC4	SH2 domain containing			
3956	-24.51	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
3957	-24.55	kd	CGS001-23650	TRIM29	-			
3958	-24.55	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
3959	-24.55	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
3960	-24.58	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
3961	-24.61	kd	CGS001-91304	C19ORF6	-			
3962	-24.62	kd	CGS001-2919	CXCL1	Endogenous ligands			
3963	-24.63	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
3964	-24.65	kd	CGS001-7184	HSP90B1	Heat shock proteins / HSPC			
3965	-24.66	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
3966	-24.68	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
3967	-24.71	kd	CGS001-255738	PCSK9	Subtilisin			
3968	-24.73	oe	ccsbBroad304_00854	IL8	-			
3969	-24.74	kd	CGS001-344	APOC2	Apolipoproteins			
3970	-24.75	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3971	-24.76	oe	ccsbBroad304_12008	NLK	nmo subfamily			
3972	-24.76	kd	CGS001-2950	GSTP1	Glutathione S-transferases			
3973	-24.77	cc		X linked mental retardation group 2 LOF	-			
3974	-24.78	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
3975	-24.79	oe	ccsbBroad304_07045	TEAD4	-			
3976	-24.8	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
3977	-24.82	kd	CGS001-54998	AURKAIP1	-			
3978	-24.85	oe	ccsbBroad304_02604	B3GNT1	-			
3979	-24.86	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
3980	-24.87	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
3981	-24.88	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
3982	-24.91	kd	CGS001-5320	PLA2G2A	Hydrolases			
3983	-24.92	oe	ccsbBroad304_04655	TRIM9	-			
3984	-24.92	kd	CGS001-4090	SMAD5	SMADs			
3985	-24.96	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
3986	-24.96	kd	CGS001-7024	TFCP2	-			
3987	-24.96	oe	ccsbBroad304_02086	PDLIM1	-			
3988	-24.98	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
3989	-24.98	kd	CGS001-2160	F11	Chymotrypsin			
3990	-25	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
3991	-25.02	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
3992	-25.03	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
3993	-25.03	oe	ccsbBroad304_02840	PISD	Decarboxylases			
3994	-25.07	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
3995	-25.08	kd	CGS001-275	AMT	-			
3996	-25.09	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
3997	-25.09	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
3998	-25.11	kd	CGS001-5771	PTPN2	Protein tyrosine phosphatases			
3999	-25.12	kd	CGS001-7534	YWHAZ	-			
4000	-25.13	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
4001	-25.15	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
4002	-25.15	kd	CGS001-23210	JMJD6	-			
4003	-25.16	kd	CGS001-116832	RPL39L	L ribosomal proteins			
4004	-25.18	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
4005	-25.21	oe	ccsbBroad304_05894	BLVRA	-			
4006	-25.21	kd	CGS001-4151	MB	-			
4007	-25.21	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
4008	-25.22	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
4009	-25.24	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
4010	-25.25	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
4011	-25.26	cp	BRD-K65910366	KUC103904N	-666			-666
4012	-25.26	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
4013	-25.27	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
4014	-25.27	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4015	-25.28	kd	CGS001-8477	GPR65	GPCR / Class A : Orphans			
4016	-25.3	kd	CGS001-199704	ZNF585A	Zinc fingers, C2H2-type			
4017	-25.31	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
4018	-25.31	kd	CGS001-54749	EPDR1	-			
4019	-25.32	oe	ccsbBroad304_10487	BPHL	-			
4020	-25.34	cc		AHSP Pathway LOF	-			
4021	-25.34	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
4022	-25.35	kd	CGS001-56731	SLC2A4RG	-			
4023	-25.35	kd	CGS001-708	C1QBP	-			
4024	-25.37	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
4025	-25.38	kd	CGS001-9643	MORF4L2	-			
4026	-25.39	kd	CGS001-3171	FOXA3	Forkhead boxes			
4027	-25.41	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
4028	-25.42	oe	ccsbBroad304_06144	EFNB3	Ephrins			
4029	-25.43	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
4030	-25.46	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
4031	-25.47	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
4032	-25.47	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
4033	-25.47	kd	CGS001-2244	FGB	Endogenous ligands			
4034	-25.49	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
4035	-25.49	kd	CGS001-125950	RAVER1	RNA binding motif (RRM) containing			
4036	-25.51	kd	CGS001-23028	KDM1A	Histone demethylase			
4037	-25.54	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
4038	-25.55	kd	CGS001-7771	ZFP112	-			
4039	-25.55	kd	CGS001-3778	KCNMA1	Calcium-activated potassium channels			
4040	-25.58	cp	BRD-A70083328	secnidazole	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Microtubule inhibitor, Antiprotozoal
4041	-25.6	oe	ccsbBroad304_03122	RHOD	-			
4042	-25.6	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
4043	-25.61	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
4044	-25.62	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
4045	-25.63	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
4046	-25.66	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
4047	-25.68	kd	CGS001-9869	SETDB1	Histone methyltransferases (HMTs)			
4048	-25.69	cc		Serpin peptidase inhibitors LOF	-			
4049	-25.69	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
4050	-25.7	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
4051	-25.72	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
4052	-25.74	kd	CGS001-23076	RRP1B	-			
4053	-25.74	kd	CGS001-2882	GPX7	-			
4054	-25.75	kd	CGS001-50810	HDGFRP3	-			
4055	-25.76	kd	CGS001-8829	NRP1	CD molecules			
4056	-25.78	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
4057	-25.78	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4058	-25.78	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
4059	-25.79	oe	ccsbBroad304_06449	ILF3	-			
4060	-25.82	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
4061	-25.83	kd	CGS001-124641	OVCA2	-			
4062	-25.85	kd	CGS001-3601	IL15RA	IL-2 receptor family			
4063	-25.87	oe	ccsbBroad304_01379	RBBP6	-			
4064	-25.87	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
4065	-25.87	kd	CGS001-27097	TAF5L	WD repeat domain containing			
4066	-25.88	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
4067	-25.89	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
4068	-25.89	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
4069	-25.91	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
4070	-25.91	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4071	-25.91	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
4072	-25.97	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
4073	-25.98	kd	CGS001-1974	EIF4A2	DEAD-boxes			
4074	-26.01	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
4075	-26.02	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
4076	-26.04	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
4077	-26.05	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
4078	-26.09	oe	ccsbBroad304_08839	IFIH1	-			
4079	-26.09	kd	CGS001-3609	ILF3	-			
4080	-26.13	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
4081	-26.13	kd	CGS001-34	ACADM	-			
4082	-26.15	kd	CGS001-1528	CYB5A	Cytochrome b genes			
4083	-26.17	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
4084	-26.17	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4085	-26.17	kd	CGS001-1196	CLK2	CDC-like kinases			
4086	-26.18	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
4087	-26.18	oe	ccsbBroad304_02419	NDRG1	-			
4088	-26.18	oe	ccsbBroad304_14174	CDKAL1	-			
4089	-26.19	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
4090	-26.2	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
4091	-26.21	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
4092	-26.22	kd	CGS001-4869	NPM1	-			
4093	-26.24	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
4094	-26.26	kd	CGS001-699	BUB1	Bub family			
4095	-26.27	kd	CGS001-9474	ATG5	-			
4096	-26.3	oe	ccsbBroad304_02884	POT1	-			
4097	-26.3	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
4098	-26.33	oe	ccsbBroad304_00985	MCL1	-			
4099	-26.33	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
4100	-26.34	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
4101	-26.37	kd	CGS001-440387	CTRB2	-			
4102	-26.37	kd	CGS001-23242	COBL	-			
4103	-26.38	oe	ccsbBroad304_02551	CPSF4	-			
4104	-26.39	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
4105	-26.39	kd	CGS001-11257	TP53TG1	-			
4106	-26.4	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
4107	-26.41	kd	CGS001-23047	PDS5B	-			
4108	-26.41	kd	CGS001-3957	LGALS2	Lectins, galactoside-binding			
4109	-26.47	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
4110	-26.47	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
4111	-26.47	kd	CGS001-3664	IRF6	-			
4112	-26.48	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
4113	-26.5	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
4114	-26.51	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
4115	-26.52	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
4116	-26.53	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
4117	-26.54	kd	CGS001-29775	CARD10	-			
4118	-26.56	oe	ccsbBroad304_03497	TXNL4B	-			
4119	-26.56	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
4120	-26.58	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4121	-26.6	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
4122	-26.6	kd	CGS001-5689	PSMB1	Proteasome subunits			
4123	-26.6	kd	CGS001-164091	PAQR7	-			
4124	-26.61	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
4125	-26.61	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
4126	-26.62	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
4127	-26.67	kd	CGS001-1978	EIF4EBP1	-			
4128	-26.68	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
4129	-26.68	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
4130	-26.7	kd	CGS001-79143	MBOAT7	-			
4131	-26.72	kd	CGS001-2113	ETS1	ETS Transcription Factors			
4132	-26.75	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
4133	-26.75	kd	CGS001-57680	CHD8	-			
4134	-26.78	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
4135	-26.79	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
4136	-26.8	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
4137	-26.8	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4138	-26.82	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
4139	-26.83	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
4140	-26.86	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
4141	-26.86	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
4142	-26.89	kd	CGS001-1504	CTRB1	-			
4143	-26.9	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
4144	-26.9	cp	BRD-K63784565	BRD-K63784565	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
4145	-26.91	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
4146	-26.93	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
4147	-26.93	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
4148	-26.94	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
4149	-26.94	kd	CGS001-1595	CYP51A1	Cytochrome P450s			
4150	-26.95	cc		Homeobox Gene GOF	-			
4151	-26.97	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
4152	-26.98	kd	CGS001-4193	MDM2	-			
4153	-27	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
4154	-27	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
4155	-27	kd	CGS001-306	ANXA3	Annexins			
4156	-27.01	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
4157	-27.01	kd	CGS001-6857	SYT1	Synaptotagmins			
4158	-27.02	kd	CGS001-4616	GADD45B	-			
4159	-27.03	oe	ccsbBroad304_01661	TFCP2	-			
4160	-27.04	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
4161	-27.07	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
4162	-27.08	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
4163	-27.1	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
4164	-27.11	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
4165	-27.12	cc		FXR antagonist	-			
4166	-27.13	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
4167	-27.17	kd	CGS001-5981	RFC1	ATPases / AAA-type			
4168	-27.17	kd	CGS001-5696	PSMB8	Proteasome (prosome, macropain) subunits			
4169	-27.21	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
4170	-27.24	kd	CGS001-29105	C16ORF80	-			
4171	-27.25	oe	ccsbBroad304_00033	ADSS	-			
4172	-27.25	kd	CGS001-2280	FKBP1A	Cis-trans-isomerases			
4173	-27.3	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
4174	-27.31	kd	CGS001-53347	UBASH3A	-			
4175	-27.32	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
4176	-27.34	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
4177	-27.34	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
4178	-27.34	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
4179	-27.34	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4180	-27.36	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
4181	-27.38	kd	CGS001-598	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4182	-27.38	kd	CGS001-64241	ABCG8	ATP binding cassette transporters / subfamily G			
4183	-27.41	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
4184	-27.41	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4185	-27.42	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
4186	-27.42	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
4187	-27.43	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
4188	-27.43	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
4189	-27.44	kd	CGS001-22794	CASC3	-			
4190	-27.45	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
4191	-27.45	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
4192	-27.47	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
4193	-27.49	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
4194	-27.49	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
4195	-27.5	oe	ccsbBroad304_01327	PSPH	-			
4196	-27.52	kd	CGS001-3608	ILF2	-			
4197	-27.56	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
4198	-27.56	oe	ccsbBroad304_06836	RAD23B	-			
4199	-27.58	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4200	-27.59	kd	CGS001-4174	MCM5	-			
4201	-27.61	oe	ccsbBroad304_03237	LEF1	-			
4202	-27.62	kd	CGS001-8848	TSC22D1	-			
4203	-27.62	kd	CGS001-7090	TLE3	WD repeat domain containing			
4204	-27.64	kd	CGS001-11315	PARK7	Parkinson disease			
4205	-27.67	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
4206	-27.67	oe	ccsbBroad304_07374	PTPLA	-			
4207	-27.68	oe	ccsbBroad304_01841	BAG6	-			
4208	-27.68	kd	CGS001-4351	MPI	-			
4209	-27.69	kd	CGS001-5993	RFX5	-			
4210	-27.69	kd	CGS001-873	CBR1	Prostaglandin synthases			
4211	-27.7	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
4212	-27.7	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
4213	-27.71	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
4214	-27.71	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4215	-27.72	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
4216	-27.75	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
4217	-27.78	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
4218	-27.79	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
4219	-27.79	kd	CGS001-9326	ZNHIT3	Zinc fingers, HIT-type			
4220	-27.8	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
4221	-27.82	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
4222	-27.83	oe	ccsbBroad304_04786	CANT1	-			
4223	-27.84	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
4224	-27.84	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
4225	-27.85	oe	ccsbBroad304_06004	CKB	-			
4226	-27.85	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
4227	-27.88	cc		Tubulin inhibitor	-			
4228	-27.89	kd	CGS001-54386	TERF2IP	-			
4229	-27.9	kd	CGS001-6654	SOS1	Rho guanine nucleotide exchange factors			
4230	-27.9	kd	CGS001-6513	SLC2A1	Solute carriers			
4231	-27.94	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
4232	-27.95	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
4233	-28	kd	CGS001-5037	PEBP1	-			
4234	-28.02	kd	CGS001-1152	CKB	-			
4235	-28.03	kd	CGS001-1376	CPT2	-			
4236	-28.04	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
4237	-28.06	kd	CGS001-84290	CAPNS2	EF-hand domain containing			
4238	-28.11	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
4239	-28.16	cp	BRD-K82795137	loratadine	Histamine receptor antagonist		HRH1, CYP2C19, CYP3A5	Histamine receptor antagonist
4240	-28.18	kd	CGS001-6391	SDHC	Mitochondrial respiratory chain complex / Complex II			
4241	-28.18	kd	CGS001-9447	AIM2	-			
4242	-28.2	oe	ccsbBroad304_08045	NOX1	-			
4243	-28.23	kd	CGS001-130497	OSR1	Zinc fingers, C2H2-type			
4244	-28.24	oe	ccsbBroad304_02231	USP6NL	-			
4245	-28.25	kd	CGS001-3421	IDH3G	-			
4246	-28.26	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
4247	-28.26	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
4248	-28.26	kd	CGS001-201799	TMEM154	-			
4249	-28.29	kd	CGS001-10314	LANCL1	-			
4250	-28.31	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
4251	-28.31	kd	CGS001-338	APOB	Apolipoproteins			
4252	-28.35	oe	ccsbBroad304_00174	BRAF	RAF family			
4253	-28.36	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
4254	-28.36	kd	CGS001-2952	GSTT1	Glutathione S-transferases / Soluble			
4255	-28.38	kd	CGS001-3161	HMMR	CD molecules			
4256	-28.41	kd	CGS001-55818	KDM3A	Histone demethylases			
4257	-28.41	kd	CGS001-2729	GCLC	-			
4258	-28.43	kd	CGS001-91392	ZNF502	Zinc fingers, C2H2-type			
4259	-28.43	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
4260	-28.44	kd	CGS001-8650	NUMB	-			
4261	-28.46	cp	BRD-A39390670	rabeprazole	ATPase inhibitor		ATP4A, CYP2C19	ATPase inhibitor, Gastrin inhibitor
4262	-28.48	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
4263	-28.48	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
4264	-28.49	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
4265	-28.51	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
4266	-28.51	oe	ccsbBroad304_05931	CAPG	-			
4267	-28.52	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
4268	-28.52	kd	CGS001-8714	ABCC3	ATP binding cassette transporters / subfamily C			
4269	-28.56	oe	ccsbBroad304_00789	HSBP1	-			
4270	-28.61	kd	CGS001-6829	SUPT5H	-			
4271	-28.62	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
4272	-28.62	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4273	-28.63	kd	CGS001-688	KLF5	Kruppel-like transcription factors			
4274	-28.67	oe	ccsbBroad304_05821	ANXA1	Annexins			
4275	-28.69	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4276	-28.7	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
4277	-28.7	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
4278	-28.76	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
4279	-28.76	kd	CGS001-9695	EDEM1	-			
4280	-28.8	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
4281	-28.8	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4282	-28.84	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
4283	-28.86	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
4284	-28.89	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
4285	-28.9	oe	ccsbBroad304_00933	LDHB	-			
4286	-28.91	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
4287	-28.92	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
4288	-28.93	oe	ccsbBroad304_10230	STK19	G11 family			
4289	-28.93	oe	ccsbBroad304_07724	KDELR2	-			
4290	-29	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
4291	-29	kd	CGS001-6926	TBX3	T-boxes			
4292	-29.01	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
4293	-29.02	kd	CGS001-5080	PAX6	Paired boxes			
4294	-29.05	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
4295	-29.05	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
4296	-29.06	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
4297	-29.06	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
4298	-29.09	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
4299	-29.09	kd	CGS001-57149	LYRM1	LYR motif containing			
4300	-29.16	kd	CGS001-4860	PNP	-			
4301	-29.18	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
4302	-29.18	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
4303	-29.21	oe	ccsbBroad304_01394	RFX4	-			
4304	-29.23	kd	CGS001-2778	GNAS	-			
4305	-29.24	oe	ccsbBroad304_06765	PRCC	-			
4306	-29.24	cp	BRD-K18523449	mestanolone	Androgenic steroid			Androgenic steroid
4307	-29.26	oe	ccsbBroad304_02822	ARFIP2	-			
4308	-29.27	oe	ccsbBroad304_02370	HRSP12	-			
4309	-29.28	kd	CGS001-23461	ABCA5	ATP binding cassette transporters / subfamily A			
4310	-29.29	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
4311	-29.3	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
4312	-29.31	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
4313	-29.33	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
4314	-29.34	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
4315	-29.34	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
4316	-29.35	oe	ccsbBroad304_02109	XPR1	-			
4317	-29.35	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
4318	-29.37	oe	ccsbBroad304_01061	NAB2	-			
4319	-29.43	oe	ccsbBroad304_07569	TRIB1	Trbl family			
4320	-29.44	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
4321	-29.45	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4322	-29.46	oe	ccsbBroad304_07820	SNW1	-			
4323	-29.47	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
4324	-29.47	kd	CGS001-26520	TIMM9	-			
4325	-29.48	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
4326	-29.48	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
4327	-29.49	oe	ccsbBroad304_05152	SSBP4	-			
4328	-29.51	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
4329	-29.52	kd	CGS001-84647	PLA2G12B	-			
4330	-29.54	oe	ccsbBroad304_07053	TFPI	-			
4331	-29.55	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
4332	-29.55	kd	CGS001-527	ATP6V0C	ATPases / V-type			
4333	-29.56	kd	CGS001-9374	PPT2	-			
4334	-29.57	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
4335	-29.6	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
4336	-29.63	kd	CGS001-1756	DMD	-			
4337	-29.66	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
4338	-29.67	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
4339	-29.68	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
4340	-29.68	kd	CGS001-7477	WNT7B	Endogenous ligands			
4341	-29.71	kd	CGS001-10227	MFSD10	-			
4342	-29.76	kd	CGS001-9322	TRIP10	-			
4343	-29.82	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
4344	-29.83	oe	ccsbBroad304_04544	RCCD1	-			
4345	-29.83	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
4346	-29.86	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
4347	-29.86	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
4348	-29.86	kd	CGS001-10845	CLPX	ATPases / AAA-type			
4349	-29.9	cp	BRD-A84134924	pancuronium	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRNA1, CHRNA2	Acetylcholine receptor antagonist
4350	-29.91	oe	ccsbBroad304_03097	CNOT7	-			
4351	-29.92	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
4352	-29.94	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
4353	-29.95	oe	ccsbBroad304_08662	MCCC1	-			
4354	-29.96	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4355	-29.97	oe	ccsbBroad304_06435	RBPJ	-			
4356	-29.97	oe	ccsbBroad304_06828	PYCR1	-			
4357	-29.98	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
4358	-29.98	kd	CGS001-29079	MED4	-			
4359	-29.99	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
4360	-29.99	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
4361	-30	kd	CGS001-29763	PACSIN3	-			
4362	-30	kd	CGS001-9404	LPXN	-			
4363	-30.01	kd	CGS001-678	ZFP36L2	RING-type (C3HC4) zinc fingers			
4364	-30.01	kd	CGS001-9710	KIAA0355	-			
4365	-30.02	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
4366	-30.05	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
4367	-30.07	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
4368	-30.07	kd	CGS001-2673	GFPT1	-			
4369	-30.08	kd	CGS001-2078	ERG	ETS Transcription Factors			
4370	-30.11	kd	CGS001-10318	TNIP1	-			
4371	-30.11	kd	CGS001-5916	RARG	Retinoic acid receptors			
4372	-30.12	kd	CGS001-113451	ADC	-			
4373	-30.13	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
4374	-30.15	cc		Akt Signaling LOF	-			
4375	-30.17	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
4376	-30.18	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4377	-30.18	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
4378	-30.18	kd	CGS001-2015	EMR1	Adhesion Class GPCRs			
4379	-30.2	oe	ccsbBroad304_03850	TRIB3	Trbl family			
4380	-30.2	kd	CGS001-6723	SRM	-			
4381	-30.22	kd	CGS001-5447	POR	-			
4382	-30.24	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
4383	-30.25	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
4384	-30.28	oe	ccsbBroad304_06670	OGG1	-			
4385	-30.29	kd	CGS001-1070	CETN3	EF-hand domain containing			
4386	-30.3	kd	CGS001-2909	ARHGAP35	Rho GTPase activating proteins			
4387	-30.32	kd	CGS001-11180	WDR6	WD repeat domain containing			
4388	-30.32	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
4389	-30.35	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
4390	-30.37	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
4391	-30.37	kd	CGS001-10284	SAP18	-			
4392	-30.39	oe	ccsbBroad304_00162	BIK	-			
4393	-30.41	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
4394	-30.41	kd	CGS001-5018	OXA1L	-			
4395	-30.46	kd	CGS001-3638	INSIG1	-			
4396	-30.48	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4397	-30.5	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
4398	-30.6	oe	ccsbBroad304_00359	CPT1A	-			
4399	-30.6	kd	CGS001-5361	PLXNA1	Plexins			
4400	-30.61	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
4401	-30.62	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
4402	-30.64	kd	CGS001-11267	SNF8	-			
4403	-30.65	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
4404	-30.65	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
4405	-30.66	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
4406	-30.66	kd	CGS001-648	BMI1	Polycomb group ring fingers			
4407	-30.67	kd	CGS001-10691	GMEB1	-			
4408	-30.69	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
4409	-30.69	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
4410	-30.7	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
4411	-30.73	kd	CGS001-2167	FABP4	Fatty acid binding protein family			
4412	-30.8	oe	ccsbBroad304_03618	OSGEP	-			
4413	-30.8	kd	CGS001-663	BNIP2	-			
4414	-30.82	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
4415	-30.82	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
4416	-30.84	kd	CGS001-10973	ASCC3	-			
4417	-30.84	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
4418	-30.87	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
4419	-30.87	kd	CGS001-10465	PPIH	-			
4420	-30.89	kd	CGS001-8874	ARHGEF7	Rho guanine nucleotide exchange factors			
4421	-30.91	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
4422	-30.92	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4423	-30.92	kd	CGS001-94103	ORMDL3	-			
4424	-30.92	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
4425	-30.94	kd	CGS001-1327	COX4I1	Mitochondrial respiratory chain complex			
4426	-30.98	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
4427	-30.99	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
4428	-31	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
4429	-31.01	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
4430	-31.02	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
4431	-31.02	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
4432	-31.04	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
4433	-31.05	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
4434	-31.06	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
4435	-31.06	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4436	-31.08	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
4437	-31.09	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
4438	-31.09	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
4439	-31.11	kd	CGS001-6272	SORT1	-			
4440	-31.12	oe	ccsbBroad304_01624	SUPV3L1	-			
4441	-31.13	oe	ccsbBroad304_03182	GLOD4	-			
4442	-31.15	kd	CGS001-10652	YKT6	-			
4443	-31.15	kd	CGS001-10001	MED6	-			
4444	-31.17	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
4445	-31.18	oe	ccsbBroad304_03129	ERO1L	-			
4446	-31.22	oe	ccsbBroad304_03113	DSE	-			
4447	-31.23	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
4448	-31.23	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
4449	-31.23	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
4450	-31.23	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
4451	-31.24	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
4452	-31.25	kd	CGS001-1488	CTBP2	-			
4453	-31.26	kd	CGS001-5294	PIK3CG	Phosphatidylinositol kinases			
4454	-31.27	kd	CGS001-9787	DLGAP5	-			
4455	-31.27	kd	CGS001-161	AP2A2	-			
4456	-31.29	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
4457	-31.29	kd	CGS001-4297	MLL	-			
4458	-31.3	kd	CGS001-5306	PITPNA	-			
4459	-31.38	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
4460	-31.38	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4461	-31.38	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4462	-31.38	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
4463	-31.39	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
4464	-31.42	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
4465	-31.42	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
4466	-31.44	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
4467	-31.46	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
4468	-31.47	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
4469	-31.47	kd	CGS001-1022	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
4470	-31.48	kd	CGS001-9589	WTAP	-			
4471	-31.5	kd	CGS001-2538	G6PC	-			
4472	-31.51	oe	ccsbBroad304_01205	PIN1	-			
4473	-31.52	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
4474	-31.53	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
4475	-31.54	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
4476	-31.58	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
