Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cc		Sodium channel blocker	-			
2	99.99	cc		Wnt family LOF	-			
3	99.99	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
4	99.98	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
5	99.98	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
6	99.98	oe	ccsbBroad304_02741	PDS5A	-			
7	99.98	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
8	99.98	oe	ccsbBroad304_02759	DICER1	-			
9	99.98	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
10	99.98	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
11	99.98	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
12	99.98	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
13	99.98	oe	ccsbBroad304_06458	IRF3	-			
14	99.98	oe	ccsbBroad304_00795	HSF2	-			
15	99.98	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
16	99.98	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
17	99.98	oe	ccsbBroad304_06278	GK	Glycerol kinases			
18	99.98	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
19	99.98	oe	ccsbBroad304_02686	COPZ1	-			
20	99.98	oe	ccsbBroad304_02143	CNOT8	-			
21	99.98	oe	ccsbBroad304_03047	BZW2	-			
22	99.98	oe	ccsbBroad304_09225	BUD13	-			
23	99.98	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
24	99.98	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
25	99.98	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
26	99.98	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
27	99.98	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
28	99.98	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
29	99.98	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
30	99.98	cp	BRD-K01649396	indatraline	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine transporter inhibitor
31	99.98	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
32	99.98	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
33	99.98	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
34	99.98	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
35	99.98	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
36	99.98	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
37	99.98	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
38	99.98	kd	CGS001-7504	XK	Blood group antigens			
39	99.98	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
40	99.98	kd	CGS001-89882	TPD52L3	-			
41	99.98	kd	CGS001-7004	TEAD4	-			
42	99.98	kd	CGS001-6895	TARBP2	-			
43	99.98	kd	CGS001-6821	SUOX	-			
44	99.98	kd	CGS001-6469	SHH	-			
45	99.98	kd	CGS001-462	SERPINC1	Serine (or cysteine) peptidase inhibitors			
46	99.98	kd	CGS001-9616	RNF7	RING-type (C3HC4) zinc fingers			
47	99.98	kd	CGS001-8635	RNASET2	-			
48	99.98	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
49	99.98	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
50	99.98	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
51	99.98	kd	CGS001-7025	NR2F1	COUP-TF-like receptors			
52	99.98	kd	CGS001-10392	NOD1	Nucleotide-binding domain and leucine rich repeat containing			
53	99.98	kd	CGS001-4830	NME1	-			
54	99.98	kd	CGS001-64863	METTL4	-			
55	99.98	kd	CGS001-84539	MCHR2	GPCR / Class A : MCH receptors			
56	99.98	kd	CGS001-3930	LBR	Tudor domain containing			
57	99.98	kd	CGS001-8692	HYAL2	-			
58	99.98	kd	CGS001-3373	HYAL1	-			
59	99.98	kd	CGS001-2937	GSS	-			
60	99.98	kd	CGS001-23401	FRAT2	-			
61	99.98	kd	CGS001-2168	FABP1	Fatty acid-binding proteins			
62	99.98	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
63	99.98	kd	CGS001-1763	DNA2	-			
64	99.98	kd	CGS001-1719	DHFR	Oxidoreductases			
65	99.98	kd	CGS001-148327	CREB3L4	basic leucine zipper proteins			
66	99.98	kd	CGS001-54805	CNNM2	-			
67	99.98	kd	CGS001-1028	CDKN1C	-			
68	99.98	kd	CGS001-55536	CDCA7L	-			
69	99.98	kd	CGS001-890	CCNA2	-			
70	99.98	kd	CGS001-8535	CBX4	-			
71	99.98	kd	CGS001-840	CASP7	Caspases			
72	99.98	kd	CGS001-837	CASP4	Caspases			
73	99.98	kd	CGS001-85027	C5ORF62	-			
74	99.98	kd	CGS001-694	BTG1	-			
75	99.98	kd	CGS001-51027	BOLA1	-			
76	99.98	kd	CGS001-367	AR	Nuclear hormone receptors			
77	99.98	kd	CGS001-55608	ANKRD10	Ankyrin repeat domain containing			
78	99.98	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
79	99.96	oe	ccsbBroad304_04891	TMEM174	-			
80	99.96	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
81	99.96	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
82	99.96	oe	ccsbBroad304_04153	PHF17	-			
83	99.96	oe	ccsbBroad304_06654	NPM1	-			
84	99.96	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
85	99.96	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
86	99.96	oe	ccsbBroad304_06291	GNAI1	-			
87	99.96	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
88	99.96	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
89	99.96	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
90	99.96	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
91	99.96	kd	CGS001-7108	TM7SF2	-			
92	99.96	kd	CGS001-23224	SYNE2	-			
93	99.96	kd	CGS001-23378	RRP8	-			
94	99.96	kd	CGS001-5091	PC	Carboxylases			
95	99.96	kd	CGS001-9500	MAGED1	-			
96	99.96	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
97	99.96	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
98	99.96	kd	CGS001-8804	CREG1	-			
99	99.96	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
100	99.96	oe	ccsbBroad304_00811	ICAM1	CD molecules			
101	99.95	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
102	99.95	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
103	99.95	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
104	99.95	oe	ccsbBroad304_02292	BCL2L11	-			
105	99.95	oe	ccsbBroad304_00146	BAD	-			
106	99.95	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
107	99.95	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
108	99.95	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
109	99.95	cp	BRD-A48261811	argatroban	Thrombin inhibitor		F2, CYP3A5	Thrombin inhibitor
110	99.95	cp	BRD-K85925969	zalcitabine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
111	99.95	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
112	99.95	kd	CGS001-285676	ZNF454	Zinc fingers, C2H2-type			
113	99.95	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
114	99.95	kd	CGS001-57761	TRIB3	Trbl family			
115	99.95	kd	CGS001-8435	SOAT2	-			
116	99.95	kd	CGS001-57154	SMURF1	-			
117	99.95	kd	CGS001-5446	PON3	Paraoxonases			
118	99.95	kd	CGS001-23139	MAST2	MAST family			
119	99.95	kd	CGS001-23030	KDM4B	Histone demethylases			
120	99.95	kd	CGS001-65123	INTS3	-			
121	99.95	kd	CGS001-55662	HIF1AN	-			
122	99.95	kd	CGS001-9759	HDAC4	Histone deacetylases			
123	99.95	kd	CGS001-1305	COL13A1	Collagens			
124	99.95	kd	CGS001-25966	C2CD2	-			
125	99.94	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
126	99.94	oe	ccsbBroad304_03604	ENOSF1	-			
127	99.94	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
128	99.94	oe	ccsbBroad304_02058	PLOD3	-			
129	99.94	oe	ccsbBroad304_08104	MED4	-			
130	99.94	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
131	99.94	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
132	99.94	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
133	99.94	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
134	99.94	kd	CGS001-6519	SLC3A1	SLC3 family			
135	99.94	kd	CGS001-6117	RPA1	-			
136	99.94	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
137	99.94	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
138	99.94	kd	CGS001-4849	CNOT3	-			
139	99.94	kd	CGS001-84811	BUD13	-			
140	99.94	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
141	99.93	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
142	99.93	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
143	99.93	oe	ccsbBroad304_07280	LAMTOR3	-			
144	99.93	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
145	99.93	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
146	99.93	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
147	99.93	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
148	99.93	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
149	99.93	kd	CGS001-10252	SPRY1	-			
150	99.93	kd	CGS001-4707	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
151	99.93	kd	CGS001-2243	FGA	Endogenous ligands			
152	99.93	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
153	99.93	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
154	99.93	kd	CGS001-538	ATP7A	ATPases / P-type			
155	99.93	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
156	99.93	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
157	99.92	oe	ccsbBroad304_00995	MECP2	-			
158	99.91	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
159	99.91	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
160	99.91	oe	ccsbBroad304_00975	MAT2A	-			
161	99.91	oe	ccsbBroad304_03023	CRCP	-			
162	99.91	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
163	99.91	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
164	99.91	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
165	99.91	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
166	99.91	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
167	99.91	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
168	99.91	kd	CGS001-121599	SPIC	ETS Transcription Factors			
169	99.91	kd	CGS001-481	ATP1B1	ATPases / P-type			
170	99.91	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
171	99.9	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
172	99.9	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
173	99.9	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
174	99.9	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
175	99.9	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
176	99.9	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
177	99.9	kd	CGS001-51097	SCCPDH	-			
178	99.9	kd	CGS001-4942	OAT	-			
179	99.9	kd	CGS001-4012	LNPEP	Aminopeptidase N			
180	99.9	kd	CGS001-2048	EPHB2	Type XIII RTKs: Ephrin receptor family			
181	99.89	cc		Potassium channel activator	-			
182	99.89	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
183	99.89	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
184	99.89	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
185	99.89	kd	CGS001-29982	NRBF2	-			
186	99.89	oe	ccsbBroad304_07688	FAM114A2	-			
187	99.88	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
188	99.88	oe	ccsbBroad304_00644	GCLC	-			
189	99.88	oe	ccsbBroad304_09054	EGFL8	-			
190	99.88	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
191	99.88	kd	CGS001-6118	RPA2	-			
192	99.88	kd	CGS001-4069	LYZ	-			
193	99.88	kd	CGS001-1069	CETN2	EF-hand domain containing			
194	99.87	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
195	99.87	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
196	99.87	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
197	99.87	cp	BRD-K11630072	carmofur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
198	99.87	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
199	99.87	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
200	99.87	kd	CGS001-118442	GPR62	GPCR / Class A : Orphans			
201	99.87	kd	CGS001-8905	AP1S2	-			
202	99.85	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
203	99.85	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
204	99.85	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
205	99.85	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
206	99.85	kd	CGS001-10237	SLC35B1	SLC35 family of nucleotide sugar transporters			
207	99.85	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
208	99.84	oe	ccsbBroad304_00964	SMAD7	SMADs			
209	99.84	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
210	99.84	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
211	99.84	kd	CGS001-51128	SAR1B	-			
212	99.83	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
213	99.83	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
214	99.83	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
215	99.83	kd	CGS001-285267	ZNF619	Zinc fingers, C2H2-type			
216	99.83	kd	CGS001-6601	SMARCC2	-			
217	99.83	kd	CGS001-79170	PRR15L	-			
218	99.83	kd	CGS001-51588	PIAS4	Zinc fingers, MIZ-type			
219	99.83	kd	CGS001-54505	DHX29	DEAH-boxes			
220	99.83	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
221	99.82	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
222	99.82	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
223	99.82	kd	CGS001-1786	DNMT1	Methyltransferases			
224	99.81	cc		Protein phosphatase catalytic subunits LOF	-			
225	99.81	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
226	99.81	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
227	99.81	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
228	99.81	kd	CGS001-83440	ADPGK	-			
229	99.79	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
230	99.79	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
231	99.79	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
232	99.79	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
233	99.79	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
234	99.79	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
235	99.78	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
236	99.77	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
237	99.77	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
238	99.77	kd	CGS001-7298	TYMS	Methyltransferases			
239	99.77	kd	CGS001-6887	TAL2	Basic helix-loop-helix proteins			
240	99.77	kd	CGS001-116535	MRGPRF	GPCR / Class A : Orphans			
241	99.76	cp	BRD-K16336526	capsaicin	TRPV agonist		TRPV1, CFTR, ENOX2	TRPV agonist
242	99.76	cp	BRD-K33483813	actarit	Interleukin receptor agonist			Interleukin receptor agonist
243	99.76	kd	CGS001-2264	FGFR4	Type V RTKs: FGF (fibroblast growth factor) receptor family			
244	99.76	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
245	99.75	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
246	99.74	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
247	99.74	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
248	99.74	oe	ccsbBroad304_09254	PAQR8	-			
249	99.74	oe	ccsbBroad304_02157	MED21	-			
250	99.73	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
251	99.73	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
252	99.73	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
253	99.73	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
254	99.72	cc		C2 domain containing LOF	-			
255	99.72	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
256	99.72	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
257	99.72	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
258	99.72	kd	CGS001-10451	VAV3	Rho guanine nucleotide exchange factors			
259	99.72	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
260	99.71	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
261	99.71	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
262	99.71	oe	ccsbBroad304_00268	CD81	CD molecules			
263	99.71	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
264	99.71	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
265	99.71	kd	CGS001-185	AGTR1	Angiotensin receptors			
266	99.7	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
267	99.7	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
268	99.7	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
269	99.7	kd	CGS001-22889	KIAA0907	-			
270	99.68	oe	ccsbBroad304_00650	GNA11	-			
271	99.68	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
272	99.67	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
273	99.67	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
274	99.66	kd	CGS001-3162	HMOX1	Haem oxygenase			
275	99.65	oe	ccsbBroad304_01699	TPD52L2	-			
276	99.65	kd	CGS001-2130	EWSR1	RNA binding motif (RRM) containing			
277	99.65	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
278	99.64	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
279	99.64	kd	CGS001-8566	PDXK	-			
280	99.64	kd	CGS001-9788	MTSS1	-			
281	99.64	kd	CGS001-25861	DFNB31	-			
282	99.64	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
283	99.63	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
284	99.62	kd	CGS001-3017	HIST1H2BD	Histones / Replication-dependent			
285	99.62	kd	CGS001-835	CASP2	Caspases			
286	99.61	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
287	99.61	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
288	99.61	kd	CGS001-7750	ZMYM2	Zinc fingers, MYM type			
289	99.6	oe	ccsbBroad304_04471	C5ORF62	-			
290	99.6	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
291	99.6	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
292	99.6	kd	CGS001-7486	WRN	-			
293	99.6	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
294	99.6	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
295	99.6	kd	CGS001-9891	NUAK1	NuaK subfamily			
296	99.6	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
297	99.59	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
298	99.59	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
299	99.59	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
300	99.59	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
301	99.59	kd	CGS001-126208	ZNF787	Zinc fingers, C2H2-type			
302	99.58	oe	ccsbBroad304_08217	SCCPDH	-			
303	99.57	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
304	99.57	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
305	99.57	kd	CGS001-56993	TOMM22	-			
306	99.56	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
307	99.56	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
308	99.56	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
309	99.55	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
310	99.55	oe	ccsbBroad304_02676	PHB2	-			
311	99.55	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
312	99.55	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
313	99.54	oe	ccsbBroad304_09708	PNLDC1	-			
314	99.54	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
315	99.54	kd	CGS001-10608	MXD4	Basic helix-loop-helix proteins			
316	99.53	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
317	99.53	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
318	99.52	kd	CGS001-10928	RALBP1	-			
319	99.52	kd	CGS001-150962	PUS10	-			
320	99.51	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
321	99.5	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
322	99.5	kd	CGS001-5194	PEX13	-			
323	99.48	cp	BRD-K41903098	diphenoxylate	Opioid receptor agonist		OPRM1, OPRD1	Opioid receptor agonist
324	99.48	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
325	99.47	oe	ccsbBroad304_06226	FTL	-			
326	99.47	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
327	99.46	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
328	99.45	kd	CGS001-51776	ZAK	MLK subfamily			
329	99.44	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
330	99.44	kd	CGS001-8050	PDHX	-			
331	99.44	kd	CGS001-3131	HLF	-			
332	99.43	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
333	99.43	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
334	99.43	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
335	99.43	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
336	99.43	kd	CGS001-5445	PON2	Paraoxonases			
337	99.42	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
338	99.42	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
339	99.42	kd	CGS001-5645	PRSS2	Serine peptidases			
340	99.41	oe	ccsbBroad304_01186	PHB	-			
341	99.41	kd	CGS001-6198	RPS6KB1	p70 subfamily			
342	99.41	kd	CGS001-2876	GPX1	-			
343	99.41	kd	CGS001-1211	CLTA	-			
344	99.4	cc		Sterol demethylase inhibitor	-			
345	99.4	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
346	99.4	oe	ccsbBroad304_02197	VPS26A	-			
347	99.4	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
348	99.4	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
349	99.39	oe	ccsbBroad304_01247	POU2AF1	-			
350	99.39	oe	ccsbBroad304_08605	PBK	TOPK family			
351	99.39	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
352	99.39	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
353	99.38	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
354	99.38	cp	BRD-A23637604	oxymetholone	Androgen receptor agonist		AR	Androgen receptor agonist
355	99.36	kd	CGS001-5378	PMS1	-			
356	99.36	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
357	99.36	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
358	99.35	kd	CGS001-29940	DSE	-			
359	99.34	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
360	99.34	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
361	99.34	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
362	99.34	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
363	99.33	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
364	99.33	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
365	99.33	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
366	99.32	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
367	99.31	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
368	99.3	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
369	99.28	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
370	99.28	kd	CGS001-23274	CLEC16A	C-type lectin domain containing			
371	99.27	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
372	99.27	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
373	99.27	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
374	99.27	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
375	99.25	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
376	99.25	kd	CGS001-29959	NRBP1	NRBP family			
377	99.24	cc		Histone deacetylases LOF	-			
378	99.24	kd	CGS001-4841	NONO	RNA binding motif (RRM) containing			
379	99.23	kd	CGS001-286075	ZNF707	Zinc fingers, C2H2-type			
380	99.23	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
381	99.21	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
382	99.21	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
383	99.21	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
384	99.19	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
385	99.19	kd	CGS001-84923	FAM104A	-			
386	99.18	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
387	99.18	kd	CGS001-5257	PHKB	-			
388	99.17	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
389	99.17	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
390	99.16	cc		CCK receptor antagonist	-			
391	99.16	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
392	99.16	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
393	99.15	oe	ccsbBroad304_01527	SGK1	SGK family			
394	99.15	oe	ccsbBroad304_10207	ERLIN1	-			
395	99.15	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
396	99.15	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
397	99.14	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
398	99.14	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
399	99.14	kd	CGS001-3776	KCNK2	Two-P potassium channels			
400	99.13	kd	CGS001-10617	STAMBP	-			
401	99.11	kd	CGS001-11319	ECD	-			
402	99.1	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
403	99.1	kd	CGS001-4232	MEST	-			
404	99.09	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
405	99.08	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
406	99.08	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
407	99.06	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
408	99.06	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
409	99.06	kd	CGS001-7727	ZNF174	Zinc fingers, C2H2-type			
410	99.05	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
411	99.05	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
412	99.04	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
413	99.03	oe	ccsbBroad304_01257	PPOX	-			
414	99.03	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
415	99.02	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
416	99.02	oe	ccsbBroad304_02026	NRP1	CD molecules			
417	99.02	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
418	99.01	cc		DNA Replication LOF	-			
419	98.99	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
420	98.99	cp	BRD-A52282606	lacidipine	Calcium channel blocker		CACNA1C	Calcium channel blocker
421	98.98	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
422	98.97	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
423	98.97	kd	CGS001-2615	LRRC32	-			
424	98.97	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
425	98.96	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
426	98.96	kd	CGS001-4781	NFIB	-			
427	98.95	kd	CGS001-5982	RFC2	ATPases / AAA-type			
428	98.94	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
429	98.94	oe	ccsbBroad304_01519	SET	-			
430	98.94	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
431	98.94	kd	CGS001-10161	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
432	98.93	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
433	98.92	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
434	98.92	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
435	98.91	oe	ccsbBroad304_07128	VHL	-			
436	98.88	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
437	98.88	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
438	98.88	kd	CGS001-337867	UBAC2	-			
439	98.88	kd	CGS001-2618	GART	Ribosyl transferases			
440	98.87	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
441	98.86	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
442	98.86	cp	BRD-K34508425	KUC103898N	-666			-666
443	98.86	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
444	98.85	cc		HIV protease inhibitor	-			
445	98.85	kd	CGS001-6472	SHMT2	-			
446	98.84	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
447	98.84	kd	CGS001-5928	RBBP4	WD repeat domain containing			
448	98.84	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
449	98.83	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
450	98.83	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
451	98.83	kd	CGS001-10308	ZNF267	Zinc fingers, C2H2-type			
452	98.83	kd	CGS001-124583	CANT1	-			
453	98.81	cp	BRD-A62890442	3-methyl-GABA	GABA aminotransferase activator			GABA aminotransferase activator
454	98.81	oe	ccsbBroad304_02047	AP1S2	-			
455	98.8	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
456	98.8	cp	BRD-A56892734	esomeprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
457	98.79	kd	CGS001-6883	TAF12	-			
458	98.79	kd	CGS001-900	CCNG1	-			
459	98.78	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
460	98.77	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
461	98.77	kd	CGS001-55311	ZNF444	Zinc fingers, C2H2-type			
462	98.76	cp	BRD-K44353683	nateglinide	Insulin secretagogue		ABCC8, KCNJ11, CYP3A4, INS, KCNJ10, PPARG	Insulin secretagogue
463	98.76	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
464	98.75	kd	CGS001-152	ADRA2C	GPCR / Class A : Adrenoceptors : alpha			
465	98.72	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
466	98.72	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
467	98.71	cp	BRD-K84566043	fenpiverinium	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
468	98.71	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
469	98.71	kd	CGS001-26292	MYCBP	-			
470	98.7	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
471	98.68	cp	BRD-A49172652	lansoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4, CYP3A5	ATPase inhibitor
472	98.68	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
473	98.68	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
474	98.68	kd	CGS001-84647	PLA2G12B	-			
475	98.68	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
476	98.67	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
477	98.67	kd	CGS001-55423	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
478	98.66	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
479	98.66	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
480	98.66	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
481	98.66	kd	CGS001-84722	PSRC1	-			
482	98.64	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
483	98.64	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
484	98.64	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
485	98.64	kd	CGS001-55226	NAT10	-			
486	98.63	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
487	98.63	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
488	98.62	kd	CGS001-718	C3	Endogenous ligands			
489	98.61	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
490	98.6	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
491	98.6	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
492	98.58	kd	CGS001-8061	FOSL1	basic leucine zipper proteins			
493	98.57	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
494	98.57	kd	CGS001-3589	IL11	Endogenous ligands			
495	98.56	kd	CGS001-83933	HDAC10	Histone deacetylases			
496	98.55	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
497	98.54	kd	CGS001-9318	COPS2	-			
498	98.53	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
499	98.52	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
500	98.51	oe	ccsbBroad304_08322	UFM1	-			
501	98.51	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
502	98.51	cp	BRD-K32398298	alprazolam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, CYP3A5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
503	98.5	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
504	98.5	kd	CGS001-5277	PIGA	Glycosyltransferase group 1 domain containing			
505	98.5	kd	CGS001-85315	PAQR8	-			
506	98.5	kd	CGS001-2072	ERCC4	-			
507	98.49	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
508	98.49	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
509	98.48	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
510	98.48	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
511	98.46	oe	ccsbBroad304_03308	YTHDF2	-			
512	98.46	kd	CGS001-6713	SQLE	Lanosterol biosynthesis pathway			
513	98.46	kd	CGS001-716	C1S	Complement system			
514	98.45	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
515	98.45	kd	CGS001-3689	ITGB2	Integrins			
516	98.45	kd	CGS001-29965	C16ORF5	-			
517	98.44	oe	ccsbBroad304_03186	GMNN	-			
518	98.43	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
519	98.39	kd	CGS001-3912	LAMB1	Laminins			
520	98.39	kd	CGS001-2896	GRN	-			
521	98.38	oe	ccsbBroad304_04064	PRR15L	-			
522	98.37	oe	ccsbBroad304_06992	SRC	Src family			
523	98.37	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
524	98.36	cc		DNA synthesis inhibitor	-			
525	98.36	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
526	98.36	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
527	98.36	kd	CGS001-5328	PLAU	Chymotrypsin			
528	98.35	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
529	98.35	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
530	98.32	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
531	98.32	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
532	98.31	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
533	98.3	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
534	98.29	kd	CGS001-10007	GNPDA1	-			
535	98.29	kd	CGS001-2159	F10	Chymotrypsin			
536	98.28	cp	BRD-A01787639	naftopidil	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
537	98.28	kd	CGS001-23	ABCF1	ATP binding cassette transporters / subfamily F			
538	98.25	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
539	98.25	oe	ccsbBroad304_00225	CAT	-			
540	98.25	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
541	98.24	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
542	98.24	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
543	98.22	oe	ccsbBroad304_06671	OPA1	-			
544	98.21	kd	CGS001-2078	ERG	ETS Transcription Factors			
545	98.18	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
546	98.17	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
547	98.17	kd	CGS001-5048	PAFAH1B1	WD repeat domain containing			
548	98.17	kd	CGS001-11140	CDC37	-			
549	98.16	oe	ccsbBroad304_06852	RBP4	Lipocalins			
550	98.16	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
551	98.16	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
552	98.16	kd	CGS001-9352	TXNL1	-			
553	98.15	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
554	98.15	kd	CGS001-439	ASNA1	-			
555	98.13	kd	CGS001-8193	DPF1	Zinc fingers, PHD-type			
556	98.12	oe	ccsbBroad304_02845	PRPF6	-			
557	98.11	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
558	98.1	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
559	98.09	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
560	98.09	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
561	98.09	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
562	98.08	oe	ccsbBroad304_03089	PACSIN3	-			
563	98.08	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
564	98.08	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
565	98.07	kd	CGS001-23142	DCUN1D4	-			
566	98.06	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
567	98.06	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
568	98.03	oe	ccsbBroad304_03739	NRIP3	-			
569	98.03	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
570	98.02	kd	CGS001-1284	COL4A2	Collagens			
571	98.02	kd	CGS001-801	CALM1	EF-hand domain containing			
572	98.01	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
573	98	cp	BRD-K50938287	sumatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1A, HTR1F, HTR1E, HTR5A, HTR6, HTR7	Serotonin receptor agonist
574	97.98	oe	ccsbBroad304_06889	RPN2	-			
575	97.98	kd	CGS001-27336	HTATSF1	RNA binding motif (RRM) containing			
576	97.96	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
577	97.95	kd	CGS001-54677	CROT	-			
578	97.94	oe	ccsbBroad304_00738	HINT1	-			
579	97.94	cp	BRD-K06878038	deferiprone	Chelating agent		CYP4F2	Chelating agent
580	97.93	kd	CGS001-8985	PLOD3	-			
581	97.92	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
582	97.92	kd	CGS001-54884	RETSAT	-			
583	97.91	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
584	97.9	kd	CGS001-9475	ROCK2	Pleckstrin homology (PH) domain containing			
585	97.89	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
586	97.88	kd	CGS001-79001	VKORC1	Oxidoreductases			
587	97.88	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
588	97.87	oe	ccsbBroad304_06318	GPER	-			
589	97.87	cp	BRD-A09495397	bicuculline	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, KCNN1	GABA receptor antagonist
590	97.87	kd	CGS001-390	RND3	-			
591	97.85	oe	ccsbBroad304_06174	ERCC1	-			
592	97.85	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
593	97.85	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
594	97.83	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
595	97.83	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
596	97.8	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
597	97.77	cc		Targets of VEGFR inhibitors GOF	-			
598	97.77	kd	CGS001-51495	PTPLAD1	-			
599	97.76	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
600	97.75	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
601	97.73	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
602	97.73	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
603	97.7	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
604	97.7	kd	CGS001-10721	POLQ	DNA polymerases			
605	97.69	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
606	97.68	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
607	97.65	kd	CGS001-2817	GPC1	Proteoglycans / Cell Surface : Glypicans			
608	97.64	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
609	97.63	kd	CGS001-9854	C2CD2L	-			
610	97.61	kd	CGS001-6775	STAT4	SH2 domain containing			
611	97.6	oe	ccsbBroad304_06998	SRPK1	SRPK family			
612	97.58	kd	CGS001-405	ARNT	Basic helix-loop-helix proteins			
613	97.57	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
614	97.57	kd	CGS001-509	ATP5C1	ATPases / F-type			
615	97.55	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
616	97.55	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
617	97.54	kd	CGS001-54815	GATAD2A	GATA zinc finger domain containing			
618	97.54	kd	CGS001-10491	CRTAP	-			
619	97.5	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
620	97.49	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
621	97.49	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
622	97.46	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
623	97.44	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
624	97.43	kd	CGS001-81539	SLC38A1	System A-like transporters			
625	97.42	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
626	97.38	oe	ccsbBroad304_01013	MIF	-			
627	97.38	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
628	97.37	cp	BRD-K85090592	pilocarpine	Acetylcholine receptor agonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor agonist
629	97.36	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
630	97.35	kd	CGS001-5327	PLAT	Chymotrypsin			
631	97.32	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
632	97.31	kd	CGS001-9261	MAPKAPK2	MAPKAPK subfamily			
633	97.27	kd	CGS001-6257	RXRB	Retinoid X receptors			
634	97.25	kd	CGS001-55193	PBRM1	Non-enzymatic BRD containing proteins			
635	97.24	oe	ccsbBroad304_03848	METTL14	-			
636	97.24	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
637	97.24	kd	CGS001-2004	ELK3	ETS Transcription Factors			
638	97.23	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
639	97.21	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
640	97.21	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
641	97.18	cc		Bromodomain Inhibitor	-			
642	97.17	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
643	97.17	kd	CGS001-539	ATP5O	ATPases / F-type			
644	97.15	kd	CGS001-3717	JAK2	Janus kinase (JakA) family			
645	97.13	oe	ccsbBroad304_00171	BNIP3L	-			
646	97.12	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
647	97.12	kd	CGS001-5045	FURIN	Subtilisin			
648	97.09	oe	ccsbBroad304_02576	MLLT11	-			
649	97.09	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
650	97.06	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
651	97.05	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
652	97.05	cp	BRD-K37516142	idebenone	Calcium channel modulator			Calcium channel modulator
653	97.04	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
654	97.04	oe	ccsbBroad304_05756	ACAA1	-			
655	97.04	kd	CGS001-2730	GCLM	-			
656	97.03	kd	CGS001-203	AK1	Adenylate kinases			
657	97	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
658	96.97	kd	CGS001-599	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
659	96.96	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
660	96.95	oe	ccsbBroad304_02217	FEZ1	-			
661	96.94	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
662	96.94	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
663	96.94	kd	CGS001-727	C5	Endogenous ligands			
664	96.93	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
665	96.93	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
666	96.91	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
667	96.9	kd	CGS001-995	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
668	96.89	oe	ccsbBroad304_00532	F11	Chymotrypsin			
669	96.87	kd	CGS001-6499	SKIV2L	-			
670	96.85	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
671	96.85	kd	CGS001-6720	SREBF1	Basic helix-loop-helix proteins			
672	96.85	kd	CGS001-57459	GATAD2B	GATA zinc finger domain containing			
673	96.84	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
674	96.84	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
675	96.83	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
676	96.83	kd	CGS001-83694	RPS6KL1	RSKL family			
677	96.78	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
678	96.78	kd	CGS001-8767	RIPK2	Receptor interacting protein kinase (RIPK) family			
679	96.77	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
680	96.77	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
681	96.72	oe	ccsbBroad304_07561	YAF2	-			
682	96.72	kd	CGS001-256364	EML3	WD repeat domain containing			
683	96.71	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
684	96.7	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
685	96.69	kd	CGS001-4121	MAN1A1	-			
