Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
2	100	oe	ccsbBroad304_06992	SRC	Src family			
3	100	kd	CGS001-200081	TXLNA	-			
4	99.98	oe	ccsbBroad304_00833	IFNG	Interferons			
5	99.98	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6	99.98	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
7	99.98	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
8	99.98	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
9	99.98	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
10	99.98	oe	ccsbBroad304_01257	PPOX	-			
11	99.98	oe	ccsbBroad304_13633	PI4KAP2	-			
12	99.98	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
13	99.98	oe	ccsbBroad304_02052	KYNU	-			
14	99.98	oe	ccsbBroad304_00880	IRF2	-			
15	99.98	oe	ccsbBroad304_00832	IFNB1	Interferons			
16	99.98	oe	ccsbBroad304_03433	DDIT4	-			
17	99.98	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
18	99.98	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
19	99.98	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
20	99.98	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
21	99.98	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
22	99.98	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
23	99.98	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
24	99.98	kd	CGS001-55179	FAIM	-			
25	99.98	kd	CGS001-9451	EIF2AK3	PEK subfamily			
26	99.98	kd	CGS001-478	ATP1A3	ATPases / P-type			
27	99.98	kd	CGS001-55608	ANKRD10	Ankyrin repeat domain containing			
28	99.98	kd	CGS001-9326	ZNHIT3	Zinc fingers, HIT-type			
29	99.98	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
30	99.98	kd	CGS001-89766	UMODL1	-			
31	99.98	kd	CGS001-10381	TUBB3	Tubulins			
32	99.98	kd	CGS001-9748	SLK	SLK subfamily			
33	99.98	kd	CGS001-8634	RTCD1	-			
34	99.98	kd	CGS001-55312	RFK	-			
35	99.98	kd	CGS001-5106	PCK2	-			
36	99.98	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
37	99.98	kd	CGS001-7181	NR2C1	Testicular receptors			
38	99.98	kd	CGS001-4077	NBR1	-			
39	99.98	kd	CGS001-9443	MED7	-			
40	99.98	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
41	99.98	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
42	99.98	kd	CGS001-2849	GPR26	GPCR / Class A : Orphans			
43	99.98	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
44	99.98	kd	CGS001-23149	FCHO1	-			
45	99.98	kd	CGS001-11124	FAF1	UBX domain containing			
46	99.98	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
47	99.98	kd	CGS001-23405	DICER1	-			
48	99.98	kd	CGS001-8804	CREG1	-			
49	99.98	kd	CGS001-55937	APOM	Apolipoproteins			
50	99.98	kd	CGS001-8644	AKR1C3	Prostaglandin synthases			
51	99.98	oe	ccsbBroad304_14011	PAPSS1	-			
52	99.98	oe	ccsbBroad304_07761	CORO1A	Coronins			
53	99.96	oe	ccsbBroad304_01699	TPD52L2	-			
54	99.96	oe	ccsbBroad304_07598	PEMT	-			
55	99.96	oe	ccsbBroad304_00811	ICAM1	CD molecules			
56	99.96	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
57	99.96	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
58	99.96	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
59	99.96	kd	CGS001-51181	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
60	99.96	kd	CGS001-10421	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
61	99.96	kd	CGS001-9531	BAG3	-			
62	99.96	oe	ccsbBroad304_05749	A2M	-			
63	99.96	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
64	99.95	cc		Structural maintenance of chromosomes proteins LOF	-			
65	99.95	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
66	99.95	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
67	99.95	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
68	99.95	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
69	99.95	kd	CGS001-25836	NIPBL	-			
70	99.95	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
71	99.95	kd	CGS001-6259	RYK	Type XV RTKs: RYK			
72	99.95	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
73	99.95	kd	CGS001-1001	CDH3	Cadherins / Major cadherins			
74	99.95	kd	CGS001-694	BTG1	-			
75	99.95	kd	CGS001-51742	ARID4B	-			
76	99.95	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
77	99.94	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
78	99.94	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
79	99.94	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
80	99.94	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
81	99.94	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
82	99.94	kd	CGS001-2073	ERCC5	-			
83	99.93	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
84	99.93	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
85	99.93	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
86	99.93	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
87	99.93	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
88	99.93	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
89	99.93	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
90	99.93	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
91	99.93	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
92	99.93	kd	CGS001-5184	PEPD	Methionyl aminopeptidase			
93	99.93	kd	CGS001-4817	NIT1	-			
94	99.93	kd	CGS001-29965	C16ORF5	-			
95	99.93	kd	CGS001-481	ATP1B1	ATPases / P-type			
96	99.92	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
97	99.92	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
98	99.92	kd	CGS001-8233	ZRSR2	RNA binding motif (RRM) containing			
99	99.92	kd	CGS001-6909	TBX2	T-boxes			
100	99.92	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
101	99.92	kd	CGS001-384	ARG2	Arginase			
102	99.9	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
103	99.9	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
104	99.9	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
105	99.9	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
106	99.9	kd	CGS001-6714	SRC	Src family			
107	99.9	kd	CGS001-9761	MLEC	-			
108	99.89	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
109	99.89	cp	BRD-A42423104	benproperine	Antitussive			Antitussive
110	99.89	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
111	99.89	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
112	99.89	kd	CGS001-5373	PMM2	-			
113	99.89	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
114	99.88	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
115	99.88	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
116	99.88	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
117	99.88	kd	CGS001-283455	KSR2	RAF family			
118	99.87	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
119	99.87	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
120	99.87	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
121	99.87	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
122	99.87	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
123	99.87	kd	CGS001-2261	FGFR3	Type V RTKs: FGF (fibroblast growth factor) receptor family			
124	99.87	kd	CGS001-6387	CXCL12	Endogenous ligands			
125	99.86	oe	ccsbBroad304_02386	EIF1B	-			
126	99.86	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
127	99.86	kd	CGS001-57406	ABHD6	Abhydrolase domain containing			
128	99.84	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
129	99.84	kd	CGS001-10494	STK25	YSK subfamily			
130	99.84	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
131	99.84	kd	CGS001-81894	SLC25A28	Miscellaneous SLC25 mitochondrial transporters			
132	99.84	kd	CGS001-5566	PRKACA	Protein kinase A			
133	99.84	kd	CGS001-122618	PLD4	-			
134	99.84	kd	CGS001-10128	LRPPRC	-			
135	99.83	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
136	99.83	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
137	99.82	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
138	99.82	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
139	99.82	kd	CGS001-677	ZFP36L1	RING-type (C3HC4) zinc fingers			
140	99.82	kd	CGS001-538	ATP7A	ATPases / P-type			
141	99.81	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
142	99.81	kd	CGS001-79006	METRN	-			
143	99.81	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
144	99.8	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
145	99.8	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
146	99.8	kd	CGS001-7027	TFDP1	-			
147	99.8	kd	CGS001-64783	RBM15	RNA binding motif (RRM) containing			
148	99.8	kd	CGS001-353345	GPR141	GPCR / Class A : Orphans			
149	99.8	kd	CGS001-2118	ETV4	ETS Transcription Factors			
150	99.8	kd	CGS001-10589	DRAP1	-			
151	99.79	kd	CGS001-8193	DPF1	Zinc fingers, PHD-type			
152	99.78	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
153	99.78	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
154	99.78	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
155	99.78	kd	CGS001-7103	TSPAN8	Tetraspanins			
156	99.78	kd	CGS001-10254	STAM2	-			
157	99.77	cc		Rho associated kinase inhibitor	-			
158	99.77	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
159	99.77	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
160	99.77	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
161	99.77	kd	CGS001-8438	RAD54L	-			
162	99.76	kd	CGS001-10383	TUBB2C	Tubulins			
163	99.76	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
164	99.76	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
165	99.75	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
166	99.75	kd	CGS001-65123	INTS3	-			
167	99.75	kd	CGS001-8573	CASK	CASK family			
168	99.74	cp	BRD-K33312228	halometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
169	99.74	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
170	99.74	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
171	99.74	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
172	99.73	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
173	99.73	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
174	99.72	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
175	99.71	oe	ccsbBroad304_06048	CRYZ	-			
176	99.71	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
177	99.71	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
178	99.7	oe	ccsbBroad304_00551	FECH	-			
179	99.7	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
180	99.7	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
181	99.7	kd	CGS001-9988	DMTF1	-			
182	99.69	cp	BRD-K56614220	clofazimine	GK0582 inhibitor			GK0582 inhibitor
183	99.69	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
184	99.69	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
185	99.68	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
186	99.68	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
187	99.66	kd	CGS001-10392	NOD1	Nucleotide-binding domain and leucine rich repeat containing			
188	99.66	kd	CGS001-64170	CARD9	-			
189	99.65	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
190	99.65	kd	CGS001-10544	PROCR	CD molecules			
191	99.64	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
192	99.64	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
193	99.63	oe	ccsbBroad304_06862	RGS3	-			
194	99.62	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
195	99.62	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
196	99.61	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
197	99.59	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
198	99.59	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
199	99.58	kd	CGS001-6897	TARS	Aminoacyl tRNA synthetases / Class II			
200	99.58	kd	CGS001-5501	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
201	99.58	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
202	99.57	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
203	99.57	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
204	99.57	oe	ccsbBroad304_06855	RDX	-			
205	99.56	oe	ccsbBroad304_06648	CNOT3	-			
206	99.56	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
207	99.56	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
208	99.56	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
209	99.54	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
210	99.54	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
211	99.54	kd	CGS001-5352	PLOD2	-			
212	99.54	oe	ccsbBroad304_06836	RAD23B	-			
213	99.53	kd	CGS001-1649	DDIT3	-			
214	99.52	kd	CGS001-5879	RAC1	Endogenous ligands			
215	99.52	kd	CGS001-1327	COX4I1	Mitochondrial respiratory chain complex			
216	99.52	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
217	99.51	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
218	99.51	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
219	99.5	kd	CGS001-23408	SIRT5	Histone deacetylases			
220	99.48	kd	CGS001-54788	DNAJB12	Heat shock proteins / DNAJ (HSP40)			
221	99.46	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
222	99.46	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
223	99.46	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
224	99.46	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
225	99.45	kd	CGS001-10413	YAP1	Hippo Signaling			
226	99.43	cp	BRD-K66412701	pazufloxacin	Topoisomerase inhibitor			Topoisomerase inhibitor
227	99.43	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
228	99.42	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
229	99.42	kd	CGS001-7267	TTC3	RING-type (C3HC4) zinc fingers			
230	99.42	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
231	99.41	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
232	99.41	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
233	99.4	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
234	99.39	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
235	99.38	oe	ccsbBroad304_00552	FEN1	-			
236	99.38	kd	CGS001-6347	CCL2	Chemokine ligands			
237	99.37	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
238	99.37	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
239	99.36	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
240	99.35	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
241	99.35	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
242	99.35	kd	CGS001-6117	RPA1	-			
243	99.35	kd	CGS001-55810	FOXJ2	Forkhead boxes			
244	99.34	kd	CGS001-3690	ITGB3	Integrins			
245	99.33	kd	CGS001-5594	MAPK1	MAPK:ERK subfamily			
246	99.33	kd	CGS001-1643	DDB2	WD repeat domain containing			
247	99.33	kd	CGS001-8945	BTRC	F-boxes / WD-40 domains			
248	99.33	kd	CGS001-435	ASL	-			
249	99.32	kd	CGS001-7020	TFAP2A	-			
250	99.31	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
251	99.3	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
252	99.3	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
253	99.28	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
254	99.28	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
255	99.28	kd	CGS001-657	BMPR1A	Type I receptor serine/threonine kinases			
256	99.27	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
257	99.27	kd	CGS001-9833	MELK	MELK subfamily			
258	99.26	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
259	99.24	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
260	99.23	kd	CGS001-140685	ZBTB46	BTB/POZ domain containing			
261	99.23	kd	CGS001-5827	PXMP2	-			
262	99.23	kd	CGS001-79143	MBOAT7	-			
263	99.23	kd	CGS001-54998	AURKAIP1	-			
264	99.22	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
265	99.22	kd	CGS001-1622	DBI	-			
266	99.21	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
267	99.21	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
268	99.21	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
269	99.21	kd	CGS001-100	ADA	Adenosine turnover			
270	99.19	kd	CGS001-10096	ACTR3	-			
271	99.18	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
272	99.16	kd	CGS001-5993	RFX5	-			
273	99.15	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
274	99.15	kd	CGS001-10105	PPIF	-			
275	99.14	kd	CGS001-4299	AFF1	-			
276	99.13	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
277	99.13	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
278	99.12	kd	CGS001-81544	GDPD5	-			
279	99.11	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
280	99.11	kd	CGS001-2355	FOSL2	basic leucine zipper proteins			
281	99.1	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
282	99.1	kd	CGS001-7001	PRDX2	-			
283	99.1	kd	CGS001-2309	FOXO3	Forkhead boxes			
284	99.1	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
285	99.09	kd	CGS001-2000	ELF4	ETS Transcription Factors			
286	99.08	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
287	99.08	kd	CGS001-3664	IRF6	-			
288	99.07	kd	CGS001-5226	PGD	-			
289	99.07	kd	CGS001-54681	P4HTM	-			
290	99.06	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
291	99.05	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
292	99.05	kd	CGS001-27097	TAF5L	WD repeat domain containing			
293	99.03	cc		Mediator complex LOF	-			
294	99.01	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
295	99.01	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
296	98.97	kd	CGS001-10943	MSL3	-			
297	98.96	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
298	98.95	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
299	98.95	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
300	98.94	kd	CGS001-3162	HMOX1	Haem oxygenase			
301	98.94	kd	CGS001-1677	DFFB	-			
302	98.94	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
303	98.93	oe	ccsbBroad304_02203	MAD2L1BP	-			
304	98.93	kd	CGS001-5378	PMS1	-			
305	98.93	kd	CGS001-10841	FTCD	-			
306	98.92	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
307	98.92	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
308	98.92	kd	CGS001-1105	CHD1	-			
309	98.88	oe	ccsbBroad304_07124	UROD	-			
310	98.87	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
311	98.86	kd	CGS001-11212	PROSC	-			
312	98.83	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
313	98.83	kd	CGS001-9519	TBPL1	-			
314	98.8	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
315	98.79	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
316	98.79	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
317	98.79	kd	CGS001-10112	KIF20A	Kinesins			
318	98.77	kd	CGS001-7172	TPMT	-			
319	98.75	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
320	98.75	kd	CGS001-3589	IL11	Endogenous ligands			
321	98.72	oe	ccsbBroad304_05948	CCND2	-			
322	98.71	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
323	98.71	kd	CGS001-25888	ZNF473	Zinc fingers, C2H2-type			
324	98.71	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
325	98.7	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
326	98.7	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
327	98.69	kd	CGS001-8874	ARHGEF7	Rho guanine nucleotide exchange factors			
328	98.65	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
329	98.64	cp	BRD-A79903587	tegafur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
330	98.63	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
331	98.63	kd	CGS001-10538	BATF	basic leucine zipper proteins			
332	98.62	cp	BRD-K04196797	oxcarbazepine	Sodium channel blocker		CYP2C19, CYP3A4, CYP3A5, SCN1A, SCN3A, SCN5A	Sodium channel blocker
333	98.62	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
334	98.62	kd	CGS001-1717	DHCR7	-			
335	98.6	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
336	98.6	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
337	98.6	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
338	98.6	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
339	98.54	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
340	98.53	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
341	98.53	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
342	98.5	kd	CGS001-5909	RAP1GAP	-			
343	98.49	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
344	98.49	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
345	98.48	kd	CGS001-5796	PTPRK	Receptor tyrosine phosphatases (RTP)			
346	98.47	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
347	98.46	kd	CGS001-9897	KIAA0196	-			
348	98.46	kd	CGS001-54541	DDIT4	-			
349	98.46	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
350	98.45	kd	CGS001-5096	PCCB	Carboxylases			
351	98.44	kd	CGS001-5920	RARRES3	-			
352	98.44	kd	CGS001-440387	CTRB2	-			
353	98.43	kd	CGS001-10765	KDM5B	Histone demethylases			
354	98.41	kd	CGS001-5351	PLOD1	-			
355	98.4	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
356	98.4	kd	CGS001-7323	UBE2D3	Ubiquitin-conjugating enzymes E2			
357	98.4	kd	CGS001-4782	NFIC	-			
358	98.39	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
359	98.38	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
360	98.37	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
361	98.35	oe	ccsbBroad304_01247	POU2AF1	-			
362	98.34	kd	CGS001-9869	SETDB1	Histone methyltransferases (HMTs)			
363	98.33	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
364	98.33	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
365	98.32	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
366	98.31	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
367	98.3	kd	CGS001-29947	DNMT3L	-			
368	98.27	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
369	98.25	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
370	98.22	kd	CGS001-2859	GPR35	GPCR / Class A : Orphans			
371	98.22	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
372	98.21	kd	CGS001-831	CAST	-			
373	98.19	oe	ccsbBroad304_00060	AMBP	Lipocalins			
374	98.17	kd	CGS001-10497	UNC13B	-			
375	98.15	kd	CGS001-100133941	CD24	CD molecules			
376	98.14	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
377	98.12	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
378	98.12	kd	CGS001-55958	KLHL9	BTB/POZ domain containing			
379	98.11	oe	ccsbBroad304_00995	MECP2	-			
380	98.11	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
381	98.1	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
382	98.09	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
383	98.06	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
384	98.05	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
385	98.04	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
386	98.04	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
387	98.04	kd	CGS001-10048	RANBP9	-			
388	98.04	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
389	98.02	kd	CGS001-2683	B4GALT1	Beta 4-glycosyltransferases			
390	98.01	kd	CGS001-23266	LPHN2	Adhesion Class GPCRs			
391	97.97	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
392	97.95	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
393	97.94	oe	ccsbBroad304_02425	CDIPT	-			
394	97.94	kd	CGS001-11331	PHB2	-			
395	97.93	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
396	97.92	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
397	97.9	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
398	97.9	kd	CGS001-8835	SOCS2	SH2 domain containing			
399	97.87	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
400	97.86	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
401	97.84	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
402	97.81	kd	CGS001-5427	POLE2	DNA polymerases			
403	97.8	kd	CGS001-79001	VKORC1	Oxidoreductases			
404	97.8	kd	CGS001-8807	IL18RAP	CD molecules			
405	97.79	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
406	97.77	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
407	97.77	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
408	97.76	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
409	97.75	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
410	97.74	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
411	97.71	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
412	97.7	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
413	97.69	kd	CGS001-5563	PRKAA2	AMPK subfamily			
414	97.68	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
415	97.67	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
416	97.67	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
417	97.65	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
418	97.65	kd	CGS001-116519	APOA5	Apolipoproteins			
419	97.64	kd	CGS001-7292	TNFSF4	CD molecules			
420	97.64	kd	CGS001-1827	RCAN1	-			
421	97.63	kd	CGS001-586	BCAT1	-			
422	97.62	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
423	97.61	kd	CGS001-149233	IL23R	IL-12 receptor family			
424	97.58	oe	ccsbBroad304_08167	DNTTIP2	-			
425	97.58	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
426	97.54	kd	CGS001-7374	UNG	-			
427	97.48	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
428	97.42	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
429	97.42	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
430	97.41	kd	CGS001-4352	MPL	Prolactin receptor family			
431	97.39	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
432	97.37	kd	CGS001-323	APBB2	-			
433	97.36	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
434	97.36	kd	CGS001-8853	ASAP2	Ankyrin repeat domain containing			
435	97.32	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
436	97.31	kd	CGS001-2782	GNB1	WD repeat domain containing			
437	97.3	oe	ccsbBroad304_00459	DPYD	-			
438	97.28	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
439	97.28	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
440	97.24	kd	CGS001-7297	TYK2	Janus kinase (JakA) family			
441	97.24	kd	CGS001-5144	PDE4D	Phosphodiesterases			
442	97.22	cc		DNA Replication LOF	-			
443	97.22	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
444	97.2	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
445	97.19	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
446	97.1	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
447	97.07	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
448	97.05	oe	ccsbBroad304_06711	PFAS	-			
449	97.04	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
450	97.03	cp	BRD-A68589262	troxipide	Glucosamine synthetase stimulant			Glucosamine synthetase stimulant
451	97.03	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
452	97.02	oe	ccsbBroad304_06090	DDOST	-			
453	97.02	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
454	97.01	oe	ccsbBroad304_06291	GNAI1	-			
455	96.99	kd	CGS001-3688	ITGB1	Integrins			
456	96.95	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
457	96.94	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
458	96.93	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
459	96.91	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
460	96.9	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
461	96.89	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
462	96.88	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
463	96.86	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
464	96.84	kd	CGS001-60493	FASTKD5	-			
465	96.82	kd	CGS001-7343	UBTF	-			
466	96.81	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
467	96.81	kd	CGS001-7272	TTK	TTK family			
468	96.8	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
469	96.77	cc		NFKB Activation GOF	-			
470	96.77	kd	CGS001-5469	MED1	-			
471	96.75	kd	CGS001-84969	TOX2	-			
472	96.75	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
473	96.69	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
474	96.66	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
475	96.64	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
476	96.63	oe	ccsbBroad304_01519	SET	-			
477	96.61	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
478	96.6	kd	CGS001-57761	TRIB3	Trbl family			
479	96.58	kd	CGS001-4316	MMP7	Matrix metallopeptidase			
480	96.56	oe	ccsbBroad304_01933	TEAD2	-			
481	96.56	kd	CGS001-3930	LBR	Tudor domain containing			
482	96.56	kd	CGS001-10196	PRMT3	Protein arginine N-methyltransferases			
483	96.55	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
484	96.53	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
485	96.52	kd	CGS001-4907	NT5E	Adenosine turnover			
486	96.5	kd	CGS001-9415	FADS2	Fatty acid desaturases			
487	96.45	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
488	96.44	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
489	96.44	kd	CGS001-81848	SPRY4	-			
490	96.44	kd	CGS001-2109	ETFB	-			
491	96.43	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
492	96.43	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
493	96.42	kd	CGS001-55422	ZNF331	Zinc fingers, C2H2-type			
494	96.42	oe	ccsbBroad304_02572	SERINC3	-			
495	96.41	kd	CGS001-2872	MKNK2	MKN subfamily			
496	96.41	kd	CGS001-808	CALM3	EF-hand domain containing			
497	96.35	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
498	96.33	cp	BRD-A37052580	physostigmine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Cholinesterase inhibitor
499	96.33	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
500	96.3	kd	CGS001-11129	CLASRP	-			
501	96.28	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
502	96.26	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
503	96.26	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
504	96.24	oe	ccsbBroad304_02032	TSC22D1	-			
505	96.24	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
506	96.23	kd	CGS001-6016	RIT1	-			
507	96.21	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
508	96.19	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
509	96.19	kd	CGS001-2817	GPC1	Proteoglycans / Cell Surface : Glypicans			
510	96.18	cc		BMP Signaling LOF	-			
511	96.16	cp	BRD-K18523449	mestanolone	Androgenic steroid			Androgenic steroid
512	96.14	kd	CGS001-23492	CBX7	-			
513	96.13	cc		DNA synthesis inhibitor	-			
514	96.11	cc		PKC activator	-			
515	96.09	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
516	96.08	kd	CGS001-54438	GFOD1	-			
517	96.08	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
518	96.07	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
519	96.07	kd	CGS001-23657	SLC7A11	Solute carriers			
520	96.06	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
521	96.06	kd	CGS001-253260	RICTOR	-			
522	96.05	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
523	96.03	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
524	96.02	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
525	96.02	kd	CGS001-22883	CLSTN1	Cadherins / Cadherin-related			
526	95.97	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
527	95.95	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
528	95.93	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
529	95.92	kd	CGS001-545	ATR	ATR subfamily			
530	95.89	kd	CGS001-9638	FEZ1	-			
531	95.86	kd	CGS001-25937	WWTR1	Hippo Signaling			
532	95.85	oe	ccsbBroad304_00816	IDE	Pitrilysin			
533	95.85	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
534	95.82	kd	CGS001-813	CALU	EF-hand domain containing			
535	95.82	kd	CGS001-1031	CDKN2C	Ankyrin repeat domain containing			
536	95.78	kd	CGS001-51014	TMED7	-			
537	95.77	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
538	95.76	kd	CGS001-2288	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
539	95.76	kd	CGS001-10891	PPARGC1A	RNA binding motif (RRM) containing			
540	95.76	kd	CGS001-1163	CKS1B	-			
541	95.73	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
542	95.73	kd	CGS001-11180	WDR6	WD repeat domain containing			
543	95.73	kd	CGS001-190	NR0B1	DAX-like receptors			
544	95.72	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
545	95.7	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
546	95.7	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
547	95.7	oe	ccsbBroad304_01146	PARN	-			
548	95.69	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
549	95.68	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
550	95.63	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
551	95.62	kd	CGS001-10174	SORBS3	-			
552	95.6	kd	CGS001-284	ANGPT1	Fibrinogen C domain containing			
553	95.59	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
554	95.54	kd	CGS001-84333	PCGF5	Polycomb group ring fingers			
555	95.54	kd	CGS001-2959	GTF2B	General transcription factors			
556	95.53	kd	CGS001-7165	TPD52L2	-			
557	95.5	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
558	95.48	kd	CGS001-8313	AXIN2	-			
559	95.46	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
560	95.46	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
561	95.45	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
562	95.45	kd	CGS001-10651	MTX2	-			
563	95.44	kd	CGS001-6715	SRD5A1	-			
564	95.43	kd	CGS001-10241	CALCOCO2	-			
565	95.41	kd	CGS001-5025	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
566	95.39	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
567	95.39	kd	CGS001-8767	RIPK2	Receptor interacting protein kinase (RIPK) family			
568	95.39	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
569	95.37	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
570	95.35	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
571	95.31	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
572	95.3	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
573	95.3	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
574	95.29	kd	CGS001-6675	UAP1	-			
575	95.28	oe	ccsbBroad304_01184	PGK1	-			
576	95.27	kd	CGS001-9637	FEZ2	-			
577	95.23	cc		Serpin peptidase inhibitors LOF	-			
578	95.22	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
579	95.2	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
580	95.2	kd	CGS001-23786	BCL2L13	-			
581	95.19	cc		Serine proteases GOF	-			
582	95.17	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
583	95.17	kd	CGS001-64858	DCLRE1B	-			
584	95.14	oe	ccsbBroad304_00568	FHL2	-			
585	95.14	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
586	95.13	kd	CGS001-23647	ARFIP2	-			
587	95.1	kd	CGS001-10190	TXNDC9	-			
588	95.07	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
589	95.06	oe	ccsbBroad304_03555	PANK4	-			
590	95.06	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
591	95.05	kd	CGS001-8894	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
592	95.03	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
593	95.03	kd	CGS001-4680	CEACAM6	CD molecules			
594	95	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
595	94.99	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
596	94.96	kd	CGS001-2230	FDX1	-			
597	94.91	cp	BRD-K44779798	miglitol	Glucosidase inhibitor		GAA, MGAM, GANAB, GANC, SLC5A4	Glucosidase inhibitor
598	94.89	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
599	94.88	cp	BRD-A71009679	KUC103420N	-666			-666
600	94.85	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
601	94.8	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
602	94.75	kd	CGS001-2280	FKBP1A	Cis-trans-isomerases			
603	94.72	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
604	94.68	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
605	94.64	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
606	94.63	oe	ccsbBroad304_08481	CEP55	-			
607	94.54	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
608	94.51	oe	ccsbBroad304_08325	LIPT1	-			
609	94.49	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
610	94.49	kd	CGS001-6241	RRM2	Ribonucleoside-diphosphate reductases			
611	94.46	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
612	94.41	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
613	94.41	kd	CGS001-9181	ARHGEF2	Rho guanine nucleotide exchange factors			
614	94.41	oe	ccsbBroad304_08480	PNPO	-			
615	94.38	oe	ccsbBroad304_10758	CTBP2	-			
616	94.37	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
617	94.34	kd	CGS001-3017	HIST1H2BD	Histones / Replication-dependent			
618	94.34	kd	CGS001-5433	POLR2D	RNA polymerase subunits			
619	94.32	kd	CGS001-54957	TXNL4B	-			
620	94.29	kd	CGS001-4869	NPM1	-			
621	94.26	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
622	94.22	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
623	94.22	kd	CGS001-2857	GPR34	GPCR / Class A : Orphans			
624	94.21	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
625	94.2	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
626	94.19	kd	CGS001-5018	OXA1L	-			
627	94.17	kd	CGS001-5982	RFC2	ATPases / AAA-type			
628	94.16	kd	CGS001-26277	TINF2	-			
629	94.14	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
630	94.13	cc		General transcription factors group 1 LOF	-			
631	94.04	kd	CGS001-10681	GNB5	WD repeat domain containing			
632	94.02	kd	CGS001-116113	FOXP4	Forkhead boxes			
633	94	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
634	93.98	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
635	93.96	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
636	93.96	kd	CGS001-516	ATP5G1	ATPases / F-type			
637	93.95	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
638	93.93	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
639	93.91	kd	CGS001-7371	UCK2	-			
640	93.88	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
641	93.84	cp	BRD-K98493452	honokiol	AKT inhibitor		ALOX5, PTGS1, PTGS2	AKT inhibitor
642	93.83	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
643	93.82	oe	ccsbBroad304_07094	TPMT	-			
644	93.8	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
645	93.8	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
646	93.79	kd	CGS001-9891	NUAK1	NuaK subfamily			
647	93.78	oe	ccsbBroad304_04038	ELOVL6	-			
648	93.74	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
649	93.73	kd	CGS001-1112	FOXN3	Forkhead boxes			
650	93.69	oe	ccsbBroad304_02110	VAPB	-			
651	93.65	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
652	93.64	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
653	93.64	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
654	93.61	oe	ccsbBroad304_03268	GMPR2	-			
655	93.6	kd	CGS001-27336	HTATSF1	RNA binding motif (RRM) containing			
656	93.58	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
657	93.56	kd	CGS001-27244	SESN1	-			
658	93.56	kd	CGS001-7965	AIMP2	-			
659	93.55	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
660	93.54	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
661	93.53	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
662	93.51	kd	CGS001-5355	PLP2	-			
663	93.49	oe	ccsbBroad304_00836	IGF2	-			
664	93.46	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
665	93.44	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
666	93.44	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
667	93.42	kd	CGS001-1508	CTSB	Cathepsins			
668	93.42	kd	CGS001-11154	AP4S1	-			
669	93.32	kd	CGS001-81550	TDRD3	Tudor domain containing			
670	93.3	oe	ccsbBroad304_07704	SUB1	-			
671	93.26	kd	CGS001-2263	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
672	93.25	oe	ccsbBroad304_07531	TANK	-			
673	93.19	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
674	93.18	cp	BRD-K33483813	actarit	Interleukin receptor agonist			Interleukin receptor agonist
675	93.13	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
676	93.13	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
677	93.09	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
678	93.09	kd	CGS001-2909	ARHGAP35	Rho GTPase activating proteins			
679	93.08	kd	CGS001-9133	CCNB2	-			
680	93.07	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
681	93.07	oe	ccsbBroad304_00077	APEX1	-			
682	93.05	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
683	93.04	cp	BRD-A94543220	bifonazole	Sterol demethylase inhibitor		CYP2B6	Sterol demethylase inhibitor
684	93.01	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
685	92.99	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
686	92.96	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
687	92.95	kd	CGS001-11073	TOPBP1	-			
688	92.94	oe	ccsbBroad304_02578	EBNA1BP2	-			
689	92.91	kd	CGS001-995	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
690	92.88	oe	ccsbBroad304_03652	EXOC2	-			
691	92.83	kd	CGS001-54512	EXOSC4	-			
692	92.82	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
693	92.75	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
694	92.75	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
695	92.73	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
696	92.73	kd	CGS001-1859	DYRK1A	Dyrk1 subfamily			
697	92.71	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
698	92.7	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
699	92.69	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
700	92.64	oe	ccsbBroad304_07252	DGKZ	-			
701	92.63	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
702	92.62	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
703	92.59	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
704	92.58	cp	BRD-A01787639	naftopidil	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
705	92.57	kd	CGS001-57521	RPTOR	WD repeat domain containing			
706	92.56	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
707	92.56	kd	CGS001-29763	PACSIN3	-			
708	92.55	oe	ccsbBroad304_03444	PAF1	-			
709	92.55	kd	CGS001-5110	PCMT1	-			
710	92.54	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
711	92.51	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
712	92.47	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
713	92.46	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
714	92.44	kd	CGS001-257397	TAB3	-			
715	92.4	oe	ccsbBroad304_02048	BCL10	-			
716	92.39	kd	CGS001-4926	NUMA1	-			
717	92.36	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
718	92.33	cc		Lipocalins GOF	-			
719	92.32	oe	ccsbBroad304_00985	MCL1	-			
720	92.28	kd	CGS001-87	ACTN1	EF-hand domain containing			
721	92.27	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
722	92.25	kd	CGS001-5036	PA2G4	-			
723	92.23	kd	CGS001-2920	CXCL2	Endogenous ligands			
724	92.2	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
725	92.19	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
726	92.17	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
727	92.17	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
728	92.14	kd	CGS001-8895	CPNE3	-			
729	92.13	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
730	92.11	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
731	92.07	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
732	92.04	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
733	92.03	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
734	92.02	oe	ccsbBroad304_01211	PKM2	-			
735	92.02	oe	ccsbBroad304_02249	KIAA0494	-			
736	92.01	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
737	92.01	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
738	91.98	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
739	91.98	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
740	91.95	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
741	91.95	kd	CGS001-3313	HSPA9	Heat shock proteins / HSP70			
742	91.94	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
743	91.92	kd	CGS001-10113	PREB	WD repeat domain containing			
744	91.92	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
745	91.9	oe	ccsbBroad304_06976	SMARCE1	-			
746	91.89	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
747	91.86	kd	CGS001-2976	GTF3C2	General transcription factors			
748	91.82	kd	CGS001-23670	TMEM2	-			
749	91.79	kd	CGS001-2264	FGFR4	Type V RTKs: FGF (fibroblast growth factor) receptor family			
750	91.73	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
751	91.71	cc		Purinergic receptors P2Y GOF	-			
752	91.7	oe	ccsbBroad304_01617	STX4	-			
753	91.67	oe	ccsbBroad304_06870	RNH1	-			
754	91.63	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
755	91.63	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
756	91.6	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
757	91.5	kd	CGS001-4092	SMAD7	SMADs			
758	91.46	kd	CGS001-999	CDH1	CD molecules			
759	91.45	kd	CGS001-7004	TEAD4	-			
760	91.41	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
761	91.39	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
762	91.34	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
763	91.3	kd	CGS001-27	ABL2	Abl family			
764	91.29	oe	ccsbBroad304_07097	TRAF1	-			
765	91.27	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
766	91.27	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
767	91.26	kd	CGS001-2242	FES	Fer family			
768	91.2	oe	ccsbBroad304_03420	TOLLIP	-			
769	91.19	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
770	91.18	kd	CGS001-10957	PNRC1	-			
771	91.18	kd	CGS001-1154	CISH	SH2 domain containing			
772	91.17	kd	CGS001-57804	POLD4	DNA polymerases			
773	91.16	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
774	91.13	kd	CGS001-10493	VAT1	-			
775	91.08	kd	CGS001-3431	SP110	Non-enzymatic BRD containing proteins			
776	91.07	kd	CGS001-1045	CDX2	Homeoboxes / ANTP class : HOXL subclass			
777	91.05	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
778	90.99	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
779	90.95	kd	CGS001-5649	RELN	-			
780	90.92	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
781	90.92	kd	CGS001-3717	JAK2	Janus kinase (JakA) family			
782	90.91	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
783	90.88	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
784	90.88	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
785	90.85	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
786	90.79	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
787	90.75	kd	CGS001-10682	EBP	-			
788	90.67	kd	CGS001-1387	CREBBP	Chromatin-modifying enzymes / K-acetyltransferases			
789	90.66	kd	CGS001-6886	TAL1	Basic helix-loop-helix proteins			
790	90.63	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
791	90.5	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
792	90.5	kd	CGS001-2950	GSTP1	Glutathione S-transferases			
793	90.48	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
794	90.46	kd	CGS001-126208	ZNF787	Zinc fingers, C2H2-type			
795	90.42	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
796	90.42	kd	CGS001-9184	BUB3	WD repeat domain containing			
797	90.41	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
798	90.41	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
799	90.39	kd	CGS001-163486	DENND1B	DENN/MADD domain containing			
800	90.35	oe	ccsbBroad304_07326	EIF2B2	-			
801	90.29	cc		Integrin subunits beta LOF	-			
802	90.28	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
803	90.15	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
804	90.12	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
805	90.07	cp	BRD-K85090592	pilocarpine	Acetylcholine receptor agonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor agonist
806	90	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
807	89.94	oe	ccsbBroad304_08152	PSAT1	-			
808	89.93	cc		Aurora kinase inhibitor	-			
809	89.92	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
810	89.92	kd	CGS001-9589	WTAP	-			
811	89.91	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
812	89.91	kd	CGS001-56998	CTNNBIP1	Catenins			
813	89.9	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
814	89.9	kd	CGS001-80758	PRR7	-			
815	89.89	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
816	89.85	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
817	89.85	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
818	89.82	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
819	89.74	oe	ccsbBroad304_02964	TIMM9	-			
820	89.7	kd	CGS001-2869	GRK5	GRK1/3 subfamily			
821	89.65	oe	ccsbBroad304_07861	COBL	-			
822	89.65	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
823	89.62	kd	CGS001-5091	PC	Carboxylases			
824	89.6	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
825	89.6	kd	CGS001-4548	MTR	-			
826	89.56	kd	CGS001-64135	IFIH1	-			
827	89.52	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
828	89.45	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
829	89.43	kd	CGS001-6429	SRSF4	RNA binding motif (RRM) containing			
830	89.37	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
831	89.36	kd	CGS001-645	BLVRB	Short chain dehydrogenase/reductase superfamily / Atypical members			
832	89.32	kd	CGS001-4709	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
833	89.32	kd	CGS001-7852	CXCR4	Chemokine receptors			
834	89.26	kd	CGS001-6282	S100A11	EF-hand domain containing			
835	89.24	kd	CGS001-826	CAPNS1	EF-hand domain containing			
836	89.24	oe	ccsbBroad304_03808	ERGIC1	-			
837	89.22	oe	ccsbBroad304_01052	MYB	-			
838	89.22	kd	CGS001-11340	EXOSC8	-			
839	89.21	kd	CGS001-7298	TYMS	Methyltransferases			
840	89.18	oe	ccsbBroad304_01701	TPI1	-			
841	89.18	kd	CGS001-822	CAPG	-			
842	89.17	kd	CGS001-1349	COX7B	Mitochondrial respiratory chain complex			
843	89.12	oe	ccsbBroad304_01174	PEX13	-			
844	89.12	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
845	89.08	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
846	89.08	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
847	89.01	cc		Tumor necrosis factor superfamily LOF	-			
848	89	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
849	88.99	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
850	88.99	kd	CGS001-6988	TCTA	-			
851	88.96	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
852	88.94	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
853	88.92	oe	ccsbBroad304_06828	PYCR1	-			
854	88.92	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
855	88.92	kd	CGS001-79885	HDAC11	Histone deacetylases			
856	88.88	kd	CGS001-10051	SMC4	Structural maintenance of chromosomes proteins			
857	88.84	kd	CGS001-7764	ZNF217	Zinc fingers, C2H2-type			
858	88.81	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
859	88.8	oe	ccsbBroad304_08662	MCCC1	-			
860	88.8	kd	CGS001-5966	REL	NFkappaB transcription factor family			
861	88.78	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
862	88.77	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
863	88.76	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
864	88.76	oe	ccsbBroad304_00116	ASS1	-			
865	88.76	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
866	88.68	kd	CGS001-2108	ETFA	-			
867	88.67	kd	CGS001-3131	HLF	-			
868	88.67	kd	CGS001-51022	GLRX2	-			
869	88.67	kd	CGS001-1152	CKB	-			
870	88.64	oe	ccsbBroad304_03950	ATG3	-			
871	88.64	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
872	88.6	oe	ccsbBroad304_01351	PEX19	-			
873	88.59	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
874	88.58	kd	CGS001-6118	RPA2	-			
875	88.51	kd	CGS001-10657	KHDRBS1	-			
876	88.45	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
877	88.45	kd	CGS001-64343	AZI2	-			
878	88.4	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
879	88.36	cp	BRD-K81855038	roxatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
880	88.35	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
881	88.35	kd	CGS001-8536	CAMK1	CAMK1 family			
882	88.35	kd	CGS001-115	ADCY9	Adenylyl cyclases			
883	88.33	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
884	88.28	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
885	88.24	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
886	88.22	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
887	88.21	kd	CGS001-1212	CLTB	-			
888	88.2	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
889	88.18	oe	ccsbBroad304_00954	LYN	Src family			
890	88.18	kd	CGS001-8031	NCOA4	-			
891	88.14	oe	ccsbBroad304_06783	LGMN	Legumain			
892	88.11	cp	BRD-K00673382	famotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
893	88.08	kd	CGS001-285267	ZNF619	Zinc fingers, C2H2-type			
894	87.97	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
895	87.95	oe	ccsbBroad304_02446	TADA3	-			
896	87.91	kd	CGS001-7088	TLE1	WD repeat domain containing			
897	87.89	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
898	87.86	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
899	87.86	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
900	87.85	oe	ccsbBroad304_02875	BRP44	-			
901	87.74	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
902	87.69	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
903	87.64	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
904	87.59	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
905	87.51	oe	ccsbBroad304_00170	BNIP1	-			
906	87.5	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
907	87.49	kd	CGS001-1490	CTGF	-			
908	87.47	kd	CGS001-3251	HPRT1	-			
909	87.45	kd	CGS001-7424	VEGFC	-			
910	87.44	kd	CGS001-5612	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
911	87.42	kd	CGS001-56889	TM9SF3	-			
912	87.33	kd	CGS001-23464	GCAT	-			
913	87.29	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
914	87.28	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
915	87.27	oe	ccsbBroad304_00542	FBP1	-			
916	87.26	kd	CGS001-6397	SEC14L1	-			
917	87.22	kd	CGS001-80762	NDFIP1	-			
918	87.15	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
919	87.14	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
920	87.1	kd	CGS001-55604	LRRC16A	-			
921	87.05	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
922	86.95	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
923	86.91	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
924	86.85	kd	CGS001-5345	SERPINF2	Serine (or cysteine) peptidase inhibitors			
925	86.84	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
926	86.79	oe	ccsbBroad304_02565	RALBP1	-			
927	86.77	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
928	86.75	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
929	86.74	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
930	86.74	kd	CGS001-11230	PRAF2	-			
931	86.71	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
932	86.67	kd	CGS001-7982	ST7	-			
933	86.67	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
934	86.66	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
935	86.64	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
936	86.61	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
937	86.58	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
938	86.57	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
939	86.57	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
940	86.53	kd	CGS001-6776	STAT5A	SH2 domain containing			
941	86.51	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
942	86.49	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
943	86.45	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
944	86.43	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
945	86.43	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
946	86.42	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
947	86.38	kd	CGS001-5223	PGAM1	-			
948	86.34	kd	CGS001-841	CASP8	Caspases			
949	86.32	kd	CGS001-123803	NTAN1	-			
950	86.3	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
951	86.23	cc		Mitochondrial complex IV LOF	-			
952	86.21	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
953	86.2	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
954	86.2	kd	CGS001-50810	HDGFRP3	-			
955	86.2	kd	CGS001-1211	CLTA	-			
956	86.17	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
957	86.16	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
958	86.14	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
959	86.14	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
960	86.13	kd	CGS001-6658	SOX3	SRY (sex determining region Y)-boxes			
961	86.12	kd	CGS001-865	CBFB	-			
962	86.05	kd	CGS001-55536	CDCA7L	-			
963	86.01	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
964	86	kd	CGS001-10142	AKAP9	A-kinase anchor proteins			
965	85.96	kd	CGS001-2002	ELK1	ETS Transcription Factors			
966	85.96	oe	ccsbBroad304_00238	CCNE1	-			
967	85.94	oe	ccsbBroad304_00963	SMAD5	SMADs			
968	85.94	kd	CGS001-10395	DLC1	Rho GTPase activating proteins			
969	85.93	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
970	85.91	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
971	85.9	kd	CGS001-2235	FECH	-			
972	85.89	oe	ccsbBroad304_06324	GPX7	-			
973	85.86	oe	ccsbBroad304_03618	OSGEP	-			
974	85.84	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
975	85.83	kd	CGS001-64147	KIF9	Kinesins			
976	85.82	oe	ccsbBroad304_00794	HSF1	-			
977	85.81	kd	CGS001-7106	TSPAN4	Tetraspanins			
978	85.81	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
979	85.79	kd	CGS001-563	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
980	85.75	kd	CGS001-9380	GRHPR	-			
981	85.74	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
982	85.71	cc		Dihydrofolate reductase inhibitor	-			
983	85.66	oe	ccsbBroad304_04399	PGBD1	-			
984	85.66	kd	CGS001-8649	LAMTOR3	-			
985	85.64	oe	ccsbBroad304_06720	PHYH	-			
986	85.63	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
987	85.63	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
988	85.59	kd	CGS001-5590	PRKCZ	Iota subfamily			
989	85.59	kd	CGS001-79135	APOO	Apolipoproteins			
990	85.52	oe	ccsbBroad304_02026	NRP1	CD molecules			
991	85.48	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
992	85.47	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
993	85.44	cp	BRD-K47278471	diphenhydramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
994	85.41	kd	CGS001-378	ARF4	ADP-ribosylation factors			
995	85.39	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
996	85.38	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
997	85.37	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
998	85.36	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
999	85.33	kd	CGS001-11140	CDC37	-			
1000	85.32	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
1001	85.26	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
1002	85.24	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
1003	85.18	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
1004	85.12	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
1005	85.07	oe	ccsbBroad304_00212	CAMLG	-			
1006	85.05	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1007	85.01	oe	ccsbBroad304_03269	CD320	CD molecules			
1008	84.99	kd	CGS001-205564	SENP5	-			
1009	84.98	kd	CGS001-6721	SREBF2	Basic helix-loop-helix proteins			
1010	84.95	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
1011	84.82	kd	CGS001-10939	AFG3L2	ATPases / AAA-type			
1012	84.8	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
1013	84.75	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
1014	84.74	kd	CGS001-54205	CYCS	-			
1015	84.71	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
1016	84.6	kd	CGS001-10099	TSPAN3	Tetraspanins			
1017	84.52	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
1018	84.51	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
1019	84.5	oe	ccsbBroad304_14242	MCCC2	-			
1020	84.42	oe	ccsbBroad304_04891	TMEM174	-			
1021	84.41	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
1022	84.4	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1023	84.39	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1024	84.35	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
1025	84.33	kd	CGS001-10475	TRIM38	-			
1026	84.33	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
1027	84.24	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
1028	84.19	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
1029	84.19	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1030	84.15	kd	CGS001-9217	VAPB	-			
1031	84.14	kd	CGS001-6643	SNX2	Sorting nexins			
1032	84.11	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
1033	84.1	kd	CGS001-5891	MOK	RCK family			
1034	84.08	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
1035	84.04	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
1036	84.03	oe	ccsbBroad304_09006	RPF1	-			
1037	83.99	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
1038	83.98	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
1039	83.97	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1040	83.97	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
1041	83.87	kd	CGS001-2580	GAK	Heat shock proteins / DNAJ (HSP40)			
1042	83.76	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
1043	83.73	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
1044	83.72	kd	CGS001-8795	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
1045	83.69	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
1046	83.69	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
1047	83.61	kd	CGS001-10795	ZNF268	Zinc fingers, C2H2-type			
1048	83.55	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
1049	83.54	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
1050	83.46	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
1051	83.45	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
1052	83.4	cc		CDK inhibitor	-			
1053	83.38	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
1054	83.38	kd	CGS001-3035	HARS	Aminoacyl tRNA synthetases / Class II			
1055	83.33	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
1056	83.31	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
1057	83.29	oe	ccsbBroad304_01661	TFCP2	-			
1058	83.26	kd	CGS001-1431	CS	-			
1059	83.21	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
1060	83.17	oe	ccsbBroad304_01034	MSH2	-			
1061	83.17	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
1062	83.15	oe	ccsbBroad304_08511	RFK	-			
1063	83.15	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
1064	83.15	kd	CGS001-1788	DNMT3A	Methyltransferases			
1065	83.14	kd	CGS001-6856	SYPL1	-			
1066	83.06	kd	CGS001-64750	SMURF2	-			
1067	83.04	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
1068	83.03	kd	CGS001-8805	TRIM24	TIF1 family			
1069	83.02	oe	ccsbBroad304_06645	NQO2	-			
1070	83.01	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
1071	82.98	kd	CGS001-11007	CCDC85B	-			
1072	82.97	kd	CGS001-7078	TIMP3	-			
1073	82.95	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
1074	82.95	kd	CGS001-4312	MMP1	Matrix metallopeptidase			
1075	82.89	kd	CGS001-2617	GARS	Aminoacyl tRNA synthetases / Class II			
1076	82.88	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
1077	82.88	kd	CGS001-2629	GBA	-			
1078	82.75	kd	CGS001-11232	POLG2	DNA polymerases			
1079	82.74	oe	ccsbBroad304_04387	MKI67IP	-			
1080	82.73	oe	ccsbBroad304_08993	DHDDS	-			