4477	-31.61	kd	CGS001-1981	EIF4G1	Parkinson disease			
4478	-31.64	oe	ccsbBroad304_02834	GABARAPL1	-			
4479	-31.64	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
4480	-31.66	oe	ccsbBroad304_00620	GCDH	-			
4481	-31.69	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
4482	-31.7	oe	ccsbBroad304_06188	F10	Chymotrypsin			
4483	-31.71	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
4484	-31.73	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
4485	-31.73	kd	CGS001-9061	PAPSS1	-			
4486	-31.74	oe	ccsbBroad304_02432	IFI30	-			
4487	-31.79	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
4488	-31.81	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
4489	-31.81	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
4490	-31.82	cc		Bromodomain Inhibitor	-			
4491	-31.82	kd	CGS001-93594	WDR67	-			
4492	-31.84	kd	CGS001-5184	PEPD	Methionyl aminopeptidase			
4493	-31.87	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
4494	-31.89	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
4495	-31.9	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
4496	-31.9	kd	CGS001-1977	EIF4E	Translation Initiation Factor 4E			
4497	-31.91	kd	CGS001-81620	CDT1	-			
4498	-31.92	kd	CGS001-8220	DGCR14	-			
4499	-31.93	kd	CGS001-9467	SH3BP5	-			
4500	-32	kd	CGS001-6119	RPA3	-			
4501	-32.04	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
4502	-32.08	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
4503	-32.1	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
4504	-32.11	kd	CGS001-3978	LIG1	-			
4505	-32.12	kd	CGS001-26227	PHGDH	-			
4506	-32.13	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
4507	-32.15	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
4508	-32.18	kd	CGS001-475	ATOX1	-			
4509	-32.22	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
4510	-32.23	cc		HOXL subclass homeoboxes LOF	-			
4511	-32.24	kd	CGS001-10672	GNA13	-			
4512	-32.25	kd	CGS001-9815	GIT2	Ankyrin repeat domain containing			
4513	-32.27	kd	CGS001-6714	SRC	Src family			
4514	-32.28	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
4515	-32.29	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
4516	-32.3	kd	CGS001-474354	LRRC18	-			
4517	-32.31	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
4518	-32.32	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
4519	-32.33	cc		RAF inhibitor	-			
4520	-32.33	kd	CGS001-9184	BUB3	WD repeat domain containing			
4521	-32.34	oe	ccsbBroad304_03112	NENF	-			
4522	-32.4	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
4523	-32.4	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
4524	-32.42	oe	ccsbBroad304_00817	IDH2	-			
4525	-32.42	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
4526	-32.45	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4527	-32.45	oe	ccsbBroad304_06292	GNAI2	-			
4528	-32.46	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
4529	-32.49	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
4530	-32.53	cp	BRD-K10065684	dantron	Laxative			Laxative
4531	-32.54	kd	CGS001-80306	MED28	-			
4532	-32.55	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
4533	-32.55	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
4534	-32.56	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
4535	-32.56	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
4536	-32.56	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
4537	-32.56	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
4538	-32.58	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
4539	-32.59	oe	ccsbBroad304_03812	PBXIP1	-			
4540	-32.59	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
4541	-32.6	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
4542	-32.61	oe	ccsbBroad304_06665	OAT	-			
4543	-32.61	cp	BRD-K44779798	miglitol	Glucosidase inhibitor		GAA, MGAM, GANAB, GANC, SLC5A4	Glucosidase inhibitor
4544	-32.63	kd	CGS001-3033	HADH	-			
4545	-32.65	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
4546	-32.65	kd	CGS001-5686	PSMA5	Proteasome subunits			
4547	-32.67	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
4548	-32.67	oe	ccsbBroad304_03728	DIABLO	-			
4549	-32.69	oe	ccsbBroad304_00941	LIG3	-			
4550	-32.72	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
4551	-32.73	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
4552	-32.74	oe	ccsbBroad304_06820	PTS	-			
4553	-32.74	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
4554	-32.79	kd	CGS001-10253	SPRY2	-			
4555	-32.82	kd	CGS001-7840	ALMS1	-			
4556	-32.83	kd	CGS001-670	BPHL	-			
4557	-32.88	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
4558	-32.88	kd	CGS001-3934	LCN2	Lipocalins			
4559	-32.9	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
4560	-32.9	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
4561	-32.91	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
4562	-32.94	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
4563	-32.96	kd	CGS001-6988	TCTA	-			
4564	-32.96	oe	ccsbBroad304_01163	PDHA1	-			
4565	-32.97	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
4566	-32.99	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
4567	-32.99	kd	CGS001-4097	MAFG	-			
4568	-32.99	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
4569	-32.99	kd	CGS001-159	ADSS	-			
4570	-33	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4571	-33.01	kd	CGS001-1855	DVL1	Dishevelled homologs			
4572	-33.08	cp	BRD-K59753975	vindesine	Tubulin inhibitor		TUBB, TUBB1	Tubulin inhibitor
4573	-33.12	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
4574	-33.15	oe	ccsbBroad304_00003	ABAT	GABA turnover			
4575	-33.17	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
4576	-33.17	cp	BRD-K39983086	loteprednol	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Phospholipase inhibitor
4577	-33.22	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
4578	-33.24	kd	CGS001-5515	PPP2CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4579	-33.26	cc		Topoisomerase inhibitor	-			
4580	-33.27	kd	CGS001-8900	CCNA1	-			
4581	-33.27	kd	CGS001-383	ARG1	Arginase			
4582	-33.29	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
4583	-33.29	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
4584	-33.3	oe	ccsbBroad304_06134	ECH1	-			
4585	-33.31	kd	CGS001-2203	FBP1	-			
4586	-33.34	oe	ccsbBroad304_02502	GNA13	-			
4587	-33.34	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4588	-33.36	kd	CGS001-8870	IER3	-			
4589	-33.39	kd	CGS001-8945	BTRC	F-boxes / WD-40 domains			
4590	-33.4	kd	CGS001-10298	PAK4	PAKB subfamily			
4591	-33.41	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
4592	-33.41	kd	CGS001-5170	PDPK1	PDK1 family			
4593	-33.49	kd	CGS001-3459	IFNGR1	Interferon receptor family			
4594	-33.5	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
4595	-33.5	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
4596	-33.51	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4597	-33.52	oe	ccsbBroad304_02249	KIAA0494	-			
4598	-33.56	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
4599	-33.57	kd	CGS001-8896	BUD31	-			
4600	-33.57	kd	CGS001-166	AES	-			
4601	-33.63	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
4602	-33.66	kd	CGS001-8543	LMO4	-			
4603	-33.67	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
4604	-33.68	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
4605	-33.7	kd	CGS001-7862	BRPF1	Non-enzymatic BRD containing proteins			
4606	-33.72	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
4607	-33.73	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
4608	-33.78	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
4609	-33.79	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
4610	-33.8	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
4611	-33.8	oe	ccsbBroad304_06663	OAS1	-			
4612	-33.81	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
4613	-33.82	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
4614	-33.85	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
4615	-33.86	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
4616	-33.86	oe	ccsbBroad304_00313	TBCB	-			
4617	-33.88	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
4618	-33.89	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4619	-33.9	kd	CGS001-3485	IGFBP2	insulin-like growth factor (IGF) binding proteins			
4620	-33.91	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
4621	-33.91	kd	CGS001-10939	AFG3L2	ATPases / AAA-type			
4622	-33.92	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
4623	-33.97	kd	CGS001-50604	IL20	Interleukins and interleukin receptors			
4624	-34.04	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
4625	-34.04	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
4626	-34.1	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
4627	-34.12	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
4628	-34.12	oe	ccsbBroad304_01101	NME1	-			
4629	-34.16	oe	ccsbBroad304_01673	TIMP3	-			
4630	-34.17	oe	ccsbBroad304_01150	PCCB	Carboxylases			
4631	-34.18	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
4632	-34.19	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
4633	-34.24	kd	CGS001-6275	S100A4	EF-hand domain containing			
4634	-34.26	oe	ccsbBroad304_00179	BTG1	-			
4635	-34.26	kd	CGS001-162699	TCEB3C	-			
4636	-34.28	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
4637	-34.28	oe	ccsbBroad304_00986	MCM2	-			
4638	-34.28	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
4639	-34.29	cc		JAK inhibitor	-			
4640	-34.29	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
4641	-34.29	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
4642	-34.33	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
4643	-34.33	kd	CGS001-132	ADK	Adenosine turnover			
4644	-34.34	oe	ccsbBroad304_05902	BNIP3	-			
4645	-34.35	oe	ccsbBroad304_01880	LAGE3	-			
4646	-34.38	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
4647	-34.39	kd	CGS001-5063	PAK3	PAKA subfamily			
4648	-34.42	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
4649	-34.44	oe	ccsbBroad304_00001	NAT1	-			
4650	-34.46	oe	ccsbBroad304_02857	BAMBI	-			
4651	-34.46	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
4652	-34.46	kd	CGS001-5962	RDX	-			
4653	-34.49	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
4654	-34.5	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
4655	-34.5	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
4656	-34.51	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
4657	-34.51	kd	CGS001-51548	SIRT6	Histone deacetylases (HDACs)			
4658	-34.53	kd	CGS001-2805	GOT1	-			
4659	-34.55	cc		Mediator complex LOF	-			
4660	-34.55	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
4661	-34.58	kd	CGS001-23014	FBXO21	F-boxes / other			
4662	-34.59	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
4663	-34.59	kd	CGS001-22938	SNW1	-			
4664	-34.62	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
4665	-34.64	oe	ccsbBroad304_02772	ICMT	-			
4666	-34.64	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
4667	-34.68	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
4668	-34.68	kd	CGS001-8649	LAMTOR3	-			
4669	-34.69	cc		Gamma secretase inhibitor	-			
4670	-34.69	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4671	-34.69	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
4672	-34.69	kd	CGS001-6184	RPN1	-			
4673	-34.74	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
4674	-34.76	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
4675	-34.76	oe	ccsbBroad304_02506	EBP	-			
4676	-34.77	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
4677	-34.77	kd	CGS001-262	AMD1	Decarboxylases			
4678	-34.78	kd	CGS001-10295	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
4679	-34.81	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
4680	-34.83	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
4681	-34.84	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
4682	-34.85	kd	CGS001-8741	TNFSF13	CD molecules			
4683	-34.86	kd	CGS001-57504	MTA3	GATA zinc finger domain containing			
4684	-34.88	oe	ccsbBroad304_08775	SQRDL	-			
4685	-34.89	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
4686	-34.9	cc		General transcription factors group 2 LOF	-			
4687	-34.9	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
4688	-34.94	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
4689	-34.94	kd	CGS001-84669	USP32	EF-hand domain containing			
4690	-34.95	oe	ccsbBroad304_02205	WTAP	-			
4691	-34.95	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
4692	-34.96	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
4693	-34.97	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
4694	-34.97	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
4695	-34.97	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4696	-34.97	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
4697	-34.99	oe	ccsbBroad304_07888	CBX6	-			
4698	-35.01	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
4699	-35.03	kd	CGS001-6675	UAP1	-			
4700	-35.05	kd	CGS001-55781	RIOK2	RIO2 subfamily			
4701	-35.07	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
4702	-35.07	kd	CGS001-2956	MSH6	-			
4703	-35.07	kd	CGS001-2745	GLRX	-			
4704	-35.08	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
4705	-35.09	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
4706	-35.09	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
4707	-35.18	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
4708	-35.19	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4709	-35.23	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
4710	-35.23	kd	CGS001-4074	M6PR	-			
4711	-35.24	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
4712	-35.25	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
4713	-35.25	kd	CGS001-84515	MCM8	-			
4714	-35.31	kd	CGS001-154	ADRB2	GPCR / Class A : Adrenoceptors : beta			
4715	-35.32	kd	CGS001-4087	SMAD2	SMADs			
4716	-35.32	kd	CGS001-23338	PHF15	-			
4717	-35.32	kd	CGS001-54623	PAF1	-			
4718	-35.36	oe	ccsbBroad304_00881	IRF5	-			
4719	-35.36	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
4720	-35.37	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
4721	-35.39	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
4722	-35.41	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
4723	-35.43	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
4724	-35.45	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
4725	-35.45	kd	CGS001-83637	ZMIZ2	Zinc fingers, MIZ-type			
4726	-35.46	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4727	-35.46	kd	CGS001-3265	HRAS	RAS subfamily			
4728	-35.48	kd	CGS001-4790	NFKB1	NFkappaB transcription factor family			
4729	-35.51	oe	ccsbBroad304_00836	IGF2	-			
4730	-35.52	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
4731	-35.55	kd	CGS001-51097	SCCPDH	-			
4732	-35.57	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
4733	-35.58	kd	CGS001-83593	RASSF5	-			
4734	-35.58	kd	CGS001-50846	DHH	-			
4735	-35.6	kd	CGS001-8027	STAM	-			
4736	-35.6	oe	ccsbBroad304_02592	KIF2C	Kinesins			
4737	-35.62	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
4738	-35.63	kd	CGS001-6812	STXBP1	-			
4739	-35.64	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
4740	-35.64	kd	CGS001-4976	OPA1	-			
4741	-35.67	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
4742	-35.68	kd	CGS001-1659	DHX8	DEAH-boxes			
4743	-35.7	kd	CGS001-8667	EIF3H	-			
4744	-35.72	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
4745	-35.72	oe	ccsbBroad304_00552	FEN1	-			
4746	-35.75	kd	CGS001-10857	PGRMC1	-			
4747	-35.8	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
4748	-35.83	oe	ccsbBroad304_02815	SSBP2	-			
4749	-35.83	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
4750	-35.85	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
4751	-35.85	kd	CGS001-51031	GLOD4	-			
4752	-35.86	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
4753	-35.87	oe	ccsbBroad304_07018	SUPT5H	-			
4754	-35.88	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
4755	-35.89	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
4756	-35.89	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
4757	-35.9	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
4758	-35.9	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
4759	-35.91	kd	CGS001-2769	GNA15	-			
4760	-35.92	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
4761	-35.94	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
4762	-35.95	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
4763	-35.96	cp	BRD-A24381660	zeranol	Estrogen receptor agonist			Estrogen receptor agonist
4764	-36	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
4765	-36.01	kd	CGS001-4683	NBN	-			
4766	-36.02	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
4767	-36.02	kd	CGS001-5621	PRNP	CD molecules			
4768	-36.06	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4769	-36.11	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
4770	-36.14	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
4771	-36.14	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4772	-36.14	kd	CGS001-7323	UBE2D3	Ubiquitin-conjugating enzymes E2			
4773	-36.16	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
4774	-36.16	kd	CGS001-51172	NAGPA	-			
4775	-36.17	kd	CGS001-10113	PREB	WD repeat domain containing			
4776	-36.19	kd	CGS001-2787	GNG5	-			
4777	-36.2	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
4778	-36.21	oe	ccsbBroad304_03037	TMEM97	-			
4779	-36.21	kd	CGS001-1975	EIF4B	RNA binding motif (RRM) containing			
4780	-36.26	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
4781	-36.27	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
4782	-36.27	kd	CGS001-6741	SSB	La ribonucleoprotein domain containing			
4783	-36.28	oe	ccsbBroad304_06225	FTH1	-			
4784	-36.28	oe	ccsbBroad304_13891	LCK	Src family			
4785	-36.29	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4786	-36.33	oe	ccsbBroad304_00147	BAG1	-			
4787	-36.35	oe	ccsbBroad304_02402	TMEM5	-			
4788	-36.35	oe	ccsbBroad304_01654	TCTA	-			
4789	-36.37	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
4790	-36.45	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
4791	-36.46	oe	ccsbBroad304_07923	LSM5	-			
4792	-36.46	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
4793	-36.54	oe	ccsbBroad304_00661	GNGT2	-			
4794	-36.61	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
4795	-36.61	kd	CGS001-1147	CHUK	IKK family			
4796	-36.62	cc		GATA Zinc finger domain containing LOF	-			
4797	-36.65	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
4798	-36.69	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
4799	-36.72	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
4800	-36.74	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
4801	-36.74	kd	CGS001-10494	STK25	YSK subfamily			
4802	-36.74	kd	CGS001-121549	ASCL4	Basic helix-loop-helix proteins			
4803	-36.78	oe	ccsbBroad304_00614	GAMT	-			
4804	-36.79	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4805	-36.85	oe	ccsbBroad304_06255	LRRC32	-			
4806	-36.86	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4807	-36.87	kd	CGS001-2475	MTOR	FRAP subfamily			
4808	-36.88	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
4809	-36.93	kd	CGS001-54899	PXK	Slob family			
4810	-36.95	cc		Glucocorticoid receptor agonist	-			
4811	-36.96	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
4812	-36.97	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
4813	-36.98	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
4814	-37	kd	CGS001-5236	PGM1	-			
4815	-37.03	kd	CGS001-9276	COPB2	WD repeat domain containing			
4816	-37.05	kd	CGS001-7052	TGM2	Transglutaminases			
4817	-37.05	kd	CGS001-9519	TBPL1	-			
4818	-37.06	kd	CGS001-2355	FOSL2	basic leucine zipper proteins			
4819	-37.07	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
4820	-37.09	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4821	-37.1	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
4822	-37.12	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
4823	-37.14	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
4824	-37.2	oe	ccsbBroad304_01948	GAS7	-			
4825	-37.2	kd	CGS001-57804	POLD4	DNA polymerases			
4826	-37.25	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
4827	-37.28	kd	CGS001-6621	SNAPC4	-			
4828	-37.32	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
4829	-37.32	kd	CGS001-602	BCL3	Ankyrin repeat domain containing			
4830	-37.39	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
4831	-37.44	oe	ccsbBroad304_01659	TERF1	-			
4832	-37.47	oe	ccsbBroad304_07101	TSC2	-			
4833	-37.53	oe	ccsbBroad304_01960	CASK	CASK family			
4834	-37.56	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
4835	-37.58	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
4836	-37.58	cp	BRD-K28849549	mesalazine	Cyclooxygenase inhibitor		PTGS1, PPARG, PTGS2, ALOX5, CHUK, CTNNB1, IKBKB, MPO, NAT1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor, Prostanoid receptor antagonist
4837	-37.59	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
4838	-37.61	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
4839	-37.66	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
4840	-37.68	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
4841	-37.7	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
4842	-37.72	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
4843	-37.76	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
4844	-37.77	oe	ccsbBroad304_02837	BHMT2	-			
4845	-37.78	kd	CGS001-3925	STMN1	-			
4846	-37.82	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
4847	-37.82	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
4848	-37.83	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
4849	-37.83	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
4850	-37.84	oe	ccsbBroad304_03961	SMURF2	-			
4851	-37.86	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
4852	-37.92	kd	CGS001-57406	ABHD6	Abhydrolase domain containing			
4853	-37.93	kd	CGS001-26149	ZNF658	Zinc fingers, C2H2-type			
4854	-37.94	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
4855	-37.95	oe	ccsbBroad304_07506	UBAP2L	-			
4856	-37.95	oe	ccsbBroad304_07890	CBX7	-			
4857	-37.96	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
4858	-37.96	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
4859	-37.99	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
4860	-38.03	oe	ccsbBroad304_02605	PAPD7	-			
4861	-38.04	kd	CGS001-163486	DENND1B	DENN/MADD domain containing			
4862	-38.07	kd	CGS001-5315	PKM2	-			
4863	-38.1	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
4864	-38.1	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
4865	-38.11	oe	ccsbBroad304_02425	CDIPT	-			
4866	-38.11	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
4867	-38.11	kd	CGS001-54811	ZNF562	Zinc fingers, C2H2-type			
4868	-38.16	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
4869	-38.16	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
4870	-38.16	kd	CGS001-54851	ANKRD49	Ankyrin repeat domain containing			
4871	-38.17	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
4872	-38.19	kd	CGS001-89766	UMODL1	-			
4873	-38.19	kd	CGS001-7167	TPI1	-			
4874	-38.2	oe	ccsbBroad304_01556	SMARCB1	-			
4875	-38.25	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
4876	-38.25	kd	CGS001-8575	PRKRA	-			
4877	-38.26	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
4878	-38.34	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
4879	-38.35	oe	ccsbBroad304_00098	ARG1	Arginase			
4880	-38.35	kd	CGS001-23266	LPHN2	Adhesion Class GPCRs			
4881	-38.41	oe	ccsbBroad304_01183	PGD	-			
4882	-38.42	oe	ccsbBroad304_04788	OVCA2	-			
4883	-38.45	kd	CGS001-7465	WEE1	WEE family			
4884	-38.45	kd	CGS001-949	SCARB1	-			
4885	-38.47	oe	ccsbBroad304_02919	KIAA1279	-			
4886	-38.49	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
4887	-38.51	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
4888	-38.52	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
4889	-38.53	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
4890	-38.56	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
4891	-38.58	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
4892	-38.58	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
4893	-38.6	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
4894	-38.63	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
4895	-38.65	oe	ccsbBroad304_02415	TUBB3	Tubulins			
4896	-38.65	oe	ccsbBroad304_07208	NRIP1	-			
4897	-38.68	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4898	-38.69	oe	ccsbBroad304_00648	GLRX	-			
4899	-38.72	oe	ccsbBroad304_02676	PHB2	-			
4900	-38.73	kd	CGS001-79080	CCDC86	-			
4901	-38.74	kd	CGS001-6271	S100A1	EF-hand domain containing			
4902	-38.74	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
4903	-38.79	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
4904	-38.79	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
4905	-38.85	oe	ccsbBroad304_07411	LPXN	-			
4906	-38.88	oe	ccsbBroad304_00006	ACADM	-			
4907	-38.89	oe	ccsbBroad304_02278	THRAP3	-			
4908	-38.92	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
4909	-38.92	oe	ccsbBroad304_07651	HEXIM1	-			
4910	-38.95	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
4911	-38.95	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
4912	-38.96	oe	ccsbBroad304_02306	PQBP1	-			
4913	-38.96	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
4914	-38.96	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
4915	-38.96	cp	BRD-K94144010	cotinine	Nicotine metabolite			Nicotine metabolite
4916	-38.99	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
4917	-39.01	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
4918	-39.03	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
4919	-39.06	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
4920	-39.06	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
4921	-39.07	kd	CGS001-7296	TXNRD1	-			
4922	-39.08	kd	CGS001-8726	EED	Neutral sphingomyelinase coupling factors			
4923	-39.09	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
4924	-39.11	oe	ccsbBroad304_07920	NUP62	-			
4925	-39.19	kd	CGS001-5253	PHF2	Histone demethylases			
4926	-39.25	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
4927	-39.28	kd	CGS001-54732	TMED9	-			
4928	-39.29	oe	ccsbBroad304_06777	PRNP	CD molecules			
4929	-39.32	kd	CGS001-30836	DNTTIP2	-			
4930	-39.38	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
4931	-39.41	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
4932	-39.45	kd	CGS001-2115	ETV1	ETS Transcription Factors			
4933	-39.48	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
4934	-39.5	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
4935	-39.5	kd	CGS001-10221	TRIB1	Trbl family			
4936	-39.53	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
4937	-39.54	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
4938	-39.55	kd	CGS001-7165	TPD52L2	-			
4939	-39.57	kd	CGS001-498	ATP5A1	ATPases / F-type			
4940	-39.6	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
4941	-39.62	kd	CGS001-3998	LMAN1	-			
4942	-39.63	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
4943	-39.67	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
4944	-39.67	kd	CGS001-4047	LSS	Lanosterol biosynthesis pathway			
4945	-39.69	oe	ccsbBroad304_01584	SPARC	-			
4946	-39.72	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
4947	-39.74	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
4948	-39.74	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
4949	-39.78	cc		Aldehyde dehydrogenases LOF	-			
4950	-39.78	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
4951	-39.78	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
4952	-39.86	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
4953	-39.9	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
4954	-39.92	cc		HRH1 antagonist	-			
4955	-39.93	kd	CGS001-545	ATR	ATR subfamily			
4956	-39.97	oe	ccsbBroad304_02702	MSRB2	-			
4957	-40	oe	ccsbBroad304_03565	ADI1	-			
4958	-40.09	kd	CGS001-6696	SPP1	Endogenous ligands			
4959	-40.12	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
4960	-40.13	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
4961	-40.13	kd	CGS001-222546	RFX6	-			
4962	-40.14	kd	CGS001-9319	TRIP13	ATPases / AAA-type			
4963	-40.17	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
4964	-40.19	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
4965	-40.19	kd	CGS001-144811	LACC1	-			
4966	-40.19	kd	CGS001-345611	IRGM	-			
4967	-40.3	kd	CGS001-8835	SOCS2	SH2 domain containing			
4968	-40.34	kd	CGS001-5612	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
4969	-40.35	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
4970	-40.38	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
4971	-40.39	kd	CGS001-1128	CHRM1	Cholinergic receptors			
4972	-40.41	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
4973	-40.42	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
4974	-40.43	oe	ccsbBroad304_01623	SUPT4H1	-			
4975	-40.43	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
4976	-40.43	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4977	-40.44	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
4978	-40.47	kd	CGS001-7157	TP53	-			
4979	-40.48	oe	ccsbBroad304_05183	TXLNA	-			
4980	-40.55	oe	ccsbBroad304_11405	UBE3C	-			
4981	-40.55	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
4982	-40.55	kd	CGS001-11336	EXOC3	-			
4983	-40.57	oe	ccsbBroad304_03980	DCLRE1B	-			
4984	-40.6	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
4985	-40.63	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
4986	-40.64	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
4987	-40.65	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
4988	-40.67	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
4989	-40.68	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
4990	-40.69	kd	CGS001-143	PARP4	Poly (ADP-ribose) polymerases			
4991	-40.7	kd	CGS001-5613	PRKX	Protein kinase A			
4992	-40.71	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
4993	-40.71	oe	ccsbBroad304_03428	EXOSC4	-			
4994	-40.72	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4995	-40.72	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
4996	-40.74	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
4997	-40.74	kd	CGS001-501	ALDH7A1	Aldehyde dehydrogenases			