686	96.69	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
687	96.66	kd	CGS001-159	ADSS	-			
688	96.64	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
689	96.62	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
690	96.61	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
691	96.6	cp	BRD-K31491153	1-phenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
692	96.59	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
693	96.58	kd	CGS001-6778	STAT6	SH2 domain containing			
694	96.57	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
695	96.57	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
696	96.56	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
697	96.51	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
698	96.51	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
699	96.51	kd	CGS001-2101	ESRRA	Estrogen-related receptors			
700	96.5	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
701	96.48	cp	BRD-K29113274	ketoconazole	Sterol demethylase inhibitor		AR, CYP19A1, CYP21A2, CYP2C19, CYP3A5, CYP3A7, KCNA10	Sterol demethylase inhibitor
702	96.48	kd	CGS001-8836	GGH	Gamma-glutamyl hydrolase			
703	96.47	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
704	96.47	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
705	96.47	kd	CGS001-7405	UVRAG	-			
706	96.46	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
707	96.46	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
708	96.45	kd	CGS001-10444	ZER1	ZYG11 cell cycle regulator family			
709	96.45	kd	CGS001-2683	B4GALT1	Beta 4-glycosyltransferases			
710	96.44	kd	CGS001-23013	SPEN	RNA binding motif (RRM) containing			
711	96.43	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
712	96.41	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
713	96.41	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
714	96.4	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
715	96.39	kd	CGS001-57661	PHRF1	Zinc fingers, PHD-type			
716	96.38	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
717	96.38	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
718	96.37	kd	CGS001-6676	SPAG4	-			
719	96.37	kd	CGS001-5992	RFX4	-			
720	96.34	kd	CGS001-26523	EIF2C1	-			
721	96.33	oe	ccsbBroad304_03164	MTERFD1	-			
722	96.33	cp	BRD-K51485625	ritonavir	HIV protease inhibitor		CYP3A4, CYP1A2, CYP2B6, CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
723	96.33	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
724	96.33	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
725	96.31	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
726	96.31	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
727	96.27	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
728	96.27	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
729	96.25	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
730	96.25	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
731	96.24	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
732	96.23	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
733	96.21	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
734	96.2	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
735	96.19	cc		Akt Signaling GOF	-			
736	96.18	oe	ccsbBroad304_06695	PCK2	-			
737	96.16	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
738	96.13	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
739	96.1	kd	CGS001-171017	ZNF384	Zinc fingers, C2H2-type			
740	96.09	kd	CGS001-26039	SS18L1	-			
741	96.09	kd	CGS001-21	ABCA3	ATP binding cassette transporters / subfamily A			
742	96.08	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
743	96.07	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
744	96.05	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
745	96.05	kd	CGS001-2181	ACSL3	Acyl-CoA synthetase family			
746	96.03	cc		MEK inhibitor	-			
747	96.03	oe	ccsbBroad304_01985	EIF3H	-			
748	96	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
749	95.99	kd	CGS001-6678	SPARC	-			
750	95.98	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
751	95.98	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
752	95.97	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
753	95.97	kd	CGS001-81848	SPRY4	-			
754	95.96	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
755	95.94	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
756	95.92	kd	CGS001-701	BUB1B	Bub family			
757	95.9	kd	CGS001-5966	REL	NFkappaB transcription factor family			
758	95.89	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
759	95.88	kd	CGS001-776	CACNA1D	Calcium channel subunits			
760	95.85	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
761	95.85	kd	CGS001-51022	GLRX2	-			
762	95.84	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
763	95.82	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
764	95.81	oe	ccsbBroad304_01617	STX4	-			
765	95.81	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
766	95.8	kd	CGS001-286380	FOXD4L3	-			
767	95.75	kd	CGS001-8727	CTNNAL1	Catenins			
768	95.74	kd	CGS001-4352	MPL	Prolactin receptor family			
769	95.71	oe	ccsbBroad304_01392	TRIM27	-			
770	95.66	oe	ccsbBroad304_01662	TFDP2	-			
771	95.66	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
772	95.66	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
773	95.65	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
774	95.61	oe	ccsbBroad304_13939	MOK	RCK family			
775	95.55	kd	CGS001-9961	MVP	-			
776	95.52	kd	CGS001-3418	IDH2	-			
777	95.51	kd	CGS001-4023	LPL	-			
778	95.49	oe	ccsbBroad304_02052	KYNU	-			
779	95.48	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
780	95.47	oe	ccsbBroad304_03372	CAB39	-			
781	95.47	kd	CGS001-164091	PAQR7	-			
782	95.44	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
783	95.4	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
784	95.4	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
785	95.4	kd	CGS001-1500	CTNND1	Catenins			
786	95.39	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
787	95.39	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
788	95.37	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
789	95.36	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
790	95.34	oe	ccsbBroad304_02367	CALCOCO2	-			
791	95.34	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
792	95.34	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
793	95.33	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
794	95.33	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
795	95.33	kd	CGS001-6309	SC5DL	-			
796	95.33	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
797	95.31	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
798	95.28	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
799	95.25	kd	CGS001-4282	MIF	-			
800	95.24	oe	ccsbBroad304_01102	NMT1	-			
801	95.23	cc		FGFR inhibitor	-			
802	95.22	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
803	95.2	oe	ccsbBroad304_03934	LEPRE1	-			
804	95.2	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
805	95.2	kd	CGS001-54851	ANKRD49	Ankyrin repeat domain containing			
806	95.19	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
807	95.17	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
808	95.17	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
809	95.15	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
810	95.14	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
811	95.14	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
812	95.05	kd	CGS001-5583	PRKCH	Eta subfamily			
813	95	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
814	95	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
815	94.99	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
816	94.98	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
817	94.98	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
818	94.96	oe	ccsbBroad304_07088	TP53	-			
819	94.94	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
820	94.93	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
821	94.9	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
822	94.89	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
823	94.87	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
824	94.86	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
825	94.85	oe	ccsbBroad304_07478	CCP110	-			
826	94.85	kd	CGS001-3176	HNMT	-			
827	94.84	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
828	94.84	kd	CGS001-930	CD19	CD molecules			
829	94.8	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
830	94.77	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
831	94.77	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
832	94.76	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
833	94.69	kd	CGS001-9847	KIAA0528	-			
834	94.68	oe	ccsbBroad304_05758	ACADSB	-			
835	94.67	kd	CGS001-5469	MED1	-			
836	94.65	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
837	94.61	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
838	94.61	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
839	94.6	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
840	94.6	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
841	94.59	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
842	94.56	kd	CGS001-114112	TXNRD3	-			
843	94.55	oe	ccsbBroad304_01401	RIT1	-			
844	94.53	kd	CGS001-53836	GPR87	GPCR / Class A : Orphans			
845	94.52	kd	CGS001-51271	UBAP1	-			
846	94.52	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
847	94.51	kd	CGS001-9415	FADS2	Fatty acid desaturases			
848	94.49	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
849	94.48	kd	CGS001-6658	SOX3	SRY (sex determining region Y)-boxes			
850	94.47	oe	ccsbBroad304_02922	TES	-			
851	94.47	kd	CGS001-8522	GAS7	-			
852	94.45	kd	CGS001-10135	NAMPT	-			
853	94.44	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
854	94.44	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
855	94.43	cc		Beta-adrenergic receptor agonist	-			
856	94.4	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
857	94.38	kd	CGS001-51719	CAB39	-			
858	94.37	kd	CGS001-10180	RBM6	G patch domain containing			
859	94.36	oe	ccsbBroad304_01923	UXT	-			
860	94.34	kd	CGS001-1910	EDNRB	Endothelin receptors			
861	94.33	cp	BRD-K33226500	indinavir	HIV protease inhibitor		CYP3A5	HIV protease inhibitor
862	94.3	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
863	94.26	cc		SRC inhibitor	-			
864	94.25	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
865	94.2	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
866	94.16	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
867	94.15	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
868	94.11	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
869	94.1	kd	CGS001-516	ATP5G1	ATPases / F-type			
870	94.08	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
871	94.08	kd	CGS001-2565	GABRG1	GABA receptors			
872	94.05	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
873	94	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
874	94	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
875	93.99	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
876	93.94	oe	ccsbBroad304_04619	GNG8	-			
877	93.93	kd	CGS001-5699	PSMB10	Proteasome (prosome, macropain) subunits			
878	93.93	kd	CGS001-7001	PRDX2	-			
879	93.91	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
880	93.89	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
881	93.88	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
882	93.85	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
883	93.81	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
884	93.81	kd	CGS001-51203	NUSAP1	-			
885	93.8	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
886	93.74	kd	CGS001-2098	ESD	-			
887	93.72	oe	ccsbBroad304_07349	MAP7	-			
888	93.67	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
889	93.66	oe	ccsbBroad304_06494	KLRC1	CD molecules			
890	93.65	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
891	93.65	kd	CGS001-113878	DTX2	RING-type (C3HC4) zinc fingers			
892	93.64	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
893	93.63	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
894	93.56	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
895	93.55	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
896	93.52	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
897	93.47	kd	CGS001-3799	KIF5B	Kinesins			
898	93.43	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
899	93.42	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
900	93.4	kd	CGS001-3419	IDH3A	-			
901	93.37	kd	CGS001-7424	VEGFC	-			
902	93.37	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
903	93.35	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
904	93.34	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
905	93.34	kd	CGS001-64943	NT5DC2	-			
906	93.33	oe	ccsbBroad304_02653	PRAF2	-			
907	93.33	cp	BRD-A42423104	benproperine	Antitussive			Antitussive
908	93.31	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
909	93.3	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
910	93.29	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
911	93.29	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
912	93.28	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
913	93.26	kd	CGS001-54472	TOLLIP	-			
914	93.26	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
915	93.26	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
916	93.25	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
917	93.25	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
918	93.25	kd	CGS001-1389	CREBL2	basic leucine zipper proteins			
919	93.24	kd	CGS001-3297	HSF1	-			
920	93.22	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
921	93.21	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
922	93.21	kd	CGS001-5066	PAM	-			
923	93.18	oe	ccsbBroad304_09006	RPF1	-			
924	93.16	oe	ccsbBroad304_08167	DNTTIP2	-			
925	93.16	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
926	93.16	kd	CGS001-9231	DLG5	-			
927	93.13	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
928	93.13	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
929	93.08	kd	CGS001-10538	BATF	basic leucine zipper proteins			
930	93.06	kd	CGS001-2295	FOXF2	Forkhead boxes			
931	92.99	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
932	92.98	oe	ccsbBroad304_06237	GAA	Glycosidases			
933	92.97	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
934	92.97	cp	BRD-K51730347	diphencyprone	Immunostimulant			Immunostimulant
935	92.89	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
936	92.89	kd	CGS001-624	BDKRB2	Bradykinin receptors			
937	92.88	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
938	92.87	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
939	92.86	kd	CGS001-8870	IER3	-			
940	92.82	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
941	92.79	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
942	92.78	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
943	92.77	kd	CGS001-2184	FAH	-			
944	92.72	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
945	92.72	cp	BRD-K82143716	flucytosine	Antifungal		DNMT1	Antifungal
946	92.72	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
947	92.66	oe	ccsbBroad304_02579	YWHAQ	-			
948	92.66	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
949	92.62	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
950	92.62	kd	CGS001-4779	NFE2L1	basic leucine zipper proteins			
951	92.59	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
952	92.56	oe	ccsbBroad304_06645	NQO2	-			
953	92.55	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
954	92.55	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
955	92.54	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
956	92.52	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
957	92.52	oe	ccsbBroad304_01211	PKM2	-			
958	92.51	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
959	92.48	kd	CGS001-2308	FOXO1	Forkhead boxes			
960	92.47	oe	ccsbBroad304_06711	PFAS	-			
961	92.45	kd	CGS001-55312	RFK	-			
962	92.43	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
963	92.43	kd	CGS001-10657	KHDRBS1	-			
964	92.42	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
965	92.37	oe	ccsbBroad304_07528	DMTF1	-			
966	92.37	kd	CGS001-103	ADAR	-			
967	92.35	kd	CGS001-2963	GTF2F2	General transcription factors			
968	92.34	kd	CGS001-10493	VAT1	-			
969	92.32	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
970	92.27	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
971	92.26	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
972	92.24	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
973	92.23	kd	CGS001-79722	ANKRD55	Ankyrin repeat domain containing			
974	92.2	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
975	92.16	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
976	92.1	oe	ccsbBroad304_01019	MLH1	-			
977	92.09	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
978	92.06	kd	CGS001-2495	FTH1	-			
979	92.03	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
980	92.02	oe	ccsbBroad304_00316	CKS1B	-			
981	92.02	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
982	92.02	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
983	91.99	kd	CGS001-5584	PRKCI	Iota subfamily			
984	91.97	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
985	91.95	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
986	91.94	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
987	91.92	kd	CGS001-27113	BBC3	-			
988	91.9	kd	CGS001-2731	GLDC	-			
989	91.89	cc		HSP inhibitor	-			
990	91.88	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
991	91.88	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
992	91.86	kd	CGS001-2261	FGFR3	Type V RTKs: FGF (fibroblast growth factor) receptor family			
993	91.85	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
994	91.82	kd	CGS001-64175	LEPRE1	-			
995	91.8	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
996	91.74	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
997	91.66	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
998	91.64	kd	CGS001-9183	ZW10	-			
999	91.64	kd	CGS001-3690	ITGB3	Integrins			
1000	91.63	kd	CGS001-5450	POU2AF1	-			
1001	91.57	cp	BRD-K49404994	levetiracetam	Calcium channel blocker		SV2A, CACNA1B, SCN1A	Calcium channel blocker
1002	91.55	kd	CGS001-474354	LRRC18	-			
1003	91.54	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
1004	91.52	kd	CGS001-3976	LIF	-			
1005	91.5	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
1006	91.48	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
1007	91.48	kd	CGS001-4712	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
1008	91.47	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
1009	91.45	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
1010	91.42	oe	ccsbBroad304_02220	MTFR1	-			
1011	91.4	oe	ccsbBroad304_07238	STK24	YSK subfamily			
1012	91.35	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
1013	91.28	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
1014	91.27	oe	ccsbBroad304_06349	HAGH	-			
1015	91.27	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
1016	91.24	oe	ccsbBroad304_02203	MAD2L1BP	-			
1017	91.23	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
1018	91.23	cp	BRD-A15914070	4-hydroxy-2-nonenal	Cytotoxic lipid peroxidation product		IKBKB	Cytotoxic lipid peroxidation product
1019	91.19	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
1020	91.19	kd	CGS001-58508	MLL3	-			
1021	91.16	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
1022	91.13	kd	CGS001-54107	POLE3	DNA polymerases			
1023	91.12	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
1024	91.11	kd	CGS001-25793	FBXO7	F-boxes / other			
1025	91.11	kd	CGS001-30	ACAA1	-			
1026	91.09	kd	CGS001-2313	FLI1	ETS Transcription Factors			
1027	91.08	kd	CGS001-55437	STRADB	STLK subfamily			
1028	91.06	kd	CGS001-408	ARRB1	-			
1029	91.03	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
1030	91.02	kd	CGS001-3995	FADS3	Fatty acid desaturases			
1031	91.01	kd	CGS001-55214	LEPREL1	-			
1032	90.97	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
1033	90.96	oe	ccsbBroad304_07363	AIFM1	-			
1034	90.96	kd	CGS001-24140	FTSJ1	-			
1035	90.95	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
1036	90.95	kd	CGS001-57026	PDXP	-			
1037	90.93	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
1038	90.92	kd	CGS001-4763	NF1	-			
1039	90.88	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
1040	90.88	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
1041	90.87	kd	CGS001-6241	RRM2	Ribonucleoside-diphosphate reductases			
1042	90.87	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
1043	90.85	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
1044	90.85	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
1045	90.84	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
1046	90.83	oe	ccsbBroad304_08840	KIF9	Kinesins			
1047	90.83	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
1048	90.82	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
1049	90.75	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
1050	90.74	kd	CGS001-9868	TOMM70A	Tetratricopeptide (TTC) repeat domain containing			
1051	90.74	kd	CGS001-9	NAT1	-			
1052	90.73	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
1053	90.7	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
1054	90.68	kd	CGS001-8726	EED	Neutral sphingomyelinase coupling factors			
1055	90.65	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
1056	90.65	oe	ccsbBroad304_00471	E2F6	-			
1057	90.64	kd	CGS001-7389	UROD	-			
1058	90.6	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
1059	90.59	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
1060	90.58	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
1061	90.56	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
1062	90.55	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
1063	90.54	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
1064	90.54	kd	CGS001-221393	GPR115	Adhesion Class GPCRs			
1065	90.53	kd	CGS001-435	ASL	-			
1066	90.51	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
1067	90.51	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
1068	90.49	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
1069	90.49	kd	CGS001-7905	REEP5	Receptor accessory proteins			
1070	90.49	kd	CGS001-55509	BATF3	basic leucine zipper proteins			
1071	90.44	kd	CGS001-7272	TTK	TTK family			
1072	90.44	kd	CGS001-4947	OAZ2	-			
1073	90.41	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
1074	90.38	kd	CGS001-468	ATF4	basic leucine zipper proteins			
1075	90.36	oe	ccsbBroad304_00147	BAG1	-			
1076	90.36	kd	CGS001-4717	NDUFC1	Mitochondrial respiratory chain complex / Complex I			
1077	90.34	oe	ccsbBroad304_03658	DCP1A	-			
1078	90.32	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
1079	90.3	kd	CGS001-122809	SOCS4	SH2 domain containing			
1080	90.28	oe	ccsbBroad304_06383	HMMR	CD molecules			
1081	90.27	oe	ccsbBroad304_05547	TMEM110	-			
1082	90.27	oe	ccsbBroad304_06013	CLPTM1	-			
1083	90.26	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
1084	90.26	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
1085	90.24	oe	ccsbBroad304_03415	GFOD1	-			
1086	90.23	kd	CGS001-5352	PLOD2	-			
1087	90.22	oe	ccsbBroad304_08694	TBX20	T-boxes			
1088	90.21	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
1089	90.17	cc		Reverse transcriptase inhibitor	-			
1090	90.17	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
1091	90.14	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
1092	90.08	oe	ccsbBroad304_08952	E2F8	-			
1093	90.08	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1094	90.08	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
1095	90.07	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
1096	90.06	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
1097	90.02	kd	CGS001-3225	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
1098	90.01	kd	CGS001-80714	PBX4	Homeoboxes / TALE class			
1099	90.01	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
1100	90	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
1101	89.94	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
1102	89.93	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
1103	89.91	cp	BRD-K04196797	oxcarbazepine	Sodium channel blocker		CYP2C19, CYP3A4, CYP3A5, SCN1A, SCN3A, SCN5A	Sodium channel blocker
1104	89.88	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
1105	89.84	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
1106	89.81	kd	CGS001-3665	IRF7	-			
1107	89.7	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
1108	89.68	oe	ccsbBroad304_00956	LYZ	-			
1109	89.65	kd	CGS001-2770	GNAI1	-			
1110	89.63	kd	CGS001-161725	OTUD7A	OTU domain containing			
1111	89.58	kd	CGS001-3376	IARS	Aminoacyl tRNA synthetases / Class I			
1112	89.57	kd	CGS001-8974	P4HA2	-			
1113	89.55	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
1114	89.54	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
1115	89.5	kd	CGS001-1810	DR1	-			
1116	89.48	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
1117	89.44	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
1118	89.44	oe	ccsbBroad304_00962	SMAD4	SMADs			
1119	89.44	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
1120	89.44	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
1121	89.44	kd	CGS001-5624	PROC	Endogenous ligands			
1122	89.44	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
1123	89.41	kd	CGS001-5979	RET	Type XIV RTKs: RET			
1124	89.39	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
1125	89.35	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
1126	89.32	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
1127	89.32	kd	CGS001-10247	HRSP12	-			
1128	89.27	cp	BRD-K99447003	enalaprilat	ACE inhibitor		ACE	ACE inhibitor
1129	89.24	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
1130	89.24	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
1131	89.22	kd	CGS001-9360	PPIG	-			
1132	89.21	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
1133	89.2	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
1134	89.2	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
1135	89.18	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
1136	89.15	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
1137	89.15	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
1138	89.13	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
1139	89.12	kd	CGS001-1635	DCTD	-			
1140	89.11	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1141	89.03	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
1142	89.02	kd	CGS001-1154	CISH	SH2 domain containing			
1143	89.01	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
1144	89.01	kd	CGS001-84759	PCGF1	Polycomb group ring fingers			
1145	88.99	kd	CGS001-56848	SPHK2	Sphingosine kinase			
1146	88.99	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1147	88.92	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
1148	88.91	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
1149	88.9	kd	CGS001-139135	PASD1	-			
1150	88.89	kd	CGS001-54881	TEX10	-			
1151	88.86	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
1152	88.86	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
1153	88.83	kd	CGS001-7082	TJP1	-			
1154	88.76	kd	CGS001-3046	HBE1	-			
1155	88.74	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
1156	88.73	kd	CGS001-4094	MAF	-			
1157	88.68	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
1158	88.67	kd	CGS001-51335	NGRN	-			
1159	88.61	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
1160	88.61	kd	CGS001-3482	IGF2R	CD molecules			
1161	88.59	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
1162	88.59	oe	ccsbBroad304_02002	RNMT	-			
1163	88.57	kd	CGS001-1843	DUSP1	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1164	88.51	kd	CGS001-11116	FGFR1OP	-			
1165	88.47	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1166	88.45	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
1167	88.43	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
1168	88.39	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
1169	88.37	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
1170	88.35	kd	CGS001-55937	APOM	Apolipoproteins			
1171	88.34	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
1172	88.33	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
1173	88.31	kd	CGS001-4507	MTAP	-			
1174	88.25	kd	CGS001-3170	FOXA2	Forkhead boxes			
1175	88.21	cc		Nucleoside reverse transcriptase inhibitor	-			
1176	88.21	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
1177	88.2	kd	CGS001-6884	TAF13	-			
1178	88.18	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
1179	88.14	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
1180	88.08	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
1181	88.02	kd	CGS001-10957	PNRC1	-			
1182	88.01	kd	CGS001-375	ARF1	ADP-ribosylation factors			
1183	88.01	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
1184	87.92	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
1185	87.91	kd	CGS001-10906	TRAFD1	-			
1186	87.9	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
1187	87.9	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
1188	87.85	oe	ccsbBroad304_03121	NRBF2	-			
1189	87.84	cp	BRD-K22009844	phenprobamate	Muscle relaxant			Muscle relaxant
1190	87.81	kd	CGS001-147837	ZNF563	Zinc fingers, C2H2-type			
1191	87.8	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
1192	87.77	kd	CGS001-4194	MDM4	-			
1193	87.74	oe	ccsbBroad304_01651	TCF7L2	-			
1194	87.72	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
1195	87.69	kd	CGS001-58497	PRUNE	-			
1196	87.67	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
1197	87.67	cp	BRD-K85503079	perospirone	Dopamine receptor antagonist		DRD2, HTR2A, DRD3, DRD4, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
1198	87.67	kd	CGS001-51655	RASD1	-			
1199	87.65	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
1200	87.64	oe	ccsbBroad304_05590	NOTCH2NL	-			
1201	87.61	kd	CGS001-7982	ST7	-			
1202	87.6	kd	CGS001-328	APEX1	-			
1203	87.55	oe	ccsbBroad304_04170	PANK2	-			
1204	87.49	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
1205	87.49	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
1206	87.46	oe	ccsbBroad304_05757	ACADS	-			
1207	87.46	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
1208	87.45	kd	CGS001-3755	KCNG1	Voltage-gated potassium channels			
1209	87.44	kd	CGS001-1984	EIF5A	-			
1210	87.4	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
1211	87.39	oe	ccsbBroad304_06286	GLUL	-			
1212	87.38	kd	CGS001-10477	UBE2E3	Ubiquitin-conjugating enzymes E2			
1213	87.37	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
1214	87.36	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
1215	87.29	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
1216	87.26	kd	CGS001-2919	CXCL1	Endogenous ligands			
1217	87.25	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
1218	87.18	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
1219	87.15	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
1220	87.11	oe	ccsbBroad304_01008	KITLG	-			
1221	87.08	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
1222	87.07	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
1223	87.06	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
1224	87.02	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
1225	87.01	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
1226	87	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
1227	87	kd	CGS001-4205	MEF2A	Myocyte enhancer factors			
1228	86.99	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
1229	86.95	kd	CGS001-8996	NOL3	-			
1230	86.95	kd	CGS001-9258	MFHAS1	-			
1231	86.93	kd	CGS001-23710	GABARAPL1	-			
1232	86.92	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
1233	86.91	cp	BRD-K62858456	lomerizine	Calcium channel blocker		ABCB1, CACNA1B, SCN5A	Calcium channel blocker
1234	86.91	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
1235	86.91	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
1236	86.89	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
1237	86.85	kd	CGS001-8480	RAE1	WD repeat domain containing			
1238	86.84	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
1239	86.76	kd	CGS001-23212	RRS1	-			
1240	86.75	oe	ccsbBroad304_02361	MFSD10	-			
1241	86.74	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
1242	86.72	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
1243	86.65	kd	CGS001-2149	F2R	Protease activated receptors			
1244	86.58	oe	ccsbBroad304_00424	DBI	-			
1245	86.45	kd	CGS001-29937	NENF	-			
1246	86.37	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
1247	86.35	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
1248	86.35	kd	CGS001-833	CARS	Aminoacyl tRNA synthetases / Class I			
1249	86.34	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
1250	86.34	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
1251	86.32	kd	CGS001-7533	YWHAH	-			
1252	86.32	kd	CGS001-323	APBB2	-			
1253	86.23	kd	CGS001-3651	PDX1	Homeoboxes / ANTP class : HOXL subclass			
1254	86.22	kd	CGS001-9455	HOMER2	-			
1255	86.15	kd	CGS001-4088	SMAD3	SMADs			
1256	86.15	kd	CGS001-286530	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
1257	86.07	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
1258	86.02	oe	ccsbBroad304_08339	CMPK1	-			
1259	86.02	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
1260	85.93	kd	CGS001-4323	MMP14	Matrix metallopeptidase			
1261	85.9	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1262	85.84	kd	CGS001-80758	PRR7	-			
1263	85.8	oe	ccsbBroad304_00063	AMPD2	-			
1264	85.78	oe	ccsbBroad304_07118	UGDH	-			
1265	85.74	kd	CGS001-10413	YAP1	Hippo Signaling			
1266	85.66	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
1267	85.66	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
1268	85.64	oe	ccsbBroad304_03357	RASD1	-			
1269	85.63	kd	CGS001-7150	TOP1	DNA Topoisomerases			
1270	85.62	cc		Tachykinin antagonist	-			
1271	85.62	cp	BRD-K34437622	BRD-K34437622	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
1272	85.61	kd	CGS001-192669	EIF2C3	-			
1273	85.57	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
1274	85.48	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
1275	85.47	kd	CGS001-117581	TWIST2	Basic helix-loop-helix proteins			
1276	85.39	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
1277	85.38	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
1278	85.32	oe	ccsbBroad304_01532	SIAH1	-			
1279	85.32	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
1280	85.31	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
1281	85.3	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
1282	85.3	kd	CGS001-1837	DTNA	-			
1283	85.29	kd	CGS001-8801	SUCLG2	-			
1284	85.28	kd	CGS001-9767	PHF16	-			
1285	85.25	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
1286	85.23	kd	CGS001-23266	LPHN2	Adhesion Class GPCRs			
1287	85.2	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
1288	85.19	cc		Na-K-Cl transporter inhibitor	-			
1289	85.18	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
1290	85.16	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1291	85.13	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
1292	85.13	oe	ccsbBroad304_10758	CTBP2	-			
1293	85.08	kd	CGS001-3203	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
1294	85.07	cc		KCNJ11 modulator	-			
1295	85.07	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
1296	85.06	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
1297	85.06	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
1298	84.91	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
1299	84.9	kd	CGS001-8800	PEX11A	-			
1300	84.79	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
1301	84.76	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
1302	84.72	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
1303	84.72	kd	CGS001-427	ASAH1	Acid ceramidase			
1304	84.71	kd	CGS001-9290	GPR55	GPCR / Class A : Orphans			
1305	84.7	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
1306	84.7	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
1307	84.67	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
1308	84.67	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
1309	84.67	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
1310	84.67	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
1311	84.64	oe	ccsbBroad304_01674	TIMP4	-			
1312	84.63	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
1313	84.63	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
1314	84.62	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
1315	84.6	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
1316	84.6	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
1317	84.59	kd	CGS001-9181	ARHGEF2	Rho guanine nucleotide exchange factors			
1318	84.57	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
1319	84.54	kd	CGS001-8864	PER2	-			
1320	84.5	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
1321	84.49	kd	CGS001-808	CALM3	EF-hand domain containing			
1322	84.45	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
1323	84.43	kd	CGS001-5428	POLG	DNA polymerases			
1324	84.42	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
1325	84.37	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
1326	84.33	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
1327	84.33	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
1328	84.32	kd	CGS001-57121	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1329	84.32	kd	CGS001-30001	ERO1L	-			
1330	84.26	kd	CGS001-1736	DKC1	-			
1331	84.26	kd	CGS001-84875	PARP10	Poly (ADP-ribose) polymerases			
1332	84.25	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
1333	84.22	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
1334	84.17	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
1335	84.12	kd	CGS001-118738	ZNF488	Zinc fingers, C2H2-type			
1336	84.12	kd	CGS001-9380	GRHPR	-			
1337	84.11	kd	CGS001-58533	SNX6	Sorting nexins			
1338	84.1	oe	ccsbBroad304_02243	DLGAP5	-			
1339	83.99	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
1340	83.9	kd	CGS001-8548	BLZF1	-			
1341	83.89	kd	CGS001-8508	NIPSNAP1	-			
1342	83.88	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
1343	83.87	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
1344	83.87	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
1345	83.83	oe	ccsbBroad304_01203	PIM1	PIM family			
1346	83.82	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
1347	83.8	kd	CGS001-9189	ZBED1	Pseudoautosomal regions / PAR1			
1348	83.76	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
1349	83.75	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
1350	83.75	kd	CGS001-65975	STK33	CAMK-unique family			
1351	83.72	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
1352	83.71	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
1353	83.67	cp	BRD-K40758068	efavirenz	HIV protease inhibitor		CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5	HIV protease inhibitor
1354	83.65	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
1355	83.62	kd	CGS001-4090	SMAD5	SMADs			
1356	83.56	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1357	83.47	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
1358	83.46	cc		Cyclins LOF	-			
1359	83.42	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
1360	83.37	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
1361	83.35	oe	ccsbBroad304_13952	SHMT2	-			
1362	83.35	kd	CGS001-275	AMT	-			
1363	83.31	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
1364	83.25	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
1365	83.22	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
1366	83.22	kd	CGS001-8428	STK24	YSK subfamily			
1367	83.19	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
1368	83.14	kd	CGS001-10887	PROKR1	GPCR / Class A : Prokineticin receptors			