1081	82.67	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
1082	82.65	oe	ccsbBroad304_02438	FAM3C	-			
1083	82.63	kd	CGS001-1936	EEF1D	-			
1084	82.62	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
1085	82.58	kd	CGS001-3675	ITGA3	Integrins			
1086	82.54	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
1087	82.54	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
1088	82.52	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
1089	82.48	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
1090	82.44	kd	CGS001-2737	GLI3	Zinc fingers, C2H2-type			
1091	82.42	kd	CGS001-4507	MTAP	-			
1092	82.4	oe	ccsbBroad304_09396	TIRAP	-			
1093	82.36	kd	CGS001-1155	TBCB	-			
1094	82.3	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1095	82.28	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
1096	82.23	oe	ccsbBroad304_02220	MTFR1	-			
1097	82.23	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
1098	82.19	kd	CGS001-79712	GTDC1	Glycosyltransferase group 1 domain containing			
1099	82.12	cp	BRD-A24191444	ifenprodil	Adrenergic receptor antagonist		GRIN1, GRIN2B	Adrenergic receptor antagonist, Glutamate receptor antagonist
1100	82.1	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
1101	82.1	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
1102	82.07	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
1103	82.07	kd	CGS001-147837	ZNF563	Zinc fingers, C2H2-type			
1104	82.05	oe	ccsbBroad304_00250	CD19	CD molecules			
1105	81.96	kd	CGS001-57121	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1106	81.95	kd	CGS001-51593	SRRT	-			
1107	81.84	kd	CGS001-152	ADRA2C	GPCR / Class A : Adrenoceptors : alpha			
1108	81.8	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
1109	81.8	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
1110	81.78	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1111	81.72	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
1112	81.7	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
1113	81.68	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
1114	81.65	kd	CGS001-1675	CFD	Complement system			
1115	81.64	kd	CGS001-6990	DYNLT3	Cytoplasmic dyneins			
1116	81.63	oe	ccsbBroad304_02419	NDRG1	-			
1117	81.53	kd	CGS001-3419	IDH3A	-			
1118	81.52	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
1119	81.49	kd	CGS001-64422	ATG3	-			
1120	81.49	kd	CGS001-4795	NFKBIL1	-			
1121	81.47	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
1122	81.45	kd	CGS001-8833	GMPS	-			
1123	81.38	kd	CGS001-51720	UIMC1	-			
1124	81.37	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
1125	81.32	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
1126	81.32	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
1127	81.31	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
1128	81.28	cp	BRD-A02189320	met-leu-phe	-666			-666
1129	81.23	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
1130	81.21	kd	CGS001-10513	APPBP2	-			
1131	81.09	cp	BRD-K44442813	pidotimod	Interferon receptor agonist			Interferon receptor agonist, Interleukin receptor agonist
1132	81.09	kd	CGS001-5550	PREP	Prolyl oligopeptidase			
1133	81.07	oe	ccsbBroad304_07478	CCP110	-			
1134	81.01	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
1135	81	kd	CGS001-56616	DIABLO	-			
1136	80.96	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
1137	80.93	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
1138	80.89	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
1139	80.89	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
1140	80.89	kd	CGS001-8896	BUD31	-			
1141	80.81	kd	CGS001-4088	SMAD3	SMADs			
1142	80.81	kd	CGS001-8635	RNASET2	-			
1143	80.8	kd	CGS001-51547	SIRT7	Histone deacetylases (HDACs)			
1144	80.77	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
1145	80.72	kd	CGS001-55163	PNPO	-			
1146	80.65	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
1147	80.55	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
1148	80.55	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
1149	80.5	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
1150	80.49	kd	CGS001-1020	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
1151	80.47	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
1152	80.41	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
1153	80.4	kd	CGS001-348	APOE	Apolipoproteins			
1154	80.38	cc		Sigma receptor antagonist	-			
1155	80.37	oe	ccsbBroad304_06140	EEF1D	-			
1156	80.36	kd	CGS001-339403	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
1157	80.36	kd	CGS001-3397	ID1	Basic helix-loop-helix proteins			
1158	80.31	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
1159	80.2	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
1160	80.19	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
1161	80.17	kd	CGS001-3670	ISL1	Homeoboxes / LIM class			
1162	80.15	kd	CGS001-1384	CRAT	-			
1163	80.14	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
1164	80.14	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
1165	80.11	kd	CGS001-10295	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
1166	80.1	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
1167	80.09	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
1168	79.99	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
1169	79.93	kd	CGS001-4436	MSH2	-			
1170	79.92	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1171	79.89	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
1172	79.81	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
1173	79.78	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
1174	79.77	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
1175	79.71	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
1176	79.71	kd	CGS001-369	ARAF	RAF family			
1177	79.68	kd	CGS001-1840	DTX1	-			
1178	79.66	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1179	79.65	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
1180	79.61	oe	ccsbBroad304_01008	KITLG	-			
1181	79.58	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
1182	79.58	kd	CGS001-5511	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1183	79.57	kd	CGS001-328	APEX1	-			
1184	79.56	kd	CGS001-57147	SCYL3	-			
1185	79.53	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1186	79.47	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
1187	79.43	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
1188	79.41	kd	CGS001-3428	IFI16	-			
1189	79.39	oe	ccsbBroad304_00665	GOT1	-			
1190	79.36	kd	CGS001-10827	FAM114A2	-			
1191	79.36	kd	CGS001-23210	JMJD6	-			
1192	79.33	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
1193	79.32	kd	CGS001-22850	ADNP2	Zinc fingers, C2H2-type			
1194	79.29	kd	CGS001-5906	RAP1A	-			
1195	79.29	kd	CGS001-3373	HYAL1	-			
1196	79.26	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
1197	79.23	kd	CGS001-835	CASP2	Caspases			
1198	79.21	kd	CGS001-1891	ECH1	-			
1199	79.2	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
1200	79.19	kd	CGS001-10888	GPR83	GPCR / Class A : Orphans			
1201	79.17	oe	ccsbBroad304_04775	NTAN1	-			
1202	79.16	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
1203	79.15	oe	ccsbBroad304_05098	MAGEB6	-			
1204	79.09	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
1205	79.01	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1206	79.01	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
1207	78.99	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1208	78.98	cp	BRD-A23637604	oxymetholone	Androgen receptor agonist		AR	Androgen receptor agonist
1209	78.98	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
1210	78.98	kd	CGS001-7150	TOP1	DNA Topoisomerases			
1211	78.93	kd	CGS001-4860	PNP	-			
1212	78.92	oe	ccsbBroad304_00941	LIG3	-			
1213	78.92	oe	ccsbBroad304_02318	KIF20A	Kinesins			
1214	78.92	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
1215	78.9	cp	BRD-K52080565	rilmenidine	Imidazoline receptor agonist		NISCH	Imidazoline receptor agonist
1216	78.82	kd	CGS001-5925	RB1	Endogenous ligands			
1217	78.72	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
1218	78.72	kd	CGS001-10670	RRAGA	-			
1219	78.71	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
1220	78.68	kd	CGS001-2805	GOT1	-			
1221	78.67	kd	CGS001-23659	PLA2G15	-			
1222	78.66	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
1223	78.62	kd	CGS001-2539	G6PD	-			
1224	78.62	oe	ccsbBroad304_00993	MDM4	-			
1225	78.57	kd	CGS001-11015	KDELR3	-			
1226	78.48	oe	ccsbBroad304_02566	MORF4L1	-			
1227	78.44	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
1228	78.41	oe	ccsbBroad304_01675	TK1	-			
1229	78.41	kd	CGS001-8891	EIF2B3	-			
1230	78.4	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1231	78.38	kd	CGS001-7360	UGP2	-			
1232	78.31	cc		IGF-1 inhibitor	-			
1233	78.31	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
1234	78.28	kd	CGS001-27346	TMEM97	-			
1235	78.27	kd	CGS001-3976	LIF	-			
1236	78.27	kd	CGS001-408	ARRB1	-			
1237	78.19	kd	CGS001-51752	ERAP1	Aminopeptidase N			
1238	78.16	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
1239	78.14	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
1240	78.09	kd	CGS001-11284	PNKP	-			
1241	78.07	kd	CGS001-8974	P4HA2	-			
1242	78.01	kd	CGS001-10645	CAMKK2	Meta subfamily			
1243	77.98	kd	CGS001-10901	DHRS4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1244	77.98	oe	ccsbBroad304_01091	NFIB	-			
1245	77.91	kd	CGS001-51495	PTPLAD1	-			
1246	77.9	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
1247	77.85	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
1248	77.79	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
1249	77.74	oe	ccsbBroad304_01398	RHEB	-			
1250	77.74	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
1251	77.69	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
1252	77.66	kd	CGS001-25	ABL1	Abl family			
1253	77.65	oe	ccsbBroad304_01165	PDK1	-			
1254	77.65	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
1255	77.64	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
1256	77.62	kd	CGS001-3488	IGFBP5	insulin-like growth factor (IGF) binding proteins			
1257	77.6	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
1258	77.6	kd	CGS001-25898	RCHY1	RING-type (C3HC4) zinc fingers			
1259	77.56	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
1260	77.55	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
1261	77.53	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
1262	77.53	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
1263	77.52	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
1264	77.51	kd	CGS001-10557	RPP38	-			
1265	77.48	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
1266	77.43	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
1267	77.41	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
1268	77.39	oe	ccsbBroad304_01163	PDHA1	-			
1269	77.38	oe	ccsbBroad304_03357	RASD1	-			
1270	77.37	kd	CGS001-55968	NSFL1C	UBX domain containing			
1271	77.36	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
1272	77.34	oe	ccsbBroad304_02956	EHF	-			
1273	77.26	kd	CGS001-513	ATP5D	ATPases / F-type			
1274	77.22	kd	CGS001-57018	CCNL1	-			
1275	77.18	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
1276	77.15	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
1277	77.14	kd	CGS001-10401	PIAS3	Zinc fingers, MIZ-type			
1278	77.12	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
1279	77.08	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
1280	77.04	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
1281	77.01	oe	ccsbBroad304_07080	TM7SF2	-			
1282	77	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
1283	76.94	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
1284	76.93	cp	BRD-K94887716	TFMPP	Serotonin receptor agonist			Serotonin receptor agonist, Serotonin receptor antagonist
1285	76.93	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
1286	76.89	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
1287	76.87	kd	CGS001-2475	MTOR	FRAP subfamily			
1288	76.85	kd	CGS001-64077	LHPP	-			
1289	76.82	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
1290	76.8	kd	CGS001-55793	FAM63A	-			
1291	76.78	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
1292	76.77	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
1293	76.69	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
1294	76.68	kd	CGS001-5194	PEX13	-			
1295	76.66	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
1296	76.64	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
1297	76.64	oe	ccsbBroad304_00648	GLRX	-			
1298	76.62	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
1299	76.59	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
1300	76.54	kd	CGS001-7525	YES1	Src family			
1301	76.48	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
1302	76.48	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
1303	76.46	kd	CGS001-29998	GLTSCR1	-			
1304	76.44	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
1305	76.41	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
1306	76.41	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1307	76.37	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
1308	76.27	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
1309	76.25	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
1310	76.2	kd	CGS001-169792	GLIS3	Zinc fingers, C2H2-type			
1311	76.2	oe	ccsbBroad304_07832	XPO7	Exportins			
1312	76.16	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
1313	76.13	kd	CGS001-7280	TUBB2A	Tubulins			
1314	76.12	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
1315	76.12	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
1316	76.12	kd	CGS001-578	BAK1	-			
1317	76.02	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
1318	75.92	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
1319	75.91	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
1320	75.91	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
1321	75.86	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
1322	75.85	kd	CGS001-5111	PCNA	-			
1323	75.85	kd	CGS001-892	CCNC	-			
1324	75.77	cp	BRD-K54316499	tolterodine	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRM1, CHRM4, CHRM5	Acetylcholine receptor antagonist
1325	75.75	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
1326	75.73	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
1327	75.65	kd	CGS001-2004	ELK3	ETS Transcription Factors			
1328	75.64	kd	CGS001-587	BCAT2	-			
1329	75.62	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
1330	75.62	kd	CGS001-2565	GABRG1	GABA receptors			
1331	75.6	kd	CGS001-8731	RNMT	-			
1332	75.52	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
1333	75.51	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
1334	75.5	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
1335	75.42	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
1336	75.41	kd	CGS001-154197	PNLDC1	-			
1337	75.38	kd	CGS001-1727	CYB5R3	-			
1338	75.37	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
1339	75.35	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
1340	75.31	kd	CGS001-23530	NNT	-			
1341	75.27	kd	CGS001-374291	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
1342	75.26	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
1343	75.26	kd	CGS001-8572	PDLIM4	-			
1344	75.17	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
1345	75.15	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
1346	75.14	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1347	75.11	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
1348	75.11	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
1349	75.07	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
1350	75.07	kd	CGS001-56916	SMARCAD1	-			
1351	75.05	cc		JAK inhibitor	-			
1352	75.01	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
1353	74.94	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
1354	74.93	kd	CGS001-56993	TOMM22	-			
1355	74.91	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1356	74.88	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
1357	74.85	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
1358	74.81	kd	CGS001-3170	FOXA2	Forkhead boxes			
1359	74.79	oe	ccsbBroad304_00617	GBA	-			
1360	74.79	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
1361	74.78	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
1362	74.75	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
1363	74.74	kd	CGS001-8061	FOSL1	basic leucine zipper proteins			
1364	74.72	kd	CGS001-9159	PCSK7	Subtilisin			
1365	74.71	kd	CGS001-10553	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
1366	74.7	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
1367	74.67	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
1368	74.59	kd	CGS001-6709	SPTAN1	EF-hand domain containing			
1369	74.54	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
1370	74.46	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
1371	74.44	kd	CGS001-4043	LRPAP1	-			
1372	74.41	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
1373	74.37	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
1374	74.33	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
1375	74.29	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
1376	74.26	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
1377	74.26	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
1378	74.24	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
1379	74.2	kd	CGS001-342926	ZNF677	Zinc fingers, C2H2-type			
1380	74.19	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
1381	74.16	oe	ccsbBroad304_08898	TRAK2	-			
1382	74.14	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
1383	74.05	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
1384	74.04	kd	CGS001-6778	STAT6	SH2 domain containing			
1385	74.01	kd	CGS001-2837	UTS2R	Urotensin receptor			
1386	73.97	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
1387	73.85	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
1388	73.83	cp	BRD-K82795137	loratadine	Histamine receptor antagonist		HRH1, CYP2C19, CYP3A5	Histamine receptor antagonist
1389	73.83	kd	CGS001-10227	MFSD10	-			
1390	73.73	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
1391	73.72	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
1392	73.72	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
1393	73.69	oe	ccsbBroad304_06282	GLDC	-			
1394	73.65	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
1395	73.65	kd	CGS001-55206	SBNO1	-			
1396	73.63	oe	ccsbBroad304_03164	MTERFD1	-			
1397	73.62	kd	CGS001-2969	GTF2I	General transcription factors			
1398	73.62	kd	CGS001-160	AP2A1	-			
1399	73.56	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
1400	73.56	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
1401	73.55	kd	CGS001-7846	TUBA1A	Tubulins			
1402	73.53	kd	CGS001-2203	FBP1	-			
1403	73.43	kd	CGS001-3460	IFNGR2	Interferon receptor family			
1404	73.43	kd	CGS001-3383	ICAM1	CD molecules			
1405	73.41	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
1406	73.37	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
1407	73.34	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
1408	73.28	kd	CGS001-84647	PLA2G12B	-			
1409	73.28	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
1410	73.18	cp	BRD-K50938287	sumatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1A, HTR1F, HTR1E, HTR5A, HTR6, HTR7	Serotonin receptor agonist
1411	73.11	kd	CGS001-132	ADK	Adenosine turnover			
1412	73.11	oe	ccsbBroad304_09615	LACC1	-			
1413	73.09	kd	CGS001-5591	PRKDC	Other PIKK family kinases			
1414	73.08	oe	ccsbBroad304_02368	TIMM17B	-			
1415	73.07	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
1416	73.06	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1417	73.06	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1418	73.05	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
1419	73.04	oe	ccsbBroad304_01183	PGD	-			
1420	73.02	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
1421	73.02	kd	CGS001-57680	CHD8	-			
1422	73.01	kd	CGS001-1312	COMT	Catecholamine turnover			
1423	72.87	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
1424	72.87	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
1425	72.82	kd	CGS001-5019	OXCT1	-			
1426	72.77	kd	CGS001-976	CD97	Adhesion Class GPCRs			
1427	72.75	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
1428	72.69	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
1429	72.69	kd	CGS001-4267	CD99	CD molecules			
1430	72.69	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1431	72.64	kd	CGS001-775	CACNA1C	Calcium channel subunits			
1432	72.63	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
1433	72.61	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
1434	72.57	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1435	72.55	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
1436	72.43	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
1437	72.42	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
1438	72.41	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
1439	72.4	kd	CGS001-162699	TCEB3C	-			
1440	72.35	kd	CGS001-3920	LAMP2	CD molecules			
1441	72.35	kd	CGS001-790	CAD	-			
1442	72.32	kd	CGS001-10915	TCERG1	-			
1443	72.27	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
1444	72.27	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
1445	72.18	kd	CGS001-375	ARF1	ADP-ribosylation factors			
1446	72.17	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1447	72.16	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
1448	72.08	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
1449	72.07	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
1450	72.06	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1451	72	kd	CGS001-8624	PSMG1	-			
1452	71.91	kd	CGS001-6810	STX4	-			
1453	71.86	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
1454	71.86	kd	CGS001-2184	FAH	-			
1455	71.8	oe	ccsbBroad304_06820	PTS	-			
1456	71.77	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
1457	71.74	cc		Norepinephrine reuptake inhibitor	-			
1458	71.74	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
1459	71.72	oe	ccsbBroad304_02596	KDELR3	-			
1460	71.69	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
1461	71.67	oe	ccsbBroad304_06852	RBP4	Lipocalins			
1462	71.66	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1463	71.64	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
1464	71.63	cc		Ribonucleotide reductase inhibitor	-			
1465	71.6	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
1466	71.42	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
1467	71.42	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
1468	71.35	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
1469	71.33	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
1470	71.28	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
1471	71.26	kd	CGS001-51684	SUFU	-			
1472	71.21	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
1473	71.18	cc		EIF Proteins LOF	-			
1474	71.18	kd	CGS001-1676	DFFA	-			
1475	71.17	oe	ccsbBroad304_00282	CDKN1A	-			
1476	71.17	kd	CGS001-1513	CTSK	Cathepsins			
1477	71.15	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
1478	71.11	kd	CGS001-4605	MYBL2	-			
1479	71.1	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
1480	71.07	kd	CGS001-2295	FOXF2	Forkhead boxes			
1481	71.02	kd	CGS001-124535	HSF5	-			
1482	71	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
1483	71	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
1484	70.99	kd	CGS001-1509	CTSD	Cathepsins			
1485	70.94	kd	CGS001-2810	SFN	-			
1486	70.9	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
1487	70.9	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
1488	70.89	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
1489	70.86	oe	ccsbBroad304_07561	YAF2	-			
1490	70.84	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
1491	70.83	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
1492	70.82	kd	CGS001-8527	DGKD	Pleckstrin homology (PH) domain containing			
1493	70.8	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1494	70.78	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
1495	70.78	kd	CGS001-28985	MCTS1	-			
1496	70.76	oe	ccsbBroad304_02815	SSBP2	-			
1497	70.76	oe	ccsbBroad304_01985	EIF3H	-			
1498	70.75	kd	CGS001-6799	SULT1A2	Sulfotransferases, cytosolic			
1499	70.73	oe	ccsbBroad304_02197	VPS26A	-			
1500	70.72	kd	CGS001-9453	GGPS1	Lanosterol biosynthesis pathway			
1501	70.71	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
1502	70.68	kd	CGS001-8678	BECN1	-			
1503	70.61	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
1504	70.58	kd	CGS001-4287	ATXN3	Ataxins			
1505	70.52	cc		Phospholipases LOF	-			
1506	70.41	oe	ccsbBroad304_02845	PRPF6	-			
1507	70.38	kd	CGS001-9926	LPGAT1	-			
1508	70.34	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
1509	70.29	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
1510	70.26	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
1511	70.25	oe	ccsbBroad304_06998	SRPK1	SRPK family			
1512	70.24	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
1513	70.22	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
1514	70.22	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
1515	70.21	kd	CGS001-4254	KITLG	-			
1516	70.19	kd	CGS001-6790	AURKA	Aurora kinase			
1517	70.13	kd	CGS001-4925	NUCB2	EF-hand domain containing			
1518	70.06	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
1519	70.05	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
1520	70.05	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
1521	70.05	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
1522	70.04	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
1523	70.02	kd	CGS001-9975	NR1D2	Rev-Erb receptors			
1524	70.02	kd	CGS001-2260	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
1525	69.99	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1526	69.98	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
1527	69.89	kd	CGS001-5613	PRKX	Protein kinase A			
1528	69.85	kd	CGS001-55644	OSGEP	-			
1529	69.84	kd	CGS001-5471	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
1530	69.81	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
1531	69.75	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1532	69.7	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
1533	69.7	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
1534	69.68	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
1535	69.68	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
1536	69.66	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
1537	69.65	kd	CGS001-140612	ZFP28	Zinc fingers, C2H2-type			
1538	69.62	kd	CGS001-701	BUB1B	Bub family			
1539	69.61	kd	CGS001-80714	PBX4	Homeoboxes / TALE class			
1540	69.57	kd	CGS001-6502	SKP2	F-boxes / Leucine-rich repeats			
1541	69.56	oe	ccsbBroad304_03554	NAT10	-			
1542	69.55	cc		Kinase anchoring proteins LOF	-			
1543	69.54	kd	CGS001-9709	HERPUD1	-			
1544	69.44	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
1545	69.39	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
1546	69.32	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
1547	69.32	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
1548	69.3	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
1549	69.19	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
1550	69.18	oe	ccsbBroad304_03874	UBL5	-			
1551	69.18	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
1552	69.16	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
1553	69.16	kd	CGS001-486	FXYD2	Ion transport regulator			
1554	69.14	oe	ccsbBroad304_00423	DAXX	-			
1555	69.1	oe	ccsbBroad304_02361	MFSD10	-			
1556	69.09	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
1557	69.08	kd	CGS001-81577	GFOD2	-			
1558	69.04	kd	CGS001-8027	STAM	-			
1559	69.02	kd	CGS001-8985	PLOD3	-			
1560	69.02	kd	CGS001-2876	GPX1	-			
1561	68.96	kd	CGS001-1810	DR1	-			
1562	68.87	oe	ccsbBroad304_13880	IDH3G	-			
1563	68.87	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
1564	68.87	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
1565	68.8	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
1566	68.73	kd	CGS001-3638	INSIG1	-			
1567	68.55	kd	CGS001-5050	PAFAH1B3	-			
1568	68.53	kd	CGS001-5198	PFAS	-			
1569	68.5	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
1570	68.46	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
1571	68.42	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
1572	68.39	cp	BRD-K46435977	valaciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
1573	68.29	kd	CGS001-1854	DUT	-			
1574	68.27	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
1575	68.24	oe	ccsbBroad304_06318	GPER	-			
1576	68.24	kd	CGS001-57154	SMURF1	-			
1577	68.22	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
1578	68.2	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
1579	68.19	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
1580	68.18	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
1581	68.16	cp	BRD-K92413528	thiazolidinecarboxylic-acid	Reducing agent			Reducing agent
1582	68.06	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
1583	68.06	kd	CGS001-271	AMPD2	-			
1584	67.95	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
1585	67.95	kd	CGS001-6654	SOS1	Rho guanine nucleotide exchange factors			
1586	67.95	kd	CGS001-11041	B3GNT1	-			
1587	67.9	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
1588	67.9	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
1589	67.81	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
1590	67.77	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
1591	67.76	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
1592	67.72	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
1593	67.66	oe	ccsbBroad304_06144	EFNB3	Ephrins			
1594	67.66	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
1595	67.66	kd	CGS001-3242	HPD	Oxidoreductases			
1596	67.62	kd	CGS001-182	JAG1	CD molecules			
1597	67.59	kd	CGS001-6050	RNH1	-			
1598	67.58	kd	CGS001-1493	CTLA4	CD molecules			
1599	67.54	kd	CGS001-306	ANXA3	Annexins			
1600	67.5	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
1601	67.43	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
1602	67.43	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
1603	67.33	kd	CGS001-11004	KIF2C	Kinesins			
1604	67.29	kd	CGS001-1407	CRY1	-			
1605	67.27	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
1606	67.22	kd	CGS001-817	CAMK2D	CAMK2 family			
1607	67.21	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
1608	67.2	kd	CGS001-29899	GPSM2	Tetratricopeptide (TTC) repeat domain containing			
1609	67.19	kd	CGS001-23161	SNX13	Sorting nexins			
1610	67.18	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
1611	67.13	kd	CGS001-11198	SUPT16H	-			
1612	67.11	kd	CGS001-5460	POU5F1	Homeoboxes / POU class			
1613	67.08	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
1614	67.07	kd	CGS001-5744	PTHLH	Endogenous ligands			
1615	67.05	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
1616	67.05	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
1617	67.02	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
1618	67	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
1619	66.97	kd	CGS001-2768	GNA12	-			
1620	66.96	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
1621	66.88	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1622	66.87	oe	ccsbBroad304_00819	IDH3B	-			
1623	66.81	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
1624	66.77	kd	CGS001-26064	RAI14	Ankyrin repeat domain containing			
1625	66.72	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
1626	66.62	oe	ccsbBroad304_00632	GGCX	Carboxylases			
1627	66.57	kd	CGS001-5608	MAP2K6	MAPKK:STE7 family			
1628	66.54	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
1629	66.5	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1630	66.49	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
1631	66.48	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
1632	66.44	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
1633	66.4	oe	ccsbBroad304_05887	CFB	Complement system			
1634	66.39	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1635	66.39	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
1636	66.38	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
1637	66.37	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
1638	66.37	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
1639	66.32	kd	CGS001-3418	IDH2	-			
1640	66.3	oe	ccsbBroad304_08023	EIF2C1	-			
1641	66.29	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
1642	66.18	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
1643	66.13	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
1644	66.11	kd	CGS001-51545	ZNF581	Zinc fingers, C2H2-type			
1645	66.1	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
1646	66.1	oe	ccsbBroad304_06383	HMMR	CD molecules			
1647	66.04	kd	CGS001-18	ABAT	GABA turnover			
1648	66.02	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
1649	66.01	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
1650	65.98	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
1651	65.84	kd	CGS001-7184	HSP90B1	Heat shock proteins / HSPC			
1652	65.81	oe	ccsbBroad304_03072	GTPBP8	-			
1653	65.77	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
1654	65.75	kd	CGS001-8802	SUCLG1	-			
1655	65.74	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
1656	65.74	kd	CGS001-113878	DTX2	RING-type (C3HC4) zinc fingers			
1657	65.7	oe	ccsbBroad304_00237	CCND3	-			
1658	65.58	oe	ccsbBroad304_05981	CDO1	-			
1659	65.58	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1660	65.57	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
1661	65.56	kd	CGS001-11319	ECD	-			
1662	65.55	kd	CGS001-1949	EFNB3	Ephrins			
1663	65.54	kd	CGS001-3421	IDH3G	-			
1664	65.52	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1665	65.47	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
1666	65.44	kd	CGS001-7016	TESK1	TESK subfamily			
1667	65.42	oe	ccsbBroad304_01101	NME1	-			
1668	65.39	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
1669	65.38	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
1670	65.33	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
1671	65.33	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1672	65.29	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
1673	65.28	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
1674	65.26	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
1675	65.25	kd	CGS001-5320	PLA2G2A	Hydrolases			
1676	65.17	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
1677	65.13	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
1678	65.1	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
1679	65.1	kd	CGS001-3778	KCNMA1	Calcium-activated potassium channels			
1680	65.06	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
1681	64.96	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
1682	64.9	kd	CGS001-1027	CDKN1B	-			
1683	64.87	kd	CGS001-10342	TFG	-			
1684	64.82	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
1685	64.8	oe	ccsbBroad304_02163	MED7	-			
1686	64.73	kd	CGS001-84159	ARID5B	-			
1687	64.7	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
1688	64.68	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
1689	64.68	kd	CGS001-9559	VPS26A	-			
1690	64.64	kd	CGS001-1837	DTNA	-			
1691	64.53	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
1692	64.49	kd	CGS001-6603	SMARCD2	-			
1693	64.48	kd	CGS001-3689	ITGB2	Integrins			
1694	64.47	oe	ccsbBroad304_02195	SPAG7	-			
1695	64.44	kd	CGS001-11243	PMF1	-			
1696	64.43	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
1697	64.34	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
1698	64.31	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
1699	64.29	kd	CGS001-80025	PANK2	-			
1700	64.28	oe	ccsbBroad304_03746	CDC42SE1	-			
1701	64.28	kd	CGS001-8569	MKNK1	MKN subfamily			
1702	64.23	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
1703	64.18	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
1704	64.16	oe	ccsbBroad304_14143	NUSAP1	-			
1705	64.15	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
1706	64.12	kd	CGS001-5624	PROC	Endogenous ligands			
1707	63.97	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
1708	63.96	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
1709	63.95	kd	CGS001-51586	MED15	-			
1710	63.95	kd	CGS001-1605	DAG1	-			
1711	63.93	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
1712	63.92	kd	CGS001-8837	CFLAR	Endogenous ligands			
1713	63.9	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
1714	63.9	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
1715	63.87	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
1716	63.82	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1717	63.78	kd	CGS001-427	ASAH1	Acid ceramidase			
1718	63.76	kd	CGS001-3416	IDE	Pitrilysin			
1719	63.75	kd	CGS001-203	AK1	Adenylate kinases			
1720	63.74	kd	CGS001-84936	ZFYVE19	Zinc fingers, FYVE domain containing			
1721	63.74	kd	CGS001-93594	WDR67	-			
1722	63.61	kd	CGS001-29915	HCFC2	-			
1723	63.59	kd	CGS001-3880	KRT19	Intermediate filaments type I, keratins (acidic)			
1724	63.53	kd	CGS001-8669	EIF3J	-			
1725	63.45	kd	CGS001-3032	HADHB	-			
1726	63.45	kd	CGS001-1974	EIF4A2	DEAD-boxes			
1727	63.41	oe	ccsbBroad304_08839	IFIH1	-			
1728	63.4	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
1729	63.39	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
1730	63.31	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
1731	63.29	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
1732	63.24	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
1733	63.24	kd	CGS001-10721	POLQ	DNA polymerases			
1734	63.16	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
1735	63.15	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
1736	63.12	kd	CGS001-27161	EIF2C2	-			
1737	63.11	kd	CGS001-25797	QPCT	Aminopeptidase Y			
1738	63.06	oe	ccsbBroad304_00501	EMD	-			
1739	63.05	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
1740	63.04	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
1741	63.02	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
1742	63.02	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
1743	63.01	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
1744	63.01	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
1745	62.94	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
1746	62.93	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
1747	62.85	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
1748	62.79	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
1749	62.74	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
1750	62.72	kd	CGS001-3995	FADS3	Fatty acid desaturases			
1751	62.67	kd	CGS001-6767	ST13	Tetratricopeptide (TTC) repeat domain containing			
1752	62.65	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
1753	62.61	kd	CGS001-1495	CTNNA1	Catenins			
1754	62.55	kd	CGS001-6884	TAF13	-			
1755	62.54	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
1756	62.54	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
1757	62.54	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
1758	62.53	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
1759	62.5	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
1760	62.48	kd	CGS001-7508	XPC	-			
1761	62.47	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
1762	62.45	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
1763	62.29	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
1764	62.27	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
1765	62.22	kd	CGS001-9797	TATDN2	-			
1766	62.21	oe	ccsbBroad304_01114	NUP88	-			
1767	62.21	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
1768	61.86	kd	CGS001-3123	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
1769	61.82	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
1770	61.81	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
1771	61.79	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
1772	61.78	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
1773	61.75	kd	CGS001-3718	JAK3	Janus kinase (JakA) family			
1774	61.72	kd	CGS001-6591	SNAI2	Snail homologs			
1775	61.7	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
1776	61.69	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
1777	61.65	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
1778	61.65	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
1779	61.62	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
1780	61.61	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
1781	61.59	kd	CGS001-4864	NPC1	-			
1782	61.57	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
1783	61.56	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
1784	61.53	kd	CGS001-3939	LDHA	-			
1785	61.52	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
1786	61.52	kd	CGS001-10058	ABCB6	ATP binding cassette transporters / subfamily B			
1787	61.45	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
1788	61.4	cc		FGFR inhibitor	-			
1789	61.37	kd	CGS001-1072	CFL1	-			
1790	61.36	oe	ccsbBroad304_06458	IRF3	-			
1791	61.34	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
1792	61.32	kd	CGS001-5997	RGS2	Endogenous ligands			
1793	61.29	kd	CGS001-2957	GTF2A1	General transcription factors			
1794	61.23	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
1795	61.17	kd	CGS001-1594	CYP27B1	Cytochrome P450s			
1796	61.16	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1797	61.16	kd	CGS001-58492	ZNF77	Zinc fingers, C2H2-type			
1798	61.15	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
1799	61.09	kd	CGS001-340371	NRBP2	NRBP family			
1800	61.04	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
1801	61.03	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
1802	61.01	oe	ccsbBroad304_00509	EPHX1	-			
1803	60.95	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
1804	60.91	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
1805	60.91	kd	CGS001-2961	GTF2E2	General transcription factors			
1806	60.89	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
1807	60.86	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
1808	60.84	kd	CGS001-11214	AKAP13	A-kinase anchor proteins			
1809	60.83	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
1810	60.82	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
1811	60.8	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
1812	60.78	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
1813	60.78	kd	CGS001-607	BCL9	-			
1814	60.75	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
1815	60.74	kd	CGS001-116832	RPL39L	L ribosomal proteins			
1816	60.67	kd	CGS001-4194	MDM4	-			
1817	60.49	oe	ccsbBroad304_07102	TSG101	-			
1818	60.46	kd	CGS001-5734	PTGER4	GPCR / Class A : Prostanoid receptors			
1819	60.45	kd	CGS001-51569	UFM1	-			
1820	60.44	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
1821	60.35	kd	CGS001-54107	POLE3	DNA polymerases			
1822	60.35	kd	CGS001-1196	CLK2	CDC-like kinases			
1823	60.34	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
1824	60.29	cp	BRD-A75935363	atracurium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
1825	60.25	kd	CGS001-3693	ITGB5	Integrins			
1826	60.25	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
1827	60.19	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
1828	60.18	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
1829	60.18	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
1830	60.18	kd	CGS001-10928	RALBP1	-			
1831	60.17	oe	ccsbBroad304_01974	RNASET2	-			
1832	60.16	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
1833	60.16	kd	CGS001-83694	RPS6KL1	RSKL family			
1834	60.15	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
1835	60.14	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
1836	60.1	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
1837	60.1	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
1838	60.05	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
1839	60	oe	ccsbBroad304_02890	SYF2	-			
1840	59.94	oe	ccsbBroad304_07651	HEXIM1	-			
1841	59.86	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
1842	59.83	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
1843	59.83	kd	CGS001-2099	ESR1	Estrogen receptors			
1844	59.82	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
1845	59.82	kd	CGS001-10476	ATP5H	ATPases / F-type			
1846	59.8	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
1847	59.76	oe	ccsbBroad304_06985	SORD	-			
1848	59.74	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
1849	59.71	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
1850	59.69	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
1851	59.69	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
1852	59.6	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
1853	59.59	oe	ccsbBroad304_00226	CAV1	-			
1854	59.58	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
1855	59.52	oe	ccsbBroad304_09503	KLHDC9	-			
1856	59.52	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
1857	59.51	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
1858	59.5	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
1859	59.49	kd	CGS001-10318	TNIP1	-			
1860	59.46	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
1861	59.43	kd	CGS001-857	CAV1	-			
1862	59.42	kd	CGS001-29984	RHOD	-			
1863	59.38	oe	ccsbBroad304_01723	TTK	TTK family			
1864	59.3	oe	ccsbBroad304_06301	GOT2	-			
1865	59.3	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
1866	59.24	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
1867	59.22	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
1868	59.19	kd	CGS001-2787	GNG5	-			
1869	59.16	cp	BRD-K13664374	dichloroacetic-acid	Pyruvate dehydrogenase kinase inhibitor		PDK1	Pyruvate dehydrogenase kinase inhibitor
1870	59.16	kd	CGS001-7024	TFCP2	-			
1871	59.05	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
1872	59.05	kd	CGS001-6793	STK10	SLK subfamily			
1873	59.04	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
1874	59.04	kd	CGS001-10632	ATP5L	ATPases / F-type			
1875	58.96	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
1876	58.96	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
1877	58.94	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
1878	58.93	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
1879	58.93	kd	CGS001-6595	SMARCA2	Non-enzymatic BRD containing proteins			
1880	58.9	oe	ccsbBroad304_02094	FIBP	-			
1881	58.85	kd	CGS001-5328	PLAU	Chymotrypsin			
1882	58.81	oe	ccsbBroad304_02579	YWHAQ	-			
1883	58.77	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
1884	58.72	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
1885	58.69	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
1886	58.67	kd	CGS001-23461	ABCA5	ATP binding cassette transporters / subfamily A			
1887	58.65	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
1888	58.61	kd	CGS001-9406	ZRANB2	Zinc fingers, RAN-binding domain containing			
1889	58.6	kd	CGS001-9261	MAPKAPK2	MAPKAPK subfamily			
1890	58.58	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
1891	58.56	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
1892	58.54	kd	CGS001-51441	YTHDF2	-			
1893	58.5	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
1894	58.43	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
1895	58.43	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
1896	58.43	kd	CGS001-7913	DEK	-			
1897	58.38	oe	ccsbBroad304_06286	GLUL	-			
1898	58.38	kd	CGS001-5660	PSAP	Endogenous ligands			
1899	58.38	kd	CGS001-23344	ESYT1	Synaptotagmins			
1900	58.31	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
1901	58.26	cc		Aminoacyl tRNA synthetases class II LOF	-			
1902	58.25	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
1903	58.23	oe	ccsbBroad304_07280	LAMTOR3	-			
1904	58.22	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
1905	58.19	oe	ccsbBroad304_01845	RDBP	-			
1906	58.16	kd	CGS001-4773	NFATC2	Nuclear factor of activated T-cells			
1907	58.1	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
1908	58.09	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
1909	58.08	cp	BRD-K22009844	phenprobamate	Muscle relaxant			Muscle relaxant
1910	58.08	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
1911	58.05	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
1912	58.02	kd	CGS001-5167	ENPP1	-			
1913	58.01	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
1914	58.01	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1915	57.98	oe	ccsbBroad304_03047	BZW2	-			
1916	57.98	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
1917	57.97	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
1918	57.95	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
1919	57.88	kd	CGS001-3895	KTN1	-			
1920	57.87	kd	CGS001-8692	HYAL2	-			
1921	57.86	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
1922	57.84	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
1923	57.81	kd	CGS001-4616	GADD45B	-			
1924	57.8	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
1925	57.79	kd	CGS001-5888	RAD51	-			
1926	57.76	oe	ccsbBroad304_06718	PFN2	-			
1927	57.69	kd	CGS001-139135	PASD1	-			
1928	57.67	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
1929	57.67	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
1930	57.63	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
1931	57.62	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
1932	57.52	kd	CGS001-55107	ANO1	Calcium activated chloride channel			
1933	57.5	oe	ccsbBroad304_02414	IRF9	-			
1934	57.41	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
1935	57.41	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
1936	57.39	oe	ccsbBroad304_01832	PAX8	Paired boxes			
1937	57.36	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
1938	57.36	kd	CGS001-8841	HDAC3	Histone deacetylases			
1939	57.3	kd	CGS001-80349	WDR61	WD repeat domain containing			
1940	57.29	cc		Androgen receptor modulator	-			
1941	57.23	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
1942	57.1	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
1943	57.09	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1944	57.01	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
1945	57	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
1946	56.93	oe	ccsbBroad304_00991	MDH1	-			
1947	56.92	kd	CGS001-54807	ZNF586	Zinc fingers, C2H2-type			
1948	56.91	kd	CGS001-25801	GCA	EF-hand domain containing			
1949	56.86	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
1950	56.78	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
1951	56.58	oe	ccsbBroad304_07401	TXNL1	-			
1952	56.53	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
1953	56.5	kd	CGS001-51347	TAOK3	TAO subfamily			
1954	56.49	oe	ccsbBroad304_06651	NOV	-			
1955	56.49	kd	CGS001-10745	PHTF1	-			
1956	56.48	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
1957	56.45	kd	CGS001-57007	CXCR7	-			
1958	56.41	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
1959	56.35	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
1960	56.34	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
1961	56.28	kd	CGS001-4069	LYZ	-			
1962	56.26	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
1963	56.23	kd	CGS001-9156	EXO1	-			
1964	56.13	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
1965	56.12	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
1966	56.1	kd	CGS001-6605	SMARCE1	-			
1967	56.08	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
1968	56.05	kd	CGS001-51776	ZAK	MLK subfamily			
1969	56.05	kd	CGS001-2023	ENO1	-			
1970	56.03	oe	ccsbBroad304_03928	RRAGC	-			
1971	56.03	kd	CGS001-8834	TMEM11	-			
1972	56	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
1973	56	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
1974	55.97	kd	CGS001-5686	PSMA5	Proteasome subunits			
1975	55.95	oe	ccsbBroad304_06234	G6PC	-			
1976	55.95	oe	ccsbBroad304_00034	AES	-			
1977	55.95	kd	CGS001-9847	KIAA0528	-			
1978	55.93	oe	ccsbBroad304_02990	LYPD3	-			
1979	55.88	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
1980	55.87	oe	ccsbBroad304_02340	SORBS3	-			
1981	55.82	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
1982	55.79	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
1983	55.77	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
1984	55.71	kd	CGS001-57657	HCN3	Cyclic nucleotide-regulated channels			
1985	55.67	oe	ccsbBroad304_06382	HMGCL	-			
1986	55.66	cc		DNA polymerase inhibitor	-			
1987	55.66	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
1988	55.65	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
1989	55.62	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
1990	55.58	kd	CGS001-1659	DHX8	DEAH-boxes			
1991	55.51	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
1992	55.49	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
1993	55.47	kd	CGS001-3053	SERPIND1	Serine (or cysteine) peptidase inhibitors			
1994	55.46	oe	ccsbBroad304_02205	WTAP	-			
1995	55.46	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
1996	55.46	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
1997	55.45	kd	CGS001-8893	EIF2B5	-			
1998	55.43	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
1999	55.41	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
2000	55.38	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
2001	55.37	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2002	55.35	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
2003	55.34	kd	CGS001-5573	PRKAR1A	Protein kinase A			
2004	55.33	kd	CGS001-6944	VPS72	-			
2005	55.32	cc		Cyclooxygenase inhibitor	-			
2006	55.14	kd	CGS001-2937	GSS	-			
2007	55.04	oe	ccsbBroad304_08878	METTL4	-			
2008	54.99	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
2009	54.98	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
2010	54.9	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
2011	54.89	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
2012	54.88	kd	CGS001-873	CBR1	Prostaglandin synthases			
2013	54.86	oe	ccsbBroad304_01019	MLH1	-			
2014	54.86	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
2015	54.72	oe	ccsbBroad304_04170	PANK2	-			
2016	54.72	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
2017	54.71	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
2018	54.61	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
2019	54.61	kd	CGS001-9788	MTSS1	-			
2020	54.55	kd	CGS001-8743	TNFSF10	CD molecules			
2021	54.55	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
2022	54.46	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
2023	54.34	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
2024	54.33	kd	CGS001-5588	PRKCQ	Delta subfamily			
2025	54.3	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
2026	54.26	oe	ccsbBroad304_07101	TSC2	-			
2027	54.26	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
2028	54.25	kd	CGS001-55143	CDCA8	-			
2029	54.23	kd	CGS001-501	ALDH7A1	Aldehyde dehydrogenases			
2030	54.23	kd	CGS001-220	ALDH1A3	Aldehyde dehydrogenases			
2031	54.11	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
2032	54.05	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
2033	54.04	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
2034	54	kd	CGS001-9500	MAGED1	-			
2035	53.98	kd	CGS001-9925	ZBTB5	BTB/POZ domain containing			
2036	53.96	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
2037	53.96	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
2038	53.95	kd	CGS001-9200	PTPLA	-			
2039	53.94	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
2040	53.86	kd	CGS001-1642	DDB1	-			
2041	53.83	kd	CGS001-22832	KIAA1009	-			
2042	53.76	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
2043	53.76	kd	CGS001-405	ARNT	Basic helix-loop-helix proteins			
2044	53.63	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
2045	53.62	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
2046	53.61	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
2047	53.57	kd	CGS001-1875	E2F5	-			
2048	53.54	cc		EGFR inhibitor	-			
2049	53.54	oe	ccsbBroad304_03264	UBAP1	-			
2050	53.53	kd	CGS001-6895	TARBP2	-			
2051	53.48	oe	ccsbBroad304_06525	LIPA	-			
2052	53.46	kd	CGS001-624	BDKRB2	Bradykinin receptors			
2053	53.42	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
2054	53.34	cp	BRD-K09471561	levofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
2055	53.34	kd	CGS001-10873	ME3	-			
2056	53.31	kd	CGS001-7295	TXN	-			
2057	53.3	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
2058	53.27	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
2059	53.26	kd	CGS001-64167	ERAP2	Aminopeptidase N			
2060	53.24	kd	CGS001-51182	HSPA14	Heat shock proteins / HSP70			
2061	53.23	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
2062	53.17	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
2063	53.13	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2064	53.13	kd	CGS001-23512	SUZ12	Zinc fingers, C2H2-type			
2065	53.05	oe	ccsbBroad304_01084	NEU1	-			
2066	53.05	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2067	52.98	oe	ccsbBroad304_01748	UFD1L	-			
2068	52.97	oe	ccsbBroad304_00469	DUT	-			
2069	52.95	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
2070	52.95	kd	CGS001-10673	TNFSF13B	CD molecules			
2071	52.92	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
2072	52.87	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
2073	52.84	kd	CGS001-28511	NKIRAS2	-			
2074	52.82	oe	ccsbBroad304_00239	CCNG1	-			
2075	52.82	kd	CGS001-10397	NDRG1	-			
2076	52.81	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
2077	52.69	kd	CGS001-159	ADSS	-			
2078	52.62	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2079	52.62	kd	CGS001-6197	RPS6KA3	RSK subfamily			
2080	52.61	kd	CGS001-7750	ZMYM2	Zinc fingers, MYM type			
2081	52.58	cc		IMPDH inhibitor	-			
2082	52.58	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
2083	52.42	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
2084	52.41	kd	CGS001-9459	ARHGEF6	Rho guanine nucleotide exchange factors			
2085	52.36	oe	ccsbBroad304_01485	SC5DL	-			
2086	52.35	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
2087	52.34	oe	ccsbBroad304_00099	ARG2	Arginase			
2088	52.28	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
2089	52.28	kd	CGS001-125965	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
2090	52.24	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2091	52.19	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
2092	52.17	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2093	52.14	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
2094	52.11	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2095	52.09	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
2096	52.09	kd	CGS001-31	ACACA	Carboxylases			
2097	52.01	kd	CGS001-23081	KDM4C	Histone demethylases			
2098	51.99	cc		Zinc fingers RanBP2 type LOF	-			
2099	51.99	kd	CGS001-2690	GHR	Prolactin receptor family			
2100	51.98	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
2101	51.88	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
2102	51.84	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
2103	51.79	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
2104	51.79	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
2105	51.77	oe	ccsbBroad304_00370	CS	-			
2106	51.76	kd	CGS001-51741	WWOX	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2107	51.75	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
2108	51.7	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
2109	51.69	kd	CGS001-3845	KRAS	RAS subfamily			
2110	51.62	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
2111	51.59	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
2112	51.55	kd	CGS001-11014	KDELR2	-			
2113	51.54	oe	ccsbBroad304_04788	OVCA2	-			
2114	51.54	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
2115	51.53	oe	ccsbBroad304_09284	UBE3B	-			
2116	51.49	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
2117	51.46	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
2118	51.45	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
2119	51.44	kd	CGS001-6257	RXRB	Retinoid X receptors			
2120	51.42	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
2121	51.37	kd	CGS001-6185	RPN2	-			
2122	51.31	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
2123	51.21	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
2124	51.2	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
2125	51.1	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
2126	51.08	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
2127	51.04	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
2128	51.04	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
2129	51.04	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2130	51.03	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
2131	51.02	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
2132	50.99	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
2133	50.98	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
2134	50.97	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
2135	50.94	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
2136	50.93	kd	CGS001-23658	LSM5	-			
2137	50.91	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2138	50.88	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
2139	50.88	oe	ccsbBroad304_09225	BUD13	-			
2140	50.85	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
2141	50.84	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
2142	50.77	kd	CGS001-3856	KRT8	Intermediate filaments type II, keratins (basic)			
2143	50.75	kd	CGS001-975	CD81	CD molecules			
2144	50.73	kd	CGS001-29880	ALG5	Glycosyltransferase family 2 domain containing			
2145	50.66	kd	CGS001-9928	KIF14	Kinesins			