4998	-40.74	oe	ccsbBroad304_06549	SMAD3	SMADs			
4999	-40.76	kd	CGS001-51734	SEPX1	-			
5000	-40.86	oe	ccsbBroad304_06094	DFFA	-			
5001	-40.86	cp	BRD-K21806131	tegaserod	Serotonin receptor partial agonist		HTR4, HTR2B, HTR2A, HTR2C	Serotonin receptor partial agonist
5002	-40.86	kd	CGS001-6822	SULT2A1	Sulfotransferases, cytosolic			
5003	-40.87	oe	ccsbBroad304_06264	GBP2	-			
5004	-40.89	kd	CGS001-6364	CCL20	Chemokine ligands			
5005	-40.94	oe	ccsbBroad304_03119	C16ORF5	-			
5006	-40.94	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
5007	-40.95	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
5008	-40.96	oe	ccsbBroad304_05439	O3FAR1	-			
5009	-40.99	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
5010	-41.01	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
5011	-41.04	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
5012	-41.05	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
5013	-41.06	oe	ccsbBroad304_00222	CASP6	Caspases			
5014	-41.06	kd	CGS001-597	BCL2A1	-			
5015	-41.07	oe	ccsbBroad304_00250	CD19	CD molecules			
5016	-41.08	cp	BRD-A80383043	BRD-A80383043	Glutamate receptor agonist		GRM1, GRM2	Glutamate receptor agonist, Glutamate receptor antagonist
5017	-41.08	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
5018	-41.09	cc		Apolipoproteins LOF	-			
5019	-41.15	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
5020	-41.16	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
5021	-41.23	kd	CGS001-80237	ELL3	-			
5022	-41.24	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
5023	-41.29	kd	CGS001-10287	RGS19	Regulators of G-protein signaling			
5024	-41.32	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
5025	-41.34	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
5026	-41.36	kd	CGS001-7132	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
5027	-41.38	cc		BMP Signaling LOF	-			
5028	-41.38	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
5029	-41.39	oe	ccsbBroad304_03232	VPS28	-			
5030	-41.41	cc		EIF Proteins LOF	-			
5031	-41.45	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
5032	-41.46	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
5033	-41.48	kd	CGS001-10452	TOMM40	-			
5034	-41.54	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
5035	-41.54	kd	CGS001-5580	PRKCD	Delta subfamily			
5036	-41.56	oe	ccsbBroad304_13813	ARAF	RAF family			
5037	-41.58	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
5038	-41.61	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
5039	-41.61	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
5040	-41.63	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
5041	-41.64	kd	CGS001-293	SLC25A6	Mitochondrial nucleotide transporter subfamily			
5042	-41.64	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
5043	-41.64	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
5044	-41.65	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
5045	-41.7	kd	CGS001-9807	IP6K1	-			
5046	-41.74	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
5047	-41.74	kd	CGS001-29915	HCFC2	-			
5048	-41.76	kd	CGS001-4837	NNMT	-			
5049	-41.88	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
5050	-41.88	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
5051	-41.89	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
5052	-41.91	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
5053	-41.93	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
5054	-41.95	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
5055	-41.95	kd	CGS001-6461	SHB	SH2 domain containing			
5056	-41.96	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
5057	-41.96	kd	CGS001-4048	LTA4H	Hydrolases			
5058	-41.97	kd	CGS001-5576	PRKAR2A	Protein kinase A			
5059	-41.98	kd	CGS001-5226	PGD	-			
5060	-42	kd	CGS001-9200	PTPLA	-			
5061	-42.06	kd	CGS001-5460	POU5F1	Homeoboxes / POU class			
5062	-42.09	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
5063	-42.1	kd	CGS001-4926	NUMA1	-			
5064	-42.11	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
5065	-42.13	oe	ccsbBroad304_06287	GM2A	-			
5066	-42.14	oe	ccsbBroad304_06952	SKP1	-			
5067	-42.14	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
5068	-42.16	cc		General transcription factors group 1 LOF	-			
5069	-42.16	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
5070	-42.17	kd	CGS001-8569	MKNK1	MKN subfamily			
5071	-42.18	oe	ccsbBroad304_02955	MYCBP	-			
5072	-42.19	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
5073	-42.21	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
5074	-42.22	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5075	-42.23	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
5076	-42.25	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
5077	-42.25	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5078	-42.3	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
5079	-42.31	cc		SRY LOF	-			
5080	-42.32	cp	BRD-K13800121	parecoxib	Cyclooxygenase inhibitor		LTF, PTGS2	Cyclooxygenase inhibitor
5081	-42.34	oe	ccsbBroad304_07727	LIAS	-			
5082	-42.34	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
5083	-42.36	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
5084	-42.36	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
5085	-42.41	kd	CGS001-2099	ESR1	Estrogen receptors			
5086	-42.45	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
5087	-42.45	kd	CGS001-29947	DNMT3L	-			
5088	-42.46	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
5089	-42.49	kd	CGS001-57222	ERGIC1	-			
5090	-42.55	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
5091	-42.61	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5092	-42.62	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5093	-42.63	kd	CGS001-8655	DYNLL1	Cytoplasmic dyneins			
5094	-42.65	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
5095	-42.66	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
5096	-42.67	kd	CGS001-5050	PAFAH1B3	-			
5097	-42.71	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
5098	-42.72	cp	BRD-A87387433	cefpodoxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5099	-42.72	kd	CGS001-5423	POLB	DNA polymerases			
5100	-42.73	cp	BRD-K30563334	rifabutin	Protein synthesis inhibitor		CYP3A4, HSP90AA1, HSP90B1	Protein synthesis inhibitor
5101	-42.76	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
5102	-42.77	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
5103	-42.79	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
5104	-42.82	kd	CGS001-533	ATP6V0B	ATPases / V-type			
5105	-42.83	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
5106	-42.83	oe	ccsbBroad304_01976	EIF4EBP3	-			
5107	-42.91	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
5108	-42.93	oe	ccsbBroad304_08055	ATP5S	-			
5109	-42.94	oe	ccsbBroad304_07843	FCHO1	-			
5110	-42.94	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
5111	-43.07	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
5112	-43.08	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
5113	-43.08	kd	CGS001-80714	PBX4	Homeoboxes / TALE class			
5114	-43.11	kd	CGS001-821	CANX	-			
5115	-43.12	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
5116	-43.12	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
5117	-43.12	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
5118	-43.13	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
5119	-43.14	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
5120	-43.15	kd	CGS001-5931	RBBP7	WD repeat domain containing			
5121	-43.17	kd	CGS001-11243	PMF1	-			
5122	-43.18	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
5123	-43.2	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
5124	-43.22	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
5125	-43.22	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
5126	-43.22	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
5127	-43.25	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
5128	-43.25	kd	CGS001-79109	MAPKAP1	-			
5129	-43.26	kd	CGS001-4751	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5130	-43.27	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
5131	-43.35	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
5132	-43.38	kd	CGS001-8438	RAD54L	-			
5133	-43.46	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
5134	-43.46	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
5135	-43.47	kd	CGS001-3119	HLA-DQB1	Immunoglobulin superfamily / C1-set domain containing			
5136	-43.49	kd	CGS001-165082	GPR113	Adhesion Class GPCRs			
5137	-43.5	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
5138	-43.53	kd	CGS001-23365	ARHGEF12	Rho guanine nucleotide exchange factors			
5139	-43.55	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
5140	-43.57	kd	CGS001-7054	TH	Amino acid hydroxylases			
5141	-43.58	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
5142	-43.66	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
5143	-43.69	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
5144	-43.7	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
5145	-43.73	oe	ccsbBroad304_01152	PCNA	-			
5146	-43.74	kd	CGS001-7040	TGFB1	Endogenous ligands			
5147	-43.75	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
5148	-43.77	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
5149	-43.78	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
5150	-43.8	cp	BRD-K89708791	rifaximin	RNA synthesis inhibitor		NR1I2, CYP3A4	RNA synthesis inhibitor
5151	-43.82	oe	ccsbBroad304_00376	CSK	Csk family			
5152	-43.86	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
5153	-43.86	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
5154	-43.87	kd	CGS001-169792	GLIS3	Zinc fingers, C2H2-type			
5155	-43.93	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
5156	-43.98	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
5157	-44	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
5158	-44	kd	CGS001-10142	AKAP9	A-kinase anchor proteins			
5159	-44.01	kd	CGS001-4245	MGAT1	-			
5160	-44.06	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5161	-44.07	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
5162	-44.07	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
5163	-44.12	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
5164	-44.15	cc		Glycogen synthase kinase inhibitor	-			
5165	-44.19	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
5166	-44.19	kd	CGS001-5422	POLA1	DNA polymerases			
5167	-44.22	oe	ccsbBroad304_00570	FIGF	-			
5168	-44.24	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5169	-44.27	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5170	-44.32	kd	CGS001-5073	PARN	-			
5171	-44.34	kd	CGS001-54541	DDIT4	-			
5172	-44.35	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
5173	-44.35	kd	CGS001-523	ATP6V1A	ATPases / V-type			
5174	-44.37	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
5175	-44.39	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5176	-44.4	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
5177	-44.45	kd	CGS001-2959	GTF2B	General transcription factors			
5178	-44.48	kd	CGS001-9512	PMPCB	-			
5179	-44.49	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
5180	-44.52	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
5181	-44.54	kd	CGS001-1105	CHD1	-			
5182	-44.56	cc		MTOR inhibitor	-			
5183	-44.57	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
5184	-44.6	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
5185	-44.64	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
5186	-44.64	kd	CGS001-55165	CEP55	-			
5187	-44.66	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
5188	-44.7	oe	ccsbBroad304_07197	PDHX	-			
5189	-44.71	kd	CGS001-8850	KAT2B	Histone acetyltransferases (HATs)			
5190	-44.72	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
5191	-44.73	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
5192	-44.73	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
5193	-44.75	kd	CGS001-1949	EFNB3	Ephrins			
5194	-44.86	oe	ccsbBroad304_03311	EVL	-			
5195	-44.91	oe	ccsbBroad304_02497	YKT6	-			
5196	-44.91	cp	BRD-K62374253	rufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
5197	-44.93	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
5198	-45.07	kd	CGS001-8651	SOCS1	SH2 domain containing			
5199	-45.1	kd	CGS001-3205	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
5200	-45.11	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
5201	-45.17	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
5202	-45.18	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
5203	-45.18	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
5204	-45.23	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
5205	-45.24	oe	ccsbBroad304_02443	HAX1	-			
5206	-45.31	oe	ccsbBroad304_06066	CTSL1	-			
5207	-45.4	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
5208	-45.43	kd	CGS001-10112	KIF20A	Kinesins			
5209	-45.49	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
5210	-45.49	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
5211	-45.5	kd	CGS001-7088	TLE1	WD repeat domain containing			
5212	-45.52	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
5213	-45.52	kd	CGS001-4697	NDUFA4	-			
5214	-45.55	kd	CGS001-3560	IL2RB	IL-2 receptor family			
5215	-45.57	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
5216	-45.6	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
5217	-45.65	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
5218	-45.66	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
5219	-45.68	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
5220	-45.68	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5221	-45.68	kd	CGS001-369	ARAF	RAF family			
5222	-45.72	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
5223	-45.77	oe	ccsbBroad304_06651	NOV	-			
5224	-45.81	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
5225	-45.81	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5226	-45.81	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
5227	-45.85	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
5228	-45.86	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
5229	-45.86	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
5230	-45.89	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
5231	-45.89	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
5232	-45.94	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5233	-46.01	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
5234	-46.07	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
5235	-46.13	oe	ccsbBroad304_00053	ALDOA	-			
5236	-46.15	kd	CGS001-6721	SREBF2	Basic helix-loop-helix proteins			
5237	-46.18	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5238	-46.27	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
5239	-46.27	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
5240	-46.28	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
5241	-46.29	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5242	-46.3	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
5243	-46.32	kd	CGS001-5433	POLR2D	RNA polymerase subunits			
5244	-46.4	kd	CGS001-6856	SYPL1	-			
5245	-46.45	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
5246	-46.46	kd	CGS001-1512	CTSH	Cathepsins			
5247	-46.5	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
5248	-46.5	oe	ccsbBroad304_06324	GPX7	-			
5249	-46.51	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
5250	-46.53	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
5251	-46.54	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
5252	-46.55	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
5253	-46.59	oe	ccsbBroad304_07827	STK38L	NDR family			
5254	-46.61	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5255	-46.62	kd	CGS001-238	ALK	Leukocyte tyrosine kinase (LTK) receptor family			
5256	-46.64	oe	ccsbBroad304_14242	MCCC2	-			
5257	-46.65	kd	CGS001-4086	SMAD1	SMADs			
5258	-46.67	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
5259	-46.67	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
5260	-46.68	cc		PI3K inhibitor	-			
5261	-46.73	kd	CGS001-6259	RYK	Type XV RTKs: RYK			
5262	-46.75	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
5263	-46.76	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
5264	-46.86	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
5265	-46.87	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
5266	-46.89	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
5267	-46.89	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5268	-46.9	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
5269	-46.92	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
5270	-46.93	oe	ccsbBroad304_04038	ELOVL6	-			
5271	-46.95	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5272	-46.98	kd	CGS001-5144	PDE4D	Phosphodiesterases			
5273	-47.02	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
5274	-47.03	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5275	-47.05	cp	BRD-K17705806	JTC-801	Opioid receptor antagonist		OPRL1	Opioid receptor antagonist
5276	-47.08	kd	CGS001-5831	PYCR1	-			
5277	-47.11	kd	CGS001-25	ABL1	Abl family			
5278	-47.18	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
5279	-47.18	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
5280	-47.2	kd	CGS001-9797	TATDN2	-			
5281	-47.21	kd	CGS001-4638	MYLK	Myosin Light Chain Kinase (MLCK) family			
5282	-47.22	kd	CGS001-64170	CARD9	-			
5283	-47.24	kd	CGS001-3551	IKBKB	IKK family			
5284	-47.24	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
5285	-47.31	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
5286	-47.37	kd	CGS001-54681	P4HTM	-			
5287	-47.37	kd	CGS001-51203	NUSAP1	-			
5288	-47.39	kd	CGS001-10383	TUBB2C	Tubulins			
5289	-47.41	oe	ccsbBroad304_02270	FAM20B	-			
5290	-47.52	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
5291	-47.55	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
5292	-47.55	kd	CGS001-6767	ST13	Tetratricopeptide (TTC) repeat domain containing			
5293	-47.61	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
5294	-47.62	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
5295	-47.62	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5296	-47.65	oe	ccsbBroad304_01640	TAF12	-			
5297	-47.7	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
5298	-47.72	kd	CGS001-5575	PRKAR1B	Protein kinase A			
5299	-47.74	oe	ccsbBroad304_04053	DERL1	-			
5300	-47.77	oe	ccsbBroad304_01845	RDBP	-			
5301	-47.78	oe	ccsbBroad304_07024	SYK	Syk family			
5302	-47.79	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
5303	-47.79	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5304	-47.8	oe	ccsbBroad304_07220	CDC45	-			
5305	-47.8	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
5306	-47.85	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
5307	-47.85	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
5308	-47.88	kd	CGS001-24148	PRPF6	-			
5309	-47.93	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
5310	-48	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
5311	-48.05	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
5312	-48.05	kd	CGS001-9159	PCSK7	Subtilisin			
5313	-48.08	cc		VEGFR inhibitor	-			
5314	-48.17	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
5315	-48.25	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
5316	-48.25	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5317	-48.26	kd	CGS001-7272	TTK	TTK family			
5318	-48.28	cp	BRD-K10670311	sulfasalazine	Antirheumatic		PTGS1, PTGS2, ACAT1, ALOX5, CHUK, IKBKB, PLA2G1B, PPARG, SLC46A1, SLC7A11, TBXAS1	Antirheumatic, NFkB pathway inhibitor
5319	-48.34	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
5320	-48.35	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
5321	-48.37	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
5322	-48.42	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
5323	-48.44	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
5324	-48.45	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
5325	-48.47	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
5326	-48.53	kd	CGS001-56882	CDC42SE1	-			
5327	-48.57	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
5328	-48.61	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
5329	-48.61	cp	BRD-A88254928	salbutamol	Adrenergic receptor agonist		ADRB2, ADRB1	Adrenergic receptor agonist
5330	-48.68	kd	CGS001-11179	ZNF277	-			
5331	-48.69	oe	ccsbBroad304_01483	SAT1	-			
5332	-48.71	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
5333	-48.74	kd	CGS001-6850	SYK	Syk family			
5334	-48.76	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
5335	-48.76	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
5336	-48.77	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
5337	-48.93	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
5338	-48.94	oe	ccsbBroad304_02018	SUCLA2	-			
5339	-48.97	oe	ccsbBroad304_04202	MED28	-			
5340	-48.98	kd	CGS001-10423	CDIPT	-			
5341	-49	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
5342	-49.01	kd	CGS001-7597	ZBTB25	BTB/POZ domain containing			
5343	-49.07	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
5344	-49.09	kd	CGS001-3708	ITPR1	Ion channels / Inositol triphosphate receptors			
5345	-49.1	kd	CGS001-56889	TM9SF3	-			
5346	-49.11	kd	CGS001-23384	SPECC1L	-			
5347	-49.13	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
5348	-49.18	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
5349	-49.18	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
5350	-49.18	kd	CGS001-813	CALU	EF-hand domain containing			
5351	-49.19	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
5352	-49.21	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
5353	-49.22	kd	CGS001-23753	SDF2L1	-			
5354	-49.24	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5355	-49.3	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
5356	-49.31	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
5357	-49.31	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
5358	-49.32	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
5359	-49.36	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
5360	-49.44	kd	CGS001-330	BIRC3	Inhibitors of apoptosis (IAP) protein family			
5361	-49.45	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
5362	-49.46	oe	ccsbBroad304_00239	CCNG1	-			
5363	-49.48	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
5364	-49.49	kd	CGS001-775	CACNA1C	Calcium channel subunits			
5365	-49.54	oe	ccsbBroad304_01769	VEGFB	-			
5366	-49.57	kd	CGS001-51293	CD320	CD molecules			
5367	-49.58	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
5368	-49.61	kd	CGS001-5255	PHKA1	-			
5369	-49.69	kd	CGS001-64135	IFIH1	-			
5370	-49.73	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
5371	-49.77	kd	CGS001-9158	FIBP	-			
5372	-49.82	kd	CGS001-5810	RAD1	-			
5373	-49.85	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
5374	-49.86	kd	CGS001-8317	CDC7	CDC7 family			
5375	-49.92	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
5376	-49.93	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
5377	-49.94	kd	CGS001-2896	GRN	-			
5378	-49.95	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
5379	-49.96	kd	CGS001-2837	UTS2R	Urotensin receptor			
5380	-50.06	kd	CGS001-2674	GFRA1	GDNF receptor family			
5381	-50.07	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
5382	-50.08	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
5383	-50.1	oe	ccsbBroad304_02298	DNM1L	-			
5384	-50.14	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
5385	-50.15	kd	CGS001-6886	TAL1	Basic helix-loop-helix proteins			
5386	-50.16	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5387	-50.17	oe	ccsbBroad304_08536	PARL	-			
5388	-50.23	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
5389	-50.25	oe	ccsbBroad304_00841	IKBKB	IKK family			
5390	-50.29	cc		Aromatase inhibitor	-			
5391	-50.31	oe	ccsbBroad304_00472	EBF1	-			
5392	-50.41	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
5393	-50.43	kd	CGS001-4439	MSH5	-			
5394	-50.44	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
5395	-50.45	oe	ccsbBroad304_09615	LACC1	-			
5396	-50.5	kd	CGS001-2597	GAPDH	-			
5397	-50.52	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
5398	-50.56	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
5399	-50.56	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
5400	-50.56	kd	CGS001-63933	CCDC90A	-			
5401	-50.57	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
5402	-50.59	cc		Leucine rich repeat kinase inhibitor	-			
5403	-50.59	kd	CGS001-6443	SGCB	-			
5404	-50.67	cp	BRD-K02227374	milnacipran	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Serotonin reuptake inhibitor
5405	-50.68	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
5406	-50.7	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
5407	-50.77	kd	CGS001-51070	NOSIP	-			
5408	-50.84	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
5409	-50.85	kd	CGS001-64750	SMURF2	-			
5410	-50.94	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
5411	-50.96	kd	CGS001-10914	PAPOLA	-			
5412	-50.97	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
5413	-50.97	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
5414	-50.97	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
5415	-51.02	oe	ccsbBroad304_00615	GAPDH	-			
5416	-51.04	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
5417	-51.13	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
5418	-51.13	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
5419	-51.15	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
5420	-51.17	oe	ccsbBroad304_10431	HADHB	-			
5421	-51.28	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
5422	-51.33	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
5423	-51.42	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
5424	-51.48	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
5425	-51.54	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
5426	-51.56	oe	ccsbBroad304_07145	ZFP161	-			
5427	-51.6	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
5428	-51.63	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
5429	-51.63	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
5430	-51.64	kd	CGS001-1854	DUT	-			
5431	-51.66	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
5432	-51.67	kd	CGS001-2957	GTF2A1	General transcription factors			
5433	-51.76	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
5434	-51.77	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
5435	-51.78	oe	ccsbBroad304_01658	PRDX2	-			
5436	-51.79	oe	ccsbBroad304_14011	PAPSS1	-			
5437	-51.79	kd	CGS001-22887	FOXJ3	Forkhead boxes			
5438	-51.83	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
5439	-51.83	kd	CGS001-9784	SNX17	Sorting nexins			
5440	-51.85	kd	CGS001-831	CAST	-			
5441	-51.87	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
5442	-51.98	kd	CGS001-84930	MASTL	MAST family			
5443	-51.99	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
5444	-52.07	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
5445	-52.09	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
5446	-52.11	oe	ccsbBroad304_01054	GADD45B	-			
5447	-52.13	kd	CGS001-1611	DAP	-			
5448	-52.15	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
5449	-52.17	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5450	-52.19	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
5451	-52.22	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
5452	-52.22	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
5453	-52.23	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
5454	-52.26	kd	CGS001-29888	STRN4	WD repeat domain containing			
5455	-52.27	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
5456	-52.33	oe	ccsbBroad304_07515	GFPT2	-			
5457	-52.34	cp	BRD-K04710043	hexamethylenebisacetamide	AKT inhibitor			AKT inhibitor, Differentiation inducer, NFkB pathway inhibitor
5458	-52.36	kd	CGS001-11015	KDELR3	-			
5459	-52.38	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
5460	-52.39	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
5461	-52.45	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
5462	-52.52	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
5463	-52.54	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
5464	-52.56	kd	CGS001-10099	TSPAN3	Tetraspanins			
5465	-52.58	cp	BRD-A01787639	naftopidil	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
5466	-52.59	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
5467	-52.65	kd	CGS001-8833	GMPS	-			
5468	-52.69	oe	ccsbBroad304_01373	RAN	-			
5469	-52.81	cp	BRD-A23359898	sibutramine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, CYP2B6, CYP2C19, CYP3A5	Serotonin reuptake inhibitor
5470	-52.89	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
5471	-52.94	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
5472	-52.95	oe	ccsbBroad304_09578	PASD1	-			
5473	-52.95	cp	BRD-K55034111	pefloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
5474	-53.01	oe	ccsbBroad304_03310	LCMT1	-			
5475	-53.04	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
5476	-53.09	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
5477	-53.1	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
5478	-53.1	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5479	-53.11	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
5480	-53.12	cc		Adenosine receptor agonist	-			
5481	-53.12	oe	ccsbBroad304_00501	EMD	-			
5482	-53.2	oe	ccsbBroad304_02572	SERINC3	-			
5483	-53.23	kd	CGS001-324	APC	Armadillo repeat containing			
5484	-53.3	oe	ccsbBroad304_07029	TADA2A	-			
5485	-53.31	oe	ccsbBroad304_02875	BRP44	-			
5486	-53.32	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
5487	-53.37	kd	CGS001-8738	CRADD	-			
5488	-53.38	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
5489	-53.43	cc		ATP synthase inhibitor	-			
5490	-53.44	oe	ccsbBroad304_02801	CASP14	Caspases			
5491	-53.44	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
5492	-53.46	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
5493	-53.49	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
5494	-53.51	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5495	-53.52	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
5496	-53.54	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
5497	-53.57	kd	CGS001-1633	DCK	-			
5498	-53.58	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
5499	-53.58	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