1369	83.13	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
1370	83.04	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1371	83.03	cp	BRD-K96134740	kitasamycin	Protein synthesis inhibitor			Protein synthesis inhibitor
1372	83.03	kd	CGS001-283455	KSR2	RAF family			
1373	83.02	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
1374	82.99	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
1375	82.99	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1376	82.99	oe	ccsbBroad304_01469	RSU1	-			
1377	82.98	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
1378	82.97	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
1379	82.9	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
1380	82.89	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
1381	82.88	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
1382	82.88	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
1383	82.84	kd	CGS001-3663	IRF5	-			
1384	82.81	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1385	82.8	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
1386	82.79	kd	CGS001-7090	TLE3	WD repeat domain containing			
1387	82.74	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
1388	82.74	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
1389	82.74	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
1390	82.73	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
1391	82.72	kd	CGS001-9817	KEAP1	Kelch-like proteins			
1392	82.66	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
1393	82.65	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
1394	82.63	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
1395	82.59	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
1396	82.58	oe	ccsbBroad304_02708	TRIM32	-			
1397	82.57	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
1398	82.56	kd	CGS001-23621	BACE1	Pepsin			
1399	82.54	cp	BRD-K44094599	tacrolimus	Calcineurin inhibitor		FKBP1A, CYP3A5, CYP3A7	Calcineurin inhibitor
1400	82.53	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
1401	82.53	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
1402	82.5	oe	ccsbBroad304_06745	PNN	-			
1403	82.5	oe	ccsbBroad304_03405	CHRAC1	-			
1404	82.5	kd	CGS001-3416	IDE	Pitrilysin			
1405	82.49	kd	CGS001-1643	DDB2	WD repeat domain containing			
1406	82.44	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1407	82.43	kd	CGS001-2242	FES	Fer family			
1408	82.41	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
1409	82.4	oe	ccsbBroad304_00155	CCND1	-			
1410	82.38	kd	CGS001-57680	CHD8	-			
1411	82.23	kd	CGS001-24148	PRPF6	-			
1412	82.22	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
1413	82.21	kd	CGS001-10476	ATP5H	ATPases / F-type			
1414	82.21	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
1415	82.18	kd	CGS001-3030	HADHA	-			
1416	82.18	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
1417	82.11	kd	CGS001-79071	ELOVL6	-			
1418	82.1	kd	CGS001-2118	ETV4	ETS Transcription Factors			
1419	82.03	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
1420	82.02	kd	CGS001-3177	SLC29A2	SLC29 family			
1421	82.01	cp	BRD-K56450366	NSC-94258	Antineoplastic		AKR1B1, CYP19A1, HSD17B1	Antineoplastic
1422	81.97	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
1423	81.95	oe	ccsbBroad304_00632	GGCX	Carboxylases			
1424	81.93	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
1425	81.89	kd	CGS001-5618	PRLR	Prolactin receptor family			
1426	81.87	kd	CGS001-11168	PSIP1	-			
1427	81.86	kd	CGS001-26959	HBP1	-			
1428	81.85	kd	CGS001-64087	MCCC2	-			
1429	81.81	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
1430	81.8	kd	CGS001-116519	APOA5	Apolipoproteins			
1431	81.79	kd	CGS001-4795	NFKBIL1	-			
1432	81.78	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
1433	81.74	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
1434	81.67	kd	CGS001-7965	AIMP2	-			
1435	81.65	cc		Wnt family GOF	-			
1436	81.65	oe	ccsbBroad304_00226	CAV1	-			
1437	81.62	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1438	81.61	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
1439	81.58	kd	CGS001-34	ACADM	-			
1440	81.54	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
1441	81.52	kd	CGS001-8878	SQSTM1	-			
1442	81.51	kd	CGS001-573	BAG1	-			
1443	81.49	kd	CGS001-54807	ZNF586	Zinc fingers, C2H2-type			
1444	81.46	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
1445	81.43	oe	ccsbBroad304_01605	SSX2	-			
1446	81.39	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
1447	81.3	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
1448	81.26	cc		GPCR Subset GOF	-			
1449	81.26	cc		Bile acid	-			
1450	81.26	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
1451	81.19	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
1452	81.07	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
1453	81.07	kd	CGS001-1468	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
1454	80.99	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
1455	80.99	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
1456	80.94	cc		Serotonin receptor antagonist	-			
1457	80.94	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
1458	80.89	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
1459	80.88	kd	CGS001-467	ATF3	basic leucine zipper proteins			
1460	80.86	kd	CGS001-4688	NCF2	Tetratricopeptide (TTC) repeat domain containing			
1461	80.84	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1462	80.84	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
1463	80.74	kd	CGS001-4916	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
1464	80.69	oe	ccsbBroad304_01398	RHEB	-			
1465	80.69	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
1466	80.62	oe	ccsbBroad304_00392	CTLA4	CD molecules			
1467	80.61	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
1468	80.6	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1469	80.59	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
1470	80.57	kd	CGS001-5710	PSMD4	Proteasome (prosome, macropain) subunits			
1471	80.53	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1472	80.51	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
1473	80.5	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
1474	80.49	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
1475	80.47	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
1476	80.42	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
1477	80.39	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
1478	80.38	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
1479	80.33	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
1480	80.32	kd	CGS001-23635	SSBP2	-			
1481	80.27	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1482	80.11	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
1483	80.07	kd	CGS001-9791	PTDSS1	-			
1484	80.05	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
1485	80.05	kd	CGS001-9587	MAD2L1BP	-			
1486	80.03	oe	ccsbBroad304_00658	GNG5	-			
1487	80.01	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
1488	80	kd	CGS001-2119	ETV5	ETS Transcription Factors			
1489	79.93	kd	CGS001-6727	SRP14	-			
1490	79.9	kd	CGS001-7342	UBP1	-			
1491	79.89	kd	CGS001-27347	STK39	FRAY subfamily			
1492	79.85	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
1493	79.85	kd	CGS001-151742	PPM1L	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1494	79.79	oe	ccsbBroad304_02057	P4HA2	-			
1495	79.77	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
1496	79.76	oe	ccsbBroad304_01661	TFCP2	-			
1497	79.75	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
1498	79.75	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1499	79.69	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
1500	79.55	kd	CGS001-8573	CASK	CASK family			
1501	79.53	oe	ccsbBroad304_00077	APEX1	-			
1502	79.53	kd	CGS001-8495	PPFIBP2	Sterile alpha motif (SAM) domain containing			
1503	79.53	oe	ccsbBroad304_07598	PEMT	-			
1504	79.52	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
1505	79.5	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
1506	79.49	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
1507	79.45	kd	CGS001-10312	TCIRG1	ATPases / V-type			
1508	79.38	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
1509	79.38	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
1510	79.31	oe	ccsbBroad304_00529	F3	CD molecules			
1511	79.21	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
1512	79.2	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
1513	79.16	cp	BRD-A37052580	physostigmine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Cholinesterase inhibitor
1514	79.16	kd	CGS001-10991	SLC38A3	System N-like transporters			
1515	79.15	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
1516	79.04	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
1517	79.04	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
1518	79.02	kd	CGS001-168374	ZNF92	Zinc fingers, C2H2-type			
1519	78.99	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1520	78.98	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
1521	78.98	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
1522	78.96	kd	CGS001-7917	BAG6	-			
1523	78.95	cc		Estrogen receptor antagonist	-			
1524	78.95	oe	ccsbBroad304_01091	NFIB	-			
1525	78.94	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
1526	78.92	kd	CGS001-1196	CLK2	CDC-like kinases			
1527	78.85	cc		Calcium channel blocker	-			
1528	78.84	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
1529	78.78	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
1530	78.78	kd	CGS001-11232	POLG2	DNA polymerases			
1531	78.74	cc		Serotonin receptor agonist	-			
1532	78.69	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
1533	78.69	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
1534	78.68	cc		TGF beta receptor inhibitor	-			
1535	78.64	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
1536	78.57	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
1537	78.57	kd	CGS001-5053	PAH	Amino acid hydroxylases			
1538	78.57	kd	CGS001-10553	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
1539	78.46	kd	CGS001-8650	NUMB	-			
1540	78.45	kd	CGS001-7936	RDBP	-			
1541	78.42	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
1542	78.39	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
1543	78.39	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
1544	78.3	kd	CGS001-9943	OXSR1	FRAY subfamily			
1545	78.28	kd	CGS001-154197	PNLDC1	-			
1546	78.22	kd	CGS001-80762	NDFIP1	-			
1547	78.21	oe	ccsbBroad304_08386	SMOX	-			
1548	78.21	kd	CGS001-87	ACTN1	EF-hand domain containing			
1549	78.1	cc		X linked mental retardation group 1 LOF	-			
1550	78.03	oe	ccsbBroad304_00390	CTGF	-			
1551	78.01	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
1552	77.99	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
1553	77.97	kd	CGS001-22891	ZNF365	Zinc fingers, C2H2-type			
1554	77.96	kd	CGS001-10810	WASF3	-			
1555	77.95	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
1556	77.95	kd	CGS001-29978	UBQLN2	Ubiquilin family			
1557	77.89	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
1558	77.85	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
1559	77.79	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
1560	77.73	kd	CGS001-664	BNIP3	-			
1561	77.7	oe	ccsbBroad304_02738	RRS1	-			
1562	77.68	kd	CGS001-58492	ZNF77	Zinc fingers, C2H2-type			
1563	77.6	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
1564	77.58	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
1565	77.57	kd	CGS001-8802	SUCLG1	-			
1566	77.54	oe	ccsbBroad304_01664	TGFA	-			
1567	77.5	kd	CGS001-253430	IPMK	-			
1568	77.47	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
1569	77.44	oe	ccsbBroad304_07851	FAM120A	-			
1570	77.44	kd	CGS001-170591	S100Z	EF-hand domain containing			
1571	77.43	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
1572	77.4	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
1573	77.39	kd	CGS001-3708	ITPR1	Ion channels / Inositol triphosphate receptors			
1574	77.38	oe	ccsbBroad304_02964	TIMM9	-			
1575	77.38	kd	CGS001-170463	SSBP4	-			
1576	77.38	kd	CGS001-5359	PLSCR1	-			
1577	77.37	kd	CGS001-353	APRT	-			
1578	77.26	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
1579	77.25	kd	CGS001-10153	CEBPZ	-			
1580	77.24	oe	ccsbBroad304_04257	SPRY4	-			
1581	77.17	kd	CGS001-4833	NME4	-			
1582	77.12	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
1583	77.06	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
1584	77.02	kd	CGS001-8669	EIF3J	-			
1585	77.01	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
1586	77.01	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
1587	76.99	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
1588	76.84	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
1589	76.81	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
1590	76.78	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
1591	76.73	kd	CGS001-10652	YKT6	-			
1592	76.68	oe	ccsbBroad304_00009	ACLY	-			
1593	76.67	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
1594	76.66	oe	ccsbBroad304_07097	TRAF1	-			
1595	76.62	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
1596	76.58	kd	CGS001-6827	SUPT4H1	-			
1597	76.53	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
1598	76.47	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
1599	76.4	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1600	76.39	kd	CGS001-2580	GAK	Heat shock proteins / DNAJ (HSP40)			
1601	76.32	oe	ccsbBroad304_04399	PGBD1	-			
1602	76.29	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
1603	76.19	kd	CGS001-10412	NSA2	-			
1604	76.17	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
1605	76.13	kd	CGS001-6813	STXBP2	-			
1606	76.12	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
1607	76.1	kd	CGS001-28512	NKIRAS1	-			
1608	76.03	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
1609	76.01	kd	CGS001-5580	PRKCD	Delta subfamily			
1610	76	oe	ccsbBroad304_07506	UBAP2L	-			
1611	75.99	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
1612	75.93	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
1613	75.91	cc		ATP synthase inhibitor	-			
1614	75.87	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
1615	75.87	kd	CGS001-5563	PRKAA2	AMPK subfamily			
1616	75.81	cp	BRD-K05350981	oligomycin-c	ATPase inhibitor		ATP5A1	ATPase inhibitor, ATP synthase inhibitor
1617	75.81	kd	CGS001-2335	FN1	Endogenous ligands			
1618	75.77	kd	CGS001-25898	RCHY1	RING-type (C3HC4) zinc fingers			
1619	75.77	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
1620	75.74	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
1621	75.74	cp	BRD-K81916719	triclabendazole	Microtubule inhibitor		DNMT1	Microtubule inhibitor
1622	75.71	oe	ccsbBroad304_01114	NUP88	-			
1623	75.71	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
1624	75.7	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
1625	75.68	oe	ccsbBroad304_06098	DHCR24	-			
1626	75.67	kd	CGS001-335	APOA1	Apolipoproteins			
1627	75.65	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
1628	75.64	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1629	75.64	kd	CGS001-23405	DICER1	-			
1630	75.63	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
1631	75.62	kd	CGS001-3065	HDAC1	Histone deacetylases			
1632	75.58	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
1633	75.58	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
1634	75.51	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
1635	75.47	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1636	75.46	kd	CGS001-23043	TNIK	MSN subfamily			
1637	75.46	kd	CGS001-3688	ITGB1	Integrins			
1638	75.44	kd	CGS001-1387	CREBBP	Chromatin-modifying enzymes / K-acetyltransferases			
1639	75.32	kd	CGS001-333929	SNAI3	Snail homologs			
1640	75.29	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1641	75.25	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1642	75.23	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
1643	75.21	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
1644	75.21	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
1645	75.21	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1646	75.12	kd	CGS001-1429	CRYZ	-			
1647	75.11	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
1648	75.11	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
1649	75.06	oe	ccsbBroad304_00464	DTNA	-			
1650	75.03	oe	ccsbBroad304_03191	NOSIP	-			
1651	74.99	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
1652	74.99	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
1653	74.99	kd	CGS001-3566	IL4R	IL-2 receptor family			
1654	74.95	kd	CGS001-23012	STK38L	NDR family			
1655	74.92	kd	CGS001-55038	CDCA4	-			
1656	74.91	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
1657	74.9	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
1658	74.89	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
1659	74.88	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1660	74.88	kd	CGS001-1738	DLD	-			
1661	74.83	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1662	74.76	oe	ccsbBroad304_02737	JMJD6	-			
1663	74.73	oe	ccsbBroad304_12106	PXK	Slob family			
1664	74.63	oe	ccsbBroad304_01372	RALB	-			
1665	74.62	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
1666	74.56	oe	ccsbBroad304_06367	HK1	-			
1667	74.52	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
1668	74.34	kd	CGS001-2717	GLA	-			
1669	74.27	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
1670	74.25	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
1671	74.22	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1672	74.17	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
1673	74.05	kd	CGS001-326	AIRE	Zinc fingers, PHD-type			
1674	73.99	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
1675	73.98	kd	CGS001-3927	LASP1	-			
1676	73.96	kd	CGS001-3094	HINT1	-			
1677	73.93	oe	ccsbBroad304_06820	PTS	-			
1678	73.91	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
1679	73.88	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
1680	73.88	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
1681	73.85	kd	CGS001-6608	SMO	GPCR / Class F : Frizzled receptors			
1682	73.83	kd	CGS001-4316	MMP7	Matrix metallopeptidase			
1683	73.72	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
1684	73.68	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
1685	73.66	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1686	73.66	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
1687	73.6	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
1688	73.59	oe	ccsbBroad304_07592	CEPT1	-			
1689	73.53	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1690	73.51	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
1691	73.46	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
1692	73.46	kd	CGS001-79006	METRN	-			
1693	73.45	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
1694	73.4	kd	CGS001-3486	IGFBP3	insulin-like growth factor (IGF) binding proteins			
1695	73.37	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
1696	73.35	cc		Homeobox Gene GOF	-			
1697	73.35	cc		Rho GTPase activating proteins LOF	-			
1698	73.34	kd	CGS001-23131	GPATCH8	G patch domain containing			
1699	73.33	kd	CGS001-595	CCND1	-			
1700	73.31	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
1701	73.27	oe	ccsbBroad304_00469	DUT	-			
1702	73.21	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
1703	73.13	kd	CGS001-2787	GNG5	-			
1704	73.12	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
1705	73.11	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
1706	73.07	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
1707	73.06	kd	CGS001-9134	CCNE2	-			
1708	73.05	kd	CGS001-8148	TAF15	RNA binding motif (RRM) containing			
1709	73.04	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
1710	72.94	oe	ccsbBroad304_04626	EGLN3	-			
1711	72.93	kd	CGS001-865	CBFB	-			
1712	72.92	oe	ccsbBroad304_07875	SPECC1L	-			
1713	72.92	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
1714	72.84	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
1715	72.83	kd	CGS001-54901	CDKAL1	-			
1716	72.8	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
1717	72.8	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
1718	72.77	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
1719	72.71	kd	CGS001-5170	PDPK1	PDK1 family			
1720	72.7	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
1721	72.63	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
1722	72.61	oe	ccsbBroad304_12008	NLK	nmo subfamily			
1723	72.61	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
1724	72.47	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
1725	72.4	kd	CGS001-975	CD81	CD molecules			
1726	72.37	oe	ccsbBroad304_07704	SUB1	-			
1727	72.37	oe	ccsbBroad304_03433	DDIT4	-			
1728	72.32	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
1729	72.31	kd	CGS001-5910	RAP1GDS1	Armadillo repeat containing			
1730	72.3	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
1731	72.3	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
1732	72.28	kd	CGS001-64783	RBM15	RNA binding motif (RRM) containing			
1733	72.25	kd	CGS001-4016	LOXL1	-			
1734	72.17	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
1735	72.14	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
1736	72.09	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
1737	72.08	kd	CGS001-7625	ZNF74	Zinc fingers, C2H2-type			
1738	72.07	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1739	72.03	kd	CGS001-26277	TINF2	-			
1740	72	kd	CGS001-5887	RAD23B	-			
1741	71.99	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
1742	71.96	oe	ccsbBroad304_02372	SPRY1	-			
1743	71.94	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
1744	71.86	kd	CGS001-80135	RPF1	-			
1745	71.85	kd	CGS001-4771	NF2	A-kinase anchor proteins			
1746	71.76	oe	ccsbBroad304_01832	PAX8	Paired boxes			
1747	71.76	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
1748	71.75	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
1749	71.66	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
1750	71.62	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
1751	71.6	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
1752	71.55	kd	CGS001-57720	GPR107	GPCR / Unclassified : 7TM orphan receptors			
1753	71.54	kd	CGS001-2071	ERCC3	General transcription factors			
1754	71.52	kd	CGS001-7415	VCP	ATPases / AAA-type			
1755	71.46	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
1756	71.44	oe	ccsbBroad304_03444	PAF1	-			
1757	71.44	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
1758	71.32	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
1759	71.24	kd	CGS001-122402	TDRD9	Tudor domain containing			
1760	71.21	oe	ccsbBroad304_13633	PI4KAP2	-			
1761	71.19	kd	CGS001-84328	LZIC	-			
1762	71.15	kd	CGS001-7852	CXCR4	Chemokine receptors			
1763	71.08	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
1764	71.06	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
1765	70.91	kd	CGS001-598	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1766	70.89	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
1767	70.86	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
1768	70.85	kd	CGS001-27035	NOX1	-			
1769	70.73	kd	CGS001-93594	WDR67	-			
1770	70.7	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
1771	70.6	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
1772	70.53	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
1773	70.52	kd	CGS001-4773	NFATC2	Nuclear factor of activated T-cells			
1774	70.39	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
1775	70.31	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
1776	70.27	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
1777	70.15	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
1778	70.15	kd	CGS001-3586	IL10	Interleukins and interleukin receptors			
1779	70.09	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1780	70.04	kd	CGS001-5612	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
1781	70.02	kd	CGS001-466	ATF1	basic leucine zipper proteins			
1782	70.01	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
1783	70.01	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
1784	69.97	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
1785	69.93	kd	CGS001-790	CAD	-			
1786	69.92	cp	BRD-K70883034	nimetazepam	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA receptor agonist
1787	69.89	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
1788	69.87	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
1789	69.84	kd	CGS001-1356	CP	-			
1790	69.74	kd	CGS001-51002	TPRKB	-			
1791	69.73	kd	CGS001-5906	RAP1A	-			
1792	69.71	oe	ccsbBroad304_02566	MORF4L1	-			
1793	69.68	oe	ccsbBroad304_03040	NKIRAS2	-			
1794	69.65	kd	CGS001-6925	TCF4	Basic helix-loop-helix proteins			
1795	69.62	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
1796	69.58	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
1797	69.53	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
1798	69.46	oe	ccsbBroad304_07140	XPC	-			
1799	69.44	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
1800	69.44	kd	CGS001-79733	E2F8	-			
1801	69.43	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
1802	69.42	oe	ccsbBroad304_02702	MSRB2	-			
1803	69.4	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
1804	69.3	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
1805	69.29	kd	CGS001-4798	NFRKB	INO80 complex subunits			
1806	69.21	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
1807	69.17	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
1808	69.09	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
1809	68.95	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
1810	68.94	oe	ccsbBroad304_00221	CASP3	Caspases			
1811	68.93	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
1812	68.9	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
1813	68.86	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
1814	68.83	oe	ccsbBroad304_03591	ETNK1	-			
1815	68.8	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
1816	68.71	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
1817	68.71	kd	CGS001-3315	HSPB1	Heat shock proteins / HSPB			
1818	68.67	oe	ccsbBroad304_03386	SPA17	-			
1819	68.66	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
1820	68.66	kd	CGS001-5049	PAFAH1B2	-			
1821	68.64	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
1822	68.61	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
1823	68.49	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
1824	68.48	kd	CGS001-397	ARHGDIB	Endogenous ligands			
1825	68.46	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
1826	68.43	oe	ccsbBroad304_00747	HLF	-			
1827	68.41	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
1828	68.34	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
1829	68.32	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
1830	68.27	oe	ccsbBroad304_00394	CTSD	Cathepsins			
1831	68.23	kd	CGS001-9061	PAPSS1	-			
1832	68.2	kd	CGS001-7078	TIMP3	-			
1833	68.2	kd	CGS001-51447	IP6K2	-			
1834	68.15	oe	ccsbBroad304_00725	HADHA	-			
1835	68.14	oe	ccsbBroad304_06048	CRYZ	-			
1836	68.06	oe	ccsbBroad304_02500	RRAGA	-			
1837	68.06	kd	CGS001-894	CCND2	-			
1838	68.04	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
1839	68.03	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
1840	67.95	kd	CGS001-586	BCAT1	-			
1841	67.94	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
1842	67.93	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
1843	67.91	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
1844	67.9	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
1845	67.85	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
1846	67.8	kd	CGS001-7866	IFRD2	-			
1847	67.79	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1848	67.78	oe	ccsbBroad304_00223	CASP9	Caspases			
1849	67.74	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
1850	67.71	kd	CGS001-638	BIK	-			
1851	67.6	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
1852	67.59	oe	ccsbBroad304_05192	SPRED2	-			
1853	67.58	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
1854	67.48	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
1855	67.47	kd	CGS001-5654	HTRA1	Serine peptidases / Serine peptidases			
1856	67.44	kd	CGS001-9738	CCP110	-			
1857	67.42	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
1858	67.41	kd	CGS001-2017	CTTN	-			
1859	67.39	kd	CGS001-2161	F12	Chymotrypsin			
1860	67.34	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
1861	67.33	kd	CGS001-19	ABCA1	ATP binding cassette transporters / subfamily A			
1862	67.28	kd	CGS001-6478	SIAH2	-			
1863	67.17	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1864	67.17	kd	CGS001-1327	COX4I1	Mitochondrial respiratory chain complex			
1865	67.09	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
1866	67.02	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
1867	66.98	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
1868	66.96	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
1869	66.95	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1870	66.95	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
1871	66.92	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
1872	66.88	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
1873	66.83	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
1874	66.8	cc		Sirtuins GOF	-			
1875	66.8	kd	CGS001-6832	SUPV3L1	-			
1876	66.79	kd	CGS001-1112	FOXN3	Forkhead boxes			
1877	66.77	kd	CGS001-10489	LRRC41	-			
1878	66.74	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
1879	66.7	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
1880	66.64	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
1881	66.47	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
1882	66.39	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
1883	66.37	oe	ccsbBroad304_00032	ADSL	-			
1884	66.31	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
1885	66.28	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
1886	66.17	oe	ccsbBroad304_02239	RASSF2	-			
1887	66.16	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
1888	66.12	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
1889	66.09	kd	CGS001-81533	ITFG1	-			
1890	65.84	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
1891	65.8	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
1892	65.78	oe	ccsbBroad304_06382	HMGCL	-			
1893	65.78	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
1894	65.7	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
1895	65.6	kd	CGS001-7280	TUBB2A	Tubulins			
1896	65.58	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
1897	65.57	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
1898	65.5	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
1899	65.41	oe	ccsbBroad304_06235	G6PD	-			
1900	65.4	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
1901	65.37	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
1902	65.35	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1903	65.27	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
1904	65.26	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
1905	65.2	kd	CGS001-1120	CHKB	-			
1906	65.15	oe	ccsbBroad304_06420	ICAM3	CD molecules			
1907	65.14	kd	CGS001-84109	QRFPR	GPCR / Class A : RF amide peptide receptors			
1908	64.98	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
1909	64.97	cc		MDM inhibitor	-			
1910	64.89	kd	CGS001-5108	PCM1	-			
1911	64.85	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
1912	64.84	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
1913	64.84	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
1914	64.8	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
1915	64.79	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
1916	64.78	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
1917	64.75	cc		RAF inhibitor	-			
1918	64.74	kd	CGS001-4668	NAGA	-			
1919	64.73	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
1920	64.69	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
1921	64.69	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
1922	64.59	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
1923	64.57	oe	ccsbBroad304_06435	RBPJ	-			
1924	64.56	kd	CGS001-60	ACTB	-			
1925	64.55	kd	CGS001-1891	ECH1	-			
1926	64.53	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
1927	64.45	kd	CGS001-51548	SIRT6	Histone deacetylases (HDACs)			
1928	64.45	kd	CGS001-4190	MDH1	-			
1929	64.39	oe	ccsbBroad304_00164	BLMH	-			
1930	64.38	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
1931	64.38	kd	CGS001-83729	INHBE	-			
1932	64.34	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
1933	64.32	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
1934	64.31	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
1935	64.29	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
1936	64.28	kd	CGS001-1647	GADD45A	-			
1937	64.13	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
1938	64.11	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
1939	64.1	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
1940	64.09	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
1941	64.03	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
1942	64.01	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
1943	63.95	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
1944	63.95	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
1945	63.86	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1946	63.86	kd	CGS001-7528	YY1	INO80 complex subunits			
1947	63.86	kd	CGS001-3909	LAMA3	Laminins			
1948	63.84	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
1949	63.78	oe	ccsbBroad304_07727	LIAS	-			
1950	63.75	kd	CGS001-7010	TEK	Type XII RTKs: TIE family of angiopoietin receptors			
1951	63.75	kd	CGS001-2000	ELF4	ETS Transcription Factors			
1952	63.75	kd	CGS001-55723	ASF1B	-			
1953	63.74	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
1954	63.74	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
1955	63.67	kd	CGS001-150094	SIK1	QIK subfamily			
1956	63.65	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
1957	63.64	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
1958	63.6	kd	CGS001-6541	SLC7A1	SLC7 family			
1959	63.56	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
1960	63.49	kd	CGS001-5106	PCK2	-			
1961	63.42	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
1962	63.29	kd	CGS001-2562	GABRB3	GABA receptors			
1963	63.27	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
1964	63.19	kd	CGS001-23530	NNT	-			
1965	63.18	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
1966	63.14	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
1967	63.11	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
1968	63.04	oe	ccsbBroad304_07884	RYBP	-			
1969	62.86	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
1970	62.81	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
1971	62.76	kd	CGS001-5578	PRKCA	Delta subfamily			
1972	62.73	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
1973	62.72	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
1974	62.71	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
1975	62.67	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
1976	62.66	oe	ccsbBroad304_07724	KDELR2	-			
1977	62.63	kd	CGS001-55634	ZNF673	-			
1978	62.6	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
1979	62.56	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
1980	62.44	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
1981	62.38	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
1982	62.35	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
1983	62.27	oe	ccsbBroad304_00106	ARRB1	-			
1984	62.27	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
1985	62.26	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
1986	62.25	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
1987	62.24	oe	ccsbBroad304_07277	RTCD1	-			
1988	62.21	kd	CGS001-4204	MECP2	-			
1989	62.2	oe	ccsbBroad304_01304	PSEN1	Presenilin			
1990	62.2	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
1991	62.19	kd	CGS001-6453	ITSN1	Rho guanine nucleotide exchange factors			
1992	62.18	oe	ccsbBroad304_09396	TIRAP	-			
1993	62.12	kd	CGS001-10138	YAF2	-			
1994	62.12	kd	CGS001-53834	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
1995	62.08	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
1996	61.96	oe	ccsbBroad304_02506	EBP	-			
1997	61.96	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
1998	61.91	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
1999	61.89	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2000	61.87	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
2001	61.85	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
2002	61.78	kd	CGS001-4594	MUT	-			
2003	61.73	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
2004	61.68	kd	CGS001-3385	ICAM3	CD molecules			
2005	61.67	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
2006	61.61	oe	ccsbBroad304_09358	MAPK1IP1L	-			
2007	61.6	kd	CGS001-2152	F3	CD molecules			
2008	61.58	oe	ccsbBroad304_00881	IRF5	-			
2009	61.55	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
2010	61.53	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
2011	61.52	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
2012	61.46	kd	CGS001-1509	CTSD	Cathepsins			
2013	61.45	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
2014	61.45	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
2015	61.36	oe	ccsbBroad304_08553	STAP2	-			
2016	61.32	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
2017	61.3	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
2018	61.28	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
2019	61.24	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
2020	61.24	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
2021	61.23	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
2022	61.22	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
2023	61.2	kd	CGS001-9412	MED21	-			
2024	61.01	kd	CGS001-1201	CLN3	-			
2025	60.99	cc		GABA receptor antagonist	-			
2026	60.94	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
2027	60.93	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
2028	60.85	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
2029	60.85	kd	CGS001-23057	NMNAT2	-			
2030	60.84	kd	CGS001-10048	RANBP9	-			
2031	60.84	kd	CGS001-843	CASP10	Caspases			
2032	60.68	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
2033	60.63	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
2034	60.62	oe	ccsbBroad304_02416	TUBB4B	-			
2035	60.59	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
2036	60.56	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
2037	60.5	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
2038	60.49	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
2039	60.47	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
2040	60.47	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
2041	60.45	kd	CGS001-51135	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
2042	60.36	kd	CGS001-4724	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
2043	60.35	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
2044	60.33	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
2045	60.31	cp	BRD-K59456551	methotrexate	Dihydrofolate reductase inhibitor		DHFR, AOX1, FOLR1, TYMS	Dihydrofolate reductase inhibitor
2046	60.3	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
2047	60.29	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
2048	60.26	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
2049	60.2	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
2050	60.18	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
2051	60.13	oe	ccsbBroad304_02368	TIMM17B	-			
2052	60.12	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
2053	60.03	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