2146	50.61	kd	CGS001-7276	TTR	-			
2147	50.47	kd	CGS001-199704	ZNF585A	Zinc fingers, C2H2-type			
2148	50.41	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
2149	50.3	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
2150	50.28	kd	CGS001-114112	TXNRD3	-			
2151	50.27	kd	CGS001-3775	KCNK1	Two-P potassium channels			
2152	50.25	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
2153	50.25	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
2154	50.24	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
2155	50.17	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
2156	50.17	kd	CGS001-8548	BLZF1	-			
2157	50.15	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2158	50.15	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
2159	50.14	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
2160	50.1	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
2161	50.06	kd	CGS001-23192	ATG4B	Aut2 peptidase			
2162	50	kd	CGS001-391013	PLA2G2C	-			
2163	49.97	kd	CGS001-23369	PUM2	-			
2164	49.95	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
2165	49.92	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
2166	49.92	kd	CGS001-58508	MLL3	-			
2167	49.91	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
2168	49.88	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
2169	49.85	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
2170	49.84	kd	CGS001-11315	PARK7	Parkinson disease			
2171	49.83	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
2172	49.81	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
2173	49.73	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
2174	49.7	kd	CGS001-50865	HEBP1	Endogenous ligands			
2175	49.68	kd	CGS001-58477	SRPRB	-			
2176	49.64	kd	CGS001-4779	NFE2L1	basic leucine zipper proteins			
2177	49.61	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
2178	49.57	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
2179	49.52	kd	CGS001-4170	MCL1	-			
2180	49.49	kd	CGS001-51380	CSAD	-			
2181	49.47	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
2182	49.45	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
2183	49.45	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
2184	49.44	kd	CGS001-2674	GFRA1	GDNF receptor family			
2185	49.34	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
2186	49.31	kd	CGS001-218	ALDH3A1	Aldehyde dehydrogenases			
2187	49.19	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2188	49.19	kd	CGS001-929	CD14	CD molecules			
2189	49.14	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
2190	49.14	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
2191	49.09	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
2192	49.06	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
2193	49.04	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
2194	49	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
2195	48.97	kd	CGS001-5335	PLCG1	Phosphoinositide-specific phospholipase C			
2196	48.95	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
2197	48.91	kd	CGS001-79170	PRR15L	-			
2198	48.84	kd	CGS001-3485	IGFBP2	insulin-like growth factor (IGF) binding proteins			
2199	48.82	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
2200	48.76	oe	ccsbBroad304_02058	PLOD3	-			
2201	48.76	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
2202	48.76	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
2203	48.7	kd	CGS001-51053	GMNN	-			
2204	48.66	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
2205	48.65	kd	CGS001-23636	NUP62	-			
2206	48.62	cp	BRD-K47780086	penciclovir	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor
2207	48.62	kd	CGS001-91392	ZNF502	Zinc fingers, C2H2-type			
2208	48.59	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
2209	48.59	kd	CGS001-9212	AURKB	Aurora kinase			
2210	48.53	kd	CGS001-112858	TP53RK	Bud32 family			
2211	48.49	oe	ccsbBroad304_07267	PDLIM4	-			
2212	48.49	oe	ccsbBroad304_06435	RBPJ	-			
2213	48.41	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
2214	48.41	kd	CGS001-1955	MEGF9	-			
2215	48.39	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
2216	48.38	kd	CGS001-5860	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
2217	48.34	kd	CGS001-79145	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
2218	48.34	kd	CGS001-54555	DDX49	DEAD-boxes			
2219	48.32	oe	ccsbBroad304_00397	CTSK	Cathepsins			
2220	48.32	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
2221	48.29	kd	CGS001-9146	HGS	Zinc fingers, FYVE domain containing			
2222	48.29	kd	CGS001-6286	S100P	EF-hand domain containing			
2223	48.13	kd	CGS001-3725	JUN	basic leucine zipper proteins			
2224	48.11	kd	CGS001-5564	PRKAB1	AMPK subfamily			
2225	48.03	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
2226	47.94	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
2227	47.94	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
2228	47.94	kd	CGS001-4067	LYN	Src family			
2229	47.93	kd	CGS001-7263	TST	-			
2230	47.9	kd	CGS001-116443	GRIN3A	Glutamate receptors			
2231	47.88	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
2232	47.87	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
2233	47.85	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
2234	47.85	kd	CGS001-10613	ERLIN1	-			
2235	47.78	kd	CGS001-4712	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
2236	47.77	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
2237	47.74	cc		Bacterial 30S ribosomal subunit inhibitor	-			
2238	47.73	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
2239	47.65	kd	CGS001-5387	PMS2P3	-			
2240	47.62	kd	CGS001-90655	TGIF2LY	Homeoboxes / TALE class			
2241	47.54	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
2242	47.53	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
2243	47.46	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
2244	47.45	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
2245	47.39	kd	CGS001-29982	NRBF2	-			
2246	47.34	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
2247	47.3	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
2248	47.25	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
2249	47.23	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
2250	47.2	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
2251	47.19	kd	CGS001-8522	GAS7	-			
2252	47.18	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
2253	47.16	kd	CGS001-7100	TLR5	Toll-like receptor family			
2254	47.08	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
2255	47.08	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
2256	47.01	kd	CGS001-253430	IPMK	-			
2257	47	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
2258	46.99	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
2259	46.94	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
2260	46.93	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
2261	46.9	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
2262	46.87	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
2263	46.85	oe	ccsbBroad304_06004	CKB	-			
2264	46.76	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
2265	46.74	kd	CGS001-2224	FDPS	Lanosterol biosynthesis pathway			
2266	46.72	kd	CGS001-8553	BHLHE40	Basic helix-loop-helix proteins			
2267	46.69	kd	CGS001-1468	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
2268	46.62	kd	CGS001-55229	PANK4	-			
2269	46.58	oe	ccsbBroad304_07363	AIFM1	-			
2270	46.54	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
2271	46.5	kd	CGS001-255877	BCL6B	BTB/POZ domain containing			
2272	46.45	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
2273	46.41	oe	ccsbBroad304_00036	AFP	-			
2274	46.36	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
2275	46.35	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
2276	46.34	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
2277	46.33	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
2278	46.33	kd	CGS001-5538	PPT1	-			
2279	46.31	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
2280	46.25	cc		RNA Polymerase Enzymes LOF	-			
2281	46.25	kd	CGS001-5981	RFC1	ATPases / AAA-type			
2282	46.24	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
2283	46.23	kd	CGS001-8738	CRADD	-			
2284	46.19	kd	CGS001-890	CCNA2	-			
2285	46.14	kd	CGS001-2523	FUT1	Fucosyltransferases			
2286	46.13	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
2287	46.12	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
2288	46.08	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
2289	46.08	kd	CGS001-10153	CEBPZ	-			
2290	46.07	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
2291	46.05	kd	CGS001-54386	TERF2IP	-			
2292	46.03	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
2293	46.02	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
2294	46	cc		CCK receptor antagonist	-			
2295	46	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
2296	45.98	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
2297	45.95	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
2298	45.86	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
2299	45.82	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2300	45.81	oe	ccsbBroad304_07506	UBAP2L	-			
2301	45.79	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
2302	45.79	oe	ccsbBroad304_02370	HRSP12	-			
2303	45.79	kd	CGS001-5447	POR	-			
2304	45.74	cp	BRD-A16444946	acarbose	Glucosidase inhibitor		GAA, MGAM, AMY2A, SI	Glucosidase inhibitor
2305	45.72	kd	CGS001-25949	SYF2	-			
2306	45.71	oe	ccsbBroad304_03173	TMED7	-			
2307	45.71	kd	CGS001-7025	NR2F1	COUP-TF-like receptors			
2308	45.67	kd	CGS001-665	BNIP3L	-			
2309	45.65	kd	CGS001-2731	GLDC	-			
2310	45.63	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
2311	45.62	oe	ccsbBroad304_02674	STK38	NDR family			
2312	45.55	cp	BRD-A39390670	rabeprazole	ATPase inhibitor		ATP4A, CYP2C19	ATPase inhibitor, Gastrin inhibitor
2313	45.54	kd	CGS001-8797	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
2314	45.5	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
2315	45.49	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
2316	45.49	kd	CGS001-11116	FGFR1OP	-			
2317	45.46	oe	ccsbBroad304_00962	SMAD4	SMADs			
2318	45.42	cp	BRD-K70883034	nimetazepam	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA receptor agonist
2319	45.38	oe	ccsbBroad304_02367	CALCOCO2	-			
2320	45.37	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
2321	45.35	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
2322	45.3	oe	ccsbBroad304_04404	TUBB6	Tubulins			
2323	45.23	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
2324	45.12	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
2325	45.11	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
2326	45.07	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
2327	45.01	oe	ccsbBroad304_00147	BAG1	-			
2328	45.01	kd	CGS001-8660	IRS2	Pleckstrin homology (PH) domain containing			
2329	44.97	oe	ccsbBroad304_05936	CASP2	Caspases			
2330	44.89	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
2331	44.88	kd	CGS001-54805	CNNM2	-			
2332	44.87	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
2333	44.87	kd	CGS001-1719	DHFR	Oxidoreductases			
2334	44.84	oe	ccsbBroad304_00329	CLTA	-			
2335	44.76	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
2336	44.74	kd	CGS001-9061	PAPSS1	-			
2337	44.72	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
2338	44.7	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
2339	44.67	kd	CGS001-5641	LGMN	Legumain			
2340	44.66	kd	CGS001-1050	CEBPA	basic leucine zipper proteins			
2341	44.65	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
2342	44.63	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2343	44.62	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
2344	44.61	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
2345	44.53	oe	ccsbBroad304_07920	NUP62	-			
2346	44.5	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
2347	44.5	oe	ccsbBroad304_01880	LAGE3	-			
2348	44.49	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2349	44.44	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
2350	44.35	kd	CGS001-1906	EDN1	Endogenous ligands			
2351	44.32	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
2352	44.3	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
2353	44.3	kd	CGS001-64080	RBKS	-			
2354	44.26	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
2355	44.23	kd	CGS001-345611	IRGM	-			
2356	44.21	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
2357	44.21	kd	CGS001-26959	HBP1	-			
2358	44.21	oe	ccsbBroad304_02554	TRAFD1	-			
2359	44.08	kd	CGS001-4610	MYCL1	-			
2360	44.03	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
2361	43.99	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
2362	43.88	kd	CGS001-64223	MLST8	WD repeat domain containing			
2363	43.84	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
2364	43.84	kd	CGS001-8566	PDXK	-			
2365	43.84	kd	CGS001-10797	MTHFD2	-			
2366	43.8	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
2367	43.79	kd	CGS001-403	ARL3	ADP-ribosylation factors			
2368	43.78	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
2369	43.77	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2370	43.77	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
2371	43.69	oe	ccsbBroad304_01035	MSH5	-			
2372	43.58	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
2373	43.55	kd	CGS001-85480	TSLP	-			
2374	43.52	kd	CGS001-10165	SLC25A13	Mitochondrial amino acid transporter subfamily			
2375	43.51	kd	CGS001-55632	G2E3	Zinc fingers, PHD-type			
2376	43.49	oe	ccsbBroad304_06535	LPL	-			
2377	43.49	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
2378	43.45	oe	ccsbBroad304_00155	CCND1	-			
2379	43.43	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
2380	43.37	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
2381	43.32	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
2382	43.22	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
2383	43.22	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2384	43.12	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
2385	43.11	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
2386	43.1	kd	CGS001-79733	E2F8	-			
2387	43.09	oe	ccsbBroad304_07128	VHL	-			
2388	43.04	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
2389	42.97	oe	ccsbBroad304_05890	BHMT	-			
2390	42.95	oe	ccsbBroad304_00446	DKC1	-			
2391	42.93	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2392	42.9	kd	CGS001-7090	TLE3	WD repeat domain containing			
2393	42.84	kd	CGS001-1457	CSNK2A1	Casein kinase 2 (CK2) family			
2394	42.83	kd	CGS001-84669	USP32	EF-hand domain containing			
2395	42.81	kd	CGS001-5062	PAK2	PAKA subfamily			
2396	42.78	kd	CGS001-337867	UBAC2	-			
2397	42.76	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
2398	42.73	oe	ccsbBroad304_02231	USP6NL	-			
2399	42.73	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
2400	42.71	kd	CGS001-472	ATM	Other PIKK family kinases			
2401	42.69	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
2402	42.68	kd	CGS001-4179	CD46	CD molecules			
2403	42.66	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
2404	42.65	oe	ccsbBroad304_03739	NRIP3	-			
2405	42.61	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2406	42.61	kd	CGS001-2936	GSR	Oxidoreductases			
2407	42.53	oe	ccsbBroad304_02741	PDS5A	-			
2408	42.46	kd	CGS001-51128	SAR1B	-			
2409	42.43	kd	CGS001-1201	CLN3	-			
2410	42.42	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
2411	42.42	oe	ccsbBroad304_02298	DNM1L	-			
2412	42.4	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
2413	42.34	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
2414	42.29	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
2415	42.29	oe	ccsbBroad304_10487	BPHL	-			
2416	42.28	kd	CGS001-7353	UFD1L	-			
2417	42.26	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2418	42.25	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
2419	42.25	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
2420	42.18	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2421	42.16	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
2422	42.14	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
2423	42.11	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
2424	42.11	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
2425	42.07	kd	CGS001-2254	FGF9	Endogenous ligands			
2426	41.96	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
2427	41.95	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2428	41.89	oe	ccsbBroad304_05985	CFL1	-			
2429	41.89	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
2430	41.88	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
2431	41.88	kd	CGS001-7314	UBB	-			
2432	41.88	kd	CGS001-115201	ATG4A	-			
2433	41.85	kd	CGS001-23013	SPEN	RNA binding motif (RRM) containing			
2434	41.84	kd	CGS001-1635	DCTD	-			
2435	41.82	oe	ccsbBroad304_12008	NLK	nmo subfamily			
2436	41.81	oe	ccsbBroad304_01960	CASK	CASK family			
2437	41.76	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
2438	41.65	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
2439	41.63	oe	ccsbBroad304_03951	NARFL	-			
2440	41.62	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
2441	41.62	oe	ccsbBroad304_08292	IP6K2	-			
2442	41.61	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
2443	41.59	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
2444	41.58	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
2445	41.51	kd	CGS001-2588	GALNS	Arylsulfatase family			
2446	41.45	kd	CGS001-8780	RIOK3	RIO3 subfamily			
2447	41.41	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
2448	41.4	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
2449	41.36	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
2450	41.3	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
2451	41.27	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
2452	41.21	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
2453	41.18	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
2454	41.16	oe	ccsbBroad304_00152	BCAT2	-			
2455	41.15	oe	ccsbBroad304_05183	TXLNA	-			
2456	41.13	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
2457	41.13	kd	CGS001-9488	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
2458	41.06	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
2459	41.04	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
2460	40.99	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2461	40.99	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
2462	40.94	kd	CGS001-7480	WNT10B	Wingless-type MMTV integration sites			
2463	40.93	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2464	40.9	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
2465	40.89	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
2466	40.82	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
2467	40.8	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
2468	40.8	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
2469	40.79	oe	ccsbBroad304_00221	CASP3	Caspases			
2470	40.77	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
2471	40.76	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
2472	40.72	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
2473	40.67	oe	ccsbBroad304_12106	PXK	Slob family			
2474	40.67	oe	ccsbBroad304_02569	BTG3	-			
2475	40.67	kd	CGS001-55176	SEC61A2	-			
2476	40.66	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2477	40.64	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
2478	40.63	kd	CGS001-2138	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2479	40.61	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
2480	40.6	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
2481	40.58	cc		Sirtuins GOF	-			
2482	40.57	oe	ccsbBroad304_07491	IP6K1	-			
2483	40.51	kd	CGS001-162	AP1B1	-			
2484	40.49	kd	CGS001-163688	CALML6	EF-hand domain containing			
2485	40.47	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
2486	40.45	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
2487	40.44	oe	ccsbBroad304_07053	TFPI	-			
2488	40.44	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
2489	40.42	kd	CGS001-23012	STK38L	NDR family			
2490	40.42	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
2491	40.4	kd	CGS001-11113	CIT	Other DMPK family kinases			
2492	40.39	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
2493	40.36	oe	ccsbBroad304_07605	LYPLA1	-			
2494	40.36	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
2495	40.34	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
2496	40.33	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
2497	40.31	kd	CGS001-8543	LMO4	-			
2498	40.31	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
2499	40.29	kd	CGS001-9868	TOMM70A	Tetratricopeptide (TTC) repeat domain containing			
2500	40.28	kd	CGS001-5058	PAK1	PAKA subfamily			
2501	40.26	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
2502	40.26	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
2503	40.26	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2504	40.24	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
2505	40.2	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
2506	40.17	kd	CGS001-53347	UBASH3A	-			
2507	40.15	kd	CGS001-5727	PTCH1	-			
2508	40.12	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2509	40.1	kd	CGS001-55556	ENOSF1	-			
2510	40.05	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
2511	40.04	kd	CGS001-55311	ZNF444	Zinc fingers, C2H2-type			
2512	39.99	kd	CGS001-5450	POU2AF1	-			
2513	39.98	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
2514	39.97	kd	CGS001-5899	RALB	-			
2515	39.95	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
2516	39.92	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
2517	39.91	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
2518	39.88	oe	ccsbBroad304_08461	CDCA4	-			
2519	39.88	kd	CGS001-1345	COX6C	Mitochondrial respiratory chain complex			
2520	39.87	kd	CGS001-1195	CLK1	CDC-like kinases			
2521	39.81	oe	ccsbBroad304_07411	LPXN	-			
2522	39.78	oe	ccsbBroad304_01576	SOAT1	-			
2523	39.72	oe	ccsbBroad304_07808	RAB11FIP2	-			
2524	39.69	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
2525	39.66	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
2526	39.64	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
2527	39.61	kd	CGS001-5621	PRNP	CD molecules			
2528	39.54	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
2529	39.54	kd	CGS001-4191	MDH2	-			
2530	39.54	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
2531	39.52	kd	CGS001-9352	TXNL1	-			
2532	39.5	oe	ccsbBroad304_01787	YES1	Src family			
2533	39.5	oe	ccsbBroad304_01724	TTR	-			
2534	39.49	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
2535	39.46	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2536	39.43	kd	CGS001-9903	KLHL21	BTB/POZ domain containing			
2537	39.36	kd	CGS001-1399	CRKL	SH2 domain containing			
2538	39.33	kd	CGS001-10554	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
2539	39.32	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
2540	39.32	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
2541	39.28	oe	ccsbBroad304_02676	PHB2	-			
2542	39.25	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
2543	39.25	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
2544	39.24	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
2545	39.23	cc		Bacterial cell wall synthesis inhibitor	-			
2546	39.21	oe	ccsbBroad304_03310	LCMT1	-			
2547	39.2	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
2548	39.18	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
2549	39.18	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
2550	39.18	kd	CGS001-158	ADSL	-			
2551	39.14	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
2552	39.1	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
2553	39.02	kd	CGS001-116931	MED12L	-			
2554	38.98	cc		Topoisomerase inhibitor	-			
2555	38.98	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
2556	38.97	oe	ccsbBroad304_08952	E2F8	-			
2557	38.94	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
2558	38.89	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
2559	38.75	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
2560	38.75	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
2561	38.73	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
2562	38.72	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
2563	38.67	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
2564	38.66	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
2565	38.6	kd	CGS001-7029	TFDP2	-			
2566	38.59	oe	ccsbBroad304_06574	MDH2	-			
2567	38.59	kd	CGS001-10456	HAX1	-			
2568	38.5	kd	CGS001-10362	HMG20B	High mobility group / Non-canonical			
2569	38.47	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
2570	38.46	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
2571	38.4	kd	CGS001-7316	UBC	-			
2572	38.34	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
2573	38.29	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2574	38.29	kd	CGS001-10914	PAPOLA	-			
2575	38.22	oe	ccsbBroad304_00966	MAFG	-			
2576	38.2	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
2577	38.2	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
2578	38.19	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
2579	38.17	cc		Dopamine receptor antagonist	-			
2580	38.17	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
2581	38.17	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
2582	38.14	cp	BRD-K10670311	sulfasalazine	Antirheumatic		PTGS1, PTGS2, ACAT1, ALOX5, CHUK, IKBKB, PLA2G1B, PPARG, SLC46A1, SLC7A11, TBXAS1	Antirheumatic, NFkB pathway inhibitor
2583	38.1	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
2584	38.08	oe	ccsbBroad304_00183	C1S	Complement system			
2585	38.06	oe	ccsbBroad304_05547	TMEM110	-			
2586	38.05	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
2587	38.02	kd	CGS001-29110	TBK1	IKK family			
2588	37.97	cc		Serotonin receptor antagonist	-			
2589	37.95	cp	BRD-K39983086	loteprednol	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Phospholipase inhibitor
2590	37.94	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
2591	37.89	kd	CGS001-7159	TP53BP2	Ankyrin repeat domain containing			
2592	37.88	kd	CGS001-50846	DHH	-			
2593	37.83	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
2594	37.83	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
2595	37.82	oe	ccsbBroad304_05135	PARP15	-			
2596	37.81	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
2597	37.8	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
2598	37.79	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
2599	37.77	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
2600	37.76	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
2601	37.74	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
2602	37.73	kd	CGS001-55722	CEP72	-			
2603	37.7	kd	CGS001-30001	ERO1L	-			
2604	37.68	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
2605	37.67	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
2606	37.67	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
2607	37.66	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
2608	37.6	kd	CGS001-5707	PSMD1	Proteasome subunits			
2609	37.56	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
2610	37.56	kd	CGS001-54815	GATAD2A	GATA zinc finger domain containing			
2611	37.55	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
2612	37.52	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
2613	37.49	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
2614	37.48	kd	CGS001-10776	ARPP19	-			
2615	37.35	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
2616	37.34	oe	ccsbBroad304_07071	TKT	-			
2617	37.16	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
2618	37.15	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
2619	37.07	kd	CGS001-2115	ETV1	ETS Transcription Factors			
2620	37.05	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
2621	36.98	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
2622	36.95	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
2623	36.92	kd	CGS001-9958	USP15	Ubiquitin-specific peptidases			
2624	36.92	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
2625	36.91	cp	BRD-K41051431	mecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2626	36.86	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
2627	36.84	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
2628	36.82	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
2629	36.82	kd	CGS001-2266	FGG	Endogenous ligands			
2630	36.81	kd	CGS001-2821	GPI	-			
2631	36.8	kd	CGS001-2119	ETV5	ETS Transcription Factors			
2632	36.73	oe	ccsbBroad304_07922	TRIM29	-			
2633	36.72	oe	ccsbBroad304_00964	SMAD7	SMADs			
2634	36.65	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
2635	36.64	kd	CGS001-7321	UBE2D1	Ubiquitin-conjugating enzymes E2			
2636	36.62	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
2637	36.61	kd	CGS001-10131	TRAP1	Heat shock proteins / HSPC			
2638	36.58	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
2639	36.56	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
2640	36.52	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
2641	36.5	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
2642	36.46	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
2643	36.45	kd	CGS001-9842	PLEKHM1	Pleckstrin homology (PH) domain containing			
2644	36.41	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
2645	36.37	kd	CGS001-51002	TPRKB	-			
2646	36.35	kd	CGS001-6434	TRA2B	RNA binding motif (RRM) containing			
2647	36.29	kd	CGS001-6773	STAT2	SH2 domain containing			
2648	36.28	kd	CGS001-27113	BBC3	-			
2649	36.2	oe	ccsbBroad304_01662	TFDP2	-			
2650	36.2	oe	ccsbBroad304_00570	FIGF	-			
2651	36.18	kd	CGS001-4905	NSF	ATPases / AAA-type			
2652	36.17	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
2653	36.11	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
2654	36.1	oe	ccsbBroad304_02115	PTTG1	-			
2655	36.1	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
2656	36.09	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
2657	36.09	oe	ccsbBroad304_00313	TBCB	-			
2658	36.08	kd	CGS001-2161	F12	Chymotrypsin			
2659	36.06	oe	ccsbBroad304_07374	PTPLA	-			
2660	36.01	kd	CGS001-1356	CP	-			
2661	36.01	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
2662	36	kd	CGS001-6787	NEK4	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2663	35.99	oe	ccsbBroad304_06178	ERCC5	-			
2664	35.98	kd	CGS001-7423	VEGFB	-			
2665	35.95	cc		Homeobox Gene GOF	-			
2666	35.91	oe	ccsbBroad304_07592	CEPT1	-			
2667	35.9	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
2668	35.87	oe	ccsbBroad304_10437	STMN1	-			
2669	35.85	kd	CGS001-3614	IMPDH1	Oxidoreductases			
2670	35.83	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2671	35.76	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
2672	35.75	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
2673	35.75	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
2674	35.74	kd	CGS001-7030	TFE3	Basic helix-loop-helix proteins			
2675	35.73	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
2676	35.73	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
2677	35.66	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
2678	35.65	kd	CGS001-5825	ABCD3	ATP binding cassette transporters / subfamily D			
2679	35.64	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
2680	35.58	kd	CGS001-2159	F10	Chymotrypsin			
2681	35.54	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
2682	35.52	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
2683	35.45	kd	CGS001-1650	DDOST	-			
2684	35.45	kd	CGS001-286075	ZNF707	Zinc fingers, C2H2-type			
2685	35.43	kd	CGS001-126823	KLHDC9	-			
2686	35.4	oe	ccsbBroad304_02018	SUCLA2	-			
2687	35.38	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
2688	35.38	kd	CGS001-345	APOC3	Apolipoproteins			
2689	35.33	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
2690	35.32	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
2691	35.31	kd	CGS001-6277	S100A6	EF-hand domain containing			
2692	35.31	kd	CGS001-5992	RFX4	-			
2693	35.27	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
2694	35.26	kd	CGS001-6827	SUPT4H1	-			
2695	35.25	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
2696	35.25	kd	CGS001-6722	SRF	-			
2697	35.24	kd	CGS001-57819	LSM2	-			
2698	35.18	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
2699	35.17	kd	CGS001-64121	RRAGC	-			
2700	35.16	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
2701	35.14	oe	ccsbBroad304_04064	PRR15L	-			
2702	35.14	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
2703	35.08	kd	CGS001-11186	RASSF1	-			
2704	35.06	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
2705	35.04	kd	CGS001-5366	PMAIP1	-			
2706	35.04	kd	CGS001-135	ADORA2A	GPCR / Class A : Adenosine receptors			
2707	34.99	kd	CGS001-3482	IGF2R	CD molecules			
2708	34.97	kd	CGS001-10614	HEXIM1	-			
2709	34.95	kd	CGS001-7474	WNT5A	Endogenous ligands			
2710	34.92	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
2711	34.91	oe	ccsbBroad304_00222	CASP6	Caspases			
2712	34.86	oe	ccsbBroad304_00626	GDI1	-			
2713	34.84	kd	CGS001-898	CCNE1	-			
2714	34.83	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
2715	34.72	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
2716	34.72	kd	CGS001-3476	IGBP1	-			
2717	34.71	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
2718	34.71	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
2719	34.7	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
2720	34.64	kd	CGS001-6804	STX1A	-			
2721	34.61	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
2722	34.61	kd	CGS001-1445	CSK	Csk family			
2723	34.59	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
2724	34.57	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
2725	34.55	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
2726	34.55	kd	CGS001-3479	IGF1	Endogenous ligands			
2727	34.53	kd	CGS001-10427	SEC24B	-			
2728	34.52	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
2729	34.48	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
2730	34.43	kd	CGS001-5894	RAF1	RAF family			
2731	34.42	kd	CGS001-161	AP2A2	-			
2732	34.36	kd	CGS001-1763	DNA2	-			
2733	34.26	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
2734	34.26	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
2735	34.22	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
2736	34.17	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
2737	34.11	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
2738	34.1	oe	ccsbBroad304_02415	TUBB3	Tubulins			
2739	34.09	oe	ccsbBroad304_08645	BCCIP	-			
2740	34.07	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
2741	34.07	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
2742	34.06	kd	CGS001-673	BRAF	RAF family			
2743	34.04	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
2744	34.04	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
2745	34.01	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
2746	34	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
2747	33.99	kd	CGS001-84811	BUD13	-			
2748	33.98	kd	CGS001-165082	GPR113	Adhesion Class GPCRs			
2749	33.97	kd	CGS001-22891	ZNF365	Zinc fingers, C2H2-type			
2750	33.92	kd	CGS001-4090	SMAD5	SMADs			
2751	33.91	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
2752	33.91	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2753	33.89	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
2754	33.89	kd	CGS001-55802	DCP1A	-			
2755	33.88	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
2756	33.88	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
2757	33.88	kd	CGS001-116535	MRGPRF	GPCR / Class A : Orphans			
2758	33.87	oe	ccsbBroad304_03961	SMURF2	-			
2759	33.8	kd	CGS001-51284	TLR7	Toll-like receptor family			
2760	33.79	oe	ccsbBroad304_00491	EIF4EBP2	-			
2761	33.77	oe	ccsbBroad304_03497	TXNL4B	-			
2762	33.76	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
2763	33.75	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
2764	33.73	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
2765	33.71	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
2766	33.66	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
2767	33.66	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
2768	33.65	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
2769	33.63	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
2770	33.63	kd	CGS001-55234	SMU1	WD repeat domain containing			
2771	33.62	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
2772	33.61	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
2773	33.6	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
2774	33.52	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
2775	33.5	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
2776	33.47	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
2777	33.44	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
2778	33.43	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2779	33.4	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
2780	33.38	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
2781	33.34	cp	BRD-K99447003	enalaprilat	ACE inhibitor		ACE	ACE inhibitor
2782	33.34	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
2783	33.24	oe	ccsbBroad304_00956	LYZ	-			
2784	33.23	kd	CGS001-5052	PRDX1	-			
2785	33.21	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
2786	33.2	kd	CGS001-5571	PRKAG1	AMPK subfamily			
2787	33.18	kd	CGS001-6303	SAT1	-			
2788	33.17	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
2789	33.16	kd	CGS001-114904	C1QTNF6	-			
2790	33.1	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
2791	33.1	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
2792	33.09	kd	CGS001-255738	PCSK9	Subtilisin			
2793	33.05	oe	ccsbBroad304_02534	UTP14A	-			
2794	32.98	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
2795	32.95	kd	CGS001-3608	ILF2	-			
2796	32.89	oe	ccsbBroad304_07178	ZFP112	-			
2797	32.89	oe	ccsbBroad304_02533	NOXA1	-			
2798	32.87	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
2799	32.85	kd	CGS001-3776	KCNK2	Two-P potassium channels			
2800	32.85	oe	ccsbBroad304_04194	ELL3	-			
2801	32.85	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
2802	32.77	kd	CGS001-23076	RRP1B	-			
2803	32.76	kd	CGS001-64219	PJA1	RING-type (C3HC4) zinc fingers			
2804	32.73	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2805	32.69	oe	ccsbBroad304_04544	RCCD1	-			
2806	32.69	kd	CGS001-4929	NR4A2	Nerve growth factor IB-like receptors			
2807	32.66	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
2808	32.66	oe	ccsbBroad304_00392	CTLA4	CD molecules			
2809	32.64	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
2810	32.63	kd	CGS001-11112	HIBADH	-			
2811	32.59	oe	ccsbBroad304_02219	MORF4L2	-			
2812	32.59	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
2813	32.56	oe	ccsbBroad304_07843	FCHO1	-			
2814	32.51	kd	CGS001-6621	SNAPC4	-			
2815	32.5	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2816	32.46	kd	CGS001-26271	FBXO5	F-boxes / other			
2817	32.42	kd	CGS001-2966	GTF2H2	General transcription factors			
2818	32.33	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
2819	32.33	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
2820	32.33	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2821	32.31	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
2822	32.3	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
2823	32.27	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
2824	32.19	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
2825	32.17	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
2826	32.16	kd	CGS001-6519	SLC3A1	SLC3 family			
2827	32.16	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
2828	32.12	kd	CGS001-9034	CCRL2	Chemokine receptors			
2829	32.05	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
2830	32.02	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
2831	31.98	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
2832	31.97	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
2833	31.97	kd	CGS001-3957	LGALS2	Lectins, galactoside-binding			
2834	31.93	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
2835	31.91	kd	CGS001-9851	KIAA0753	-			
2836	31.89	oe	ccsbBroad304_13903	MTAP	-			
2837	31.84	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
2838	31.81	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
2839	31.75	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
2840	31.72	oe	ccsbBroad304_07890	CBX7	-			
2841	31.69	kd	CGS001-4143	MAT1A	-			
2842	31.67	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
2843	31.67	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
2844	31.63	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
2845	31.57	oe	ccsbBroad304_02109	XPR1	-			
2846	31.56	oe	ccsbBroad304_09054	EGFL8	-			
2847	31.56	kd	CGS001-27076	LYPD3	-			
2848	31.48	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
2849	31.46	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2850	31.43	oe	ccsbBroad304_04257	SPRY4	-			
2851	31.4	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
2852	31.38	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
2853	31.37	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
2854	31.31	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
2855	31.28	kd	CGS001-6757	SSX2	-			
2856	31.24	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
2857	31.24	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
2858	31.2	kd	CGS001-2053	EPHX2	-			
2859	31.17	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
2860	31.15	kd	CGS001-8772	FADD	-			
2861	31.14	oe	ccsbBroad304_00865	ILF2	-			
2862	31.1	oe	ccsbBroad304_02285	MED6	-			
2863	31.07	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
2864	31.06	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
2865	31.05	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
2866	31.05	kd	CGS001-6885	MAP3K7	MAPKKK:TAK1 subfamily			
2867	31.04	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
2868	31.02	kd	CGS001-3109	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
2869	31.01	oe	ccsbBroad304_07024	SYK	Syk family			
2870	30.94	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
2871	30.93	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
2872	30.92	oe	ccsbBroad304_08553	STAP2	-			
2873	30.92	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
2874	30.92	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
2875	30.9	kd	CGS001-10887	PROKR1	GPCR / Class A : Prokineticin receptors			
2876	30.87	cc		Integrin subunits alpha LOF	-			
2877	30.84	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
2878	30.81	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
2879	30.79	kd	CGS001-2548	GAA	Glycosidases			
2880	30.63	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
2881	30.62	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
2882	30.49	kd	CGS001-9189	ZBED1	Pseudoautosomal regions / PAR1			
2883	30.44	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
2884	30.44	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
2885	30.36	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2886	30.36	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
2887	30.31	oe	ccsbBroad304_07662	NPRL2	-			
2888	30.3	kd	CGS001-2274	FHL2	-			
2889	30.29	kd	CGS001-6813	STXBP2	-			
2890	30.28	kd	CGS001-10616	RBCK1	RING-type (C3HC4) zinc fingers			
2891	30.27	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
2892	30.23	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
2893	30.23	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
2894	30.22	kd	CGS001-79581	GPR172A	-			
2895	30.22	kd	CGS001-9700	ESPL1	-			
2896	30.21	kd	CGS001-5618	PRLR	Prolactin receptor family			
2897	30.18	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
2898	30.17	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
2899	30.15	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
2900	30.15	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
2901	30.14	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
2902	30.13	kd	CGS001-26136	TES	-			
2903	30.13	kd	CGS001-2834	PRLHR	GPCR / Class A : RF amide peptide receptors			
2904	30.09	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
2905	30.07	oe	ccsbBroad304_02239	RASSF2	-			
2906	30.06	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
2907	30.05	cc		FLT3 inhibitor	-			
2908	30.05	kd	CGS001-118738	ZNF488	Zinc fingers, C2H2-type			
2909	30.03	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
2910	29.99	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
2911	29.96	kd	CGS001-9308	CD83	CD molecules			
2912	29.95	kd	CGS001-7862	BRPF1	Non-enzymatic BRD containing proteins			
2913	29.94	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
2914	29.93	kd	CGS001-2878	GPX3	-			
2915	29.92	kd	CGS001-8435	SOAT2	-			
2916	29.89	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
2917	29.89	kd	CGS001-1633	DCK	-			
2918	29.86	kd	CGS001-23463	ICMT	-			
2919	29.85	kd	CGS001-122809	SOCS4	SH2 domain containing			
2920	29.83	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
2921	29.82	kd	CGS001-10971	YWHAQ	-			
2922	29.82	kd	CGS001-2769	GNA15	-			
2923	29.79	kd	CGS001-124641	OVCA2	-			
2924	29.77	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
2925	29.76	cc		Glycogen synthase kinase inhibitor	-			
2926	29.76	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
2927	29.76	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
2928	29.74	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
2929	29.68	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
2930	29.66	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
2931	29.59	kd	CGS001-5217	PFN2	-			
2932	29.59	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
2933	29.57	oe	ccsbBroad304_08322	UFM1	-			
2934	29.57	oe	ccsbBroad304_00888	ITPK1	-			
2935	29.57	kd	CGS001-85315	PAQR8	-			
2936	29.56	kd	CGS001-2155	F7	Chymotrypsin			
2937	29.55	kd	CGS001-23401	FRAT2	-			
2938	29.52	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
2939	29.5	kd	CGS001-57720	GPR107	GPCR / Unclassified : 7TM orphan receptors			
2940	29.44	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2941	29.42	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
2942	29.39	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
2943	29.38	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
2944	29.38	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
2945	29.37	oe	ccsbBroad304_01061	NAB2	-			
2946	29.36	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
2947	29.27	kd	CGS001-901	CCNG2	-			
2948	29.26	kd	CGS001-2160	F11	Chymotrypsin			
2949	29.25	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
2950	29.22	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
2951	29.21	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
2952	29.19	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
2953	29.16	cc		X linked mental retardation group 2 LOF	-			
2954	29.16	kd	CGS001-55011	PIH1D1	-			
2955	29.15	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
2956	29.14	cp	BRD-K69650333	idarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
2957	29.13	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
2958	29.13	kd	CGS001-3958	LGALS3	Endogenous ligands			
2959	29.09	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
2960	29.09	kd	CGS001-80306	MED28	-			
2961	29.07	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
2962	29.07	kd	CGS001-23576	DDAH1	Dimethylarginine dimethylaminohydrolases			
2963	29.06	kd	CGS001-9014	TAF1B	-			
2964	29.05	oe	ccsbBroad304_02243	DLGAP5	-			
2965	29.03	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2966	29.01	oe	ccsbBroad304_05963	CD44	CD molecules			
2967	29	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
2968	28.99	kd	CGS001-55577	NAGK	-			
2969	28.97	kd	CGS001-2052	EPHX1	-			
2970	28.96	oe	ccsbBroad304_02653	PRAF2	-			
2971	28.95	kd	CGS001-966	CD59	CD molecules			
2972	28.93	kd	CGS001-9770	RASSF2	-			
2973	28.92	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
2974	28.92	kd	CGS001-9218	VAPA	-			
2975	28.92	kd	CGS001-221393	GPR115	Adhesion Class GPCRs			
2976	28.87	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
2977	28.87	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
2978	28.78	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
2979	28.77	kd	CGS001-8295	TRRAP	TRRAP subfamily			
2980	28.76	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
2981	28.75	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
2982	28.74	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
2983	28.65	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
2984	28.62	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
2985	28.55	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
2986	28.47	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
2987	28.47	kd	CGS001-10434	LYPLA1	-			
2988	28.46	kd	CGS001-22894	DIS3	-			
2989	28.45	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
2990	28.4	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
2991	28.39	cp	BRD-A84134924	pancuronium	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRNA1, CHRNA2	Acetylcholine receptor antagonist
2992	28.37	cc		Imidazoline ligand	-			
2993	28.34	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
2994	28.29	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
2995	28.25	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
2996	28.22	kd	CGS001-178	AGL	-			
2997	28.19	oe	ccsbBroad304_00489	EHHADH	-			
2998	28.19	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
2999	28.16	kd	CGS001-26039	SS18L1	-			
3000	28.14	kd	CGS001-55328	RNLS	-			
3001	28.1	kd	CGS001-4781	NFIB	-			
3002	28.09	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
3003	28.05	kd	CGS001-11162	NUDT6	Nudix motif containing			
3004	28.02	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
3005	28.01	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
3006	28.01	kd	CGS001-5445	PON2	Paraoxonases			
3007	27.99	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
3008	27.97	kd	CGS001-5723	PSPH	-			
3009	27.94	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
3010	27.87	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
3011	27.86	cc		LIM class homeoboxes GOF	-			
3012	27.84	oe	ccsbBroad304_06089	DDIT3	-			
3013	27.84	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
3014	27.84	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
3015	27.81	kd	CGS001-8576	STK16	NAK family			
3016	27.8	oe	ccsbBroad304_03980	DCLRE1B	-			
3017	27.79	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
3018	27.77	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
3019	27.77	kd	CGS001-221391	OPN5	GPCR / Class A : Opsin receptors			
3020	27.74	cc		VEGFR inhibitor	-			
3021	27.72	kd	CGS001-83999	KREMEN1	-			
3022	27.71	kd	CGS001-597	BCL2A1	-			
3023	27.67	kd	CGS001-5682	PSMA1	Proteasome subunits			
3024	27.66	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
3025	27.65	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
3026	27.62	kd	CGS001-3487	IGFBP4	insulin-like growth factor (IGF) binding proteins			
3027	27.61	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
3028	27.6	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
3029	27.56	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
3030	27.51	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
3031	27.49	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
3032	27.44	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
3033	27.42	kd	CGS001-125950	RAVER1	RNA binding motif (RRM) containing			
3034	27.4	kd	CGS001-114609	TIRAP	-			
3035	27.32	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
3036	27.28	oe	ccsbBroad304_00841	IKBKB	IKK family			
3037	27.25	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
3038	27.24	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
3039	27.23	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
3040	27.21	kd	CGS001-55033	FKBP14	EF-hand domain containing			
3041	27.2	kd	CGS001-3029	HAGH	-			
3042	27.15	kd	CGS001-11136	SLC7A9	SLC7 family			
3043	27.1	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
3044	27.05	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
3045	27.04	kd	CGS001-21	ABCA3	ATP binding cassette transporters / subfamily A			
3046	27.01	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
3047	27	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3048	27	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
3049	27	kd	CGS001-8836	GGH	Gamma-glutamyl hydrolase			
3050	26.99	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
3051	26.98	oe	ccsbBroad304_00020	ACY1	-			
3052	26.95	oe	ccsbBroad304_06562	MAT1A	-			
3053	26.92	kd	CGS001-10253	SPRY2	-			
3054	26.9	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
3055	26.83	oe	ccsbBroad304_07018	SUPT5H	-			
3056	26.82	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
3057	26.81	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
3058	26.81	kd	CGS001-433	ASGR2	C-type lectin domain containing			
3059	26.76	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
3060	26.75	kd	CGS001-10969	EBNA1BP2	-			
3061	26.73	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
3062	26.69	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
3063	26.67	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
3064	26.65	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
3065	26.62	kd	CGS001-22794	CASC3	-			
3066	26.56	oe	ccsbBroad304_02801	CASP14	Caspases			
3067	26.56	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
3068	26.5	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
3069	26.43	kd	CGS001-80351	TNKS2	Ankyrin repeat domain containing			
3070	26.43	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
3071	26.42	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
3072	26.42	kd	CGS001-23242	COBL	-			
3073	26.4	oe	ccsbBroad304_01623	SUPT4H1	-			
3074	26.36	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
3075	26.33	kd	CGS001-55718	POLR3E	RNA polymerase subunits			
3076	26.31	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
3077	26.29	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
3078	26.28	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
3079	26.25	kd	CGS001-2786	GNG4	-			
3080	26.24	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
3081	26.22	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
3082	26.2	kd	CGS001-79902	NUP85	-			
3083	26.15	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
3084	26.14	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3085	26.13	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
3086	26.12	kd	CGS001-51096	UTP18	WD repeat domain containing			
3087	26.11	oe	ccsbBroad304_02276	MVP	-			
3088	26.06	kd	CGS001-10468	FST	-			
3089	26.04	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
3090	25.92	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3091	25.89	kd	CGS001-22978	NT5C2	Adenosine turnover			
3092	25.86	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
3093	25.85	kd	CGS001-5230	PGK1	-			
3094	25.84	kd	CGS001-55765	C1ORF106	-			
3095	25.83	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
3096	25.83	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
3097	25.82	oe	ccsbBroad304_05758	ACADSB	-			
3098	25.82	kd	CGS001-54106	TLR9	Toll-like receptor family			
3099	25.74	cc		Supressors of cytokine signaling GOF	-			
3100	25.73	kd	CGS001-7037	TFRC	CD molecules			
3101	25.71	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
3102	25.68	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
3103	25.66	oe	ccsbBroad304_01038	MSRA	-			
3104	25.64	kd	CGS001-5653	KLK6	Chymotrypsin			
3105	25.62	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
3106	25.57	kd	CGS001-4671	NAIP	Inhibitors of apoptosis (IAP) protein family			
3107	25.54	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
3108	25.54	kd	CGS001-10198	MPHOSPH9	-			
3109	25.48	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
3110	25.47	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
3111	25.45	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
3112	25.45	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
3113	25.43	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
3114	25.39	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
3115	25.37	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
3116	25.36	kd	CGS001-1655	DDX5	DEAD-boxes			
3117	25.3	kd	CGS001-7155	TOP2B	DNA Topoisomerases			
3118	25.28	kd	CGS001-1376	CPT2	-			
3119	25.27	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
3120	25.26	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
3121	25.24	kd	CGS001-80237	ELL3	-			
3122	25.24	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
3123	25.22	oe	ccsbBroad304_00650	GNA11	-			
3124	25.21	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
3125	25.18	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
3126	25.17	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
3127	25.16	kd	CGS001-833	CARS	Aminoacyl tRNA synthetases / Class I			
3128	25.1	kd	CGS001-8431	NR0B2	DAX-like receptors			
3129	25.07	cc		Cyclin dependent kinases LOF	-			
3130	25.06	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
3131	25.05	kd	CGS001-4300	MLLT3	-			
3132	24.99	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
3133	24.99	kd	CGS001-2879	GPX4	-			
3134	24.96	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
3135	24.88	cc		Poly ADP ribose polymerases LOF	-			
3136	24.86	oe	ccsbBroad304_06745	PNN	-			
3137	24.81	kd	CGS001-3821	KLRC1	CD molecules			
3138	24.77	oe	ccsbBroad304_07851	FAM120A	-			
3139	24.75	kd	CGS001-3127	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
3140	24.74	kd	CGS001-55082	ARGLU1	-			
3141	24.73	kd	CGS001-10672	GNA13	-			
3142	24.66	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
3143	24.66	kd	CGS001-2931	GSK3A	GSK subfamily			
3144	24.65	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
3145	24.62	kd	CGS001-10452	TOMM40	-			
3146	24.52	kd	CGS001-8503	PIK3R3	Phosphatidylinositol kinases			
3147	24.52	oe	ccsbBroad304_02496	MTX2	-			
3148	24.47	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
3149	24.43	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
3150	24.43	kd	CGS001-54899	PXK	Slob family			
3151	24.41	kd	CGS001-5446	PON3	Paraoxonases			
3152	24.38	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
3153	24.38	kd	CGS001-4171	MCM2	-			
3154	24.36	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
3155	24.33	kd	CGS001-9213	XPR1	-			
3156	24.29	kd	CGS001-2538	G6PC	-			
3157	24.28	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
3158	24.23	kd	CGS001-5045	FURIN	Subtilisin			
3159	24.22	kd	CGS001-23451	SF3B1	-			
3160	24.17	oe	ccsbBroad304_00447	DLD	-			
3161	24.15	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
3162	24.12	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
3163	24.09	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
3164	24.04	kd	CGS001-2010	EMD	-			
3165	24.02	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
3166	23.98	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
3167	23.95	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
3168	23.95	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
3169	23.95	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
3170	23.95	kd	CGS001-4976	OPA1	-			
3171	23.87	kd	CGS001-26086	GPSM1	Tetratricopeptide (TTC) repeat domain containing			
3172	23.69	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
3173	23.67	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
3174	23.65	kd	CGS001-7079	TIMP4	-			
3175	23.64	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
3176	23.59	kd	CGS001-26292	MYCBP	-			
3177	23.58	oe	ccsbBroad304_03113	DSE	-			
3178	23.52	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3179	23.49	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
3180	23.49	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
3181	23.41	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
3182	23.37	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
3183	23.35	kd	CGS001-10001	MED6	-			
3184	23.33	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
3185	23.32	oe	ccsbBroad304_05757	ACADS	-			
3186	23.3	kd	CGS001-10725	NFAT5	Nuclear factor of activated T-cells			
3187	23.29	oe	ccsbBroad304_07017	SUOX	-			
3188	23.25	kd	CGS001-4129	MAOB	Catecholamine turnover			
3189	23.24	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
3190	23.18	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
3191	23.17	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
3192	23.16	kd	CGS001-9655	SOCS5	SH2 domain containing			
3193	23.11	kd	CGS001-6625	SNRNP70	RNA binding motif (RRM) containing			
3194	23.1	oe	ccsbBroad304_01672	TIMP2	-			
3195	23.08	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
3196	23.07	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
3197	22.98	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
3198	22.9	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
3199	22.86	cp	BRD-A49172652	lansoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4, CYP3A5	ATPase inhibitor
3200	22.86	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3201	22.84	oe	ccsbBroad304_03878	SENP2	-			
3202	22.84	kd	CGS001-23028	KDM1A	Histone demethylase			
3203	22.83	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
3204	22.81	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
3205	22.79	kd	CGS001-347736	NME9	-			
3206	22.79	oe	ccsbBroad304_08825	LHPP	-			
3207	22.76	kd	CGS001-83593	RASSF5	-			
3208	22.71	kd	CGS001-390	RND3	-			
3209	22.64	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
3210	22.61	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