5500	-53.58	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
5501	-53.6	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
5502	-53.67	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
5503	-53.68	oe	ccsbBroad304_00572	FKBP3	-			
5504	-53.69	kd	CGS001-5571	PRKAG1	AMPK subfamily			
5505	-53.71	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
5506	-53.72	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
5507	-53.75	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
5508	-53.77	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
5509	-53.79	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
5510	-53.81	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
5511	-53.86	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
5512	-53.91	kd	CGS001-7474	WNT5A	Endogenous ligands			
5513	-53.93	kd	CGS001-7295	TXN	-			
5514	-53.93	kd	CGS001-6050	RNH1	-			
5515	-54.04	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
5516	-54.07	kd	CGS001-115201	ATG4A	-			
5517	-54.14	kd	CGS001-10437	IFI30	-			
5518	-54.17	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
5519	-54.17	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
5520	-54.18	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
5521	-54.18	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
5522	-54.19	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
5523	-54.21	oe	ccsbBroad304_03615	ZNF673	-			
5524	-54.21	oe	ccsbBroad304_00231	CBFB	-			
5525	-54.21	kd	CGS001-29083	GTPBP8	-			
5526	-54.27	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
5527	-54.29	kd	CGS001-4092	SMAD7	SMADs			
5528	-54.32	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
5529	-54.37	cc		Minor histocompatibility antigens LOF	-			
5530	-54.37	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
5531	-54.44	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
5532	-54.54	kd	CGS001-7105	TSPAN6	Tetraspanins			
5533	-54.56	kd	CGS001-9180	OSMR	IL-6 receptor family			
5534	-54.6	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
5535	-54.61	oe	ccsbBroad304_06159	CTTN	-			
5536	-54.62	oe	ccsbBroad304_01166	PDK2	PDHK family			
5537	-54.62	kd	CGS001-3821	KLRC1	CD molecules			
5538	-54.67	kd	CGS001-50865	HEBP1	Endogenous ligands			
5539	-54.69	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
5540	-54.72	cc		HSP inhibitor	-			
5541	-54.78	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
5542	-54.82	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
5543	-54.86	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
5544	-54.86	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
5545	-54.88	oe	ccsbBroad304_07287	HYAL2	-			
5546	-54.89	oe	ccsbBroad304_04387	MKI67IP	-			
5547	-54.9	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
5548	-54.94	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5549	-54.98	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
5550	-55.04	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
5551	-55.1	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
5552	-55.1	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
5553	-55.11	oe	ccsbBroad304_01748	UFD1L	-			
5554	-55.11	kd	CGS001-116113	FOXP4	Forkhead boxes			
5555	-55.14	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
5556	-55.16	kd	CGS001-7013	TERF1	-			
5557	-55.17	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
5558	-55.18	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
5559	-55.18	kd	CGS001-3242	HPD	Oxidoreductases			
5560	-55.21	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
5561	-55.22	kd	CGS001-586	BCAT1	-			
5562	-55.24	oe	ccsbBroad304_07320	SQSTM1	-			
5563	-55.3	oe	ccsbBroad304_01951	BLZF1	-			
5564	-55.34	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
5565	-55.35	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
5566	-55.37	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
5567	-55.39	kd	CGS001-8678	BECN1	-			
5568	-55.45	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
5569	-55.49	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
5570	-55.51	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
5571	-55.51	kd	CGS001-8572	PDLIM4	-			
5572	-55.52	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
5573	-55.55	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
5574	-55.56	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5575	-55.58	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
5576	-55.59	cc		Calcium channel blocker	-			
5577	-55.62	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
5578	-55.68	oe	ccsbBroad304_03772	CCNL1	-			
5579	-55.7	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
5580	-55.7	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
5581	-55.71	kd	CGS001-7311	UBA52	L ribosomal proteins			
5582	-55.72	kd	CGS001-160	AP2A1	-			
5583	-55.73	cp	BRD-K66896231	BRD-K66896231	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5584	-55.87	cp	BRD-K00673382	famotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
5585	-55.98	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
5586	-56.15	cc		Protein synthesis inhibitor	-			
5587	-56.15	kd	CGS001-8935	SKAP2	Pleckstrin homology (PH) domain containing			
5588	-56.19	oe	ccsbBroad304_10491	PFKL	-			
5589	-56.19	oe	ccsbBroad304_07267	PDLIM4	-			
5590	-56.21	kd	CGS001-7345	UCHL1	Ubiquitin C-terminal hydrolase			
5591	-56.22	kd	CGS001-351	APP	Endogenous ligands			
5592	-56.23	cc		Norepinephrine reuptake inhibitor	-			
5593	-56.27	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
5594	-56.27	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
5595	-56.35	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
5596	-56.41	kd	CGS001-6446	SGK1	SGK family			
5597	-56.45	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
5598	-56.49	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
5599	-56.51	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
5600	-56.54	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
5601	-56.55	kd	CGS001-11284	PNKP	-			
5602	-56.57	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
5603	-56.57	oe	ccsbBroad304_02368	TIMM17B	-			
5604	-56.6	oe	ccsbBroad304_00446	DKC1	-			
5605	-56.64	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
5606	-56.67	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
5607	-56.72	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
5608	-56.73	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
5609	-56.73	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
5610	-56.73	kd	CGS001-10174	SORBS3	-			
5611	-56.79	kd	CGS001-220	ALDH1A3	Aldehyde dehydrogenases			
5612	-56.89	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
5613	-56.9	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
5614	-56.92	cc		PPAR receptor agonist	-			
5615	-56.92	oe	ccsbBroad304_08898	TRAK2	-			
5616	-56.92	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
5617	-56.96	kd	CGS001-10111	RAD50	-			
5618	-57.01	kd	CGS001-51284	TLR7	Toll-like receptor family			
5619	-57.05	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
5620	-57.12	kd	CGS001-8453	CUL2	-			
5621	-57.13	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
5622	-57.13	kd	CGS001-10827	FAM114A2	-			
5623	-57.17	oe	ccsbBroad304_07252	DGKZ	-			
5624	-57.18	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
5625	-57.19	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
5626	-57.22	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
5627	-57.23	cc		Tricyclic antidepressant	-			
5628	-57.25	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
5629	-57.27	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
5630	-57.3	kd	CGS001-23549	DNPEP	Aminopeptidase I			
5631	-57.34	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
5632	-57.34	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
5633	-57.36	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
5634	-57.36	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
5635	-57.41	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
5636	-57.45	kd	CGS001-9133	CCNB2	-			
5637	-57.46	kd	CGS001-5336	PLCG2	Phosphoinositide-specific phospholipase C			
5638	-57.47	kd	CGS001-10153	CEBPZ	-			
5639	-57.5	kd	CGS001-136	ADORA2B	GPCR / Class A : Adenosine receptors			
5640	-57.51	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
5641	-57.62	kd	CGS001-55163	PNPO	-			
5642	-57.63	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
5643	-57.64	kd	CGS001-8233	ZRSR2	RNA binding motif (RRM) containing			
5644	-57.77	kd	CGS001-3992	FADS1	Fatty acid desaturases			
5645	-57.81	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
5646	-57.81	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
5647	-57.86	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
5648	-57.88	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
5649	-57.9	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
5650	-57.91	oe	ccsbBroad304_10240	CROT	-			
5651	-57.92	oe	ccsbBroad304_05098	MAGEB6	-			
5652	-58.01	kd	CGS001-2872	MKNK2	MKN subfamily			
5653	-58.02	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
5654	-58.03	kd	CGS001-2967	GTF2H3	General transcription factors			
5655	-58.06	kd	CGS001-4967	OGDH	-			
5656	-58.06	kd	CGS001-9988	DMTF1	-			
5657	-58.07	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
5658	-58.08	oe	ccsbBroad304_06008	AP2M1	-			
5659	-58.1	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
5660	-58.14	kd	CGS001-6502	SKP2	F-boxes / Leucine-rich repeats			
5661	-58.17	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
5662	-58.18	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
5663	-58.19	kd	CGS001-50943	FOXP3	Forkhead boxes			
5664	-58.21	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
5665	-58.28	kd	CGS001-8841	HDAC3	Histone deacetylases			
5666	-58.32	kd	CGS001-11331	PHB2	-			
5667	-58.34	cp	BRD-A75935363	atracurium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
5668	-58.35	kd	CGS001-64223	MLST8	WD repeat domain containing			
5669	-58.38	kd	CGS001-2806	GOT2	-			
5670	-58.46	kd	CGS001-310	ANXA7	Annexins			
5671	-58.5	cp	BRD-K92870997	pterostilbene	Cyclooxygenase inhibitor		FAAH, PPARA, PTGS1, PTGS2	Cyclooxygenase inhibitor, PPAR receptor agonist
5672	-58.51	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
5673	-58.53	cc		Estrogen receptor agonist	-			
5674	-58.62	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
5675	-58.71	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
5676	-58.8	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5677	-58.81	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
5678	-58.81	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5679	-58.89	oe	ccsbBroad304_00626	GDI1	-			
5680	-58.9	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
5681	-58.96	oe	ccsbBroad304_08292	IP6K2	-			
5682	-58.96	kd	CGS001-5159	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5683	-58.99	kd	CGS001-5345	SERPINF2	Serine (or cysteine) peptidase inhibitors			
5684	-58.99	kd	CGS001-5033	P4HA1	-			
5685	-59.01	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
5686	-59.11	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
5687	-59.11	kd	CGS001-301	ANXA1	Annexins			
5688	-59.14	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
5689	-59.15	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
5690	-59.17	kd	CGS001-327	APEH	Prolyl oligopeptidase			
5691	-59.22	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
5692	-59.22	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
5693	-59.23	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
5694	-59.24	kd	CGS001-10013	HDAC6	Histone deacetylases			
5695	-59.31	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
5696	-59.34	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
5697	-59.35	kd	CGS001-2057	EPOR	Prolactin receptor family			
5698	-59.36	oe	ccsbBroad304_02864	PRDX5	-			
5699	-59.39	kd	CGS001-7314	UBB	-			
5700	-59.39	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
5701	-59.41	kd	CGS001-9748	SLK	SLK subfamily			
5702	-59.42	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
5703	-59.43	kd	CGS001-5914	RARA	Retinoic acid receptors			
5704	-59.45	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
5705	-59.5	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
5706	-59.54	kd	CGS001-1499	CTNNB1	Catenins			
5707	-59.55	kd	CGS001-8824	CES2	Carboxylesterases			
5708	-59.56	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5709	-59.57	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
5710	-59.58	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
5711	-59.68	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
5712	-59.69	oe	ccsbBroad304_14020	SH3BP5	-			
5713	-59.69	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
5714	-59.7	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
5715	-59.7	kd	CGS001-54925	ZNF434	-			
5716	-59.72	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
5717	-59.72	kd	CGS001-221188	GPR114	Adhesion Class GPCRs			
5718	-59.73	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
5719	-59.76	cp	BRD-K97752965	nicorandil	Nitric oxide donor		ABCC9, KCNJ11, KCNJ8	Nitric oxide donor, Potassium channel activator
5720	-59.8	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
5721	-59.8	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
5722	-59.86	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
5723	-59.88	kd	CGS001-3832	KIF11	Kinesins			
5724	-59.91	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
5725	-59.92	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
5726	-59.93	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
5727	-60.05	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
5728	-60.08	oe	ccsbBroad304_01234	POLB	DNA polymerases			
5729	-60.12	kd	CGS001-10018	BCL2L11	-			
5730	-60.13	oe	ccsbBroad304_03625	HIF1AN	-			
5731	-60.15	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
5732	-60.16	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
5733	-60.21	kd	CGS001-283	ANG	Ribonucleases, RNase A			
5734	-60.24	cc		P38 MAPK inhibitor	-			
5735	-60.24	kd	CGS001-3673	ITGA2	Integrins			
5736	-60.33	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
5737	-60.33	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
5738	-60.34	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
5739	-60.37	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5740	-60.38	kd	CGS001-23244	PDS5A	-			
5741	-60.39	kd	CGS001-3481	IGF2	-			
5742	-60.4	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
5743	-60.46	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
5744	-60.5	oe	ccsbBroad304_02032	TSC22D1	-			
5745	-60.51	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
5746	-60.53	oe	ccsbBroad304_00542	FBP1	-			
5747	-60.56	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5748	-60.6	kd	CGS001-7016	TESK1	TESK subfamily			
5749	-60.61	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5750	-60.61	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
5751	-60.63	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
5752	-60.64	kd	CGS001-9641	IKBKE	IKK family			
5753	-60.67	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
5754	-60.68	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
5755	-60.74	kd	CGS001-27034	ACAD8	-			
5756	-60.77	kd	CGS001-26128	KIAA1279	-			
5757	-60.8	kd	CGS001-641	BLM	-			
5758	-60.83	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
5759	-60.86	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
5760	-60.93	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
5761	-60.93	kd	CGS001-51282	SCAND1	-			
5762	-60.93	kd	CGS001-55239	OGFOD1	-			
5763	-60.95	oe	ccsbBroad304_07094	TPMT	-			
5764	-61.03	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
5765	-61.05	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
5766	-61.06	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
5767	-61.08	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
5768	-61.09	kd	CGS001-111	ADCY5	Adenylate cyclases			
5769	-61.14	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
5770	-61.17	oe	ccsbBroad304_10437	STMN1	-			
5771	-61.25	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
5772	-61.29	oe	ccsbBroad304_00112	ASNA1	-			
5773	-61.3	kd	CGS001-11200	CHEK2	CHK1 subfamily			
5774	-61.32	cp	BRD-K50866992	tropisetron	Serotonin receptor antagonist		HTR3A, GLRA1, GLRA2, GLRB, HTR4	Serotonin receptor antagonist
5775	-61.35	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
5776	-61.37	cc		EGFR inhibitor	-			
5777	-61.39	kd	CGS001-3487	IGFBP4	insulin-like growth factor (IGF) binding proteins			
5778	-61.41	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
5779	-61.44	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
5780	-61.44	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
5781	-61.44	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
5782	-61.54	cc		Non Homologous End Joining LOF	-			
5783	-61.61	kd	CGS001-2773	GNAI3	-			
5784	-61.64	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
5785	-61.66	kd	CGS001-80150	ASRGL1	-			
5786	-61.67	oe	ccsbBroad304_03479	YTHDF1	-			
5787	-61.68	kd	CGS001-65263	PYCRL	-			
5788	-61.75	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
5789	-61.77	oe	ccsbBroad304_03808	ERGIC1	-			
5790	-61.86	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
5791	-61.86	kd	CGS001-8313	AXIN2	-			
5792	-61.89	kd	CGS001-1936	EEF1D	-			
5793	-61.9	kd	CGS001-79947	DHDDS	-			
5794	-61.91	kd	CGS001-2863	GPR39	GPCR / Class A : Orphans			
5795	-61.92	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
5796	-61.92	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
5797	-61.92	kd	CGS001-8503	PIK3R3	Phosphatidylinositol kinases			
5798	-61.94	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
5799	-61.96	oe	ccsbBroad304_03080	C16ORF80	-			
5800	-62.02	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
5801	-62.05	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
5802	-62.06	oe	ccsbBroad304_00492	EIF5A	-			
5803	-62.11	oe	ccsbBroad304_06683	FURIN	Subtilisin			
5804	-62.14	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
5805	-62.14	kd	CGS001-3074	HEXB	-			
5806	-62.21	kd	CGS001-6622	SNCA	Parkinson disease			
5807	-62.25	kd	CGS001-353345	GPR141	GPCR / Class A : Orphans			
5808	-62.26	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
5809	-62.28	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
5810	-62.3	oe	ccsbBroad304_02218	IKBKE	IKK family			
5811	-62.3	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
5812	-62.31	kd	CGS001-375133	PI4KAP2	-			
5813	-62.33	kd	CGS001-2782	GNB1	WD repeat domain containing			
5814	-62.36	oe	ccsbBroad304_00036	AFP	-			
5815	-62.37	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
5816	-62.37	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
5817	-62.37	kd	CGS001-991	CDC20	WD repeat domain containing			
5818	-62.39	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
5819	-62.39	kd	CGS001-27244	SESN1	-			
5820	-62.39	kd	CGS001-2230	FDX1	-			
5821	-62.41	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
5822	-62.43	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
5823	-62.51	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
5824	-62.55	kd	CGS001-55612	FERMT1	Fermitins			
5825	-62.56	oe	ccsbBroad304_06565	MB	-			
5826	-62.65	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
5827	-62.68	kd	CGS001-1844	DUSP2	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
5828	-62.7	cp	BRD-K41051431	mecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5829	-62.72	kd	CGS001-5501	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5830	-62.74	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
5831	-62.76	oe	ccsbBroad304_05890	BHMT	-			
5832	-62.79	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5833	-62.84	kd	CGS001-11164	NUDT5	Nudix motif containing			
5834	-62.85	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
5835	-62.88	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
5836	-62.93	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
5837	-62.93	oe	ccsbBroad304_03235	TUBD1	Tubulins			
5838	-62.95	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
5839	-62.98	kd	CGS001-54536	EXOC6	-			
5840	-63	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
5841	-63	kd	CGS001-79258	MMEL1	-			
5842	-63.03	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
5843	-63.1	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
5844	-63.1	kd	CGS001-4077	NBR1	-			
5845	-63.17	kd	CGS001-2247	FGF2	Endogenous ligands			
5846	-63.22	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
5847	-63.26	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
5848	-63.32	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
5849	-63.38	kd	CGS001-6520	SLC3A2	SLC3 family			
5850	-63.4	kd	CGS001-6793	STK10	SLK subfamily			
5851	-63.41	oe	ccsbBroad304_00038	AGL	-			
5852	-63.42	kd	CGS001-9377	COX5A	Mitochondrial respiratory chain complex			
5853	-63.45	kd	CGS001-1398	CRK	SH2 domain containing			
5854	-63.55	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
5855	-63.58	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
5856	-63.61	oe	ccsbBroad304_00389	CTBP1	-			
5857	-63.66	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
5858	-63.72	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
5859	-63.73	kd	CGS001-6929	TCF3	Basic helix-loop-helix proteins			
5860	-63.79	cc		NFkB pathway inhibitor	-			
5861	-63.79	kd	CGS001-257397	TAB3	-			
5862	-63.84	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
5863	-63.84	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
5864	-63.85	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5865	-63.87	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
5866	-63.9	kd	CGS001-2197	FAU	S ribosomal proteins			
5867	-63.9	kd	CGS001-133690	CAPSL	EF-hand domain containing			
5868	-63.93	kd	CGS001-2969	GTF2I	General transcription factors			
5869	-63.95	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
5870	-63.98	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
5871	-64.01	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
5872	-64.02	cc		Serotonin receptor antagonist	-			
5873	-64.1	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
5874	-64.12	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
5875	-64.12	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
5876	-64.13	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
5877	-64.14	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
5878	-64.14	kd	CGS001-1051	CEBPB	basic leucine zipper proteins			
5879	-64.14	kd	CGS001-55256	ADI1	-			
5880	-64.15	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
5881	-64.17	kd	CGS001-6617	SNAPC1	-			
5882	-64.18	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
5883	-64.19	kd	CGS001-847	CAT	-			
5884	-64.25	kd	CGS001-9568	GABBR2	GABA receptors			
5885	-64.27	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
5886	-64.29	cp	BRD-K39621635	artemether	Antimalarial		ATP1A1, CYP2B6, CYP2C19, CYP3A5	Antimalarial
5887	-64.32	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5888	-64.33	oe	ccsbBroad304_07754	FGFR1OP	-			
5889	-64.34	oe	ccsbBroad304_01754	UCK2	-			
5890	-64.34	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
5891	-64.37	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
5892	-64.38	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
5893	-64.42	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
5894	-64.43	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
5895	-64.45	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
5896	-64.48	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
5897	-64.55	kd	CGS001-51460	SFMBT1	Sterile alpha motif (SAM) domain containing			
5898	-64.67	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
5899	-64.68	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
5900	-64.71	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
5901	-64.76	kd	CGS001-22894	DIS3	-			
5902	-64.77	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
5903	-64.78	kd	CGS001-3725	JUN	basic leucine zipper proteins			
5904	-64.81	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5905	-64.85	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
5906	-64.9	kd	CGS001-1859	DYRK1A	Dyrk1 subfamily			
5907	-64.96	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
5908	-65.02	kd	CGS001-5997	RGS2	Endogenous ligands			
5909	-65.03	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
5910	-65.05	oe	ccsbBroad304_01930	CUL2	-			
5911	-65.13	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
5912	-65.14	kd	CGS001-1163	CKS1B	-			
5913	-65.15	kd	CGS001-10523	CHERP	G patch domain containing			
5914	-65.16	kd	CGS001-1119	CHKA	-			
5915	-65.17	kd	CGS001-11157	LSM6	-			
5916	-65.22	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
5917	-65.38	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
5918	-65.43	kd	CGS001-25949	SYF2	-			
5919	-65.43	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
5920	-65.47	kd	CGS001-1173	AP2M1	-			
5921	-65.5	oe	ccsbBroad304_00874	INS	-			
5922	-65.52	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
5923	-65.56	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
5924	-65.56	oe	ccsbBroad304_02229	TRAM2	-			
5925	-65.61	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
5926	-65.62	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
5927	-65.64	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
5928	-65.66	cp	BRD-K52020312	metronidazole	DNA inhibitor		CYP2C8, CYP2E1, CYP3A5, CYP3A7	DNA inhibitor, Antiprotozoal
5929	-65.68	oe	ccsbBroad304_07326	EIF2B2	-			
5930	-65.77	kd	CGS001-3034	HAL	-			
5931	-65.8	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
5932	-65.8	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
5933	-65.81	cc		Mitochondrial complex IV LOF	-			
5934	-65.88	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
5935	-65.89	oe	ccsbBroad304_07887	GCAT	-			
5936	-65.94	kd	CGS001-657	BMPR1A	Type I receptor serine/threonine kinases			
5937	-65.97	kd	CGS001-23466	CBX6	-			
5938	-66	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
5939	-66.04	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
5940	-66.08	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
5941	-66.08	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
5942	-66.1	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
5943	-66.18	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
5944	-66.26	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
5945	-66.32	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
5946	-66.33	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
5947	-66.35	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
5948	-66.36	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
5949	-66.37	cp	BRD-K09471561	levofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
5950	-66.39	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
5951	-66.41	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
5952	-66.51	kd	CGS001-5096	PCCB	Carboxylases			
5953	-66.55	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
5954	-66.67	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
5955	-66.77	kd	CGS001-2023	ENO1	-			
5956	-66.79	cp	BRD-K32744045	disulfiram	Aldehyde dehydrogenase inhibitor		ALDH2, ALDH1A2, ALDH5A1, ALDH7A1, CYP2E1, DBH, DNMT1, TRPA1	Aldehyde dehydrogenase inhibitor, TRPV agonist, DNA methyltransferase inhibitor
5957	-66.8	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
5958	-66.82	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
5959	-66.85	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
5960	-66.87	cc		Interleukins GOF	-			
5961	-66.89	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
5962	-66.96	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
5963	-66.96	kd	CGS001-1515	CTSL2	-			
5964	-67.01	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
5965	-67.03	kd	CGS001-7057	THBS1	-			
5966	-67.04	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
5967	-67.06	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
5968	-67.08	cp	BRD-A02189320	met-leu-phe	-666			-666
5969	-67.08	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
5970	-67.13	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
5971	-67.16	oe	ccsbBroad304_08596	EAPP	-			
5972	-67.2	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
5973	-67.2	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
5974	-67.23	kd	CGS001-10397	NDRG1	-			
5975	-67.23	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
5976	-67.24	kd	CGS001-54438	GFOD1	-			
5977	-67.25	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
5978	-67.26	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
5979	-67.3	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
5980	-67.32	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
5981	-67.39	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
5982	-67.44	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
5983	-67.45	kd	CGS001-6193	RPS5	S ribosomal proteins			
5984	-67.52	kd	CGS001-79921	TCEAL4	-			
5985	-67.53	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5986	-67.59	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
5987	-67.61	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
5988	-67.63	oe	ccsbBroad304_06870	RNH1	-			
5989	-67.64	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
5990	-67.65	kd	CGS001-5595	MAPK3	MAPK:ERK subfamily			
5991	-67.71	kd	CGS001-5932	RBBP8	-			
5992	-67.72	kd	CGS001-4671	NAIP	Inhibitors of apoptosis (IAP) protein family			
5993	-67.78	kd	CGS001-3226	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
5994	-67.81	kd	CGS001-9552	SPAG7	-			
5995	-67.86	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
5996	-67.93	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
5997	-67.95	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5998	-67.98	kd	CGS001-55746	NUP133	-			
5999	-68.01	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
6000	-68.06	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
6001	-68.09	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
6002	-68.11	kd	CGS001-7919	DDX39B	DEAD-boxes			
6003	-68.12	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
6004	-68.17	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6005	-68.26	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
6006	-68.3	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
6007	-68.3	kd	CGS001-2760	GM2A	-			