2054	60	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
2055	59.96	kd	CGS001-523	ATP6V1A	ATPases / V-type			
2056	59.94	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
2057	59.89	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
2058	59.85	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
2059	59.85	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
2060	59.77	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
2061	59.76	kd	CGS001-3032	HADHB	-			
2062	59.71	kd	CGS001-23534	TNPO3	Importins			
2063	59.64	kd	CGS001-23509	POFUT1	Fucosyltransferases			
2064	59.63	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
2065	59.63	kd	CGS001-10269	ZMPSTE24	-			
2066	59.59	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
2067	59.51	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
2068	59.46	oe	ccsbBroad304_02487	TXNIP	-			
2069	59.32	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
2070	59.23	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
2071	59.23	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
2072	59.22	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
2073	59.12	kd	CGS001-10845	CLPX	ATPases / AAA-type			
2074	59.09	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
2075	59.06	cc		Dihydrofolate reductase inhibitor	-			
2076	59.06	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
2077	59.04	kd	CGS001-25987	TSKU	-			
2078	59.03	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
2079	58.95	kd	CGS001-8467	SMARCA5	-			
2080	58.93	kd	CGS001-23743	BHMT2	-			
2081	58.89	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
2082	58.89	kd	CGS001-2010	EMD	-			
2083	58.86	kd	CGS001-11343	MGLL	Endocannabinoid turnover			
2084	58.85	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
2085	58.85	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
2086	58.84	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
2087	58.84	kd	CGS001-8829	NRP1	CD molecules			
2088	58.82	kd	CGS001-1390	CREM	basic leucine zipper proteins			
2089	58.77	kd	CGS001-114904	C1QTNF6	-			
2090	58.75	kd	CGS001-56889	TM9SF3	-			
2091	58.73	oe	ccsbBroad304_02414	IRF9	-			
2092	58.7	kd	CGS001-5594	MAPK1	MAPK:ERK subfamily			
2093	58.63	oe	ccsbBroad304_00617	GBA	-			
2094	58.63	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2095	58.57	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
2096	58.57	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
2097	58.57	kd	CGS001-10014	HDAC5	Histone deacetylases			
2098	58.54	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
2099	58.54	kd	CGS001-4176	MCM7	-			
2100	58.49	oe	ccsbBroad304_02340	SORBS3	-			
2101	58.48	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
2102	58.44	cc		Sigma receptor antagonist	-			
2103	58.43	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
2104	58.41	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
2105	58.4	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
2106	58.37	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2107	58.32	kd	CGS001-11015	KDELR3	-			
2108	58.29	oe	ccsbBroad304_00034	AES	-			
2109	58.24	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
2110	58.24	kd	CGS001-1029	CDKN2A	-			
2111	58.17	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
2112	58.14	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
2113	58.05	kd	CGS001-23647	ARFIP2	-			
2114	58.04	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
2115	58.03	kd	CGS001-4245	MGAT1	-			
2116	58.02	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
2117	58.01	cc		FOS transcription factor family GOF	-			
2118	58	cp	BRD-K60690191	MPEP	Glutamate receptor antagonist		GRM5, GRM1, GRM4	Glutamate receptor antagonist
2119	57.94	kd	CGS001-7337	UBE3A	-			
2120	57.86	oe	ccsbBroad304_01962	STK16	NAK family			
2121	57.86	kd	CGS001-9687	GREB1	-			
2122	57.86	kd	CGS001-27241	BBS9	-			
2123	57.81	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
2124	57.8	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
2125	57.78	kd	CGS001-64376	IKZF5	IKAROS zinc fingers			
2126	57.71	kd	CGS001-4860	PNP	-			
2127	57.67	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
2128	57.62	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
2129	57.57	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
2130	57.55	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
2131	57.52	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2132	57.52	kd	CGS001-5981	RFC1	ATPases / AAA-type			
2133	57.52	kd	CGS001-4548	MTR	-			
2134	57.44	kd	CGS001-10987	COPS5	-			
2135	57.41	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2136	57.41	kd	CGS001-6304	SATB1	Homeoboxes / CUT class			
2137	57.39	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
2138	57.28	oe	ccsbBroad304_00376	CSK	Csk family			
2139	57.28	kd	CGS001-56922	MCCC1	-			
2140	57.27	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
2141	57.24	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
2142	57.23	oe	ccsbBroad304_06282	GLDC	-			
2143	57.19	oe	ccsbBroad304_03910	CCDC90A	-			
2144	57.13	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
2145	57.12	kd	CGS001-134187	POU5F2	Homeoboxes / POU class			
2146	57.09	oe	ccsbBroad304_08660	SMARCAD1	-			
2147	57.05	kd	CGS001-51727	CMPK1	-			
2148	57.02	kd	CGS001-58528	RRAGD	-			
2149	56.92	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2150	56.81	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
2151	56.8	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
2152	56.75	oe	ccsbBroad304_05948	CCND2	-			
2153	56.69	kd	CGS001-8022	LHX3	Homeoboxes / LIM class			
2154	56.69	kd	CGS001-57657	HCN3	Cyclic nucleotide-regulated channels			
2155	56.64	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
2156	56.59	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
2157	56.59	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
2158	56.56	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
2159	56.55	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
2160	56.44	cc		Lipocalins GOF	-			
2161	56.39	kd	CGS001-54407	SLC38A2	System A-like transporters			
2162	56.37	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
2163	56.36	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
2164	56.36	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
2165	56.32	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
2166	56.3	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
2167	56.29	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
2168	56.26	oe	ccsbBroad304_03056	MCTS1	-			
2169	56.24	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
2170	56.14	kd	CGS001-9900	SV2A	Major facilitator superfamily (MFS) of transporters			
2171	56.08	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
2172	56.08	kd	CGS001-2194	FASN	Short chain dehydrogenase/reductase superfamily / Atypical members			
2173	56.04	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
2174	55.99	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
2175	55.98	kd	CGS001-5920	RARRES3	-			
2176	55.97	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2177	55.94	kd	CGS001-2710	GK	Glycerol kinases			
2178	55.69	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
2179	55.63	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
2180	55.61	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
2181	55.54	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
2182	55.53	kd	CGS001-51347	TAOK3	TAO subfamily			
2183	55.51	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
2184	55.44	oe	ccsbBroad304_08839	IFIH1	-			
2185	55.43	kd	CGS001-5771	PTPN2	Protein tyrosine phosphatases			
2186	55.42	oe	ccsbBroad304_02017	PEX11A	-			
2187	55.42	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
2188	55.27	kd	CGS001-10096	ACTR3	-			
2189	55.24	kd	CGS001-344	APOC2	Apolipoproteins			
2190	55.17	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
2191	55.14	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
2192	55.13	kd	CGS001-55837	EAPP	-			
2193	55.12	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2194	55.1	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
2195	55.03	kd	CGS001-7511	XPNPEP1	Methionyl aminopeptidase			
2196	54.99	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
2197	54.94	oe	ccsbBroad304_03573	BRF2	-			
2198	54.89	oe	ccsbBroad304_03858	SRPRB	-			
2199	54.88	kd	CGS001-9221	NOLC1	-			
2200	54.86	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
2201	54.85	oe	ccsbBroad304_05745	CD24	CD molecules			
2202	54.83	kd	CGS001-211	ALAS1	-			
2203	54.78	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
2204	54.78	kd	CGS001-10681	GNB5	WD repeat domain containing			
2205	54.73	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2206	54.49	oe	ccsbBroad304_01754	UCK2	-			
2207	54.48	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
2208	54.46	kd	CGS001-3958	LGALS3	Endogenous ligands			
2209	54.44	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
2210	54.42	oe	ccsbBroad304_06642	NIT1	-			
2211	54.4	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
2212	54.38	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
2213	54.32	kd	CGS001-9748	SLK	SLK subfamily			
2214	54.28	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
2215	54.28	kd	CGS001-478	ATP1A3	ATPases / P-type			
2216	54.21	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
2217	54.19	kd	CGS001-8720	MBTPS1	Subtilisin			
2218	54.19	kd	CGS001-51601	LIPT1	-			
2219	54.14	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
2220	54.14	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
2221	54.11	kd	CGS001-819	CAMLG	-			
2222	54.06	kd	CGS001-4046	LSP1	-			
2223	54.05	kd	CGS001-3417	IDH1	-			
2224	53.97	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
2225	53.96	kd	CGS001-8089	YEATS4	-			
2226	53.94	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
2227	53.91	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
2228	53.87	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
2229	53.87	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
2230	53.83	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
2231	53.81	kd	CGS001-183	AGT	Endogenous ligands			
2232	53.78	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
2233	53.73	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
2234	53.7	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
2235	53.7	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
2236	53.7	kd	CGS001-54998	AURKAIP1	-			
2237	53.66	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
2238	53.61	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
2239	53.55	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
2240	53.55	oe	ccsbBroad304_02446	TADA3	-			
2241	53.55	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
2242	53.52	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
2243	53.43	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2244	53.38	oe	ccsbBroad304_06134	ECH1	-			
2245	53.36	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2246	53.35	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
2247	53.35	kd	CGS001-84333	PCGF5	Polycomb group ring fingers			
2248	53.32	oe	ccsbBroad304_00626	GDI1	-			
2249	53.2	oe	ccsbBroad304_02133	CD83	CD molecules			
2250	53.14	kd	CGS001-3939	LDHA	-			
2251	53.13	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
2252	53.11	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
2253	53.08	oe	ccsbBroad304_00162	BIK	-			
2254	53.06	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
2255	53.04	kd	CGS001-11315	PARK7	Parkinson disease			
2256	53.03	oe	ccsbBroad304_02596	KDELR3	-			
2257	53	kd	CGS001-8743	TNFSF10	CD molecules			
2258	52.97	oe	ccsbBroad304_01139	PA2G4	-			
2259	52.91	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
2260	52.9	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
2261	52.88	kd	CGS001-9459	ARHGEF6	Rho guanine nucleotide exchange factors			
2262	52.81	oe	ccsbBroad304_01143	PAFAH1B3	-			
2263	52.8	oe	ccsbBroad304_14011	PAPSS1	-			
2264	52.66	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
2265	52.64	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
2266	52.63	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
2267	52.6	kd	CGS001-2203	FBP1	-			
2268	52.59	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
2269	52.58	oe	ccsbBroad304_06845	RARRES3	-			
2270	52.56	cp	BRD-A24543851	nornicotine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2271	52.51	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
2272	52.48	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
2273	52.4	kd	CGS001-8777	MPDZ	-			
2274	52.37	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
2275	52.36	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
2276	52.33	kd	CGS001-1493	CTLA4	CD molecules			
2277	52.27	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
2278	52.24	kd	CGS001-9869	SETDB1	Histone methyltransferases (HMTs)			
2279	52.23	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2280	52.22	kd	CGS001-22934	RPIA	-			
2281	52.21	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
2282	52.2	oe	ccsbBroad304_00418	CD55	CD molecules			
2283	52.2	kd	CGS001-4905	NSF	ATPases / AAA-type			
2284	52.18	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
2285	52.14	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
2286	52.14	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
2287	52.06	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
2288	52.05	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
2289	52.05	kd	CGS001-571	BACH1	BTB/POZ domain containing			
2290	52.04	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
2291	52.03	kd	CGS001-1363	CPE	Carboxypeptidase A			
2292	52.02	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
2293	52	kd	CGS001-1497	CTNS	-			
2294	51.99	kd	CGS001-9710	KIAA0355	-			
2295	51.92	oe	ccsbBroad304_00054	ALDOC	-			
2296	51.92	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
2297	51.88	kd	CGS001-2976	GTF3C2	General transcription factors			
2298	51.88	kd	CGS001-27109	ATP5S	-			
2299	51.85	cp	BRD-K96740444	itopride	Dopamine receptor antagonist		DRD2, ACHE, CHRM3	Dopamine receptor antagonist
2300	51.85	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2301	51.85	kd	CGS001-10513	APPBP2	-			
2302	51.74	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
2303	51.7	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
2304	51.69	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
2305	51.64	kd	CGS001-3609	ILF3	-			
2306	51.63	kd	CGS001-283150	FOXR1	Forkhead boxes			
2307	51.59	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
2308	51.59	cp	BRD-A16444946	acarbose	Glucosidase inhibitor		GAA, MGAM, AMY2A, SI	Glucosidase inhibitor
2309	51.56	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
2310	51.56	cp	BRD-K32311154	nifekalant	Potassium channel blocker			Potassium channel blocker
2311	51.52	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
2312	51.51	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
2313	51.46	oe	ccsbBroad304_06720	PHYH	-			
2314	51.34	kd	CGS001-3455	IFNAR2	Interferon receptor family			
2315	51.33	kd	CGS001-6829	SUPT5H	-			
2316	51.32	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
2317	51.28	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
2318	51.27	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
2319	51.25	oe	ccsbBroad304_01576	SOAT1	-			
2320	51.19	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
2321	51.12	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
2322	51.11	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
2323	51.11	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2324	51.1	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
2325	51.1	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
2326	51.06	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
2327	50.94	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
2328	50.91	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
2329	50.85	kd	CGS001-55869	HDAC8	Histone deacetylases			
2330	50.8	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
2331	50.79	cp	BRD-M47937986	cefatrizine	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2332	50.76	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
2333	50.75	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
2334	50.75	kd	CGS001-3053	SERPIND1	Serine (or cysteine) peptidase inhibitors			
2335	50.73	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
2336	50.72	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
2337	50.7	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
2338	50.68	oe	ccsbBroad304_00550	FDXR	-			
2339	50.64	kd	CGS001-8409	UXT	-			
2340	50.58	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
2341	50.46	oe	ccsbBroad304_02822	ARFIP2	-			
2342	50.33	oe	ccsbBroad304_01174	PEX13	-			
2343	50.28	kd	CGS001-11004	KIF2C	Kinesins			
2344	50.25	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
2345	50.22	kd	CGS001-11331	PHB2	-			
2346	50.21	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
2347	50.21	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
2348	50.12	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
2349	50.06	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
2350	50.02	oe	ccsbBroad304_02345	TXNDC9	-			
2351	50.02	kd	CGS001-80349	WDR61	WD repeat domain containing			
2352	50.01	oe	ccsbBroad304_07017	SUOX	-			
2353	49.96	kd	CGS001-205564	SENP5	-			
2354	49.9	kd	CGS001-6196	RPS6KA2	RSK subfamily			
2355	49.77	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
2356	49.76	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
2357	49.76	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
2358	49.6	kd	CGS001-8531	CSDA	-			
2359	49.49	kd	CGS001-4303	FOXO4	Forkhead boxes			
2360	49.44	oe	ccsbBroad304_03266	ERGIC2	-			
2361	49.4	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
2362	49.38	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
2363	49.37	kd	CGS001-7158	TP53BP1	-			
2364	49.35	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
2365	49.31	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
2366	49.29	kd	CGS001-1045	CDX2	Homeoboxes / ANTP class : HOXL subclass			
2367	49.27	kd	CGS001-10474	TADA3	-			
2368	49.26	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
2369	49.25	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
2370	49.24	oe	ccsbBroad304_03097	CNOT7	-			
2371	49.19	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
2372	49.11	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
2373	49.1	kd	CGS001-8894	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2374	49.09	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
2375	49.03	kd	CGS001-5294	PIK3CG	Phosphatidylinositol kinases			
2376	49.03	kd	CGS001-11007	CCDC85B	-			
2377	48.99	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
2378	48.94	kd	CGS001-9128	PRPF4	WD repeat domain containing			
2379	48.9	kd	CGS001-151126	ZNF385B	-			
2380	48.83	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
2381	48.76	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
2382	48.74	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
2383	48.64	oe	ccsbBroad304_13499	KSR2	RAF family			
2384	48.6	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
2385	48.56	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
2386	48.55	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
2387	48.5	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
2388	48.5	cp	BRD-K62374253	rufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
2389	48.49	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
2390	48.47	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
2391	48.45	kd	CGS001-1756	DMD	-			
2392	48.41	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
2393	48.35	cc		Aminoacyl tRNA synthetases class II LOF	-			
2394	48.33	kd	CGS001-10010	TANK	-			
2395	48.29	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
2396	48.24	kd	CGS001-9955	HS3ST3A1	Sulfotransferases, membrane-bound			
2397	48.2	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
2398	47.99	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
2399	47.96	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
2400	47.86	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
2401	47.84	kd	CGS001-10059	DNM1L	-			
2402	47.81	kd	CGS001-2160	F11	Chymotrypsin			
2403	47.79	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
2404	47.73	kd	CGS001-23585	TMEM50A	-			
2405	47.64	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
2406	47.63	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
2407	47.61	cp	BRD-K37814297	acepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
2408	47.57	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2409	47.55	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
2410	47.55	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
2411	47.51	cp	BRD-A87125127	3-matida	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2412	47.5	kd	CGS001-23429	RYBP	-			
2413	47.47	kd	CGS001-23038	WDTC1	DDB1 and CUL4 associated factors			
2414	47.38	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
2415	47.33	kd	CGS001-255738	PCSK9	Subtilisin			
2416	47.26	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
2417	47.24	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
2418	47.23	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
2419	47.18	kd	CGS001-28985	MCTS1	-			
2420	47.11	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
2421	46.99	cc		PKC activator	-			
2422	46.98	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
2423	46.94	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
2424	46.89	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
2425	46.86	kd	CGS001-4172	MCM3	-			
2426	46.78	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
2427	46.74	oe	ccsbBroad304_00038	AGL	-			
2428	46.74	oe	ccsbBroad304_03450	TMED9	-			
2429	46.74	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
2430	46.69	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
2431	46.66	kd	CGS001-115727	RASGRP4	EF-hand domain containing			
2432	46.64	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
2433	46.64	kd	CGS001-6988	TCTA	-			
2434	46.63	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
2435	46.62	kd	CGS001-55191	NADSYN1	-			
2436	46.61	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
2437	46.61	cp	BRD-K82357231	desloratadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2438	46.6	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
2439	46.6	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
2440	46.58	kd	CGS001-4856	NOV	-			
2441	46.54	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
2442	46.53	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2443	46.48	oe	ccsbBroad304_09821	TMEM154	-			
2444	46.48	oe	ccsbBroad304_02580	TMED10	-			
2445	46.45	kd	CGS001-7465	WEE1	WEE family			
2446	46.43	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2447	46.39	kd	CGS001-2113	ETS1	ETS Transcription Factors			
2448	46.35	cp	BRD-K99063460	didanosine	Nucleoside reverse transcriptase inhibitor		PNP	Nucleoside reverse transcriptase inhibitor
2449	46.32	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
2450	46.31	kd	CGS001-57406	ABHD6	Abhydrolase domain containing			
2451	46.29	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
2452	46.25	kd	CGS001-1622	DBI	-			
2453	46.23	oe	ccsbBroad304_04406	PLA2G12B	-			
2454	46.23	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
2455	46.23	kd	CGS001-201799	TMEM154	-			
2456	46.22	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
2457	46.21	kd	CGS001-10628	TXNIP	-			
2458	46.15	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
2459	46.13	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
2460	46.08	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
2461	46.08	kd	CGS001-4782	NFIC	-			
2462	46.05	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
2463	46.05	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
2464	46.03	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
2465	45.98	cp	BRD-K86003836	flubendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
2466	45.96	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
2467	45.96	kd	CGS001-5300	PIN1	-			
2468	45.92	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
2469	45.89	oe	ccsbBroad304_00620	GCDH	-			
2470	45.81	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
2471	45.78	kd	CGS001-3676	ITGA4	Integrins			
2472	45.77	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
2473	45.75	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
2474	45.63	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
2475	45.58	oe	ccsbBroad304_06837	RAF1	RAF family			
2476	45.48	kd	CGS001-4700	NDUFA6	LYR motif containing			
2477	45.47	kd	CGS001-10745	PHTF1	-			
2478	45.47	kd	CGS001-9146	HGS	Zinc fingers, FYVE domain containing			
2479	45.46	kd	CGS001-6603	SMARCD2	-			
2480	45.38	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
2481	45.37	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
2482	45.36	cc		HDAC inhibitor	-			
2483	45.32	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
2484	45.31	kd	CGS001-23386	NUDCD3	-			
2485	45.3	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
2486	45.28	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
2487	45.21	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
2488	45.14	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
2489	45.14	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
2490	45.1	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
2491	45.07	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
2492	45.02	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
2493	45.02	kd	CGS001-4175	MCM6	-			
2494	44.97	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
2495	44.95	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
2496	44.92	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2497	44.92	kd	CGS001-135	ADORA2A	GPCR / Class A : Adenosine receptors			
2498	44.86	kd	CGS001-7035	TFPI	-			
2499	44.85	oe	ccsbBroad304_02306	PQBP1	-			
2500	44.76	kd	CGS001-2857	GPR34	GPCR / Class A : Orphans			
2501	44.75	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
2502	44.62	cc		Thymidylate synthase inhibitor	-			
2503	44.59	oe	ccsbBroad304_08825	LHPP	-			
2504	44.58	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
2505	44.57	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
2506	44.56	kd	CGS001-2810	SFN	-			
2507	44.51	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
2508	44.49	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
2509	44.48	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
2510	44.4	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
2511	44.39	kd	CGS001-9787	DLGAP5	-			
2512	44.37	kd	CGS001-2834	PRLHR	GPCR / Class A : RF amide peptide receptors			
2513	44.18	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
2514	44.17	kd	CGS001-80351	TNKS2	Ankyrin repeat domain containing			
2515	44.13	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
2516	44.1	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
2517	44.08	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
2518	43.97	kd	CGS001-83439	TCF7L1	-			
2519	43.97	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
2520	43.95	oe	ccsbBroad304_03113	DSE	-			
2521	43.93	kd	CGS001-5581	PRKCE	Eta subfamily			
2522	43.9	cp	BRD-K46742498	alosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
2523	43.9	kd	CGS001-6277	S100A6	EF-hand domain containing			
2524	43.89	kd	CGS001-811	CALR	-			
2525	43.86	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
2526	43.85	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
2527	43.81	oe	ccsbBroad304_00883	ISG20	-			
2528	43.81	kd	CGS001-3251	HPRT1	-			
2529	43.79	oe	ccsbBroad304_03155	DHH	-			
2530	43.76	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
2531	43.7	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
2532	43.69	oe	ccsbBroad304_03746	CDC42SE1	-			
2533	43.65	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
2534	43.51	cp	BRD-A24191444	ifenprodil	Adrenergic receptor antagonist		GRIN1, GRIN2B	Adrenergic receptor antagonist, Glutamate receptor antagonist
2535	43.46	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
2536	43.43	oe	ccsbBroad304_02605	PAPD7	-			
2537	43.41	cp	BRD-K29653726	topiramate	Carbonic anhydrase inhibitor		CA2, CA4, GRIK1, CA1, CA12, CA7, CYP2C19, CYP3A4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA1, SCN1A, SCN5A	Carbonic anhydrase inhibitor, Glutamate receptor antagonist, Kainate receptor antagonist
2538	43.39	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
2539	43.37	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
2540	43.32	kd	CGS001-2355	FOSL2	basic leucine zipper proteins			
2541	43.31	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
2542	43.29	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
2543	43.27	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
2544	43.27	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
2545	43.26	oe	ccsbBroad304_06089	DDIT3	-			
2546	43.25	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
2547	43.23	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
2548	43.13	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
2549	42.9	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
2550	42.87	oe	ccsbBroad304_07616	ZNF238	-			
2551	42.85	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
2552	42.85	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
2553	42.71	oe	ccsbBroad304_08775	SQRDL	-			
2554	42.65	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
2555	42.65	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
2556	42.64	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
2557	42.63	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
2558	42.54	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
2559	42.51	kd	CGS001-25925	ZNF521	Zinc fingers, C2H2-type			
2560	42.51	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2561	42.48	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2562	42.47	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
2563	42.46	kd	CGS001-1173	AP2M1	-			
2564	42.38	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2565	42.38	kd	CGS001-3596	IL13	Interleukins and interleukin receptors			
2566	42.32	oe	ccsbBroad304_02501	DCTN6	-			
2567	42.31	oe	ccsbBroad304_06294	GNAZ	-			
2568	42.29	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
2569	42.2	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
2570	42.18	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
2571	42.15	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
2572	42.13	oe	ccsbBroad304_05135	PARP15	-			
2573	42.1	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
2574	42.08	oe	ccsbBroad304_01371	RALA	-			
2575	42.04	oe	ccsbBroad304_01038	MSRA	-			
2576	41.97	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
2577	41.96	kd	CGS001-488	ATP2A2	Calcium-ATPases			
2578	41.94	kd	CGS001-23588	KLHDC2	-			
2579	41.93	oe	ccsbBroad304_06518	LDHA	-			
2580	41.89	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
2581	41.82	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
2582	41.81	oe	ccsbBroad304_05823	ANXA2	Annexins			
2583	41.8	kd	CGS001-823	CAPN1	EF-hand domain containing			
2584	41.74	oe	ccsbBroad304_06828	PYCR1	-			
2585	41.72	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
2586	41.69	kd	CGS001-471	ATIC	-			
2587	41.61	kd	CGS001-29083	GTPBP8	-			
2588	41.59	cp	BRD-A80928489	1-monopalmitin	P-glycoprotein inhibitor		ABCB1	P-glycoprotein inhibitor
2589	41.57	kd	CGS001-374291	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
2590	41.52	oe	ccsbBroad304_07362	NMI	-			
2591	41.47	oe	ccsbBroad304_00420	DAP	-			
2592	41.44	cp	BRD-K93618743	ipriflavone	Bone resorption inhibitor			Bone resorption inhibitor
2593	41.42	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
2594	41.42	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
2595	41.33	kd	CGS001-5689	PSMB1	Proteasome subunits			
2596	41.26	kd	CGS001-11243	PMF1	-			
2597	41.25	kd	CGS001-342926	ZNF677	Zinc fingers, C2H2-type			
2598	41.22	kd	CGS001-2523	FUT1	Fucosyltransferases			
2599	41.14	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
2600	41.13	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
2601	41.03	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
2602	41.01	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
2603	40.98	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2604	40.95	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2605	40.94	kd	CGS001-4836	NMT1	-			
2606	40.89	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
2607	40.88	oe	ccsbBroad304_07808	RAB11FIP2	-			
2608	40.85	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2609	40.85	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
2610	40.85	kd	CGS001-4125	MAN2B1	-			
2611	40.81	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
2612	40.8	oe	ccsbBroad304_00564	FGR	Src family			
2613	40.78	kd	CGS001-546	ATRX	-			
2614	40.78	kd	CGS001-154	ADRB2	GPCR / Class A : Adrenoceptors : beta			
2615	40.74	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2616	40.66	kd	CGS001-10078	TSSC4	-			
2617	40.66	kd	CGS001-7100	TLR5	Toll-like receptor family			
2618	40.62	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
2619	40.62	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
2620	40.61	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
2621	40.56	oe	ccsbBroad304_00112	ASNA1	-			
2622	40.56	kd	CGS001-2212	FCGR2A	CD molecules			
2623	40.51	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
2624	40.5	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
2625	40.47	cp	BRD-A87387433	cefpodoxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2626	40.46	oe	ccsbBroad304_03951	NARFL	-			
2627	40.45	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
2628	40.42	oe	ccsbBroad304_04194	ELL3	-			
2629	40.39	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
2630	40.39	kd	CGS001-4331	MNAT1	RING-type (C3HC4) zinc fingers			
2631	40.38	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
2632	40.33	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
2633	40.31	kd	CGS001-5004	ORM1	Lipocalins			
2634	40.22	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
2635	40.16	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
2636	40.13	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
2637	40.08	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
2638	40.08	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
2639	40.06	oe	ccsbBroad304_07605	LYPLA1	-			
2640	40.06	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
2641	40.06	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
2642	40.01	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
2643	39.95	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
2644	39.92	kd	CGS001-10587	TXNRD2	-			
2645	39.91	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
2646	39.82	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
2647	39.82	kd	CGS001-3458	IFNG	Interferons			
2648	39.81	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
2649	39.69	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
2650	39.64	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
2651	39.63	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
2652	39.63	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
2653	39.61	kd	CGS001-2859	GPR35	GPCR / Class A : Orphans			
2654	39.58	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
2655	39.58	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
2656	39.45	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
2657	39.43	oe	ccsbBroad304_01215	PLAUR	CD molecules			
2658	39.4	cc		PRD class homeoboxes and psudogenes LOF	-			
2659	39.37	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
2660	39.37	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
2661	39.35	kd	CGS001-22933	SIRT2	Histone deacetylases			
2662	39.28	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
2663	39.28	kd	CGS001-6434	TRA2B	RNA binding motif (RRM) containing			
2664	39.24	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
2665	39.22	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
2666	39.22	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
2667	39.21	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
2668	39.21	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
2669	39.19	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
2670	39.15	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
2671	39.15	kd	CGS001-10165	SLC25A13	Mitochondrial amino acid transporter subfamily			
2672	39.13	kd	CGS001-51720	UIMC1	-			
2673	39.13	kd	CGS001-9131	AIFM1	-			
2674	39.11	oe	ccsbBroad304_03859	ENOPH1	-			
2675	39.1	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
2676	39.06	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
2677	39.06	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2678	39.03	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
2679	39.03	kd	CGS001-25874	BRP44	-			
2680	39.02	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
2681	39.02	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
2682	39.02	kd	CGS001-6709	SPTAN1	EF-hand domain containing			
2683	39	oe	ccsbBroad304_02313	ACTR3	-			
2684	38.98	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
2685	38.97	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
2686	38.95	cp	BRD-A23359898	sibutramine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, CYP2B6, CYP2C19, CYP3A5	Serotonin reuptake inhibitor
2687	38.92	kd	CGS001-79139	DERL1	-			
2688	38.91	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
2689	38.9	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
2690	38.82	kd	CGS001-140612	ZFP28	Zinc fingers, C2H2-type			
2691	38.81	kd	CGS001-2767	GNA11	-			
2692	38.8	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
2693	38.77	cc		PI3K Signaling LOF	-			
2694	38.75	kd	CGS001-10523	CHERP	G patch domain containing			
2695	38.7	kd	CGS001-1050	CEBPA	basic leucine zipper proteins			
2696	38.57	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
2697	38.55	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
2698	38.55	kd	CGS001-1955	MEGF9	-			
2699	38.53	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
2700	38.53	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
2701	38.53	kd	CGS001-6009	RHEB	-			
2702	38.52	oe	ccsbBroad304_02554	TRAFD1	-			
2703	38.51	oe	ccsbBroad304_07531	TANK	-			
2704	38.48	kd	CGS001-9276	COPB2	WD repeat domain containing			
2705	38.43	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
2706	38.41	kd	CGS001-5467	PPARD	Nuclear hormone receptors			
2707	38.39	kd	CGS001-6199	RPS6KB2	p70 subfamily			
2708	38.31	kd	CGS001-51160	VPS28	-			
2709	38.31	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
2710	38.29	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
2711	38.28	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
2712	38.26	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
2713	38.26	kd	CGS001-55324	ABCF3	ATP binding cassette transporters / subfamily F			
2714	38.19	oe	ccsbBroad304_02110	VAPB	-			
2715	38.18	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
2716	38.16	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
2717	38.08	kd	CGS001-1534	CYB561	Cytochrome b genes			
2718	38.04	cc		IGF-1 inhibitor	-			
2719	38.04	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
2720	38.03	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
2721	38.02	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
2722	38.02	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
2723	38.01	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
2724	38	kd	CGS001-2869	GRK5	GRK1/3 subfamily			
2725	37.89	kd	CGS001-51284	TLR7	Toll-like receptor family			
2726	37.89	kd	CGS001-9184	BUB3	WD repeat domain containing			
2727	37.82	oe	ccsbBroad304_01101	NME1	-			