3211	22.56	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
3212	22.47	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
3213	22.39	kd	CGS001-9871	SEC24D	-			
3214	22.32	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
3215	22.32	kd	CGS001-51750	RTEL1	-			
3216	22.28	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
3217	22.27	cp	BRD-K52020312	metronidazole	DNA inhibitor		CYP2C8, CYP2E1, CYP3A5, CYP3A7	DNA inhibitor, Antiprotozoal
3218	22.19	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
3219	22.18	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
3220	22.16	kd	CGS001-2581	GALC	-			
3221	22.15	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
3222	22.1	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3223	22.04	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
3224	22.02	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
3225	22.01	kd	CGS001-6491	STIL	-			
3226	21.99	kd	CGS001-210	ALAD	-			
3227	21.95	cp	BRD-K32311154	nifekalant	Potassium channel blocker			Potassium channel blocker
3228	21.94	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
3229	21.93	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
3230	21.9	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
3231	21.9	kd	CGS001-89882	TPD52L3	-			
3232	21.8	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
3233	21.77	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
3234	21.75	oe	ccsbBroad304_05821	ANXA1	Annexins			
3235	21.73	kd	CGS001-727	C5	Endogenous ligands			
3236	21.69	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
3237	21.67	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
3238	21.64	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
3239	21.63	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
3240	21.62	kd	CGS001-2747	GLUD2	-			
3241	21.61	kd	CGS001-10477	UBE2E3	Ubiquitin-conjugating enzymes E2			
3242	21.59	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
3243	21.59	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
3244	21.58	kd	CGS001-57822	GRHL3	-			
3245	21.46	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
3246	21.42	kd	CGS001-9900	SV2A	Major facilitator superfamily (MFS) of transporters			
3247	21.39	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
3248	21.33	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
3249	21.33	kd	CGS001-54442	KCTD5	-			
3250	21.31	cp	BRD-K02227374	milnacipran	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Serotonin reuptake inhibitor
3251	21.16	cc		PI3K inhibitor	-			
3252	21.09	kd	CGS001-51268	PIPOX	-			
3253	21.07	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
3254	21.01	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
3255	20.92	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
3256	20.91	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
3257	20.91	kd	CGS001-8717	TRADD	-			
3258	20.89	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
3259	20.86	kd	CGS001-91304	C19ORF6	-			
3260	20.77	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
3261	20.75	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
3262	20.74	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3263	20.71	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
3264	20.69	oe	ccsbBroad304_06739	PLOD1	-			
3265	20.68	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
3266	20.65	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
3267	20.65	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
3268	20.61	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3269	20.6	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
3270	20.6	kd	CGS001-10626	TRIM16	Tripartite motif containing			
3271	20.59	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
3272	20.53	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
3273	20.53	kd	CGS001-23509	POFUT1	Fucosyltransferases			
3274	20.42	kd	CGS001-3265	HRAS	RAS subfamily			
3275	20.39	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
3276	20.36	kd	CGS001-9412	MED21	-			
3277	20.34	kd	CGS001-54556	ING3	Zinc fingers, PHD-type			
3278	20.28	kd	CGS001-7182	NR2C2	Testicular receptors			
3279	20.17	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3280	20.16	kd	CGS001-7086	TKT	-			
3281	20.15	kd	CGS001-8850	KAT2B	Histone acetyltransferases (HATs)			
3282	20.11	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
3283	20.04	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
3284	20.04	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
3285	20	kd	CGS001-637	BID	Endogenous ligands			
3286	19.98	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
3287	19.98	kd	CGS001-383	ARG1	Arginase			
3288	19.93	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
3289	19.92	kd	CGS001-10269	ZMPSTE24	-			
3290	19.91	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
3291	19.9	kd	CGS001-5664	PSEN2	Presenilin			
3292	19.84	oe	ccsbBroad304_08536	PARL	-			
3293	19.77	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
3294	19.72	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
3295	19.7	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
3296	19.66	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
3297	19.62	kd	CGS001-7035	TFPI	-			
3298	19.6	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
3299	19.6	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
3300	19.59	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
3301	19.58	kd	CGS001-4174	MCM5	-			
3302	19.57	kd	CGS001-139760	GPR119	GPCR / Class A : Orphans			
3303	19.55	kd	CGS001-23743	BHMT2	-			
3304	19.52	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
3305	19.5	kd	CGS001-3364	HUS1	-			
3306	19.49	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
3307	19.44	kd	CGS001-1861	TOR1A	-			
3308	19.41	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
3309	19.39	oe	ccsbBroad304_04675	ATG4A	-			
3310	19.27	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
3311	19.21	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
3312	19.21	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
3313	19.18	cc		Sterol demethylase inhibitor	-			
3314	19.18	kd	CGS001-11142	PKIG	-			
3315	19.17	cp	BRD-K00532621	midazolam	Benzodiazepine receptor agonist		CYP3A5, CYP3A7, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3	Benzodiazepine receptor agonist
3316	19.15	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
3317	19.13	kd	CGS001-3909	LAMA3	Laminins			
3318	19.1	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
3319	19.09	kd	CGS001-8905	AP1S2	-			
3320	19.04	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
3321	19.01	kd	CGS001-6477	SIAH1	-			
3322	19	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
3323	19	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
3324	19	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
3325	18.99	kd	CGS001-23761	PISD	Decarboxylases			
3326	18.96	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
3327	18.89	kd	CGS001-204851	HIPK1	HIPK subfamily			
3328	18.88	kd	CGS001-10775	POP4	-			
3329	18.88	kd	CGS001-26298	EHF	-			
3330	18.81	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
3331	18.8	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
3332	18.79	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
3333	18.72	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
3334	18.71	kd	CGS001-5361	PLXNA1	Plexins			
3335	18.68	kd	CGS001-604	BCL6	BTB/POZ domain containing			
3336	18.66	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
3337	18.66	kd	CGS001-54505	DHX29	DEAH-boxes			
3338	18.59	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
3339	18.57	kd	CGS001-6632	SNRPD1	-			
3340	18.54	kd	CGS001-3098	HK1	-			
3341	18.5	kd	CGS001-3576	IL8	-			
3342	18.49	oe	ccsbBroad304_00394	CTSD	Cathepsins			
3343	18.49	kd	CGS001-11320	MGAT4A	-			
3344	18.45	kd	CGS001-7013	TERF1	-			
3345	18.43	kd	CGS001-9943	OXSR1	FRAY subfamily			
3346	18.3	kd	CGS001-3673	ITGA2	Integrins			
3347	18.25	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
3348	18.25	cp	BRD-K33226500	indinavir	HIV protease inhibitor		CYP3A5	HIV protease inhibitor
3349	18.24	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
3350	18.23	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
3351	18.21	kd	CGS001-930	CD19	CD molecules			
3352	18.18	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
3353	18.12	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
3354	18.03	kd	CGS001-51422	PRKAG2	AMPK subfamily			
3355	18.02	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
3356	17.98	kd	CGS001-2172	FABP6	Fatty acid binding protein family			
3357	17.86	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
3358	17.84	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
3359	17.77	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
3360	17.73	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
3361	17.69	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3362	17.62	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
3363	17.59	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
3364	17.54	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3365	17.53	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
3366	17.48	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
3367	17.44	kd	CGS001-1503	CTPS	-			
3368	17.38	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
3369	17.37	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
3370	17.35	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
3371	17.32	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
3372	17.31	kd	CGS001-79080	CCDC86	-			
3373	17.3	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
3374	17.18	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
3375	17.16	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
3376	17.07	oe	ccsbBroad304_04649	ADC	-			
3377	16.96	kd	CGS001-23635	SSBP2	-			
3378	16.95	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
3379	16.92	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
3380	16.88	cc		PDGFR/KIT inhibitor	-			
3381	16.84	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
3382	16.69	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
3383	16.57	kd	CGS001-6193	RPS5	S ribosomal proteins			
3384	16.54	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
3385	16.51	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
3386	16.51	kd	CGS001-6196	RPS6KA2	RSK subfamily			
3387	16.48	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
3388	16.47	cc		Nucleoporin LOF	-			
3389	16.47	oe	ccsbBroad304_02218	IKBKE	IKK family			
3390	16.44	kd	CGS001-7428	VHL	-			
3391	16.43	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
3392	16.4	cc		AHSP Pathway LOF	-			
3393	16.4	kd	CGS001-10606	PAICS	-			
3394	16.27	kd	CGS001-533	ATP6V0B	ATPases / V-type			
3395	16.15	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3396	16.1	kd	CGS001-10444	ZER1	ZYG11 cell cycle regulator family			
3397	16.09	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
3398	16.04	kd	CGS001-7405	UVRAG	-			
3399	16	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
3400	15.98	kd	CGS001-9221	NOLC1	-			
3401	15.92	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
3402	15.88	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
3403	15.52	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
3404	15.47	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3405	15.47	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
3406	15.46	kd	CGS001-6098	ROS1	Type XVII RTKs: ROS receptors			
3407	15.27	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
3408	15.25	kd	CGS001-7076	TIMP1	-			
3409	15.21	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
3410	15.17	kd	CGS001-367	AR	Nuclear hormone receptors			
3411	15.15	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
3412	15.11	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
3413	15.09	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
3414	15.02	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
3415	14.91	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
3416	14.86	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
3417	14.67	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
3418	14.65	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
3419	14.6	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
3420	14.33	kd	CGS001-5567	PRKACB	Protein kinase A			
3421	14.25	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
3422	14.25	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
3423	14.2	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
3424	14.2	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
3425	14.07	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3426	14.06	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
3427	13.98	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
3428	13.94	kd	CGS001-58533	SNX6	Sorting nexins			
3429	13.85	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
3430	13.77	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
3431	13.71	kd	CGS001-51071	DERA	-			
3432	13.61	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
3433	13.48	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
3434	13.45	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
3435	13.39	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
3436	13.39	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
3437	13.28	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
3438	13.27	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
3439	13.16	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
3440	13.16	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
3441	13.14	kd	CGS001-55526	DHTKD1	-			
3442	13.11	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
3443	12.86	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
3444	12.78	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
3445	12.74	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
3446	12.73	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3447	12.43	cc		Calmodulin antagonist	-			
3448	12.4	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
3449	12.35	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
3450	12.34	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
3451	12.32	kd	CGS001-955	ENTPD6	-			
3452	12.31	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
3453	12.28	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
3454	12.24	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
3455	12.12	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
3456	11.95	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
3457	11.93	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
3458	11.84	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
3459	11.8	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3460	11.69	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
3461	11.64	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
3462	11.63	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
3463	11.62	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
3464	11.57	kd	CGS001-10123	ARL4C	ADP-ribosylation factors			
3465	11.36	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
3466	11.29	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
3467	11.24	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
3468	11.18	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
3469	11	kd	CGS001-4172	MCM3	-			
3470	10.74	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
3471	10.59	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
3472	10.57	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
3473	10.45	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
3474	10.41	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
3475	10.24	kd	CGS001-6850	SYK	Syk family			
3476	10.17	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
3477	10.08	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
3478	9.89	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
3479	9.64	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
3480	9.63	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
3481	9.56	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
3482	9.44	kd	CGS001-23536	ADAT1	-			
3483	9.35	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
3484	9.33	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
3485	9.3	cc		HIV protease inhibitor	-			
3486	8.88	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
3487	8.74	kd	CGS001-22887	FOXJ3	Forkhead boxes			
3488	8.62	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
3489	8.53	cp	BRD-K23369905	oxiconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3490	8.23	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
3491	8.07	kd	CGS001-1647	GADD45A	-			
3492	8.06	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
3493	7.69	cc		PARP inhibitor	-			
3494	7.17	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
3495	7.03	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
3496	5.81	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3497	4.46	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
3498	-3.08	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
3499	-4.64	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
3500	-4.89	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
3501	-5.36	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
3502	-5.65	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
3503	-6.39	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3504	-6.44	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
3505	-6.77	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
3506	-7.55	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3507	-7.62	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3508	-8.01	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
3509	-8.11	cc		MEK inhibitor	-			
3510	-8.17	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
3511	-8.27	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
3512	-8.44	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
3513	-8.51	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
3514	-8.66	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
3515	-8.69	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
3516	-8.96	kd	CGS001-4087	SMAD2	SMADs			
3517	-9.1	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
3518	-9.17	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
3519	-9.29	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
3520	-9.33	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
3521	-9.36	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
3522	-9.4	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
3523	-9.4	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
3524	-9.67	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
3525	-9.7	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
3526	-9.75	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
3527	-9.76	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
3528	-9.76	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
3529	-9.77	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
3530	-9.88	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
3531	-9.93	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
3532	-9.99	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
3533	-10.18	kd	CGS001-6919	TCEA2	-			
3534	-10.25	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
3535	-10.25	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
3536	-10.34	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
3537	-10.38	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
3538	-10.43	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
3539	-10.54	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3540	-10.65	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
3541	-10.66	kd	CGS001-641	BLM	-			
3542	-10.75	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
3543	-10.96	kd	CGS001-5689	PSMB1	Proteasome subunits			
3544	-11.03	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
3545	-11.04	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
3546	-11.15	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
3547	-11.24	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
3548	-11.29	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
3549	-11.39	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
3550	-11.39	kd	CGS001-6772	STAT1	SH2 domain containing			
3551	-11.52	oe	ccsbBroad304_03177	FIS1	-			
3552	-11.53	cp	BRD-A39172021	ampiroxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3553	-11.57	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
3554	-11.58	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
3555	-11.6	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3556	-11.81	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
3557	-11.93	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
3558	-12.01	kd	CGS001-7157	TP53	-			
3559	-12.09	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
3560	-12.22	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
3561	-12.22	kd	CGS001-998	CDC42	-			
3562	-12.32	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3563	-12.44	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
3564	-12.49	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
3565	-12.53	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
3566	-12.64	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
3567	-12.65	kd	CGS001-124583	CANT1	-			
3568	-12.7	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
3569	-12.78	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
3570	-12.81	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
3571	-12.83	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
3572	-12.84	kd	CGS001-1528	CYB5A	Cytochrome b genes			
3573	-12.9	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
3574	-12.9	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3575	-12.94	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
3576	-13	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
3577	-13.03	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
3578	-13.1	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
3579	-13.12	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
3580	-13.13	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
3581	-13.16	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
3582	-13.27	cc		Toll like receptors LOF	-			
3583	-13.31	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
3584	-13.32	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
3585	-13.35	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3586	-13.36	kd	CGS001-1429	CRYZ	-			
3587	-13.37	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
3588	-13.44	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
3589	-13.46	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3590	-13.53	kd	CGS001-55256	ADI1	-			
3591	-13.6	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
3592	-13.62	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
3593	-13.74	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
3594	-13.75	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
3595	-13.82	kd	CGS001-3329	HSPD1	Heat Shock Proteins / Chaperonins			
3596	-13.83	cc		Mitogen activated protein kinases LOF	-			
3597	-13.86	cc		Cyclins LOF	-			
3598	-13.87	kd	CGS001-7018	TF	-			
3599	-13.94	kd	CGS001-1026	CDKN1A	-			
3600	-13.95	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
3601	-13.96	kd	CGS001-51222	ZNF219	Zinc fingers, C2H2-type			
3602	-14.04	cp	BRD-K94144010	cotinine	Nicotine metabolite			Nicotine metabolite
3603	-14.07	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
3604	-14.21	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3605	-14.23	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
3606	-14.32	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
3607	-14.32	kd	CGS001-25842	ASF1A	-			
3608	-14.34	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
3609	-14.35	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
3610	-14.36	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
3611	-14.39	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
3612	-14.43	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
3613	-14.43	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
3614	-14.43	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
3615	-14.44	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
3616	-14.48	kd	CGS001-147686	ZNF418	Zinc fingers, C2H2-type			
3617	-14.55	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
3618	-14.58	kd	CGS001-7097	TLR2	Toll-like receptor family			
3619	-14.6	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
3620	-14.62	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
3621	-14.65	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
3622	-14.65	kd	CGS001-4221	MEN1	-			
3623	-14.67	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
3624	-14.79	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
3625	-14.84	cc		T-type calcium channel blocker	-			
3626	-14.87	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
3627	-14.87	kd	CGS001-1616	DAXX	-			
3628	-14.88	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
3629	-14.93	oe	ccsbBroad304_08709	SCYL3	-			
3630	-15.02	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
3631	-15.03	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
3632	-15.03	cp	BRD-K55034111	pefloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
3633	-15.07	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
3634	-15.07	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
3635	-15.14	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
3636	-15.2	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3637	-15.36	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
3638	-15.42	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
3639	-15.5	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
3640	-15.53	kd	CGS001-10250	SRRM1	-			
3641	-15.53	kd	CGS001-5253	PHF2	Histone demethylases			
3642	-15.55	kd	CGS001-10221	TRIB1	Trbl family			
3643	-15.58	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
3644	-15.61	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
3645	-15.72	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
3646	-15.79	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
3647	-15.79	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
3648	-15.84	kd	CGS001-28960	DCPS	-			
3649	-15.85	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
3650	-15.87	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
3651	-15.92	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
3652	-15.93	kd	CGS001-5810	RAD1	-			
3653	-15.95	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
3654	-15.97	kd	CGS001-4734	NEDD4	-			
3655	-15.99	kd	CGS001-124626	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3656	-15.99	kd	CGS001-51292	GMPR2	-			
3657	-16	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
3658	-16.02	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
3659	-16.07	kd	CGS001-5575	PRKAR1B	Protein kinase A			
3660	-16.07	kd	CGS001-56922	MCCC1	-			
3661	-16.1	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
3662	-16.11	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
3663	-16.12	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
3664	-16.15	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
3665	-16.18	cc		SMAD family LOF	-			
3666	-16.31	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
3667	-16.37	kd	CGS001-25861	DFNB31	-			
3668	-16.39	kd	CGS001-839	CASP6	Caspases			
3669	-16.55	oe	ccsbBroad304_07557	NAMPT	-			
3670	-16.57	cc		Tricyclic antidepressant	-			
3671	-16.58	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
3672	-16.6	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
3673	-16.61	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
3674	-16.7	kd	CGS001-4485	MST1	-			
3675	-16.74	cp	BRD-K89708791	rifaximin	RNA synthesis inhibitor		NR1I2, CYP3A4	RNA synthesis inhibitor
3676	-16.74	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3677	-16.75	kd	CGS001-55191	NADSYN1	-			
3678	-16.77	cp	BRD-K81916719	triclabendazole	Microtubule inhibitor		DNMT1	Microtubule inhibitor
3679	-16.83	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
3680	-16.85	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
3681	-16.87	cc		Sodium channel blocker	-			
3682	-16.98	kd	CGS001-7840	ALMS1	-			
3683	-17.04	kd	CGS001-11200	CHEK2	CHK1 subfamily			
3684	-17.05	cp	BRD-K34437622	BRD-K34437622	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
3685	-17.19	cc		FOS transcription factor family GOF	-			
3686	-17.19	oe	ccsbBroad304_00854	IL8	-			
3687	-17.2	kd	CGS001-4208	MEF2C	Myocyte enhancer factors			
3688	-17.22	oe	ccsbBroad304_00009	ACLY	-			
3689	-17.23	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
3690	-17.28	kd	CGS001-4947	OAZ2	-			
3691	-17.3	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
3692	-17.32	kd	CGS001-2864	FFAR1	Fatty acid receptors			
3693	-17.35	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
3694	-17.38	kd	CGS001-4086	SMAD1	SMADs			
3695	-17.41	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
3696	-17.42	kd	CGS001-57459	GATAD2B	GATA zinc finger domain containing			
3697	-17.44	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
3698	-17.44	kd	CGS001-8720	MBTPS1	Subtilisin			
3699	-17.48	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
3700	-17.49	cp	BRD-A00520476	otenzepad	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
3701	-17.53	kd	CGS001-10523	CHERP	G patch domain containing			
3702	-17.57	kd	CGS001-375133	PI4KAP2	-			
3703	-17.6	cc		FXR antagonist	-			
3704	-17.64	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
3705	-17.65	oe	ccsbBroad304_04655	TRIM9	-			
3706	-17.66	cc		Wnt family GOF	-			
3707	-17.67	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
3708	-17.67	kd	CGS001-2167	FABP4	Fatty acid binding protein family			
3709	-17.78	kd	CGS001-3481	IGF2	-			
3710	-17.87	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
3711	-17.9	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
3712	-17.96	oe	ccsbBroad304_05745	CD24	CD molecules			
3713	-17.98	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
3714	-18.02	kd	CGS001-302	ANXA2	Annexins			
3715	-18.05	kd	CGS001-1504	CTRB1	-			
3716	-18.09	oe	ccsbBroad304_06837	RAF1	RAF family			
3717	-18.1	cc		Akt Signaling LOF	-			
3718	-18.11	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
3719	-18.13	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
3720	-18.14	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
3721	-18.14	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3722	-18.14	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
3723	-18.14	kd	CGS001-389421	LIN28B	-			
3724	-18.16	kd	CGS001-6832	SUPV3L1	-			
3725	-18.19	kd	CGS001-65263	PYCRL	-			
3726	-18.22	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
3727	-18.22	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3728	-18.25	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
3729	-18.25	kd	CGS001-79947	DHDDS	-			
3730	-18.3	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
3731	-18.31	kd	CGS001-9318	COPS2	-			
3732	-18.36	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3733	-18.37	kd	CGS001-2114	ETS2	ETS Transcription Factors			
3734	-18.41	kd	CGS001-5654	HTRA1	Serine peptidases / Serine peptidases			
3735	-18.42	kd	CGS001-54623	PAF1	-			
3736	-18.52	kd	CGS001-1515	CTSL2	-			
3737	-18.58	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
3738	-18.58	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3739	-18.59	cc		MTOR inhibitor	-			
3740	-18.61	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
3741	-18.65	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
3742	-18.7	kd	CGS001-143187	VTI1A	-			
3743	-18.71	oe	ccsbBroad304_03658	DCP1A	-			
3744	-18.72	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
3745	-18.75	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
3746	-18.78	kd	CGS001-26191	PTPN22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
3747	-18.79	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
3748	-18.8	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
3749	-18.8	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
3750	-18.81	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3751	-18.85	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
3752	-18.85	kd	CGS001-2885	GRB2	SH2 domain containing			
3753	-18.87	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
3754	-18.87	kd	CGS001-444	ASPH	-			
3755	-18.88	cp	BRD-K73196317	urapidil	Adrenergic receptor antagonist		HTR1A	Adrenergic receptor antagonist
3756	-18.89	kd	CGS001-4023	LPL	-			
3757	-18.92	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
3758	-18.97	kd	CGS001-4837	NNMT	-			
3759	-19.08	oe	ccsbBroad304_02086	PDLIM1	-			
3760	-19.11	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
3761	-19.17	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
3762	-19.21	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
3763	-19.26	kd	CGS001-151126	ZNF385B	-			
3764	-19.3	oe	ccsbBroad304_02278	THRAP3	-			
3765	-19.35	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3766	-19.37	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
3767	-19.38	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
3768	-19.4	oe	ccsbBroad304_10846	GGT1	CD molecules			
3769	-19.4	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
3770	-19.41	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
3771	-19.46	kd	CGS001-3163	HMOX2	Haem oxygenase			
3772	-19.59	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3773	-19.66	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
3774	-19.78	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
3775	-19.79	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
3776	-19.8	kd	CGS001-10020	GNE	-			
3777	-19.81	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
3778	-19.84	oe	ccsbBroad304_02605	PAPD7	-			
3779	-19.84	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
3780	-19.87	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
3781	-19.88	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
3782	-19.89	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
3783	-19.97	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
3784	-19.97	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
3785	-20.02	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
3786	-20.03	kd	CGS001-4047	LSS	Lanosterol biosynthesis pathway			
3787	-20.05	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3788	-20.05	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3789	-20.06	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
3790	-20.06	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
3791	-20.06	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
3792	-20.07	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
3793	-20.11	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
3794	-20.12	oe	ccsbBroad304_00102	RND3	-			
3795	-20.16	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
3796	-20.18	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
3797	-20.19	kd	CGS001-63892	THADA	-			
3798	-20.2	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
3799	-20.2	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
3800	-20.21	kd	CGS001-79109	MAPKAP1	-			
3801	-20.26	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
3802	-20.27	oe	ccsbBroad304_06663	OAS1	-			
3803	-20.29	kd	CGS001-6932	TCF7	-			
3804	-20.29	kd	CGS001-2673	GFPT1	-			
3805	-20.34	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3806	-20.35	kd	CGS001-8655	DYNLL1	Cytoplasmic dyneins			
3807	-20.37	kd	CGS001-1981	EIF4G1	Parkinson disease			
3808	-20.38	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
3809	-20.38	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
3810	-20.4	oe	ccsbBroad304_02838	SDF2L1	-			
3811	-20.41	kd	CGS001-5595	MAPK3	MAPK:ERK subfamily			
3812	-20.44	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
3813	-20.46	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
3814	-20.56	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
3815	-20.57	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
3816	-20.57	kd	CGS001-388650	FAM69A	-			
3817	-20.58	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
3818	-20.61	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
3819	-20.62	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
3820	-20.63	kd	CGS001-6258	RXRG	Retinoid X receptors			
3821	-20.63	kd	CGS001-5579	PRKCB	Alpha subfamily			
3822	-20.66	oe	ccsbBroad304_00986	MCM2	-			
3823	-20.66	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
3824	-20.69	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3825	-20.7	oe	ccsbBroad304_00376	CSK	Csk family			
3826	-20.7	kd	CGS001-3169	FOXA1	Forkhead boxes			
3827	-20.72	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
3828	-20.74	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
3829	-20.75	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
3830	-20.77	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
3831	-20.78	kd	CGS001-581	BAX	-			
3832	-20.8	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
3833	-20.93	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
3834	-20.94	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
3835	-20.95	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
3836	-20.97	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
3837	-20.98	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
3838	-20.99	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
3839	-21.05	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
3840	-21.06	oe	ccsbBroad304_10207	ERLIN1	-			
3841	-21.06	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
3842	-21.06	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
3843	-21.07	kd	CGS001-55832	CAND1	-			
3844	-21.08	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
3845	-21.1	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
3846	-21.11	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
3847	-21.12	kd	CGS001-26149	ZNF658	Zinc fingers, C2H2-type			
3848	-21.2	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
3849	-21.2	kd	CGS001-5160	PDHA1	-			
3850	-21.2	kd	CGS001-760	CA2	Carbonic anhydrases			
3851	-21.21	kd	CGS001-8446	DUSP11	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
3852	-21.23	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
3853	-21.27	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
3854	-21.35	kd	CGS001-64781	CERK	Ceramide kinase			
3855	-21.36	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
3856	-21.37	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
3857	-21.42	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
3858	-21.43	kd	CGS001-9252	RPS6KA5	MSK subfamily			
3859	-21.45	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
3860	-21.47	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
3861	-21.5	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
3862	-21.54	oe	ccsbBroad304_03798	PHTF2	-			
3863	-21.55	kd	CGS001-6541	SLC7A1	SLC7 family			
3864	-21.55	kd	CGS001-652	BMP4	Bone morphogenetic proteins			
3865	-21.57	kd	CGS001-1869	E2F1	-			
3866	-21.58	kd	CGS001-56675	NRIP3	-			
3867	-21.59	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
3868	-21.6	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
3869	-21.63	kd	CGS001-29079	MED4	-			
3870	-21.65	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
3871	-21.67	cc		Canonical high mobility group proteins LOF	-			
3872	-21.68	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
3873	-21.74	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
3874	-21.8	kd	CGS001-222546	RFX6	-			
3875	-21.8	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
3876	-21.81	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
3877	-21.82	oe	ccsbBroad304_00115	ASPH	-			
3878	-21.83	kd	CGS001-9512	PMPCB	-			
3879	-21.85	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
3880	-21.86	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
3881	-21.9	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
3882	-21.91	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
3883	-22	oe	ccsbBroad304_08684	CXCR7	-			
3884	-22.01	kd	CGS001-83637	ZMIZ2	Zinc fingers, MIZ-type			
3885	-22.03	kd	CGS001-64175	LEPRE1	-			
3886	-22.13	kd	CGS001-2348	FOLR1	-			
3887	-22.14	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
3888	-22.19	kd	CGS001-7389	UROD	-			
3889	-22.19	kd	CGS001-7099	TLR4	Toll-like receptor family			
3890	-22.19	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
3891	-22.22	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
3892	-22.24	oe	ccsbBroad304_00053	ALDOA	-			
3893	-22.25	kd	CGS001-57215	THAP11	THAP (C2CH-type zinc finger) domain containing			
3894	-22.25	kd	CGS001-5916	RARG	Retinoic acid receptors			
3895	-22.29	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
3896	-22.29	kd	CGS001-1119	CHKA	-			
3897	-22.31	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
3898	-22.31	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
3899	-22.35	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
3900	-22.37	oe	ccsbBroad304_02589	COPS5	-			
3901	-22.37	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
3902	-22.4	kd	CGS001-3783	KCNN4	Calcium-activated potassium channels			
3903	-22.4	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
3904	-22.41	kd	CGS001-2877	GPX2	-			
3905	-22.45	kd	CGS001-3155	HMGCL	-			
3906	-22.46	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
3907	-22.48	kd	CGS001-9641	IKBKE	IKK family			
3908	-22.49	cp	BRD-A43082555	loxoprofen	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
3909	-22.49	kd	CGS001-5883	RAD9A	-			
3910	-22.52	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
3911	-22.55	kd	CGS001-8467	SMARCA5	-			
3912	-22.57	cp	BRD-K29653726	topiramate	Carbonic anhydrase inhibitor		CA2, CA4, GRIK1, CA1, CA12, CA7, CYP2C19, CYP3A4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA1, SCN1A, SCN5A	Carbonic anhydrase inhibitor, Glutamate receptor antagonist, Kainate receptor antagonist
3913	-22.58	kd	CGS001-8453	CUL2	-			
3914	-22.61	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
3915	-22.63	cc		Gamma secretase inhibitor	-			
3916	-22.63	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
3917	-22.67	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
3918	-22.68	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
3919	-22.73	kd	CGS001-6821	SUOX	-			
3920	-22.78	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3921	-22.78	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
3922	-22.81	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
3923	-22.81	oe	ccsbBroad304_02843	FTSJ1	-			
3924	-22.81	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
3925	-22.82	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
3926	-22.82	kd	CGS001-708	C1QBP	-			
3927	-22.88	kd	CGS001-79258	MMEL1	-			
3928	-22.91	oe	ccsbBroad304_11405	UBE3C	-			
3929	-22.91	kd	CGS001-83933	HDAC10	Histone deacetylases			
3930	-22.91	kd	CGS001-55612	FERMT1	Fermitins			
3931	-23.01	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
3932	-23.02	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
3933	-23.04	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
3934	-23.06	kd	CGS001-7486	WRN	-			
3935	-23.07	oe	ccsbBroad304_00184	C2	Complement system			
3936	-23.08	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
3937	-23.09	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
3938	-23.1	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
3939	-23.13	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
3940	-23.14	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
3941	-23.15	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
3942	-23.15	cp	BRD-K25310650	ormetoprim	Bacterial antifolate			Bacterial antifolate
3943	-23.16	kd	CGS001-6364	CCL20	Chemokine ligands			
3944	-23.2	oe	ccsbBroad304_06765	PRCC	-			
3945	-23.22	kd	CGS001-467	ATF3	basic leucine zipper proteins			
3946	-23.25	kd	CGS001-399664	MEX3D	Mex-3 homologs			
3947	-23.27	kd	CGS001-10587	TXNRD2	-			
3948	-23.29	kd	CGS001-10019	SH2B3	Pleckstrin homology (PH) domain containing			
3949	-23.3	kd	CGS001-10607	TBL3	WD repeat domain containing			
3950	-23.31	kd	CGS001-2735	GLI1	Zinc fingers, C2H2-type			
3951	-23.37	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
3952	-23.39	kd	CGS001-9945	GFPT2	-			
3953	-23.42	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
3954	-23.44	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3955	-23.45	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
3956	-23.45	kd	CGS001-2495	FTH1	-			
3957	-23.47	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
3958	-23.47	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
3959	-23.51	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
3960	-23.52	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
3961	-23.6	oe	ccsbBroad304_00223	CASP9	Caspases			
3962	-23.61	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3963	-23.64	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
3964	-23.65	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
3965	-23.66	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
3966	-23.67	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
3967	-23.68	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
3968	-23.68	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
3969	-23.71	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
3970	-23.73	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
3971	-23.75	oe	ccsbBroad304_09833	SENP5	-			
3972	-23.75	kd	CGS001-5931	RBBP7	WD repeat domain containing			
3973	-23.76	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3974	-23.76	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
3975	-23.77	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
3976	-23.79	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3977	-23.81	kd	CGS001-3956	LGALS1	Endogenous ligands			
3978	-23.82	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
3979	-23.84	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
3980	-23.86	kd	CGS001-1028	CDKN1C	-			
3981	-23.89	kd	CGS001-602	BCL3	Ankyrin repeat domain containing			
3982	-23.94	kd	CGS001-811	CALR	-			
3983	-23.95	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
3984	-23.96	kd	CGS001-10465	PPIH	-			
3985	-23.97	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
3986	-24.08	kd	CGS001-50604	IL20	Interleukins and interleukin receptors			
3987	-24.08	oe	ccsbBroad304_06264	GBP2	-			
3988	-24.11	oe	ccsbBroad304_07219	CDC7	CDC7 family			
3989	-24.11	kd	CGS001-11182	SLC2A6	Solute carriers			
3990	-24.12	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
3991	-24.14	kd	CGS001-595	CCND1	-			
3992	-24.17	kd	CGS001-11343	MGLL	Endocannabinoid turnover			
3993	-24.18	kd	CGS001-23102	TBC1D2B	-			
3994	-24.2	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
3995	-24.21	kd	CGS001-22954	TRIM32	-			
3996	-24.23	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
3997	-24.23	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
3998	-24.28	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
3999	-24.29	kd	CGS001-50808	AK3	-			
4000	-24.3	kd	CGS001-6464	SHC1	SH2 domain containing			
4001	-24.31	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
4002	-24.35	oe	ccsbBroad304_00424	DBI	-			
4003	-24.35	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
4004	-24.35	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
4005	-24.36	oe	ccsbBroad304_00471	E2F6	-			
4006	-24.37	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
4007	-24.37	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
4008	-24.41	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
4009	-24.42	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
4010	-24.42	kd	CGS001-2987	GUK1	-			
4011	-24.43	kd	CGS001-5710	PSMD4	Proteasome (prosome, macropain) subunits			
4012	-24.45	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
4013	-24.46	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
4014	-24.46	kd	CGS001-2147	F2	Endogenous ligands			
4015	-24.47	kd	CGS001-55634	ZNF673	-			
4016	-24.5	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
4017	-24.51	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
4018	-24.53	oe	ccsbBroad304_02955	MYCBP	-			
4019	-24.54	kd	CGS001-6304	SATB1	Homeoboxes / CUT class			
4020	-24.55	kd	CGS001-10608	MXD4	Basic helix-loop-helix proteins			
4021	-24.57	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
4022	-24.58	oe	ccsbBroad304_01754	UCK2	-			
4023	-24.58	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4024	-24.6	oe	ccsbBroad304_03450	TMED9	-			
4025	-24.64	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
4026	-24.65	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
4027	-24.66	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
4028	-24.68	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
4029	-24.71	kd	CGS001-10955	SERINC3	-			
4030	-24.72	oe	ccsbBroad304_01658	PRDX2	-			
4031	-24.72	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
4032	-24.73	oe	ccsbBroad304_07515	GFPT2	-			
4033	-24.76	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
4034	-24.77	kd	CGS001-6646	SOAT1	-			
4035	-24.77	kd	CGS001-861	RUNX1	-			
4036	-24.77	kd	CGS001-221895	JAZF1	Zinc fingers, C2H2-type			
4037	-24.78	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
4038	-24.8	kd	CGS001-5577	PRKAR2B	Protein kinase A			
4039	-24.88	kd	CGS001-1036	CDO1	-			
4040	-24.89	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
4041	-24.89	oe	ccsbBroad304_02432	IFI30	-			
4042	-24.9	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
4043	-24.91	kd	CGS001-9688	NUP93	-			
4044	-24.94	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
4045	-24.95	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
4046	-24.99	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
4047	-25.02	kd	CGS001-4175	MCM6	-			
4048	-25.03	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
4049	-25.05	oe	ccsbBroad304_01234	POLB	DNA polymerases			
4050	-25.05	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
4051	-25.05	kd	CGS001-4144	MAT2A	-			
4052	-25.07	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
4053	-25.08	kd	CGS001-8741	TNFSF13	CD molecules			
4054	-25.11	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
4055	-25.12	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
4056	-25.13	kd	CGS001-81539	SLC38A1	System A-like transporters			
4057	-25.14	kd	CGS001-4841	NONO	RNA binding motif (RRM) containing			
4058	-25.15	oe	ccsbBroad304_04616	ORMDL3	-			
4059	-25.15	kd	CGS001-191	AHCY	Adenosine turnover			
4060	-25.15	oe	ccsbBroad304_01577	SOD1	-			
4061	-25.16	kd	CGS001-23057	NMNAT2	-			
4062	-25.2	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
4063	-25.23	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
4064	-25.25	kd	CGS001-5033	P4HA1	-			
4065	-25.3	kd	CGS001-2963	GTF2F2	General transcription factors			
4066	-25.31	kd	CGS001-5134	PDCD2	Zinc fingers, MYND-type			
4067	-25.36	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
4068	-25.38	kd	CGS001-10084	PQBP1	-			
4069	-25.39	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
4070	-25.41	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
4071	-25.41	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
4072	-25.42	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
4073	-25.44	cp	BRD-K96740444	itopride	Dopamine receptor antagonist		DRD2, ACHE, CHRM3	Dopamine receptor antagonist
4074	-25.46	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
4075	-25.47	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
4076	-25.47	kd	CGS001-9612	NCOR2	-			
4077	-25.49	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
4078	-25.5	kd	CGS001-7727	ZNF174	Zinc fingers, C2H2-type			
4079	-25.51	cp	BRD-K33106058	cytarabine	Ribonucleotide reductase inhibitor		POLB, POLA1	Ribonucleotide reductase inhibitor
4080	-25.51	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
4081	-25.54	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
4082	-25.56	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
4083	-25.56	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
4084	-25.58	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
4085	-25.58	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
4086	-25.61	cp	BRD-K63265447	docetaxel	Tubulin inhibitor		TUBB, BCL2, MAP2, MAP4, MAPT, NR1I2, TUBB1	Tubulin inhibitor
4087	-25.61	oe	ccsbBroad304_02306	PQBP1	-			
4088	-25.65	oe	ccsbBroad304_04490	RSPH1	-			
4089	-25.68	kd	CGS001-93185	IGSF8	CD molecules			
4090	-25.69	cp	BRD-A68888262	azelastine	Histamine receptor antagonist		HRH1, CYP2C19	Histamine receptor antagonist
4091	-25.69	kd	CGS001-285676	ZNF454	Zinc fingers, C2H2-type			
4092	-25.69	kd	CGS001-4089	SMAD4	SMADs			
4093	-25.69	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
4094	-25.7	kd	CGS001-1948	EFNB2	Ephrins			
4095	-25.71	kd	CGS001-259	AMBP	Lipocalins			
4096	-25.74	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
4097	-25.75	kd	CGS001-5300	PIN1	-			
4098	-25.76	cc		Bacterial DNA gyrase inhibitor	-			
4099	-25.76	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
4100	-25.77	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
4101	-25.78	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
4102	-25.78	kd	CGS001-5411	PNN	-			
4103	-25.79	kd	CGS001-8848	TSC22D1	-			
4104	-25.81	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
4105	-25.81	kd	CGS001-23118	TAB2	-			
4106	-25.81	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
4107	-25.83	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
4108	-25.87	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
4109	-25.91	oe	ccsbBroad304_05590	NOTCH2NL	-			
4110	-25.92	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
4111	-25.95	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
4112	-25.96	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
4113	-25.99	kd	CGS001-56731	SLC2A4RG	-			
4114	-25.99	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
4115	-26	kd	CGS001-84930	MASTL	MAST family			
4116	-26.01	oe	ccsbBroad304_00101	RHOC	-			
4117	-26.04	kd	CGS001-4968	OGG1	-			
4118	-26.07	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
4119	-26.07	kd	CGS001-4688	NCF2	Tetratricopeptide (TTC) repeat domain containing			
4120	-26.08	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
4121	-26.12	cp	BRD-K07237224	moclobemide	Monoamine oxidase inhibitor		MAOA, CYP2C19, MAOB	Monoamine oxidase inhibitor
4122	-26.13	oe	ccsbBroad304_09881	RFX6	-			
4123	-26.13	oe	ccsbBroad304_05907	BUB1B	Bub family			
4124	-26.13	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
4125	-26.13	kd	CGS001-498	ATP5A1	ATPases / F-type			
4126	-26.13	kd	CGS001-283	ANG	Ribonucleases, RNase A			
4127	-26.15	oe	ccsbBroad304_00657	GNG4	-			
4128	-26.16	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
4129	-26.17	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
4130	-26.17	kd	CGS001-84288	EFCAB2	EF-hand domain containing			
4131	-26.25	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
4132	-26.25	kd	CGS001-3705	ITPK1	-			
4133	-26.25	kd	CGS001-1398	CRK	SH2 domain containing			
4134	-26.27	kd	CGS001-944	TNFSF8	CD molecules			
4135	-26.27	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
4136	-26.27	kd	CGS001-3281	HSBP1	-			
4137	-26.27	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
4138	-26.28	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
4139	-26.29	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
4140	-26.31	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
4141	-26.36	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
4142	-26.39	oe	ccsbBroad304_06889	RPN2	-			
4143	-26.41	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
4144	-26.46	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
4145	-26.46	kd	CGS001-8089	YEATS4	-			
4146	-26.52	kd	CGS001-54749	EPDR1	-			
4147	-26.53	kd	CGS001-3074	HEXB	-			
4148	-26.54	cc		PKC inhibitor	-			
4149	-26.56	kd	CGS001-3161	HMMR	CD molecules			
4150	-26.57	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
4151	-26.57	kd	CGS001-93134	ZNF561	Zinc fingers, C2H2-type			
4152	-26.61	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
4153	-26.68	oe	ccsbBroad304_09195	MCM8	-			
4154	-26.7	oe	ccsbBroad304_05439	O3FAR1	-			
4155	-26.71	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
4156	-26.72	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
4157	-26.73	kd	CGS001-23043	TNIK	MSN subfamily			
4158	-26.73	kd	CGS001-5663	PSEN1	Presenilin			
4159	-26.73	kd	CGS001-2664	GDI1	-			
4160	-26.74	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
4161	-26.75	kd	CGS001-7185	TRAF1	-			
4162	-26.77	cc		General transcription factors group 2 LOF	-			
4163	-26.77	kd	CGS001-22905	EPN2	-			
4164	-26.78	kd	CGS001-51655	RASD1	-			
4165	-26.82	cp	BRD-K40758068	efavirenz	HIV protease inhibitor		CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5	HIV protease inhibitor
4166	-26.83	kd	CGS001-11267	SNF8	-			
4167	-26.85	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
4168	-26.86	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
4169	-26.91	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
4170	-26.91	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
4171	-26.91	kd	CGS001-5371	PML	RING-type (C3HC4) zinc fingers			
4172	-26.98	cp	BRD-K44353683	nateglinide	Insulin secretagogue		ABCC8, KCNJ11, CYP3A4, INS, KCNJ10, PPARG	Insulin secretagogue
4173	-26.98	kd	CGS001-6741	SSB	La ribonucleoprotein domain containing			
4174	-26.98	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
4175	-26.99	oe	ccsbBroad304_09708	PNLDC1	-			
4176	-26.99	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
4177	-27	kd	CGS001-54566	EPB41L4B	-			
4178	-27.01	kd	CGS001-4724	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
4179	-27.03	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
4180	-27.06	kd	CGS001-5211	PFKL	-			
4181	-27.08	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
4182	-27.08	kd	CGS001-54925	ZNF434	-			
4183	-27.09	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
4184	-27.1	cc		Interleukins GOF	-			
4185	-27.1	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
4186	-27.1	kd	CGS001-51174	TUBD1	Tubulins			
4187	-27.11	kd	CGS001-133522	PPARGC1B	RNA binding motif (RRM) containing			
4188	-27.12	kd	CGS001-390980	ZNF805	Zinc fingers, C2H2-type			
4189	-27.15	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
4190	-27.15	kd	CGS001-51601	LIPT1	-			
4191	-27.16	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4192	-27.16	kd	CGS001-103	ADAR	-			
4193	-27.19	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
4194	-27.2	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
4195	-27.21	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
4196	-27.21	kd	CGS001-4074	M6PR	-			
4197	-27.24	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
4198	-27.24	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
4199	-27.25	kd	CGS001-5264	PHYH	-			
4200	-27.31	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
4201	-27.34	kd	CGS001-471	ATIC	-			
4202	-27.36	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
4203	-27.38	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
4204	-27.39	cp	BRD-K59456551	methotrexate	Dihydrofolate reductase inhibitor		DHFR, AOX1, FOLR1, TYMS	Dihydrofolate reductase inhibitor
4205	-27.43	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
4206	-27.43	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
4207	-27.47	oe	ccsbBroad304_04465	RERG	-			
4208	-27.48	kd	CGS001-2277	FIGF	-			
4209	-27.49	oe	ccsbBroad304_00933	LDHB	-			
4210	-27.49	kd	CGS001-6822	SULT2A1	Sulfotransferases, cytosolic			
4211	-27.49	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
4212	-27.49	kd	CGS001-55214	LEPREL1	-			
4213	-27.51	cc		C2 domain containing protein kinases LOF	-			
4214	-27.51	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
4215	-27.55	oe	ccsbBroad304_03112	NENF	-			
4216	-27.61	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
4217	-27.62	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
4218	-27.67	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
4219	-27.68	kd	CGS001-2168	FABP1	Fatty acid-binding proteins			
4220	-27.68	oe	ccsbBroad304_03040	NKIRAS2	-			
4221	-27.7	oe	ccsbBroad304_00262	CD59	CD molecules			
4222	-27.7	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
4223	-27.73	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
4224	-27.75	kd	CGS001-388	RHOB	-			
4225	-27.85	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
4226	-27.85	cp	BRD-K37814297	acepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
4227	-27.89	kd	CGS001-4833	NME4	-			
4228	-27.99	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
4229	-28.01	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
4230	-28.03	kd	CGS001-5824	PEX19	-			
4231	-28.04	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
4232	-28.06	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
4233	-28.06	kd	CGS001-9807	IP6K1	-			
4234	-28.07	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
4235	-28.07	kd	CGS001-819	CAMLG	-			
4236	-28.08	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
4237	-28.12	cc		ATP synthase inhibitor	-			
4238	-28.12	kd	CGS001-7158	TP53BP1	-			
4239	-28.15	oe	ccsbBroad304_05528	TICAM2	-			
4240	-28.16	kd	CGS001-2882	GPX7	-			
4241	-28.16	kd	CGS001-718	C3	Endogenous ligands			
4242	-28.17	oe	ccsbBroad304_07217	AXIN2	-			
4243	-28.18	kd	CGS001-5362	PLXNA2	Plexins			