6008	-68.31	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
6009	-68.31	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
6010	-68.32	cc		Cannabinoid receptor agonist	-			
6011	-68.32	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
6012	-68.35	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
6013	-68.36	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6014	-68.41	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
6015	-68.41	kd	CGS001-5682	PSMA1	Proteasome subunits			
6016	-68.43	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6017	-68.45	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
6018	-68.45	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
6019	-68.46	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
6020	-68.57	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
6021	-68.68	oe	ccsbBroad304_01593	SRP14	-			
6022	-68.69	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
6023	-68.75	kd	CGS001-2629	GBA	-			
6024	-68.77	kd	CGS001-57147	SCYL3	-			
6025	-68.78	kd	CGS001-7020	TFAP2A	-			
6026	-68.79	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
6027	-68.94	cp	BRD-K82109576	vincristine	Tubulin inhibitor		TUBB, TUBA4A	Tubulin inhibitor
6028	-68.95	kd	CGS001-6897	TARS	Aminoacyl tRNA synthetases / Class II			
6029	-68.95	kd	CGS001-2558	GABRA5	GABA receptors			
6030	-68.95	kd	CGS001-1213	CLTC	-			
6031	-68.95	kd	CGS001-998	CDC42	-			
6032	-68.98	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
6033	-68.99	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
6034	-69.02	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6035	-69.04	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
6036	-69.04	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
6037	-69.04	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
6038	-69.1	cc		Progesterone receptor antagonist	-			
6039	-69.13	kd	CGS001-8853	ASAP2	Ankyrin repeat domain containing			
6040	-69.16	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
6041	-69.19	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
6042	-69.22	kd	CGS001-6387	CXCL12	Endogenous ligands			
6043	-69.22	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
6044	-69.29	oe	ccsbBroad304_04616	ORMDL3	-			
6045	-69.36	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
6046	-69.36	kd	CGS001-84634	KISS1R	GPCR / Class A : RF amide peptide receptors			
6047	-69.42	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
6048	-69.44	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
6049	-69.45	kd	CGS001-2958	GTF2A2	General transcription factors			
6050	-69.47	oe	ccsbBroad304_00987	MCM3	-			
6051	-69.48	kd	CGS001-29916	SNX11	Sorting nexins			
6052	-69.56	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
6053	-69.56	kd	CGS001-1027	CDKN1B	-			
6054	-69.58	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
6055	-69.63	kd	CGS001-1314	COPA	Endogenous ligands			
6056	-69.64	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6057	-69.66	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
6058	-69.67	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
6059	-69.69	kd	CGS001-7480	WNT10B	Wingless-type MMTV integration sites			
6060	-69.71	kd	CGS001-7431	VIM	Intermediate filaments type III			
6061	-69.71	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
6062	-69.73	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
6063	-69.74	kd	CGS001-57018	CCNL1	-			
6064	-69.78	kd	CGS001-9929	JOSD1	-			
6065	-69.82	kd	CGS001-4801	NFYB	-			
6066	-69.9	kd	CGS001-5217	PFN2	-			
6067	-69.9	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6068	-69.96	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
6069	-70.03	oe	ccsbBroad304_02115	PTTG1	-			
6070	-70.03	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
6071	-70.04	kd	CGS001-11040	PIM2	PIM family			
6072	-70.07	kd	CGS001-10972	TMED10	-			
6073	-70.12	kd	CGS001-26298	EHF	-			
6074	-70.16	oe	ccsbBroad304_07600	NSA2	-			
6075	-70.19	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
6076	-70.24	oe	ccsbBroad304_00462	DR1	-			
6077	-70.24	kd	CGS001-23102	TBC1D2B	-			
6078	-70.25	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
6079	-70.26	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
6080	-70.4	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
6081	-70.4	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
6082	-70.41	cc		NFKB Activation GOF	-			
6083	-70.5	oe	ccsbBroad304_03933	CARD9	-			
6084	-70.5	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
6085	-70.5	kd	CGS001-7421	VDR	Vitamin D receptors			
6086	-70.5	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
6087	-70.51	kd	CGS001-6663	SOX10	SRY (sex determining region Y)-boxes			
6088	-70.52	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
6089	-70.55	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
6090	-70.55	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
6091	-70.57	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
6092	-70.65	cc		HIF activator	-			
6093	-70.65	kd	CGS001-2182	ACSL4	Acyl-CoA synthetase family			
6094	-70.7	kd	CGS001-64422	ATG3	-			
6095	-70.71	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
6096	-70.74	kd	CGS001-10020	GNE	-			
6097	-70.79	kd	CGS001-2944	GSTM1	Glutathione S-transferases / Soluble			
6098	-70.82	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
6099	-70.88	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
6100	-70.89	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
6101	-70.9	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
6102	-70.9	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
6103	-70.92	kd	CGS001-10084	PQBP1	-			
6104	-70.93	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
6105	-70.93	kd	CGS001-999	CDH1	CD molecules			
6106	-70.95	kd	CGS001-3569	IL6	Interferons			
6107	-70.99	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
6108	-71	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
6109	-71.01	oe	ccsbBroad304_02578	EBNA1BP2	-			
6110	-71.04	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
6111	-71.05	kd	CGS001-5230	PGK1	-			
6112	-71.05	oe	ccsbBroad304_07119	UGP2	-			
6113	-71.06	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
6114	-71.08	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
6115	-71.16	kd	CGS001-84159	ARID5B	-			
6116	-71.17	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
6117	-71.27	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
6118	-71.37	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
6119	-71.38	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
6120	-71.38	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
6121	-71.39	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
6122	-71.4	kd	CGS001-2849	GPR26	GPCR / Class A : Orphans			
6123	-71.42	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
6124	-71.45	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
6125	-71.46	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
6126	-71.46	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
6127	-71.46	kd	CGS001-2021	ENDOG	-			
6128	-71.53	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
6129	-71.54	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
6130	-71.56	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
6131	-71.56	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
6132	-71.58	cc		Cyclooxygenase inhibitor	-			
6133	-71.6	kd	CGS001-5110	PCMT1	-			
6134	-71.64	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
6135	-71.64	kd	CGS001-1026	CDKN1A	-			
6136	-71.64	kd	CGS001-3281	HSBP1	-			
6137	-71.65	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
6138	-71.66	kd	CGS001-3660	IRF2	-			
6139	-71.68	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
6140	-71.73	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
6141	-71.75	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
6142	-71.79	kd	CGS001-5565	PRKAB2	AMPK subfamily			
6143	-71.82	oe	ccsbBroad304_00651	GNAI3	-			
6144	-71.86	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
6145	-71.89	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
6146	-71.91	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
6147	-71.95	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
6148	-71.98	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
6149	-71.98	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
6150	-72	cc		RNA Polymerase Enzymes LOF	-			
6151	-72.01	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
6152	-72.04	cc		Ribonucleotide reductase inhibitor	-			
6153	-72.05	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
6154	-72.07	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6155	-72.13	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
6156	-72.19	kd	CGS001-4835	NQO2	-			
6157	-72.22	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
6158	-72.23	cp	BRD-K23369905	oxiconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6159	-72.27	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
6160	-72.29	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
6161	-72.35	oe	ccsbBroad304_00551	FECH	-			
6162	-72.45	oe	ccsbBroad304_08137	HOOK2	-			
6163	-72.51	oe	ccsbBroad304_00397	CTSK	Cathepsins			
6164	-72.51	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6165	-72.58	oe	ccsbBroad304_06301	GOT2	-			
6166	-72.59	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
6167	-72.61	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
6168	-72.63	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
6169	-72.66	oe	ccsbBroad304_04465	RERG	-			
6170	-72.66	kd	CGS001-7276	TTR	-			
6171	-72.68	kd	CGS001-51441	YTHDF2	-			
6172	-72.73	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
6173	-72.75	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
6174	-72.75	kd	CGS001-4709	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6175	-72.76	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
6176	-72.8	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
6177	-72.81	cp	BRD-K46742498	alosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
6178	-73	kd	CGS001-486	FXYD2	Ion transport regulator			
6179	-73	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
6180	-73.01	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
6181	-73.04	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6182	-73.08	kd	CGS001-388677	NOTCH2NL	-			
6183	-73.13	kd	CGS001-7415	VCP	ATPases / AAA-type			
6184	-73.18	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6185	-73.2	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
6186	-73.21	kd	CGS001-10813	UTP14A	-			
6187	-73.23	oe	ccsbBroad304_02596	KDELR3	-			
6188	-73.23	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
6189	-73.23	kd	CGS001-9967	THRAP3	-			
6190	-73.26	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
6191	-73.32	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
6192	-73.36	oe	ccsbBroad304_02756	RRP8	-			
6193	-73.43	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
6194	-73.44	kd	CGS001-6599	SMARCC1	-			
6195	-73.46	kd	CGS001-5411	PNN	-			
6196	-73.47	oe	ccsbBroad304_03570	QRSL1	-			
6197	-73.47	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
6198	-73.5	kd	CGS001-5511	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6199	-73.52	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
6200	-73.52	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
6201	-73.54	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
6202	-73.56	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
6203	-73.57	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
6204	-73.57	kd	CGS001-124626	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6205	-73.59	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
6206	-73.6	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
6207	-73.61	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
6208	-73.63	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
6209	-73.67	cp	BRD-K33106058	cytarabine	Ribonucleotide reductase inhibitor		POLB, POLA1	Ribonucleotide reductase inhibitor
6210	-73.68	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
6211	-73.73	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
6212	-73.76	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6213	-73.79	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
6214	-73.8	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
6215	-73.83	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
6216	-73.88	kd	CGS001-5707	PSMD1	Proteasome subunits			
6217	-73.89	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
6218	-73.94	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
6219	-73.97	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
6220	-74	kd	CGS001-6204	RPS10	S ribosomal proteins			
6221	-74.02	kd	CGS001-5209	PFKFB3	-			
6222	-74.04	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
6223	-74.04	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
6224	-74.08	kd	CGS001-290	ANPEP	Aminopeptidase N			
6225	-74.1	oe	ccsbBroad304_00991	MDH1	-			
6226	-74.15	kd	CGS001-7541	ZFP161	-			
6227	-74.17	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
6228	-74.18	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
6229	-74.19	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
6230	-74.2	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
6231	-74.22	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
6232	-74.23	kd	CGS001-2145	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
6233	-74.25	kd	CGS001-2735	GLI1	Zinc fingers, C2H2-type			
6234	-74.25	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
6235	-74.27	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
6236	-74.28	kd	CGS001-8914	TIMELESS	-			
6237	-74.32	kd	CGS001-6491	STIL	-			
6238	-74.4	oe	ccsbBroad304_07922	TRIM29	-			
6239	-74.41	kd	CGS001-22	ABCB7	ATP binding cassette transporters / subfamily B			
6240	-74.49	cp	BRD-K82147103	lofepramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
6241	-74.53	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
6242	-74.54	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
6243	-74.57	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
6244	-74.58	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
6245	-74.59	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
6246	-74.59	kd	CGS001-139760	GPR119	GPCR / Class A : Orphans			
6247	-74.68	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
6248	-74.73	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
6249	-74.75	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
6250	-74.75	kd	CGS001-83448	PUS7L	-			
6251	-74.77	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
6252	-74.79	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
6253	-74.86	cp	BRD-K53220666	trimetozine	Sedative			Sedative
6254	-74.86	kd	CGS001-35	ACADS	-			
6255	-74.91	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
6256	-74.95	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
6257	-74.96	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
6258	-75.05	kd	CGS001-10969	EBNA1BP2	-			
6259	-75.05	kd	CGS001-56005	C19ORF10	-			
6260	-75.13	oe	ccsbBroad304_07511	KIF14	Kinesins			
6261	-75.14	kd	CGS001-3383	ICAM1	CD molecules			
6262	-75.17	cp	BRD-K69650333	idarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
6263	-75.17	kd	CGS001-5045	FURIN	Subtilisin			
6264	-75.18	kd	CGS001-55011	PIH1D1	-			
6265	-75.25	oe	ccsbBroad304_06523	LIG1	-			
6266	-75.27	kd	CGS001-515	ATP5F1	ATPases / F-type			
6267	-75.3	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
6268	-75.32	kd	CGS001-7428	VHL	-			
6269	-75.32	kd	CGS001-51005	AMDHD2	-			
6270	-75.33	kd	CGS001-9945	GFPT2	-			
6271	-75.35	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6272	-75.41	oe	ccsbBroad304_06996	SRM	-			
6273	-75.44	kd	CGS001-5805	PTS	-			
6274	-75.48	oe	ccsbBroad304_07178	ZFP112	-			
6275	-75.48	kd	CGS001-5188	PET112	-			
6276	-75.5	cc		NADH ubiquinone oxidoreductase supernumerary subunits LOF	-			
6277	-75.51	oe	ccsbBroad304_07861	COBL	-			
6278	-75.57	kd	CGS001-115	ADCY9	Adenylyl cyclases			
6279	-75.61	kd	CGS001-572	BAD	-			
6280	-75.62	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6281	-75.64	oe	ccsbBroad304_02219	MORF4L2	-			
6282	-75.65	kd	CGS001-10285	SMNDC1	Tudor domain containing			
6283	-75.68	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
6284	-75.7	kd	CGS001-2746	GLUD1	-			
6285	-75.7	kd	CGS001-1072	CFL1	-			
6286	-75.78	oe	ccsbBroad304_01002	METTL1	-			
6287	-75.79	kd	CGS001-6493	SIM2	Basic helix-loop-helix proteins			
6288	-75.87	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6289	-75.88	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
6290	-75.89	cc		Angiotensin receptor antagonist	-			
6291	-75.93	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
6292	-75.94	oe	ccsbBroad304_06040	CRY1	-			
6293	-75.95	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
6294	-75.96	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
6295	-75.97	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
6296	-75.98	kd	CGS001-1386	ATF2	basic leucine zipper proteins			
6297	-76.01	kd	CGS001-5566	PRKACA	Protein kinase A			
6298	-76.04	oe	ccsbBroad304_06525	LIPA	-			
6299	-76.09	kd	CGS001-7251	TSG101	-			
6300	-76.2	kd	CGS001-178	AGL	-			
6301	-76.24	cc		Cyclin dependent kinases LOF	-			
6302	-76.28	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
6303	-76.32	kd	CGS001-2100	ESR2	Estrogen receptors			
6304	-76.33	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
6305	-76.35	kd	CGS001-22832	KIAA1009	-			
6306	-76.36	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
6307	-76.37	oe	ccsbBroad304_06126	TSC22D3	-			
6308	-76.39	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6309	-76.43	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
6310	-76.47	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
6311	-76.48	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
6312	-76.5	oe	ccsbBroad304_07071	TKT	-			
6313	-76.52	oe	ccsbBroad304_02788	PRAME	-			
6314	-76.52	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
6315	-76.53	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6316	-76.53	kd	CGS001-51096	UTP18	WD repeat domain containing			
6317	-76.62	kd	CGS001-4144	MAT2A	-			
6318	-76.63	cc		Cell Cycle Inhibition GOF	-			
6319	-76.63	oe	ccsbBroad304_06133	TOR1A	-			
6320	-76.63	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6321	-76.65	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
6322	-76.67	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
6323	-76.68	cc		Imidazoline ligand	-			
6324	-76.69	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
6325	-76.7	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
6326	-76.73	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
6327	-76.75	oe	ccsbBroad304_00833	IFNG	Interferons			
6328	-76.78	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
6329	-76.78	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
6330	-76.8	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
6331	-76.8	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
6332	-76.81	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
6333	-76.82	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
6334	-76.84	kd	CGS001-3572	IL6ST	IL-6 receptor family			
6335	-76.92	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
6336	-76.93	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
6337	-76.93	kd	CGS001-59343	SENP2	-			
6338	-76.94	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
6339	-76.97	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
6340	-76.97	oe	ccsbBroad304_00262	CD59	CD molecules			
6341	-76.98	oe	ccsbBroad304_07632	PROCR	CD molecules			
6342	-76.99	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
6343	-77	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
6344	-77.02	cp	BRD-K73991644	isoquercetin	Aldose reductase inhibitor		AKR1B1, ACE	Aldose reductase inhibitor
6345	-77.04	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
6346	-77.04	oe	ccsbBroad304_00690	GRN	-			
6347	-77.06	kd	CGS001-2677	GGCX	Carboxylases			
6348	-77.07	oe	ccsbBroad304_07401	TXNL1	-			
6349	-77.07	kd	CGS001-5498	PPOX	-			
6350	-77.09	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
6351	-77.13	kd	CGS001-6788	STK3	MST subfamily			
6352	-77.19	oe	ccsbBroad304_04379	LZIC	-			
6353	-77.2	cc		Rho associated kinase inhibitor	-			
6354	-77.2	oe	ccsbBroad304_10212	GRHL3	-			
6355	-77.25	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
6356	-77.27	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
6357	-77.31	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
6358	-77.36	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
6359	-77.45	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6360	-77.5	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
6361	-77.51	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
6362	-77.57	oe	ccsbBroad304_00085	APRT	-			
6363	-77.6	kd	CGS001-944	TNFSF8	CD molecules			
6364	-77.62	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
6365	-77.64	kd	CGS001-6909	TBX2	T-boxes			
6366	-77.68	kd	CGS001-50808	AK3	-			
6367	-77.69	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
6368	-77.69	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
6369	-77.77	kd	CGS001-56654	NPDC1	-			
6370	-77.8	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
6371	-77.8	kd	CGS001-50813	COPS7A	-			
6372	-77.86	cp	BRD-K44442813	pidotimod	Interferon receptor agonist			Interferon receptor agonist, Interleukin receptor agonist
6373	-77.9	kd	CGS001-26993	AKAP8L	-			
6374	-77.91	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
6375	-77.94	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
6376	-77.96	kd	CGS001-5663	PSEN1	Presenilin			
6377	-78.03	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
6378	-78.06	oe	ccsbBroad304_02175	MAGED1	-			
6379	-78.08	cp	BRD-K88701661	dimercaptosuccinic-acid	Chelating agent		DNMT1	Chelating agent
6380	-78.13	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
6381	-78.13	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
6382	-78.14	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
6383	-78.25	cc		Lysine acetyltransferases LOF	-			
6384	-78.25	kd	CGS001-4931	NVL	ATPases / AAA-type			
6385	-78.29	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
6386	-78.29	kd	CGS001-5538	PPT1	-			
6387	-78.33	kd	CGS001-150280	HORMAD2	-			
6388	-78.34	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6389	-78.38	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6390	-78.41	kd	CGS001-7077	TIMP2	-			
6391	-78.42	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
6392	-78.43	kd	CGS001-4436	MSH2	-			
6393	-78.44	cc		Bacterial 30S ribosomal subunit inhibitor	-			
6394	-78.44	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
6395	-78.49	cc		Phospholipases LOF	-			
6396	-78.5	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
6397	-78.52	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
6398	-78.55	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
6399	-78.55	kd	CGS001-7103	TSPAN8	Tetraspanins			
6400	-78.6	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
6401	-78.61	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
6402	-78.64	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
6403	-78.66	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
6404	-78.67	kd	CGS001-5329	PLAUR	CD molecules			
6405	-78.68	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
6406	-78.79	kd	CGS001-2274	FHL2	-			
6407	-78.81	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
6408	-78.82	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
6409	-78.85	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
6410	-78.87	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
6411	-78.88	oe	ccsbBroad304_06855	RDX	-			
6412	-78.91	kd	CGS001-10950	BTG3	-			
6413	-78.92	cp	BRD-K51671335	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
6414	-78.93	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
6415	-78.98	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
6416	-78.99	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
6417	-79.02	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
6418	-79.05	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
6419	-79.11	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
6420	-79.12	oe	ccsbBroad304_02458	STK25	YSK subfamily			
6421	-79.14	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
6422	-79.15	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
6423	-79.19	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
6424	-79.2	kd	CGS001-7076	TIMP1	-			
6425	-79.21	cp	BRD-A41450521	tosufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6426	-79.22	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
6427	-79.26	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
6428	-79.33	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
6429	-79.34	kd	CGS001-205	AK4	Adenylate kinases			
6430	-79.35	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
6431	-79.36	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
6432	-79.38	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
6433	-79.4	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
6434	-79.47	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
6435	-79.49	oe	ccsbBroad304_00491	EIF4EBP2	-			
6436	-79.5	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
6437	-79.54	kd	CGS001-3669	ISG20	-			
6438	-79.6	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
6439	-79.63	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
6440	-79.66	oe	ccsbBroad304_09281	TPD52L3	-			
6441	-79.69	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
6442	-79.7	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
6443	-79.79	cc		HDAC inhibitor	-			
6444	-79.84	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
6445	-79.84	kd	CGS001-644	BLVRA	-			
6446	-79.88	oe	ccsbBroad304_01034	MSH2	-			
6447	-79.92	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
6448	-79.92	kd	CGS001-3612	IMPA1	Inositol monophosphatase			
6449	-79.93	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
6450	-79.95	cp	BRD-K15519488	CS-110266	Dopamine receptor agonist		SLC6A3	Dopamine receptor agonist
6451	-79.95	kd	CGS001-7915	ALDH5A1	Aldehyde dehydrogenases			
6452	-79.96	kd	CGS001-2752	GLUL	-			
6453	-79.96	kd	CGS001-607	BCL9	-			
6454	-79.97	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
6455	-80	oe	ccsbBroad304_06103	DMD	-			
6456	-80.01	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6457	-80.07	kd	CGS001-6934	TCF7L2	-			
6458	-80.09	kd	CGS001-8826	IQGAP1	-			
6459	-80.1	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
6460	-80.15	oe	ccsbBroad304_00819	IDH3B	-			
6461	-80.2	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
6462	-80.27	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
6463	-80.29	kd	CGS001-4221	MEN1	-			
6464	-80.31	kd	CGS001-4605	MYBL2	-			
6465	-80.36	kd	CGS001-5293	PIK3CD	Phosphatidylinositol kinases			
6466	-80.42	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
6467	-80.43	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
6468	-80.44	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
6469	-80.47	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6470	-80.47	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
6471	-80.49	oe	ccsbBroad304_02287	GNPDA1	-			
6472	-80.5	oe	ccsbBroad304_02869	ASF1A	-			
6473	-80.54	kd	CGS001-3479	IGF1	Endogenous ligands			
6474	-80.55	cc		Serine proteases GOF	-			
6475	-80.55	kd	CGS001-11230	PRAF2	-			
6476	-80.56	kd	CGS001-8731	RNMT	-			
6477	-80.56	kd	CGS001-1727	CYB5R3	-			
6478	-80.58	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
6479	-80.59	kd	CGS001-5054	SERPINE1	Serine (or cysteine) peptidase inhibitors			
6480	-80.61	kd	CGS001-169436	C9ORF96	-			
6481	-80.63	oe	ccsbBroad304_04752	IKBIP	-			
6482	-80.66	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
6483	-80.67	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
6484	-80.68	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
6485	-80.71	kd	CGS001-84547	PGBD1	-			
6486	-80.73	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
6487	-80.73	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
6488	-80.73	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
6489	-80.75	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
6490	-80.76	kd	CGS001-2287	FKBP3	-			
6491	-80.77	oe	ccsbBroad304_03696	C19ORF10	-			
6492	-80.79	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
6493	-80.83	kd	CGS001-10775	POP4	-			
6494	-80.87	kd	CGS001-537	ATP6AP1	-			
6495	-80.89	kd	CGS001-25937	WWTR1	Hippo Signaling			
6496	-80.9	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
6497	-80.95	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
6498	-80.97	kd	CGS001-445	ASS1	-			
6499	-81.09	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
6500	-81.11	oe	ccsbBroad304_03506	AURKAIP1	-			
6501	-81.12	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
6502	-81.15	kd	CGS001-2621	GAS6	-			
6503	-81.23	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
6504	-81.24	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
6505	-81.31	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
6506	-81.36	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
6507	-81.4	kd	CGS001-57721	METTL14	-			
6508	-81.45	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
6509	-81.46	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
6510	-81.46	kd	CGS001-204	AK2	Adenylate kinases			
6511	-81.47	kd	CGS001-3845	KRAS	RAS subfamily			
6512	-81.51	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
6513	-81.54	kd	CGS001-283150	FOXR1	Forkhead boxes			
6514	-81.54	kd	CGS001-642	BLMH	-			
6515	-81.56	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
6516	-81.62	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
6517	-81.65	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
6518	-81.65	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
6519	-81.68	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
6520	-81.73	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
6521	-81.74	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
6522	-81.76	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
6523	-81.81	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
6524	-81.81	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
6525	-81.85	oe	ccsbBroad304_02271	LPGAT1	-			