2728	37.78	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
2729	37.73	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
2730	37.72	cc		Norepinephrine reuptake inhibitor	-			
2731	37.72	cp	BRD-A84134924	pancuronium	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRNA1, CHRNA2	Acetylcholine receptor antagonist
2732	37.69	kd	CGS001-5962	RDX	-			
2733	37.65	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
2734	37.63	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
2735	37.61	kd	CGS001-79090	TRAPPC6A	Trafficking protein particle complex			
2736	37.51	kd	CGS001-7054	TH	Amino acid hydroxylases			
2737	37.51	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
2738	37.5	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
2739	37.49	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2740	37.46	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
2741	37.45	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
2742	37.37	kd	CGS001-5693	PSMB5	Proteasome subunits			
2743	37.31	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
2744	37.29	oe	ccsbBroad304_02526	POP4	-			
2745	37.27	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
2746	37.18	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
2747	37.13	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
2748	37.11	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
2749	37.11	kd	CGS001-84775	ZNF607	Zinc fingers, C2H2-type			
2750	37.09	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
2751	37.09	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
2752	37.05	kd	CGS001-23384	SPECC1L	-			
2753	37.03	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
2754	37	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
2755	36.99	kd	CGS001-271	AMPD2	-			
2756	36.98	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2757	36.95	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
2758	36.94	cc		PI3K inhibitor	-			
2759	36.92	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
2760	36.83	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
2761	36.81	oe	ccsbBroad304_03533	CDCA8	-			
2762	36.77	oe	ccsbBroad304_00313	TBCB	-			
2763	36.75	oe	ccsbBroad304_00120	ATOX1	-			
2764	36.73	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
2765	36.73	kd	CGS001-10401	PIAS3	Zinc fingers, MIZ-type			
2766	36.71	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
2767	36.71	kd	CGS001-7343	UBTF	-			
2768	36.7	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
2769	36.7	kd	CGS001-64319	FBRS	-			
2770	36.66	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
2771	36.63	kd	CGS001-4048	LTA4H	Hydrolases			
2772	36.6	kd	CGS001-2769	GNA15	-			
2773	36.58	kd	CGS001-3608	ILF2	-			
2774	36.57	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
2775	36.57	kd	CGS001-84527	ZNF559	Zinc fingers, C2H2-type			
2776	36.56	kd	CGS001-1605	DAG1	-			
2777	36.52	oe	ccsbBroad304_02386	EIF1B	-			
2778	36.49	kd	CGS001-129685	TAF8	-			
2779	36.44	cc		Mitogen activated protein kinases LOF	-			
2780	36.42	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2781	36.41	oe	ccsbBroad304_00519	ETFB	-			
2782	36.38	oe	ccsbBroad304_01672	TIMP2	-			
2783	36.37	kd	CGS001-6098	ROS1	Type XVII RTKs: ROS receptors			
2784	36.36	cp	BRD-A79903587	tegafur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
2785	36.36	kd	CGS001-54623	PAF1	-			
2786	36.33	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
2787	36.33	kd	CGS001-79960	PHF17	-			
2788	36.33	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
2789	36.33	kd	CGS001-9447	AIM2	-			
2790	36.3	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
2791	36.28	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
2792	36.19	oe	ccsbBroad304_01131	OXCT1	-			
2793	36.18	oe	ccsbBroad304_07094	TPMT	-			
2794	36.18	kd	CGS001-1384	CRAT	-			
2795	36.18	kd	CGS001-629	CFB	Complement system			
2796	36.15	kd	CGS001-64077	LHPP	-			
2797	36.14	oe	ccsbBroad304_00183	C1S	Complement system			
2798	36.12	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
2799	36.1	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
2800	36.07	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
2801	36.04	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
2802	36	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
2803	35.98	oe	ccsbBroad304_00709	GUK1	-			
2804	35.98	kd	CGS001-166	AES	-			
2805	35.97	kd	CGS001-3205	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
2806	35.94	cp	BRD-K10670311	sulfasalazine	Antirheumatic		PTGS1, PTGS2, ACAT1, ALOX5, CHUK, IKBKB, PLA2G1B, PPARG, SLC46A1, SLC7A11, TBXAS1	Antirheumatic, NFkB pathway inhibitor
2807	35.93	kd	CGS001-3054	HCFC1	-			
2808	35.86	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
2809	35.85	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
2810	35.83	oe	ccsbBroad304_03118	NRBP1	NRBP family			
2811	35.79	oe	ccsbBroad304_05038	HORMAD2	-			
2812	35.79	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2813	35.79	kd	CGS001-29911	HOOK2	-			
2814	35.77	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
2815	35.74	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2816	35.72	kd	CGS001-55278	QRSL1	-			
2817	35.69	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
2818	35.68	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
2819	35.65	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
2820	35.64	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
2821	35.62	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
2822	35.61	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
2823	35.55	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
2824	35.55	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2825	35.51	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
2826	35.5	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
2827	35.48	kd	CGS001-91975	ZNF300	Zinc fingers, C2H2-type			
2828	35.47	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
2829	35.47	kd	CGS001-51014	TMED7	-			
2830	35.44	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
2831	35.44	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
2832	35.41	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
2833	35.38	kd	CGS001-29984	RHOD	-			
2834	35.37	oe	ccsbBroad304_04490	RSPH1	-			
2835	35.36	kd	CGS001-10641	NPRL2	-			
2836	35.34	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
2837	35.32	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
2838	35.28	kd	CGS001-6787	NEK4	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2839	35.27	oe	ccsbBroad304_00985	MCL1	-			
2840	35.25	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
2841	35.24	kd	CGS001-7184	HSP90B1	Heat shock proteins / HSPC			
2842	35.22	oe	ccsbBroad304_02349	MPHOSPH9	-			
2843	35.15	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2844	35.13	oe	ccsbBroad304_02249	KIAA0494	-			
2845	35.08	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
2846	35.08	kd	CGS001-25949	SYF2	-			
2847	35.07	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
2848	34.97	kd	CGS001-10023	FRAT1	-			
2849	34.96	oe	ccsbBroad304_05947	CCNC	-			
2850	34.95	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
2851	34.92	kd	CGS001-3459	IFNGR1	Interferon receptor family			
2852	34.87	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
2853	34.87	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2854	34.79	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
2855	34.78	kd	CGS001-3487	IGFBP4	insulin-like growth factor (IGF) binding proteins			
2856	34.72	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
2857	34.71	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
2858	34.7	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
2859	34.7	oe	ccsbBroad304_07220	CDC45	-			
2860	34.69	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
2861	34.69	kd	CGS001-79902	NUP85	-			
2862	34.68	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
2863	34.63	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
2864	34.63	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
2865	34.62	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
2866	34.61	kd	CGS001-2645	GCK	Hexokinases			
2867	34.61	kd	CGS001-3169	FOXA1	Forkhead boxes			
2868	34.6	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
2869	34.58	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
2870	34.57	cp	BRD-A96107863	nisoldipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNB2, CYP3A5	Calcium channel blocker
2871	34.56	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
2872	34.53	kd	CGS001-57157	PHTF2	-			
2873	34.52	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
2874	34.47	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
2875	34.44	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
2876	34.44	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
2877	34.42	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
2878	34.41	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
2879	34.38	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
2880	34.37	oe	ccsbBroad304_01701	TPI1	-			
2881	34.37	oe	ccsbBroad304_00954	LYN	Src family			
2882	34.36	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
2883	34.35	oe	ccsbBroad304_00053	ALDOA	-			
2884	34.35	oe	ccsbBroad304_03179	BOLA1	-			
2885	34.34	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
2886	34.3	kd	CGS001-23344	ESYT1	Synaptotagmins			
2887	34.28	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
2888	34.25	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
2889	34.25	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
2890	34.23	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
2891	34.21	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
2892	34.19	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2893	34.17	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
2894	34.15	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
2895	34.04	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
2896	34.02	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
2897	34.01	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
2898	34.01	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
2899	33.98	kd	CGS001-54386	TERF2IP	-			
2900	33.97	oe	ccsbBroad304_01066	NDUFA4	-			
2901	33.97	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
2902	33.96	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
2903	33.96	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2904	33.95	kd	CGS001-26036	ZNF451	Zinc fingers, C2H2-type			
2905	33.87	oe	ccsbBroad304_08461	CDCA4	-			
2906	33.87	kd	CGS001-11129	CLASRP	-			
2907	33.83	cp	BRD-K18895904	olanzapine	Dopamine receptor antagonist		DRD2, HTR2A, HTR2C, DRD1, DRD3, DRD4, HRH1, HTR1A, HTR1B, HTR1D, HTR1E, HTR6, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C8, DRD5, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH2, HRH4, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
2908	33.68	kd	CGS001-51684	SUFU	-			
2909	33.65	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
2910	33.65	kd	CGS001-7862	BRPF1	Non-enzymatic BRD containing proteins			
2911	33.64	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
2912	33.62	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
2913	33.56	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
2914	33.54	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
2915	33.53	kd	CGS001-4904	YBX1	-			
2916	33.52	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
2917	33.52	kd	CGS001-5577	PRKAR2B	Protein kinase A			
2918	33.51	kd	CGS001-10058	ABCB6	ATP binding cassette transporters / subfamily B			
2919	33.49	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
2920	33.46	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
2921	33.44	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
2922	33.43	oe	ccsbBroad304_08426	TEX10	-			
2923	33.43	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
2924	33.4	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
2925	33.4	kd	CGS001-4091	SMAD6	SMADs			
2926	33.37	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
2927	33.35	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
2928	33.35	kd	CGS001-84878	ZBTB45	BTB/POZ domain containing			
2929	33.33	kd	CGS001-3978	LIG1	-			
2930	33.27	oe	ccsbBroad304_06225	FTH1	-			
2931	33.21	kd	CGS001-9632	SEC24C	-			
2932	33.17	kd	CGS001-2581	GALC	-			
2933	33.11	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
2934	33.11	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
2935	33.1	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
2936	33.09	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
2937	33.09	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
2938	33.02	kd	CGS001-10475	TRIM38	-			
2939	33	oe	ccsbBroad304_08797	FASTKD5	-			
2940	32.99	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
2941	32.98	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
2942	32.96	cc		Bacterial DNA gyrase inhibitor	-			
2943	32.96	oe	ccsbBroad304_01716	TSN	-			
2944	32.96	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
2945	32.96	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
2946	32.93	kd	CGS001-3516	RBPJ	-			
2947	32.93	kd	CGS001-593	BCKDHA	-			
2948	32.9	kd	CGS001-5727	PTCH1	-			
2949	32.86	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
2950	32.86	kd	CGS001-23576	DDAH1	Dimethylarginine dimethylaminohydrolases			
2951	32.83	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
2952	32.8	kd	CGS001-2806	GOT2	-			
2953	32.68	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
2954	32.67	oe	ccsbBroad304_03112	NENF	-			
2955	32.65	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
2956	32.64	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
2957	32.63	kd	CGS001-23223	RRP12	-			
2958	32.61	oe	ccsbBroad304_06085	DCK	-			
2959	32.6	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
2960	32.59	cc		AHSP Pathway LOF	-			
2961	32.55	kd	CGS001-143	PARP4	Poly (ADP-ribose) polymerases			
2962	32.54	kd	CGS001-218	ALDH3A1	Aldehyde dehydrogenases			
2963	32.52	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
2964	32.43	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
2965	32.42	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2966	32.42	kd	CGS001-79796	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
2967	32.4	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2968	32.38	oe	ccsbBroad304_03874	UBL5	-			
2969	32.37	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
2970	32.34	oe	ccsbBroad304_04387	MKI67IP	-			
2971	32.34	oe	ccsbBroad304_05981	CDO1	-			
2972	32.31	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
2973	32.31	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
2974	32.28	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
2975	32.28	kd	CGS001-55577	NAGK	-			
2976	32.26	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
2977	32.24	kd	CGS001-375318	AQP12A	Ion channels / Aquaporins			
2978	32.22	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
2979	32.14	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
2980	32.08	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
2981	32	kd	CGS001-22937	SCAP	WD repeat domain containing			
2982	31.99	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
2983	31.96	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
2984	31.93	kd	CGS001-55958	KLHL9	BTB/POZ domain containing			
2985	31.92	oe	ccsbBroad304_10437	STMN1	-			
2986	31.84	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
2987	31.82	kd	CGS001-7099	TLR4	Toll-like receptor family			
2988	31.82	kd	CGS001-8204	NRIP1	-			
2989	31.8	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
2990	31.79	kd	CGS001-84365	MKI67IP	-			
2991	31.78	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
2992	31.78	kd	CGS001-10891	PPARGC1A	RNA binding motif (RRM) containing			
2993	31.76	oe	ccsbBroad304_06140	EEF1D	-			
2994	31.73	kd	CGS001-221391	OPN5	GPCR / Class A : Opsin receptors			
2995	31.73	kd	CGS001-976	CD97	Adhesion Class GPCRs			
2996	31.69	oe	ccsbBroad304_01960	CASK	CASK family			
2997	31.66	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
2998	31.66	kd	CGS001-8649	LAMTOR3	-			
2999	31.6	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3000	31.59	oe	ccsbBroad304_00447	DLD	-			
3001	31.56	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
3002	31.56	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
3003	31.51	kd	CGS001-5590	PRKCZ	Iota subfamily			
3004	31.51	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
3005	31.47	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
3006	31.44	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
3007	31.42	kd	CGS001-5223	PGAM1	-			
3008	31.4	kd	CGS001-51031	GLOD4	-			
3009	31.34	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
3010	31.32	kd	CGS001-4122	MAN2A2	-			
3011	31.24	kd	CGS001-7311	UBA52	L ribosomal proteins			
3012	31.23	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
3013	31.11	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
3014	31.1	oe	ccsbBroad304_10212	GRHL3	-			
3015	31.09	kd	CGS001-6455	SH3GL1	-			
3016	31.04	kd	CGS001-6251	RSU1	-			
3017	30.95	oe	ccsbBroad304_00509	EPHX1	-			
3018	30.91	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
3019	30.9	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
3020	30.9	kd	CGS001-8453	CUL2	-			
3021	30.85	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
3022	30.85	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
3023	30.84	oe	ccsbBroad304_06095	DFFB	-			
3024	30.82	kd	CGS001-2538	G6PC	-			
3025	30.82	kd	CGS001-213	ALB	-			
3026	30.76	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
3027	30.75	kd	CGS001-9898	UBAP2L	-			
3028	30.75	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
3029	30.73	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
3030	30.73	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
3031	30.73	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
3032	30.69	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
3033	30.66	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
3034	30.66	cp	BRD-K82795137	loratadine	Histamine receptor antagonist		HRH1, CYP2C19, CYP3A5	Histamine receptor antagonist
3035	30.62	kd	CGS001-2052	EPHX1	-			
3036	30.57	oe	ccsbBroad304_02399	TNIP1	-			
3037	30.56	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
3038	30.55	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
3039	30.54	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
3040	30.53	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
3041	30.53	kd	CGS001-2786	GNG4	-			
3042	30.52	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
3043	30.51	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
3044	30.49	kd	CGS001-10955	SERINC3	-			
3045	30.49	kd	CGS001-4287	ATXN3	Ataxins			
3046	30.49	kd	CGS001-2	A2M	-			
3047	30.44	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
3048	30.44	kd	CGS001-10196	PRMT3	Protein arginine N-methyltransferases			
3049	30.43	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
3050	30.42	kd	CGS001-29116	MYLIP	-			
3051	30.39	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
3052	30.37	kd	CGS001-5682	PSMA1	Proteasome subunits			
3053	30.36	kd	CGS001-8477	GPR65	GPCR / Class A : Orphans			
3054	30.35	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
3055	30.35	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
3056	30.32	kd	CGS001-8505	PARG	-			
3057	30.3	kd	CGS001-29110	TBK1	IKK family			
3058	30.29	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
3059	30.27	kd	CGS001-3364	HUS1	-			
3060	30.26	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
3061	30.23	kd	CGS001-22841	RAB11FIP2	-			
3062	30.21	kd	CGS001-9441	MED26	-			
3063	30.2	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3064	30.19	kd	CGS001-10765	KDM5B	Histone demethylases			
3065	30.18	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
3066	30.18	kd	CGS001-3339	HSPG2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3067	30.17	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
3068	30.17	kd	CGS001-2260	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
3069	30.17	kd	CGS001-1642	DDB1	-			
3070	30.14	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
3071	30.13	kd	CGS001-2237	FEN1	-			
3072	30.08	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
3073	30.08	kd	CGS001-5018	OXA1L	-			
3074	30.07	kd	CGS001-2356	FPGS	-			
3075	30.06	oe	ccsbBroad304_00370	CS	-			
3076	30.04	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
3077	30.02	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
3078	30.01	kd	CGS001-5899	RALB	-			
3079	30	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
3080	29.97	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
3081	29.96	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
3082	29.95	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
3083	29.95	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
3084	29.94	kd	CGS001-3638	INSIG1	-			
3085	29.93	kd	CGS001-8463	TEAD2	-			
3086	29.84	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
3087	29.84	kd	CGS001-1152	CKB	-			
3088	29.83	oe	ccsbBroad304_02533	NOXA1	-			
3089	29.83	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3090	29.82	kd	CGS001-2534	FYN	Src family			
3091	29.79	oe	ccsbBroad304_02534	UTP14A	-			
3092	29.77	kd	CGS001-10973	ASCC3	-			
3093	29.76	oe	ccsbBroad304_01374	RAP1A	-			
3094	29.74	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
3095	29.74	kd	CGS001-23650	TRIM29	-			
3096	29.71	kd	CGS001-23523	CABIN1	-			
3097	29.67	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
3098	29.66	kd	CGS001-1827	RCAN1	-			
3099	29.64	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
3100	29.61	oe	ccsbBroad304_03072	GTPBP8	-			
3101	29.59	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
3102	29.56	cc		Toll like receptors LOF	-			
3103	29.56	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
3104	29.55	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
3105	29.55	kd	CGS001-10250	SRRM1	-			
3106	29.54	kd	CGS001-717	C2	Complement system			
3107	29.53	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
3108	29.52	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
3109	29.51	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
3110	29.51	kd	CGS001-23408	SIRT5	Histone deacetylases			
3111	29.49	oe	ccsbBroad304_00033	ADSS	-			
3112	29.49	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
3113	29.49	kd	CGS001-116443	GRIN3A	Glutamate receptors			
3114	29.43	oe	ccsbBroad304_07768	NISCH	-			
3115	29.43	kd	CGS001-7175	TPR	-			
3116	29.42	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
3117	29.4	cc		Leucine rich repeat kinase inhibitor	-			
3118	29.38	oe	ccsbBroad304_05152	SSBP4	-			
3119	29.36	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
3120	29.32	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
3121	29.3	kd	CGS001-3682	ITGAE	Integrins			
3122	29.29	kd	CGS001-5427	POLE2	DNA polymerases			
3123	29.28	oe	ccsbBroad304_08055	ATP5S	-			
3124	29.27	kd	CGS001-79618	HMBOX1	Homeoboxes / HNF class			
3125	29.23	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
3126	29.22	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
3127	29.21	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
3128	29.2	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
3129	29.17	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
3130	29.17	kd	CGS001-51564	HDAC7	Histone deacetylases			
3131	29.16	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
3132	29.16	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
3133	29.15	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
3134	29.12	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
3135	29.11	oe	ccsbBroad304_01976	EIF4EBP3	-			
3136	29.06	kd	CGS001-7296	TXNRD1	-			
3137	29.05	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
3138	29.04	kd	CGS001-9374	PPT2	-			
3139	29.03	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
3140	28.97	kd	CGS001-6804	STX1A	-			
3141	28.96	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
3142	28.94	kd	CGS001-100133941	CD24	CD molecules			
3143	28.92	kd	CGS001-10202	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3144	28.83	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3145	28.81	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
3146	28.8	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
3147	28.79	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
3148	28.76	oe	ccsbBroad304_07820	SNW1	-			
3149	28.73	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
3150	28.72	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
3151	28.7	oe	ccsbBroad304_07050	TFAP2A	-			
3152	28.6	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
3153	28.59	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
3154	28.58	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
3155	28.51	kd	CGS001-4680	CEACAM6	CD molecules			
3156	28.49	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3157	28.42	kd	CGS001-5546	PRCC	-			
3158	28.41	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
3159	28.36	kd	CGS001-22921	MSRB2	-			
3160	28.35	kd	CGS001-84433	CARD11	-			
3161	28.31	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
3162	28.3	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
3163	28.28	oe	ccsbBroad304_00060	AMBP	Lipocalins			
3164	28.26	kd	CGS001-11014	KDELR2	-			
3165	28.25	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
3166	28.18	cc		V type ATPases LOF	-			
3167	28.17	kd	CGS001-8527	DGKD	Pleckstrin homology (PH) domain containing			
3168	28.17	kd	CGS001-22794	CASC3	-			
3169	28.16	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
3170	28.14	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
3171	28.14	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
3172	28.12	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
3173	28.12	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
3174	28.09	kd	CGS001-4173	MCM4	-			
3175	28.08	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
3176	28.04	kd	CGS001-6856	SYPL1	-			
3177	28.02	kd	CGS001-2167	FABP4	Fatty acid binding protein family			
3178	28.01	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
3179	28.01	kd	CGS001-3654	IRAK1	Interleukin-1 receptor-associated kinase (IRAK) family			
3180	27.99	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
3181	27.97	cp	BRD-K52080565	rilmenidine	Imidazoline receptor agonist		NISCH	Imidazoline receptor agonist
3182	27.95	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
3183	27.95	kd	CGS001-5690	PSMB2	Proteasome subunits			
3184	27.93	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
3185	27.92	kd	CGS001-2959	GTF2B	General transcription factors			
3186	27.91	kd	CGS001-51001	MTERFD1	-			
3187	27.88	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
3188	27.88	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
3189	27.88	kd	CGS001-444	ASPH	-			
3190	27.84	kd	CGS001-3778	KCNMA1	Calcium-activated potassium channels			
3191	27.84	kd	CGS001-657	BMPR1A	Type I receptor serine/threonine kinases			
3192	27.8	kd	CGS001-10400	PEMT	-			
3193	27.75	kd	CGS001-10494	STK25	YSK subfamily			
3194	27.71	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
3195	27.7	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
3196	27.68	kd	CGS001-5993	RFX5	-			
3197	27.67	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
3198	27.51	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
3199	27.47	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
3200	27.45	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
3201	27.44	kd	CGS001-1460	CSNK2B	Casein kinase 2 (CK2) family			
3202	27.44	kd	CGS001-1349	COX7B	Mitochondrial respiratory chain complex			
3203	27.41	kd	CGS001-4846	NOS3	Nitric oxide synthases			
3204	27.36	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
3205	27.32	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
3206	27.32	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
3207	27.32	kd	CGS001-60528	ELAC2	-			
3208	27.31	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3209	27.3	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
3210	27.3	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
3211	27.29	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
3212	27.22	oe	ccsbBroad304_02890	SYF2	-			
3213	27.2	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
3214	27.19	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
3215	27.18	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
3216	27.17	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
3217	27.17	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
3218	27.17	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
3219	27.12	kd	CGS001-699	BUB1	Bub family			
3220	27.07	kd	CGS001-284	ANGPT1	Fibrinogen C domain containing			
3221	27.02	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
3222	27	kd	CGS001-10670	RRAGA	-			
3223	26.99	oe	ccsbBroad304_02589	COPS5	-			
3224	26.98	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
3225	26.96	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
3226	26.92	oe	ccsbBroad304_01613	STK11	LKB subfamily			
3227	26.9	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
3228	26.86	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
3229	26.85	kd	CGS001-5883	RAD9A	-			
3230	26.85	kd	CGS001-648	BMI1	Polycomb group ring fingers			
3231	26.83	oe	ccsbBroad304_08481	CEP55	-			
3232	26.82	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3233	26.78	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
3234	26.78	kd	CGS001-817	CAMK2D	CAMK2 family			
3235	26.74	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
3236	26.74	kd	CGS001-2617	GARS	Aminoacyl tRNA synthetases / Class II			
3237	26.64	kd	CGS001-51520	LARS	Aminoacyl tRNA synthetases / Class I			
3238	26.61	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
3239	26.61	kd	CGS001-383	ARG1	Arginase			
3240	26.58	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
3241	26.56	oe	ccsbBroad304_07890	CBX7	-			
3242	26.55	kd	CGS001-10972	TMED10	-			
3243	26.52	kd	CGS001-3957	LGALS2	Lectins, galactoside-binding			
3244	26.51	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
3245	26.49	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
3246	26.49	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
3247	26.46	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
3248	26.43	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
3249	26.41	kd	CGS001-9375	TM9SF2	-			
3250	26.4	kd	CGS001-6605	SMARCE1	-			
3251	26.38	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
3252	26.38	kd	CGS001-7029	TFDP2	-			
3253	26.37	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
3254	26.37	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
3255	26.33	kd	CGS001-5743	PTGS2	Cyclooxygenase			
3256	26.3	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
3257	26.27	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3258	26.26	kd	CGS001-1974	EIF4A2	DEAD-boxes			
3259	26.25	kd	CGS001-1051	CEBPB	basic leucine zipper proteins			
3260	26.22	kd	CGS001-23649	POLA2	DNA polymerases			
3261	26.21	kd	CGS001-563	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
3262	26.13	kd	CGS001-6046	BRD2	Bromodomain kinase (BRDK) family			
3263	26.08	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
3264	26.07	cc		Phospholipases GOF	-			
3265	26.05	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
3266	26.03	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
3267	25.98	kd	CGS001-23670	TMEM2	-			
3268	25.97	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
3269	25.91	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
3270	25.91	kd	CGS001-306	ANXA3	Annexins			
3271	25.9	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
3272	25.9	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
3273	25.89	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
3274	25.85	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
3275	25.8	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
3276	25.8	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
3277	25.8	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
3278	25.79	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
3279	25.78	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
3280	25.78	cp	BRD-K18523449	mestanolone	Androgenic steroid			Androgenic steroid
3281	25.73	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
3282	25.68	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
3283	25.67	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
3284	25.67	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
3285	25.66	oe	ccsbBroad304_00624	GCK	Hexokinases			
3286	25.65	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
3287	25.64	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
3288	25.61	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
3289	25.6	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
3290	25.58	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
3291	25.58	kd	CGS001-9519	TBPL1	-			
3292	25.57	oe	ccsbBroad304_00102	RND3	-			
3293	25.55	kd	CGS001-9541	CIR1	-			
3294	25.53	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
3295	25.52	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
3296	25.5	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
3297	25.46	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
3298	25.45	kd	CGS001-10329	TMEM5	-			
3299	25.44	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
3300	25.35	oe	ccsbBroad304_07197	PDHX	-			
3301	25.3	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3302	25.19	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
3303	25.15	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
3304	25.15	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
3305	25.14	oe	ccsbBroad304_00359	CPT1A	-			
3306	25.13	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
3307	25.12	kd	CGS001-9709	HERPUD1	-			
3308	25.1	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
3309	25.07	oe	ccsbBroad304_06789	PSEN2	Presenilin			
3310	25.07	kd	CGS001-23076	RRP1B	-			
3311	25.06	kd	CGS001-2729	GCLC	-			
3312	25.06	kd	CGS001-2247	FGF2	Endogenous ligands			
3313	24.97	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
3314	24.9	kd	CGS001-10379	IRF9	-			
3315	24.88	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
3316	24.87	oe	ccsbBroad304_02173	ATG5	-			
3317	24.87	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
3318	24.84	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
3319	24.83	kd	CGS001-23753	SDF2L1	-			
3320	24.81	kd	CGS001-308	ANXA5	Annexins			
3321	24.79	kd	CGS001-8780	RIOK3	RIO3 subfamily			
3322	24.77	kd	CGS001-5915	RARB	Retinoic acid receptors			
3323	24.73	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3324	24.71	cp	BRD-A70083328	secnidazole	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Microtubule inhibitor, Antiprotozoal
3325	24.7	kd	CGS001-11113	CIT	Other DMPK family kinases			
3326	24.67	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
3327	24.65	oe	ccsbBroad304_02604	B3GNT1	-			
3328	24.64	oe	ccsbBroad304_00941	LIG3	-			
3329	24.62	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
3330	24.58	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
3331	24.57	kd	CGS001-1594	CYP27B1	Cytochrome P450s			
3332	24.53	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
3333	24.5	kd	CGS001-5432	POLR2C	RNA polymerase subunits			
3334	24.49	kd	CGS001-10795	ZNF268	Zinc fingers, C2H2-type			
3335	24.49	kd	CGS001-2155	F7	Chymotrypsin			
3336	24.47	kd	CGS001-23536	ADAT1	-			
3337	24.46	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
3338	24.43	kd	CGS001-8892	EIF2B2	-			
3339	24.37	kd	CGS001-4170	MCL1	-			
3340	24.37	kd	CGS001-6927	HNF1A	Homeoboxes / HNF class			
3341	24.36	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
3342	24.34	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
3343	24.34	kd	CGS001-10481	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
3344	24.32	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
3345	24.32	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
3346	24.32	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
3347	24.31	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
3348	24.3	kd	CGS001-1345	COX6C	Mitochondrial respiratory chain complex			
3349	24.28	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
3350	24.26	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
3351	24.25	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
3352	24.23	oe	ccsbBroad304_02990	LYPD3	-			
3353	24.22	kd	CGS001-2015	EMR1	Adhesion Class GPCRs			
3354	24.22	kd	CGS001-9474	ATG5	-			
3355	24.2	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
3356	24.2	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
3357	24.17	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
3358	24.08	cc		JAK inhibitor	-			
3359	24.03	oe	ccsbBroad304_05907	BUB1B	Bub family			
3360	24.01	kd	CGS001-5164	PDK2	PDHK family			
3361	23.99	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3362	23.98	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
3363	23.98	kd	CGS001-2266	FGG	Endogenous ligands			
3364	23.93	kd	CGS001-1440	CSF3	Endogenous ligands			
3365	23.9	kd	CGS001-80274	SCUBE1	-			
3366	23.89	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
3367	23.88	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
3368	23.87	kd	CGS001-527	ATP6V0C	ATPases / V-type			
3369	23.85	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
3370	23.83	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
3371	23.82	cc		Poly ADP ribose polymerases LOF	-			
3372	23.78	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
3373	23.78	kd	CGS001-7105	TSPAN6	Tetraspanins			
3374	23.74	kd	CGS001-336	APOA2	Apolipoproteins			
3375	23.74	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
3376	23.73	kd	CGS001-64170	CARD9	-			
3377	23.72	kd	CGS001-2990	GUSB	-			
3378	23.71	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
3379	23.69	kd	CGS001-222546	RFX6	-			
3380	23.68	kd	CGS001-1820	ARID3A	-			
3381	23.67	oe	ccsbBroad304_09756	PAQR7	-			
3382	23.65	cc		BCL inhibitor	-			
3383	23.63	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
3384	23.62	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
3385	23.6	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
3386	23.57	kd	CGS001-29105	C16ORF80	-			
3387	23.56	kd	CGS001-6885	MAP3K7	MAPKKK:TAK1 subfamily			
3388	23.54	kd	CGS001-10554	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
3389	23.52	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3390	23.49	cc		Vesicular Transport LOF	-			
3391	23.42	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
3392	23.4	oe	ccsbBroad304_02633	LSM6	-			
3393	23.38	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
3394	23.36	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
3395	23.26	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
3396	23.21	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
3397	23.16	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
3398	23.16	kd	CGS001-2956	MSH6	-			
3399	23.16	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3400	23.13	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
3401	23.13	kd	CGS001-9322	TRIP10	-			
3402	23.12	kd	CGS001-283450	C12ORF51	-			
3403	23.09	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
3404	23.06	kd	CGS001-7248	TSC1	-			
3405	23.05	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
3406	23.01	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
3407	23	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
3408	23	kd	CGS001-901	CCNG2	-			
3409	22.97	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
3410	22.97	kd	CGS001-1856	DVL2	Dishevelled homologs			
3411	22.94	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
3412	22.94	kd	CGS001-1718	DHCR24	-			
3413	22.88	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
3414	22.84	kd	CGS001-64750	SMURF2	-			