4244	-28.28	oe	ccsbBroad304_06777	PRNP	CD molecules			
4245	-28.28	kd	CGS001-1497	CTNS	-			
4246	-28.3	kd	CGS001-7003	TEAD1	-			
4247	-28.3	kd	CGS001-1314	COPA	Endogenous ligands			
4248	-28.31	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
4249	-28.33	oe	ccsbBroad304_03237	LEF1	-			
4250	-28.33	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
4251	-28.35	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
4252	-28.39	kd	CGS001-5910	RAP1GDS1	Armadillo repeat containing			
4253	-28.4	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
4254	-28.41	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
4255	-28.43	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
4256	-28.45	oe	ccsbBroad304_07050	TFAP2A	-			
4257	-28.46	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
4258	-28.46	kd	CGS001-4704	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4259	-28.51	kd	CGS001-164091	PAQR7	-			
4260	-28.51	kd	CGS001-2773	GNAI3	-			
4261	-28.52	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
4262	-28.54	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4263	-28.55	oe	ccsbBroad304_02136	COPS2	-			
4264	-28.56	oe	ccsbBroad304_06188	F10	Chymotrypsin			
4265	-28.56	kd	CGS001-1512	CTSH	Cathepsins			
4266	-28.6	oe	ccsbBroad304_02452	NXF1	-			
4267	-28.6	kd	CGS001-7032	TFF2	-			
4268	-28.62	oe	ccsbBroad304_01379	RBBP6	-			
4269	-28.62	kd	CGS001-8935	SKAP2	Pleckstrin homology (PH) domain containing			
4270	-28.63	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
4271	-28.64	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
4272	-28.67	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
4273	-28.7	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
4274	-28.7	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
4275	-28.71	oe	ccsbBroad304_12226	NAGK	-			
4276	-28.73	cc		MCM family LOF	-			
4277	-28.73	kd	CGS001-170591	S100Z	EF-hand domain containing			
4278	-28.73	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
4279	-28.77	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
4280	-28.79	oe	ccsbBroad304_02884	POT1	-			
4281	-28.81	kd	CGS001-6251	RSU1	-			
4282	-28.81	kd	CGS001-80274	SCUBE1	-			
4283	-28.82	cc		Vitamin D receptor agonist	-			
4284	-28.82	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
4285	-28.85	oe	ccsbBroad304_02738	RRS1	-			
4286	-28.86	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
4287	-28.89	kd	CGS001-226	ALDOA	-			
4288	-29	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
4289	-29	kd	CGS001-84109	QRFPR	GPCR / Class A : RF amide peptide receptors			
4290	-29.02	kd	CGS001-29968	PSAT1	-			
4291	-29.03	kd	CGS001-5163	PDK1	-			
4292	-29.05	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
4293	-29.05	kd	CGS001-23466	CBX6	-			
4294	-29.07	oe	ccsbBroad304_01142	PAFAH1B2	-			
4295	-29.07	kd	CGS001-7083	TK1	-			
4296	-29.09	kd	CGS001-169436	C9ORF96	-			
4297	-29.1	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
4298	-29.1	kd	CGS001-2752	GLUL	-			
4299	-29.14	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
4300	-29.14	kd	CGS001-94234	FOXQ1	Forkhead boxes			
4301	-29.16	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
4302	-29.18	kd	CGS001-9690	UBE3C	-			
4303	-29.2	cc		Na-K-Cl transporter inhibitor	-			
4304	-29.2	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
4305	-29.21	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
4306	-29.23	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
4307	-29.27	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
4308	-29.3	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
4309	-29.31	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
4310	-29.35	kd	CGS001-4547	MTTP	-			
4311	-29.38	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
4312	-29.38	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
4313	-29.38	kd	CGS001-900	CCNG1	-			
4314	-29.4	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
4315	-29.42	kd	CGS001-54659	UGT1A3	UDP glucuronosyltransferases			
4316	-29.44	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
4317	-29.44	oe	ccsbBroad304_06294	GNAZ	-			
4318	-29.53	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
4319	-29.61	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
4320	-29.63	oe	ccsbBroad304_00389	CTBP1	-			
4321	-29.65	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
4322	-29.66	cp	BRD-K01649396	indatraline	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine transporter inhibitor
4323	-29.66	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
4324	-29.69	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
4325	-29.73	kd	CGS001-168374	ZNF92	Zinc fingers, C2H2-type			
4326	-29.75	kd	CGS001-7089	TLE2	WD repeat domain containing			
4327	-29.78	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
4328	-29.82	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
4329	-29.84	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
4330	-29.89	kd	CGS001-23475	QPRT	-			
4331	-29.9	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
4332	-29.9	kd	CGS001-5306	PITPNA	-			
4333	-29.92	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
4334	-29.94	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
4335	-29.99	kd	CGS001-1209	CLPTM1	-			
4336	-30.02	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
4337	-30.08	kd	CGS001-286380	FOXD4L3	-			
4338	-30.13	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
4339	-30.15	oe	ccsbBroad304_01613	STK11	LKB subfamily			
4340	-30.16	oe	ccsbBroad304_01855	NCOA4	-			
4341	-30.16	kd	CGS001-55290	BRF2	-			
4342	-30.19	oe	ccsbBroad304_01962	STK16	NAK family			
4343	-30.22	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
4344	-30.28	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
4345	-30.3	kd	CGS001-84634	KISS1R	GPCR / Class A : RF amide peptide receptors			
4346	-30.34	kd	CGS001-256281	NUDT14	Nudix motif containing			
4347	-30.4	kd	CGS001-222894	FERD3L	Basic helix-loop-helix proteins			
4348	-30.41	oe	ccsbBroad304_02772	ICMT	-			
4349	-30.41	kd	CGS001-4700	NDUFA6	LYR motif containing			
4350	-30.42	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
4351	-30.42	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
4352	-30.42	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
4353	-30.46	oe	ccsbBroad304_01413	RPA2	-			
4354	-30.46	oe	ccsbBroad304_03266	ERGIC2	-			
4355	-30.46	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
4356	-30.46	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
4357	-30.51	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
4358	-30.53	oe	ccsbBroad304_03155	DHH	-			
4359	-30.53	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
4360	-30.55	kd	CGS001-5269	SERPINB6	Serine (or cysteine) peptidase inhibitors			
4361	-30.58	oe	ccsbBroad304_07875	SPECC1L	-			
4362	-30.59	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
4363	-30.62	oe	ccsbBroad304_03428	EXOSC4	-			
4364	-30.62	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
4365	-30.63	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
4366	-30.64	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
4367	-30.64	kd	CGS001-662	BNIP1	-			
4368	-30.65	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
4369	-30.66	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
4370	-30.67	cp	BRD-K06388322	pramipexole	Dopamine receptor agonist		DRD3, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4371	-30.68	kd	CGS001-837	CASP4	Caspases			
4372	-30.7	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
4373	-30.71	kd	CGS001-213	ALB	-			
4374	-30.72	kd	CGS001-10451	VAV3	Rho guanine nucleotide exchange factors			
4375	-30.72	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
4376	-30.72	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
4377	-30.76	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
4378	-30.76	kd	CGS001-11168	PSIP1	-			
4379	-30.77	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
4380	-30.79	kd	CGS001-51520	LARS	Aminoacyl tRNA synthetases / Class I			
4381	-30.82	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
4382	-30.82	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
4383	-30.85	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
4384	-30.86	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
4385	-30.87	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
4386	-30.9	kd	CGS001-836	CASP3	Caspases			
4387	-30.91	oe	ccsbBroad304_07569	TRIB1	Trbl family			
4388	-30.92	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
4389	-30.93	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
4390	-30.96	kd	CGS001-6599	SMARCC1	-			
4391	-30.97	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
4392	-30.98	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
4393	-30.99	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
4394	-31	oe	ccsbBroad304_02230	HERPUD1	-			
4395	-31	kd	CGS001-57048	PLSCR3	-			
4396	-31.02	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
4397	-31.02	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
4398	-31.03	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
4399	-31.03	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
4400	-31.08	oe	ccsbBroad304_13598	NRBP2	NRBP family			
4401	-31.08	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
4402	-31.08	kd	CGS001-3588	IL10RB	IL-10 receptor family			
4403	-31.09	oe	ccsbBroad304_02398	LANCL1	-			
4404	-31.11	kd	CGS001-94235	GNG8	-			
4405	-31.12	kd	CGS001-81611	ANP32E	ANP32 acidic nuclear phosphoproteins			
4406	-31.13	kd	CGS001-2232	FDXR	-			
4407	-31.16	kd	CGS001-4255	MGMT	-			
4408	-31.17	oe	ccsbBroad304_01394	RFX4	-			
4409	-31.17	kd	CGS001-6887	TAL2	Basic helix-loop-helix proteins			
4410	-31.18	oe	ccsbBroad304_01673	TIMP3	-			
4411	-31.18	kd	CGS001-439	ASNA1	-			
4412	-31.22	kd	CGS001-2781	GNAZ	-			
4413	-31.26	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
4414	-31.28	kd	CGS001-22934	RPIA	-			
4415	-31.3	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
4416	-31.31	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
4417	-31.36	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
4418	-31.36	kd	CGS001-144811	LACC1	-			
4419	-31.38	kd	CGS001-717	C2	Complement system			
4420	-31.39	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
4421	-31.44	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
4422	-31.45	oe	ccsbBroad304_02708	TRIM32	-			
4423	-31.45	kd	CGS001-25925	ZNF521	Zinc fingers, C2H2-type			
4424	-31.45	oe	ccsbBroad304_07220	CDC45	-			
4425	-31.48	cp	BRD-A88254928	salbutamol	Adrenergic receptor agonist		ADRB2, ADRB1	Adrenergic receptor agonist
4426	-31.49	kd	CGS001-6443	SGCB	-			
4427	-31.5	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
4428	-31.52	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
4429	-31.55	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
4430	-31.55	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
4431	-31.61	oe	ccsbBroad304_06349	HAGH	-			
4432	-31.61	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
4433	-31.61	kd	CGS001-6520	SLC3A2	SLC3 family			
4434	-31.61	kd	CGS001-5763	PTMS	-			
4435	-31.64	cp	BRD-K62374253	rufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4436	-31.65	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
4437	-31.71	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
4438	-31.71	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
4439	-31.71	kd	CGS001-8226	HDHD1	-			
4440	-31.72	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
4441	-31.73	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
4442	-31.74	kd	CGS001-2243	FGA	Endogenous ligands			
4443	-31.74	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4444	-31.75	kd	CGS001-4751	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4445	-31.78	kd	CGS001-8449	DHX16	DEAH-boxes			
4446	-31.81	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
4447	-31.87	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
4448	-31.91	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
4449	-31.92	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
4450	-31.92	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
4451	-31.94	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
4452	-31.95	oe	ccsbBroad304_00113	ASNS	-			
4453	-31.95	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
4454	-31.97	oe	ccsbBroad304_00532	F11	Chymotrypsin			
4455	-31.98	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
4456	-31.98	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
4457	-31.99	oe	ccsbBroad304_06420	ICAM3	CD molecules			
4458	-31.99	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
4459	-32	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
4460	-32.01	cc		PRD class homeoboxes and psudogenes LOF	-			
4461	-32.01	kd	CGS001-6732	SRPK1	SRPK family			
4462	-32.03	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
4463	-32.03	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
4464	-32.04	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
4465	-32.06	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
4466	-32.08	oe	ccsbBroad304_02526	POP4	-			
4467	-32.09	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
4468	-32.1	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
4469	-32.12	oe	ccsbBroad304_03858	SRPRB	-			
4470	-32.14	oe	ccsbBroad304_00118	ATIC	-			
4471	-32.16	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
4472	-32.17	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4473	-32.2	kd	CGS001-4245	MGAT1	-			
4474	-32.22	kd	CGS001-151742	PPM1L	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
4475	-32.25	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
4476	-32.26	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
4477	-32.27	kd	CGS001-2057	EPOR	Prolactin receptor family			
4478	-32.28	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
4479	-32.34	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
4480	-32.35	oe	ccsbBroad304_07798	EXOC3	-			
4481	-32.35	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
4482	-32.39	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
4483	-32.4	cc		NADH ubiquinone oxidoreductase supernumerary subunits LOF	-			
4484	-32.42	kd	CGS001-2760	GM2A	-			
4485	-32.45	kd	CGS001-29940	DSE	-			
4486	-32.47	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
4487	-32.47	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
4488	-32.49	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
4489	-32.5	kd	CGS001-3458	IFNG	Interferons			
4490	-32.54	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
4491	-32.57	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
4492	-32.57	kd	CGS001-634	CEACAM1	CD molecules			
4493	-32.59	kd	CGS001-102	ADAM10	ADAM metallopeptidase domain containing			
4494	-32.6	oe	ccsbBroad304_06278	GK	Glycerol kinases			
4495	-32.61	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
4496	-32.62	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
4497	-32.63	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
4498	-32.63	kd	CGS001-818	CAMK2G	CAMK2 family			
4499	-32.67	kd	CGS001-11254	SLC6A14	Glycine transporter subfamily			
4500	-32.72	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
4501	-32.77	kd	CGS001-8505	PARG	-			
4502	-32.79	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
4503	-32.82	kd	CGS001-2017	CTTN	-			
4504	-32.84	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
4505	-32.84	kd	CGS001-7296	TXNRD1	-			
4506	-32.85	cp	BRD-K16336526	capsaicin	TRPV agonist		TRPV1, CFTR, ENOX2	TRPV agonist
4507	-32.87	oe	ccsbBroad304_08660	SMARCAD1	-			
4508	-32.89	kd	CGS001-2079	ERH	-			
4509	-32.9	oe	ccsbBroad304_02047	AP1S2	-			
4510	-32.9	kd	CGS001-3799	KIF5B	Kinesins			
4511	-32.92	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
4512	-32.93	kd	CGS001-8575	PRKRA	-			
4513	-32.95	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
4514	-32.99	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
4515	-33.03	cp	BRD-A23359898	sibutramine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, CYP2B6, CYP2C19, CYP3A5	Serotonin reuptake inhibitor
4516	-33.03	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
4517	-33.08	kd	CGS001-5202	PFDN2	-			
4518	-33.1	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
4519	-33.12	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
4520	-33.13	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
4521	-33.17	oe	ccsbBroad304_00728	HBE1	-			
4522	-33.18	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
4523	-33.18	kd	CGS001-3651	PDX1	Homeoboxes / ANTP class : HOXL subclass			
4524	-33.19	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
4525	-33.19	kd	CGS001-27109	ATP5S	-			
4526	-33.2	kd	CGS001-7444	VRK2	Vaccina related kinase (VRK) family			
4527	-33.25	oe	ccsbBroad304_06494	KLRC1	CD molecules			
4528	-33.25	kd	CGS001-35	ACADS	-			
4529	-33.27	oe	ccsbBroad304_01186	PHB	-			
4530	-33.27	oe	ccsbBroad304_00472	EBF1	-			
4531	-33.28	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
4532	-33.33	oe	ccsbBroad304_01674	TIMP4	-			
4533	-33.33	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4534	-33.33	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
4535	-33.37	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
4536	-33.39	kd	CGS001-55038	CDCA4	-			
4537	-33.4	oe	ccsbBroad304_03372	CAB39	-			
4538	-33.41	kd	CGS001-2077	ERF	ETS Transcription Factors			
4539	-33.42	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
4540	-33.42	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
4541	-33.46	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
4542	-33.48	kd	CGS001-11344	TWF2	Twinfilin subfamily			
4543	-33.49	kd	CGS001-9961	MVP	-			
4544	-33.49	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
4545	-33.49	kd	CGS001-192669	EIF2C3	-			
4546	-33.5	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
4547	-33.51	kd	CGS001-5277	PIGA	Glycosyltransferase group 1 domain containing			
4548	-33.53	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
4549	-33.53	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
4550	-33.55	oe	ccsbBroad304_02372	SPRY1	-			
4551	-33.55	kd	CGS001-3685	ITGAV	Integrins			
4552	-33.56	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
4553	-33.57	oe	ccsbBroad304_05823	ANXA2	Annexins			
4554	-33.59	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
4555	-33.6	oe	ccsbBroad304_01556	SMARCB1	-			
4556	-33.6	oe	ccsbBroad304_00225	CAT	-			
4557	-33.62	kd	CGS001-2592	GALT	-			
4558	-33.62	kd	CGS001-2308	FOXO1	Forkhead boxes			
4559	-33.63	cc		Cell Cycle Inhibition GOF	-			
4560	-33.63	kd	CGS001-118442	GPR62	GPCR / Class A : Orphans			
4561	-33.69	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
4562	-33.7	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
4563	-33.71	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
4564	-33.71	kd	CGS001-9020	MAP3K14	MAPKKK:STE-unique family			
4565	-33.72	kd	CGS001-3570	IL6R	IL-6 receptor family			
4566	-33.73	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
4567	-33.75	kd	CGS001-2	A2M	-			
4568	-33.76	oe	ccsbBroad304_03089	PACSIN3	-			
4569	-33.83	kd	CGS001-6696	SPP1	Endogenous ligands			
4570	-33.84	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
4571	-33.88	kd	CGS001-114785	MBD6	-			
4572	-33.89	oe	ccsbBroad304_00359	CPT1A	-			
4573	-33.9	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
4574	-33.9	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
4575	-33.9	cp	BRD-K13800121	parecoxib	Cyclooxygenase inhibitor		LTF, PTGS2	Cyclooxygenase inhibitor
4576	-33.93	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
4577	-34.01	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
4578	-34.03	oe	ccsbBroad304_03625	HIF1AN	-			
4579	-34.04	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
4580	-34.05	oe	ccsbBroad304_00960	SMAD1	SMADs			
4581	-34.08	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
4582	-34.08	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
4583	-34.08	oe	ccsbBroad304_00931	LCN2	Lipocalins			
4584	-34.09	oe	ccsbBroad304_04471	C5ORF62	-			
4585	-34.09	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
4586	-34.11	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
4587	-34.17	kd	CGS001-1120	CHKB	-			
4588	-34.18	oe	ccsbBroad304_13952	SHMT2	-			
4589	-34.21	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
4590	-34.22	oe	ccsbBroad304_07140	XPC	-			
4591	-34.23	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
4592	-34.25	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
4593	-34.25	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
4594	-34.25	kd	CGS001-4791	NFKB2	NFkappaB transcription factor family			
4595	-34.26	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
4596	-34.27	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
4597	-34.27	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
4598	-34.28	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
4599	-34.28	kd	CGS001-3486	IGFBP3	insulin-like growth factor (IGF) binding proteins			
4600	-34.29	oe	ccsbBroad304_00874	INS	-			
4601	-34.29	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
4602	-34.29	kd	CGS001-664	BNIP3	-			
4603	-34.31	oe	ccsbBroad304_07884	RYBP	-			
4604	-34.33	kd	CGS001-22949	PTGR1	-			
4605	-34.34	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
4606	-34.35	kd	CGS001-3269	HRH1	Histamine receptors			
4607	-34.37	kd	CGS001-64863	METTL4	-			
4608	-34.39	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
4609	-34.45	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
4610	-34.47	kd	CGS001-7039	TGFA	-			
4611	-34.48	kd	CGS001-1604	CD55	CD molecules			
4612	-34.49	kd	CGS001-5695	PSMB7	Proteasome subunits			
4613	-34.49	kd	CGS001-3119	HLA-DQB1	Immunoglobulin superfamily / C1-set domain containing			
4614	-34.5	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
4615	-34.5	kd	CGS001-4097	MAFG	-			
4616	-34.51	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
4617	-34.54	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
4618	-34.54	kd	CGS001-22	ABCB7	ATP binding cassette transporters / subfamily B			
4619	-34.56	cp	BRD-K92870997	pterostilbene	Cyclooxygenase inhibitor		FAAH, PPARA, PTGS1, PTGS2	Cyclooxygenase inhibitor, PPAR receptor agonist
4620	-34.57	kd	CGS001-840	CASP7	Caspases			
4621	-34.6	oe	ccsbBroad304_03812	PBXIP1	-			
4622	-34.6	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
4623	-34.62	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
4624	-34.63	kd	CGS001-4351	MPI	-			
4625	-34.64	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
4626	-34.65	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
4627	-34.66	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
4628	-34.67	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
4629	-34.67	kd	CGS001-11157	LSM6	-			
4630	-34.71	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
4631	-34.71	kd	CGS001-23030	KDM4B	Histone demethylases			
4632	-34.75	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
4633	-34.76	oe	ccsbBroad304_08093	DCPS	-			
4634	-34.76	kd	CGS001-8803	SUCLA2	-			
4635	-34.78	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
4636	-34.79	kd	CGS001-4121	MAN1A1	-			
4637	-34.85	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
4638	-34.85	kd	CGS001-9650	MTFR1	-			
4639	-34.86	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
4640	-34.86	kd	CGS001-8477	GPR65	GPCR / Class A : Orphans			
4641	-34.88	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
4642	-34.91	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
4643	-34.92	kd	CGS001-64087	MCCC2	-			
4644	-34.93	oe	ccsbBroad304_08392	EXOC6	-			
4645	-34.94	oe	ccsbBroad304_00490	EIF4EBP1	-			
4646	-34.97	kd	CGS001-6857	SYT1	Synaptotagmins			
4647	-35.01	oe	ccsbBroad304_07277	RTCD1	-			
4648	-35.02	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
4649	-35.03	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
4650	-35.04	kd	CGS001-23365	ARHGEF12	Rho guanine nucleotide exchange factors			
4651	-35.06	kd	CGS001-3516	RBPJ	-			
4652	-35.07	kd	CGS001-5451	POU2F1	Homeoboxes / POU class			
4653	-35.17	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
4654	-35.19	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
4655	-35.23	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
4656	-35.24	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
4657	-35.24	kd	CGS001-5515	PPP2CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4658	-35.26	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
4659	-35.27	kd	CGS001-55723	ASF1B	-			
4660	-35.27	oe	ccsbBroad304_07768	NISCH	-			
4661	-35.28	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
4662	-35.3	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
4663	-35.32	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
4664	-35.32	kd	CGS001-7056	THBD	CD molecules			
4665	-35.33	kd	CGS001-2098	ESD	-			
4666	-35.38	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
4667	-35.39	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4668	-35.39	oe	ccsbBroad304_01841	BAG6	-			
4669	-35.4	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
4670	-35.41	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
4671	-35.41	kd	CGS001-7919	DDX39B	DEAD-boxes			
4672	-35.47	oe	ccsbBroad304_00464	DTNA	-			
4673	-35.48	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
4674	-35.52	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4675	-35.55	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
4676	-35.56	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
4677	-35.62	kd	CGS001-10010	TANK	-			
4678	-35.63	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
4679	-35.64	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
4680	-35.64	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
4681	-35.64	kd	CGS001-9374	PPT2	-			
4682	-35.65	kd	CGS001-2744	GLS	Ankyrin repeat domain containing			
4683	-35.69	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
4684	-35.71	kd	CGS001-166793	ZBTB49	BTB/POZ domain containing			
4685	-35.73	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
4686	-35.73	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
4687	-35.74	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
4688	-35.8	kd	CGS001-7471	WNT1	Endogenous ligands			
4689	-35.81	kd	CGS001-27125	AFF4	-			
4690	-35.82	kd	CGS001-6499	SKIV2L	-			
4691	-35.83	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
4692	-35.86	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
4693	-35.86	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
4694	-35.86	kd	CGS001-3553	IL1B	Interleukins and interleukin receptors			
4695	-35.87	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
4696	-35.9	kd	CGS001-6421	SFPQ	RNA binding motif (RRM) containing			
4697	-35.9	kd	CGS001-56139	PCDHA10	Cadherins / Protocadherins : Clustered			
4698	-35.9	kd	CGS001-644	BLVRA	-			
4699	-35.91	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
4700	-35.95	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
4701	-35.96	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
4702	-35.96	kd	CGS001-5054	SERPINE1	Serine (or cysteine) peptidase inhibitors			
4703	-35.97	kd	CGS001-1389	CREBL2	basic leucine zipper proteins			
4704	-36	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
4705	-36.01	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
4706	-36.01	oe	ccsbBroad304_03506	AURKAIP1	-			
4707	-36.03	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
4708	-36.03	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
4709	-36.08	oe	ccsbBroad304_00120	ATOX1	-			
4710	-36.14	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
4711	-36.14	kd	CGS001-57616	TSHZ3	Teashirt zinc fingers			
4712	-36.14	kd	CGS001-11336	EXOC3	-			
4713	-36.15	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
4714	-36.16	kd	CGS001-3420	IDH3B	-			
4715	-36.19	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
4716	-36.21	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
4717	-36.24	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
4718	-36.27	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
4719	-36.28	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
4720	-36.36	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
4721	-36.36	kd	CGS001-9887	SMG7	-			
4722	-36.39	kd	CGS001-2697	GJA1	Ion channels / Gap junction proteins (connexins)			
4723	-36.4	oe	ccsbBroad304_06993	SRD5A1	-			
4724	-36.4	kd	CGS001-3203	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
4725	-36.42	kd	CGS001-63874	ABHD4	Abhydrolase domain containing			
4726	-36.43	oe	ccsbBroad304_08104	MED4	-			
4727	-36.45	oe	ccsbBroad304_03122	RHOD	-			
4728	-36.46	kd	CGS001-2015	EMR1	Adhesion Class GPCRs			
4729	-36.47	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
4730	-36.48	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
4731	-36.48	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
4732	-36.48	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
4733	-36.51	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
4734	-36.56	kd	CGS001-55054	ATG16L1	WD repeat domain containing			
4735	-36.63	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
4736	-36.63	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
4737	-36.65	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
4738	-36.65	kd	CGS001-8220	DGCR14	-			
4739	-36.68	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
4740	-36.7	cc		Lysine acetyltransferases LOF	-			
4741	-36.78	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
4742	-36.79	kd	CGS001-7431	VIM	Intermediate filaments type III			
4743	-36.8	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
4744	-36.8	kd	CGS001-5442	POLRMT	-			
4745	-36.87	kd	CGS001-10285	SMNDC1	Tudor domain containing			
4746	-36.91	kd	CGS001-10245	TIMM17B	-			
4747	-36.91	kd	CGS001-9158	FIBP	-			
4748	-36.92	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
4749	-36.95	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
4750	-37	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
4751	-37	kd	CGS001-2863	GPR39	GPCR / Class A : Orphans			
4752	-37.01	oe	ccsbBroad304_02313	ACTR3	-			
4753	-37.01	oe	ccsbBroad304_02922	TES	-			
4754	-37.04	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
4755	-37.06	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
4756	-37.07	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4757	-37.09	kd	CGS001-330	BIRC3	Inhibitors of apoptosis (IAP) protein family			
4758	-37.12	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
4759	-37.14	oe	ccsbBroad304_02484	PAICS	-			
4760	-37.15	cc		Trace amine receptors LOF	-			
4761	-37.15	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
4762	-37.15	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
4763	-37.2	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
4764	-37.25	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
4765	-37.25	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
4766	-37.3	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
4767	-37.3	kd	CGS001-4594	MUT	-			
4768	-37.31	cc		HDAC inhibitor	-			
4769	-37.31	oe	ccsbBroad304_06103	DMD	-			
4770	-37.32	kd	CGS001-6622	SNCA	Parkinson disease			
4771	-37.35	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
4772	-37.36	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
4773	-37.37	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
4774	-37.38	kd	CGS001-1962	EHHADH	-			
4775	-37.41	kd	CGS001-117581	TWIST2	Basic helix-loop-helix proteins			
4776	-37.41	kd	CGS001-5105	PCK1	-			
4777	-37.42	kd	CGS001-6271	S100A1	EF-hand domain containing			
4778	-37.43	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
4779	-37.43	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
4780	-37.43	kd	CGS001-10097	ACTR2	-			
4781	-37.44	kd	CGS001-10018	BCL2L11	-			
4782	-37.46	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
4783	-37.47	kd	CGS001-4798	NFRKB	INO80 complex subunits			
4784	-37.51	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
4785	-37.51	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
4786	-37.51	oe	ccsbBroad304_06386	HNMT	-			
4787	-37.58	oe	ccsbBroad304_00150	BAX	-			
4788	-37.58	kd	CGS001-83440	ADPGK	-			
4789	-37.6	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
4790	-37.63	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
4791	-37.65	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
4792	-37.66	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
4793	-37.68	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
4794	-37.72	kd	CGS001-10237	SLC35B1	SLC35 family of nucleotide sugar transporters			
4795	-37.81	oe	ccsbBroad304_07012	STK3	MST subfamily			
4796	-37.81	kd	CGS001-10287	RGS19	Regulators of G-protein signaling			
4797	-37.83	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
4798	-37.84	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
4799	-37.86	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
4800	-37.88	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
4801	-37.91	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
4802	-37.97	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4803	-37.97	kd	CGS001-23753	SDF2L1	-			
4804	-37.98	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
4805	-37.98	kd	CGS001-11019	LIAS	-			
4806	-38.01	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
4807	-38.01	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4808	-38.02	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
4809	-38.03	oe	ccsbBroad304_03533	CDCA8	-			
4810	-38.03	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
4811	-38.04	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
4812	-38.04	kd	CGS001-84759	PCGF1	Polycomb group ring fingers			
4813	-38.07	kd	CGS001-121599	SPIC	ETS Transcription Factors			
4814	-38.09	kd	CGS001-9867	PJA2	RING-type (C3HC4) zinc fingers			
4815	-38.09	kd	CGS001-8639	AOC3	Oxidoreductases			
4816	-38.1	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
4817	-38.14	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
4818	-38.16	kd	CGS001-84775	ZNF607	Zinc fingers, C2H2-type			
4819	-38.17	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
4820	-38.17	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4821	-38.17	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4822	-38.19	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
4823	-38.2	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
4824	-38.2	kd	CGS001-84878	ZBTB45	BTB/POZ domain containing			
4825	-38.24	oe	ccsbBroad304_00620	GCDH	-			
4826	-38.26	oe	ccsbBroad304_06225	FTH1	-			
4827	-38.27	kd	CGS001-2990	GUSB	-			
4828	-38.29	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
4829	-38.3	kd	CGS001-57026	PDXP	-			
4830	-38.31	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
4831	-38.31	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
4832	-38.36	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
4833	-38.4	kd	CGS001-29978	UBQLN2	Ubiquilin family			
4834	-38.43	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
4835	-38.45	oe	ccsbBroad304_02502	GNA13	-			
4836	-38.45	kd	CGS001-1606	DGKA	EF-hand domain containing			
4837	-38.47	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
4838	-38.48	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
4839	-38.49	kd	CGS001-6647	SOD1	-			
4840	-38.52	oe	ccsbBroad304_02133	CD83	CD molecules			
4841	-38.54	kd	CGS001-4016	LOXL1	-			
4842	-38.58	kd	CGS001-24148	PRPF6	-			
4843	-38.59	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4844	-38.63	oe	ccsbBroad304_07923	LSM5	-			
4845	-38.63	kd	CGS001-1460	CSNK2B	Casein kinase 2 (CK2) family			
4846	-38.63	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
4847	-38.65	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
4848	-38.66	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
4849	-38.71	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
4850	-38.73	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
4851	-38.73	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
4852	-38.75	oe	ccsbBroad304_02485	STAMBP	-			
4853	-38.75	kd	CGS001-29105	C16ORF80	-			
4854	-38.76	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
4855	-38.77	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
4856	-38.8	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
4857	-38.9	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
4858	-38.9	kd	CGS001-54490	UGT2B28	UDP glucuronosyltransferases			
4859	-38.94	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
4860	-38.94	oe	ccsbBroad304_03186	GMNN	-			
4861	-39.03	kd	CGS001-335	APOA1	Apolipoproteins			
4862	-39.04	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
4863	-39.04	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
4864	-39.06	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
4865	-39.07	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
4866	-39.08	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
4867	-39.09	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4868	-39.09	kd	CGS001-2618	GART	Ribosyl transferases			
4869	-39.12	kd	CGS001-22908	SACM1L	-			
4870	-39.13	kd	CGS001-5338	PLD2	Hydrolases			
4871	-39.14	kd	CGS001-55324	ABCF3	ATP binding cassette transporters / subfamily F			
4872	-39.15	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
4873	-39.15	kd	CGS001-5336	PLCG2	Phosphoinositide-specific phospholipase C			
4874	-39.17	kd	CGS001-8650	NUMB	-			
4875	-39.18	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4876	-39.18	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4877	-39.19	kd	CGS001-7187	TRAF3	-			
4878	-39.2	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
4879	-39.22	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
4880	-39.28	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
4881	-39.29	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
4882	-39.32	oe	ccsbBroad304_06683	FURIN	Subtilisin			
4883	-39.34	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
4884	-39.37	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
4885	-39.4	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
4886	-39.4	kd	CGS001-80777	CYB5B	-			
4887	-39.46	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
4888	-39.49	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
4889	-39.61	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
4890	-39.66	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
4891	-39.68	kd	CGS001-2568	GABRP	GABA receptors			
4892	-39.71	kd	CGS001-10161	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
4893	-39.72	kd	CGS001-2181	ACSL3	Acyl-CoA synthetase family			
4894	-39.74	oe	ccsbBroad304_02175	MAGED1	-			
4895	-39.74	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
4896	-39.75	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
4897	-39.77	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
4898	-39.78	oe	ccsbBroad304_01374	RAP1A	-			
4899	-39.78	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
4900	-39.86	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
4901	-39.9	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
4902	-39.91	cp	BRD-K96471533	nitazoxanide	Pyruvate ferredoxin oxidoreductase inhibitor			Pyruvate ferredoxin oxidoreductase inhibitor
4903	-39.91	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
4904	-39.95	kd	CGS001-55876	GSDMB	-			
4905	-40.04	cc		V type ATPases LOF	-			
4906	-40.05	kd	CGS001-2710	GK	Glycerol kinases			
4907	-40.06	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
4908	-40.08	kd	CGS001-284119	PTRF	-			
4909	-40.09	cp	BRD-K22947005	dexbrompheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4910	-40.1	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
4911	-40.11	kd	CGS001-3998	LMAN1	-			
4912	-40.13	cc		Proteasome Pathway LOF	-			
4913	-40.13	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
4914	-40.14	oe	ccsbBroad304_06066	CTSL1	-			
4915	-40.15	kd	CGS001-7511	XPNPEP1	Methionyl aminopeptidase			
4916	-40.16	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
4917	-40.18	kd	CGS001-5164	PDK2	PDHK family			
4918	-40.21	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
4919	-40.23	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
4920	-40.24	cp	BRD-K22227508	targinine	Nitric oxide synthase inhibitor		NOS2, NOS3	Nitric oxide synthase inhibitor
4921	-40.25	oe	ccsbBroad304_07466	VGLL4	-			
4922	-40.25	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
4923	-40.3	kd	CGS001-130497	OSR1	Zinc fingers, C2H2-type			
4924	-40.3	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
4925	-40.32	kd	CGS001-117154	DACH2	-			
4926	-40.37	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
4927	-40.38	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
4928	-40.39	kd	CGS001-8334	HIST1H2AC	Histones / Replication-dependent			
4929	-40.4	oe	ccsbBroad304_00006	ACADM	-			
4930	-40.43	kd	CGS001-476	ATP1A1	ATPases / P-type			
4931	-40.47	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4932	-40.48	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
4933	-40.49	kd	CGS001-6775	STAT4	SH2 domain containing			
4934	-40.5	kd	CGS001-5743	PTGS2	Cyclooxygenase			
4935	-40.52	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
4936	-40.54	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
4937	-40.54	kd	CGS001-843	CASP10	Caspases			
4938	-40.58	cp	BRD-K04710043	hexamethylenebisacetamide	AKT inhibitor			AKT inhibitor, Differentiation inducer, NFkB pathway inhibitor
4939	-40.61	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
4940	-40.62	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
4941	-40.65	oe	ccsbBroad304_01102	NMT1	-			
4942	-40.66	oe	ccsbBroad304_00518	ETFA	-			
4943	-40.66	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
4944	-40.66	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
4945	-40.69	kd	CGS001-25793	FBXO7	F-boxes / other			
4946	-40.72	kd	CGS001-140465	MYL6B	EF-hand domain containing			
4947	-40.73	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
4948	-40.76	oe	ccsbBroad304_06464	ITGB2	Integrins			
4949	-40.78	kd	CGS001-9341	VAMP3	Vesicle-associated membrane proteins			
4950	-40.79	oe	ccsbBroad304_03570	QRSL1	-			
4951	-40.81	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
4952	-40.82	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4953	-40.87	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
4954	-40.87	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
4955	-40.91	kd	CGS001-6418	SET	-			
4956	-40.93	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
4957	-40.93	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
4958	-40.97	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
4959	-40.98	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
4960	-41	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
4961	-41.02	oe	ccsbBroad304_05980	CDKN1B	-			
4962	-41.07	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
4963	-41.11	kd	CGS001-7468	WHSC1	Zinc fingers, PHD-type			
4964	-41.12	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
4965	-41.2	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
4966	-41.22	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
4967	-41.25	cp	BRD-K60160658	tiagabine	GABA uptake inhibitor		SLC6A1, CYP2C19	GABA uptake inhibitor
4968	-41.26	kd	CGS001-57157	PHTF2	-			
4969	-41.27	kd	CGS001-663	BNIP2	-			
4970	-41.28	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
4971	-41.33	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4972	-41.34	cc		GPCR Subset GOF	-			
4973	-41.36	kd	CGS001-60528	ELAC2	-			
4974	-41.39	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
4975	-41.41	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
4976	-41.45	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
4977	-41.46	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
4978	-41.46	kd	CGS001-54499	TMCO1	-			
4979	-41.47	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
4980	-41.47	kd	CGS001-201799	TMEM154	-			
4981	-41.47	kd	CGS001-27148	STK36	Unc-51-like kinase (ULK) family			
4982	-41.52	oe	ccsbBroad304_06174	ERCC1	-			
4983	-41.53	oe	ccsbBroad304_01180	PFKFB3	-			
4984	-41.53	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
4985	-41.61	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
4986	-41.62	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
4987	-41.62	kd	CGS001-406	ARNTL	Basic helix-loop-helix proteins			
4988	-41.64	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
4989	-41.65	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4990	-41.65	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
4991	-41.67	kd	CGS001-29946	SERTAD3	-			
4992	-41.68	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
4993	-41.69	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
4994	-41.71	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
4995	-41.73	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
4996	-41.74	kd	CGS001-5193	PEX12	-			
4997	-41.74	kd	CGS001-8714	ABCC3	ATP binding cassette transporters / subfamily C			
4998	-41.75	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
4999	-41.79	kd	CGS001-1756	DMD	-			
5000	-41.8	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
5001	-41.85	kd	CGS001-382	ARF6	ADP-ribosylation factors			
5002	-41.88	oe	ccsbBroad304_01532	SIAH1	-			
5003	-41.91	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
5004	-41.91	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
5005	-41.95	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
5006	-41.95	oe	ccsbBroad304_08055	ATP5S	-			
5007	-41.95	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
5008	-42.01	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
5009	-42.01	oe	ccsbBroad304_01392	TRIM27	-			
5010	-42.03	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
5011	-42.03	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5012	-42.04	kd	CGS001-650	BMP2	Bone morphogenetic proteins			
5013	-42.08	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
5014	-42.09	kd	CGS001-1305	COL13A1	Collagens			
5015	-42.15	oe	ccsbBroad304_13998	PDXK	-			
5016	-42.18	oe	ccsbBroad304_02143	CNOT8	-			
5017	-42.18	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
5018	-42.21	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
5019	-42.22	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
5020	-42.23	kd	CGS001-2287	FKBP3	-			
5021	-42.25	cp	BRD-K88679075	methandriol	Androgenic steroid			Androgenic steroid
5022	-42.27	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
5023	-42.28	oe	ccsbBroad304_03696	C19ORF10	-			
5024	-42.3	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
5025	-42.31	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
5026	-42.33	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
5027	-42.34	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
5028	-42.36	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
5029	-42.36	kd	CGS001-8900	CCNA1	-			
5030	-42.39	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
5031	-42.39	kd	CGS001-5962	RDX	-			
5032	-42.41	kd	CGS001-4790	NFKB1	NFkappaB transcription factor family			
5033	-42.44	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
5034	-42.45	oe	ccsbBroad304_01013	MIF	-			
5035	-42.47	oe	ccsbBroad304_00462	DR1	-			
5036	-42.51	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
5037	-42.53	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
5038	-42.56	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
5039	-42.57	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
5040	-42.59	kd	CGS001-7866	IFRD2	-			
5041	-42.6	oe	ccsbBroad304_00709	GUK1	-			
5042	-42.6	kd	CGS001-5293	PIK3CD	Phosphatidylinositol kinases			
5043	-42.7	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
5044	-42.72	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
5045	-42.73	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
5046	-42.73	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
5047	-42.76	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
5048	-42.78	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
5049	-42.8	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
5050	-42.84	kd	CGS001-185	AGTR1	Angiotensin receptors			
5051	-42.86	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
5052	-42.91	kd	CGS001-84365	MKI67IP	-			
5053	-42.93	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
5054	-42.96	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5055	-42.96	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
5056	-42.96	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
5057	-43.01	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
5058	-43.02	kd	CGS001-66008	TRAK2	-			
5059	-43.03	kd	CGS001-2967	GTF2H3	General transcription factors			
5060	-43.05	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
5061	-43.06	kd	CGS001-151306	GPBAR1	Bile acid receptor			
5062	-43.11	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
5063	-43.12	oe	ccsbBroad304_07197	PDHX	-			
5064	-43.14	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
5065	-43.18	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
5066	-43.19	kd	CGS001-10398	MYL9	EF-hand domain containing			
5067	-43.21	kd	CGS001-85004	RERG	-			
5068	-43.23	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
5069	-43.25	oe	ccsbBroad304_07887	GCAT	-			
5070	-43.26	kd	CGS001-51027	BOLA1	-			
5071	-43.27	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
5072	-43.29	kd	CGS001-1645	AKR1C1	Aldo-keto reductases			
5073	-43.34	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
5074	-43.43	oe	ccsbBroad304_01164	PDHB	-			
5075	-43.44	kd	CGS001-1030	CDKN2B	-			
5076	-43.45	cc		SRC inhibitor	-			
5077	-43.47	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
5078	-43.47	oe	ccsbBroad304_02017	PEX11A	-			
5079	-43.51	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
5080	-43.51	kd	CGS001-5777	PTPN6	Protein tyrosine phosphatases			
5081	-43.52	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
5082	-43.53	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
5083	-43.53	kd	CGS001-4522	MTHFD1	-			
5084	-43.54	oe	ccsbBroad304_03118	NRBP1	NRBP family			
5085	-43.56	kd	CGS001-10390	CEPT1	-			
5086	-43.6	oe	ccsbBroad304_06695	PCK2	-			
5087	-43.63	kd	CGS001-4292	MLH1	-			
5088	-43.65	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
5089	-43.65	kd	CGS001-5645	PRSS2	Serine peptidases			
5090	-43.7	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
5091	-43.7	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
5092	-43.74	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5093	-43.75	kd	CGS001-5004	ORM1	Lipocalins			
5094	-43.75	kd	CGS001-55379	LRRC59	-			
5095	-43.76	kd	CGS001-1284	COL4A2	Collagens			
5096	-43.8	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
5097	-43.83	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
5098	-43.83	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
5099	-43.86	kd	CGS001-3149	HMGB3	High-mobility group / Canonical			
5100	-43.92	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
5101	-43.92	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
5102	-43.92	kd	CGS001-286530	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
5103	-43.93	kd	CGS001-55129	ANO10	Calcium activated chloride channel			
5104	-43.95	oe	ccsbBroad304_01930	CUL2	-			
5105	-43.95	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
5106	-43.95	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
5107	-43.99	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
5108	-44.01	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
5109	-44.03	cp	BRD-K84955386	hyperoside	Glucosidase inhibitor		ACE, AKR1B1, GAA	Glucosidase inhibitor
5110	-44.03	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
5111	-44.04	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
5112	-44.05	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
5113	-44.05	kd	CGS001-5887	RAD23B	-			
5114	-44.06	kd	CGS001-54472	TOLLIP	-			
5115	-44.11	kd	CGS001-10423	CDIPT	-			
5116	-44.13	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
5117	-44.15	kd	CGS001-5422	POLA1	DNA polymerases			
5118	-44.19	kd	CGS001-5049	PAFAH1B2	-			
5119	-44.2	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
5120	-44.22	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
5121	-44.22	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
5122	-44.24	cp	BRD-K39391626	ethylestrenol	Progesterone receptor agonist		AR	Progesterone receptor agonist
5123	-44.27	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
5124	-44.28	oe	ccsbBroad304_02857	BAMBI	-			
5125	-44.29	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
5126	-44.32	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
5127	-44.33	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
5128	-44.36	cp	BRD-K18895904	olanzapine	Dopamine receptor antagonist		DRD2, HTR2A, HTR2C, DRD1, DRD3, DRD4, HRH1, HTR1A, HTR1B, HTR1D, HTR1E, HTR6, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C8, DRD5, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH2, HRH4, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
5129	-44.39	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
5130	-44.42	oe	ccsbBroad304_02834	GABARAPL1	-			
5131	-44.44	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
5132	-44.44	kd	CGS001-5209	PFKFB3	-			
5133	-44.46	kd	CGS001-23581	CASP14	Caspases			
5134	-44.47	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
5135	-44.51	oe	ccsbBroad304_07287	HYAL2	-			
5136	-44.52	kd	CGS001-949	SCARB1	-			
5137	-44.56	kd	CGS001-6678	SPARC	-			
5138	-44.58	oe	ccsbBroad304_06523	LIG1	-			
5139	-44.58	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
5140	-44.58	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
5141	-44.58	kd	CGS001-3575	IL7R	IL-2 receptor family			
5142	-44.59	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
5143	-44.6	kd	CGS001-11044	PAPD7	-			
5144	-44.63	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
5145	-44.66	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
5146	-44.67	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
5147	-44.68	oe	ccsbBroad304_01271	PPT1	-			
5148	-44.7	kd	CGS001-9122	SLC16A4	SLC16 family of monocarboxylate transporters			
5149	-44.75	kd	CGS001-148103	ZNF599	Zinc fingers, C2H2-type			
5150	-44.77	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
5151	-44.85	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
5152	-44.88	kd	CGS001-2634	GBP2	-			
5153	-44.89	oe	ccsbBroad304_07814	SACM1L	-			
5154	-44.89	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
5155	-44.96	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
5156	-44.96	kd	CGS001-6601	SMARCC2	-			
5157	-44.96	kd	CGS001-211	ALAS1	-			
5158	-44.97	oe	ccsbBroad304_00164	BLMH	-			
5159	-44.99	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
5160	-45	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
5161	-45	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
5162	-45	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
5163	-45.01	kd	CGS001-338557	O3FAR1	-			
5164	-45.02	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
5165	-45.02	kd	CGS001-1831	TSC22D3	-			
5166	-45.04	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5167	-45.06	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
5168	-45.13	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
5169	-45.16	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
5170	-45.16	kd	CGS001-3665	IRF7	-			
5171	-45.16	kd	CGS001-133690	CAPSL	EF-hand domain containing			
5172	-45.17	cc		TGF beta receptor inhibitor	-			
5173	-45.2	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
5174	-45.21	kd	CGS001-7247	TSN	-			
5175	-45.21	kd	CGS001-4638	MYLK	Myosin Light Chain Kinase (MLCK) family			
5176	-45.28	cc		Angiotensin receptor antagonist	-			
5177	-45.29	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
5178	-45.29	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
5179	-45.31	kd	CGS001-3171	FOXA3	Forkhead boxes			
5180	-45.33	kd	CGS001-9791	PTDSS1	-			
5181	-45.36	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
5182	-45.39	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
5183	-45.42	kd	CGS001-9813	KIAA0494	-			
5184	-45.42	kd	CGS001-6723	SRM	-			
5185	-45.43	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
5186	-45.47	kd	CGS001-54884	RETSAT	-			
5187	-45.55	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
5188	-45.56	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
5189	-45.56	kd	CGS001-9111	NMI	-			
5190	-45.57	kd	CGS001-65243	ZNF643	-			
5191	-45.58	oe	ccsbBroad304_05763	ACTB	-			
5192	-45.59	kd	CGS001-3586	IL10	Interleukins and interleukin receptors			
5193	-45.59	kd	CGS001-3339	HSPG2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5194	-45.6	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
5195	-45.61	cc		KCNJ11 modulator	-			
5196	-45.63	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
5197	-45.64	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
5198	-45.66	kd	CGS001-3692	EIF6	-			
5199	-45.67	oe	ccsbBroad304_07889	QPRT	-			
5200	-45.67	kd	CGS001-8667	EIF3H	-			
5201	-45.68	kd	CGS001-4931	NVL	ATPases / AAA-type			
5202	-45.68	kd	CGS001-9643	MORF4L2	-			
5203	-45.69	oe	ccsbBroad304_02553	BLCAP	-			
5204	-45.75	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
5205	-45.79	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
5206	-45.82	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
5207	-45.87	kd	CGS001-1843	DUSP1	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
5208	-45.89	kd	CGS001-9180	OSMR	IL-6 receptor family			
5209	-45.9	kd	CGS001-2828	GPR4	GPCR / Class A : Orphans			
5210	-45.91	kd	CGS001-55872	PBK	TOPK family			
5211	-45.92	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
5212	-45.93	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
5213	-45.98	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5214	-45.98	kd	CGS001-7421	VDR	Vitamin D receptors			
5215	-45.98	kd	CGS001-2593	GAMT	-			
5216	-45.99	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
5217	-45.99	kd	CGS001-51172	NAGPA	-			
5218	-46.01	cp	BRD-K15842202	eudesmic-acid	-666			-666
5219	-46.01	kd	CGS001-161725	OTUD7A	OTU domain containing			
5220	-46.03	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
5221	-46.06	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
5222	-46.08	oe	ccsbBroad304_06845	RARRES3	-			
5223	-46.1	kd	CGS001-22796	COG2	Components of oligomeric golgi complex			
5224	-46.12	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
5225	-46.17	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
5226	-46.17	kd	CGS001-23650	TRIM29	-			
5227	-46.19	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
5228	-46.19	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
5229	-46.2	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
5230	-46.2	cp	BRD-K10065684	dantron	Laxative			Laxative
5231	-46.2	kd	CGS001-51588	PIAS4	Zinc fingers, MIZ-type			
5232	-46.21	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
5233	-46.22	oe	ccsbBroad304_06975	SMARCC2	-			
5234	-46.24	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
5235	-46.24	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
5236	-46.28	kd	CGS001-6514	SLC2A2	Solute carriers			
5237	-46.31	oe	ccsbBroad304_01205	PIN1	-			
5238	-46.36	kd	CGS001-8986	RPS6KA4	MSK subfamily			
5239	-46.43	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
5240	-46.45	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5241	-46.48	kd	CGS001-4711	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
5242	-46.49	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
5243	-46.5	kd	CGS001-25824	PRDX5	-			
5244	-46.51	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
5245	-46.54	oe	ccsbBroad304_00100	RHOA	-			
5246	-46.54	kd	CGS001-11164	NUDT5	Nudix motif containing			
5247	-46.55	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
5248	-46.55	cp	BRD-A70083328	secnidazole	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Microtubule inhibitor, Antiprotozoal
5249	-46.56	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
5250	-46.6	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
5251	-46.6	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
5252	-46.62	oe	ccsbBroad304_02822	ARFIP2	-			
5253	-46.66	oe	ccsbBroad304_01618	STXBP1	-			
5254	-46.67	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5255	-46.74	oe	ccsbBroad304_00231	CBFB	-			
5256	-46.75	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
5257	-46.75	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5258	-46.8	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
5259	-46.82	kd	CGS001-1978	EIF4EBP1	-			
5260	-46.87	oe	ccsbBroad304_06350	HAL	-			
5261	-46.87	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
5262	-46.87	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
5263	-46.88	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
5264	-46.89	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
5265	-46.9	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
5266	-46.9	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
5267	-46.93	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
5268	-46.94	cp	BRD-K65910366	KUC103904N	-666			-666
5269	-46.95	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
5270	-46.97	kd	CGS001-4190	MDH1	-			
5271	-46.98	kd	CGS001-27297	CRCP	-			
5272	-47.03	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
5273	-47.03	kd	CGS001-9787	DLGAP5	-			
5274	-47.06	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
5275	-47.06	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
5276	-47.08	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5277	-47.11	kd	CGS001-6188	RPS3	S ribosomal proteins			
5278	-47.13	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