6526	-81.87	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
6527	-81.88	oe	ccsbBroad304_02276	MVP	-			
6528	-81.89	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
6529	-81.92	cp	BRD-K66412701	pazufloxacin	Topoisomerase inhibitor			Topoisomerase inhibitor
6530	-81.95	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
6531	-81.99	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
6532	-82.01	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
6533	-82.01	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
6534	-82.02	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
6535	-82.04	kd	CGS001-9020	MAP3K14	MAPKKK:STE-unique family			
6536	-82.12	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
6537	-82.14	kd	CGS001-8659	ALDH4A1	Aldehyde dehydrogenases			
6538	-82.21	kd	CGS001-10651	MTX2	-			
6539	-82.23	cp	BRD-M41783010	acamprosate	Glutamate receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B, GRM5	Glutamate receptor antagonist
6540	-82.26	cc		Dopamine receptor antagonist	-			
6541	-82.27	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
6542	-82.28	kd	CGS001-5743	PTGS2	Cyclooxygenase			
6543	-82.28	kd	CGS001-5690	PSMB2	Proteasome subunits			
6544	-82.3	kd	CGS001-1452	CSNK1A1	Casein kinase 1 (CK1) family			
6545	-82.31	kd	CGS001-4927	NUP88	-			
6546	-82.32	cc		Canonical high mobility group proteins LOF	-			
6547	-82.35	kd	CGS001-3123	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
6548	-82.36	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
6549	-82.4	kd	CGS001-7128	TNFAIP3	OTU domain containing			
6550	-82.45	kd	CGS001-348	APOE	Apolipoproteins			
6551	-82.46	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
6552	-82.46	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
6553	-82.47	kd	CGS001-3593	IL12B	Interleukins and interleukin receptors			
6554	-82.49	oe	ccsbBroad304_02373	SPRY2	-			
6555	-82.52	kd	CGS001-8772	FADD	-			
6556	-82.54	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6557	-82.54	kd	CGS001-1616	DAXX	-			
6558	-82.56	oe	ccsbBroad304_02405	TFG	-			
6559	-82.65	kd	CGS001-6307	MSMO1	Fatty acid hydroxylase domain containing			
6560	-82.67	cc		CDK inhibitor	-			
6561	-82.72	oe	ccsbBroad304_00969	MAGEA10	-			
6562	-82.73	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
6563	-82.76	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
6564	-82.81	oe	ccsbBroad304_08093	DCPS	-			
6565	-82.81	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
6566	-82.83	cc		Tumor necrosis factor superfamily LOF	-			
6567	-82.83	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
6568	-82.84	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
6569	-82.85	oe	ccsbBroad304_06739	PLOD1	-			
6570	-82.85	kd	CGS001-2744	GLS	Ankyrin repeat domain containing			
6571	-82.86	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
6572	-82.88	kd	CGS001-5355	PLP2	-			
6573	-82.88	kd	CGS001-55107	ANO1	Calcium activated chloride channel			
6574	-82.93	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
6575	-82.93	kd	CGS001-10525	HYOU1	Heat shock proteins / HSP70			
6576	-83	oe	ccsbBroad304_06464	ITGB2	Integrins			
6577	-83.02	cc		Integrin subunits alpha LOF	-			
6578	-83.02	kd	CGS001-7263	TST	-			
6579	-83.06	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
6580	-83.09	cc		Reverse transcriptase inhibitor	-			
6581	-83.12	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
6582	-83.15	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
6583	-83.19	oe	ccsbBroad304_01052	MYB	-			
6584	-83.28	cc		Supressors of cytokine signaling GOF	-			
6585	-83.3	oe	ccsbBroad304_06178	ERCC5	-			
6586	-83.31	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
6587	-83.31	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
6588	-83.35	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
6589	-83.38	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
6590	-83.4	kd	CGS001-5058	PAK1	PAKA subfamily			
6591	-83.43	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
6592	-83.47	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6593	-83.48	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6594	-83.48	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
6595	-83.48	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
6596	-83.53	cp	BRD-A71009679	KUC103420N	-666			-666
6597	-83.53	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
6598	-83.53	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
6599	-83.54	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
6600	-83.59	oe	ccsbBroad304_02831	SGK3	SGK family			
6601	-83.64	kd	CGS001-9805	SCRN1	-			
6602	-83.66	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
6603	-83.66	kd	CGS001-10769	PLK2	Polo-like kinase (PLK) family			
6604	-83.73	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
6605	-83.73	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
6606	-83.74	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
6607	-83.79	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
6608	-83.83	kd	CGS001-8334	HIST1H2AC	Histones / Replication-dependent			
6609	-83.87	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
6610	-83.88	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
6611	-83.9	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
6612	-83.94	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
6613	-83.95	kd	CGS001-6258	RXRG	Retinoid X receptors			
6614	-84.02	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
6615	-84.04	cp	BRD-K63343048	orlistat	Lipase inhibitor		PNLIP, DAGLA, FASN, LIPF, CNR1, DAGLB	Lipase inhibitor
6616	-84.04	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
6617	-84.05	oe	ccsbBroad304_02671	ECD	-			
6618	-84.08	kd	CGS001-8634	RTCD1	-			
6619	-84.08	kd	CGS001-1195	CLK1	CDC-like kinases			
6620	-84.09	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
6621	-84.12	kd	CGS001-7267	TTC3	RING-type (C3HC4) zinc fingers			
6622	-84.13	kd	CGS001-9867	PJA2	RING-type (C3HC4) zinc fingers			
6623	-84.14	cp	BRD-K22947005	dexbrompheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6624	-84.16	kd	CGS001-5781	PTPN11	Protein tyrosine phosphatases			
6625	-84.16	kd	CGS001-54584	GNB1L	WD repeat domain containing			
6626	-84.17	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
6627	-84.18	oe	ccsbBroad304_00652	GNAS	-			
6628	-84.19	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
6629	-84.23	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
6630	-84.26	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
6631	-84.34	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
6632	-84.35	kd	CGS001-11124	FAF1	UBX domain containing			
6633	-84.37	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
6634	-84.39	kd	CGS001-7270	TTF1	-			
6635	-84.41	oe	ccsbBroad304_08684	CXCR7	-			
6636	-84.42	cp	BRD-A11990600	lorazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, TSPO	Benzodiazepine receptor agonist
6637	-84.46	oe	ccsbBroad304_07102	TSG101	-			
6638	-84.47	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
6639	-84.48	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6640	-84.49	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
6641	-84.52	kd	CGS001-51053	GMNN	-			
6642	-84.53	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
6643	-84.56	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
6644	-84.58	oe	ccsbBroad304_00210	CALR	-			
6645	-84.6	kd	CGS001-25819	CCRN4L	-			
6646	-84.61	oe	ccsbBroad304_05528	TICAM2	-			
6647	-84.61	kd	CGS001-53343	NUDT9	Nudix motif containing			
6648	-84.62	kd	CGS001-6871	TADA2A	-			
6649	-84.63	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
6650	-84.64	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
6651	-84.65	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
6652	-84.68	kd	CGS001-10131	TRAP1	Heat shock proteins / HSPC			
6653	-84.68	kd	CGS001-55699	IARS2	Aminoacyl tRNA synthetases / Class I			
6654	-84.7	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
6655	-84.84	oe	ccsbBroad304_00118	ATIC	-			
6656	-84.87	kd	CGS001-8797	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
6657	-84.88	kd	CGS001-10434	LYPLA1	-			
6658	-84.92	kd	CGS001-340371	NRBP2	NRBP family			
6659	-84.93	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
6660	-84.98	kd	CGS001-54821	ERCC6L	-			
6661	-84.99	kd	CGS001-7032	TFF2	-			
6662	-85.03	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6663	-85.04	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6664	-85.05	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
6665	-85.07	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6666	-85.13	kd	CGS001-7764	ZNF217	Zinc fingers, C2H2-type			
6667	-85.13	kd	CGS001-23566	LPAR3	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6668	-85.14	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
6669	-85.19	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
6670	-85.24	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
6671	-85.25	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
6672	-85.3	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
6673	-85.33	oe	ccsbBroad304_08480	PNPO	-			
6674	-85.36	cc		Interleukin receptors LOF	-			
6675	-85.37	kd	CGS001-11044	PAPD7	-			
6676	-85.37	kd	CGS001-23081	KDM4C	Histone demethylases			
6677	-85.37	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
6678	-85.48	kd	CGS001-94234	FOXQ1	Forkhead boxes			
6679	-85.52	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
6680	-85.54	cc		SMAD family LOF	-			
6681	-85.55	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
6682	-85.56	oe	ccsbBroad304_05194	LIPH	-			
6683	-85.56	kd	CGS001-5693	PSMB5	Proteasome subunits			
6684	-85.58	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
6685	-85.63	kd	CGS001-85442	KNDC1	-			
6686	-85.66	oe	ccsbBroad304_14047	TACC3	-			
6687	-85.67	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
6688	-85.67	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
6689	-85.67	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
6690	-85.69	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
6691	-85.7	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6692	-85.73	kd	CGS001-5723	PSPH	-			
6693	-85.74	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
6694	-85.74	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
6695	-85.83	cc		Proteasome Pathway LOF	-			
6696	-85.87	oe	ccsbBroad304_05887	CFB	Complement system			
6697	-85.91	oe	ccsbBroad304_00430	GADD45A	-			
6698	-85.91	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
6699	-85.96	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
6700	-86	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
6701	-86	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
6702	-86.02	oe	ccsbBroad304_07491	IP6K1	-			
6703	-86.02	cp	BRD-A92630576	trimebutine	Opioid receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Opioid receptor agonist
6704	-86.02	kd	CGS001-2781	GNAZ	-			
6705	-86.03	oe	ccsbBroad304_07800	EXOSC8	-			
6706	-86.03	kd	CGS001-5562	PRKAA1	AMPK subfamily			
6707	-86.07	oe	ccsbBroad304_01146	PARN	-			
6708	-86.19	kd	CGS001-3312	HSPA8	Heat shock proteins / HSP70			
6709	-86.26	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
6710	-86.28	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6711	-86.29	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
6712	-86.39	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
6713	-86.44	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
6714	-86.48	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
6715	-86.48	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
6716	-86.49	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
6717	-86.51	kd	CGS001-55631	LRRC40	-			
6718	-86.52	kd	CGS001-8702	B4GALT4	Beta 4-glycosyltransferases			
6719	-86.54	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
6720	-86.56	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
6721	-86.57	kd	CGS001-206358	SLC36A1	SLC36 family of proton-coupled amino acid transporters			
6722	-86.66	oe	ccsbBroad304_06985	SORD	-			
6723	-86.66	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
6724	-86.67	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
6725	-86.72	oe	ccsbBroad304_07548	TSSC4	-			
6726	-86.72	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
6727	-86.73	kd	CGS001-6595	SMARCA2	Non-enzymatic BRD containing proteins			
6728	-86.74	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6729	-86.77	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
6730	-86.78	kd	CGS001-2037	EPB41L2	-			
6731	-86.79	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
6732	-86.8	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
6733	-86.87	cp	BRD-K19462402	buflomedil	Adrenergic receptor antagonist		CACNA1C	Adrenergic receptor antagonist, Calcium channel blocker
6734	-86.89	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
6735	-86.9	oe	ccsbBroad304_02285	MED6	-			
6736	-86.9	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
6737	-86.92	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
6738	-86.95	cp	BRD-K96471533	nitazoxanide	Pyruvate ferredoxin oxidoreductase inhibitor			Pyruvate ferredoxin oxidoreductase inhibitor
6739	-87.02	kd	CGS001-56647	BCCIP	-			
6740	-87.07	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
6741	-87.07	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
6742	-87.1	kd	CGS001-65243	ZNF643	-			
6743	-87.12	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
6744	-87.13	oe	ccsbBroad304_03732	NPDC1	-			
6745	-87.13	kd	CGS001-11182	SLC2A6	Solute carriers			
6746	-87.18	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
6747	-87.19	oe	ccsbBroad304_00549	FDX1	-			
6748	-87.19	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
6749	-87.28	oe	ccsbBroad304_02581	ASCC3	-			
6750	-87.28	kd	CGS001-47	ACLY	-			
6751	-87.32	kd	CGS001-2737	GLI3	Zinc fingers, C2H2-type			
6752	-87.34	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
6753	-87.36	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6754	-87.37	kd	CGS001-7321	UBE2D1	Ubiquitin-conjugating enzymes E2			
6755	-87.39	kd	CGS001-5829	PXN	-			
6756	-87.42	cp	BRD-K29530284	amlexanox	Histamine receptor modulator		FGF1, IL3, S100A12, S100A13	Histamine receptor modulator
6757	-87.42	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
6758	-87.44	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
6759	-87.46	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6760	-87.48	oe	ccsbBroad304_05985	CFL1	-			
6761	-87.48	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
6762	-87.49	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
6763	-87.5	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
6764	-87.52	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
6765	-87.52	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
6766	-87.54	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
6767	-87.55	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
6768	-87.55	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
6769	-87.57	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
6770	-87.58	kd	CGS001-2568	GABRP	GABA receptors			
6771	-87.59	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
6772	-87.6	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
6773	-87.62	kd	CGS001-23046	KIF21B	Kinesins			
6774	-87.63	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
6775	-87.64	kd	CGS001-57616	TSHZ3	Teashirt zinc fingers			
6776	-87.65	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
6777	-87.66	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
6778	-87.68	kd	CGS001-4664	NAB1	-			
6779	-87.7	kd	CGS001-6772	STAT1	SH2 domain containing			
6780	-87.72	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
6781	-87.76	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
6782	-87.76	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
6783	-87.8	kd	CGS001-8807	IL18RAP	CD molecules			
6784	-87.86	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
6785	-87.87	kd	CGS001-5901	RAN	-			
6786	-87.88	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
6787	-87.93	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
6788	-87.93	cp	BRD-K39391626	ethylestrenol	Progesterone receptor agonist		AR	Progesterone receptor agonist
6789	-88.02	oe	ccsbBroad304_02677	PDAP1	-			
6790	-88.02	oe	ccsbBroad304_02838	SDF2L1	-			
6791	-88.04	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
6792	-88.06	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
6793	-88.11	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
6794	-88.14	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
6795	-88.15	kd	CGS001-112812	FDX1L	-			
6796	-88.16	oe	ccsbBroad304_02173	ATG5	-			
6797	-88.18	cc		Calmodulin antagonist	-			
6798	-88.18	oe	ccsbBroad304_08023	EIF2C1	-			
6799	-88.18	kd	CGS001-7027	TFDP1	-			
6800	-88.18	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
6801	-88.2	kd	CGS001-9697	TRAM2	-			
6802	-88.2	kd	CGS001-2852	GPER	-			
6803	-88.23	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
6804	-88.24	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
6805	-88.26	oe	ccsbBroad304_08426	TEX10	-			
6806	-88.27	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6807	-88.31	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
6808	-88.38	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
6809	-88.45	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
6810	-88.46	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
6811	-88.48	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
6812	-88.53	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
6813	-88.56	cc		G2 M Checkpoint LOF	-			
6814	-88.56	oe	ccsbBroad304_04490	RSPH1	-			
6815	-88.61	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
6816	-88.63	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
6817	-88.64	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6818	-88.65	oe	ccsbBroad304_00818	IDH3A	-			
6819	-88.68	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
6820	-88.69	oe	ccsbBroad304_00152	BCAT2	-			
6821	-88.69	kd	CGS001-18	ABAT	GABA turnover			
6822	-88.71	oe	ccsbBroad304_00490	EIF4EBP1	-			
6823	-88.73	kd	CGS001-2277	FIGF	-			
6824	-88.74	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
6825	-88.74	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
6826	-88.75	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
6827	-88.76	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
6828	-88.79	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
6829	-88.8	oe	ccsbBroad304_00115	ASPH	-			
6830	-88.81	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
6831	-88.83	kd	CGS001-9770	RASSF2	-			
6832	-88.88	kd	CGS001-55500	ETNK1	-			
6833	-88.89	kd	CGS001-406	ARNTL	Basic helix-loop-helix proteins			
6834	-88.93	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
6835	-88.93	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
6836	-88.97	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
6837	-88.98	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
6838	-89	kd	CGS001-85004	RERG	-			
6839	-89.06	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
6840	-89.07	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
6841	-89.1	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6842	-89.13	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
6843	-89.15	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
6844	-89.17	cp	BRD-K70358946	aripiprazole	Serotonin receptor agonist		DRD2, HTR1A, HTR2A, HRH1, HTR1B, HTR1D, HTR2C, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR1E, HTR3A, HTR6, HTR7	Serotonin receptor agonist, Serotonin receptor antagonist
6845	-89.17	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
6846	-89.18	cp	BRD-K94887716	TFMPP	Serotonin receptor agonist			Serotonin receptor agonist, Serotonin receptor antagonist
6847	-89.19	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
6848	-89.21	kd	CGS001-8576	STK16	NAK family			
6849	-89.23	kd	CGS001-10544	PROCR	CD molecules			
6850	-89.25	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
6851	-89.27	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
6852	-89.3	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
6853	-89.32	kd	CGS001-5373	PMM2	-			
6854	-89.32	kd	CGS001-79581	GPR172A	-			
6855	-89.33	cc		Baculoviral IAP repeat domain containing LOF	-			
6856	-89.36	kd	CGS001-1020	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
6857	-89.37	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
6858	-89.39	cp	BRD-K49668410	clarithromycin	Bacterial 50S ribosomal subunit inhibitor		CYP2C19, CYP3A4, CYP3A5, CYP3A7	Bacterial 50S ribosomal subunit inhibitor
6859	-89.41	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
6860	-89.43	kd	CGS001-955	ENTPD6	-			
6861	-89.43	kd	CGS001-23786	BCL2L13	-			
6862	-89.46	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
6863	-89.48	oe	ccsbBroad304_01271	PPT1	-			
6864	-89.51	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
6865	-89.57	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
6866	-89.63	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
6867	-89.63	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
6868	-89.64	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
6869	-89.66	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
6870	-89.69	kd	CGS001-960	CD44	CD molecules			
6871	-89.71	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
6872	-89.73	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
6873	-89.78	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
6874	-89.82	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
6875	-89.82	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
6876	-89.84	oe	ccsbBroad304_02045	BUD31	-			
6877	-89.89	kd	CGS001-26574	AATF	-			
6878	-89.91	oe	ccsbBroad304_06538	LSP1	-			
6879	-89.92	kd	CGS001-10557	RPP38	-			
6880	-89.95	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
6881	-89.96	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
6882	-90.06	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
6883	-90.06	kd	CGS001-400	ARL1	ADP-ribosylation factors			
6884	-90.07	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
6885	-90.07	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
6886	-90.08	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
6887	-90.12	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
6888	-90.17	oe	ccsbBroad304_06569	MCM5	-			
6889	-90.17	kd	CGS001-7292	TNFSF4	CD molecules			
6890	-90.26	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
6891	-90.29	kd	CGS001-3988	LIPA	-			
6892	-90.3	kd	CGS001-7172	TPMT	-			
6893	-90.31	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
6894	-90.32	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
6895	-90.33	oe	ccsbBroad304_01147	PC	Carboxylases			
6896	-90.35	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
6897	-90.36	kd	CGS001-27102	EIF2AK1	Other PEK family kinases			
6898	-90.39	cc		Benzodiazepine receptor agonist	-			
6899	-90.39	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
6900	-90.39	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
6901	-90.42	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
6902	-90.42	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
6903	-90.43	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
6904	-90.43	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
6905	-90.44	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
6906	-90.44	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
6907	-90.46	kd	CGS001-84619	ZGPAT	G patch domain containing			
6908	-90.48	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
6909	-90.51	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
6910	-90.59	kd	CGS001-5744	PTHLH	Endogenous ligands			
6911	-90.61	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
6912	-90.62	cc		IKK inhibitor	-			
6913	-90.62	kd	CGS001-3985	LIMK2	LIMK subfamily			
6914	-90.63	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
6915	-90.63	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
6916	-90.64	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
6917	-90.65	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
6918	-90.67	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
6919	-90.67	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
6920	-90.69	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6921	-90.71	kd	CGS001-122618	PLD4	-			
6922	-90.72	cc		PDGFR/KIT inhibitor	-			
6923	-90.73	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
6924	-90.73	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
6925	-90.73	kd	CGS001-54915	YTHDF1	-			
6926	-90.75	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
6927	-90.75	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
6928	-90.78	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
6929	-90.85	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6930	-90.92	oe	ccsbBroad304_02804	KLHDC2	-			
6931	-90.95	oe	ccsbBroad304_02862	CCRN4L	-			
6932	-90.98	oe	ccsbBroad304_01862	YEATS4	-			
6933	-90.99	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
6934	-90.99	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
6935	-90.99	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
6936	-91.01	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
6937	-91.03	kd	CGS001-3309	HSPA5	Heat shock proteins / HSP70			
6938	-91.09	oe	ccsbBroad304_02674	STK38	NDR family			
6939	-91.09	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
6940	-91.1	kd	CGS001-1831	TSC22D3	-			
6941	-91.18	kd	CGS001-4968	OGG1	-			
6942	-91.19	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
6943	-91.23	kd	CGS001-6790	AURKA	Aurora kinase			
6944	-91.24	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
6945	-91.24	kd	CGS001-677	ZFP36L1	RING-type (C3HC4) zinc fingers			
6946	-91.25	kd	CGS001-3066	HDAC2	Histone deacetylases			
6947	-91.26	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
6948	-91.26	kd	CGS001-6625	SNRNP70	RNA binding motif (RRM) containing			
6949	-91.28	kd	CGS001-3248	HPGD	Prostaglandin synthases			
6950	-91.31	kd	CGS001-6421	SFPQ	RNA binding motif (RRM) containing			
6951	-91.32	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
6952	-91.35	kd	CGS001-4811	NID1	-			
6953	-91.38	kd	CGS001-5684	PSMA3	Proteasome subunits			
6954	-91.4	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
6955	-91.4	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
6956	-91.42	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
6957	-91.44	kd	CGS001-10051	SMC4	Structural maintenance of chromosomes proteins			
6958	-91.45	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
6959	-91.46	cp	BRD-A20589515	dihydroxyphenylglycine	Glutamate receptor agonist		GRM1	Glutamate receptor agonist
6960	-91.47	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6961	-91.49	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
6962	-91.53	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6963	-91.54	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
6964	-91.54	kd	CGS001-51593	SRRT	-			
6965	-91.55	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
6966	-91.56	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
6967	-91.58	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
6968	-91.61	cp	BRD-K00532621	midazolam	Benzodiazepine receptor agonist		CYP3A5, CYP3A7, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3	Benzodiazepine receptor agonist
6969	-91.65	oe	ccsbBroad304_05763	ACTB	-			
6970	-91.66	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
6971	-91.74	kd	CGS001-6647	SOD1	-			
6972	-91.75	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
6973	-91.79	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
6974	-91.8	oe	ccsbBroad304_00020	ACY1	-			
6975	-91.83	cp	BRD-A95696820	acadesine	AMPK activator			AMPK activator
6976	-91.84	oe	ccsbBroad304_00116	ASS1	-			
6977	-91.85	kd	CGS001-23325	KIAA1033	-			
6978	-91.89	kd	CGS001-6670	SP3	Specificity protein transcription factors			
6979	-91.91	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
6980	-91.91	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
6981	-91.91	kd	CGS001-10921	RNPS1	RNA binding motif (RRM) containing			
6982	-91.95	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
6983	-91.95	kd	CGS001-10190	TXNDC9	-			
6984	-91.96	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
6985	-91.97	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
6986	-91.98	kd	CGS001-7466	WFS1	-			
6987	-91.99	oe	ccsbBroad304_00816	IDE	Pitrilysin			
6988	-92.01	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
6989	-92.04	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
6990	-92.04	kd	CGS001-28960	DCPS	-			
6991	-92.07	oe	ccsbBroad304_00099	ARG2	Arginase			
6992	-92.08	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
6993	-92.08	kd	CGS001-8295	TRRAP	TRRAP subfamily			
6994	-92.1	kd	CGS001-6194	RPS6	S ribosomal proteins			
6995	-92.15	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
6996	-92.18	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
6997	-92.22	kd	CGS001-6303	SAT1	-			
6998	-92.22	kd	CGS001-635	BHMT	-			
6999	-92.23	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
7000	-92.25	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
7001	-92.27	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
7002	-92.27	kd	CGS001-51182	HSPA14	Heat shock proteins / HSP70			
7003	-92.28	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
7004	-92.29	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
7005	-92.32	kd	CGS001-23118	TAB2	-			
7006	-92.35	cp	BRD-K98493452	honokiol	AKT inhibitor		ALOX5, PTGS1, PTGS2	AKT inhibitor
7007	-92.36	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
7008	-92.4	cc		FOS transcription factor family GOF	-			
7009	-92.4	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
7010	-92.42	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
7011	-92.43	kd	CGS001-9212	AURKB	Aurora kinase			
7012	-92.46	cp	BRD-A39172021	ampiroxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
7013	-92.46	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
7014	-92.49	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
7015	-92.49	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
7016	-92.51	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
7017	-92.51	kd	CGS001-8431	NR0B2	DAX-like receptors			
7018	-92.52	cc		Kruppel like transcription factors LOF	-			
7019	-92.55	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