3415	22.81	kd	CGS001-4751	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3416	22.8	kd	CGS001-7181	NR2C1	Testicular receptors			
3417	22.79	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
3418	22.75	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
3419	22.74	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
3420	22.69	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
3421	22.68	kd	CGS001-81894	SLC25A28	Miscellaneous SLC25 mitochondrial transporters			
3422	22.68	kd	CGS001-11162	NUDT6	Nudix motif containing			
3423	22.65	kd	CGS001-7079	TIMP4	-			
3424	22.64	oe	ccsbBroad304_03177	FIS1	-			
3425	22.61	kd	CGS001-5264	PHYH	-			
3426	22.61	kd	CGS001-5019	OXCT1	-			
3427	22.59	kd	CGS001-8833	GMPS	-			
3428	22.5	kd	CGS001-578	BAK1	-			
3429	22.47	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
3430	22.41	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
3431	22.39	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
3432	22.38	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
3433	22.36	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
3434	22.35	kd	CGS001-1644	DDC	Catecholamine turnover			
3435	22.33	oe	ccsbBroad304_02857	BAMBI	-			
3436	22.33	kd	CGS001-1066	CES1	Carboxylesterases			
3437	22.31	kd	CGS001-115650	TNFRSF13C	Tumour necrosis factor (TNF) receptor family			
3438	22.3	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
3439	22.3	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
3440	22.28	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
3441	22.25	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
3442	22.22	kd	CGS001-5050	PAFAH1B3	-			
3443	22.21	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
3444	22.2	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
3445	22.14	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
3446	22.11	kd	CGS001-6146	RPL22	L ribosomal proteins			
3447	22.1	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
3448	22.09	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
3449	22.04	kd	CGS001-125919	ZNF543	Zinc fingers, C2H2-type			
3450	22.04	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
3451	22.03	kd	CGS001-1314	COPA	Endogenous ligands			
3452	22	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3453	21.98	kd	CGS001-4151	MB	-			
3454	21.96	oe	ccsbBroad304_00865	ILF2	-			
3455	21.96	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
3456	21.96	kd	CGS001-5329	PLAUR	CD molecules			
3457	21.94	kd	CGS001-1677	DFFB	-			
3458	21.91	kd	CGS001-2864	FFAR1	Fatty acid receptors			
3459	21.85	oe	ccsbBroad304_04457	TOX2	-			
3460	21.83	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
3461	21.82	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
3462	21.81	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3463	21.8	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
3464	21.76	kd	CGS001-3269	HRH1	Histamine receptors			
3465	21.74	kd	CGS001-4208	MEF2C	Myocyte enhancer factors			
3466	21.69	kd	CGS001-6617	SNAPC1	-			
3467	21.68	kd	CGS001-10841	FTCD	-			
3468	21.67	oe	ccsbBroad304_02496	MTX2	-			
3469	21.6	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
3470	21.58	oe	ccsbBroad304_03773	CIAPIN1	-			
3471	21.57	kd	CGS001-3456	IFNB1	Interferons			
3472	21.51	kd	CGS001-55802	DCP1A	-			
3473	21.44	kd	CGS001-1111	CHEK1	CHK1 subfamily			
3474	21.42	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
3475	21.42	kd	CGS001-5591	PRKDC	Other PIKK family kinases			
3476	21.41	kd	CGS001-36	ACADSB	-			
3477	21.39	kd	CGS001-347736	NME9	-			
3478	21.3	kd	CGS001-2805	GOT1	-			
3479	21.29	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
3480	21.28	kd	CGS001-6757	SSX2	-			
3481	21.21	kd	CGS001-5817	PVR	Immunoglobulin superfamily / C2-set domain containing			
3482	21.19	kd	CGS001-6929	TCF3	Basic helix-loop-helix proteins			
3483	21.11	kd	CGS001-190	NR0B1	DAX-like receptors			
3484	21.05	kd	CGS001-1879	EBF1	-			
3485	21.04	kd	CGS001-10318	TNIP1	-			
3486	21.02	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
3487	20.93	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
3488	20.91	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
3489	20.9	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
3490	20.89	kd	CGS001-26086	GPSM1	Tetratricopeptide (TTC) repeat domain containing			
3491	20.87	oe	ccsbBroad304_00993	MDM4	-			
3492	20.86	kd	CGS001-57521	RPTOR	WD repeat domain containing			
3493	20.77	oe	ccsbBroad304_00161	BID	Endogenous ligands			
3494	20.74	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
3495	20.72	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
3496	20.69	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
3497	20.68	kd	CGS001-3783	KCNN4	Calcium-activated potassium channels			
3498	20.68	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
3499	20.67	kd	CGS001-11179	ZNF277	-			
3500	20.65	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
3501	20.63	kd	CGS001-10097	ACTR2	-			
3502	20.62	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
3503	20.61	kd	CGS001-6932	TCF7	-			
3504	20.57	kd	CGS001-4072	EPCAM	CD molecules			
3505	20.57	kd	CGS001-9774	BCLAF1	-			
3506	20.54	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
3507	20.5	kd	CGS001-5236	PGM1	-			
3508	20.49	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
3509	20.48	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
3510	20.46	kd	CGS001-29079	MED4	-			
3511	20.32	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
3512	20.31	kd	CGS001-8655	DYNLL1	Cytoplasmic dyneins			
3513	20.25	oe	ccsbBroad304_06290	GNA15	-			
3514	20.25	oe	ccsbBroad304_01872	DGCR14	-			
3515	20.25	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
3516	20.23	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
3517	20.21	oe	ccsbBroad304_07766	RASSF1	-			
3518	20.1	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
3519	20.1	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
3520	20.07	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
3521	20.07	kd	CGS001-58477	SRPRB	-			
3522	20.05	cc		Proteasome Pathway LOF	-			
3523	20.05	kd	CGS001-81611	ANP32E	ANP32 acidic nuclear phosphoproteins			
3524	20.04	oe	ccsbBroad304_02834	GABARAPL1	-			
3525	20.04	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
3526	20.03	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
3527	19.98	kd	CGS001-256281	NUDT14	Nudix motif containing			
3528	19.98	kd	CGS001-9700	ESPL1	-			
3529	19.97	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
3530	19.93	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
3531	19.89	kd	CGS001-1070	CETN3	EF-hand domain containing			
3532	19.86	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3533	19.86	kd	CGS001-6286	S100P	EF-hand domain containing			
3534	19.85	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
3535	19.8	kd	CGS001-6652	SORD	-			
3536	19.74	oe	ccsbBroad304_01208	PITPNA	-			
3537	19.7	kd	CGS001-7572	ZNF24	Zinc fingers, C2H2-type			
3538	19.7	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
3539	19.69	kd	CGS001-84971	ATG4D	-			
3540	19.66	kd	CGS001-167826	OLIG3	Basic helix-loop-helix proteins			
3541	19.64	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
3542	19.59	kd	CGS001-7039	TGFA	-			
3543	19.58	oe	ccsbBroad304_02756	RRP8	-			
3544	19.58	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
3545	19.52	kd	CGS001-11336	EXOC3	-			
3546	19.48	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
3547	19.48	kd	CGS001-3601	IL15RA	IL-2 receptor family			
3548	19.46	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
3549	19.41	kd	CGS001-3565	IL4	Interleukins and interleukin receptors			
3550	19.39	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
3551	19.36	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
3552	19.35	kd	CGS001-7374	UNG	-			
3553	19.33	kd	CGS001-23512	SUZ12	Zinc fingers, C2H2-type			
3554	19.32	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
3555	19.24	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
3556	19.16	kd	CGS001-3029	HAGH	-			
3557	19.1	kd	CGS001-149233	IL23R	IL-12 receptor family			
3558	19.09	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
3559	19.08	oe	ccsbBroad304_04649	ADC	-			
3560	19.08	kd	CGS001-10295	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
3561	19.05	kd	CGS001-2145	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
3562	18.96	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
3563	18.91	oe	ccsbBroad304_00794	HSF1	-			
3564	18.88	oe	ccsbBroad304_02425	CDIPT	-			
3565	18.86	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
3566	18.85	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
3567	18.82	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
3568	18.81	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
3569	18.8	kd	CGS001-4837	NNMT	-			
3570	18.8	kd	CGS001-51182	HSPA14	Heat shock proteins / HSP70			
3571	18.8	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
3572	18.78	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
3573	18.73	kd	CGS001-2138	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
3574	18.7	kd	CGS001-1407	CRY1	-			
3575	18.67	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
3576	18.62	kd	CGS001-4299	AFF1	-			
3577	18.6	kd	CGS001-9655	SOCS5	SH2 domain containing			
3578	18.57	kd	CGS001-581	BAX	-			
3579	18.52	kd	CGS001-10094	ARPC3	Actin related protein 2/3 complex subunits			
3580	18.48	oe	ccsbBroad304_03420	TOLLIP	-			
3581	18.45	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
3582	18.44	kd	CGS001-11198	SUPT16H	-			
3583	18.39	kd	CGS001-55234	SMU1	WD repeat domain containing			
3584	18.38	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
3585	18.35	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
3586	18.31	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
3587	18.23	kd	CGS001-29968	PSAT1	-			
3588	18.17	kd	CGS001-5653	KLK6	Chymotrypsin			
3589	18.15	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
3590	18.05	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
3591	17.99	kd	CGS001-390212	GPR152	GPCR / Class A : Orphans			
3592	17.96	kd	CGS001-10465	PPIH	-			
3593	17.96	kd	CGS001-3612	IMPA1	Inositol monophosphatase			
3594	17.9	oe	ccsbBroad304_00816	IDE	Pitrilysin			
3595	17.9	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
3596	17.89	kd	CGS001-133522	PPARGC1B	RNA binding motif (RRM) containing			
3597	17.86	kd	CGS001-3155	HMGCL	-			
3598	17.77	oe	ccsbBroad304_02136	COPS2	-			
3599	17.76	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
3600	17.73	kd	CGS001-5950	RBP4	Lipocalins			
3601	17.69	kd	CGS001-1445	CSK	Csk family			
3602	17.67	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
3603	17.62	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
3604	17.61	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
3605	17.55	kd	CGS001-23028	KDM1A	Histone demethylase			
3606	17.53	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
3607	17.49	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
3608	17.49	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
3609	17.48	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
3610	17.38	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
3611	17.34	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3612	17.33	kd	CGS001-4893	NRAS	RAS subfamily			
3613	17.32	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
3614	17.31	cc		IMPDH inhibitor	-			
3615	17.29	cc		PKC inhibitor	-			
3616	17.25	kd	CGS001-57665	RDH14	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3617	17.23	kd	CGS001-11257	TP53TG1	-			
3618	17.16	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
3619	17.14	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
3620	17.04	kd	CGS001-51222	ZNF219	Zinc fingers, C2H2-type			
3621	17.04	kd	CGS001-1606	DGKA	EF-hand domain containing			
3622	17.04	kd	CGS001-836	CASP3	Caspases			
3623	16.87	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
3624	16.85	kd	CGS001-892	CCNC	-			
3625	16.84	kd	CGS001-3827	KNG1	Endogenous ligands			
3626	16.84	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
3627	16.83	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
3628	16.8	kd	CGS001-23314	SATB2	Homeoboxes / CUT class			
3629	16.76	kd	CGS001-25801	GCA	EF-hand domain containing			
3630	16.66	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
3631	16.63	kd	CGS001-158	ADSL	-			
3632	16.61	cc		HMGCR inhibitor	-			
3633	16.58	kd	CGS001-10128	LRPPRC	-			
3634	16.48	kd	CGS001-506	ATP5B	ATPases / F-type			
3635	16.43	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
3636	16.39	kd	CGS001-5987	TRIM27	-			
3637	16.38	kd	CGS001-80314	EPC1	-			
3638	16.37	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
3639	16.21	kd	CGS001-54541	DDIT4	-			
3640	16.2	cc		Aurora kinase inhibitor	-			
3641	16.06	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
3642	15.99	kd	CGS001-771	CA12	Carbonic anhydrases			
3643	15.96	oe	ccsbBroad304_13903	MTAP	-			
3644	15.93	kd	CGS001-822	CAPG	-			
3645	15.88	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
3646	15.75	kd	CGS001-662	BNIP1	-			
3647	15.71	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
3648	15.71	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3649	15.62	kd	CGS001-5933	RBL1	-			
3650	15.55	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
3651	15.51	kd	CGS001-4711	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
3652	15.47	kd	CGS001-10725	NFAT5	Nuclear factor of activated T-cells			
3653	15.42	cc		FLT3 inhibitor	-			
3654	15.39	kd	CGS001-22949	PTGR1	-			
3655	15.39	kd	CGS001-1184	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
3656	15.37	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3657	15.18	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
3658	15.13	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
3659	15.1	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
3660	15.06	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
3661	15.06	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
3662	15.01	kd	CGS001-3123	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
3663	15	kd	CGS001-5894	RAF1	RAF family			
3664	14.97	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
3665	14.97	kd	CGS001-1036	CDO1	-			
3666	14.94	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
3667	14.91	kd	CGS001-124535	HSF5	-			
3668	14.82	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
3669	14.74	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
3670	14.7	oe	ccsbBroad304_02092	SYNGR3	-			
3671	14.67	oe	ccsbBroad304_05963	CD44	CD molecules			
3672	14.67	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
3673	14.55	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
3674	14.53	kd	CGS001-1906	EDN1	Endogenous ligands			
3675	14.43	oe	ccsbBroad304_06777	PRNP	CD molecules			
3676	14.41	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
3677	14.38	oe	ccsbBroad304_01035	MSH5	-			
3678	14.29	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
3679	14.17	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3680	14.06	kd	CGS001-2289	FKBP5	Tetratricopeptide (TTC) repeat domain containing			
3681	14.05	cc		General transcription factors group 1 LOF	-			
3682	14.05	kd	CGS001-3119	HLA-DQB1	Immunoglobulin superfamily / C1-set domain containing			
3683	14.04	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
3684	13.81	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
3685	13.81	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
3686	13.8	kd	CGS001-6810	STX4	-			
3687	13.77	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
3688	13.53	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
3689	13.52	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
3690	13.48	kd	CGS001-23192	ATG4B	Aut2 peptidase			
3691	13.43	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
3692	13.33	kd	CGS001-2263	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
3693	13.29	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
3694	13.28	kd	CGS001-7771	ZFP112	-			
3695	13.1	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
3696	13.06	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
3697	13.02	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
3698	12.96	kd	CGS001-6464	SHC1	SH2 domain containing			
3699	12.69	oe	ccsbBroad304_06180	ESD	-			
3700	12.68	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
3701	12.65	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
3702	12.65	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3703	12.64	oe	ccsbBroad304_05749	A2M	-			
3704	12.63	kd	CGS001-545	ATR	ATR subfamily			
3705	12.42	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
3706	12.22	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
3707	12.21	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
3708	12.17	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
3709	11.97	kd	CGS001-83737	ITCH	-			
3710	11.85	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
3711	11.79	kd	CGS001-262	AMD1	Decarboxylases			
3712	11.76	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
3713	11.59	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
3714	11.58	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
3715	11.52	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3716	11.51	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
3717	11.5	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
3718	11.41	kd	CGS001-4929	NR4A2	Nerve growth factor IB-like receptors			
3719	11.3	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
3720	11.27	kd	CGS001-5925	RB1	Endogenous ligands			
3721	11.2	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
3722	11.13	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
3723	11.08	kd	CGS001-56731	SLC2A4RG	-			
3724	10.94	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
3725	10.91	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
3726	10.83	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
3727	10.73	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
3728	10.55	cp	BRD-K30563334	rifabutin	Protein synthesis inhibitor		CYP3A4, HSP90AA1, HSP90B1	Protein synthesis inhibitor
3729	10.48	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
3730	10.46	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
3731	10.29	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
3732	10.21	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
3733	9.94	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
3734	9.81	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
3735	9.57	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
3736	9.55	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
3737	9.52	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
3738	9.5	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
3739	9.24	cc		BMP Signaling LOF	-			
3740	8.95	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
3741	8.95	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
3742	8.33	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
3743	7.72	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3744	7.65	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
3745	7.47	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
3746	7.47	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
3747	7.27	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
3748	7.14	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
3749	6.95	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3750	6.76	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
3751	6.57	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
3752	6.15	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
3753	6.1	kd	CGS001-8536	CAMK1	CAMK1 family			
3754	5.24	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
3755	4.99	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
3756	4.55	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
3757	2.34	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
3758	-3.68	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
3759	-4.92	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
3760	-4.97	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
3761	-5.23	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
3762	-5.49	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
3763	-5.69	oe	ccsbBroad304_07012	STK3	MST subfamily			
3764	-6.04	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
3765	-6.06	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
3766	-6.21	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
3767	-6.71	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
3768	-6.75	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
3769	-6.81	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
3770	-7	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
3771	-7.08	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
3772	-7.26	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
3773	-7.29	oe	ccsbBroad304_06424	IFI16	-			
3774	-7.43	cc		Rho associated kinase inhibitor	-			
3775	-7.46	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
3776	-7.56	kd	CGS001-2475	MTOR	FRAP subfamily			
3777	-7.74	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
3778	-7.85	oe	ccsbBroad304_05937	CASP7	Caspases			
3779	-7.93	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
3780	-8.16	kd	CGS001-9156	EXO1	-			
3781	-8.81	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
3782	-8.97	kd	CGS001-2674	GFRA1	GDNF receptor family			
3783	-8.99	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
3784	-9.11	kd	CGS001-3932	LCK	Src family			
3785	-9.15	oe	ccsbBroad304_08392	EXOC6	-			
3786	-9.2	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
3787	-9.37	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
3788	-9.45	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
3789	-9.64	kd	CGS001-5062	PAK2	PAKA subfamily			
3790	-9.65	oe	ccsbBroad304_02592	KIF2C	Kinesins			
3791	-9.69	oe	ccsbBroad304_07662	NPRL2	-			
3792	-9.75	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3793	-9.87	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
3794	-9.96	kd	CGS001-3163	HMOX2	Haem oxygenase			
3795	-10.06	oe	ccsbBroad304_02018	SUCLA2	-			
3796	-10.26	kd	CGS001-5573	PRKAR1A	Protein kinase A			
3797	-10.36	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
3798	-10.46	oe	ccsbBroad304_02032	TSC22D1	-			
3799	-10.47	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
3800	-10.5	oe	ccsbBroad304_06004	CKB	-			
3801	-10.52	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
3802	-10.54	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
3803	-10.54	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
3804	-10.65	kd	CGS001-2287	FKBP3	-			
3805	-10.69	kd	CGS001-8681	JMJD7-PLA2G4B	-			
3806	-10.71	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
3807	-10.72	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
3808	-10.82	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
3809	-10.92	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
3810	-10.95	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
3811	-11.07	oe	ccsbBroad304_02415	TUBB3	Tubulins			
3812	-11.14	cc		NADH ubiquinone oxidoreductase supernumerary subunits LOF	-			
3813	-11.17	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
3814	-11.2	kd	CGS001-3675	ITGA3	Integrins			
3815	-11.24	oe	ccsbBroad304_00179	BTG1	-			
3816	-11.25	oe	ccsbBroad304_03615	ZNF673	-			
3817	-11.34	oe	ccsbBroad304_01724	TTR	-			
3818	-11.4	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
3819	-11.55	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
3820	-11.61	kd	CGS001-6776	STAT5A	SH2 domain containing			
3821	-11.85	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
3822	-11.9	kd	CGS001-5411	PNN	-			
3823	-11.99	oe	ccsbBroad304_02270	FAM20B	-			
3824	-12.02	kd	CGS001-4602	MYB	-			
3825	-12.03	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
3826	-12.15	cc		DNA dependent protein kinase inhibitor	-			
3827	-12.16	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
3828	-12.24	kd	CGS001-32	ACACB	Carboxylases			
3829	-12.34	kd	CGS001-10632	ATP5L	ATPases / F-type			
3830	-12.42	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
3831	-12.44	kd	CGS001-115201	ATG4A	-			
3832	-12.49	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
3833	-12.64	oe	ccsbBroad304_07208	NRIP1	-			
3834	-12.64	oe	ccsbBroad304_04190	CCDC92	-			
3835	-12.84	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
3836	-12.87	oe	ccsbBroad304_01485	SC5DL	-			
3837	-12.89	cc		HOXL subclass homeoboxes LOF	-			
3838	-12.89	kd	CGS001-1869	E2F1	-			
3839	-12.92	kd	CGS001-5575	PRKAR1B	Protein kinase A			
3840	-12.97	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
3841	-13.01	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
3842	-13.04	cp	BRD-K25310650	ormetoprim	Bacterial antifolate			Bacterial antifolate
3843	-13.08	kd	CGS001-4790	NFKB1	NFkappaB transcription factor family			
3844	-13.11	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
3845	-13.19	kd	CGS001-93185	IGSF8	CD molecules			
3846	-13.2	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
3847	-13.21	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
3848	-13.22	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
3849	-13.23	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
3850	-13.29	kd	CGS001-10253	SPRY2	-			
3851	-13.3	oe	ccsbBroad304_08802	ELAC2	-			
3852	-13.36	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
3853	-13.37	cc		Potassium channel blocker	-			
3854	-13.38	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
3855	-13.42	kd	CGS001-4292	MLH1	-			
3856	-13.45	kd	CGS001-2932	GSK3B	GSK subfamily			
3857	-13.69	cc		Aldehyde dehydrogenases LOF	-			
3858	-13.74	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
3859	-13.74	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
3860	-13.82	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
3861	-13.85	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3862	-13.92	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
3863	-13.97	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
3864	-13.99	kd	CGS001-3664	IRF6	-			
3865	-14	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
3866	-14.01	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
3867	-14.05	cc		General transcription factors group 2 LOF	-			
3868	-14.05	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
3869	-14.13	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
3870	-14.14	oe	ccsbBroad304_00876	INSIG1	-			
3871	-14.14	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
3872	-14.28	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
3873	-14.39	oe	ccsbBroad304_06916	SCP2	-			
3874	-14.39	kd	CGS001-4697	NDUFA4	-			
3875	-14.41	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
3876	-14.45	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
3877	-14.49	oe	ccsbBroad304_13880	IDH3G	-			
3878	-14.72	cp	BRD-K32744045	disulfiram	Aldehyde dehydrogenase inhibitor		ALDH2, ALDH1A2, ALDH5A1, ALDH7A1, CYP2E1, DBH, DNMT1, TRPA1	Aldehyde dehydrogenase inhibitor, TRPV agonist, DNA methyltransferase inhibitor
3879	-14.72	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
3880	-14.84	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
3881	-14.88	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
3882	-14.92	kd	CGS001-10873	ME3	-			
3883	-14.93	kd	CGS001-25	ABL1	Abl family			
3884	-14.94	kd	CGS001-10289	EIF1B	-			
3885	-15.18	oe	ccsbBroad304_01769	VEGFB	-			
3886	-15.21	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
3887	-15.24	kd	CGS001-403	ARL3	ADP-ribosylation factors			
3888	-15.26	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
3889	-15.26	kd	CGS001-7423	VEGFB	-			
3890	-15.27	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
3891	-15.28	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
3892	-15.32	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
3893	-15.38	kd	CGS001-1105	CHD1	-			
3894	-15.39	cc		Minor histocompatibility antigens LOF	-			
3895	-15.4	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
3896	-15.4	kd	CGS001-6364	CCL20	Chemokine ligands			
3897	-15.41	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
3898	-15.43	kd	CGS001-23066	CAND2	-			
3899	-15.45	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
3900	-15.49	oe	ccsbBroad304_03853	LSM2	-			
3901	-15.51	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
3902	-15.61	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
3903	-15.63	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
3904	-15.63	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
3905	-15.7	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
3906	-15.73	kd	CGS001-85004	RERG	-			
3907	-15.74	kd	CGS001-5052	PRDX1	-			
3908	-15.75	kd	CGS001-2987	GUK1	-			
3909	-15.77	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
3910	-15.8	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
3911	-15.84	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
3912	-15.86	kd	CGS001-10472	ZNF238	-			
3913	-15.88	kd	CGS001-2837	UTS2R	Urotensin receptor			
3914	-15.89	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
3915	-15.9	kd	CGS001-93349	SP140L	Zinc fingers, PHD-type			
3916	-15.96	oe	ccsbBroad304_01623	SUPT4H1	-			
3917	-15.96	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
3918	-15.96	kd	CGS001-5361	PLXNA1	Plexins			
3919	-16	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3920	-16.04	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
3921	-16.07	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
3922	-16.1	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
3923	-16.18	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
3924	-16.19	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
3925	-16.4	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
3926	-16.41	kd	CGS001-210	ALAD	-			
3927	-16.42	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
3928	-16.43	kd	CGS001-10013	HDAC6	Histone deacetylases			
3929	-16.45	cc		Dopamine receptor antagonist	-			
3930	-16.61	kd	CGS001-6715	SRD5A1	-			
3931	-16.62	kd	CGS001-11200	CHEK2	CHK1 subfamily			
3932	-16.63	kd	CGS001-11164	NUDT5	Nudix motif containing			
3933	-16.67	cp	BRD-K47780086	penciclovir	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor
3934	-16.75	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
3935	-16.75	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
3936	-16.77	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
3937	-16.82	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
3938	-16.83	oe	ccsbBroad304_04294	ATG10	-			
3939	-16.88	kd	CGS001-5163	PDK1	-			
3940	-16.89	kd	CGS001-2099	ESR1	Estrogen receptors			
3941	-16.99	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
3942	-17.03	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
3943	-17.04	kd	CGS001-54498	SMOX	-			
3944	-17.05	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
3945	-17.08	cc		Glycogen synthase kinase inhibitor	-			
3946	-17.09	kd	CGS001-644	BLVRA	-			
3947	-17.19	kd	CGS001-10398	MYL9	EF-hand domain containing			
3948	-17.21	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
3949	-17.25	kd	CGS001-391013	PLA2G2C	-			
3950	-17.27	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
3951	-17.31	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
3952	-17.33	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
3953	-17.33	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
3954	-17.35	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
3955	-17.36	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
3956	-17.37	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
3957	-17.38	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
3958	-17.4	kd	CGS001-222894	FERD3L	Basic helix-loop-helix proteins			
3959	-17.42	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
3960	-17.44	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
3961	-17.46	kd	CGS001-5501	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3962	-17.48	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
3963	-17.48	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
3964	-17.49	oe	ccsbBroad304_01556	SMARCB1	-			
3965	-17.49	kd	CGS001-2254	FGF9	Endogenous ligands			
3966	-17.5	kd	CGS001-160	AP2A1	-			
3967	-17.52	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
3968	-17.54	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
3969	-17.54	kd	CGS001-5881	RAC3	Endogenous ligands			
3970	-17.59	kd	CGS001-1287	COL4A5	Collagens			
3971	-17.6	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
3972	-17.63	oe	ccsbBroad304_09615	LACC1	-			
3973	-17.63	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
3974	-17.63	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
3975	-17.67	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
3976	-17.68	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
3977	-17.74	kd	CGS001-55011	PIH1D1	-			
3978	-17.76	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
3979	-17.76	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
3980	-17.77	kd	CGS001-57504	MTA3	GATA zinc finger domain containing			
3981	-17.77	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
3982	-17.8	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
3983	-17.88	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3984	-17.89	kd	CGS001-384	ARG2	Arginase			
3985	-17.93	kd	CGS001-1854	DUT	-			
3986	-17.94	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
3987	-17.97	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
3988	-17.99	kd	CGS001-54899	PXK	Slob family			
3989	-18.03	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
3990	-18.08	kd	CGS001-3895	KTN1	-			
3991	-18.1	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
3992	-18.1	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
3993	-18.14	kd	CGS001-55500	ETNK1	-			
3994	-18.19	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
3995	-18.2	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3996	-18.2	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
3997	-18.21	kd	CGS001-28511	NKIRAS2	-			
3998	-18.22	kd	CGS001-3428	IFI16	-			
3999	-18.23	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
4000	-18.24	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
4001	-18.27	kd	CGS001-84290	CAPNS2	EF-hand domain containing			
4002	-18.28	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4003	-18.3	kd	CGS001-221895	JAZF1	Zinc fingers, C2H2-type			
4004	-18.31	kd	CGS001-4255	MGMT	-			
4005	-18.38	oe	ccsbBroad304_01142	PAFAH1B2	-			
4006	-18.39	oe	ccsbBroad304_06301	GOT2	-			
4007	-18.42	kd	CGS001-7471	WNT1	Endogenous ligands			
4008	-18.44	kd	CGS001-51172	NAGPA	-			
4009	-18.5	kd	CGS001-338557	O3FAR1	-			
4010	-18.52	oe	ccsbBroad304_00150	BAX	-			
4011	-18.52	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
4012	-18.53	kd	CGS001-5336	PLCG2	Phosphoinositide-specific phospholipase C			
4013	-18.59	kd	CGS001-7263	TST	-			
4014	-18.65	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
4015	-18.65	kd	CGS001-3670	ISL1	Homeoboxes / LIM class			
4016	-18.67	kd	CGS001-5226	PGD	-			
4017	-18.7	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
4018	-18.71	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
4019	-18.91	kd	CGS001-1499	CTNNB1	Catenins			
4020	-18.92	kd	CGS001-51079	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
4021	-18.94	kd	CGS001-53343	NUDT9	Nudix motif containing			
4022	-18.97	kd	CGS001-7353	UFD1L	-			
4023	-18.97	kd	CGS001-56139	PCDHA10	Cadherins / Protocadherins : Clustered			
4024	-18.98	kd	CGS001-7187	TRAF3	-			
4025	-19.01	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
4026	-19.04	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
4027	-19.06	kd	CGS001-4143	MAT1A	-			
4028	-19.08	kd	CGS001-7083	TK1	-			
4029	-19.08	kd	CGS001-50808	AK3	-			
4030	-19.09	cc		GATA Zinc finger domain containing LOF	-			
4031	-19.09	kd	CGS001-2002	ELK1	ETS Transcription Factors			
4032	-19.12	kd	CGS001-3127	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
4033	-19.12	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
4034	-19.13	kd	CGS001-998	CDC42	-			
4035	-19.14	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
4036	-19.14	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
4037	-19.21	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4038	-19.22	oe	ccsbBroad304_02231	USP6NL	-			
4039	-19.23	kd	CGS001-57018	CCNL1	-			
4040	-19.27	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4041	-19.34	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
4042	-19.37	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
4043	-19.37	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
4044	-19.39	kd	CGS001-83593	RASSF5	-			
4045	-19.4	oe	ccsbBroad304_00489	EHHADH	-			
4046	-19.4	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
4047	-19.43	kd	CGS001-9111	NMI	-			
4048	-19.45	oe	ccsbBroad304_01675	TK1	-			
4049	-19.46	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
4050	-19.47	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
4051	-19.49	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
4052	-19.5	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
4053	-19.5	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
4054	-19.53	kd	CGS001-55810	FOXJ2	Forkhead boxes			
4055	-19.57	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
4056	-19.59	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4057	-19.61	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
4058	-19.62	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4059	-19.63	kd	CGS001-2773	GNAI3	-			
4060	-19.64	kd	CGS001-5134	PDCD2	Zinc fingers, MYND-type			
4061	-19.65	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
4062	-19.66	cc		Topoisomerase inhibitor	-			
4063	-19.69	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
4064	-19.72	kd	CGS001-2550	GABBR1	GABA receptors			
4065	-19.73	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
4066	-19.74	oe	ccsbBroad304_07827	STK38L	NDR family			
4067	-19.74	oe	ccsbBroad304_02716	NMNAT2	-			
4068	-19.74	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4069	-19.75	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
4070	-19.75	kd	CGS001-5660	PSAP	Endogenous ligands			
4071	-19.77	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
4072	-19.79	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
4073	-19.8	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
4074	-19.83	kd	CGS001-8848	TSC22D1	-			
4075	-19.85	kd	CGS001-8543	LMO4	-			
4076	-19.87	kd	CGS001-50943	FOXP3	Forkhead boxes			
4077	-19.88	oe	ccsbBroad304_00783	HPRT1	-			
4078	-19.89	kd	CGS001-2232	FDXR	-			
4079	-19.92	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
4080	-19.96	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
4081	-19.99	kd	CGS001-7159	TP53BP2	Ankyrin repeat domain containing			
4082	-20.02	kd	CGS001-2882	GPX7	-			
4083	-20.03	kd	CGS001-23014	FBXO21	F-boxes / other			
4084	-20.06	kd	CGS001-327	APEH	Prolyl oligopeptidase			
4085	-20.08	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
4086	-20.09	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
4087	-20.11	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4088	-20.2	kd	CGS001-140690	CTCFL	Zinc fingers, C2H2-type			
4089	-20.2	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
4090	-20.21	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
4091	-20.22	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
4092	-20.25	cp	BRD-K39983086	loteprednol	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Phospholipase inhibitor
4093	-20.27	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
4094	-20.27	kd	CGS001-11340	EXOSC8	-			
4095	-20.29	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
4096	-20.29	kd	CGS001-23466	CBX6	-			
4097	-20.32	cc		Lysine acetyltransferases LOF	-			
4098	-20.32	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
4099	-20.38	cp	BRD-K66896231	BRD-K66896231	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