5279	-47.15	kd	CGS001-290	ANPEP	Aminopeptidase N			
5280	-47.18	oe	ccsbBroad304_03191	NOSIP	-			
5281	-47.2	cp	BRD-K96134740	kitasamycin	Protein synthesis inhibitor			Protein synthesis inhibitor
5282	-47.21	kd	CGS001-7728	ZNF175	Zinc fingers, C2H2-type			
5283	-47.22	kd	CGS001-23014	FBXO21	F-boxes / other			
5284	-47.25	kd	CGS001-5432	POLR2C	RNA polymerase subunits			
5285	-47.26	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
5286	-47.27	kd	CGS001-5881	RAC3	Endogenous ligands			
5287	-47.28	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
5288	-47.29	oe	ccsbBroad304_04379	LZIC	-			
5289	-47.31	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
5290	-47.38	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
5291	-47.39	kd	CGS001-598	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5292	-47.45	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
5293	-47.54	oe	ccsbBroad304_02458	STK25	YSK subfamily			
5294	-47.54	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
5295	-47.55	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
5296	-47.55	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
5297	-47.55	kd	CGS001-8872	CDC123	-			
5298	-47.56	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
5299	-47.58	oe	ccsbBroad304_01131	OXCT1	-			
5300	-47.6	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
5301	-47.61	oe	ccsbBroad304_00510	EPHX2	-			
5302	-47.69	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
5303	-47.73	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
5304	-47.74	oe	ccsbBroad304_08775	SQRDL	-			
5305	-47.74	kd	CGS001-5562	PRKAA1	AMPK subfamily			
5306	-47.75	kd	CGS001-1736	DKC1	-			
5307	-47.76	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
5308	-47.77	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
5309	-47.79	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
5310	-47.8	kd	CGS001-134187	POU5F2	Homeoboxes / POU class			
5311	-47.81	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
5312	-47.82	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5313	-47.82	kd	CGS001-6720	SREBF1	Basic helix-loop-helix proteins			
5314	-47.85	kd	CGS001-112812	FDX1L	-			
5315	-47.87	oe	ccsbBroad304_03308	YTHDF2	-			
5316	-47.87	kd	CGS001-28964	GIT1	Ankyrin repeat domain containing			
5317	-47.92	kd	CGS001-57326	PBXIP1	-			
5318	-47.95	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
5319	-47.95	kd	CGS001-9231	DLG5	-			
5320	-47.96	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
5321	-47.99	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
5322	-48.01	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
5323	-48.01	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
5324	-48.04	cc		Baculoviral IAP repeat domain containing LOF	-			
5325	-48.04	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
5326	-48.05	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
5327	-48.06	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
5328	-48.06	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
5329	-48.09	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5330	-48.1	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
5331	-48.14	kd	CGS001-4811	NID1	-			
5332	-48.15	kd	CGS001-9404	LPXN	-			
5333	-48.18	cp	BRD-K88304388	dextrorphan	Glutamate receptor antagonist		OPRM1, OPRK1, OPRD1, GRIN1, HTR1A, SLC6A2	Glutamate receptor antagonist
5334	-48.19	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
5335	-48.2	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
5336	-48.21	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
5337	-48.26	kd	CGS001-51135	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
5338	-48.29	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
5339	-48.32	kd	CGS001-2113	ETS1	ETS Transcription Factors			
5340	-48.33	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
5341	-48.33	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
5342	-48.34	kd	CGS001-11333	PDAP1	-			
5343	-48.37	cp	BRD-K37516142	idebenone	Calcium channel modulator			Calcium channel modulator
5344	-48.37	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
5345	-48.38	kd	CGS001-3708	ITPR1	Ion channels / Inositol triphosphate receptors			
5346	-48.39	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
5347	-48.4	kd	CGS001-57396	CLK4	CDC-like kinases			
5348	-48.41	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
5349	-48.52	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5350	-48.52	kd	CGS001-5255	PHKA1	-			
5351	-48.56	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
5352	-48.57	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
5353	-48.64	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
5354	-48.68	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
5355	-48.68	kd	CGS001-9337	CNOT8	-			
5356	-48.71	kd	CGS001-9918	NCAPD2	-			
5357	-48.72	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
5358	-48.73	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
5359	-48.74	oe	ccsbBroad304_00975	MAT2A	-			
5360	-48.74	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
5361	-48.74	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
5362	-48.77	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
5363	-48.77	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
5364	-48.81	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
5365	-48.82	cp	BRD-K37798499	etoposide	Topoisomerase inhibitor		TOP2A, CYP2E1, CYP3A5, TOP2B	Topoisomerase inhibitor
5366	-48.85	kd	CGS001-26227	PHGDH	-			
5367	-48.89	kd	CGS001-4046	LSP1	-			
5368	-48.91	cp	BRD-K82147103	lofepramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
5369	-48.91	kd	CGS001-57167	SALL4	Zinc fingers, C2H2-type			
5370	-48.91	kd	CGS001-29959	NRBP1	NRBP family			
5371	-48.95	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
5372	-48.96	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
5373	-49.01	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
5374	-49.01	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
5375	-49.05	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
5376	-49.1	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5377	-49.15	kd	CGS001-51734	SEPX1	-			
5378	-49.18	oe	ccsbBroad304_00032	ADSL	-			
5379	-49.18	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
5380	-49.19	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
5381	-49.21	kd	CGS001-9270	ITGB1BP1	-			
5382	-49.21	kd	CGS001-474354	LRRC18	-			
5383	-49.21	kd	CGS001-9815	GIT2	Ankyrin repeat domain containing			
5384	-49.22	kd	CGS001-4323	MMP14	Matrix metallopeptidase			
5385	-49.23	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
5386	-49.24	oe	ccsbBroad304_07688	FAM114A2	-			
5387	-49.28	oe	ccsbBroad304_02345	TXNDC9	-			
5388	-49.33	oe	ccsbBroad304_07275	PSMG1	-			
5389	-49.38	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
5390	-49.39	oe	ccsbBroad304_07827	STK38L	NDR family			
5391	-49.4	kd	CGS001-9898	UBAP2L	-			
5392	-49.41	cc		Non Homologous End Joining LOF	-			
5393	-49.41	oe	ccsbBroad304_14174	CDKAL1	-			
5394	-49.42	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
5395	-49.44	oe	ccsbBroad304_03615	ZNF673	-			
5396	-49.44	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
5397	-49.44	kd	CGS001-4664	NAB1	-			
5398	-49.45	oe	ccsbBroad304_06133	TOR1A	-			
5399	-49.46	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
5400	-49.49	oe	ccsbBroad304_02173	ATG5	-			
5401	-49.52	kd	CGS001-23224	SYNE2	-			
5402	-49.57	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
5403	-49.58	kd	CGS001-4176	MCM7	-			
5404	-49.62	kd	CGS001-1386	ATF2	basic leucine zipper proteins			
5405	-49.63	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
5406	-49.63	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
5407	-49.66	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
5408	-49.73	kd	CGS001-2767	GNA11	-			
5409	-49.75	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
5410	-49.83	kd	CGS001-3579	CXCR2	Chemokine receptors			
5411	-49.88	kd	CGS001-523	ATP6V1A	ATPases / V-type			
5412	-49.89	oe	ccsbBroad304_13939	MOK	RCK family			
5413	-49.93	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
5414	-49.96	kd	CGS001-5684	PSMA3	Proteasome subunits			
5415	-49.97	kd	CGS001-84290	CAPNS2	EF-hand domain containing			
5416	-50.02	kd	CGS001-10325	RRAGB	-			
5417	-50.11	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
5418	-50.13	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
5419	-50.17	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
5420	-50.19	oe	ccsbBroad304_00615	GAPDH	-			
5421	-50.22	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
5422	-50.26	cp	BRD-K66206289	lobeline	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist
5423	-50.32	oe	ccsbBroad304_02487	TXNIP	-			
5424	-50.32	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5425	-50.34	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
5426	-50.35	kd	CGS001-6652	SORD	-			
5427	-50.39	kd	CGS001-150280	HORMAD2	-			
5428	-50.44	oe	ccsbBroad304_02686	COPZ1	-			
5429	-50.45	oe	ccsbBroad304_06367	HK1	-			
5430	-50.5	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
5431	-50.56	kd	CGS001-5092	PCBD1	-			
5432	-50.59	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
5433	-50.66	oe	ccsbBroad304_03235	TUBD1	Tubulins			
5434	-50.69	cc		Akt Signaling GOF	-			
5435	-50.71	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
5436	-50.72	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
5437	-50.72	kd	CGS001-10014	HDAC5	Histone deacetylases			
5438	-50.74	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
5439	-50.74	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
5440	-50.74	kd	CGS001-571	BACH1	BTB/POZ domain containing			
5441	-50.75	kd	CGS001-1499	CTNNB1	Catenins			
5442	-50.77	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
5443	-50.8	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
5444	-50.8	kd	CGS001-7917	BAG6	-			
5445	-50.81	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
5446	-50.82	cc		BCL inhibitor	-			
5447	-50.84	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
5448	-50.86	kd	CGS001-2783	GNB2	WD repeat domain containing			
5449	-50.86	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5450	-50.88	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
5451	-50.88	kd	CGS001-9131	AIFM1	-			
5452	-50.95	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
5453	-50.98	kd	CGS001-7251	TSG101	-			
5454	-51.03	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
5455	-51.06	oe	ccsbBroad304_01304	PSEN1	Presenilin			
5456	-51.07	kd	CGS001-4439	MSH5	-			
5457	-51.07	kd	CGS001-896	CCND3	-			
5458	-51.1	kd	CGS001-25942	SIN3A	-			
5459	-51.11	cc		HSP inhibitor	-			
5460	-51.16	oe	ccsbBroad304_00268	CD81	CD molecules			
5461	-51.16	kd	CGS001-1514	CTSL1	-			
5462	-51.17	kd	CGS001-10111	RAD50	-			
5463	-51.18	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
5464	-51.18	kd	CGS001-4835	NQO2	-			
5465	-51.2	kd	CGS001-23510	KCTD2	-			
5466	-51.22	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
5467	-51.24	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
5468	-51.24	oe	ccsbBroad304_00430	GADD45A	-			
5469	-51.33	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
5470	-51.35	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
5471	-51.37	kd	CGS001-10460	TACC3	-			
5472	-51.38	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
5473	-51.4	kd	CGS001-5580	PRKCD	Delta subfamily			
5474	-51.42	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
5475	-51.42	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5476	-51.42	kd	CGS001-4094	MAF	-			
5477	-51.45	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
5478	-51.47	cc		Glucocorticoid receptor agonist	-			
5479	-51.49	kd	CGS001-3912	LAMB1	Laminins			
5480	-51.5	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
5481	-51.5	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
5482	-51.51	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
5483	-51.51	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5484	-51.57	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
5485	-51.58	cp	BRD-K29113274	ketoconazole	Sterol demethylase inhibitor		AR, CYP19A1, CYP21A2, CYP2C19, CYP3A5, CYP3A7, KCNA10	Sterol demethylase inhibitor
5486	-51.59	kd	CGS001-4482	MSRA	-			
5487	-51.6	kd	CGS001-22938	SNW1	-			
5488	-51.61	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
5489	-51.65	kd	CGS001-5188	PET112	-			
5490	-51.66	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
5491	-51.69	oe	ccsbBroad304_02862	CCRN4L	-			
5492	-51.7	kd	CGS001-5428	POLG	DNA polymerases			
5493	-51.72	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
5494	-51.73	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
5495	-51.74	kd	CGS001-5245	PHB	-			
5496	-51.74	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
5497	-51.76	kd	CGS001-2621	GAS6	-			
5498	-51.77	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
5499	-51.77	kd	CGS001-59286	UBL5	-			
5500	-51.78	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
5501	-51.79	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5502	-51.79	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
5503	-51.79	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
5504	-51.82	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
5505	-51.93	kd	CGS001-10007	GNPDA1	-			
5506	-51.96	oe	ccsbBroad304_02405	TFG	-			
5507	-51.97	oe	ccsbBroad304_13891	LCK	Src family			
5508	-51.97	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5509	-52.01	kd	CGS001-24138	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
5510	-52.06	kd	CGS001-84539	MCHR2	GPCR / Class A : MCH receptors			
5511	-52.07	oe	ccsbBroad304_05192	SPRED2	-			
5512	-52.07	cp	BRD-K43236057	piceid	ICAM1 inhibitor		GAA, XDH	ICAM1 inhibitor
5513	-52.12	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
5514	-52.16	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
5515	-52.17	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
5516	-52.19	oe	ccsbBroad304_14047	TACC3	-			
5517	-52.19	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
5518	-52.22	oe	ccsbBroad304_00550	FDXR	-			
5519	-52.24	kd	CGS001-115727	RASGRP4	EF-hand domain containing			
5520	-52.25	kd	CGS001-3832	KIF11	Kinesins			
5521	-52.26	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
5522	-52.27	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5523	-52.29	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
5524	-52.3	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
5525	-52.31	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5526	-52.37	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
5527	-52.37	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
5528	-52.39	kd	CGS001-83729	INHBE	-			
5529	-52.4	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5530	-52.41	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
5531	-52.43	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
5532	-52.45	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
5533	-52.47	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
5534	-52.49	kd	CGS001-89910	UBE3B	-			
5535	-52.5	kd	CGS001-10094	ARPC3	Actin related protein 2/3 complex subunits			
5536	-52.52	oe	ccsbBroad304_02497	YKT6	-			
5537	-52.52	kd	CGS001-4363	ABCC1	ATP binding cassette transporters / subfamily C			
5538	-52.57	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
5539	-52.58	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
5540	-52.61	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
5541	-52.63	kd	CGS001-148327	CREB3L4	basic leucine zipper proteins			
5542	-52.64	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
5543	-52.65	oe	ccsbBroad304_00881	IRF5	-			
5544	-52.72	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
5545	-52.75	kd	CGS001-55662	HIF1AN	-			
5546	-52.76	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
5547	-52.77	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
5548	-52.8	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
5549	-52.83	kd	CGS001-53836	GPR87	GPCR / Class A : Orphans			
5550	-52.86	cc		PKA inhibitor	-			
5551	-52.86	oe	ccsbBroad304_00072	ANXA7	Annexins			
5552	-52.86	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
5553	-52.87	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
5554	-52.95	oe	ccsbBroad304_01215	PLAUR	CD molecules			
5555	-52.99	kd	CGS001-400	ARL1	ADP-ribosylation factors			
5556	-53.03	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
5557	-53.04	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
5558	-53.05	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
5559	-53.09	oe	ccsbBroad304_06253	GALT	-			
5560	-53.09	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
5561	-53.1	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
5562	-53.1	kd	CGS001-572	BAD	-			
5563	-53.11	oe	ccsbBroad304_02576	MLLT11	-			
5564	-53.13	kd	CGS001-8050	PDHX	-			
5565	-53.14	kd	CGS001-7337	UBE3A	-			
5566	-53.16	oe	ccsbBroad304_02443	HAX1	-			
5567	-53.16	kd	CGS001-9360	PPIG	-			
5568	-53.18	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
5569	-53.2	kd	CGS001-10482	NXF1	-			
5570	-53.21	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
5571	-53.31	kd	CGS001-54108	CHRAC1	-			
5572	-53.32	oe	ccsbBroad304_08802	ELAC2	-			
5573	-53.32	kd	CGS001-4706	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
5574	-53.36	kd	CGS001-3046	HBE1	-			
5575	-53.37	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
5576	-53.4	oe	ccsbBroad304_05194	LIPH	-			
5577	-53.43	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
5578	-53.43	oe	ccsbBroad304_06462	ITGAE	Integrins			
5579	-53.44	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
5580	-53.44	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
5581	-53.49	cp	BRD-K99063460	didanosine	Nucleoside reverse transcriptase inhibitor		PNP	Nucleoside reverse transcriptase inhibitor
5582	-53.5	kd	CGS001-9290	GPR55	GPCR / Class A : Orphans			
5583	-53.52	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
5584	-53.53	kd	CGS001-1051	CEBPB	basic leucine zipper proteins			
5585	-53.58	oe	ccsbBroad304_02271	LPGAT1	-			
5586	-53.59	cc		MDM inhibitor	-			
5587	-53.63	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
5588	-53.63	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
5589	-53.63	kd	CGS001-10474	TADA3	-			
5590	-53.66	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
5591	-53.68	kd	CGS001-4615	MYD88	-			
5592	-53.7	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
5593	-53.71	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
5594	-53.74	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
5595	-53.75	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
5596	-53.81	oe	ccsbBroad304_01143	PAFAH1B3	-			
5597	-53.81	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
5598	-53.84	kd	CGS001-4904	YBX1	-			
5599	-53.84	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
5600	-53.86	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
5601	-53.87	oe	ccsbBroad304_07349	MAP7	-			
5602	-53.87	kd	CGS001-55631	LRRC40	-			
5603	-53.88	kd	CGS001-23710	GABARAPL1	-			
5604	-53.91	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
5605	-53.95	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
5606	-54.01	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
5607	-54.03	oe	ccsbBroad304_03591	ETNK1	-			
5608	-54.03	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
5609	-54.04	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
5610	-54.05	kd	CGS001-7342	UBP1	-			
5611	-54.12	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
5612	-54.14	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
5613	-54.19	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
5614	-54.19	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
5615	-54.23	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
5616	-54.28	oe	ccsbBroad304_05902	BNIP3	-			
5617	-54.31	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
5618	-54.35	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
5619	-54.37	cp	BRD-K28849549	mesalazine	Cyclooxygenase inhibitor		PTGS1, PPARG, PTGS2, ALOX5, CHUK, CTNNB1, IKBKB, MPO, NAT1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor, Prostanoid receptor antagonist
5620	-54.39	kd	CGS001-5586	PKN2	Protein kinase N (PKN) family			
5621	-54.39	kd	CGS001-2677	GGCX	Carboxylases			
5622	-54.4	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
5623	-54.41	oe	ccsbBroad304_02012	FADD	-			
5624	-54.42	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
5625	-54.45	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
5626	-54.45	kd	CGS001-10933	MORF4L1	-			
5627	-54.49	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
5628	-54.52	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5629	-54.54	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
5630	-54.59	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
5631	-54.6	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
5632	-54.62	kd	CGS001-1029	CDKN2A	-			
5633	-54.64	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
5634	-54.69	kd	CGS001-6493	SIM2	Basic helix-loop-helix proteins			
5635	-54.7	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
5636	-54.75	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
5637	-54.76	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
5638	-54.76	kd	CGS001-390212	GPR152	GPCR / Class A : Orphans			
5639	-54.8	kd	CGS001-55500	ETNK1	-			
5640	-54.82	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
5641	-54.84	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
5642	-54.86	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
5643	-54.86	kd	CGS001-9759	HDAC4	Histone deacetylases			
5644	-54.91	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
5645	-54.97	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
5646	-54.99	kd	CGS001-6917	TCEA1	General transcription factors			
5647	-55	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
5648	-55.09	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
5649	-55.09	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
5650	-55.1	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
5651	-55.13	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5652	-55.14	kd	CGS001-54536	EXOC6	-			
5653	-55.16	kd	CGS001-2313	FLI1	ETS Transcription Factors			
5654	-55.19	cc		EMSY complex LOF	-			
5655	-55.24	kd	CGS001-64943	NT5DC2	-			
5656	-55.25	kd	CGS001-2212	FCGR2A	CD molecules			
5657	-55.27	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
5658	-55.29	kd	CGS001-60	ACTB	-			
5659	-55.3	kd	CGS001-2149	F2R	Protease activated receptors			
5660	-55.31	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
5661	-55.31	kd	CGS001-2550	GABBR1	GABA receptors			
5662	-55.32	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
5663	-55.33	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
5664	-55.38	kd	CGS001-22933	SIRT2	Histone deacetylases			
5665	-55.4	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
5666	-55.41	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
5667	-55.44	kd	CGS001-445	ASS1	-			
5668	-55.46	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
5669	-55.47	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
5670	-55.47	kd	CGS001-3569	IL6	Interferons			
5671	-55.51	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
5672	-55.53	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
5673	-55.55	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
5674	-55.56	oe	ccsbBroad304_05937	CASP7	Caspases			
5675	-55.57	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
5676	-55.57	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
5677	-55.59	cp	BRD-K86887724	dofetilide	Potassium channel blocker		KCNH2, KCNH1, KCNJ12, KCNK2	Potassium channel blocker
5678	-55.6	oe	ccsbBroad304_00795	HSF2	-			
5679	-55.6	kd	CGS001-22921	MSRB2	-			
5680	-55.67	cp	BRD-A16934955	nalbuphine	Opioid receptor agonist		OPRD1, OPRK1, OPRM1	Opioid receptor agonist, Opioid receptor antagonist
5681	-55.68	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
5682	-55.69	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
5683	-55.72	kd	CGS001-9128	PRPF4	WD repeat domain containing			
5684	-55.74	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
5685	-55.76	cp	BRD-K85503079	perospirone	Dopamine receptor antagonist		DRD2, HTR2A, DRD3, DRD4, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
5686	-55.77	kd	CGS001-10257	ABCC4	ATP binding cassette transporters / subfamily C			
5687	-55.79	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
5688	-55.83	kd	CGS001-3177	SLC29A2	SLC29 family			
5689	-55.83	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
5690	-55.86	kd	CGS001-2078	ERG	ETS Transcription Factors			
5691	-55.87	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
5692	-55.89	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
5693	-55.93	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
5694	-55.96	oe	ccsbBroad304_00001	NAT1	-			
5695	-56.01	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
5696	-56.01	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
5697	-56.01	kd	CGS001-91433	RCCD1	-			
5698	-56.08	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
5699	-56.08	oe	ccsbBroad304_04190	CCDC92	-			
5700	-56.1	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
5701	-56.12	oe	ccsbBroad304_02580	TMED10	-			
5702	-56.13	oe	ccsbBroad304_08426	TEX10	-			
5703	-56.14	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
5704	-56.18	oe	ccsbBroad304_05152	SSBP4	-			
5705	-56.19	oe	ccsbBroad304_06237	GAA	Glycosidases			
5706	-56.19	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
5707	-56.23	oe	ccsbBroad304_00644	GCLC	-			
5708	-56.25	oe	ccsbBroad304_02919	KIAA1279	-			
5709	-56.25	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
5710	-56.31	kd	CGS001-23534	TNPO3	Importins			
5711	-56.31	kd	CGS001-4683	NBN	-			
5712	-56.32	kd	CGS001-1374	CPT1A	-			
5713	-56.36	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
5714	-56.4	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
5715	-56.41	oe	ccsbBroad304_01872	DGCR14	-			
5716	-56.47	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5717	-56.48	kd	CGS001-205	AK4	Adenylate kinases			
5718	-56.51	oe	ccsbBroad304_01002	METTL1	-			
5719	-56.51	oe	ccsbBroad304_02804	KLHDC2	-			
5720	-56.53	oe	ccsbBroad304_03641	ASF1B	-			
5721	-56.56	kd	CGS001-4771	NF2	A-kinase anchor proteins			
5722	-56.58	kd	CGS001-4946	OAZ1	-			
5723	-56.64	kd	CGS001-10202	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5724	-56.67	kd	CGS001-85442	KNDC1	-			
5725	-56.68	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
5726	-56.7	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
5727	-56.72	kd	CGS001-57149	LYRM1	LYR motif containing			
5728	-56.74	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
5729	-56.8	oe	ccsbBroad304_09358	MAPK1IP1L	-			
5730	-56.86	cc		HRH1 antagonist	-			
5731	-56.9	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
5732	-56.91	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
5733	-56.92	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
5734	-56.92	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
5735	-57.02	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
5736	-57.02	kd	CGS001-91975	ZNF300	Zinc fingers, C2H2-type			
5737	-57.02	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5738	-57.2	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
5739	-57.27	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
5740	-57.27	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
5741	-57.28	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
5742	-57.3	cp	BRD-K17705806	JTC-801	Opioid receptor antagonist		OPRL1	Opioid receptor antagonist
5743	-57.31	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
5744	-57.36	oe	ccsbBroad304_09254	PAQR8	-			
5745	-57.37	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
5746	-57.37	kd	CGS001-2071	ERCC3	General transcription factors			
5747	-57.39	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
5748	-57.42	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
5749	-57.53	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
5750	-57.54	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
5751	-57.55	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
5752	-57.56	oe	ccsbBroad304_07029	TADA2A	-			
5753	-57.56	kd	CGS001-546	ATRX	-			
5754	-57.59	kd	CGS001-716	C1S	Complement system			
5755	-57.66	oe	ccsbBroad304_07118	UGDH	-			
5756	-57.74	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
5757	-57.8	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
5758	-57.8	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
5759	-57.81	kd	CGS001-6208	RPS14	S ribosomal proteins			
5760	-57.82	kd	CGS001-26128	KIAA1279	-			
5761	-57.83	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5762	-57.84	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
5763	-57.85	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
5764	-57.86	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
5765	-57.86	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
5766	-57.9	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
5767	-57.92	kd	CGS001-51031	GLOD4	-			
5768	-57.92	kd	CGS001-54811	ZNF562	Zinc fingers, C2H2-type			
5769	-57.97	cp	BRD-K46742498	alosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5770	-57.99	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
5771	-58.07	oe	ccsbBroad304_00809	HUS1	-			
5772	-58.08	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
5773	-58.08	oe	ccsbBroad304_08605	PBK	TOPK family			
5774	-58.11	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
5775	-58.12	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
5776	-58.14	oe	ccsbBroad304_06287	GM2A	-			
5777	-58.17	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
5778	-58.2	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
5779	-58.2	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
5780	-58.21	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
5781	-58.21	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
5782	-58.26	kd	CGS001-8829	NRP1	CD molecules			
5783	-58.3	kd	CGS001-2745	GLRX	-			
5784	-58.31	kd	CGS001-2101	ESRRA	Estrogen-related receptors			
5785	-58.33	cc		ATPase inhibitor	-			
5786	-58.34	oe	ccsbBroad304_08365	CYCS	-			
5787	-58.34	kd	CGS001-8525	DGKZ	-			
5788	-58.34	oe	ccsbBroad304_00810	HYAL1	-			
5789	-58.35	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
5790	-58.38	kd	CGS001-8318	CDC45	-			
5791	-58.39	kd	CGS001-3560	IL2RB	IL-2 receptor family			
5792	-58.41	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
5793	-58.43	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
5794	-58.43	kd	CGS001-3800	KIF5C	Kinesins			
5795	-58.45	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
5796	-58.49	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
5797	-58.49	kd	CGS001-5565	PRKAB2	AMPK subfamily			
5798	-58.52	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
5799	-58.54	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
5800	-58.56	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
5801	-58.57	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
5802	-58.57	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
5803	-58.63	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
5804	-58.64	kd	CGS001-54498	SMOX	-			
5805	-58.65	oe	ccsbBroad304_06098	DHCR24	-			
5806	-58.67	oe	ccsbBroad304_01584	SPARC	-			
5807	-58.69	kd	CGS001-222	ALDH3B2	Aldehyde dehydrogenases			
5808	-58.72	cc		Bile acid	-			
5809	-58.73	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
5810	-58.75	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
5811	-58.76	oe	ccsbBroad304_02702	MSRB2	-			
5812	-58.78	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
5813	-58.86	cp	BRD-K85030058	benactyzine	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
5814	-58.87	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
5815	-58.87	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
5816	-58.88	kd	CGS001-57504	MTA3	GATA zinc finger domain containing			
5817	-58.89	oe	ccsbBroad304_13813	ARAF	RAF family			
5818	-58.94	kd	CGS001-9354	UBE4A	U-box domain containing			
5819	-58.96	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
5820	-58.99	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
5821	-59.01	kd	CGS001-27241	BBS9	-			
5822	-59.04	oe	ccsbBroad304_02671	ECD	-			
5823	-59.06	kd	CGS001-9474	ATG5	-			
5824	-59.08	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
5825	-59.1	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5826	-59.11	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
5827	-59.13	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
5828	-59.13	kd	CGS001-23549	DNPEP	Aminopeptidase I			
5829	-59.17	oe	ccsbBroad304_06642	NIT1	-			
5830	-59.2	oe	ccsbBroad304_02716	NMNAT2	-			
5831	-59.21	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
5832	-59.24	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
5833	-59.25	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
5834	-59.25	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
5835	-59.28	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
5836	-59.29	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
5837	-59.33	oe	ccsbBroad304_02349	MPHOSPH9	-			
5838	-59.34	oe	ccsbBroad304_00783	HPRT1	-			
5839	-59.35	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
5840	-59.36	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
5841	-59.37	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
5842	-59.38	kd	CGS001-4763	NF1	-			
5843	-59.39	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
5844	-59.41	kd	CGS001-6195	RPS6KA1	RSK subfamily			
5845	-59.46	cp	BRD-A07395371	esmolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
5846	-59.49	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
5847	-59.5	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
5848	-59.54	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
5849	-59.68	kd	CGS001-10617	STAMBP	-			
5850	-59.69	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
5851	-59.69	kd	CGS001-23411	SIRT1	Histone deacetylases			
5852	-59.73	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
5853	-59.83	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
5854	-59.87	oe	ccsbBroad304_01001	MEST	-			
5855	-59.9	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
5856	-59.95	oe	ccsbBroad304_04534	HN1L	-			
5857	-59.97	cc		IKK inhibitor	-			
5858	-60.04	kd	CGS001-6256	RXRA	Retinoid X receptors			
5859	-60.09	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
5860	-60.15	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
5861	-60.16	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
5862	-60.17	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
5863	-60.28	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
5864	-60.3	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
5865	-60.36	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
5866	-60.37	kd	CGS001-9774	BCLAF1	-			
5867	-60.42	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
5868	-60.44	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5869	-60.54	kd	CGS001-10138	YAF2	-			
5870	-60.56	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
5871	-60.58	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
5872	-60.6	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
5873	-60.6	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
5874	-60.61	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
5875	-60.62	oe	ccsbBroad304_00003	ABAT	GABA turnover			
5876	-60.62	kd	CGS001-25913	POT1	-			
5877	-60.66	kd	CGS001-1644	DDC	Catecholamine turnover			
5878	-60.68	kd	CGS001-2919	CXCL1	Endogenous ligands			
5879	-60.72	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
5880	-60.74	oe	ccsbBroad304_01632	SYPL1	-			
5881	-60.75	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
5882	-60.75	kd	CGS001-29102	DROSHA	-			
5883	-60.79	oe	ccsbBroad304_00957	M6PR	-			
5884	-60.79	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
5885	-60.79	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
5886	-60.8	kd	CGS001-10298	PAK4	PAKB subfamily			
5887	-60.83	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
5888	-60.89	kd	CGS001-3593	IL12B	Interleukins and interleukin receptors			
5889	-60.9	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
5890	-60.97	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
5891	-60.97	kd	CGS001-2645	GCK	Hexokinases			
5892	-60.99	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
5893	-61.01	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
5894	-61.01	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
5895	-61.03	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
5896	-61.04	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
5897	-61.05	kd	CGS001-5087	PBX1	Homeoboxes / TALE class			
5898	-61.08	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
5899	-61.11	kd	CGS001-79960	PHF17	-			
5900	-61.12	kd	CGS001-55437	STRADB	STLK subfamily			
5901	-61.15	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
5902	-61.17	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
5903	-61.18	oe	ccsbBroad304_02057	P4HA2	-			
5904	-61.18	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
5905	-61.19	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
5906	-61.19	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
5907	-61.2	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
5908	-61.21	cc		Targets of VEGFR inhibitors GOF	-			
5909	-61.23	oe	ccsbBroad304_08266	PIPOX	-			
5910	-61.26	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
5911	-61.27	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
5912	-61.28	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
5913	-61.32	kd	CGS001-4329	ALDH6A1	Aldehyde dehydrogenases			
5914	-61.34	kd	CGS001-1975	EIF4B	RNA binding motif (RRM) containing			
5915	-61.35	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
5916	-61.36	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
5917	-61.36	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
5918	-61.38	kd	CGS001-23355	VPS8	-			
5919	-61.4	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
5920	-61.43	kd	CGS001-7572	ZNF24	Zinc fingers, C2H2-type			
5921	-61.46	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
5922	-61.53	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
5923	-61.54	cp	BRD-K82143716	flucytosine	Antifungal		DNMT1	Antifungal
5924	-61.54	kd	CGS001-219333	USP12	Ubiquitin-specific peptidases			
5925	-61.56	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
5926	-61.62	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
5927	-61.64	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
5928	-61.68	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
5929	-61.69	kd	CGS001-9140	ATG12	-			
5930	-61.79	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
5931	-61.79	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
5932	-61.8	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
5933	-61.82	oe	ccsbBroad304_10491	PFKL	-			
5934	-61.86	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
5935	-61.86	kd	CGS001-1066	CES1	Carboxylesterases			
5936	-61.87	kd	CGS001-54407	SLC38A2	System A-like transporters			
5937	-61.89	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
5938	-61.92	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
5939	-61.92	kd	CGS001-10314	LANCL1	-			
5940	-61.93	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
5941	-61.95	kd	CGS001-23066	CAND2	-			
5942	-61.96	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
5943	-62.02	oe	ccsbBroad304_01152	PCNA	-			
5944	-62.03	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
5945	-62.03	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
5946	-62.05	cc		Aldehyde dehydrogenases LOF	-			
5947	-62.06	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
5948	-62.09	kd	CGS001-4282	MIF	-			
5949	-62.1	kd	CGS001-3297	HSF1	-			
5950	-62.12	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
5951	-62.13	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5952	-62.15	kd	CGS001-84971	ATG4D	-			
5953	-62.17	cp	BRD-K21806131	tegaserod	Serotonin receptor partial agonist		HTR4, HTR2B, HTR2A, HTR2C	Serotonin receptor partial agonist
5954	-62.18	oe	ccsbBroad304_05947	CCNC	-			
5955	-62.19	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
5956	-62.2	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
5957	-62.21	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
5958	-62.21	kd	CGS001-1844	DUSP2	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
5959	-62.25	oe	ccsbBroad304_07119	UGP2	-			
5960	-62.26	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
5961	-62.3	cp	BRD-K49668410	clarithromycin	Bacterial 50S ribosomal subunit inhibitor		CYP2C19, CYP3A4, CYP3A5, CYP3A7	Bacterial 50S ribosomal subunit inhibitor
5962	-62.3	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
5963	-62.34	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
5964	-62.34	kd	CGS001-56647	BCCIP	-			
5965	-62.37	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
5966	-62.39	kd	CGS001-170463	SSBP4	-			
5967	-62.4	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
5968	-62.4	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
5969	-62.43	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
5970	-62.44	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
5971	-62.5	kd	CGS001-4665	NAB2	-			
5972	-62.6	kd	CGS001-11329	STK38	NDR family			
5973	-62.62	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
5974	-62.62	kd	CGS001-3676	ITGA4	Integrins			
5975	-62.68	kd	CGS001-4122	MAN2A2	-			
5976	-62.72	oe	ccsbBroad304_06136	ECHS1	-			
5977	-62.72	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
5978	-62.76	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
5979	-62.77	kd	CGS001-399694	SHC4	SH2 domain containing			
5980	-62.78	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
5981	-62.79	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
5982	-62.83	kd	CGS001-5690	PSMB2	Proteasome subunits			
5983	-62.91	kd	CGS001-10400	PEMT	-			
5984	-62.93	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
5985	-62.93	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
5986	-62.94	kd	CGS001-326	AIRE	Zinc fingers, PHD-type			
5987	-62.96	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
5988	-62.97	cc		Histone deacetylases LOF	-			
5989	-62.98	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
5990	-62.98	kd	CGS001-8192	CLPP	ATPases / AAA-type			
5991	-63	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
5992	-63.03	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
5993	-63.03	kd	CGS001-23387	SIK3	QIK subfamily			
5994	-63.06	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
5995	-63.09	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
5996	-63.09	kd	CGS001-23046	KIF21B	Kinesins			
5997	-63.09	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
5998	-63.1	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
5999	-63.12	kd	CGS001-79618	HMBOX1	Homeoboxes / HNF class			
6000	-63.17	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
6001	-63.19	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
6002	-63.19	kd	CGS001-4232	MEST	-			
6003	-63.21	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
6004	-63.23	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
6005	-63.25	oe	ccsbBroad304_01066	NDUFA4	-			
6006	-63.25	kd	CGS001-5987	TRIM27	-			
6007	-63.28	kd	CGS001-1488	CTBP2	-			
6008	-63.29	kd	CGS001-10991	SLC38A3	System N-like transporters			
6009	-63.29	kd	CGS001-293	SLC25A6	Mitochondrial nucleotide transporter subfamily			
6010	-63.39	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
6011	-63.39	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
6012	-63.41	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
6013	-63.42	kd	CGS001-1198	CLK3	CDC-like kinases			
6014	-63.44	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
6015	-63.45	oe	ccsbBroad304_01640	TAF12	-			
6016	-63.46	kd	CGS001-6223	RPS19	S ribosomal proteins			
6017	-63.47	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
6018	-63.48	kd	CGS001-11179	ZNF277	-			
6019	-63.49	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6020	-63.49	kd	CGS001-10898	CPSF4	-			
6021	-63.59	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
6022	-63.6	kd	CGS001-7057	THBS1	-			
6023	-63.64	kd	CGS001-7270	TTF1	-			
6024	-63.68	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
6025	-63.68	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
6026	-63.69	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
6027	-63.71	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
6028	-63.71	kd	CGS001-3654	IRAK1	Interleukin-1 receptor-associated kinase (IRAK) family			
6029	-63.73	kd	CGS001-27102	EIF2AK1	Other PEK family kinases			
6030	-63.74	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
6031	-63.77	kd	CGS001-84527	ZNF559	Zinc fingers, C2H2-type			
6032	-63.8	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
6033	-63.84	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
6034	-63.87	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
6035	-63.88	kd	CGS001-23047	PDS5B	-			
6036	-63.92	kd	CGS001-57665	RDH14	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6037	-63.93	kd	CGS001-351	APP	Endogenous ligands			
6038	-63.97	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
6039	-63.99	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
6040	-64.01	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
6041	-64.01	kd	CGS001-1879	EBF1	-			
6042	-64.03	kd	CGS001-79722	ANKRD55	Ankyrin repeat domain containing			
6043	-64.04	kd	CGS001-10472	ZNF238	-			
6044	-64.07	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6045	-64.07	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
6046	-64.07	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
6047	-64.12	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
6048	-64.17	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
6049	-64.18	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
6050	-64.19	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
6051	-64.2	kd	CGS001-113451	ADC	-			
6052	-64.23	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
6053	-64.24	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
6054	-64.25	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
6055	-64.29	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
6056	-64.29	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
6057	-64.32	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6058	-64.33	oe	ccsbBroad304_06565	MB	-			
6059	-64.35	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
6060	-64.4	kd	CGS001-8659	ALDH4A1	Aldehyde dehydrogenases			
6061	-64.42	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
6062	-64.42	kd	CGS001-109	ADCY3	Adenylyl cyclases			
6063	-64.45	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6064	-64.49	kd	CGS001-333929	SNAI3	Snail homologs			
6065	-64.5	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6066	-64.52	kd	CGS001-29116	MYLIP	-			
6067	-64.53	kd	CGS001-7533	YWHAH	-			
6068	-64.55	oe	ccsbBroad304_06292	GNAI2	-			
6069	-64.56	oe	ccsbBroad304_00652	GNAS	-			
6070	-64.56	kd	CGS001-162655	ZNF519	Zinc fingers, C2H2-type			
6071	-64.56	kd	CGS001-7849	PAX8	Paired boxes			
6072	-64.57	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
6073	-64.59	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
6074	-64.6	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
6075	-64.61	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
6076	-64.62	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
6077	-64.65	kd	CGS001-2182	ACSL4	Acyl-CoA synthetase family			
6078	-64.67	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
6079	-64.69	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
6080	-64.72	oe	ccsbBroad304_05038	HORMAD2	-			
6081	-64.79	kd	CGS001-6871	TADA2A	-			
6082	-64.81	oe	ccsbBroad304_03232	VPS28	-			
6083	-64.83	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
6084	-64.87	kd	CGS001-9854	C2CD2L	-			
6085	-64.87	kd	CGS001-5699	PSMB10	Proteasome (prosome, macropain) subunits			
6086	-64.89	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
6087	-64.91	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
6088	-64.92	oe	ccsbBroad304_06134	ECH1	-			
6089	-64.94	oe	ccsbBroad304_03405	CHRAC1	-			
6090	-64.95	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
6091	-64.95	kd	CGS001-51719	CAB39	-			
6092	-64.96	kd	CGS001-8702	B4GALT4	Beta 4-glycosyltransferases			
6093	-64.97	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
6094	-64.98	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
6095	-64.99	kd	CGS001-4331	MNAT1	RING-type (C3HC4) zinc fingers			
6096	-65.06	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
6097	-65.14	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
6098	-65.21	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
6099	-65.23	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
6100	-65.24	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
6101	-65.25	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
6102	-65.26	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
6103	-65.27	cc		SRY LOF	-			
6104	-65.29	oe	ccsbBroad304_02501	DCTN6	-			
6105	-65.31	kd	CGS001-55165	CEP55	-			
6106	-65.32	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
6107	-65.33	kd	CGS001-65975	STK33	CAMK-unique family			
6108	-65.35	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
6109	-65.37	kd	CGS001-51176	LEF1	-			
6110	-65.4	kd	CGS001-275	AMT	-			
6111	-65.41	oe	ccsbBroad304_07727	LIAS	-			
6112	-65.48	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
6113	-65.49	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
6114	-65.49	kd	CGS001-10906	TRAFD1	-			
6115	-65.5	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
6116	-65.51	cc		GATA Zinc finger domain containing LOF	-			
6117	-65.51	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
6118	-65.51	kd	CGS001-23274	CLEC16A	C-type lectin domain containing			
6119	-65.52	kd	CGS001-84515	MCM8	-			
6120	-65.55	kd	CGS001-10023	FRAT1	-			
6121	-65.64	kd	CGS001-4200	ME2	-			
6122	-65.65	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
6123	-65.68	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
6124	-65.69	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
6125	-65.72	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
6126	-65.77	kd	CGS001-6469	SHH	-			
6127	-65.81	oe	ccsbBroad304_01148	PCBD1	-			
6128	-65.81	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
6129	-65.84	kd	CGS001-79139	DERL1	-			
6130	-65.85	cc		RAF inhibitor	-			
6131	-65.85	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
6132	-65.87	cc		HIF activator	-			
6133	-65.94	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
6134	-65.96	cp	BRD-A52282606	lacidipine	Calcium channel blocker		CACNA1C	Calcium channel blocker
6135	-65.97	oe	ccsbBroad304_09281	TPD52L3	-			
6136	-65.97	oe	ccsbBroad304_03573	BRF2	-			
6137	-65.98	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
6138	-65.99	kd	CGS001-573	BAG1	-			
6139	-66.03	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
6140	-66.11	kd	CGS001-3455	IFNAR2	Interferon receptor family			
6141	-66.16	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
6142	-66.16	oe	ccsbBroad304_01651	TCF7L2	-			
6143	-66.17	kd	CGS001-2067	ERCC1	-			
6144	-66.2	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
6145	-66.22	kd	CGS001-2194	FASN	Short chain dehydrogenase/reductase superfamily / Atypical members			
6146	-66.3	oe	ccsbBroad304_14291	GDPD5	-			
6147	-66.3	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
6148	-66.3	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
6149	-66.3	kd	CGS001-81620	CDT1	-			
6150	-66.31	kd	CGS001-122402	TDRD9	Tudor domain containing			
6151	-66.31	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
6152	-66.33	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
6153	-66.41	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
6154	-66.42	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
6155	-66.45	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
6156	-66.46	oe	ccsbBroad304_02399	TNIP1	-			
6157	-66.5	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
6158	-66.51	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
6159	-66.53	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
6160	-66.55	kd	CGS001-3932	LCK	Src family			
6161	-66.6	oe	ccsbBroad304_10230	STK19	G11 family			
6162	-66.6	kd	CGS001-6189	RPS3A	S ribosomal proteins			
6163	-66.6	kd	CGS001-4893	NRAS	RAS subfamily			
6164	-66.62	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
6165	-66.62	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
6166	-66.71	kd	CGS001-9319	TRIP13	ATPases / AAA-type			
6167	-66.72	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
6168	-66.74	kd	CGS001-350	APOH	Apolipoproteins			
6169	-66.77	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
6170	-66.78	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
6171	-66.78	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
6172	-66.78	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
6173	-66.79	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
6174	-66.82	kd	CGS001-55226	NAT10	-			
6175	-66.82	kd	CGS001-3590	IL11RA	IL-6 receptor family			
6176	-66.84	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
6177	-66.87	kd	CGS001-5813	PURA	-			
6178	-66.9	kd	CGS001-23223	RRP12	-			
6179	-66.91	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
6180	-66.91	kd	CGS001-310	ANXA7	Annexins			
6181	-66.93	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
6182	-66.93	kd	CGS001-29928	TIMM22	-			
6183	-66.97	oe	ccsbBroad304_07888	CBX6	-			
6184	-66.97	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
6185	-66.98	kd	CGS001-1184	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
6186	-67	kd	CGS001-3456	IFNB1	Interferons			
6187	-67.06	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
6188	-67.08	kd	CGS001-29775	CARD10	-			
6189	-67.1	oe	ccsbBroad304_06996	SRM	-			
6190	-67.1	kd	CGS001-3226	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
6191	-67.11	kd	CGS001-3176	HNMT	-			
6192	-67.13	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
6193	-67.14	kd	CGS001-2853	GPR31	GPCR / Class A : Orphans			
6194	-67.15	kd	CGS001-10412	NSA2	-			
6195	-67.2	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
6196	-67.2	kd	CGS001-55012	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
6197	-67.26	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
6198	-67.29	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
6199	-67.32	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6200	-67.34	kd	CGS001-10312	TCIRG1	ATPases / V-type			
6201	-67.39	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
6202	-67.41	oe	ccsbBroad304_00549	FDX1	-			
6203	-67.41	cp	BRD-K39621635	artemether	Antimalarial		ATP1A1, CYP2B6, CYP2C19, CYP3A5	Antimalarial
6204	-67.45	kd	CGS001-978	CDA	-			
6205	-67.54	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
6206	-67.56	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
6207	-67.56	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
6208	-67.58	oe	ccsbBroad304_03772	CCNL1	-			
6209	-67.61	cp	BRD-K10961822	latanoprost	Prostanoid receptor agonist		PTGFR	Prostanoid receptor agonist
6210	-67.65	kd	CGS001-2145	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
6211	-67.68	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
6212	-67.68	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
6213	-67.75	kd	CGS001-90861	HN1L	-			
6214	-67.84	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
6215	-67.85	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
6216	-67.86	kd	CGS001-9687	GREB1	-			
6217	-67.87	kd	CGS001-891	CCNB1	-			
6218	-67.88	kd	CGS001-8824	CES2	Carboxylesterases			
6219	-67.92	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
6220	-67.95	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
6221	-67.95	kd	CGS001-53632	PRKAG3	AMPK subfamily			
6222	-67.96	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
6223	-67.97	oe	ccsbBroad304_08339	CMPK1	-			
6224	-67.99	kd	CGS001-51530	ZC3HC1	Zinc fingers, C3HC-type			
6225	-67.99	kd	CGS001-1910	EDNRB	Endothelin receptors			
6226	-68	kd	CGS001-7915	ALDH5A1	Aldehyde dehydrogenases			
6227	-68	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
6228	-68.06	kd	CGS001-8800	PEX11A	-			
6229	-68.12	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
6230	-68.13	oe	ccsbBroad304_03910	CCDC90A	-			
6231	-68.15	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
6232	-68.17	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
6233	-68.19	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
6234	-68.2	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
6235	-68.23	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
6236	-68.24	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
6237	-68.28	kd	CGS001-171017	ZNF384	Zinc fingers, C2H2-type			
6238	-68.35	kd	CGS001-32	ACACB	Carboxylases			
6239	-68.36	kd	CGS001-515	ATP5F1	ATPases / F-type			
6240	-68.37	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
6241	-68.39	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
6242	-68.42	oe	ccsbBroad304_06639	NFYB	-			
6243	-68.45	kd	CGS001-2558	GABRA5	GABA receptors			
6244	-68.46	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
6245	-68.53	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
6246	-68.54	cp	BRD-A35519318	benidipine	Calcium channel blocker		CACNA1C, CACNA1G, CYP3A5	Calcium channel blocker
6247	-68.55	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
6248	-68.6	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
6249	-68.62	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
6250	-68.64	cc		Vesicular Transport LOF	-			
6251	-68.64	oe	ccsbBroad304_02373	SPRY2	-			
6252	-68.65	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
6253	-68.68	oe	ccsbBroad304_04457	TOX2	-			
6254	-68.69	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
6255	-68.75	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
6256	-68.77	oe	ccsbBroad304_09954	PTRF	-			
6257	-68.81	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
6258	-68.81	kd	CGS001-30	ACAA1	-			
6259	-68.81	oe	ccsbBroad304_09095	PUS7L	-			
6260	-68.81	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
6261	-68.86	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
6262	-68.92	kd	CGS001-5159	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6263	-68.97	kd	CGS001-7535	ZAP70	Syk family			
6264	-69.04	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
6265	-69.09	kd	CGS001-6929	TCF3	Basic helix-loop-helix proteins			
6266	-69.13	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
6267	-69.13	kd	CGS001-23597	ACOT9	Acyl CoA thioesterases			
6268	-69.14	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6269	-69.14	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
6270	-69.14	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
6271	-69.19	oe	ccsbBroad304_00614	GAMT	-			
6272	-69.21	oe	ccsbBroad304_02217	FEZ1	-			
6273	-69.22	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
6274	-69.22	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
6275	-69.22	kd	CGS001-5359	PLSCR1	-			
6276	-69.26	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
6277	-69.27	oe	ccsbBroad304_02287	GNPDA1	-			
6278	-69.27	kd	CGS001-3601	IL15RA	IL-2 receptor family			
6279	-69.29	kd	CGS001-5930	RBBP6	-			
6280	-69.29	kd	CGS001-10437	IFI30	-			
6281	-69.38	kd	CGS001-94103	ORMDL3	-			
6282	-69.4	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
6283	-69.42	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
6284	-69.43	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
6285	-69.43	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
6286	-69.48	kd	CGS001-55139	ANKZF1	Ankyrin repeat domain containing			
6287	-69.49	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
6288	-69.49	cp	BRD-K27184429	levocetirizine	Histamine receptor antagonist		HRH1, CXCL8	Histamine receptor antagonist
6289	-69.52	kd	CGS001-9170	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6290	-69.55	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
6291	-69.61	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
6292	-69.61	kd	CGS001-25874	BRP44	-			
6293	-69.62	kd	CGS001-7108	TM7SF2	-			
6294	-69.64	oe	ccsbBroad304_02626	PKIG	-			
6295	-69.64	oe	ccsbBroad304_00249	CD14	CD molecules			
6296	-69.65	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
6297	-69.66	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
6298	-69.78	cp	BRD-K50866992	tropisetron	Serotonin receptor antagonist		HTR3A, GLRA1, GLRA2, GLRB, HTR4	Serotonin receptor antagonist
6299	-69.79	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
6300	-69.79	cp	BRD-K51730347	diphencyprone	Immunostimulant			Immunostimulant
6301	-69.81	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
6302	-69.86	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
6303	-69.93	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
6304	-69.93	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
6305	-69.95	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
6306	-70.03	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
6307	-70.03	kd	CGS001-308	ANXA5	Annexins			
6308	-70.05	kd	CGS001-9784	SNX17	Sorting nexins			
6309	-70.09	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
6310	-70.1	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