7020	-92.55	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
7021	-92.55	kd	CGS001-2678	GGT1	CD molecules			
7022	-92.57	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
7023	-92.58	cp	BRD-K81855038	roxatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
7024	-92.59	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
7025	-92.6	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
7026	-92.67	oe	ccsbBroad304_04775	NTAN1	-			
7027	-92.67	oe	ccsbBroad304_02438	FAM3C	-			
7028	-92.68	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
7029	-92.68	oe	ccsbBroad304_06172	EPS8	-			
7030	-92.73	oe	ccsbBroad304_07490	SCRN1	-			
7031	-92.73	kd	CGS001-3329	HSPD1	Heat Shock Proteins / Chaperonins			
7032	-92.74	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
7033	-92.75	kd	CGS001-3615	IMPDH2	Oxidoreductases			
7034	-92.77	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
7035	-92.79	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
7036	-92.81	kd	CGS001-253260	RICTOR	-			
7037	-92.82	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
7038	-92.84	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
7039	-92.87	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
7040	-92.87	kd	CGS001-115650	TNFRSF13C	Tumour necrosis factor (TNF) receptor family			
7041	-92.91	kd	CGS001-57215	THAP11	THAP (C2CH-type zinc finger) domain containing			
7042	-92.93	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
7043	-92.93	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
7044	-92.96	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
7045	-92.96	kd	CGS001-81544	GDPD5	-			
7046	-92.97	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
7047	-92.97	oe	ccsbBroad304_06639	NFYB	-			
7048	-92.97	kd	CGS001-9308	CD83	CD molecules			
7049	-92.99	oe	ccsbBroad304_08325	LIPT1	-			
7050	-92.99	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
7051	-93	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
7052	-93.01	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
7053	-93.02	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
7054	-93.03	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
7055	-93.04	oe	ccsbBroad304_09503	KLHDC9	-			
7056	-93.04	kd	CGS001-1508	CTSB	Cathepsins			
7057	-93.04	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
7058	-93.09	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7059	-93.1	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
7060	-93.11	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
7061	-93.14	cp	BRD-A43082555	loxoprofen	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
7062	-93.15	kd	CGS001-55486	PARL	-			
7063	-93.18	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
7064	-93.19	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
7065	-93.2	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
7066	-93.2	kd	CGS001-55139	ANKZF1	Ankyrin repeat domain containing			
7067	-93.22	kd	CGS001-347736	NME9	-			
7068	-93.23	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
7069	-93.27	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
7070	-93.3	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
7071	-93.3	kd	CGS001-2643	GCH1	-			
7072	-93.33	oe	ccsbBroad304_02357	SSX3	-			
7073	-93.35	cc		Heat shock 70kDa proteins LOF	-			
7074	-93.35	oe	ccsbBroad304_14291	GDPD5	-			
7075	-93.38	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
7076	-93.38	kd	CGS001-226	ALDOA	-			
7077	-93.39	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
7078	-93.39	cp	BRD-K48932581	cetraxate	Mucus protecting agent		GAST	Mucus protecting agent
7079	-93.42	kd	CGS001-9443	MED7	-			
7080	-93.45	cc		Structural maintenance of chromosomes proteins LOF	-			
7081	-93.45	kd	CGS001-10616	RBCK1	RING-type (C3HC4) zinc fingers			
7082	-93.46	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
7083	-93.5	oe	ccsbBroad304_06718	PFN2	-			
7084	-93.5	oe	ccsbBroad304_00070	ANXA5	Annexins			
7085	-93.51	kd	CGS001-3945	LDHB	-			
7086	-93.53	cc		Zinc fingers RanBP2 type LOF	-			
7087	-93.53	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
7088	-93.58	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
7089	-93.59	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
7090	-93.61	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
7091	-93.63	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
7092	-93.63	cp	BRD-K47278471	diphenhydramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
7093	-93.63	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
7094	-93.67	kd	CGS001-2172	FABP6	Fatty acid binding protein family			
7095	-93.68	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
7096	-93.68	kd	CGS001-7879	RAB7A	RAB, member RAS oncogene			
7097	-93.69	oe	ccsbBroad304_03798	PHTF2	-			
7098	-93.7	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
7099	-93.7	oe	ccsbBroad304_00832	IFNB1	Interferons			
7100	-93.71	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
7101	-93.74	kd	CGS001-2771	GNAI2	-			
7102	-93.75	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
7103	-93.75	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
7104	-93.75	kd	CGS001-9531	BAG3	-			
7105	-93.76	oe	ccsbBroad304_13998	PDXK	-			
7106	-93.78	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
7107	-93.78	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
7108	-93.81	kd	CGS001-6632	SNRPD1	-			
7109	-93.82	kd	CGS001-84936	ZFYVE19	Zinc fingers, FYVE domain containing			
7110	-93.84	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
7111	-93.84	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
7112	-93.84	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
7113	-93.85	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
7114	-93.86	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
7115	-93.86	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
7116	-93.87	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
7117	-93.88	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
7118	-93.91	oe	ccsbBroad304_01180	PFKFB3	-			
7119	-93.93	cp	BRD-K33312228	halometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
7120	-94	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
7121	-94	oe	ccsbBroad304_02484	PAICS	-			
7122	-94.02	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
7123	-94.02	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
7124	-94.02	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
7125	-94.04	oe	ccsbBroad304_00600	FYN	Src family			
7126	-94.04	kd	CGS001-1155	TBCB	-			
7127	-94.04	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
7128	-94.04	kd	CGS001-10671	DCTN6	-			
7129	-94.11	kd	CGS001-1514	CTSL1	-			
7130	-94.13	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
7131	-94.13	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
7132	-94.15	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
7133	-94.15	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
7134	-94.17	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
7135	-94.19	kd	CGS001-11254	SLC6A14	Glycine transporter subfamily			
7136	-94.22	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
7137	-94.23	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
7138	-94.29	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
7139	-94.33	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
7140	-94.35	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
7141	-94.36	oe	ccsbBroad304_00810	HYAL1	-			
7142	-94.36	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
7143	-94.36	kd	CGS001-9761	MLEC	-			
7144	-94.37	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
7145	-94.38	kd	CGS001-5900	RALGDS	-			
7146	-94.39	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
7147	-94.44	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
7148	-94.44	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
7149	-94.47	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
7150	-94.5	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
7151	-94.5	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
7152	-94.51	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
7153	-94.52	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
7154	-94.54	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
7155	-94.54	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
7156	-94.54	kd	CGS001-10626	TRIM16	Tripartite motif containing			
7157	-94.54	kd	CGS001-1645	AKR1C1	Aldo-keto reductases			
7158	-94.55	kd	CGS001-23678	SGK3	SGK family			
7159	-94.58	kd	CGS001-51174	TUBD1	Tubulins			
7160	-94.58	kd	CGS001-388	RHOB	-			
7161	-94.6	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
7162	-94.6	oe	ccsbBroad304_06888	RPN1	-			
7163	-94.6	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
7164	-94.6	kd	CGS001-54512	EXOSC4	-			
7165	-94.61	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
7166	-94.62	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
7167	-94.65	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
7168	-94.66	oe	ccsbBroad304_00238	CCNE1	-			
7169	-94.66	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
7170	-94.67	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7171	-94.7	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
7172	-94.7	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
7173	-94.74	oe	ccsbBroad304_00957	M6PR	-			
7174	-94.75	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
7175	-94.75	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
7176	-94.78	kd	CGS001-54108	CHRAC1	-			
7177	-94.79	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
7178	-94.8	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
7179	-94.8	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
7180	-94.81	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
7181	-94.82	oe	ccsbBroad304_00728	HBE1	-			
7182	-94.83	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
7183	-94.84	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
7184	-94.85	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
7185	-94.88	oe	ccsbBroad304_02890	SYF2	-			
7186	-94.88	oe	ccsbBroad304_02716	NMNAT2	-			
7187	-94.88	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
7188	-94.89	kd	CGS001-1717	DHCR7	-			
7189	-94.9	oe	ccsbBroad304_09833	SENP5	-			
7190	-94.91	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
7191	-94.91	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
7192	-94.91	kd	CGS001-55379	LRRC59	-			
7193	-94.98	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
7194	-95.01	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
7195	-95.03	kd	CGS001-9851	KIAA0753	-			
7196	-95.03	kd	CGS001-1875	E2F5	-			
7197	-95.05	kd	CGS001-558	AXL	Fibronectin type III domain containing			
7198	-95.09	oe	ccsbBroad304_01164	PDHB	-			
7199	-95.1	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
7200	-95.11	oe	ccsbBroad304_08266	PIPOX	-			
7201	-95.12	cc		Vesicular Transport LOF	-			
7202	-95.12	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
7203	-95.13	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
7204	-95.16	kd	CGS001-54659	UGT1A3	UDP glucuronosyltransferases			
7205	-95.17	kd	CGS001-2079	ERH	-			
7206	-95.18	kd	CGS001-54205	CYCS	-			
7207	-95.19	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
7208	-95.19	oe	ccsbBroad304_04534	HN1L	-			
7209	-95.21	kd	CGS001-4234	METTL1	-			
7210	-95.22	kd	CGS001-57396	CLK4	CDC-like kinases			
7211	-95.23	cp	BRD-K86887724	dofetilide	Potassium channel blocker		KCNH2, KCNH1, KCNJ12, KCNK2	Potassium channel blocker
7212	-95.24	kd	CGS001-56916	SMARCAD1	-			
7213	-95.25	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
7214	-95.28	kd	CGS001-6129	RPL7	L ribosomal proteins			
7215	-95.32	oe	ccsbBroad304_06976	SMARCE1	-			
7216	-95.33	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
7217	-95.33	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
7218	-95.36	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
7219	-95.37	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
7220	-95.39	oe	ccsbBroad304_08346	COQ3	-			
7221	-95.39	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
7222	-95.39	kd	CGS001-5796	PTPRK	Receptor tyrosine phosphatases (RTP)			
7223	-95.4	kd	CGS001-80025	PANK2	-			
7224	-95.42	kd	CGS001-6207	RPS13	S ribosomal proteins			
7225	-95.46	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
7226	-95.47	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
7227	-95.49	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
7228	-95.51	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
7229	-95.52	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
7230	-95.55	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
7231	-95.55	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
7232	-95.57	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
7233	-95.57	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
7234	-95.57	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
7235	-95.57	kd	CGS001-3590	IL11RA	IL-6 receptor family			
7236	-95.59	kd	CGS001-51752	ERAP1	Aminopeptidase N			
7237	-95.6	kd	CGS001-8717	TRADD	-			
7238	-95.62	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
7239	-95.62	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
7240	-95.63	oe	ccsbBroad304_00888	ITPK1	-			
7241	-95.63	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
7242	-95.63	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7243	-95.63	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
7244	-95.64	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
7245	-95.67	kd	CGS001-3476	IGBP1	-			
7246	-95.68	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
7247	-95.68	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
7248	-95.69	kd	CGS001-26271	FBXO5	F-boxes / other			
7249	-95.69	kd	CGS001-11325	DDX42	DEAD-boxes			
7250	-95.72	kd	CGS001-84969	TOX2	-			
7251	-95.75	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
7252	-95.75	kd	CGS001-5245	PHB	-			
7253	-95.76	kd	CGS001-100	ADA	Adenosine turnover			
7254	-95.77	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
7255	-95.77	oe	ccsbBroad304_01222	PLP2	-			
7256	-95.78	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
7257	-95.8	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
7258	-95.82	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
7259	-95.83	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
7260	-95.84	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
7261	-95.86	kd	CGS001-54861	SNRK	SNRK subfamily			
7262	-95.91	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
7263	-95.94	oe	ccsbBroad304_00237	CCND3	-			
7264	-95.94	kd	CGS001-23196	FAM120A	-			
7265	-95.96	kd	CGS001-4610	MYCL1	-			
7266	-95.98	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
7267	-95.99	kd	CGS001-55120	FANCL	Fanconi anemia, complementation groups			
7268	-96.01	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
7269	-96.01	kd	CGS001-51466	EVL	-			
7270	-96.04	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
7271	-96.05	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
7272	-96.06	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
7273	-96.1	kd	CGS001-8192	CLPP	ATPases / AAA-type			
7274	-96.12	kd	CGS001-9813	KIAA0494	-			
7275	-96.14	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
7276	-96.14	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
7277	-96.14	kd	CGS001-1312	COMT	Catecholamine turnover			
7278	-96.15	kd	CGS001-27076	LYPD3	-			
7279	-96.16	cp	BRD-K22227508	targinine	Nitric oxide synthase inhibitor		NOS2, NOS3	Nitric oxide synthase inhibitor
7280	-96.16	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
7281	-96.2	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
7282	-96.2	oe	ccsbBroad304_02956	EHF	-			
7283	-96.2	kd	CGS001-3431	SP110	Non-enzymatic BRD containing proteins			
7284	-96.21	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
7285	-96.22	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
7286	-96.24	kd	CGS001-9712	USP6NL	-			
7287	-96.24	kd	CGS001-5986	RFNG	Beta 3-glycosyltransferases			
7288	-96.24	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
7289	-96.25	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
7290	-96.26	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
7291	-96.27	cc		T-type calcium channel blocker	-			
7292	-96.27	kd	CGS001-28511	NKIRAS2	-			
7293	-96.27	kd	CGS001-4191	MDH2	-			
7294	-96.27	kd	CGS001-3575	IL7R	IL-2 receptor family			
7295	-96.28	cp	BRD-K73196317	urapidil	Adrenergic receptor antagonist		HTR1A	Adrenergic receptor antagonist
7296	-96.29	kd	CGS001-1950	EGF	-			
7297	-96.3	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
7298	-96.3	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
7299	-96.31	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
7300	-96.31	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
7301	-96.33	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7302	-96.34	kd	CGS001-4953	ODC1	Decarboxylases			
7303	-96.34	kd	CGS001-8893	EIF2B5	-			
7304	-96.35	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
7305	-96.35	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
7306	-96.36	oe	ccsbBroad304_00510	EPHX2	-			
7307	-96.37	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
7308	-96.39	kd	CGS001-3313	HSPA9	Heat shock proteins / HSP70			
7309	-96.42	oe	ccsbBroad304_09095	PUS7L	-			
7310	-96.42	kd	CGS001-10645	CAMKK2	Meta subfamily			
7311	-96.42	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
7312	-96.42	kd	CGS001-433	ASGR2	C-type lectin domain containing			
7313	-96.43	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
7314	-96.43	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
7315	-96.44	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
7316	-96.44	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
7317	-96.45	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
7318	-96.48	cp	BRD-A68888262	azelastine	Histamine receptor antagonist		HRH1, CYP2C19	Histamine receptor antagonist
7319	-96.49	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
7320	-96.5	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
7321	-96.52	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
7322	-96.52	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
7323	-96.52	cp	BRD-K81169441	cerivastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A5	HMGCR inhibitor
7324	-96.52	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
7325	-96.53	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
7326	-96.56	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
7327	-96.58	oe	ccsbBroad304_07337	TAF1B	-			
7328	-96.58	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
7329	-96.58	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
7330	-96.59	kd	CGS001-5664	PSEN2	Presenilin			
7331	-96.6	kd	CGS001-4200	ME2	-			
7332	-96.61	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
7333	-96.62	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
7334	-96.63	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
7335	-96.65	cp	BRD-K92413528	thiazolidinecarboxylic-acid	Reducing agent			Reducing agent
7336	-96.65	kd	CGS001-54957	TXNL4B	-			
7337	-96.67	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
7338	-96.67	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
7339	-96.67	kd	CGS001-10254	STAM2	-			
7340	-96.69	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
7341	-96.69	kd	CGS001-7358	UGDH	-			
7342	-96.7	cc		IL4 Pathway LOF	-			
7343	-96.7	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
7344	-96.72	kd	CGS001-10915	TCERG1	-			
7345	-96.72	kd	CGS001-896	CCND3	-			
7346	-96.74	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
7347	-96.76	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
7348	-96.76	cp	BRD-K06388322	pramipexole	Dopamine receptor agonist		DRD3, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
7349	-96.76	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
7350	-96.77	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
7351	-96.78	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
7352	-96.78	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
7353	-96.8	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
7354	-96.8	kd	CGS001-191	AHCY	Adenosine turnover			
7355	-96.82	cp	BRD-K54316499	tolterodine	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRM1, CHRM4, CHRM5	Acetylcholine receptor antagonist
7356	-96.83	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
7357	-96.83	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
7358	-96.86	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
7359	-96.88	oe	ccsbBroad304_03767	TOMM22	-			
7360	-96.88	oe	ccsbBroad304_07834	GGA2	-			
7361	-96.89	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
7362	-96.89	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
7363	-96.89	kd	CGS001-440	ASNS	-			
7364	-96.9	oe	ccsbBroad304_07889	QPRT	-			
7365	-96.9	kd	CGS001-3670	ISL1	Homeoboxes / LIM class			
7366	-96.91	cc		Nucleoporin LOF	-			
7367	-96.91	cp	BRD-A64297288	amlodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, ABCG2, CA1, CACNA1B, CACNA1S, CACNA2D3, CACNB1, CACNB2, SMPD1	Calcium channel blocker
7368	-96.91	kd	CGS001-9451	EIF2AK3	PEK subfamily			
7369	-96.92	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
7370	-96.93	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
7371	-96.93	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
7372	-96.94	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
7373	-96.94	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
7374	-96.94	cp	BRD-K88679075	methandriol	Androgenic steroid			Androgenic steroid
7375	-96.97	oe	ccsbBroad304_01663	TFF2	-			
7376	-96.97	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
7377	-96.98	kd	CGS001-4708	NDUFB2	Mitochondrial respiratory chain complex / Complex I			
7378	-97.01	kd	CGS001-5025	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
7379	-97.02	kd	CGS001-9406	ZRANB2	Zinc fingers, RAN-binding domain containing			
7380	-97.03	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
7381	-97.03	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
7382	-97.04	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
7383	-97.04	oe	ccsbBroad304_01855	NCOA4	-			
7384	-97.05	cp	BRD-K49481516	galantamine	Acetylcholinesterase inhibitor		ACHE, BCHE, CHRNA1, CHRNA10, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNA9, CHRNB1, CHRNB2, CHRNB3, CHRNB4, CHRND, CHRNE, CHRNG	Acetylcholinesterase inhibitor
7385	-97.06	cp	BRD-A12560204	nitrendipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1H, CACNA1S, CACNA2D2, CACNB2, CACNG1, KCNN4	Calcium channel blocker
7386	-97.08	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
7387	-97.09	kd	CGS001-6591	SNAI2	Snail homologs			
7388	-97.09	kd	CGS001-8031	NCOA4	-			
7389	-97.11	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
7390	-97.12	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
7391	-97.13	kd	CGS001-25989	ULK3	Unc-51-like kinase (ULK) family			
7392	-97.14	kd	CGS001-10460	TACC3	-			
7393	-97.14	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
7394	-97.15	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
7395	-97.15	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
7396	-97.15	kd	CGS001-89910	UBE3B	-			
7397	-97.17	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
7398	-97.18	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
7399	-97.18	kd	CGS001-3775	KCNK1	Two-P potassium channels			
7400	-97.18	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
7401	-97.19	kd	CGS001-90861	HN1L	-			
7402	-97.2	oe	ccsbBroad304_05980	CDKN1B	-			
7403	-97.2	kd	CGS001-11333	PDAP1	-			
7404	-97.22	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
7405	-97.22	kd	CGS001-6500	SKP1	-			
7406	-97.22	kd	CGS001-387	RHOA	-			
7407	-97.23	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
7408	-97.24	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
7409	-97.24	oe	ccsbBroad304_00809	HUS1	-			
7410	-97.24	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
7411	-97.24	kd	CGS001-8525	DGKZ	-			
7412	-97.25	cc		DNA dependent protein kinase inhibitor	-			
7413	-97.25	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
7414	-97.25	kd	CGS001-64167	ERAP2	Aminopeptidase N			
7415	-97.26	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
7416	-97.28	oe	ccsbBroad304_03652	EXOC2	-			
7417	-97.29	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
7418	-97.29	cp	BRD-K84955386	hyperoside	Glucosidase inhibitor		ACE, AKR1B1, GAA	Glucosidase inhibitor
7419	-97.29	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
7420	-97.31	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
7421	-97.32	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
7422	-97.32	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
7423	-97.33	oe	ccsbBroad304_01413	RPA2	-			
7424	-97.33	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
7425	-97.34	oe	ccsbBroad304_00960	SMAD1	SMADs			
7426	-97.34	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
7427	-97.34	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
7428	-97.34	kd	CGS001-5777	PTPN6	Protein tyrosine phosphatases			
7429	-97.35	kd	CGS001-6418	SET	-			
7430	-97.35	oe	ccsbBroad304_02138	TRIP10	-			
7431	-97.39	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
7432	-97.4	kd	CGS001-56998	CTNNBIP1	Catenins			
7433	-97.42	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
7434	-97.42	kd	CGS001-55620	STAP2	-			
7435	-97.42	kd	CGS001-7849	PAX8	Paired boxes			
7436	-97.43	kd	CGS001-8834	TMEM11	-			
7437	-97.43	kd	CGS001-6894	TARBP1	-			
7438	-97.45	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
7439	-97.46	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
7440	-97.49	kd	CGS001-91433	RCCD1	-			
7441	-97.49	kd	CGS001-7913	DEK	-			
7442	-97.49	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
7443	-97.52	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
7444	-97.53	cp	BRD-K88304388	dextrorphan	Glutamate receptor antagonist		OPRM1, OPRK1, OPRD1, GRIN1, HTR1A, SLC6A2	Glutamate receptor antagonist
7445	-97.53	kd	CGS001-6337	SCNN1A	Epithelial sodium channels (ENaC)			
7446	-97.54	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
7447	-97.54	kd	CGS001-9124	PDLIM1	-			
7448	-97.54	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
7449	-97.55	cc		LIM class homeoboxes GOF	-			
7450	-97.56	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7451	-97.58	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
7452	-97.58	kd	CGS001-1453	CSNK1D	Casein kinase 1 (CK1) family			
7453	-97.59	kd	CGS001-9688	NUP93	-			
7454	-97.59	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
7455	-97.59	kd	CGS001-8915	BCL10	-			
7456	-97.61	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
7457	-97.61	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
7458	-97.62	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
7459	-97.63	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
7460	-97.63	oe	ccsbBroad304_00518	ETFA	-			
7461	-97.64	kd	CGS001-23239	PHLPP1	Pleckstrin homology (PH) domain containing			
7462	-97.64	kd	CGS001-9275	BCL7B	-			
7463	-97.66	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
7464	-97.67	kd	CGS001-7037	TFRC	CD molecules			
7465	-97.69	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
7466	-97.7	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
7467	-97.71	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
7468	-97.73	oe	ccsbBroad304_00515	ERH	-			
7469	-97.73	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
7470	-97.73	kd	CGS001-3693	ITGB5	Integrins			
7471	-97.73	kd	CGS001-8837	CFLAR	Endogenous ligands			
7472	-97.74	oe	ccsbBroad304_03264	UBAP1	-			
7473	-97.74	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
7474	-97.75	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
7475	-97.75	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
7476	-97.75	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7477	-97.76	cc		DNA polymerase inhibitor	-			
7478	-97.76	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
7479	-97.76	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
7480	-97.77	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
7481	-97.77	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
7482	-97.77	cp	BRD-K46435977	valaciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
7483	-97.78	cc		Potassium channel blocker	-			
7484	-97.78	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
7485	-97.79	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
7486	-97.8	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
7487	-97.8	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
7488	-97.82	cc		Bacterial cell wall synthesis inhibitor	-			
7489	-97.84	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
7490	-97.85	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
7491	-97.86	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
7492	-97.86	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
7493	-97.86	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
7494	-97.86	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
7495	-97.87	kd	CGS001-9453	GGPS1	Lanosterol biosynthesis pathway			
7496	-97.89	cp	BRD-K83144676	olmesartan	Angiotensin antagonist		AGTR1	Angiotensin antagonist
7497	-97.91	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
7498	-97.92	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
7499	-97.94	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
7500	-97.94	oe	ccsbBroad304_00398	CTSL2	-			
7501	-97.94	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
7502	-97.95	oe	ccsbBroad304_03640	CEP72	-			
7503	-97.95	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
7504	-97.95	oe	ccsbBroad304_05936	CASP2	Caspases			
7505	-97.96	kd	CGS001-219333	USP12	Ubiquitin-specific peptidases			
7506	-97.98	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
7507	-97.98	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
7508	-97.98	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
7509	-97.99	kd	CGS001-23211	ZC3H4	Zinc fingers, CCCH-type domain containing			
7510	-97.99	kd	CGS001-23475	QPRT	-			
7511	-97.99	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
7512	-98	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
7513	-98.01	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
7514	-98.02	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
7515	-98.03	kd	CGS001-23581	CASP14	Caspases			
7516	-98.04	kd	CGS001-57048	PLSCR3	-			