4100	-20.39	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
4101	-20.4	kd	CGS001-399694	SHC4	SH2 domain containing			
4102	-20.42	kd	CGS001-4976	OPA1	-			
4103	-20.51	kd	CGS001-64147	KIF9	Kinesins			
4104	-20.57	kd	CGS001-8569	MKNK1	MKN subfamily			
4105	-20.59	cc		G2 M Checkpoint LOF	-			
4106	-20.59	cc		Apolipoproteins LOF	-			
4107	-20.63	cc		X linked mental retardation group 2 LOF	-			
4108	-20.63	kd	CGS001-54108	CHRAC1	-			
4109	-20.64	kd	CGS001-1195	CLK1	CDC-like kinases			
4110	-20.65	kd	CGS001-10682	EBP	-			
4111	-20.67	kd	CGS001-148103	ZNF599	Zinc fingers, C2H2-type			
4112	-20.74	kd	CGS001-11041	B3GNT1	-			
4113	-20.76	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
4114	-20.76	kd	CGS001-64135	IFIH1	-			
4115	-20.76	kd	CGS001-64241	ABCG8	ATP binding cassette transporters / subfamily G			
4116	-20.78	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
4117	-20.79	oe	ccsbBroad304_06993	SRD5A1	-			
4118	-20.79	kd	CGS001-2147	F2	Endogenous ligands			
4119	-20.8	oe	ccsbBroad304_03173	TMED7	-			
4120	-20.8	oe	ccsbBroad304_00459	DPYD	-			
4121	-20.8	kd	CGS001-637	BID	Endogenous ligands			
4122	-20.82	kd	CGS001-6850	SYK	Syk family			
4123	-20.84	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
4124	-20.87	kd	CGS001-10287	RGS19	Regulators of G-protein signaling			
4125	-20.87	kd	CGS001-1374	CPT1A	-			
4126	-20.9	kd	CGS001-5805	PTS	-			
4127	-20.94	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
4128	-20.97	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
4129	-20.98	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
4130	-20.98	kd	CGS001-1030	CDKN2B	-			
4131	-21.01	kd	CGS001-55139	ANKZF1	Ankyrin repeat domain containing			
4132	-21.05	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
4133	-21.1	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
4134	-21.1	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
4135	-21.13	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
4136	-21.13	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
4137	-21.13	kd	CGS001-3560	IL2RB	IL-2 receptor family			
4138	-21.13	kd	CGS001-94235	GNG8	-			
4139	-21.18	kd	CGS001-91304	C19ORF6	-			
4140	-21.19	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
4141	-21.19	kd	CGS001-3481	IGF2	-			
4142	-21.2	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
4143	-21.2	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
4144	-21.27	oe	ccsbBroad304_03544	FAIM	-			
4145	-21.31	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
4146	-21.31	kd	CGS001-5621	PRNP	CD molecules			
4147	-21.36	kd	CGS001-8835	SOCS2	SH2 domain containing			
4148	-21.37	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4149	-21.48	kd	CGS001-9133	CCNB2	-			
4150	-21.51	cc		MTOR inhibitor	-			
4151	-21.51	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
4152	-21.55	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
4153	-21.58	oe	ccsbBroad304_08878	METTL4	-			
4154	-21.61	kd	CGS001-1128	CHRM1	Cholinergic receptors			
4155	-21.63	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
4156	-21.63	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
4157	-21.69	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
4158	-21.7	kd	CGS001-3312	HSPA8	Heat shock proteins / HSP70			
4159	-21.7	kd	CGS001-2957	GTF2A1	General transcription factors			
4160	-21.72	oe	ccsbBroad304_00006	ACADM	-			
4161	-21.76	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
4162	-21.77	kd	CGS001-182	JAG1	CD molecules			
4163	-21.81	kd	CGS001-10921	RNPS1	RNA binding motif (RRM) containing			
4164	-21.82	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
4165	-21.82	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
4166	-21.84	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
4167	-21.86	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
4168	-21.87	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
4169	-21.9	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
4170	-21.91	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
4171	-21.91	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
4172	-21.92	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
4173	-21.94	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
4174	-21.94	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
4175	-21.95	kd	CGS001-5292	PIM1	PIM family			
4176	-21.96	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
4177	-21.98	kd	CGS001-6917	TCEA1	General transcription factors			
4178	-21.99	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
4179	-22	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
4180	-22.02	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
4181	-22.03	kd	CGS001-3460	IFNGR2	Interferon receptor family			
4182	-22.06	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
4183	-22.08	oe	ccsbBroad304_00118	ATIC	-			
4184	-22.1	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4185	-22.11	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
4186	-22.15	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
4187	-22.2	kd	CGS001-7031	TFF1	-			
4188	-22.24	kd	CGS001-11180	WDR6	WD repeat domain containing			
4189	-22.24	kd	CGS001-4144	MAT2A	-			
4190	-22.25	kd	CGS001-59343	SENP2	-			
4191	-22.26	oe	ccsbBroad304_06855	RDX	-			
4192	-22.26	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
4193	-22.26	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
4194	-22.27	kd	CGS001-56882	CDC42SE1	-			
4195	-22.28	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
4196	-22.3	kd	CGS001-4547	MTTP	-			
4197	-22.33	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
4198	-22.38	kd	CGS001-3718	JAK3	Janus kinase (JakA) family			
4199	-22.39	oe	ccsbBroad304_02674	STK38	NDR family			
4200	-22.39	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
4201	-22.39	kd	CGS001-1633	DCK	-			
4202	-22.4	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
4203	-22.42	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
4204	-22.43	kd	CGS001-27148	STK36	Unc-51-like kinase (ULK) family			
4205	-22.46	cp	BRD-A64297288	amlodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, ABCG2, CA1, CACNA1B, CACNA1S, CACNA2D3, CACNB1, CACNB2, SMPD1	Calcium channel blocker
4206	-22.5	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
4207	-22.5	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4208	-22.51	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
4209	-22.56	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
4210	-22.57	kd	CGS001-8031	NCOA4	-			
4211	-22.6	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
4212	-22.6	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
4213	-22.62	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4214	-22.65	oe	ccsbBroad304_14020	SH3BP5	-			
4215	-22.67	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
4216	-22.69	cc		FXR antagonist	-			
4217	-22.7	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
4218	-22.73	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
4219	-22.73	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
4220	-22.76	kd	CGS001-10221	TRIB1	Trbl family			
4221	-22.77	kd	CGS001-3934	LCN2	Lipocalins			
4222	-22.77	kd	CGS001-81620	CDT1	-			
4223	-22.78	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
4224	-22.79	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
4225	-22.82	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
4226	-22.86	kd	CGS001-89766	UMODL1	-			
4227	-22.87	oe	ccsbBroad304_01180	PFKFB3	-			
4228	-22.94	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
4229	-22.94	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
4230	-22.95	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
4231	-23	kd	CGS001-5562	PRKAA1	AMPK subfamily			
4232	-23.04	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
4233	-23.06	kd	CGS001-7056	THBD	CD molecules			
4234	-23.09	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
4235	-23.1	kd	CGS001-7057	THBS1	-			
4236	-23.13	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
4237	-23.26	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
4238	-23.26	kd	CGS001-5037	PEBP1	-			
4239	-23.26	kd	CGS001-23210	JMJD6	-			
4240	-23.29	kd	CGS001-3553	IL1B	Interleukins and interleukin receptors			
4241	-23.29	kd	CGS001-8192	CLPP	ATPases / AAA-type			
4242	-23.36	oe	ccsbBroad304_02094	FIBP	-			
4243	-23.37	oe	ccsbBroad304_02318	KIF20A	Kinesins			
4244	-23.37	oe	ccsbBroad304_00329	CLTA	-			
4245	-23.39	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
4246	-23.4	kd	CGS001-5479	PPIB	-			
4247	-23.42	kd	CGS001-3856	KRT8	Intermediate filaments type II, keratins (basic)			
4248	-23.43	kd	CGS001-8945	BTRC	F-boxes / WD-40 domains			
4249	-23.43	kd	CGS001-338	APOB	Apolipoproteins			
4250	-23.45	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
4251	-23.46	oe	ccsbBroad304_01163	PDHA1	-			
4252	-23.48	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
4253	-23.5	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
4254	-23.51	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
4255	-23.51	kd	CGS001-5167	ENPP1	-			
4256	-23.53	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
4257	-23.54	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
4258	-23.56	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
4259	-23.58	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
4260	-23.59	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
4261	-23.61	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
4262	-23.61	kd	CGS001-1611	DAP	-			
4263	-23.62	oe	ccsbBroad304_01641	TAF13	-			
4264	-23.64	kd	CGS001-5695	PSMB7	Proteasome subunits			
4265	-23.67	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
4266	-23.68	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
4267	-23.69	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
4268	-23.7	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
4269	-23.71	cc		Mediator complex LOF	-			
4270	-23.71	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
4271	-23.72	oe	ccsbBroad304_02831	SGK3	SGK family			
4272	-23.74	oe	ccsbBroad304_06651	NOV	-			
4273	-23.75	kd	CGS001-3660	IRF2	-			
4274	-23.76	kd	CGS001-55143	CDCA8	-			
4275	-23.78	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
4276	-23.8	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
4277	-23.82	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
4278	-23.82	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
4279	-23.83	kd	CGS001-54732	TMED9	-			
4280	-23.85	oe	ccsbBroad304_01560	SNAPC1	-			
4281	-23.85	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
4282	-23.89	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
4283	-23.91	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
4284	-23.92	kd	CGS001-123803	NTAN1	-			
4285	-23.95	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
4286	-24	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
4287	-24.03	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
4288	-24.07	kd	CGS001-604	BCL6	BTB/POZ domain containing			
4289	-24.09	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
4290	-24.1	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
4291	-24.13	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
4292	-24.13	oe	ccsbBroad304_12226	NAGK	-			
4293	-24.16	oe	ccsbBroad304_06008	AP2M1	-			
4294	-24.18	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
4295	-24.2	kd	CGS001-10943	MSL3	-			
4296	-24.21	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
4297	-24.21	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
4298	-24.22	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
4299	-24.25	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
4300	-24.26	kd	CGS001-7016	TESK1	TESK subfamily			
4301	-24.28	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
4302	-24.29	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
4303	-24.3	kd	CGS001-10198	MPHOSPH9	-			
4304	-24.31	kd	CGS001-7086	TKT	-			
4305	-24.32	kd	CGS001-4193	MDM2	-			
4306	-24.36	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
4307	-24.39	kd	CGS001-18	ABAT	GABA turnover			
4308	-24.42	cc		Retinoid receptor agonist	-			
4309	-24.43	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
4310	-24.44	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
4311	-24.44	kd	CGS001-5423	POLB	DNA polymerases			
4312	-24.45	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
4313	-24.46	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
4314	-24.49	kd	CGS001-3485	IGFBP2	insulin-like growth factor (IGF) binding proteins			
4315	-24.49	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
4316	-24.49	kd	CGS001-79947	DHDDS	-			
4317	-24.5	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
4318	-24.52	oe	ccsbBroad304_09354	IGSF8	CD molecules			
4319	-24.53	kd	CGS001-2950	GSTP1	Glutathione S-transferases			
4320	-24.53	oe	ccsbBroad304_02432	IFI30	-			
4321	-24.59	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
4322	-24.6	cp	BRD-K55034111	pefloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4323	-24.61	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
4324	-24.61	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
4325	-24.62	kd	CGS001-392	ARHGAP1	Rho GTPase activating proteins			
4326	-24.64	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
4327	-24.65	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
4328	-24.65	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
4329	-24.67	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
4330	-24.67	kd	CGS001-1398	CRK	SH2 domain containing			
4331	-24.68	kd	CGS001-3880	KRT19	Intermediate filaments type I, keratins (acidic)			
4332	-24.68	kd	CGS001-8317	CDC7	CDC7 family			
4333	-24.69	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
4334	-24.7	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
4335	-24.71	kd	CGS001-6696	SPP1	Endogenous ligands			
4336	-24.71	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
4337	-24.73	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
4338	-24.73	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4339	-24.74	kd	CGS001-6184	RPN1	-			
4340	-24.76	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
4341	-24.78	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
4342	-24.81	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
4343	-24.86	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
4344	-24.86	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
4345	-24.88	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
4346	-24.89	kd	CGS001-162699	TCEB3C	-			
4347	-24.91	kd	CGS001-4179	CD46	CD molecules			
4348	-24.95	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
4349	-24.95	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4350	-24.95	oe	ccsbBroad304_07045	TEAD4	-			
4351	-24.96	kd	CGS001-7484	WNT9B	Wingless-type MMTV integration sites			
4352	-24.96	kd	CGS001-3956	LGALS1	Endogenous ligands			
4353	-25.01	kd	CGS001-10691	GMEB1	-			
4354	-25.03	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
4355	-25.04	kd	CGS001-5918	RARRES1	-			
4356	-25.05	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
4357	-25.07	kd	CGS001-558	AXL	Fibronectin type III domain containing			
4358	-25.17	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
4359	-25.18	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
4360	-25.19	kd	CGS001-10314	LANCL1	-			
4361	-25.2	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
4362	-25.21	kd	CGS001-634	CEACAM1	CD molecules			
4363	-25.22	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
4364	-25.24	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
4365	-25.26	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
4366	-25.26	cp	BRD-K57930253	nitrazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, SCN1A	Benzodiazepine receptor agonist
4367	-25.27	kd	CGS001-4869	NPM1	-			
4368	-25.28	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4369	-25.28	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
4370	-25.29	kd	CGS001-5535	PPP3R2	EF-hand domain containing			
4371	-25.3	kd	CGS001-64425	POLR1E	RNA polymerase subunits			
4372	-25.31	oe	ccsbBroad304_02438	FAM3C	-			
4373	-25.35	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
4374	-25.37	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
4375	-25.38	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
4376	-25.42	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
4377	-25.42	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
4378	-25.46	kd	CGS001-2778	GNAS	-			
4379	-25.47	oe	ccsbBroad304_01148	PCBD1	-			
4380	-25.47	kd	CGS001-965	CD58	CD molecules			
4381	-25.5	oe	ccsbBroad304_10487	BPHL	-			
4382	-25.52	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
4383	-25.53	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
4384	-25.55	oe	ccsbBroad304_00098	ARG1	Arginase			
4385	-25.59	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
4386	-25.61	kd	CGS001-642	BLMH	-			
4387	-25.62	kd	CGS001-9263	STK17A	Death-associated kinase (DAPK) family			
4388	-25.69	kd	CGS001-8226	HDHD1	-			
4389	-25.71	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
4390	-25.72	kd	CGS001-23242	COBL	-			
4391	-25.74	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
4392	-25.74	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
4393	-25.74	cp	BRD-K33106058	cytarabine	Ribonucleotide reductase inhibitor		POLB, POLA1	Ribonucleotide reductase inhibitor
4394	-25.76	kd	CGS001-486	FXYD2	Ion transport regulator			
4395	-25.77	oe	ccsbBroad304_02271	LPGAT1	-			
4396	-25.77	kd	CGS001-22938	SNW1	-			
4397	-25.77	kd	CGS001-6195	RPS6KA1	RSK subfamily			
4398	-25.77	kd	CGS001-2967	GTF2H3	General transcription factors			
4399	-25.78	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
4400	-25.78	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
4401	-25.79	kd	CGS001-861	RUNX1	-			
4402	-25.82	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
4403	-25.83	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
4404	-25.85	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4405	-25.87	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
4406	-25.88	oe	ccsbBroad304_02843	FTSJ1	-			
4407	-25.88	kd	CGS001-3845	KRAS	RAS subfamily			
4408	-25.88	kd	CGS001-597	BCL2A1	-			
4409	-25.93	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
4410	-25.93	oe	ccsbBroad304_00690	GRN	-			
4411	-25.94	oe	ccsbBroad304_04655	TRIM9	-			
4412	-25.94	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4413	-25.96	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
4414	-26.02	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
4415	-26.03	kd	CGS001-22887	FOXJ3	Forkhead boxes			
4416	-26.06	oe	ccsbBroad304_03122	RHOD	-			
4417	-26.06	kd	CGS001-7013	TERF1	-			
4418	-26.09	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
4419	-26.09	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
4420	-26.11	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
4421	-26.11	kd	CGS001-57149	LYRM1	LYR motif containing			
4422	-26.12	oe	ccsbBroad304_03878	SENP2	-			
4423	-26.13	oe	ccsbBroad304_00880	IRF2	-			
4424	-26.14	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4425	-26.14	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
4426	-26.16	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4427	-26.27	kd	CGS001-9568	GABBR2	GABA receptors			
4428	-26.28	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
4429	-26.28	kd	CGS001-150280	HORMAD2	-			
4430	-26.28	kd	CGS001-650	BMP2	Bone morphogenetic proteins			
4431	-26.32	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
4432	-26.35	cp	BRD-A24381660	zeranol	Estrogen receptor agonist			Estrogen receptor agonist
4433	-26.35	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
4434	-26.36	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
4435	-26.38	kd	CGS001-2952	GSTT1	Glutathione S-transferases / Soluble			
4436	-26.43	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
4437	-26.47	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
4438	-26.49	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
4439	-26.5	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
4440	-26.51	kd	CGS001-4683	NBN	-			
4441	-26.56	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
4442	-26.57	kd	CGS001-8295	TRRAP	TRRAP subfamily			
4443	-26.57	kd	CGS001-3551	IKBKB	IKK family			
4444	-26.61	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4445	-26.64	kd	CGS001-7846	TUBA1A	Tubulins			
4446	-26.67	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
4447	-26.69	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
4448	-26.71	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
4449	-26.72	kd	CGS001-1163	CKS1B	-			
4450	-26.74	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
4451	-26.75	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
4452	-26.82	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
4453	-26.84	kd	CGS001-109	ADCY3	Adenylyl cyclases			
4454	-26.86	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
4455	-26.86	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
4456	-26.86	kd	CGS001-688	KLF5	Kruppel-like transcription factors			
4457	-26.86	kd	CGS001-2592	GALT	-			
4458	-26.88	kd	CGS001-3705	ITPK1	-			
4459	-26.98	kd	CGS001-440387	CTRB2	-			
4460	-26.99	kd	CGS001-10001	MED6	-			
4461	-27	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
4462	-27	kd	CGS001-8408	ULK1	Unc-51-like kinase (ULK) family			
4463	-27.01	kd	CGS001-4329	ALDH6A1	Aldehyde dehydrogenases			
4464	-27.02	kd	CGS001-6275	S100A4	EF-hand domain containing			
4465	-27.03	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
4466	-27.07	oe	ccsbBroad304_07024	SYK	Syk family			
4467	-27.08	kd	CGS001-5357	PLS1	EF-hand domain containing			
4468	-27.11	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4469	-27.11	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
4470	-27.12	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
4471	-27.13	cp	BRD-K47278471	diphenhydramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4472	-27.16	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
4473	-27.16	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
4474	-27.16	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
4475	-27.18	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
4476	-27.19	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
4477	-27.2	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
4478	-27.2	kd	CGS001-4047	LSS	Lanosterol biosynthesis pathway			
4479	-27.21	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
4480	-27.21	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
4481	-27.21	kd	CGS001-22894	DIS3	-			
4482	-27.24	oe	ccsbBroad304_07326	EIF2B2	-			
4483	-27.24	kd	CGS001-5447	POR	-			
4484	-27.28	oe	ccsbBroad304_02509	GMEB1	-			
4485	-27.3	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4486	-27.32	kd	CGS001-5931	RBBP7	WD repeat domain containing			
4487	-27.32	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
4488	-27.34	kd	CGS001-51451	LCMT1	-			
4489	-27.38	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
4490	-27.41	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
4491	-27.42	oe	ccsbBroad304_03950	ATG3	-			
4492	-27.44	cp	BRD-K17705806	JTC-801	Opioid receptor antagonist		OPRL1	Opioid receptor antagonist
4493	-27.44	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4494	-27.47	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
4495	-27.47	kd	CGS001-3309	HSPA5	Heat shock proteins / HSP70			
4496	-27.48	kd	CGS001-7157	TP53	-			
4497	-27.49	kd	CGS001-163486	DENND1B	DENN/MADD domain containing			
4498	-27.49	oe	ccsbBroad304_07275	PSMG1	-			
4499	-27.5	cp	BRD-A39390670	rabeprazole	ATPase inhibitor		ATP4A, CYP2C19	ATPase inhibitor, Gastrin inhibitor
4500	-27.51	kd	CGS001-8807	IL18RAP	CD molecules			
4501	-27.54	kd	CGS001-3421	IDH3G	-			
4502	-27.54	kd	CGS001-56647	BCCIP	-			
4503	-27.6	kd	CGS001-10434	LYPLA1	-			
4504	-27.61	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
4505	-27.63	kd	CGS001-2853	GPR31	GPCR / Class A : Orphans			
4506	-27.63	kd	CGS001-8659	ALDH4A1	Aldehyde dehydrogenases			
4507	-27.65	kd	CGS001-54556	ING3	Zinc fingers, PHD-type			
4508	-27.67	kd	CGS001-9770	RASSF2	-			
4509	-27.67	kd	CGS001-113451	ADC	-			
4510	-27.68	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4511	-27.69	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
4512	-27.72	cc		Thromboxane receptor antagonist	-			
4513	-27.74	cp	BRD-A92630576	trimebutine	Opioid receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Opioid receptor agonist
4514	-27.75	oe	ccsbBroad304_04544	RCCD1	-			
4515	-27.75	kd	CGS001-7534	YWHAZ	-			
4516	-27.75	kd	CGS001-10914	PAPOLA	-			
4517	-27.76	cc		Cannabinoid receptor agonist	-			
4518	-27.82	kd	CGS001-5686	PSMA5	Proteasome subunits			
4519	-27.85	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
4520	-27.87	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
4521	-27.93	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
4522	-27.97	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
4523	-27.98	kd	CGS001-163688	CALML6	EF-hand domain containing			
4524	-28	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4525	-28.02	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
4526	-28.04	kd	CGS001-56916	SMARCAD1	-			
4527	-28.07	kd	CGS001-3945	LDHB	-			
4528	-28.07	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
4529	-28.08	cp	BRD-K44779798	miglitol	Glucosidase inhibitor		GAA, MGAM, GANAB, GANC, SLC5A4	Glucosidase inhibitor
4530	-28.11	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
4531	-28.12	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
4532	-28.13	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
4533	-28.14	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
4534	-28.14	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
4535	-28.15	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
4536	-28.17	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
4537	-28.2	kd	CGS001-7525	YES1	Src family			
4538	-28.2	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
4539	-28.2	kd	CGS001-2852	GPER	-			
4540	-28.23	cc		PDGFR/KIT inhibitor	-			
4541	-28.23	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
4542	-28.26	kd	CGS001-8841	HDAC3	Histone deacetylases			
4543	-28.29	kd	CGS001-27244	SESN1	-			
4544	-28.3	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
4545	-28.3	oe	ccsbBroad304_06648	CNOT3	-			
4546	-28.33	kd	CGS001-841	CASP8	Caspases			
4547	-28.34	oe	ccsbBroad304_03269	CD320	CD molecules			
4548	-28.34	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
4549	-28.35	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
4550	-28.35	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
4551	-28.36	oe	ccsbBroad304_01054	GADD45B	-			
4552	-28.38	kd	CGS001-7597	ZBTB25	BTB/POZ domain containing			
4553	-28.4	kd	CGS001-5708	PSMD2	Proteasome subunits			
4554	-28.43	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
4555	-28.44	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
4556	-28.44	kd	CGS001-2958	GTF2A2	General transcription factors			
4557	-28.48	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
4558	-28.49	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
4559	-28.52	kd	CGS001-3579	CXCR2	Chemokine receptors			
4560	-28.55	kd	CGS001-1453	CSNK1D	Casein kinase 1 (CK1) family			
4561	-28.59	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
4562	-28.63	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
4563	-28.63	kd	CGS001-23161	SNX13	Sorting nexins			
4564	-28.64	cc		Mitochondrial complex IV LOF	-			
4565	-28.65	kd	CGS001-53347	UBASH3A	-			
4566	-28.65	kd	CGS001-944	TNFSF8	CD molecules			
4567	-28.66	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
4568	-28.69	cc		Heat shock 70kDa proteins LOF	-			
4569	-28.69	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
4570	-28.69	kd	CGS001-144811	LACC1	-			
4571	-28.71	kd	CGS001-139760	GPR119	GPCR / Class A : Orphans			
4572	-28.72	kd	CGS001-7421	VDR	Vitamin D receptors			
4573	-28.72	kd	CGS001-50810	HDGFRP3	-			
4574	-28.73	kd	CGS001-4482	MSRA	-			
4575	-28.79	oe	ccsbBroad304_03479	YTHDF1	-			
4576	-28.82	kd	CGS001-54659	UGT1A3	UDP glucuronosyltransferases			
4577	-28.83	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
4578	-28.86	oe	ccsbBroad304_07219	CDC7	CDC7 family			
4579	-28.86	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
4580	-28.86	kd	CGS001-55818	KDM3A	Histone demethylases			
4581	-28.88	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
4582	-28.9	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
4583	-28.93	kd	CGS001-5888	RAD51	-			
4584	-28.94	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
4585	-28.96	oe	ccsbBroad304_03037	TMEM97	-			
4586	-28.97	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
4587	-28.98	kd	CGS001-200879	LIPH	-			
4588	-28.99	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
4589	-29	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
4590	-29.03	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
4591	-29.05	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
4592	-29.07	kd	CGS001-6812	STXBP1	-			
4593	-29.07	kd	CGS001-6347	CCL2	Chemokine ligands			
4594	-29.09	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
4595	-29.09	oe	ccsbBroad304_07920	NUP62	-			
4596	-29.09	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
4597	-29.09	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
4598	-29.1	kd	CGS001-91392	ZNF502	Zinc fingers, C2H2-type			
4599	-29.11	cc		S100 calcium binding proteins LOF	-			
4600	-29.11	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
4601	-29.12	oe	ccsbBroad304_08645	BCCIP	-			
4602	-29.12	oe	ccsbBroad304_00501	EMD	-			
4603	-29.13	oe	ccsbBroad304_08116	TBK1	IKK family			
4604	-29.15	oe	ccsbBroad304_07569	TRIB1	Trbl family			
4605	-29.16	kd	CGS001-4946	OAZ1	-			
4606	-29.19	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
4607	-29.19	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
4608	-29.2	cc		EMSY complex LOF	-			
4609	-29.21	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
4610	-29.21	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
4611	-29.21	kd	CGS001-7077	TIMP2	-			
4612	-29.21	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
4613	-29.22	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
4614	-29.23	kd	CGS001-10113	PREB	WD repeat domain containing			
4615	-29.26	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
4616	-29.27	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
4617	-29.28	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
4618	-29.29	kd	CGS001-8805	TRIM24	TIF1 family			
4619	-29.29	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
4620	-29.31	oe	ccsbBroad304_10846	GGT1	CD molecules			
4621	-29.33	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
4622	-29.33	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
4623	-29.34	oe	ccsbBroad304_03310	LCMT1	-			
4624	-29.35	kd	CGS001-55722	CEP72	-			
4625	-29.36	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
4626	-29.36	oe	ccsbBroad304_00572	FKBP3	-			
4627	-29.4	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
4628	-29.44	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
4629	-29.44	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4630	-29.47	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
4631	-29.48	oe	ccsbBroad304_00819	IDH3B	-			
4632	-29.49	kd	CGS001-7024	TFCP2	-			
4633	-29.5	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
4634	-29.52	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
4635	-29.52	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
4636	-29.54	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
4637	-29.54	kd	CGS001-9319	TRIP13	ATPases / AAA-type			
4638	-29.55	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
4639	-29.55	kd	CGS001-10284	SAP18	-			
4640	-29.56	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
4641	-29.56	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
4642	-29.57	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
4643	-29.57	oe	ccsbBroad304_04786	CANT1	-			
4644	-29.57	kd	CGS001-4171	MCM2	-			
4645	-29.59	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
4646	-29.6	oe	ccsbBroad304_01948	GAS7	-			
4647	-29.6	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
4648	-29.61	oe	ccsbBroad304_01841	BAG6	-			
4649	-29.61	oe	ccsbBroad304_03641	ASF1B	-			
4650	-29.61	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
4651	-29.61	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
4652	-29.62	kd	CGS001-23581	CASP14	Caspases			
4653	-29.69	cc		EIF Proteins LOF	-			
4654	-29.72	kd	CGS001-23355	VPS8	-			
4655	-29.72	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
4656	-29.73	kd	CGS001-9140	ATG12	-			
4657	-29.75	kd	CGS001-79885	HDAC11	Histone deacetylases			
4658	-29.78	oe	ccsbBroad304_08346	COQ3	-			
4659	-29.78	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
4660	-29.8	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
4661	-29.82	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
4662	-29.89	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
4663	-29.92	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
4664	-29.93	kd	CGS001-51547	SIRT7	Histone deacetylases (HDACs)			
4665	-29.98	oe	ccsbBroad304_08709	SCYL3	-			
4666	-29.98	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
4667	-29.99	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4668	-29.99	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
4669	-30	kd	CGS001-9967	THRAP3	-			
4670	-30.02	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
4671	-30.03	oe	ccsbBroad304_03696	C19ORF10	-			
4672	-30.04	kd	CGS001-5511	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4673	-30.14	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
4674	-30.15	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
4675	-30.15	kd	CGS001-9815	GIT2	Ankyrin repeat domain containing			
4676	-30.15	kd	CGS001-2073	ERCC5	-			
4677	-30.16	kd	CGS001-23464	GCAT	-			
4678	-30.17	cp	BRD-K50866992	tropisetron	Serotonin receptor antagonist		HTR3A, GLRA1, GLRA2, GLRB, HTR4	Serotonin receptor antagonist
4679	-30.18	kd	CGS001-22944	KIN	-			
4680	-30.18	kd	CGS001-26128	KIAA1279	-			
4681	-30.2	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
4682	-30.23	kd	CGS001-22930	RAB3GAP1	-			
4683	-30.24	oe	ccsbBroad304_00949	LRPAP1	-			
4684	-30.25	kd	CGS001-1999	ELF3	ETS Transcription Factors			
4685	-30.27	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
4686	-30.27	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
4687	-30.3	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
4688	-30.3	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
4689	-30.33	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
4690	-30.36	oe	ccsbBroad304_03497	TXNL4B	-			
4691	-30.36	oe	ccsbBroad304_14242	MCCC2	-			
4692	-30.36	kd	CGS001-1595	CYP51A1	Cytochrome P450s			
4693	-30.39	oe	ccsbBroad304_00931	LCN2	Lipocalins			
4694	-30.41	oe	ccsbBroad304_02419	NDRG1	-			
4695	-30.41	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
4696	-30.41	kd	CGS001-5338	PLD2	Hydrolases			
4697	-30.44	kd	CGS001-11284	PNKP	-			
4698	-30.47	oe	ccsbBroad304_01624	SUPV3L1	-			
4699	-30.47	oe	ccsbBroad304_02840	PISD	Decarboxylases			
4700	-30.5	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
4701	-30.53	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
4702	-30.59	oe	ccsbBroad304_03618	OSGEP	-			
4703	-30.61	oe	ccsbBroad304_06862	RGS3	-			
4704	-30.68	oe	ccsbBroad304_01394	RFX4	-			
4705	-30.68	oe	ccsbBroad304_03933	CARD9	-			
4706	-30.7	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
4707	-30.71	cp	BRD-K53220666	trimetozine	Sedative			Sedative
4708	-30.71	kd	CGS001-8896	BUD31	-			
4709	-30.72	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
4710	-30.73	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
4711	-30.76	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
4712	-30.76	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4713	-30.76	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
4714	-30.76	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
4715	-30.77	cp	BRD-A35519318	benidipine	Calcium channel blocker		CACNA1C, CACNA1G, CYP3A5	Calcium channel blocker
4716	-30.77	kd	CGS001-515	ATP5F1	ATPases / F-type			
4717	-30.77	kd	CGS001-7915	ALDH5A1	Aldehyde dehydrogenases			
4718	-30.78	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
4719	-30.8	kd	CGS001-2793	GNGT2	-			
4720	-30.8	kd	CGS001-999	CDH1	CD molecules			
4721	-30.81	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
4722	-30.82	cc		Tumor necrosis factor superfamily LOF	-			
4723	-30.83	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
4724	-30.84	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
4725	-30.84	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
4726	-30.86	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
4727	-30.88	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4728	-30.91	kd	CGS001-26520	TIMM9	-			
4729	-30.91	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
4730	-30.91	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
4731	-30.94	kd	CGS001-345	APOC3	Apolipoproteins			
4732	-30.96	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
4733	-31.01	oe	ccsbBroad304_03182	GLOD4	-			
4734	-31.02	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
4735	-31.07	kd	CGS001-1504	CTRB1	-			
4736	-31.08	kd	CGS001-7428	VHL	-			
4737	-31.09	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
4738	-31.1	kd	CGS001-1649	DDIT3	-			
4739	-31.1	kd	CGS001-839	CASP6	Caspases			
4740	-31.11	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
4741	-31.11	cp	BRD-K69650333	idarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4742	-31.12	kd	CGS001-1514	CTSL1	-			
4743	-31.18	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
4744	-31.19	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
4745	-31.19	oe	ccsbBroad304_05902	BNIP3	-			
4746	-31.2	oe	ccsbBroad304_02578	EBNA1BP2	-			
4747	-31.2	kd	CGS001-2056	EPO	Endogenous ligands			
4748	-31.23	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
4749	-31.25	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
4750	-31.26	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
4751	-31.31	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
4752	-31.33	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
4753	-31.33	kd	CGS001-6788	STK3	MST subfamily			
4754	-31.36	oe	ccsbBroad304_00446	DKC1	-			
4755	-31.43	oe	ccsbBroad304_02012	FADD	-			
4756	-31.43	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
4757	-31.44	kd	CGS001-1659	DHX8	DEAH-boxes			
4758	-31.45	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
4759	-31.48	cp	BRD-K56614220	clofazimine	GK0582 inhibitor			GK0582 inhibitor
4760	-31.5	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
4761	-31.52	oe	ccsbBroad304_08993	DHDDS	-			
4762	-31.54	oe	ccsbBroad304_00036	AFP	-			
4763	-31.56	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
4764	-31.57	oe	ccsbBroad304_06975	SMARCC2	-			
4765	-31.57	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
4766	-31.58	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
4767	-31.58	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
4768	-31.59	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
4769	-31.63	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
4770	-31.65	kd	CGS001-3098	HK1	-			
4771	-31.68	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
4772	-31.69	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
4773	-31.69	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
4774	-31.7	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
4775	-31.71	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
4776	-31.72	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
4777	-31.78	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
4778	-31.8	kd	CGS001-9158	FIBP	-			
4779	-31.81	oe	ccsbBroad304_06144	EFNB3	Ephrins			