6311	-70.11	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
6312	-70.14	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
6313	-70.2	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
6314	-70.22	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
6315	-70.24	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
6316	-70.24	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
6317	-70.25	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
6318	-70.27	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
6319	-70.28	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
6320	-70.47	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
6321	-70.52	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
6322	-70.54	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6323	-70.57	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
6324	-70.57	kd	CGS001-3054	HCFC1	-			
6325	-70.62	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
6326	-70.63	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
6327	-70.65	oe	ccsbBroad304_00146	BAD	-			
6328	-70.65	kd	CGS001-203523	ZNF449	Zinc fingers, C2H2-type			
6329	-70.73	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
6330	-70.8	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
6331	-70.81	kd	CGS001-147948	ZNF582	Zinc fingers, C2H2-type			
6332	-70.82	oe	ccsbBroad304_02759	DICER1	-			
6333	-70.82	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6334	-70.84	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
6335	-70.85	oe	ccsbBroad304_01166	PDK2	PDHK family			
6336	-70.85	kd	CGS001-3225	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
6337	-70.87	kd	CGS001-7879	RAB7A	RAB, member RAS oncogene			
6338	-70.89	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
6339	-70.91	kd	CGS001-1951	CELSR3	Cadherins / Major cadherins			
6340	-70.94	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
6341	-70.97	kd	CGS001-771	CA12	Carbonic anhydrases			
6342	-71.05	kd	CGS001-6391	SDHC	Mitochondrial respiratory chain complex / Complex II			
6343	-71.08	oe	ccsbBroad304_00818	IDH3A	-			
6344	-71.11	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
6345	-71.12	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
6346	-71.14	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
6347	-71.19	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
6348	-71.27	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
6349	-71.34	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
6350	-71.35	oe	ccsbBroad304_07511	KIF14	Kinesins			
6351	-71.41	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
6352	-71.45	kd	CGS001-7756	ZNF207	Zinc fingers, C2H2-type			
6353	-71.46	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
6354	-71.5	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
6355	-71.5	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
6356	-71.51	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
6357	-71.52	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
6358	-71.55	kd	CGS001-206358	SLC36A1	SLC36 family of proton-coupled amino acid transporters			
6359	-71.57	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
6360	-71.59	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
6361	-71.6	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
6362	-71.61	oe	ccsbBroad304_03934	LEPRE1	-			
6363	-71.66	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
6364	-71.66	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
6365	-71.67	kd	CGS001-9276	COPB2	WD repeat domain containing			
6366	-71.71	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
6367	-71.72	kd	CGS001-8428	STK24	YSK subfamily			
6368	-71.72	kd	CGS001-4297	MLL	-			
6369	-71.73	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
6370	-71.74	cc		Protein phosphatase catalytic subunits LOF	-			
6371	-71.74	cp	BRD-K32744045	disulfiram	Aldehyde dehydrogenase inhibitor		ALDH2, ALDH1A2, ALDH5A1, ALDH7A1, CYP2E1, DBH, DNMT1, TRPA1	Aldehyde dehydrogenase inhibitor, TRPV agonist, DNA methyltransferase inhibitor
6372	-71.75	oe	ccsbBroad304_00070	ANXA5	Annexins			
6373	-71.78	kd	CGS001-10695	CNPY3	Trinucleotide (CAG) repeat containing			
6374	-71.79	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
6375	-71.8	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
6376	-71.81	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
6377	-71.81	kd	CGS001-9232	PTTG1	-			
6378	-71.81	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
6379	-71.81	kd	CGS001-80347	COASY	-			
6380	-71.82	oe	ccsbBroad304_06670	OGG1	-			
6381	-71.84	kd	CGS001-2770	GNAI1	-			
6382	-71.9	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
6383	-71.92	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
6384	-71.93	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
6385	-71.94	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
6386	-71.95	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
6387	-71.96	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
6388	-71.98	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
6389	-72.06	kd	CGS001-6204	RPS10	S ribosomal proteins			
6390	-72.07	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
6391	-72.08	kd	CGS001-9447	AIM2	-			
6392	-72.13	kd	CGS001-5817	PVR	Immunoglobulin superfamily / C2-set domain containing			
6393	-72.14	kd	CGS001-10447	FAM3C	-			
6394	-72.19	oe	ccsbBroad304_01593	SRP14	-			
6395	-72.19	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
6396	-72.19	kd	CGS001-5037	PEBP1	-			
6397	-72.21	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
6398	-72.22	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
6399	-72.22	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
6400	-72.26	kd	CGS001-6663	SOX10	SRY (sex determining region Y)-boxes			
6401	-72.27	oe	ccsbBroad304_02869	ASF1A	-			
6402	-72.33	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
6403	-72.35	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
6404	-72.35	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
6405	-72.36	kd	CGS001-2056	EPO	Endogenous ligands			
6406	-72.42	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
6407	-72.43	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
6408	-72.44	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
6409	-72.44	kd	CGS001-167826	OLIG3	Basic helix-loop-helix proteins			
6410	-72.49	cc		Potassium channel blocker	-			
6411	-72.5	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
6412	-72.5	kd	CGS001-54901	CDKAL1	-			
6413	-72.51	kd	CGS001-5928	RBBP4	WD repeat domain containing			
6414	-72.54	kd	CGS001-54915	YTHDF1	-			
6415	-72.55	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
6416	-72.55	kd	CGS001-2678	GGT1	CD molecules			
6417	-72.59	oe	ccsbBroad304_06665	OAT	-			
6418	-72.64	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
6419	-72.64	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
6420	-72.71	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
6421	-72.77	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
6422	-72.8	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
6423	-72.8	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
6424	-72.8	kd	CGS001-1903	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
6425	-72.85	kd	CGS001-147179	WIPF2	-			
6426	-72.85	kd	CGS001-440	ASNS	-			
6427	-72.86	cc		G2 M Checkpoint LOF	-			
6428	-72.9	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
6429	-72.93	kd	CGS001-8878	SQSTM1	-			
6430	-72.94	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
6431	-72.98	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
6432	-72.99	kd	CGS001-25885	POLR1A	RNA polymerase subunits			
6433	-73.01	cp	BRD-K29530284	amlexanox	Histamine receptor modulator		FGF1, IL3, S100A12, S100A13	Histamine receptor modulator
6434	-73.03	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
6435	-73.04	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
6436	-73.18	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
6437	-73.18	kd	CGS001-10769	PLK2	Polo-like kinase (PLK) family			
6438	-73.19	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
6439	-73.19	kd	CGS001-7357	UGCG	Glycosyltransferase family 2 domain containing			
6440	-73.23	kd	CGS001-9767	PHF16	-			
6441	-73.25	oe	ccsbBroad304_09756	PAQR7	-			
6442	-73.26	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
6443	-73.26	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
6444	-73.26	kd	CGS001-55715	DOK4	Pleckstrin homology (PH) domain containing			
6445	-73.28	oe	ccsbBroad304_01373	RAN	-			
6446	-73.34	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
6447	-73.34	kd	CGS001-11188	NISCH	-			
6448	-73.34	kd	CGS001-6500	SKP1	-			
6449	-73.37	kd	CGS001-4199	ME1	-			
6450	-73.39	kd	CGS001-6925	TCF4	Basic helix-loop-helix proteins			
6451	-73.4	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
6452	-73.4	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
6453	-73.42	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
6454	-73.51	oe	ccsbBroad304_06235	G6PD	-			
6455	-73.51	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
6456	-73.51	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
6457	-73.54	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
6458	-73.57	oe	ccsbBroad304_01527	SGK1	SGK family			
6459	-73.59	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
6460	-73.62	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
6461	-73.64	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
6462	-73.67	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
6463	-73.71	kd	CGS001-8409	UXT	-			
6464	-73.74	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6465	-73.78	kd	CGS001-51451	LCMT1	-			
6466	-73.79	kd	CGS001-85027	C5ORF62	-			
6467	-73.81	oe	ccsbBroad304_00112	ASNA1	-			
6468	-73.82	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
6469	-73.84	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
6470	-73.85	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
6471	-73.86	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
6472	-73.88	oe	ccsbBroad304_02357	SSX3	-			
6473	-73.9	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
6474	-73.91	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
6475	-73.91	oe	ccsbBroad304_02737	JMJD6	-			
6476	-73.95	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
6477	-73.96	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
6478	-73.96	kd	CGS001-2237	FEN1	-			
6479	-73.97	kd	CGS001-26993	AKAP8L	-			
6480	-73.98	cc		Rho GTPase activating proteins LOF	-			
6481	-74.01	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
6482	-74.04	kd	CGS001-5831	PYCR1	-			
6483	-74.07	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
6484	-74.07	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
6485	-74.09	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
6486	-74.09	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
6487	-74.09	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
6488	-74.12	kd	CGS001-2958	GTF2A2	General transcription factors			
6489	-74.13	kd	CGS001-79850	FAM57A	-			
6490	-74.14	kd	CGS001-1069	CETN2	EF-hand domain containing			
6491	-74.16	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
6492	-74.16	kd	CGS001-2932	GSK3B	GSK subfamily			
6493	-74.19	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
6494	-74.2	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
6495	-74.2	kd	CGS001-5915	RARB	Retinoic acid receptors			
6496	-74.23	oe	ccsbBroad304_07088	TP53	-			
6497	-74.24	kd	CGS001-9919	SEC16A	-			
6498	-74.27	oe	ccsbBroad304_02581	ASCC3	-			
6499	-74.28	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
6500	-74.28	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
6501	-74.28	kd	CGS001-2197	FAU	S ribosomal proteins			
6502	-74.29	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6503	-74.31	cp	BRD-K81169441	cerivastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A5	HMGCR inhibitor
6504	-74.31	kd	CGS001-23314	SATB2	Homeoboxes / CUT class			
6505	-74.32	oe	ccsbBroad304_04053	DERL1	-			
6506	-74.36	kd	CGS001-3927	LASP1	-			
6507	-74.4	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
6508	-74.43	oe	ccsbBroad304_03565	ADI1	-			
6509	-74.52	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
6510	-74.52	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
6511	-74.55	cc		DNA dependent protein kinase inhibitor	-			
6512	-74.57	kd	CGS001-678	ZFP36L2	RING-type (C3HC4) zinc fingers			
6513	-74.57	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
6514	-74.59	kd	CGS001-51311	TLR8	Toll-like receptor family			
6515	-74.6	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
6516	-74.62	oe	ccsbBroad304_01469	RSU1	-			
6517	-74.64	oe	ccsbBroad304_03311	EVL	-			
6518	-74.64	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
6519	-74.66	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
6520	-74.69	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
6521	-74.71	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
6522	-74.72	kd	CGS001-1841	DTYMK	-			
6523	-74.73	kd	CGS001-2562	GABRB3	GABA receptors			
6524	-74.83	kd	CGS001-5066	PAM	-			
6525	-74.83	kd	CGS001-2639	GCDH	-			
6526	-74.85	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
6527	-74.87	cc		Retinoid receptor agonist	-			
6528	-74.87	kd	CGS001-10308	ZNF267	Zinc fingers, C2H2-type			
6529	-74.88	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
6530	-74.9	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
6531	-74.91	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
6532	-74.95	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
6533	-74.95	kd	CGS001-3298	HSF2	-			
6534	-74.96	kd	CGS001-5581	PRKCE	Eta subfamily			
6535	-74.96	kd	CGS001-4758	NEU1	-			
6536	-74.97	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
6537	-74.98	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
6538	-74.99	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
6539	-75.01	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
6540	-75.05	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
6541	-75.06	oe	ccsbBroad304_00987	MCM3	-			
6542	-75.11	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
6543	-75.13	kd	CGS001-125919	ZNF543	Zinc fingers, C2H2-type			
6544	-75.14	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
6545	-75.14	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
6546	-75.2	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
6547	-75.21	oe	ccsbBroad304_03080	C16ORF80	-			
6548	-75.22	kd	CGS001-10973	ASCC3	-			
6549	-75.23	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
6550	-75.24	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
6551	-75.25	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
6552	-75.25	oe	ccsbBroad304_00690	GRN	-			
6553	-75.26	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
6554	-75.27	kd	CGS001-23621	BACE1	Pepsin			
6555	-75.27	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
6556	-75.34	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
6557	-75.36	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
6558	-75.37	cp	BRD-A24381660	zeranol	Estrogen receptor agonist			Estrogen receptor agonist
6559	-75.4	kd	CGS001-6513	SLC2A1	Solute carriers			
6560	-75.4	kd	CGS001-2852	GPER	-			
6561	-75.45	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
6562	-75.48	kd	CGS001-83439	TCF7L1	-			
6563	-75.5	kd	CGS001-593	BCKDHA	-			
6564	-75.52	oe	ccsbBroad304_01923	UXT	-			
6565	-75.52	kd	CGS001-149428	BNIPL	-			
6566	-75.55	kd	CGS001-661	POLR3D	RNA polymerase subunits			
6567	-75.59	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
6568	-75.6	cc		Thymidylate synthase inhibitor	-			
6569	-75.6	cc		Reverse transcriptase inhibitor	-			
6570	-75.64	oe	ccsbBroad304_03097	CNOT7	-			
6571	-75.64	kd	CGS001-56882	CDC42SE1	-			
6572	-75.65	oe	ccsbBroad304_01371	RALA	-			
6573	-75.66	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6574	-75.67	oe	ccsbBroad304_02045	BUD31	-			
6575	-75.67	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
6576	-75.68	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
6577	-75.72	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
6578	-75.77	kd	CGS001-2887	GRB10	Pleckstrin homology (PH) domain containing			
6579	-75.78	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
6580	-75.78	kd	CGS001-64921	CASD1	-			
6581	-75.79	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
6582	-75.84	kd	CGS001-3205	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
6583	-75.89	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
6584	-75.92	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
6585	-75.95	kd	CGS001-57721	METTL14	-			
6586	-75.96	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
6587	-75.96	kd	CGS001-3572	IL6ST	IL-6 receptor family			
6588	-75.97	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
6589	-75.99	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
6590	-76	oe	ccsbBroad304_01664	TGFA	-			
6591	-76	kd	CGS001-2247	FGF2	Endogenous ligands			
6592	-76.02	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
6593	-76.03	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
6594	-76.03	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
6595	-76.1	kd	CGS001-5480	PPIC	-			
6596	-76.13	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
6597	-76.13	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
6598	-76.13	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
6599	-76.17	kd	CGS001-4708	NDUFB2	Mitochondrial respiratory chain complex / Complex I			
6600	-76.19	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
6601	-76.19	kd	CGS001-8463	TEAD2	-			
6602	-76.19	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
6603	-76.2	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6604	-76.2	kd	CGS001-136	ADORA2B	GPCR / Class A : Adenosine receptors			
6605	-76.21	kd	CGS001-5583	PRKCH	Eta subfamily			
6606	-76.23	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
6607	-76.23	kd	CGS001-10379	IRF9	-			
6608	-76.24	kd	CGS001-9917	FAM20B	-			
6609	-76.27	oe	ccsbBroad304_02864	PRDX5	-			
6610	-76.27	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
6611	-76.31	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
6612	-76.31	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
6613	-76.35	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
6614	-76.35	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
6615	-76.36	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
6616	-76.43	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
6617	-76.47	oe	ccsbBroad304_03933	CARD9	-			
6618	-76.47	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
6619	-76.48	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6620	-76.49	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
6621	-76.5	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
6622	-76.51	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
6623	-76.52	kd	CGS001-2806	GOT2	-			
6624	-76.55	cc		PI3K Signaling LOF	-			
6625	-76.6	kd	CGS001-59343	SENP2	-			
6626	-76.64	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
6627	-76.69	kd	CGS001-5875	RABGGTA	Prenyltransferase alpha subunit repeat containing			
6628	-76.7	kd	CGS001-3596	IL13	Interleukins and interleukin receptors			
6629	-76.71	kd	CGS001-10813	UTP14A	-			
6630	-76.72	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
6631	-76.77	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
6632	-76.78	cp	BRD-A41450521	tosufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6633	-76.78	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
6634	-76.78	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
6635	-76.84	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
6636	-76.87	oe	ccsbBroad304_01054	GADD45B	-			
6637	-76.88	cc		NFkB pathway inhibitor	-			
6638	-76.9	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
6639	-76.94	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
6640	-76.95	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
6641	-77.04	kd	CGS001-9541	CIR1	-			
6642	-77.1	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
6643	-77.13	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
6644	-77.16	kd	CGS001-2072	ERCC4	-			
6645	-77.18	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6646	-77.2	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6647	-77.23	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
6648	-77.24	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
6649	-77.29	kd	CGS001-30836	DNTTIP2	-			
6650	-77.31	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
6651	-77.31	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
6652	-77.32	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
6653	-77.34	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
6654	-77.35	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
6655	-77.39	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
6656	-77.39	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6657	-77.44	kd	CGS001-1999	ELF3	ETS Transcription Factors			
6658	-77.51	oe	ccsbBroad304_02500	RRAGA	-			
6659	-77.51	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
6660	-77.54	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
6661	-77.54	kd	CGS001-5357	PLS1	EF-hand domain containing			
6662	-77.55	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
6663	-77.57	kd	CGS001-7771	ZFP112	-			
6664	-77.58	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
6665	-77.58	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6666	-77.62	kd	CGS001-1131	CHRM3	Cholinergic receptors			
6667	-77.64	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
6668	-77.64	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
6669	-77.68	kd	CGS001-5901	RAN	-			
6670	-77.7	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
6671	-77.72	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
6672	-77.73	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
6673	-77.74	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
6674	-77.74	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
6675	-77.81	cc		HMGCR inhibitor	-			
6676	-77.83	kd	CGS001-319100	TAAR6	GPCR / Class A : Trace amine associated receptors			
6677	-77.84	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
6678	-77.85	kd	CGS001-6608	SMO	GPCR / Class F : Frizzled receptors			
6679	-77.89	kd	CGS001-23678	SGK3	SGK family			
6680	-77.92	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
6681	-77.94	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
6682	-78	cp	BRD-K05350981	oligomycin-c	ATPase inhibitor		ATP5A1	ATPase inhibitor, ATP synthase inhibitor
6683	-78.01	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
6684	-78.03	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
6685	-78.07	kd	CGS001-5636	PRPSAP2	-			
6686	-78.09	oe	ccsbBroad304_00418	CD55	CD molecules			
6687	-78.11	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
6688	-78.12	kd	CGS001-388677	NOTCH2NL	-			
6689	-78.14	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
6690	-78.16	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
6691	-78.16	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
6692	-78.18	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
6693	-78.2	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
6694	-78.23	oe	ccsbBroad304_13499	KSR2	RAF family			
6695	-78.23	kd	CGS001-5829	PXN	-			
6696	-78.25	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
6697	-78.29	kd	CGS001-6009	RHEB	-			
6698	-78.31	oe	ccsbBroad304_04619	GNG8	-			
6699	-78.31	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
6700	-78.31	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
6701	-78.35	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
6702	-78.4	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
6703	-78.41	kd	CGS001-6198	RPS6KB1	p70 subfamily			
6704	-78.41	kd	CGS001-51079	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
6705	-78.42	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
6706	-78.45	kd	CGS001-2512	FTL	-			
6707	-78.49	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
6708	-78.49	kd	CGS001-9134	CCNE2	-			
6709	-78.5	kd	CGS001-991	CDC20	WD repeat domain containing			
6710	-78.52	kd	CGS001-3315	HSPB1	Heat shock proteins / HSPB			
6711	-78.55	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
6712	-78.56	kd	CGS001-27347	STK39	FRAY subfamily			
6713	-78.62	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
6714	-78.62	kd	CGS001-63948	DMRTB1	-			
6715	-78.64	cc		Nucleoside reverse transcriptase inhibitor	-			
6716	-78.66	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
6717	-78.7	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6718	-78.71	kd	CGS001-58478	ENOPH1	-			
6719	-78.75	cc		Estrogen receptor antagonist	-			
6720	-78.75	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
6721	-78.78	kd	CGS001-506	ATP5B	ATPases / F-type			
6722	-78.79	kd	CGS001-2730	GCLM	-			
6723	-78.81	kd	CGS001-4717	NDUFC1	Mitochondrial respiratory chain complex / Complex I			
6724	-78.83	kd	CGS001-3682	ITGAE	Integrins			
6725	-78.84	oe	ccsbBroad304_07800	EXOSC8	-			
6726	-78.86	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
6727	-78.87	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
6728	-78.89	oe	ccsbBroad304_00398	CTSL2	-			
6729	-78.92	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
6730	-78.99	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
6731	-79.02	cc		Thromboxane receptor antagonist	-			
6732	-79.03	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
6733	-79.05	kd	CGS001-1362	CPD	Carboxypeptidase A			
6734	-79.07	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
6735	-79.09	cp	BRD-A56892734	esomeprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
6736	-79.12	oe	ccsbBroad304_01401	RIT1	-			
6737	-79.13	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
6738	-79.13	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
6739	-79.15	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6740	-79.16	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6741	-79.2	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
6742	-79.2	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
6743	-79.2	kd	CGS001-283450	C12ORF51	-			
6744	-79.24	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
6745	-79.25	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
6746	-79.26	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6747	-79.27	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
6748	-79.28	oe	ccsbBroad304_00063	AMPD2	-			
6749	-79.3	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
6750	-79.35	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
6751	-79.35	oe	ccsbBroad304_03056	MCTS1	-			
6752	-79.35	cp	BRD-K84566043	fenpiverinium	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6753	-79.42	kd	CGS001-3417	IDH1	-			
6754	-79.47	kd	CGS001-3925	STMN1	-			
6755	-79.48	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
6756	-79.48	kd	CGS001-3376	IARS	Aminoacyl tRNA synthetases / Class I			
6757	-79.52	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
6758	-79.56	oe	ccsbBroad304_02402	TMEM5	-			
6759	-79.56	kd	CGS001-6713	SQLE	Lanosterol biosynthesis pathway			
6760	-79.57	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
6761	-79.57	kd	CGS001-2130	EWSR1	RNA binding motif (RRM) containing			
6762	-79.58	kd	CGS001-4801	NFYB	-			
6763	-79.63	kd	CGS001-216	ALDH1A1	Aldehyde dehydrogenases			
6764	-79.65	kd	CGS001-2542	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
6765	-79.66	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
6766	-79.66	kd	CGS001-79796	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
6767	-79.69	kd	CGS001-95	ACY1	-			
6768	-79.71	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
6769	-79.73	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
6770	-79.73	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
6771	-79.74	cp	BRD-K97752965	nicorandil	Nitric oxide donor		ABCC9, KCNJ11, KCNJ8	Nitric oxide donor, Potassium channel activator
6772	-79.75	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
6773	-79.77	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
6774	-79.77	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
6775	-79.79	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
6776	-79.86	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
6777	-79.88	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6778	-79.94	kd	CGS001-80150	ASRGL1	-			
6779	-79.95	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
6780	-79.98	kd	CGS001-7534	YWHAZ	-			
6781	-80.01	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
6782	-80.01	kd	CGS001-25819	CCRN4L	-			
6783	-80.07	oe	ccsbBroad304_03604	ENOSF1	-			
6784	-80.1	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
6785	-80.11	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
6786	-80.11	kd	CGS001-10059	DNM1L	-			
6787	-80.11	kd	CGS001-5257	PHKB	-			
6788	-80.2	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
6789	-80.21	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
6790	-80.23	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6791	-80.28	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
6792	-80.3	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
6793	-80.33	oe	ccsbBroad304_03848	METTL14	-			
6794	-80.35	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
6795	-80.35	kd	CGS001-1737	DLAT	-			
6796	-80.37	kd	CGS001-23566	LPAR3	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6797	-80.38	oe	ccsbBroad304_00529	F3	CD molecules			
6798	-80.38	oe	ccsbBroad304_02837	BHMT2	-			
6799	-80.38	kd	CGS001-256364	EML3	WD repeat domain containing			
6800	-80.39	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
6801	-80.39	kd	CGS001-54861	SNRK	SNRK subfamily			
6802	-80.41	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6803	-80.42	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
6804	-80.45	kd	CGS001-344	APOC2	Apolipoproteins			
6805	-80.47	kd	CGS001-7415	VCP	ATPases / AAA-type			
6806	-80.48	kd	CGS001-1287	COL4A5	Collagens			
6807	-80.5	kd	CGS001-8764	TNFRSF14	Tumour necrosis factor (TNF) receptor family			
6808	-80.51	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
6809	-80.52	kd	CGS001-64376	IKZF5	IKAROS zinc fingers			
6810	-80.56	kd	CGS001-64710	NUCKS1	-			
6811	-80.57	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
6812	-80.61	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
6813	-80.62	cp	BRD-K85925969	zalcitabine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
6814	-80.62	kd	CGS001-327	APEH	Prolyl oligopeptidase			
6815	-80.65	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
6816	-80.66	oe	ccsbBroad304_10431	HADHB	-			
6817	-80.66	kd	CGS001-8270	LAGE3	-			
6818	-80.67	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6819	-80.7	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
6820	-80.7	kd	CGS001-26523	EIF2C1	-			
6821	-80.71	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
6822	-80.72	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
6823	-80.76	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6824	-80.77	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
6825	-80.81	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
6826	-80.84	oe	ccsbBroad304_02157	MED21	-			
6827	-80.84	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
6828	-80.88	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
6829	-80.94	oe	ccsbBroad304_08596	EAPP	-			
6830	-80.94	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
6831	-80.94	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
6832	-80.96	kd	CGS001-5063	PAK3	PAKA subfamily			
6833	-80.97	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
6834	-80.98	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6835	-81.03	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
6836	-81.04	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6837	-81.09	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
6838	-81.13	kd	CGS001-81621	KAZALD1	Immunoglobulin superfamily / I-set domain containing			
6839	-81.13	kd	CGS001-3669	ISG20	-			
6840	-81.14	kd	CGS001-415116	PIM3	PIM family			
6841	-81.17	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6842	-81.17	kd	CGS001-4193	MDM2	-			
6843	-81.19	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
6844	-81.19	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
6845	-81.2	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
6846	-81.21	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
6847	-81.25	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
6848	-81.26	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6849	-81.29	oe	ccsbBroad304_08386	SMOX	-			
6850	-81.35	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
6851	-81.35	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
6852	-81.39	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
6853	-81.42	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
6854	-81.45	kd	CGS001-84433	CARD11	-			
6855	-81.46	kd	CGS001-7082	TJP1	-			
6856	-81.48	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
6857	-81.56	oe	ccsbBroad304_05756	ACAA1	-			
6858	-81.56	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
6859	-81.61	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
6860	-81.61	kd	CGS001-5805	PTS	-			
6861	-81.65	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
6862	-81.66	oe	ccsbBroad304_01560	SNAPC1	-			
6863	-81.66	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
6864	-81.71	kd	CGS001-29911	HOOK2	-			
6865	-81.73	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
6866	-81.74	oe	ccsbBroad304_00564	FGR	Src family			
6867	-81.74	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
6868	-81.75	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
6869	-81.77	cp	BRD-K86003836	flubendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
6870	-81.79	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
6871	-81.8	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6872	-81.82	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
6873	-81.83	cc		Aromatase inhibitor	-			
6874	-81.84	kd	CGS001-8942	KYNU	-			
6875	-81.86	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
6876	-81.89	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
6877	-81.9	oe	ccsbBroad304_04294	ATG10	-			
6878	-81.91	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
6879	-81.92	oe	ccsbBroad304_07600	NSA2	-			
6880	-81.93	kd	CGS001-10013	HDAC6	Histone deacetylases			
6881	-81.94	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
6882	-81.95	kd	CGS001-629	CFB	Complement system			
6883	-82	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
6884	-82	kd	CGS001-9429	ABCG2	ATP binding cassette transporters / subfamily G			
6885	-82.02	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
6886	-82.02	kd	CGS001-5294	PIK3CG	Phosphatidylinositol kinases			
6887	-82.14	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6888	-82.14	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
6889	-82.15	oe	ccsbBroad304_07834	GGA2	-			
6890	-82.18	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
6891	-82.18	kd	CGS001-2335	FN1	Endogenous ligands			
6892	-82.19	kd	CGS001-57192	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
6893	-82.2	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
6894	-82.22	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
6895	-82.28	kd	CGS001-4234	METTL1	-			
6896	-82.28	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
6897	-82.31	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
6898	-82.41	cp	BRD-K41903098	diphenoxylate	Opioid receptor agonist		OPRM1, OPRD1	Opioid receptor agonist
6899	-82.41	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
6900	-82.45	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
6901	-82.46	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
6902	-82.46	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
6903	-82.49	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
6904	-82.49	kd	CGS001-4718	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
6905	-82.52	kd	CGS001-375449	MAST4	MAST family			
6906	-82.54	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
6907	-82.55	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
6908	-82.57	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
6909	-82.58	oe	ccsbBroad304_01624	SUPV3L1	-			
6910	-82.63	oe	ccsbBroad304_06255	LRRC32	-			
6911	-82.64	kd	CGS001-883	CCBL1	Hydrogen sulphide synthesis			
6912	-82.65	oe	ccsbBroad304_00961	SMAD2	SMADs			
6913	-82.65	kd	CGS001-5479	PPIB	-			
6914	-82.66	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6915	-82.7	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
6916	-82.75	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
6917	-82.77	kd	CGS001-4205	MEF2A	Myocyte enhancer factors			
6918	-82.78	oe	ccsbBroad304_03386	SPA17	-			
6919	-82.78	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
6920	-82.81	kd	CGS001-5921	RASA1	Pleckstrin homology (PH) domain containing			
6921	-82.82	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
6922	-82.85	kd	CGS001-4012	LNPEP	Aminopeptidase N			
6923	-82.94	oe	ccsbBroad304_00316	CKS1B	-			
6924	-82.95	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
6925	-82.97	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6926	-82.98	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
6927	-83.01	oe	ccsbBroad304_07145	ZFP161	-			
6928	-83.01	kd	CGS001-50943	FOXP3	Forkhead boxes			
6929	-83.02	kd	CGS001-9441	MED26	-			
6930	-83.02	kd	CGS001-558	AXL	Fibronectin type III domain containing			
6931	-83.05	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
6932	-83.06	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6933	-83.08	kd	CGS001-55193	PBRM1	Non-enzymatic BRD containing proteins			
6934	-83.09	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
6935	-83.09	kd	CGS001-5627	PROS1	-			
6936	-83.1	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
6937	-83.14	kd	CGS001-93349	SP140L	Zinc fingers, PHD-type			
6938	-83.14	kd	CGS001-51727	CMPK1	-			
6939	-83.15	oe	ccsbBroad304_02604	B3GNT1	-			
6940	-83.15	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
6941	-83.15	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
6942	-83.15	kd	CGS001-10755	GIPC1	-			
6943	-83.18	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
6944	-83.22	oe	ccsbBroad304_02789	ADAT1	-			
6945	-83.22	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
6946	-83.25	kd	CGS001-55278	QRSL1	-			
6947	-83.28	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
6948	-83.31	kd	CGS001-1950	EGF	-			
6949	-83.41	kd	CGS001-7054	TH	Amino acid hydroxylases			
6950	-83.43	kd	CGS001-3672	ITGA1	Integrins			
6951	-83.45	kd	CGS001-3827	KNG1	Endogenous ligands			
6952	-83.48	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
6953	-83.51	kd	CGS001-3034	HAL	-			
6954	-83.53	cp	BRD-K83144676	olmesartan	Angiotensin antagonist		AGTR1	Angiotensin antagonist
6955	-83.54	kd	CGS001-1856	DVL2	Dishevelled homologs			
6956	-83.57	cp	BRD-A96107863	nisoldipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNB2, CYP3A5	Calcium channel blocker
6957	-83.6	kd	CGS001-1820	ARID3A	-			
6958	-83.61	oe	ccsbBroad304_00210	CALR	-			
6959	-83.64	cp	BRD-K44094599	tacrolimus	Calcineurin inhibitor		FKBP1A, CYP3A5, CYP3A7	Calcineurin inhibitor
6960	-83.65	oe	ccsbBroad304_06952	SKP1	-			
6961	-83.66	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
6962	-83.66	kd	CGS001-1070	CETN3	EF-hand domain containing			
6963	-83.7	kd	CGS001-51070	NOSIP	-			
6964	-83.72	kd	CGS001-200734	SPRED2	-			
6965	-83.76	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
6966	-83.77	oe	ccsbBroad304_10240	CROT	-			
6967	-83.78	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
6968	-83.78	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
6969	-83.79	oe	ccsbBroad304_00171	BNIP3L	-			
6970	-83.8	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
6971	-83.8	kd	CGS001-2746	GLUD1	-			
6972	-83.81	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
6973	-83.87	kd	CGS001-509	ATP5C1	ATPases / F-type			
6974	-83.88	kd	CGS001-262	AMD1	Decarboxylases			
6975	-83.91	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
6976	-83.93	oe	ccsbBroad304_08879	CASD1	-			
6977	-83.93	cp	BRD-K51485625	ritonavir	HIV protease inhibitor		CYP3A4, CYP1A2, CYP2B6, CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
6978	-83.93	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
6979	-83.97	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
6980	-83.97	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
6981	-83.97	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6982	-83.98	kd	CGS001-55818	KDM3A	Histone demethylases			
6983	-83.99	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
6984	-84	kd	CGS001-9375	TM9SF2	-			
6985	-84.02	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
6986	-84.05	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
6987	-84.1	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
6988	-84.13	oe	ccsbBroad304_00033	ADSS	-			
6989	-84.13	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
6990	-84.19	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
6991	-84.19	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
6992	-84.21	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
6993	-84.21	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
6994	-84.22	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
6995	-84.23	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
6996	-84.23	kd	CGS001-7528	YY1	INO80 complex subunits			
6997	-84.25	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
6998	-84.26	kd	CGS001-847	CAT	-			
6999	-84.28	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
7000	-84.3	oe	ccsbBroad304_09035	COASY	-			
7001	-84.31	cp	BRD-K66896231	BRD-K66896231	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
7002	-84.31	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
7003	-84.32	kd	CGS001-5696	PSMB8	Proteasome (prosome, macropain) subunits			
7004	-84.33	kd	CGS001-638	BIK	-			
7005	-84.34	oe	ccsbBroad304_01716	TSN	-			
7006	-84.34	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
7007	-84.35	oe	ccsbBroad304_06095	DFFB	-			
7008	-84.37	kd	CGS001-648	BMI1	Polycomb group ring fingers			
7009	-84.37	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
7010	-84.39	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
7011	-84.39	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
7012	-84.4	cp	BRD-A11990600	lorazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, TSPO	Benzodiazepine receptor agonist
7013	-84.41	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
7014	-84.45	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
7015	-84.45	kd	CGS001-9955	HS3ST3A1	Sulfotransferases, membrane-bound			
7016	-84.46	oe	ccsbBroad304_03119	C16ORF5	-			
7017	-84.53	oe	ccsbBroad304_06226	FTL	-			
7018	-84.59	oe	ccsbBroad304_03853	LSM2	-			
7019	-84.6	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
7020	-84.6	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
7021	-84.61	kd	CGS001-4072	EPCAM	CD molecules			
7022	-84.61	kd	CGS001-527	ATP6V0C	ATPases / V-type			
7023	-84.62	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
7024	-84.62	kd	CGS001-22818	COPZ1	-			
7025	-84.66	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
7026	-84.69	cp	BRD-K59753975	vindesine	Tubulin inhibitor		TUBB, TUBB1	Tubulin inhibitor
7027	-84.69	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
7028	-84.72	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
7029	-84.73	kd	CGS001-6199	RPS6KB2	p70 subfamily			
7030	-84.79	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
7031	-84.8	kd	CGS001-1545	CYP1B1	Cytochrome P450s			
7032	-84.8	kd	CGS001-353	APRT	-			
7033	-84.85	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
7034	-84.87	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
7035	-84.88	kd	CGS001-10857	PGRMC1	-			
7036	-84.9	kd	CGS001-6927	HNF1A	Homeoboxes / HNF class			
7037	-84.91	oe	ccsbBroad304_06126	TSC22D3	-			
7038	-84.91	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
7039	-84.92	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
7040	-84.92	kd	CGS001-1062	CENPE	Kinesins			
7041	-84.93	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
7042	-84.94	kd	CGS001-1390	CREM	basic leucine zipper proteins			
7043	-84.94	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
7044	-84.97	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
7045	-84.98	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
7046	-85	kd	CGS001-5918	RARRES1	-			
7047	-85.03	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
7048	-85.05	kd	CGS001-9475	ROCK2	Pleckstrin homology (PH) domain containing			
7049	-85.08	oe	ccsbBroad304_01372	RALB	-			
7050	-85.1	oe	ccsbBroad304_01951	BLZF1	-			
7051	-85.11	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
7052	-85.13	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
7053	-85.14	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
7054	-85.14	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
7055	-85.15	oe	ccsbBroad304_00054	ALDOC	-			
7056	-85.18	oe	ccsbBroad304_00817	IDH2	-			
7057	-85.19	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
7058	-85.19	kd	CGS001-55239	OGFOD1	-			
7059	-85.23	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
7060	-85.23	oe	ccsbBroad304_01976	EIF4EBP3	-			
7061	-85.24	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
7062	-85.26	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
7063	-85.27	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
7064	-85.27	kd	CGS001-5578	PRKCA	Delta subfamily			
7065	-85.31	oe	ccsbBroad304_00747	HLF	-			
7066	-85.31	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
7067	-85.31	kd	CGS001-6272	SORT1	-			
7068	-85.35	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7069	-85.36	cc		S100 calcium binding proteins LOF	-			
7070	-85.37	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
7071	-85.37	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
7072	-85.38	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
7073	-85.38	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7074	-85.4	kd	CGS001-6194	RPS6	S ribosomal proteins			
7075	-85.41	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
7076	-85.42	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
7077	-85.43	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
7078	-85.43	kd	CGS001-6774	STAT3	SH2 domain containing			
7079	-85.44	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
7080	-85.45	oe	ccsbBroad304_08694	TBX20	T-boxes			
7081	-85.46	kd	CGS001-24140	FTSJ1	-			
7082	-85.47	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
7083	-85.49	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
7084	-85.5	cp	BRD-K93618743	ipriflavone	Bone resorption inhibitor			Bone resorption inhibitor
7085	-85.5	kd	CGS001-27034	ACAD8	-			
7086	-85.55	oe	ccsbBroad304_04202	MED28	-			
7087	-85.55	kd	CGS001-462	SERPINC1	Serine (or cysteine) peptidase inhibitors			
7088	-85.67	kd	CGS001-3615	IMPDH2	Oxidoreductases			
7089	-85.71	kd	CGS001-11151	CORO1A	Coronins			
7090	-85.74	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
7091	-85.75	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
7092	-85.75	kd	CGS001-1213	CLTC	-			
7093	-85.76	cc		Beta-adrenergic receptor agonist	-			
7094	-85.78	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
7095	-85.78	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
7096	-85.84	kd	CGS001-7541	ZFP161	-			
7097	-85.84	kd	CGS001-55907	CMAS	-			
7098	-85.85	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
7099	-85.88	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
7100	-85.89	kd	CGS001-57057	TBX20	T-boxes			
7101	-85.91	cc		Phospholipases GOF	-			
7102	-85.91	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
7103	-85.93	kd	CGS001-5979	RET	Type XIV RTKs: RET			
7104	-85.94	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
7105	-85.95	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
7106	-85.96	cp	BRD-K63343048	orlistat	Lipase inhibitor		PNLIP, DAGLA, FASN, LIPF, CNR1, DAGLB	Lipase inhibitor
7107	-85.99	kd	CGS001-7693	ZNF134	Zinc fingers, C2H2-type			
7108	-86	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
7109	-86.03	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
7110	-86.03	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
7111	-86.06	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
7112	-86.06	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
7113	-86.08	kd	CGS001-2793	GNGT2	-			
7114	-86.1	cp	BRD-K70358946	aripiprazole	Serotonin receptor agonist		DRD2, HTR1A, HTR2A, HRH1, HTR1B, HTR1D, HTR2C, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR1E, HTR3A, HTR6, HTR7	Serotonin receptor agonist, Serotonin receptor antagonist
7115	-86.13	oe	ccsbBroad304_03732	NPDC1	-			
7116	-86.13	kd	CGS001-129685	TAF8	-			
7117	-86.16	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
7118	-86.16	kd	CGS001-23252	OTUD3	OTU domain containing			
7119	-86.17	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
7120	-86.17	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
7121	-86.18	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
7122	-86.2	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
7123	-86.21	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
7124	-86.22	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
7125	-86.27	kd	CGS001-8826	IQGAP1	-			
7126	-86.28	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
7127	-86.29	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
7128	-86.29	kd	CGS001-54584	GNB1L	WD repeat domain containing			
7129	-86.35	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
7130	-86.51	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
7131	-86.54	oe	ccsbBroad304_06040	CRY1	-			
7132	-86.64	kd	CGS001-9632	SEC24C	-			
7133	-86.65	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
7134	-86.67	kd	CGS001-3945	LDHB	-			
7135	-86.7	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
7136	-86.72	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
7137	-86.85	cp	BRD-K82109576	vincristine	Tubulin inhibitor		TUBB, TUBA4A	Tubulin inhibitor
7138	-86.89	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
7139	-86.93	kd	CGS001-1111	CHEK1	CHK1 subfamily			
7140	-86.94	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7141	-86.97	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
7142	-86.98	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
7143	-87.03	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
7144	-87.1	kd	CGS001-2100	ESR2	Estrogen receptors			
7145	-87.14	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
7146	-87.15	kd	CGS001-51282	SCAND1	-			
7147	-87.15	kd	CGS001-56005	C19ORF10	-			
7148	-87.19	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
7149	-87.2	oe	ccsbBroad304_03544	FAIM	-			
7150	-87.21	kd	CGS001-3755	KCNG1	Voltage-gated potassium channels			
7151	-87.23	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
7152	-87.28	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
7153	-87.28	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
7154	-87.29	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
7155	-87.3	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
7156	-87.32	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
7157	-87.36	kd	CGS001-5933	RBL1	-			
7158	-87.39	cc		Cannabinoid receptor agonist	-			
7159	-87.43	kd	CGS001-221188	GPR114	Adhesion Class GPCRs			
7160	-87.43	kd	CGS001-111	ADCY5	Adenylate cyclases			
7161	-87.46	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
7162	-87.46	kd	CGS001-5970	RELA	NFkappaB transcription factor family			
7163	-87.48	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
7164	-87.49	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
7165	-87.56	kd	CGS001-4173	MCM4	-			
7166	-87.56	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
7167	-87.58	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
7168	-87.59	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
7169	-87.59	oe	ccsbBroad304_00085	APRT	-			
7170	-87.61	kd	CGS001-5927	KDM5A	Histone demethylases			
7171	-87.66	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
7172	-87.68	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
7173	-87.7	oe	ccsbBroad304_06013	CLPTM1	-			
7174	-87.7	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
7175	-87.71	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
7176	-87.72	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
7177	-87.74	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
7178	-87.76	kd	CGS001-5693	PSMB5	Proteasome subunits			
7179	-87.82	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
7180	-87.85	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
7181	-87.89	cp	BRD-K49404994	levetiracetam	Calcium channel blocker		SV2A, CACNA1B, SCN1A	Calcium channel blocker
7182	-87.96	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
7183	-88	cp	BRD-A24543851	nornicotine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
7184	-88.01	kd	CGS001-3612	IMPA1	Inositol monophosphatase			
7185	-88.04	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
7186	-88.05	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
7187	-88.1	kd	CGS001-8022	LHX3	Homeoboxes / LIM class			
7188	-88.13	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7189	-88.16	kd	CGS001-5236	PGM1	-			
7190	-88.19	cc		GABA receptor antagonist	-			
7191	-88.19	kd	CGS001-55423	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
7192	-88.23	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7193	-88.24	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
7194	-88.26	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
7195	-88.28	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
7196	-88.3	oe	ccsbBroad304_01139	PA2G4	-			
7197	-88.3	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
7198	-88.31	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
7199	-88.34	oe	ccsbBroad304_02509	GMEB1	-			
7200	-88.35	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
7201	-88.35	kd	CGS001-47	ACLY	-			
7202	-88.35	oe	ccsbBroad304_07820	SNW1	-			
7203	-88.36	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
7204	-88.38	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
7205	-88.38	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
7206	-88.39	cc		Estrogen receptor agonist	-			
7207	-88.39	kd	CGS001-56834	GPR137	GPCR / Unclassified : 7TM orphan receptors			
7208	-88.4	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
7209	-88.42	kd	CGS001-2597	GAPDH	-			
7210	-88.46	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
7211	-88.46	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
7212	-88.49	cc		X linked mental retardation group 1 LOF	-			
7213	-88.49	kd	CGS001-336	APOA2	Apolipoproteins			
7214	-88.52	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
7215	-88.55	kd	CGS001-7484	WNT9B	Wingless-type MMTV integration sites			
7216	-88.57	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
7217	-88.59	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
7218	-88.6	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
7219	-88.62	oe	ccsbBroad304_01659	TERF1	-			
7220	-88.64	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
7221	-88.65	cp	BRD-K62858456	lomerizine	Calcium channel blocker		ABCB1, CACNA1B, SCN5A	Calcium channel blocker
7222	-88.68	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
7223	-88.74	oe	ccsbBroad304_08217	SCCPDH	-			
7224	-88.78	kd	CGS001-4303	FOXO4	Forkhead boxes			
7225	-88.8	kd	CGS001-51271	UBAP1	-			
7226	-88.82	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
7227	-88.83	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
7228	-88.83	kd	CGS001-5228	PGF	-			
7229	-88.93	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
7230	-88.94	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
7231	-88.94	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
7232	-88.94	kd	CGS001-19	ABCA1	ATP binding cassette transporters / subfamily A			
7233	-88.96	cc		P38 MAPK inhibitor	-			
7234	-89	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
7235	-89	kd	CGS001-84875	PARP10	Poly (ADP-ribose) polymerases			
7236	-89.01	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
7237	-89.06	kd	CGS001-10691	GMEB1	-			
7238	-89.07	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
7239	-89.08	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
7240	-89.09	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
7241	-89.12	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
7242	-89.15	kd	CGS001-5688	PSMA7	Proteasome subunits			
7243	-89.16	kd	CGS001-94239	H2AFV	Histones / Replication-independent			
7244	-89.17	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
7245	-89.19	kd	CGS001-5708	PSMD2	Proteasome subunits			
7246	-89.19	kd	CGS001-4916	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
7247	-89.22	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
7248	-89.22	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
7249	-89.24	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
7250	-89.25	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
7251	-89.25	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
7252	-89.27	kd	CGS001-50	ACO2	-			
7253	-89.34	kd	CGS001-25987	TSKU	-			
7254	-89.38	kd	CGS001-6894	TARBP1	-			
7255	-89.39	cp	BRD-K48932581	cetraxate	Mucus protecting agent		GAST	Mucus protecting agent
7256	-89.39	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
7257	-89.41	kd	CGS001-150094	SIK1	QIK subfamily			
7258	-89.42	kd	CGS001-25825	BACE2	Pepsin			
7259	-89.43	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
7260	-89.44	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
7261	-89.47	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
7262	-89.48	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
7263	-89.49	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
7264	-89.5	kd	CGS001-8464	SUPT3H	-			
7265	-89.51	kd	CGS001-3992	FADS1	Fatty acid desaturases			
7266	-89.51	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
7267	-89.52	cp	BRD-A64297288	amlodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, ABCG2, CA1, CACNA1B, CACNA1S, CACNA2D3, CACNB1, CACNB2, SMPD1	Calcium channel blocker
7268	-89.52	kd	CGS001-10247	HRSP12	-			
7269	-89.55	cc		Ubiquitin-specific peptidases LOF	-			
7270	-89.55	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
7271	-89.58	oe	ccsbBroad304_00420	DAP	-			
7272	-89.58	kd	CGS001-8651	SOCS1	SH2 domain containing			
7273	-89.59	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
7274	-89.6	kd	CGS001-3609	ILF3	-			
7275	-89.62	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
7276	-89.63	kd	CGS001-3985	LIMK2	LIMK subfamily			
7277	-89.64	oe	ccsbBroad304_08045	NOX1	-			
7278	-89.65	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
7279	-89.66	oe	ccsbBroad304_02138	TRIP10	-			
7280	-89.66	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
7281	-89.67	oe	ccsbBroad304_03773	CIAPIN1	-			
7282	-89.67	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
7283	-89.68	oe	ccsbBroad304_02677	PDAP1	-			
7284	-89.68	kd	CGS001-1452	CSNK1A1	Casein kinase 1 (CK1) family			
7285	-89.69	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
7286	-89.74	oe	ccsbBroad304_01105	PNP	-			
7287	-89.76	oe	ccsbBroad304_04786	CANT1	-			
7288	-89.76	kd	CGS001-84923	FAM104A	-			
7289	-89.81	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
7290	-89.83	oe	ccsbBroad304_09578	PASD1	-			
7291	-89.84	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
7292	-89.86	oe	ccsbBroad304_03479	YTHDF1	-			
7293	-89.86	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
7294	-89.91	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
7295	-89.92	oe	ccsbBroad304_00492	EIF5A	-			
7296	-89.92	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
7297	-89.93	kd	CGS001-3030	HADHA	-			
7298	-89.94	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
7299	-89.95	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
7300	-89.97	oe	ccsbBroad304_01150	PCCB	Carboxylases			
7301	-89.99	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
7302	-90.05	kd	CGS001-9275	BCL7B	-			
7303	-90.07	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
7304	-90.13	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
7305	-90.14	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
7306	-90.15	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
7307	-90.16	kd	CGS001-2524	FUT2	Fucosyltransferases			
7308	-90.17	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
7309	-90.18	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
7310	-90.18	kd	CGS001-51460	SFMBT1	Sterile alpha motif (SAM) domain containing			
7311	-90.19	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
7312	-90.2	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
7313	-90.2	oe	ccsbBroad304_07208	NRIP1	-			
7314	-90.21	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
7315	-90.25	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
7316	-90.26	kd	CGS001-169841	ZNF169	Zinc fingers, C2H2-type			
7317	-90.29	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
7318	-90.39	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
7319	-90.41	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
7320	-90.41	oe	ccsbBroad304_00098	ARG1	Arginase			
7321	-90.44	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
7322	-90.47	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
7323	-90.47	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
7324	-90.48	kd	CGS001-79174	CRELD2	-			