7517	-98.1	kd	CGS001-23761	PISD	Decarboxylases			
7518	-98.11	oe	ccsbBroad304_08152	PSAT1	-			
7519	-98.13	kd	CGS001-8803	SUCLA2	-			
7520	-98.13	kd	CGS001-805	CALM2	EF-hand domain containing			
7521	-98.14	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
7522	-98.14	kd	CGS001-5366	PMAIP1	-			
7523	-98.15	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
7524	-98.15	kd	CGS001-4067	LYN	Src family			
7525	-98.16	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
7526	-98.16	kd	CGS001-5930	RBBP6	-			
7527	-98.17	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
7528	-98.17	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7529	-98.18	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
7530	-98.18	kd	CGS001-22796	COG2	Components of oligomeric golgi complex			
7531	-98.19	kd	CGS001-3553	IL1B	Interleukins and interleukin receptors			
7532	-98.2	oe	ccsbBroad304_01632	SYPL1	-			
7533	-98.2	kd	CGS001-7185	TRAF1	-			
7534	-98.21	cp	BRD-K85030058	benactyzine	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
7535	-98.22	kd	CGS001-27	ABL2	Abl family			
7536	-98.23	oe	ccsbBroad304_09881	RFX6	-			
7537	-98.23	oe	ccsbBroad304_02789	ADAT1	-			
7538	-98.24	cc		PKA inhibitor	-			
7539	-98.27	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
7540	-98.28	cp	BRD-K60160658	tiagabine	GABA uptake inhibitor		SLC6A1, CYP2C19	GABA uptake inhibitor
7541	-98.29	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
7542	-98.3	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
7543	-98.3	kd	CGS001-2153	F5	Blood coagulation components			
7544	-98.3	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
7545	-98.32	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
7546	-98.35	cc		Proteasome inhibitor	-			
7547	-98.35	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
7548	-98.38	kd	CGS001-4637	MYL6	EF-hand domain containing			
7549	-98.38	kd	CGS001-8446	DUSP11	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7550	-98.39	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
7551	-98.41	kd	CGS001-1662	DDX10	DEAD-boxes			
7552	-98.42	oe	ccsbBroad304_06136	ECHS1	-			
7553	-98.43	oe	ccsbBroad304_02163	MED7	-			
7554	-98.45	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
7555	-98.46	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
7556	-98.46	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
7557	-98.46	kd	CGS001-28969	BZW2	-			
7558	-98.48	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
7559	-98.49	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
7560	-98.49	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
7561	-98.5	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
7562	-98.5	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
7563	-98.51	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
7564	-98.53	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
7565	-98.55	kd	CGS001-54788	DNAJB12	Heat shock proteins / DNAJ (HSP40)			
7566	-98.56	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
7567	-98.56	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
7568	-98.56	kd	CGS001-55765	C1ORF106	-			
7569	-98.57	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
7570	-98.57	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7571	-98.58	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
7572	-98.59	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
7573	-98.59	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
7574	-98.59	oe	ccsbBroad304_04292	INHBE	-			
7575	-98.59	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
7576	-98.6	kd	CGS001-652	BMP4	Bone morphogenetic proteins			
7577	-98.6	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
7578	-98.61	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
7579	-98.61	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
7580	-98.62	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
7581	-98.63	kd	CGS001-55556	ENOSF1	-			
7582	-98.64	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
7583	-98.64	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
7584	-98.64	kd	CGS001-10046	MAMLD1	-			
7585	-98.65	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
7586	-98.66	oe	ccsbBroad304_00072	ANXA7	Annexins			
7587	-98.66	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
7588	-98.67	cc		Kinase anchoring proteins LOF	-			
7589	-98.67	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
7590	-98.68	oe	ccsbBroad304_07466	VGLL4	-			
7591	-98.68	oe	ccsbBroad304_06562	MAT1A	-			
7592	-98.68	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
7593	-98.71	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7594	-98.72	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
7595	-98.72	kd	CGS001-9871	SEC24D	-			
7596	-98.73	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
7597	-98.73	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
7598	-98.73	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
7599	-98.75	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
7600	-98.76	kd	CGS001-50814	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7601	-98.77	cp	BRD-K90733503	cefalexin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7602	-98.77	cp	BRD-K07237224	moclobemide	Monoamine oxidase inhibitor		MAOA, CYP2C19, MAOB	Monoamine oxidase inhibitor
7603	-98.77	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
7604	-98.77	kd	CGS001-2961	GTF2E2	General transcription factors			
7605	-98.78	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
7606	-98.79	kd	CGS001-9833	MELK	MELK subfamily			
7607	-98.8	oe	ccsbBroad304_01933	TEAD2	-			
7608	-98.8	oe	ccsbBroad304_09035	COASY	-			
7609	-98.8	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
7610	-98.8	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
7611	-98.82	kd	CGS001-64080	RBKS	-			
7612	-98.84	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
7613	-98.84	kd	CGS001-2353	FOS	basic leucine zipper proteins			
7614	-98.85	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
7615	-98.86	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
7616	-98.86	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
7617	-98.86	kd	CGS001-6188	RPS3	S ribosomal proteins			
7618	-98.87	cp	BRD-A00520476	otenzepad	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
7619	-98.87	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
7620	-98.88	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
7621	-98.89	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
7622	-98.89	kd	CGS001-8891	EIF2B3	-			
7623	-98.9	kd	CGS001-64121	RRAGC	-			
7624	-98.91	kd	CGS001-2821	GPI	-			
7625	-98.91	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
7626	-98.91	kd	CGS001-378	ARF4	ADP-ribosylation factors			
7627	-98.93	cp	BRD-K10961822	latanoprost	Prostanoid receptor agonist		PTGFR	Prostanoid receptor agonist
7628	-98.93	kd	CGS001-5695	PSMB7	Proteasome subunits			
7629	-98.93	kd	CGS001-3149	HMGB3	High-mobility group / Canonical			
7630	-98.93	kd	CGS001-966	CD59	CD molecules			
7631	-98.94	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
7632	-98.94	kd	CGS001-3420	IDH3B	-			
7633	-98.94	kd	CGS001-64858	DCLRE1B	-			
7634	-98.95	kd	CGS001-116931	MED12L	-			
7635	-98.96	oe	ccsbBroad304_00100	RHOA	-			
7636	-98.96	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
7637	-98.97	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
7638	-98.97	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
7639	-98.98	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
7640	-98.99	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7641	-98.99	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
7642	-99	kd	CGS001-83999	KREMEN1	-			
7643	-99.02	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
7644	-99.02	kd	CGS001-31	ACACA	Carboxylases			
7645	-99.04	oe	ccsbBroad304_00963	SMAD5	SMADs			
7646	-99.04	cp	BRD-K94649603	taxifolin	Opioid receptor antagonist		APOB, APP, HMGCR	Opioid receptor antagonist
7647	-99.05	oe	ccsbBroad304_00249	CD14	CD molecules			
7648	-99.06	kd	CGS001-8639	AOC3	Oxidoreductases			
7649	-99.07	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
7650	-99.07	kd	CGS001-6256	RXRA	Retinoid X receptors			
7651	-99.07	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
7652	-99.08	oe	ccsbBroad304_07814	SACM1L	-			
7653	-99.08	kd	CGS001-6223	RPS19	S ribosomal proteins			
7654	-99.09	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
7655	-99.09	oe	ccsbBroad304_00150	BAX	-			
7656	-99.09	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
7657	-99.09	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
7658	-99.1	kd	CGS001-415116	PIM3	PIM family			
7659	-99.11	oe	ccsbBroad304_00170	BNIP1	-			
7660	-99.11	kd	CGS001-143187	VTI1A	-			
7661	-99.11	kd	CGS001-5763	PTMS	-			
7662	-99.13	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
7663	-99.14	cc		Ribosomal 40s Subunit LOF	-			
7664	-99.14	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
7665	-99.14	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
7666	-99.14	kd	CGS001-93134	ZNF561	Zinc fingers, C2H2-type			
7667	-99.14	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
7668	-99.14	kd	CGS001-5708	PSMD2	Proteasome subunits			
7669	-99.15	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
7670	-99.15	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
7671	-99.15	kd	CGS001-6477	SIAH1	-			
7672	-99.16	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
7673	-99.16	kd	CGS001-7316	UBC	-			
7674	-99.16	kd	CGS001-25824	PRDX5	-			
7675	-99.16	kd	CGS001-10447	FAM3C	-			
7676	-99.17	kd	CGS001-7444	VRK2	Vaccina related kinase (VRK) family			
7677	-99.17	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
7678	-99.18	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
7679	-99.18	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
7680	-99.18	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
7681	-99.18	kd	CGS001-2885	GRB2	SH2 domain containing			
7682	-99.19	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
7683	-99.21	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
7684	-99.21	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
7685	-99.22	oe	ccsbBroad304_07832	XPO7	Exportins			
7686	-99.22	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
7687	-99.22	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
7688	-99.23	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
7689	-99.23	kd	CGS001-11136	SLC7A9	SLC7 family			
7690	-99.23	kd	CGS001-2114	ETS2	ETS Transcription Factors			
7691	-99.24	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
7692	-99.26	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
7693	-99.26	kd	CGS001-8942	KYNU	-			
7694	-99.26	oe	ccsbBroad304_01618	STXBP1	-			
7695	-99.27	kd	CGS001-4522	MTHFD1	-			
7696	-99.27	kd	CGS001-79094	CHAC1	-			
7697	-99.28	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
7698	-99.28	kd	CGS001-5891	MOK	RCK family			
7699	-99.28	kd	CGS001-2588	GALNS	Arylsulfatase family			
7700	-99.29	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
7701	-99.29	kd	CGS001-1362	CPD	Carboxypeptidase A			
7702	-99.3	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
7703	-99.3	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
7704	-99.3	kd	CGS001-5371	PML	RING-type (C3HC4) zinc fingers			
7705	-99.3	kd	CGS001-472	ATM	Other PIKK family kinases			
7706	-99.3	kd	CGS001-39	ACAT2	Lanosterol biosynthesis pathway			
7707	-99.31	oe	ccsbBroad304_08365	CYCS	-			
7708	-99.31	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
7709	-99.31	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
7710	-99.31	oe	ccsbBroad304_06253	GALT	-			
7711	-99.32	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
7712	-99.32	kd	CGS001-9143	SYNGR3	-			
7713	-99.33	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
7714	-99.33	kd	CGS001-5480	PPIC	-			
7715	-99.33	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
7716	-99.34	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
7717	-99.34	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
7718	-99.34	kd	CGS001-7357	UGCG	Glycosyltransferase family 2 domain containing			
7719	-99.34	kd	CGS001-10797	MTHFD2	-			
7720	-99.35	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
7721	-99.35	kd	CGS001-3672	ITGA1	Integrins			
7722	-99.36	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
7723	-99.36	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
7724	-99.36	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
7725	-99.36	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
7726	-99.36	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
7727	-99.36	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
7728	-99.37	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7729	-99.37	kd	CGS001-79073	TMEM109	-			
7730	-99.38	kd	CGS001-1399	CRKL	SH2 domain containing			
7731	-99.39	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
7732	-99.39	kd	CGS001-6919	TCEA2	-			
7733	-99.39	kd	CGS001-5211	PFKL	-			
7734	-99.39	kd	CGS001-5105	PCK1	-			
7735	-99.39	kd	CGS001-4485	MST1	-			
7736	-99.39	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
7737	-99.4	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
7738	-99.4	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
7739	-99.4	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
7740	-99.4	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
7741	-99.4	kd	CGS001-6208	RPS14	S ribosomal proteins			
7742	-99.4	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
7743	-99.4	kd	CGS001-11215	AKAP11	A-kinase anchor proteins			
7744	-99.42	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
7745	-99.42	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
7746	-99.42	kd	CGS001-661	POLR3D	RNA polymerase subunits			
7747	-99.42	kd	CGS001-23658	LSM5	-			
7748	-99.44	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
7749	-99.45	oe	ccsbBroad304_09284	UBE3B	-			
7750	-99.45	oe	ccsbBroad304_00423	DAXX	-			
7751	-99.45	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
7752	-99.45	kd	CGS001-25888	ZNF473	Zinc fingers, C2H2-type			
7753	-99.46	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
7754	-99.46	kd	CGS001-6201	RPS7	S ribosomal proteins			
7755	-99.47	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
7756	-99.47	kd	CGS001-55176	SEC61A2	-			
7757	-99.47	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
7758	-99.47	kd	CGS001-673	BRAF	RAF family			
7759	-99.48	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
7760	-99.48	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
7761	-99.48	kd	CGS001-10898	CPSF4	-			
7762	-99.49	oe	ccsbBroad304_01084	NEU1	-			
7763	-99.5	oe	ccsbBroad304_07662	NPRL2	-			
7764	-99.5	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
7765	-99.5	kd	CGS001-2768	GNA12	-			
7766	-99.5	kd	CGS001-1725	DHPS	-			
7767	-99.5	kd	CGS001-6936	C2ORF3	-			
7768	-99.51	kd	CGS001-1062	CENPE	Kinesins			
7769	-99.52	kd	CGS001-64921	CASD1	-			
7770	-99.53	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
7771	-99.53	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
7772	-99.53	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
7773	-99.53	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
7774	-99.54	oe	ccsbBroad304_00645	GCLM	-			
7775	-99.54	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
7776	-99.54	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
7777	-99.54	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
7778	-99.54	kd	CGS001-2634	GBP2	-			
7779	-99.54	kd	CGS001-9337	CNOT8	-			
7780	-99.55	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
7781	-99.55	cp	BRD-K13664374	dichloroacetic-acid	Pyruvate dehydrogenase kinase inhibitor		PDK1	Pyruvate dehydrogenase kinase inhibitor
7782	-99.55	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
7783	-99.55	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
7784	-99.55	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
7785	-99.56	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
7786	-99.56	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
7787	-99.56	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
7788	-99.56	kd	CGS001-10975	UQCR11	Mitochondrial respiratory chain complex / Complex III			
7789	-99.56	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
7790	-99.58	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
7791	-99.59	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
7792	-99.59	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
7793	-99.6	oe	ccsbBroad304_08452	PIH1D1	-			
7794	-99.61	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
7795	-99.61	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
7796	-99.61	kd	CGS001-2224	FDPS	Lanosterol biosynthesis pathway			
7797	-99.62	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
7798	-99.62	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
7799	-99.62	kd	CGS001-8624	PSMG1	-			
7800	-99.62	kd	CGS001-11142	PKIG	-			
7801	-99.62	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
7802	-99.62	kd	CGS001-665	BNIP3L	-			
7803	-99.63	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
7804	-99.64	oe	ccsbBroad304_07124	UROD	-			
7805	-99.64	kd	CGS001-1655	DDX5	DEAD-boxes			
7806	-99.65	oe	ccsbBroad304_03554	NAT10	-			
7807	-99.66	oe	ccsbBroad304_02565	RALBP1	-			
7808	-99.66	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
7809	-99.66	kd	CGS001-27161	EIF2C2	-			
7810	-99.66	kd	CGS001-80777	CYB5B	-			
7811	-99.66	kd	CGS001-55832	CAND1	-			
7812	-99.68	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
7813	-99.68	kd	CGS001-4938	OAS1	-			
7814	-99.68	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
7815	-99.7	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
7816	-99.7	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
7817	-99.7	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
7818	-99.7	kd	CGS001-23075	SWAP70	EF-hand domain containing			
7819	-99.7	kd	CGS001-6646	SOAT1	-			
7820	-99.71	cc		Ubiquitin-specific peptidases LOF	-			
7821	-99.71	kd	CGS001-9958	USP15	Ubiquitin-specific peptidases			
7822	-99.71	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
7823	-99.72	oe	ccsbBroad304_06386	HNMT	-			
7824	-99.72	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
7825	-99.72	kd	CGS001-390980	ZNF805	Zinc fingers, C2H2-type			
7826	-99.73	oe	ccsbBroad304_01577	SOD1	-			
7827	-99.73	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
7828	-99.73	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
7829	-99.73	kd	CGS001-9341	VAMP3	Vesicle-associated membrane proteins			
7830	-99.73	kd	CGS001-2235	FECH	-			
7831	-99.73	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
7832	-99.74	oe	ccsbBroad304_08879	CASD1	-			
7833	-99.74	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
7834	-99.74	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
7835	-99.74	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
7836	-99.74	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
7837	-99.74	kd	CGS001-2030	SLC29A1	SLC29 family			
7838	-99.74	kd	CGS001-3685	ITGAV	Integrins			
7839	-99.74	kd	CGS001-2539	G6PD	-			
7840	-99.74	kd	CGS001-1212	CLTB	-			
7841	-99.75	oe	ccsbBroad304_00961	SMAD2	SMADs			
7842	-99.76	oe	ccsbBroad304_03555	PANK4	-			
7843	-99.76	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
7844	-99.76	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
7845	-99.76	kd	CGS001-26191	PTPN22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
7846	-99.76	kd	CGS001-10943	MSL3	-			
7847	-99.76	kd	CGS001-929	CD14	CD molecules			
7848	-99.77	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
7849	-99.77	kd	CGS001-5927	KDM5A	Histone demethylases			
7850	-99.77	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
7851	-99.77	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
7852	-99.78	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7853	-99.78	kd	CGS001-51024	FIS1	-			
7854	-99.78	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
7855	-99.78	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
7856	-99.79	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
7857	-99.79	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
7858	-99.79	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
7859	-99.79	kd	CGS001-9270	ITGB1BP1	-			
7860	-99.79	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
7861	-99.8	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
7862	-99.81	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
7863	-99.81	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
7864	-99.81	kd	CGS001-1728	NQO1	-			
7865	-99.81	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
7866	-99.82	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
7867	-99.82	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
7868	-99.82	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
7869	-99.83	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
7870	-99.83	kd	CGS001-51465	UBE2J1	Ubiquitin-conjugating enzymes E2			
7871	-99.83	kd	CGS001-5387	PMS2P3	-			
7872	-99.84	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
7873	-99.84	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
7874	-99.84	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
7875	-99.84	cp	BRD-K15916496	clotrimazole	Cytochrome P450 inhibitor		KCNN4, CYP3A4, CYP51A1, NR1I2, NR1I3, TRPM2, TRPM4, TRPM8	Cytochrome P450 inhibitor, Imidazoline receptor ligand
7876	-99.84	kd	CGS001-57167	SALL4	Zinc fingers, C2H2-type			
7877	-99.84	kd	CGS001-4718	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
7878	-99.85	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
7879	-99.85	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
7880	-99.85	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
7881	-99.85	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
7882	-99.86	kd	CGS001-4907	NT5E	Adenosine turnover			
7883	-99.87	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
7884	-99.87	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
7885	-99.87	kd	CGS001-147948	ZNF582	Zinc fingers, C2H2-type			
7886	-99.87	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
7887	-99.87	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
7888	-99.87	kd	CGS001-8644	AKR1C3	Prostaglandin synthases			
7889	-99.87	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
7890	-99.88	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
7891	-99.88	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
7892	-99.88	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
7893	-99.88	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
7894	-99.88	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
7895	-99.88	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
7896	-99.88	kd	CGS001-59286	UBL5	-			
7897	-99.88	kd	CGS001-5879	RAC1	Endogenous ligands			
7898	-99.88	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
7899	-99.88	kd	CGS001-3588	IL10RB	IL-10 receptor family			
7900	-99.88	kd	CGS001-2067	ERCC1	-			
7901	-99.89	oe	ccsbBroad304_03928	RRAGC	-			
7902	-99.89	oe	ccsbBroad304_01395	RFX5	-			
7903	-99.89	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
7904	-99.89	kd	CGS001-79862	ZNF669	Zinc fingers, C2H2-type			
7905	-99.89	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
7906	-99.89	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
7907	-99.89	kd	CGS001-54556	ING3	Zinc fingers, PHD-type			
7908	-99.89	kd	CGS001-84890	ADO	-			
7909	-99.89	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
7910	-99.9	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
7911	-99.9	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
7912	-99.9	oe	ccsbBroad304_02626	PKIG	-			
7913	-99.9	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
7914	-99.9	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
7915	-99.9	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
7916	-99.9	kd	CGS001-11212	PROSC	-			
7917	-99.9	kd	CGS001-4704	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7918	-99.9	kd	CGS001-513	ATP5D	ATPases / F-type			
7919	-99.91	oe	ccsbBroad304_01105	PNP	-			
7920	-99.91	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
7921	-99.91	kd	CGS001-55872	PBK	TOPK family			
7922	-99.91	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
7923	-99.91	kd	CGS001-818	CAMK2G	CAMK2 family			
7924	-99.91	kd	CGS001-259	AMBP	Lipocalins			
7925	-99.93	oe	ccsbBroad304_06234	G6PC	-			
7926	-99.93	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
7927	-99.93	cp	BRD-K37798499	etoposide	Topoisomerase inhibitor		TOP2A, CYP2E1, CYP3A5, TOP2B	Topoisomerase inhibitor
7928	-99.93	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7929	-99.93	kd	CGS001-112858	TP53RK	Bud32 family			
7930	-99.93	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
7931	-99.93	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
7932	-99.93	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
7933	-99.94	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
7934	-99.94	oe	ccsbBroad304_06535	LPL	-			
7935	-99.94	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
7936	-99.94	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
7937	-99.94	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
7938	-99.94	kd	CGS001-79711	IPO4	Importins			
7939	-99.94	kd	CGS001-3692	EIF6	-			
7940	-99.94	kd	CGS001-5610	EIF2AK2	Other PEK family kinases			
7941	-99.95	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
7942	-99.95	oe	ccsbBroad304_01165	PDK1	-			
7943	-99.95	oe	ccsbBroad304_02398	LANCL1	-			
7944	-99.95	oe	ccsbBroad304_00657	GNG4	-			
7945	-99.95	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
7946	-99.95	kd	CGS001-63892	THADA	-			
7947	-99.95	kd	CGS001-6777	STAT5B	SH2 domain containing			
7948	-99.95	kd	CGS001-5608	MAP2K6	MAPKK:STE7 family			
7949	-99.95	kd	CGS001-23499	MACF1	EF-hand domain containing			
7950	-99.95	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
7951	-99.95	kd	CGS001-230	ALDOC	-			
7952	-99.95	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
7953	-99.95	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
7954	-99.96	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
7955	-99.96	oe	ccsbBroad304_01001	MEST	-			
7956	-99.96	oe	ccsbBroad304_06574	MDH2	-			
7957	-99.96	oe	ccsbBroad304_06350	HAL	-			
7958	-99.96	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
7959	-99.96	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
7960	-99.96	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
7961	-99.96	oe	ccsbBroad304_08888	ACD	-			
7962	-99.96	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
7963	-99.96	cp	BRD-A16934955	nalbuphine	Opioid receptor agonist		OPRD1, OPRK1, OPRM1	Opioid receptor agonist, Opioid receptor antagonist
7964	-99.96	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
7965	-99.96	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
7966	-99.96	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
7967	-99.96	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
7968	-99.96	kd	CGS001-10497	UNC13B	-			
7969	-99.96	kd	CGS001-6794	STK11	LKB subfamily			
7970	-99.96	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
7971	-99.96	kd	CGS001-5351	PLOD1	-			
7972	-99.96	kd	CGS001-79187	FSD1	Fibronectin type III domain containing			
7973	-99.96	kd	CGS001-1962	EHHADH	-			
7974	-99.96	kd	CGS001-22818	COPZ1	-			
7975	-99.96	kd	CGS001-7832	BTG2	-			
7976	-99.96	kd	CGS001-50	ACO2	-			
7977	-99.98	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
7978	-99.98	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
7979	-99.98	oe	ccsbBroad304_01723	TTK	TTK family			
7980	-99.98	oe	ccsbBroad304_00101	RHOC	-			
7981	-99.98	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
7982	-99.98	oe	ccsbBroad304_14143	NUSAP1	-			
7983	-99.98	oe	ccsbBroad304_13598	NRBP2	NRBP family			
7984	-99.98	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
7985	-99.98	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
7986	-99.98	oe	ccsbBroad304_00568	FHL2	-			
7987	-99.98	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
7988	-99.98	oe	ccsbBroad304_06090	DDOST	-			
7989	-99.98	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
7990	-99.98	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
7991	-99.98	oe	ccsbBroad304_00113	ASNS	-			
7992	-99.98	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
7993	-99.98	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
7994	-99.98	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
7995	-99.98	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
7996	-99.98	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
7997	-99.98	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
7998	-99.98	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
7999	-99.98	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
8000	-99.98	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
8001	-99.98	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
8002	-99.98	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
8003	-99.98	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
8004	-99.98	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
8005	-99.98	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
8006	-99.98	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
8007	-99.98	kd	CGS001-203523	ZNF449	Zinc fingers, C2H2-type			
8008	-99.98	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
8009	-99.98	kd	CGS001-10342	TFG	-			
8010	-99.98	kd	CGS001-7018	TF	-			
8011	-99.98	kd	CGS001-4089	SMAD4	SMADs			
8012	-99.98	kd	CGS001-5636	PRPSAP2	-			
8013	-99.98	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
8014	-99.98	kd	CGS001-55718	POLR3E	RNA polymerase subunits			
8015	-99.98	kd	CGS001-5335	PLCG1	Phosphoinositide-specific phospholipase C			
8016	-99.98	kd	CGS001-5586	PKN2	Protein kinase N (PKN) family			
8017	-99.98	kd	CGS001-51586	MED15	-			
8018	-99.98	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
8019	-99.98	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
8020	-99.98	kd	CGS001-3109	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
8021	-99.98	kd	CGS001-94239	H2AFV	Histones / Replication-independent			
8022	-99.98	kd	CGS001-2966	GTF2H2	General transcription factors			
8023	-99.98	kd	CGS001-1806	DPYD	-			
8024	-99.98	kd	CGS001-54555	DDX49	DEAD-boxes			
8025	-99.98	kd	CGS001-760	CA2	Carbonic anhydrases			
8026	-99.98	kd	CGS001-350	APOH	Apolipoproteins			
8027	-99.98	kd	CGS001-95	ACY1	-			
8028	-99.98	oe	ccsbBroad304_02452	NXF1	-			