7325	-90.48	kd	CGS001-7132	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
7326	-90.5	cc		Interleukin receptors LOF	-			
7327	-90.51	oe	ccsbBroad304_14020	SH3BP5	-			
7328	-90.51	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
7329	-90.53	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
7330	-90.55	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
7331	-90.56	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
7332	-90.57	kd	CGS001-55699	IARS2	Aminoacyl tRNA synthetases / Class I			
7333	-90.59	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
7334	-90.59	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
7335	-90.61	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
7336	-90.61	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7337	-90.64	kd	CGS001-10078	TSSC4	-			
7338	-90.64	kd	CGS001-3691	ITGB4	Integrins			
7339	-90.65	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
7340	-90.65	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
7341	-90.74	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
7342	-90.74	oe	ccsbBroad304_06449	ILF3	-			
7343	-90.75	kd	CGS001-642	BLMH	-			
7344	-90.76	oe	ccsbBroad304_00645	GCLM	-			
7345	-90.76	kd	CGS001-7040	TGFB1	Endogenous ligands			
7346	-90.78	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
7347	-90.79	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
7348	-90.8	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
7349	-90.84	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
7350	-90.87	oe	ccsbBroad304_02668	PNKP	-			
7351	-90.9	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
7352	-90.9	oe	ccsbBroad304_00876	INSIG1	-			
7353	-90.92	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
7354	-90.94	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
7355	-90.96	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
7356	-90.96	kd	CGS001-1786	DNMT1	Methyltransferases			
7357	-90.98	kd	CGS001-10289	EIF1B	-			
7358	-90.98	kd	CGS001-55111	PLEKHJ1	Pleckstrin homology (PH) domain containing			
7359	-91	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
7360	-91.04	kd	CGS001-140690	CTCFL	Zinc fingers, C2H2-type			
7361	-91.08	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
7362	-91.11	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
7363	-91.11	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
7364	-91.16	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
7365	-91.16	kd	CGS001-6648	SOD2	-			
7366	-91.17	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
7367	-91.17	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
7368	-91.19	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
7369	-91.21	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
7370	-91.21	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
7371	-91.27	cc		Ribosomal 40s Subunit LOF	-			
7372	-91.27	cp	BRD-M41783010	acamprosate	Glutamate receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B, GRM5	Glutamate receptor antagonist
7373	-91.28	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
7374	-91.29	kd	CGS001-55127	HEATR1	-			
7375	-91.29	kd	CGS001-2776	GNAQ	-			
7376	-91.3	kd	CGS001-3309	HSPA5	Heat shock proteins / HSP70			
7377	-91.3	kd	CGS001-9568	GABBR2	GABA receptors			
7378	-91.3	kd	CGS001-64241	ABCG8	ATP binding cassette transporters / subfamily G			
7379	-91.32	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
7380	-91.37	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
7381	-91.38	oe	ccsbBroad304_07045	TEAD4	-			
7382	-91.42	oe	ccsbBroad304_01147	PC	Carboxylases			
7383	-91.42	oe	ccsbBroad304_08346	COQ3	-			
7384	-91.43	oe	ccsbBroad304_01605	SSX2	-			
7385	-91.43	kd	CGS001-6184	RPN1	-			
7386	-91.44	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
7387	-91.46	cc		Bromodomain Inhibitor	-			
7388	-91.47	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
7389	-91.49	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
7390	-91.51	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
7391	-91.54	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
7392	-91.56	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7393	-91.57	kd	CGS001-5950	RBP4	Lipocalins			
7394	-91.58	kd	CGS001-7465	WEE1	WEE family			
7395	-91.59	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
7396	-91.6	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
7397	-91.61	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
7398	-91.63	kd	CGS001-488	ATP2A2	Calcium-ATPases			
7399	-91.64	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
7400	-91.68	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
7401	-91.69	kd	CGS001-183	AGT	Endogenous ligands			
7402	-91.72	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
7403	-91.74	kd	CGS001-134288	TMEM174	-			
7404	-91.75	cc		Tubulin inhibitor	-			
7405	-91.76	oe	ccsbBroad304_00658	GNG5	-			
7406	-91.78	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
7407	-91.78	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
7408	-91.78	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
7409	-91.78	kd	CGS001-89765	RSPH1	-			
7410	-91.78	kd	CGS001-2615	LRRC32	-			
7411	-91.79	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
7412	-91.81	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
7413	-91.81	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
7414	-91.82	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
7415	-91.86	kd	CGS001-54851	ANKRD49	Ankyrin repeat domain containing			
7416	-91.88	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
7417	-91.92	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
7418	-91.95	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
7419	-91.95	kd	CGS001-51701	NLK	nmo subfamily			
7420	-91.96	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
7421	-92.02	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
7422	-92.02	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
7423	-92.03	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
7424	-92.06	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
7425	-92.06	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
7426	-92.09	kd	CGS001-2244	FGB	Endogenous ligands			
7427	-92.11	kd	CGS001-204	AK2	Adenylate kinases			
7428	-92.15	kd	CGS001-10962	MLLT11	-			
7429	-92.17	oe	ccsbBroad304_01769	VEGFB	-			
7430	-92.17	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
7431	-92.18	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
7432	-92.22	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
7433	-92.23	oe	ccsbBroad304_01395	RFX5	-			
7434	-92.24	cp	BRD-K90733503	cefalexin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7435	-92.25	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
7436	-92.25	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
7437	-92.27	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
7438	-92.29	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
7439	-92.29	kd	CGS001-375346	TMEM110	-			
7440	-92.3	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
7441	-92.31	kd	CGS001-7936	RDBP	-			
7442	-92.31	kd	CGS001-55509	BATF3	basic leucine zipper proteins			
7443	-92.32	cp	BRD-K73991644	isoquercetin	Aldose reductase inhibitor		AKR1B1, ACE	Aldose reductase inhibitor
7444	-92.33	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
7445	-92.34	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
7446	-92.36	oe	ccsbBroad304_07766	RASSF1	-			
7447	-92.37	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
7448	-92.38	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
7449	-92.38	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
7450	-92.39	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
7451	-92.4	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
7452	-92.43	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
7453	-92.46	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
7454	-92.46	kd	CGS001-22944	KIN	-			
7455	-92.48	cp	BRD-K06878038	deferiprone	Chelating agent		CYP4F2	Chelating agent
7456	-92.48	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
7457	-92.48	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
7458	-92.49	kd	CGS001-10919	EHMT2	Histone methyltransferases			
7459	-92.57	cc		Calcium channel blocker	-			
7460	-92.57	cp	BRD-K53220666	trimetozine	Sedative			Sedative
7461	-92.61	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
7462	-92.64	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
7463	-92.64	kd	CGS001-8317	CDC7	CDC7 family			
7464	-92.65	oe	ccsbBroad304_01347	RAD1	-			
7465	-92.66	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
7466	-92.66	kd	CGS001-54677	CROT	-			
7467	-92.69	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
7468	-92.72	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
7469	-92.72	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
7470	-92.74	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
7471	-92.75	kd	CGS001-5898	RALA	-			
7472	-92.76	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
7473	-92.77	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
7474	-92.77	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
7475	-92.77	kd	CGS001-5610	EIF2AK2	Other PEK family kinases			
7476	-92.79	oe	ccsbBroad304_07632	PROCR	CD molecules			
7477	-92.8	oe	ccsbBroad304_07754	FGFR1OP	-			
7478	-92.81	oe	ccsbBroad304_07616	ZNF238	-			
7479	-92.82	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
7480	-92.82	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
7481	-92.83	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
7482	-92.84	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
7483	-92.86	kd	CGS001-53343	NUDT9	Nudix motif containing			
7484	-92.87	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
7485	-92.92	kd	CGS001-9	NAT1	-			
7486	-92.94	kd	CGS001-6670	SP3	Specificity protein transcription factors			
7487	-92.98	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
7488	-93	oe	ccsbBroad304_00883	ISG20	-			
7489	-93	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
7490	-93.03	oe	ccsbBroad304_00390	CTGF	-			
7491	-93.03	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
7492	-93.04	oe	ccsbBroad304_06424	IFI16	-			
7493	-93.04	kd	CGS001-539	ATP5O	ATPases / F-type			
7494	-93.05	oe	ccsbBroad304_10212	GRHL3	-			
7495	-93.07	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
7496	-93.08	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
7497	-93.08	kd	CGS001-39	ACAT2	Lanosterol biosynthesis pathway			
7498	-93.09	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
7499	-93.1	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
7500	-93.13	kd	CGS001-6926	TBX3	T-boxes			
7501	-93.15	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
7502	-93.15	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
7503	-93.15	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
7504	-93.15	kd	CGS001-8801	SUCLG2	-			
7505	-93.15	kd	CGS001-3559	IL2RA	IL-2 receptor family			
7506	-93.15	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7507	-93.16	kd	CGS001-54658	UGT1A1	UDP glucuronosyltransferases			
7508	-93.17	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
7509	-93.17	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
7510	-93.19	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
7511	-93.2	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
7512	-93.21	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
7513	-93.23	kd	CGS001-3980	LIG3	-			
7514	-93.25	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
7515	-93.28	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
7516	-93.29	kd	CGS001-10975	UQCR11	Mitochondrial respiratory chain complex / Complex III			
7517	-93.3	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
7518	-93.32	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
7519	-93.32	kd	CGS001-2944	GSTM1	Glutathione S-transferases / Soluble			
7520	-93.33	cp	BRD-K49481516	galantamine	Acetylcholinesterase inhibitor		ACHE, BCHE, CHRNA1, CHRNA10, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNA9, CHRNB1, CHRNB2, CHRNB3, CHRNB4, CHRND, CHRNE, CHRNG	Acetylcholinesterase inhibitor
7521	-93.33	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
7522	-93.33	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
7523	-93.35	cp	BRD-K94649603	taxifolin	Opioid receptor antagonist		APOB, APP, HMGCR	Opioid receptor antagonist
7524	-93.38	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
7525	-93.38	kd	CGS001-965	CD58	CD molecules			
7526	-93.39	cc		Proteasome inhibitor	-			
7527	-93.42	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
7528	-93.42	kd	CGS001-3312	HSPA8	Heat shock proteins / HSP70			
7529	-93.44	kd	CGS001-1440	CSF3	Endogenous ligands			
7530	-93.46	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
7531	-93.47	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
7532	-93.47	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
7533	-93.48	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
7534	-93.55	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
7535	-93.56	kd	CGS001-6924	TCEB3	-			
7536	-93.57	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
7537	-93.58	kd	CGS001-6201	RPS7	S ribosomal proteins			
7538	-93.6	oe	ccsbBroad304_06518	LDHA	-			
7539	-93.6	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
7540	-93.61	kd	CGS001-5900	RALGDS	-			
7541	-93.63	kd	CGS001-6598	SMARCB1	-			
7542	-93.63	kd	CGS001-4953	ODC1	Decarboxylases			
7543	-93.63	kd	CGS001-230	ALDOC	-			
7544	-93.64	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
7545	-93.66	kd	CGS001-4637	MYL6	EF-hand domain containing			
7546	-93.67	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
7547	-93.67	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
7548	-93.68	kd	CGS001-6788	STK3	MST subfamily			
7549	-93.69	oe	ccsbBroad304_08452	PIH1D1	-			
7550	-93.7	kd	CGS001-34	ACADM	-			
7551	-93.71	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
7552	-93.74	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
7553	-93.75	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
7554	-93.78	kd	CGS001-7597	ZBTB25	BTB/POZ domain containing			
7555	-93.8	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
7556	-93.87	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
7557	-93.9	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
7558	-93.92	oe	ccsbBroad304_07320	SQSTM1	-			
7559	-93.97	cc		Heat shock 70kDa proteins LOF	-			
7560	-93.97	kd	CGS001-688	KLF5	Kruppel-like transcription factors			
7561	-93.98	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
7562	-94	oe	ccsbBroad304_01862	YEATS4	-			
7563	-94.02	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7564	-94.04	cc		HOXL subclass homeoboxes LOF	-			
7565	-94.04	oe	ccsbBroad304_02633	LSM6	-			
7566	-94.04	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
7567	-94.07	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
7568	-94.07	kd	CGS001-4830	NME1	-			
7569	-94.12	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
7570	-94.14	cp	BRD-K57930253	nitrazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, SCN1A	Benzodiazepine receptor agonist
7571	-94.14	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
7572	-94.17	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
7573	-94.19	oe	ccsbBroad304_06180	ESD	-			
7574	-94.19	kd	CGS001-9967	THRAP3	-			
7575	-94.25	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
7576	-94.29	kd	CGS001-823	CAPN1	EF-hand domain containing			
7577	-94.31	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
7578	-94.31	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
7579	-94.32	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
7580	-94.33	oe	ccsbBroad304_00486	EFNB2	Ephrins			
7581	-94.33	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
7582	-94.33	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
7583	-94.34	kd	CGS001-150962	PUS10	-			
7584	-94.35	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
7585	-94.35	kd	CGS001-10652	YKT6	-			
7586	-94.35	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
7587	-94.37	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
7588	-94.38	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
7589	-94.38	kd	CGS001-5073	PARN	-			
7590	-94.42	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
7591	-94.44	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
7592	-94.44	kd	CGS001-4204	MECP2	-			
7593	-94.46	kd	CGS001-8864	PER2	-			
7594	-94.52	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
7595	-94.54	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
7596	-94.55	kd	CGS001-5467	PPARD	Nuclear hormone receptors			
7597	-94.56	kd	CGS001-6233	RPS27A	S ribosomal proteins			
7598	-94.59	kd	CGS001-2021	ENDOG	-			
7599	-94.59	kd	CGS001-7832	BTG2	-			
7600	-94.59	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
7601	-94.61	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
7602	-94.64	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
7603	-94.67	kd	CGS001-1738	DLD	-			
7604	-94.68	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
7605	-94.7	cp	BRD-A92630576	trimebutine	Opioid receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Opioid receptor agonist
7606	-94.71	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
7607	-94.78	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
7608	-94.79	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
7609	-94.81	kd	CGS001-64333	ARHGAP9	Rho GTPase activating proteins			
7610	-94.82	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
7611	-94.82	oe	ccsbBroad304_03850	TRIB3	Trbl family			
7612	-94.83	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
7613	-94.83	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
7614	-94.84	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
7615	-94.86	oe	ccsbBroad304_06549	SMAD3	SMADs			
7616	-94.86	oe	ccsbBroad304_00515	ERH	-			
7617	-94.87	kd	CGS001-9817	KEAP1	Kelch-like proteins			
7618	-94.91	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
7619	-94.91	kd	CGS001-5053	PAH	Amino acid hydroxylases			
7620	-94.91	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
7621	-94.94	oe	ccsbBroad304_00661	GNGT2	-			
7622	-94.94	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
7623	-94.95	kd	CGS001-6472	SHMT2	-			
7624	-94.96	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
7625	-94.96	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
7626	-94.96	kd	CGS001-4938	OAS1	-			
7627	-94.96	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
7628	-94.97	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
7629	-95	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
7630	-95.01	kd	CGS001-2643	GCH1	-			
7631	-95.03	kd	CGS001-5914	RARA	Retinoic acid receptors			
7632	-95.04	kd	CGS001-6275	S100A4	EF-hand domain containing			
7633	-95.05	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
7634	-95.07	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
7635	-95.09	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
7636	-95.14	oe	ccsbBroad304_06888	RPN1	-			
7637	-95.14	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
7638	-95.14	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
7639	-95.14	kd	CGS001-2956	MSH6	-			
7640	-95.16	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
7641	-95.17	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
7642	-95.18	oe	ccsbBroad304_06290	GNA15	-			
7643	-95.18	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
7644	-95.24	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
7645	-95.24	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7646	-95.27	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7647	-95.27	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
7648	-95.27	cp	BRD-K34508425	KUC103898N	-666			-666
7649	-95.28	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
7650	-95.33	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
7651	-95.33	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
7652	-95.33	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
7653	-95.33	oe	ccsbBroad304_01654	TCTA	-			
7654	-95.36	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
7655	-95.36	kd	CGS001-10525	HYOU1	Heat shock proteins / HSP70			
7656	-95.38	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
7657	-95.38	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
7658	-95.42	kd	CGS001-8495	PPFIBP2	Sterile alpha motif (SAM) domain containing			
7659	-95.5	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
7660	-95.5	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
7661	-95.52	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
7662	-95.52	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
7663	-95.54	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
7664	-95.54	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
7665	-95.54	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
7666	-95.55	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
7667	-95.57	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
7668	-95.65	oe	ccsbBroad304_08840	KIF9	Kinesins			
7669	-95.65	oe	ccsbBroad304_04626	EGLN3	-			
7670	-95.65	kd	CGS001-9978	RBX1	RING-type (C3HC4) zinc fingers			
7671	-95.72	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
7672	-95.74	kd	CGS001-5292	PIM1	PIM family			
7673	-95.74	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
7674	-95.78	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
7675	-95.79	kd	CGS001-26574	AATF	-			
7676	-95.8	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
7677	-95.8	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
7678	-95.8	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
7679	-95.81	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
7680	-95.82	kd	CGS001-2771	GNAI2	-			
7681	-95.84	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
7682	-95.85	kd	CGS001-7248	TSC1	-			
7683	-95.85	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
7684	-95.86	kd	CGS001-29888	STRN4	WD repeat domain containing			
7685	-95.88	kd	CGS001-1874	E2F4	-			
7686	-95.9	kd	CGS001-6342	SCP2	-			
7687	-95.9	kd	CGS001-2353	FOS	basic leucine zipper proteins			
7688	-95.91	kd	CGS001-6794	STK11	LKB subfamily			
7689	-95.92	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
7690	-95.93	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
7691	-95.95	kd	CGS001-8408	ULK1	Unc-51-like kinase (ULK) family			
7692	-96	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
7693	-96	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
7694	-96	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
7695	-96	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
7696	-96.02	oe	ccsbBroad304_02788	PRAME	-			
7697	-96.02	oe	ccsbBroad304_02551	CPSF4	-			
7698	-96.02	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
7699	-96.03	kd	CGS001-55781	RIOK2	RIO2 subfamily			
7700	-96.04	kd	CGS001-84547	PGBD1	-			
7701	-96.09	cc		Benzodiazepine receptor agonist	-			
7702	-96.1	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
7703	-96.1	cp	BRD-A12560204	nitrendipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1H, CACNA1S, CACNA2D2, CACNB2, CACNG1, KCNN4	Calcium channel blocker
7704	-96.1	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
7705	-96.12	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
7706	-96.13	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
7707	-96.13	oe	ccsbBroad304_06172	EPS8	-			
7708	-96.14	kd	CGS001-7077	TIMP2	-			
7709	-96.15	cc		Wnt family LOF	-			
7710	-96.15	oe	ccsbBroad304_02002	RNMT	-			
7711	-96.16	kd	CGS001-51290	ERGIC2	-			
7712	-96.17	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
7713	-96.19	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
7714	-96.2	cp	BRD-K19462402	buflomedil	Adrenergic receptor antagonist		CACNA1C	Adrenergic receptor antagonist, Calcium channel blocker
7715	-96.2	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
7716	-96.22	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
7717	-96.22	kd	CGS001-6446	SGK1	SGK family			
7718	-96.23	kd	CGS001-23196	FAM120A	-			
7719	-96.25	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
7720	-96.27	kd	CGS001-3659	IRF1	-			
7721	-96.28	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
7722	-96.28	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
7723	-96.3	kd	CGS001-10972	TMED10	-			
7724	-96.31	kd	CGS001-3248	HPGD	Prostaglandin synthases			
7725	-96.32	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
7726	-96.33	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
7727	-96.34	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
7728	-96.34	kd	CGS001-1173	AP2M1	-			
7729	-96.37	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
7730	-96.37	oe	ccsbBroad304_03037	TMEM97	-			
7731	-96.38	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
7732	-96.39	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
7733	-96.39	cp	BRD-K82357231	desloratadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
7734	-96.4	kd	CGS001-5771	PTPN2	Protein tyrosine phosphatases			
7735	-96.4	kd	CGS001-5080	PAX6	Paired boxes			
7736	-96.41	kd	CGS001-23139	MAST2	MAST family			
7737	-96.42	cp	BRD-A48261811	argatroban	Thrombin inhibitor		F2, CYP3A5	Thrombin inhibitor
7738	-96.42	kd	CGS001-1725	DHPS	-			
7739	-96.43	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
7740	-96.44	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
7741	-96.45	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
7742	-96.5	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
7743	-96.5	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
7744	-96.52	cp	BRD-A87387433	cefpodoxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7745	-96.52	kd	CGS001-7358	UGDH	-			
7746	-96.55	oe	ccsbBroad304_04752	IKBIP	-			
7747	-96.55	kd	CGS001-6936	C2ORF3	-			
7748	-96.55	kd	CGS001-670	BPHL	-			
7749	-96.58	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
7750	-96.6	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
7751	-96.6	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
7752	-96.6	kd	CGS001-2153	F5	Blood coagulation components			
7753	-96.61	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
7754	-96.61	kd	CGS001-51805	COQ3	-			
7755	-96.63	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
7756	-96.64	cc		Tachykinin antagonist	-			
7757	-96.67	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
7758	-96.7	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7759	-96.71	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
7760	-96.71	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
7761	-96.72	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
7762	-96.72	kd	CGS001-25989	ULK3	Unc-51-like kinase (ULK) family			
7763	-96.75	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
7764	-96.76	kd	CGS001-6908	TBP	General transcription factors			
7765	-96.77	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
7766	-96.77	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
7767	-96.79	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
7768	-96.79	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7769	-96.82	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
7770	-96.82	kd	CGS001-7345	UCHL1	Ubiquitin C-terminal hydrolase			
7771	-96.83	kd	CGS001-1997	ELF1	ETS Transcription Factors			
7772	-96.85	kd	CGS001-4697	NDUFA4	-			
7773	-96.86	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
7774	-96.87	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
7775	-96.88	kd	CGS001-10284	SAP18	-			
7776	-96.89	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
7777	-96.9	kd	CGS001-8204	NRIP1	-			
7778	-96.93	kd	CGS001-10923	SUB1	-			
7779	-96.95	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
7780	-96.97	oe	ccsbBroad304_09821	TMEM154	-			
7781	-96.97	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
7782	-96.99	kd	CGS001-392	ARHGAP1	Rho GTPase activating proteins			
7783	-97.02	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
7784	-97.03	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
7785	-97.05	oe	ccsbBroad304_01641	TAF13	-			
7786	-97.06	kd	CGS001-10921	RNPS1	RNA binding motif (RRM) containing			
7787	-97.06	kd	CGS001-23077	MYCBP2	-			
7788	-97.07	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
7789	-97.07	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
7790	-97.07	oe	ccsbBroad304_03129	ERO1L	-			
7791	-97.07	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
7792	-97.09	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
7793	-97.11	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
7794	-97.11	oe	ccsbBroad304_00969	MAGEA10	-			
7795	-97.14	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
7796	-97.14	oe	ccsbBroad304_02292	BCL2L11	-			
7797	-97.15	kd	CGS001-23239	PHLPP1	Pleckstrin homology (PH) domain containing			
7798	-97.17	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
7799	-97.19	oe	ccsbBroad304_06008	AP2M1	-			
7800	-97.19	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
7801	-97.2	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
7802	-97.21	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
7803	-97.21	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
7804	-97.21	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
7805	-97.23	kd	CGS001-4707	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
7806	-97.28	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
7807	-97.28	kd	CGS001-1718	DHCR24	-			
7808	-97.29	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
7809	-97.31	oe	ccsbBroad304_06085	DCK	-			
7810	-97.35	oe	ccsbBroad304_06789	PSEN2	Presenilin			
7811	-97.36	kd	CGS001-51447	IP6K2	-			
7812	-97.37	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
7813	-97.38	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
7814	-97.4	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
7815	-97.4	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
7816	-97.4	kd	CGS001-23338	PHF15	-			
7817	-97.42	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
7818	-97.43	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
7819	-97.43	cp	BRD-K11630072	carmofur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
7820	-97.43	kd	CGS001-84328	LZIC	-			
7821	-97.45	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
7822	-97.46	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
7823	-97.46	kd	CGS001-27035	NOX1	-			
7824	-97.49	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
7825	-97.5	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
7826	-97.51	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
7827	-97.52	oe	ccsbBroad304_08137	HOOK2	-			
7828	-97.54	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
7829	-97.55	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
7830	-97.56	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
7831	-97.56	kd	CGS001-1892	ECHS1	-			
7832	-97.57	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
7833	-97.58	kd	CGS001-6611	SMS	-			
7834	-97.59	oe	ccsbBroad304_06916	SCP2	-			
7835	-97.6	kd	CGS001-51293	CD320	CD molecules			
7836	-97.63	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
7837	-97.66	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
7838	-97.7	kd	CGS001-29883	CNOT7	-			
7839	-97.72	oe	ccsbBroad304_07528	DMTF1	-			
7840	-97.73	kd	CGS001-58528	RRAGD	-			
7841	-97.77	oe	ccsbBroad304_03121	NRBF2	-			
7842	-97.78	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
7843	-97.78	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
7844	-97.79	kd	CGS001-6337	SCNN1A	Epithelial sodium channels (ENaC)			
7845	-97.8	cc		PPAR receptor agonist	-			
7846	-97.81	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
7847	-97.81	kd	CGS001-57787	MARK4	MARK subfamily			
7848	-97.82	oe	ccsbBroad304_02270	FAM20B	-			
7849	-97.87	oe	ccsbBroad304_05931	CAPG	-			
7850	-97.87	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
7851	-97.87	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
7852	-97.87	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
7853	-97.88	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
7854	-97.88	oe	ccsbBroad304_06159	CTTN	-			
7855	-97.89	kd	CGS001-5934	RBL2	-			
7856	-97.9	cc		Progesterone receptor antagonist	-			
7857	-97.9	kd	CGS001-55486	PARL	-			
7858	-97.92	kd	CGS001-115650	TNFRSF13C	Tumour necrosis factor (TNF) receptor family			
7859	-97.92	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
7860	-97.93	kd	CGS001-79711	IPO4	Importins			
7861	-97.94	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
7862	-97.98	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
7863	-97.98	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
7864	-97.98	kd	CGS001-5932	RBBP8	-			
7865	-97.99	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
7866	-97.99	kd	CGS001-375318	AQP12A	Ion channels / Aquaporins			
7867	-98.02	kd	CGS001-3551	IKBKB	IKK family			
7868	-98.03	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
7869	-98.04	oe	ccsbBroad304_04406	PLA2G12B	-			
7870	-98.05	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
7871	-98.05	kd	CGS001-6309	SC5DL	-			
7872	-98.06	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
7873	-98.06	kd	CGS001-143	PARP4	Poly (ADP-ribose) polymerases			
7874	-98.07	oe	ccsbBroad304_07238	STK24	YSK subfamily			
7875	-98.1	kd	CGS001-238	ALK	Leukocyte tyrosine kinase (LTK) receptor family			
7876	-98.11	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
7877	-98.11	kd	CGS001-6207	RPS13	S ribosomal proteins			
7878	-98.12	oe	ccsbBroad304_07337	TAF1B	-			
7879	-98.12	oe	ccsbBroad304_07362	NMI	-			
7880	-98.12	oe	ccsbBroad304_03182	GLOD4	-			
7881	-98.13	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
7882	-98.13	kd	CGS001-2778	GNAS	-			
7883	-98.16	kd	CGS001-64094	SMOC2	EF-hand domain containing			
7884	-98.16	kd	CGS001-9455	HOMER2	-			
7885	-98.17	oe	ccsbBroad304_01483	SAT1	-			
7886	-98.18	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
7887	-98.18	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
7888	-98.19	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
7889	-98.19	kd	CGS001-8727	CTNNAL1	Catenins			
7890	-98.2	cc		Nucleophosmin inhibitor	-			
7891	-98.21	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
7892	-98.21	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
7893	-98.22	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
7894	-98.22	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
7895	-98.22	kd	CGS001-1977	EIF4E	Translation Initiation Factor 4E			
7896	-98.23	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
7897	-98.23	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
7898	-98.26	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
7899	-98.28	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
7900	-98.29	cc		Leucine rich repeat kinase inhibitor	-			
7901	-98.3	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
7902	-98.3	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
7903	-98.34	oe	ccsbBroad304_06654	NPM1	-			
7904	-98.35	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
7905	-98.36	oe	ccsbBroad304_00600	FYN	Src family			
7906	-98.36	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
7907	-98.36	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
7908	-98.36	kd	CGS001-8892	EIF2B2	-			
7909	-98.36	kd	CGS001-1363	CPE	Carboxypeptidase A			
7910	-98.37	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
7911	-98.37	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
7912	-98.37	kd	CGS001-154	ADRB2	GPCR / Class A : Adrenoceptors : beta			
7913	-98.37	oe	ccsbBroad304_00106	ARRB1	-			
7914	-98.38	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
7915	-98.38	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
7916	-98.41	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
7917	-98.42	cc		Adenosine receptor agonist	-			
7918	-98.42	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
7919	-98.42	kd	CGS001-4967	OGDH	-			
7920	-98.44	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
7921	-98.44	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
7922	-98.46	kd	CGS001-3566	IL4R	IL-2 receptor family			
7923	-98.46	kd	CGS001-53834	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
7924	-98.46	kd	CGS001-54821	ERCC6L	-			
7925	-98.46	oe	ccsbBroad304_06671	OPA1	-			
7926	-98.47	cc		Protein synthesis inhibitor	-			
7927	-98.47	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
7928	-98.48	kd	CGS001-11031	RAB31	RAB, member RAS oncogene			
7929	-98.48	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
7930	-98.49	oe	ccsbBroad304_01208	PITPNA	-			
7931	-98.5	oe	ccsbBroad304_00789	HSBP1	-			
7932	-98.5	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
7933	-98.52	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
7934	-98.52	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
7935	-98.52	kd	CGS001-2356	FPGS	-			
7936	-98.53	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
7937	-98.55	oe	ccsbBroad304_03179	BOLA1	-			
7938	-98.55	kd	CGS001-7504	XK	Blood group antigens			
7939	-98.55	kd	CGS001-6210	RPS15A	S ribosomal proteins			
7940	-98.57	kd	CGS001-51548	SIRT6	Histone deacetylases (HDACs)			
7941	-98.57	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
7942	-98.58	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
7943	-98.58	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
7944	-98.58	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
7945	-98.59	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
7946	-98.59	oe	ccsbBroad304_01327	PSPH	-			
7947	-98.6	oe	ccsbBroad304_02756	RRP8	-			
7948	-98.6	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
7949	-98.6	kd	CGS001-6829	SUPT5H	-			
7950	-98.6	kd	CGS001-3934	LCN2	Lipocalins			
7951	-98.61	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
7952	-98.62	oe	ccsbBroad304_02416	TUBB4B	-			
7953	-98.62	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
7954	-98.62	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
7955	-98.62	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
7956	-98.65	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
7957	-98.65	kd	CGS001-960	CD44	CD molecules			
7958	-98.67	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
7959	-98.68	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
7960	-98.68	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
7961	-98.68	kd	CGS001-1611	DAP	-			
7962	-98.69	kd	CGS001-7625	ZNF74	Zinc fingers, C2H2-type			
7963	-98.69	kd	CGS001-64425	POLR1E	RNA polymerase subunits			
7964	-98.69	kd	CGS001-4048	LTA4H	Hydrolases			
7965	-98.71	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
7966	-98.71	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
7967	-98.72	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
7968	-98.72	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
7969	-98.73	oe	ccsbBroad304_00038	AGL	-			
7970	-98.73	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
7971	-98.74	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
7972	-98.74	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
7973	-98.75	kd	CGS001-55893	ZNF395	Zinc fingers, C2H2-type			
7974	-98.76	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
7975	-98.76	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
7976	-98.79	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
7977	-98.79	kd	CGS001-51466	EVL	-			
7978	-98.8	kd	CGS001-7249	TSC2	-			
7979	-98.8	kd	CGS001-51005	AMDHD2	-			
7980	-98.81	kd	CGS001-25805	BAMBI	-			
7981	-98.82	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
7982	-98.82	kd	CGS001-1806	DPYD	-			
7983	-98.82	kd	CGS001-301	ANXA1	Annexins			
7984	-98.83	cc		Serotonin receptor agonist	-			
7985	-98.83	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
7986	-98.83	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
7987	-98.83	kd	CGS001-2048	EPHB2	Type XIII RTKs: Ephrin receptor family			
7988	-98.86	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
7989	-98.87	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
7990	-98.87	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
7991	-98.87	kd	CGS001-6617	SNAPC1	-			
7992	-98.87	kd	CGS001-5048	PAFAH1B1	WD repeat domain containing			
7993	-98.87	kd	CGS001-8915	BCL10	-			
7994	-98.88	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
7995	-98.89	kd	CGS001-10135	NAMPT	-			
7996	-98.89	kd	CGS001-1022	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
7997	-98.91	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
7998	-98.91	kd	CGS001-8140	SLC7A5	SLC7 family			
7999	-98.91	oe	ccsbBroad304_03917	RBKS	-			
8000	-98.92	cc		Minor histocompatibility antigens LOF	-			
8001	-98.92	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
8002	-98.93	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
8003	-98.93	kd	CGS001-89845	ABCC10	ATP binding cassette transporters / subfamily C			
8004	-98.94	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
8005	-98.95	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
8006	-98.95	kd	CGS001-4125	MAN2B1	-			
8007	-98.97	kd	CGS001-8148	TAF15	RNA binding motif (RRM) containing			
8008	-98.98	oe	ccsbBroad304_09354	IGSF8	CD molecules			
8009	-98.98	oe	ccsbBroad304_08888	ACD	-			
8010	-98.99	oe	ccsbBroad304_01222	PLP2	-			
8011	-98.99	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
8012	-98.99	kd	CGS001-2030	SLC29A1	SLC29 family			
8013	-99	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
8014	-99	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
8015	-99	kd	CGS001-1487	CTBP1	-			
8016	-99.01	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
8017	-99.03	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
8018	-99.03	kd	CGS001-6307	MSMO1	Fatty acid hydroxylase domain containing			
8019	-99.03	kd	CGS001-11215	AKAP11	A-kinase anchor proteins			
8020	-99.04	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
8021	-99.04	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
8022	-99.04	kd	CGS001-699	BUB1	Bub family			
8023	-99.05	kd	CGS001-55770	EXOC2	-			
8024	-99.06	kd	CGS001-10481	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
8025	-99.07	oe	ccsbBroad304_01948	GAS7	-			
8026	-99.07	kd	CGS001-54732	TMED9	-			
8027	-99.07	kd	CGS001-58472	SQRDL	-			
8028	-99.08	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
8029	-99.09	cc		Potassium channel activator	-			
8030	-99.1	oe	ccsbBroad304_00710	GUSB	-			
8031	-99.12	cp	BRD-K32398298	alprazolam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, CYP3A5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
8032	-99.12	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
8033	-99.12	kd	CGS001-1595	CYP51A1	Cytochrome P450s			
8034	-99.13	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
8035	-99.13	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
8036	-99.13	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
8037	-99.15	oe	ccsbBroad304_03023	CRCP	-			
8038	-99.16	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
8039	-99.16	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
8040	-99.17	kd	CGS001-8726	EED	Neutral sphingomyelinase coupling factors			
8041	-99.19	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
8042	-99.19	kd	CGS001-7031	TFF1	-			
8043	-99.19	kd	CGS001-5546	PRCC	-			
8044	-99.19	kd	CGS001-8535	CBX4	-			
8045	-99.21	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
8046	-99.22	cp	BRD-M47937986	cefatrizine	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
8047	-99.22	kd	CGS001-1453	CSNK1D	Casein kinase 1 (CK1) family			
8048	-99.23	cp	BRD-K30563334	rifabutin	Protein synthesis inhibitor		CYP3A4, HSP90AA1, HSP90B1	Protein synthesis inhibitor
8049	-99.23	kd	CGS001-7128	TNFAIP3	OTU domain containing			
8050	-99.23	kd	CGS001-11325	DDX42	DEAD-boxes			
8051	-99.24	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
8052	-99.24	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
8053	-99.25	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
8054	-99.25	kd	CGS001-6934	TCF7L2	-			
8055	-99.25	kd	CGS001-23649	POLA2	DNA polymerases			
8056	-99.25	kd	CGS001-3565	IL4	Interleukins and interleukin receptors			
8057	-99.28	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
8058	-99.28	kd	CGS001-899	CCNF	F-boxes / other			
8059	-99.29	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
8060	-99.29	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
8061	-99.29	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
8062	-99.31	kd	CGS001-64754	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
8063	-99.31	kd	CGS001-6453	ITSN1	Rho guanine nucleotide exchange factors			
8064	-99.33	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
8065	-99.33	kd	CGS001-387	RHOA	-			
8066	-99.34	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
8067	-99.34	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
8068	-99.34	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
8069	-99.35	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
8070	-99.35	kd	CGS001-2289	FKBP5	Tetratricopeptide (TTC) repeat domain containing			
8071	-99.36	oe	ccsbBroad304_02092	SYNGR3	-			
8072	-99.36	kd	CGS001-6777	STAT5B	SH2 domain containing			
8073	-99.36	kd	CGS001-6217	RPS16	S ribosomal proteins			
8074	-99.37	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
8075	-99.39	kd	CGS001-3663	IRF5	-			
8076	-99.4	kd	CGS001-3988	LIPA	-			
8077	-99.41	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
8078	-99.42	kd	CGS001-23075	SWAP70	EF-hand domain containing			
8079	-99.43	oe	ccsbBroad304_03767	TOMM22	-			
8080	-99.43	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
8081	-99.43	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
8082	-99.43	kd	CGS001-57661	PHRF1	Zinc fingers, PHD-type			
8083	-99.43	kd	CGS001-10641	NPRL2	-			
8084	-99.43	kd	CGS001-3033	HADH	-			
8085	-99.44	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
8086	-99.45	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
8087	-99.46	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
8088	-99.46	kd	CGS001-2717	GLA	-			
8089	-99.46	kd	CGS001-397	ARHGDIB	Endogenous ligands			
8090	-99.47	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
8091	-99.49	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
8092	-99.49	kd	CGS001-4602	MYB	-			
8093	-99.49	kd	CGS001-7477	WNT7B	Endogenous ligands			
8094	-99.5	oe	ccsbBroad304_02840	PISD	Decarboxylases			
8095	-99.52	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
8096	-99.52	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
8097	-99.52	kd	CGS001-9322	TRIP10	-			
8098	-99.53	kd	CGS001-5576	PRKAR2A	Protein kinase A			
8099	-99.53	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
8100	-99.54	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
8101	-99.54	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
8102	-99.54	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
8103	-99.54	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
8104	-99.54	kd	CGS001-5869	RAB5B	RAB, member RAS oncogene			
8105	-99.54	kd	CGS001-5162	PDHB	-			
8106	-99.56	oe	ccsbBroad304_07548	TSSC4	-			
8107	-99.56	kd	CGS001-2152	F3	CD molecules			
8108	-99.56	kd	CGS001-805	CALM2	EF-hand domain containing			
8109	-99.57	kd	CGS001-80212	CCDC92	-			
8110	-99.58	kd	CGS001-4836	NMT1	-			
8111	-99.58	kd	CGS001-9258	MFHAS1	-			
8112	-99.58	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
8113	-99.59	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
8114	-99.59	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
8115	-99.59	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
8116	-99.59	kd	CGS001-84108	PCGF6	Polycomb group ring fingers			
8117	-99.59	kd	CGS001-55120	FANCL	Fanconi anemia, complementation groups			
8118	-99.6	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
8119	-99.6	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
8120	-99.6	kd	CGS001-2952	GSTT1	Glutathione S-transferases / Soluble			
8121	-99.61	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
8122	-99.62	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
8123	-99.62	kd	CGS001-1534	CYB561	Cytochrome b genes			
8124	-99.63	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
8125	-99.63	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
8126	-99.63	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
8127	-99.63	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
8128	-99.64	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
8129	-99.64	kd	CGS001-6883	TAF12	-			
8130	-99.65	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
8131	-99.65	kd	CGS001-8312	AXIN1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
8132	-99.65	kd	CGS001-475	ATOX1	-			
8133	-99.66	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
8134	-99.66	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
8135	-99.66	kd	CGS001-3897	L1CAM	CD molecules			
8136	-99.66	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
8137	-99.68	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
8138	-99.68	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
8139	-99.68	oe	ccsbBroad304_08116	TBK1	IKK family			
8140	-99.68	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
8141	-99.68	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
8142	-99.68	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
8143	-99.68	kd	CGS001-7010	TEK	Type XII RTKs: TIE family of angiopoietin receptors			
8144	-99.68	kd	CGS001-8531	CSDA	-			
8145	-99.69	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
8146	-99.69	kd	CGS001-7311	UBA52	L ribosomal proteins			
8147	-99.69	kd	CGS001-10628	TXNIP	-			
8148	-99.7	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
8149	-99.7	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
8150	-99.71	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
8151	-99.71	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
8152	-99.71	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
8153	-99.72	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
8154	-99.72	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
8155	-99.72	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
8156	-99.72	kd	CGS001-4151	MB	-			
8157	-99.74	cp	BRD-K15916496	clotrimazole	Cytochrome P450 inhibitor		KCNN4, CYP3A4, CYP51A1, NR1I2, NR1I3, TRPM2, TRPM4, TRPM8	Cytochrome P450 inhibitor, Imidazoline receptor ligand
8158	-99.74	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
8159	-99.74	kd	CGS001-4091	SMAD6	SMADs			
8160	-99.75	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
8161	-99.75	kd	CGS001-4846	NOS3	Nitric oxide synthases			
8162	-99.75	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
8163	-99.76	oe	ccsbBroad304_00161	BID	Endogenous ligands			
8164	-99.76	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
8165	-99.76	kd	CGS001-5315	PKM2	-			
8166	-99.76	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
8167	-99.76	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
8168	-99.77	cc		IL4 Pathway LOF	-			
8169	-99.77	kd	CGS001-1876	E2F6	-			
8170	-99.77	kd	CGS001-23429	RYBP	-			
8171	-99.78	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
8172	-99.78	oe	ccsbBroad304_03640	CEP72	-			
8173	-99.78	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
8174	-99.78	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
8175	-99.78	kd	CGS001-283150	FOXR1	Forkhead boxes			
8176	-99.79	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
8177	-99.79	kd	CGS001-9929	JOSD1	-			
8178	-99.79	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
8179	-99.8	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
8180	-99.8	oe	ccsbBroad304_00725	HADHA	-			
8181	-99.8	oe	ccsbBroad304_06094	DFFA	-			
8182	-99.8	kd	CGS001-51465	UBE2J1	Ubiquitin-conjugating enzymes E2			
8183	-99.8	kd	CGS001-8859	STK19	G11 family			
8184	-99.8	kd	CGS001-5327	PLAT	Chymotrypsin			
8185	-99.81	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
8186	-99.81	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
8187	-99.81	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
8188	-99.81	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
8189	-99.81	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
8190	-99.81	kd	CGS001-6203	RPS9	S ribosomal proteins			
8191	-99.81	kd	CGS001-55869	HDAC8	Histone deacetylases			
8192	-99.81	kd	CGS001-324	APC	Armadillo repeat containing			
8193	-99.81	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
8194	-99.82	cc		Progesterone receptor agonist	-			
8195	-99.82	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
8196	-99.82	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
8197	-99.82	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
8198	-99.82	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
8199	-99.82	kd	CGS001-3978	LIG1	-			
8200	-99.82	kd	CGS001-23523	CABIN1	-			
8201	-99.82	oe	ccsbBroad304_00174	BRAF	RAF family			
8202	-99.83	cc		Kruppel like transcription factors LOF	-			
8203	-99.83	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
8204	-99.83	kd	CGS001-51160	VPS28	-			
8205	-99.83	kd	CGS001-6455	SH3GL1	-			
8206	-99.83	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
8207	-99.83	kd	CGS001-1728	NQO1	-			
8208	-99.83	kd	CGS001-2534	FYN	Src family			
8209	-99.83	kd	CGS001-537	ATP6AP1	-			
8210	-99.84	oe	ccsbBroad304_03859	ENOPH1	-			
8211	-99.84	oe	ccsbBroad304_03415	GFOD1	-			
8212	-99.84	oe	ccsbBroad304_08797	FASTKD5	-			
8213	-99.84	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
8214	-99.84	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
8215	-99.84	kd	CGS001-50814	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
8216	-99.84	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
8217	-99.84	kd	CGS001-3094	HINT1	-			
8218	-99.84	kd	CGS001-2059	EPS8	-			
8219	-99.84	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
8220	-99.85	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
8221	-99.86	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
8222	-99.86	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
8223	-99.86	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
8224	-99.86	kd	CGS001-7167	TPI1	-			
8225	-99.86	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
8226	-99.87	cc		Apolipoproteins LOF	-			
8227	-99.87	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
8228	-99.87	oe	ccsbBroad304_03728	DIABLO	-			
8229	-99.87	kd	CGS001-23499	MACF1	EF-hand domain containing			
8230	-99.87	kd	CGS001-6129	RPL7	L ribosomal proteins			
8231	-99.87	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
8232	-99.88	oe	ccsbBroad304_04153	PHF17	-			
8233	-99.88	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
8234	-99.88	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
8235	-99.88	oe	ccsbBroad304_00572	FKBP3	-			
8236	-99.88	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
8237	-99.88	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
8238	-99.88	kd	CGS001-6817	SULT1A1	Sulfotransferases, cytosolic			
8239	-99.88	kd	CGS001-8681	JMJD7-PLA2G4B	-			
8240	-99.88	kd	CGS001-3459	IFNGR1	Interferon receptor family			
8241	-99.88	kd	CGS001-599	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
8242	-99.89	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
8243	-99.89	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
8244	-99.89	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
8245	-99.89	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
8246	-99.89	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
8247	-99.89	kd	CGS001-9263	STK17A	Death-associated kinase (DAPK) family			
8248	-99.89	kd	CGS001-6285	S100B	EF-hand domain containing			
8249	-99.89	kd	CGS001-3661	IRF3	-			
8250	-99.89	kd	CGS001-3199	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
8251	-99.89	kd	CGS001-821	CANX	-			
8252	-99.9	oe	ccsbBroad304_02592	KIF2C	Kinesins			
8253	-99.9	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
8254	-99.9	kd	CGS001-80314	EPC1	-			
8255	-99.9	kd	CGS001-10987	COPS5	-			
8256	-99.9	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
8257	-99.9	kd	CGS001-166	AES	-			
8258	-99.9	oe	ccsbBroad304_05894	BLVRA	-			
8259	-99.9	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
8260	-99.92	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
8261	-99.92	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
8262	-99.92	kd	CGS001-5535	PPP3R2	EF-hand domain containing			
8263	-99.92	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
8264	-99.93	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
8265	-99.93	kd	CGS001-7466	WFS1	-			
8266	-99.93	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
8267	-99.93	kd	CGS001-5498	PPOX	-			
8268	-99.93	kd	CGS001-4552	MTRR	-			
8269	-99.93	kd	CGS001-3660	IRF2	-			
8270	-99.93	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
8271	-99.94	oe	ccsbBroad304_07724	KDELR2	-			
8272	-99.94	oe	ccsbBroad304_04292	INHBE	-			
8273	-99.94	oe	ccsbBroad304_00179	BTG1	-			
8274	-99.94	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
8275	-99.94	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
8276	-99.94	kd	CGS001-6119	RPA3	-			
8277	-99.94	kd	CGS001-9616	RNF7	RING-type (C3HC4) zinc fingers			
8278	-99.94	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
8279	-99.94	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
8280	-99.94	kd	CGS001-11040	PIM2	PIM family			
8281	-99.94	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
8282	-99.94	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
8283	-99.95	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
8284	-99.95	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
8285	-99.95	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
8286	-99.95	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
8287	-99.95	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
8288	-99.95	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
8289	-99.95	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
8290	-99.95	kd	CGS001-10252	SPRY1	-			
8291	-99.95	kd	CGS001-56848	SPHK2	Sphingosine kinase			
8292	-99.95	kd	CGS001-5329	PLAUR	CD molecules			
8293	-99.95	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
8294	-99.96	oe	ccsbBroad304_00519	ETFB	-			
8295	-99.96	oe	ccsbBroad304_01663	TFF2	-			
8296	-99.96	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
8297	-99.96	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
8298	-99.96	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
8299	-99.96	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
8300	-99.96	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
8301	-99.96	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
8302	-99.96	kd	CGS001-3065	HDAC1	Histone deacetylases			
8303	-99.96	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
8304	-99.96	kd	CGS001-894	CCND2	-			
8305	-99.96	kd	CGS001-121549	ASCL4	Basic helix-loop-helix proteins			
8306	-99.96	oe	ccsbBroad304_00949	LRPAP1	-			
8307	-99.97	oe	ccsbBroad304_06569	MCM5	-			
8308	-99.98	oe	ccsbBroad304_01203	PIM1	PIM family			
8309	-99.98	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
8310	-99.98	oe	ccsbBroad304_00738	HINT1	-			
8311	-99.98	oe	ccsbBroad304_00651	GNAI3	-			
8312	-99.98	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
8313	-99.98	oe	ccsbBroad304_02229	TRAM2	-			
8314	-99.98	oe	ccsbBroad304_02831	SGK3	SGK family			
8315	-99.98	oe	ccsbBroad304_07490	SCRN1	-			
8316	-99.98	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
8317	-99.98	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
8318	-99.98	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
8319	-99.98	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
8320	-99.98	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
8321	-99.98	oe	ccsbBroad304_06538	LSP1	-			
8322	-99.98	oe	ccsbBroad304_00624	GCK	Hexokinases			
8323	-99.98	oe	ccsbBroad304_00162	BIK	-			
8324	-99.98	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
8325	-99.98	cp	BRD-K51671335	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
8326	-99.98	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
8327	-99.98	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
8328	-99.98	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
8329	-99.98	kd	CGS001-7052	TGM2	Transglutaminases			
8330	-99.98	kd	CGS001-10214	SSX3	-			
8331	-99.98	kd	CGS001-6478	SIAH2	-			
8332	-99.98	kd	CGS001-6146	RPL22	L ribosomal proteins			
8333	-99.98	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
8334	-99.98	kd	CGS001-5423	POLB	DNA polymerases			
8335	-99.98	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
8336	-99.98	kd	CGS001-200879	LIPH	-			
8337	-99.98	kd	CGS001-9870	KIAA0317	-			
8338	-99.98	kd	CGS001-83737	ITCH	-			
8339	-99.98	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
8340	-99.98	kd	CGS001-51564	HDAC7	Histone deacetylases			
8341	-99.98	kd	CGS001-3066	HDAC2	Histone deacetylases			
8342	-99.98	kd	CGS001-2896	GRN	-			
8343	-99.98	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
8344	-99.98	kd	CGS001-1632	ECI1	-			
8345	-99.98	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
8346	-99.98	kd	CGS001-1128	CHRM1	Cholinergic receptors			
8347	-99.98	kd	CGS001-801	CALM1	EF-hand domain containing			
8348	-99.98	kd	CGS001-6046	BRD2	Bromodomain kinase (BRDK) family			
8349	-99.98	kd	CGS001-635	BHMT	-			
8350	-99.98	kd	CGS001-338	APOB	Apolipoproteins			
8351	-99.98	kd	CGS001-174	AFP	-			
8352	-99.98	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
8353	-99.98	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
8354	-99.98	oe	ccsbBroad304_02506	EBP	-			
8355	-99.99	kd	CGS001-5170	PDPK1	PDK1 family			
8356	-100	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
8357	-100	kd	CGS001-468	ATF4	basic leucine zipper proteins			
8358	-100	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