4780	-31.81	kd	CGS001-7360	UGP2	-			
4781	-31.85	oe	ccsbBroad304_02485	STAMBP	-			
4782	-31.86	kd	CGS001-91433	RCCD1	-			
4783	-31.88	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
4784	-31.88	kd	CGS001-3590	IL11RA	IL-6 receptor family			
4785	-31.91	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
4786	-31.92	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
4787	-31.92	kd	CGS001-4297	MLL	-			
4788	-31.94	kd	CGS001-8853	ASAP2	Ankyrin repeat domain containing			
4789	-31.95	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
4790	-31.96	oe	ccsbBroad304_06670	OGG1	-			
4791	-31.98	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
4792	-32.01	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
4793	-32.01	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
4794	-32.02	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
4795	-32.06	oe	ccsbBroad304_00282	CDKN1A	-			
4796	-32.12	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4797	-32.13	oe	ccsbBroad304_08596	EAPP	-			
4798	-32.13	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
4799	-32.16	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
4800	-32.17	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
4801	-32.17	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
4802	-32.18	kd	CGS001-4351	MPI	-			
4803	-32.22	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
4804	-32.23	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
4805	-32.24	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
4806	-32.26	kd	CGS001-4097	MAFG	-			
4807	-32.3	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
4808	-32.31	kd	CGS001-2677	GGCX	Carboxylases			
4809	-32.33	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
4810	-32.34	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
4811	-32.36	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4812	-32.36	kd	CGS001-1386	ATF2	basic leucine zipper proteins			
4813	-32.39	oe	ccsbBroad304_06188	F10	Chymotrypsin			
4814	-32.4	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
4815	-32.41	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
4816	-32.44	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
4817	-32.44	oe	ccsbBroad304_03980	DCLRE1B	-			
4818	-32.44	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
4819	-32.45	cp	BRD-K00673382	famotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
4820	-32.47	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
4821	-32.48	oe	ccsbBroad304_06665	OAT	-			
4822	-32.49	cp	BRD-K10065684	dantron	Laxative			Laxative
4823	-32.5	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
4824	-32.51	kd	CGS001-10939	AFG3L2	ATPases / AAA-type			
4825	-32.53	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
4826	-32.55	kd	CGS001-7840	ALMS1	-			
4827	-32.59	oe	ccsbBroad304_07515	GFPT2	-			
4828	-32.6	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
4829	-32.63	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4830	-32.64	oe	ccsbBroad304_06836	RAD23B	-			
4831	-32.65	oe	ccsbBroad304_06952	SKP1	-			
4832	-32.65	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
4833	-32.66	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
4834	-32.66	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
4835	-32.66	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
4836	-32.67	cp	BRD-K89708791	rifaximin	RNA synthesis inhibitor		NR1I2, CYP3A4	RNA synthesis inhibitor
4837	-32.68	kd	CGS001-9637	FEZ2	-			
4838	-32.68	kd	CGS001-1452	CSNK1A1	Casein kinase 1 (CK1) family			
4839	-32.7	kd	CGS001-55165	CEP55	-			
4840	-32.79	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
4841	-32.79	kd	CGS001-23047	PDS5B	-			
4842	-32.82	kd	CGS001-4191	MDH2	-			
4843	-32.85	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
4844	-32.85	oe	ccsbBroad304_04053	DERL1	-			
4845	-32.86	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
4846	-32.9	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
4847	-32.91	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
4848	-32.91	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
4849	-32.95	oe	ccsbBroad304_07053	TFPI	-			
4850	-32.95	kd	CGS001-27297	CRCP	-			
4851	-32.96	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
4852	-32.98	oe	ccsbBroad304_02086	PDLIM1	-			
4853	-33.04	oe	ccsbBroad304_05194	LIPH	-			
4854	-33.07	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4855	-33.19	cc		Interleukin receptors LOF	-			
4856	-33.21	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
4857	-33.22	kd	CGS001-2277	FIGF	-			
4858	-33.25	oe	ccsbBroad304_05931	CAPG	-			
4859	-33.27	oe	ccsbBroad304_03237	LEF1	-			
4860	-33.27	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
4861	-33.28	oe	ccsbBroad304_07557	NAMPT	-			
4862	-33.3	kd	CGS001-4605	MYBL2	-			
4863	-33.32	oe	ccsbBroad304_06870	RNH1	-			
4864	-33.32	cp	BRD-K82147103	lofepramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
4865	-33.32	kd	CGS001-1528	CYB5A	Cytochrome b genes			
4866	-33.33	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
4867	-33.35	kd	CGS001-7693	ZNF134	Zinc fingers, C2H2-type			
4868	-33.36	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
4869	-33.36	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
4870	-33.38	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
4871	-33.38	kd	CGS001-54512	EXOSC4	-			
4872	-33.4	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
4873	-33.42	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
4874	-33.45	kd	CGS001-5162	PDHB	-			
4875	-33.48	kd	CGS001-6050	RNH1	-			
4876	-33.49	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
4877	-33.49	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
4878	-33.5	kd	CGS001-10672	GNA13	-			
4879	-33.51	oe	ccsbBroad304_06324	GPX7	-			
4880	-33.51	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
4881	-33.54	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
4882	-33.55	kd	CGS001-4671	NAIP	Inhibitors of apoptosis (IAP) protein family			
4883	-33.58	oe	ccsbBroad304_01347	RAD1	-			
4884	-33.58	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
4885	-33.59	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
4886	-33.6	kd	CGS001-10971	YWHAQ	-			
4887	-33.63	kd	CGS001-169792	GLIS3	Zinc fingers, C2H2-type			
4888	-33.64	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
4889	-33.66	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
4890	-33.67	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
4891	-33.68	cc		Akt Signaling LOF	-			
4892	-33.7	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
4893	-33.71	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
4894	-33.72	kd	CGS001-204	AK2	Adenylate kinases			
4895	-33.76	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
4896	-33.76	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
4897	-33.81	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
4898	-33.85	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
4899	-33.86	oe	ccsbBroad304_07761	CORO1A	Coronins			
4900	-33.87	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
4901	-33.87	kd	CGS001-1975	EIF4B	RNA binding motif (RRM) containing			
4902	-33.88	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
4903	-33.88	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
4904	-33.89	kd	CGS001-84669	USP32	EF-hand domain containing			
4905	-33.9	oe	ccsbBroad304_02837	BHMT2	-			
4906	-33.92	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
4907	-33.94	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4908	-33.96	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
4909	-33.96	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
4910	-33.98	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
4911	-34.01	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
4912	-34.01	oe	ccsbBroad304_01673	TIMP3	-			
4913	-34.01	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
4914	-34.04	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
4915	-34.06	oe	ccsbBroad304_02230	HERPUD1	-			
4916	-34.09	oe	ccsbBroad304_02869	ASF1A	-			
4917	-34.09	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
4918	-34.09	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
4919	-34.16	kd	CGS001-7103	TSPAN8	Tetraspanins			
4920	-34.17	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
4921	-34.2	cp	BRD-K00532621	midazolam	Benzodiazepine receptor agonist		CYP3A5, CYP3A7, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3	Benzodiazepine receptor agonist
4922	-34.21	oe	ccsbBroad304_02373	SPRY2	-			
4923	-34.21	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
4924	-34.21	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
4925	-34.22	oe	ccsbBroad304_03917	RBKS	-			
4926	-34.22	oe	ccsbBroad304_00986	MCM2	-			
4927	-34.22	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4928	-34.23	kd	CGS001-1841	DTYMK	-			
4929	-34.25	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
4930	-34.3	kd	CGS001-57787	MARK4	MARK subfamily			
4931	-34.31	kd	CGS001-2969	GTF2I	General transcription factors			
4932	-34.34	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
4933	-34.35	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
4934	-34.35	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
4935	-34.36	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
4936	-34.36	kd	CGS001-29763	PACSIN3	-			
4937	-34.37	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
4938	-34.41	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
4939	-34.43	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
4940	-34.43	kd	CGS001-3383	ICAM1	CD molecules			
4941	-34.47	kd	CGS001-5898	RALA	-			
4942	-34.48	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
4943	-34.5	oe	ccsbBroad304_00818	IDH3A	-			
4944	-34.5	kd	CGS001-1022	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
4945	-34.52	oe	ccsbBroad304_00665	GOT1	-			
4946	-34.54	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4947	-34.54	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
4948	-34.55	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
4949	-34.56	kd	CGS001-670	BPHL	-			
4950	-34.58	kd	CGS001-5198	PFAS	-			
4951	-34.58	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
4952	-34.62	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
4953	-34.62	kd	CGS001-147179	WIPF2	-			
4954	-34.63	cc		Vitamin D receptor agonist	-			
4955	-34.64	kd	CGS001-2744	GLS	Ankyrin repeat domain containing			
4956	-34.67	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
4957	-34.68	oe	ccsbBroad304_02205	WTAP	-			
4958	-34.68	kd	CGS001-2639	GCDH	-			
4959	-34.7	cp	BRD-K94887716	TFMPP	Serotonin receptor agonist			Serotonin receptor agonist, Serotonin receptor antagonist
4960	-34.77	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
4961	-34.78	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
4962	-34.79	oe	ccsbBroad304_01146	PARN	-			
4963	-34.79	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
4964	-34.82	kd	CGS001-5649	RELN	-			
4965	-34.82	kd	CGS001-6790	AURKA	Aurora kinase			
4966	-34.84	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
4967	-34.89	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
4968	-34.89	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
4969	-34.89	kd	CGS001-200734	SPRED2	-			
4970	-34.93	oe	ccsbBroad304_03129	ERO1L	-			
4971	-34.93	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
4972	-34.98	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
4973	-34.99	kd	CGS001-3074	HEXB	-			
4974	-35	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4975	-35	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
4976	-35.01	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
4977	-35.06	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
4978	-35.09	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4979	-35.09	kd	CGS001-9326	ZNHIT3	Zinc fingers, HIT-type			
4980	-35.09	kd	CGS001-7020	TFAP2A	-			
4981	-35.1	oe	ccsbBroad304_07651	HEXIM1	-			
4982	-35.13	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
4983	-35.14	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4984	-35.14	kd	CGS001-10099	TSPAN3	Tetraspanins			
4985	-35.15	kd	CGS001-5707	PSMD1	Proteasome subunits			
4986	-35.17	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
4987	-35.18	kd	CGS001-115	ADCY9	Adenylyl cyclases			
4988	-35.2	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
4989	-35.25	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
4990	-35.25	kd	CGS001-5831	PYCR1	-			
4991	-35.27	kd	CGS001-1981	EIF4G1	Parkinson disease			
4992	-35.28	oe	ccsbBroad304_00239	CCNG1	-			
4993	-35.29	oe	ccsbBroad304_02553	BLCAP	-			
4994	-35.31	kd	CGS001-79143	MBOAT7	-			
4995	-35.32	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
4996	-35.32	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
4997	-35.33	cc		HRH1 antagonist	-			
4998	-35.36	oe	ccsbBroad304_02862	CCRN4L	-			
4999	-35.36	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
5000	-35.37	kd	CGS001-4616	GADD45B	-			
5001	-35.43	kd	CGS001-178	AGL	-			
5002	-35.45	oe	ccsbBroad304_09954	PTRF	-			
5003	-35.46	kd	CGS001-537	ATP6AP1	-			
5004	-35.49	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
5005	-35.5	kd	CGS001-501	ALDH7A1	Aldehyde dehydrogenases			
5006	-35.53	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
5007	-35.56	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
5008	-35.58	kd	CGS001-10397	NDRG1	-			
5009	-35.59	kd	CGS001-607	BCL9	-			
5010	-35.64	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
5011	-35.64	kd	CGS001-7167	TPI1	-			
5012	-35.67	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
5013	-35.67	kd	CGS001-11124	FAF1	UBX domain containing			
5014	-35.69	cp	BRD-K27184429	levocetirizine	Histamine receptor antagonist		HRH1, CXCL8	Histamine receptor antagonist
5015	-35.71	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
5016	-35.71	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
5017	-35.76	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
5018	-35.81	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
5019	-35.82	kd	CGS001-10390	CEPT1	-			
5020	-35.83	kd	CGS001-84547	PGBD1	-			
5021	-35.83	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5022	-35.84	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
5023	-35.86	oe	ccsbBroad304_03506	AURKAIP1	-			
5024	-35.91	cc		Nucleophosmin inhibitor	-			
5025	-35.96	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
5026	-36.01	oe	ccsbBroad304_08325	LIPT1	-			
5027	-36.04	oe	ccsbBroad304_08480	PNPO	-			
5028	-36.05	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
5029	-36.05	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5030	-36.06	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5031	-36.13	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
5032	-36.14	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
5033	-36.14	kd	CGS001-2100	ESR2	Estrogen receptors			
5034	-36.16	kd	CGS001-1515	CTSL2	-			
5035	-36.2	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
5036	-36.24	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
5037	-36.33	kd	CGS001-10227	MFSD10	-			
5038	-36.34	oe	ccsbBroad304_00966	MAFG	-			
5039	-36.35	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
5040	-36.35	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
5041	-36.36	kd	CGS001-6233	RPS27A	S ribosomal proteins			
5042	-36.37	oe	ccsbBroad304_06765	PRCC	-			
5043	-36.41	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
5044	-36.42	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
5045	-36.43	cp	BRD-K28849549	mesalazine	Cyclooxygenase inhibitor		PTGS1, PPARG, PTGS2, ALOX5, CHUK, CTNNB1, IKBKB, MPO, NAT1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor, Prostanoid receptor antagonist
5046	-36.44	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
5047	-36.45	oe	ccsbBroad304_02668	PNKP	-			
5048	-36.45	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
5049	-36.47	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
5050	-36.49	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
5051	-36.5	kd	CGS001-2280	FKBP1A	Cis-trans-isomerases			
5052	-36.51	kd	CGS001-1977	EIF4E	Translation Initiation Factor 4E			
5053	-36.52	cp	BRD-K85030058	benactyzine	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
5054	-36.53	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
5055	-36.56	oe	ccsbBroad304_07267	PDLIM4	-			
5056	-36.56	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
5057	-36.57	kd	CGS001-93487	MAPK1IP1L	-			
5058	-36.61	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
5059	-36.62	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
5060	-36.63	kd	CGS001-6461	SHB	SH2 domain containing			
5061	-36.7	kd	CGS001-4267	CD99	CD molecules			
5062	-36.72	kd	CGS001-4638	MYLK	Myosin Light Chain Kinase (MLCK) family			
5063	-36.73	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
5064	-36.75	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5065	-36.75	kd	CGS001-6259	RYK	Type XV RTKs: RYK			
5066	-36.76	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
5067	-36.8	cp	BRD-A94543220	bifonazole	Sterol demethylase inhibitor		CYP2B6	Sterol demethylase inhibitor
5068	-36.81	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
5069	-36.85	oe	ccsbBroad304_01379	RBBP6	-			
5070	-36.85	kd	CGS001-23461	ABCA5	ATP binding cassette transporters / subfamily A			
5071	-36.9	cp	BRD-K29530284	amlexanox	Histamine receptor modulator		FGF1, IL3, S100A12, S100A13	Histamine receptor modulator
5072	-36.91	oe	ccsbBroad304_04038	ELOVL6	-			
5073	-36.96	oe	ccsbBroad304_02572	SERINC3	-			
5074	-36.97	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
5075	-36.97	kd	CGS001-29916	SNX11	Sorting nexins			
5076	-37.03	oe	ccsbBroad304_01787	YES1	Src family			
5077	-37.06	kd	CGS001-56675	NRIP3	-			
5078	-37.07	oe	ccsbBroad304_02229	TRAM2	-			
5079	-37.09	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5080	-37.09	kd	CGS001-10381	TUBB3	Tubulins			
5081	-37.1	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
5082	-37.15	oe	ccsbBroad304_01584	SPARC	-			
5083	-37.16	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
5084	-37.17	kd	CGS001-3691	ITGB4	Integrins			
5085	-37.18	oe	ccsbBroad304_03235	TUBD1	Tubulins			
5086	-37.23	oe	ccsbBroad304_01084	NEU1	-			
5087	-37.24	kd	CGS001-978	CDA	-			
5088	-37.29	kd	CGS001-26574	AATF	-			
5089	-37.3	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
5090	-37.31	oe	ccsbBroad304_03808	ERGIC1	-			
5091	-37.31	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
5092	-37.35	oe	ccsbBroad304_03565	ADI1	-			
5093	-37.35	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
5094	-37.36	cp	BRD-K63343048	orlistat	Lipase inhibitor		PNLIP, DAGLA, FASN, LIPF, CNR1, DAGLB	Lipase inhibitor
5095	-37.36	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
5096	-37.37	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
5097	-37.37	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
5098	-37.39	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
5099	-37.43	kd	CGS001-6675	UAP1	-			
5100	-37.44	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
5101	-37.47	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
5102	-37.49	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
5103	-37.51	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
5104	-37.52	cc		Progesterone receptor agonist	-			
5105	-37.52	kd	CGS001-949	SCARB1	-			
5106	-37.52	kd	CGS001-4074	M6PR	-			
5107	-37.54	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
5108	-37.59	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
5109	-37.59	kd	CGS001-25913	POT1	-			
5110	-37.65	kd	CGS001-8572	PDLIM4	-			
5111	-37.66	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
5112	-37.68	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
5113	-37.68	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
5114	-37.69	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
5115	-37.72	cc		SRY LOF	-			
5116	-37.76	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
5117	-37.77	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
5118	-37.78	kd	CGS001-9212	AURKB	Aurora kinase			
5119	-37.83	kd	CGS001-1632	ECI1	-			
5120	-37.87	kd	CGS001-3925	STMN1	-			
5121	-37.92	kd	CGS001-26993	AKAP8L	-			
5122	-37.95	kd	CGS001-6714	SRC	Src family			
5123	-37.97	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
5124	-37.99	kd	CGS001-27102	EIF2AK1	Other PEK family kinases			
5125	-38.03	kd	CGS001-7249	TSC2	-			
5126	-38.1	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
5127	-38.11	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
5128	-38.13	oe	ccsbBroad304_00001	NAT1	-			
5129	-38.14	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
5130	-38.14	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
5131	-38.21	kd	CGS001-883	CCBL1	Hydrogen sulphide synthesis			
5132	-38.26	cc		IL4 Pathway LOF	-			
5133	-38.29	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
5134	-38.31	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
5135	-38.32	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
5136	-38.36	kd	CGS001-55699	IARS2	Aminoacyl tRNA synthetases / Class I			
5137	-38.39	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
5138	-38.4	kd	CGS001-3593	IL12B	Interleukins and interleukin receptors			
5139	-38.41	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
5140	-38.43	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
5141	-38.45	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
5142	-38.47	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
5143	-38.49	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
5144	-38.55	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
5145	-38.59	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
5146	-38.63	kd	CGS001-134288	TMEM174	-			
5147	-38.66	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
5148	-38.67	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
5149	-38.69	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
5150	-38.71	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
5151	-38.73	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
5152	-38.74	kd	CGS001-126823	KLHDC9	-			
5153	-38.81	cp	BRD-K43236057	piceid	ICAM1 inhibitor		GAA, XDH	ICAM1 inhibitor
5154	-38.83	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
5155	-38.83	oe	ccsbBroad304_06090	DDOST	-			
5156	-38.85	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
5157	-38.91	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
5158	-38.91	kd	CGS001-2909	ARHGAP35	Rho GTPase activating proteins			
5159	-38.95	kd	CGS001-4791	NFKB2	NFkappaB transcription factor family			
5160	-38.95	kd	CGS001-10018	BCL2L11	-			
5161	-38.96	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
5162	-38.99	kd	CGS001-8900	CCNA1	-			
5163	-39.01	kd	CGS001-5684	PSMA3	Proteasome subunits			
5164	-39.02	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
5165	-39.02	kd	CGS001-6500	SKP1	-			
5166	-39.06	kd	CGS001-4086	SMAD1	SMADs			
5167	-39.06	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
5168	-39.06	kd	CGS001-10525	HYOU1	Heat shock proteins / HSP70			
5169	-39.1	oe	ccsbBroad304_07287	HYAL2	-			
5170	-39.1	kd	CGS001-6934	TCF7L2	-			
5171	-39.17	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
5172	-39.18	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
5173	-39.21	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
5174	-39.22	oe	ccsbBroad304_02788	PRAME	-			
5175	-39.23	oe	ccsbBroad304_02195	SPAG7	-			
5176	-39.24	kd	CGS001-89910	UBE3B	-			
5177	-39.24	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
5178	-39.27	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
5179	-39.28	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
5180	-39.28	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
5181	-39.31	kd	CGS001-50865	HEBP1	Endogenous ligands			
5182	-39.32	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
5183	-39.36	oe	ccsbBroad304_06549	SMAD3	SMADs			
5184	-39.37	oe	ccsbBroad304_11405	UBE3C	-			
5185	-39.37	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
5186	-39.39	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
5187	-39.4	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
5188	-39.45	kd	CGS001-9200	PTPLA	-			
5189	-39.47	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
5190	-39.47	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
5191	-39.48	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
5192	-39.5	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
5193	-39.51	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
5194	-39.51	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
5195	-39.52	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
5196	-39.52	cp	BRD-K52020312	metronidazole	DNA inhibitor		CYP2C8, CYP2E1, CYP3A5, CYP3A7	DNA inhibitor, Antiprotozoal
5197	-39.52	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
5198	-39.53	oe	ccsbBroad304_02048	BCL10	-			
5199	-39.59	kd	CGS001-1495	CTNNA1	Catenins			
5200	-39.66	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
5201	-39.67	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
5202	-39.72	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
5203	-39.75	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
5204	-39.85	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
5205	-39.85	kd	CGS001-7323	UBE2D3	Ubiquitin-conjugating enzymes E2			
5206	-39.88	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
5207	-39.93	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
5208	-39.96	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
5209	-40.01	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
5210	-40.01	kd	CGS001-6119	RPA3	-			
5211	-40.22	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
5212	-40.22	kd	CGS001-7040	TGFB1	Endogenous ligands			
5213	-40.22	kd	CGS001-8525	DGKZ	-			
5214	-40.23	cc		NFKB Activation GOF	-			
5215	-40.26	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
5216	-40.31	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
5217	-40.34	kd	CGS001-80347	COASY	-			
5218	-40.38	kd	CGS001-1978	EIF4EBP1	-			
5219	-40.39	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
5220	-40.44	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
5221	-40.54	kd	CGS001-7132	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
5222	-40.57	oe	ccsbBroad304_00933	LDHB	-			
5223	-40.57	kd	CGS001-58472	SQRDL	-			
5224	-40.58	oe	ccsbBroad304_00486	EFNB2	Ephrins			
5225	-40.6	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
5226	-40.61	kd	CGS001-8702	B4GALT4	Beta 4-glycosyltransferases			
5227	-40.63	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5228	-40.66	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
5229	-40.69	oe	ccsbBroad304_09195	MCM8	-			
5230	-40.69	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
5231	-40.73	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
5232	-40.76	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
5233	-40.77	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
5234	-40.83	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
5235	-40.86	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
5236	-40.88	kd	CGS001-6897	TARS	Aminoacyl tRNA synthetases / Class II			
5237	-40.95	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
5238	-40.97	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
5239	-40.98	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
5240	-41.02	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
5241	-41.05	oe	ccsbBroad304_05183	TXLNA	-			
5242	-41.07	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
5243	-41.09	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
5244	-41.12	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
5245	-41.16	kd	CGS001-1645	AKR1C1	Aldo-keto reductases			
5246	-41.19	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
5247	-41.2	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
5248	-41.27	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5249	-41.28	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
5250	-41.3	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
5251	-41.3	kd	CGS001-54106	TLR9	Toll-like receptor family			
5252	-41.32	kd	CGS001-5997	RGS2	Endogenous ligands			
5253	-41.35	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
5254	-41.37	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
5255	-41.37	oe	ccsbBroad304_00710	GUSB	-			
5256	-41.44	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
5257	-41.45	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
5258	-41.47	kd	CGS001-2782	GNB1	WD repeat domain containing			
5259	-41.53	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
5260	-41.64	oe	ccsbBroad304_01183	PGD	-			
5261	-41.67	kd	CGS001-348	APOE	Apolipoproteins			
5262	-41.69	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
5263	-41.74	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
5264	-41.76	kd	CGS001-5571	PRKAG1	AMPK subfamily			
5265	-41.77	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
5266	-41.8	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
5267	-41.81	kd	CGS001-8738	CRADD	-			
5268	-41.83	kd	CGS001-80150	ASRGL1	-			
5269	-41.84	oe	ccsbBroad304_07600	NSA2	-			
5270	-41.92	oe	ccsbBroad304_04788	OVCA2	-			
5271	-41.92	kd	CGS001-22978	NT5C2	Adenosine turnover			
5272	-41.93	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
5273	-41.98	oe	ccsbBroad304_02502	GNA13	-			
5274	-41.98	cp	BRD-K94144010	cotinine	Nicotine metabolite			Nicotine metabolite
5275	-42.02	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
5276	-42.03	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
5277	-42.03	kd	CGS001-4067	LYN	Src family			
5278	-42.12	cp	BRD-K70358946	aripiprazole	Serotonin receptor agonist		DRD2, HTR1A, HTR2A, HRH1, HTR1B, HTR1D, HTR2C, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR1E, HTR3A, HTR6, HTR7	Serotonin receptor agonist, Serotonin receptor antagonist
5279	-42.19	kd	CGS001-6663	SOX10	SRY (sex determining region Y)-boxes			
5280	-42.2	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
5281	-42.21	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
5282	-42.22	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
5283	-42.24	oe	ccsbBroad304_02278	THRAP3	-			
5284	-42.24	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
5285	-42.4	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
5286	-42.4	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
5287	-42.4	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
5288	-42.4	kd	CGS001-3669	ISG20	-			
5289	-42.41	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
5290	-42.43	kd	CGS001-124641	OVCA2	-			
5291	-42.44	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
5292	-42.46	cc		MCM family LOF	-			
5293	-42.47	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
5294	-42.49	oe	ccsbBroad304_02402	TMEM5	-			
5295	-42.49	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
5296	-42.5	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
5297	-42.51	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
5298	-42.52	kd	CGS001-9643	MORF4L2	-			
5299	-42.54	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
5300	-42.54	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
5301	-42.59	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
5302	-42.65	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
5303	-42.65	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
5304	-42.65	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
5305	-42.74	kd	CGS001-2745	GLRX	-			
5306	-42.75	kd	CGS001-9552	SPAG7	-			
5307	-42.77	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
5308	-42.81	kd	CGS001-4300	MLLT3	-			
5309	-42.82	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
5310	-42.83	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
5311	-42.83	oe	ccsbBroad304_00836	IGF2	-			
5312	-42.85	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
5313	-42.86	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
5314	-42.9	oe	ccsbBroad304_06683	FURIN	Subtilisin			
5315	-42.91	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
5316	-42.95	oe	ccsbBroad304_06264	GBP2	-			
5317	-43.02	cp	BRD-K73991644	isoquercetin	Aldose reductase inhibitor		AKR1B1, ACE	Aldose reductase inhibitor
5318	-43.03	kd	CGS001-3265	HRAS	RAS subfamily			
5319	-43.04	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
5320	-43.1	oe	ccsbBroad304_07411	LPXN	-			
5321	-43.15	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
5322	-43.15	kd	CGS001-238	ALK	Leukocyte tyrosine kinase (LTK) receptor family			
5323	-43.19	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5324	-43.2	oe	ccsbBroad304_02581	ASCC3	-			
5325	-43.24	oe	ccsbBroad304_00184	C2	Complement system			
5326	-43.32	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
5327	-43.37	oe	ccsbBroad304_04404	TUBB6	Tubulins			
5328	-43.42	oe	ccsbBroad304_02815	SSBP2	-			
5329	-43.42	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
5330	-43.43	oe	ccsbBroad304_01002	METTL1	-			
5331	-43.43	oe	ccsbBroad304_00003	ABAT	GABA turnover			
5332	-43.51	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
5333	-43.52	kd	CGS001-2746	GLUD1	-			
5334	-43.54	oe	ccsbBroad304_00728	HBE1	-			
5335	-43.57	kd	CGS001-9784	SNX17	Sorting nexins			
5336	-43.58	cc		VEGFR inhibitor	-			
5337	-43.58	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
5338	-43.61	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
5339	-43.62	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
5340	-43.64	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5341	-43.72	cc		Cell Cycle Inhibition GOF	-			
5342	-43.74	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
5343	-43.78	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
5344	-43.81	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
5345	-43.84	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
5346	-43.88	oe	ccsbBroad304_07843	FCHO1	-			
5347	-43.88	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
5348	-43.89	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
5349	-43.91	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
5350	-43.91	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
5351	-43.92	kd	CGS001-5110	PCMT1	-			
5352	-43.94	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
5353	-43.99	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
5354	-44	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
5355	-44.04	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
5356	-44.04	kd	CGS001-51071	DERA	-			
5357	-44.08	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
5358	-44.15	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
5359	-44.15	kd	CGS001-498	ATP5A1	ATPases / F-type			
5360	-44.17	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
5361	-44.18	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
5362	-44.18	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
5363	-44.22	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
5364	-44.22	kd	CGS001-5253	PHF2	Histone demethylases			
5365	-44.23	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
5366	-44.24	kd	CGS001-80306	MED28	-			
5367	-44.26	kd	CGS001-3985	LIMK2	LIMK subfamily			
5368	-44.27	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
5369	-44.28	kd	CGS001-116832	RPL39L	L ribosomal proteins			
5370	-44.3	cp	BRD-A68589262	troxipide	Glucosamine synthetase stimulant			Glucosamine synthetase stimulant
5371	-44.33	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
5372	-44.34	oe	ccsbBroad304_09503	KLHDC9	-			
5373	-44.39	kd	CGS001-8576	STK16	NAK family			
5374	-44.4	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
5375	-44.51	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
5376	-44.56	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
5377	-44.56	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
5378	-44.59	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
5379	-44.66	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
5380	-44.66	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
5381	-44.66	kd	CGS001-83999	KREMEN1	-			
5382	-44.68	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
5383	-44.72	cp	BRD-K02227374	milnacipran	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Serotonin reuptake inhibitor
5384	-44.74	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5385	-44.75	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
5386	-44.78	kd	CGS001-26298	EHF	-			
5387	-44.84	kd	CGS001-10482	NXF1	-			
5388	-44.86	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
5389	-44.87	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
5390	-44.9	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
5391	-44.9	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
5392	-44.94	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
5393	-44.96	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
5394	-45	cc		Ribonucleotide reductase inhibitor	-			
5395	-45.01	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
5396	-45.03	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
5397	-45.04	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
5398	-45.04	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
5399	-45.12	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5400	-45.15	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
5401	-45.16	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
5402	-45.16	kd	CGS001-10421	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5403	-45.19	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
5404	-45.25	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
5405	-45.31	oe	ccsbBroad304_01373	RAN	-			
5406	-45.33	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5407	-45.33	kd	CGS001-10084	PQBP1	-			
5408	-45.34	kd	CGS001-9870	KIAA0317	-			
5409	-45.35	kd	CGS001-64121	RRAGC	-			
5410	-45.42	kd	CGS001-7316	UBC	-			
5411	-45.42	kd	CGS001-8651	SOCS1	SH2 domain containing			
5412	-45.5	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5413	-45.51	kd	CGS001-3171	FOXA3	Forkhead boxes			
5414	-45.56	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
5415	-45.56	kd	CGS001-1512	CTSH	Cathepsins			
5416	-45.57	kd	CGS001-23499	MACF1	EF-hand domain containing			
5417	-45.62	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
5418	-45.64	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
5419	-45.64	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
5420	-45.68	kd	CGS001-55907	CMAS	-			
5421	-45.71	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
5422	-45.78	oe	ccsbBroad304_00552	FEN1	-			
5423	-45.79	kd	CGS001-64710	NUCKS1	-			
5424	-45.83	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
5425	-45.86	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5426	-45.89	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
5427	-45.91	oe	ccsbBroad304_01205	PIN1	-			
5428	-45.92	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
5429	-45.94	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
5430	-45.97	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
5431	-45.97	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
5432	-45.98	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5433	-46.02	oe	ccsbBroad304_00430	GADD45A	-			
5434	-46.06	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
5435	-46.07	oe	ccsbBroad304_14174	CDKAL1	-			
5436	-46.08	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
5437	-46.12	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
5438	-46.17	kd	CGS001-641	BLM	-			
5439	-46.19	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5440	-46.22	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
5441	-46.23	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
5442	-46.29	kd	CGS001-6598	SMARCB1	-			
5443	-46.33	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
5444	-46.35	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
5445	-46.35	kd	CGS001-220	ALDH1A3	Aldehyde dehydrogenases			
5446	-46.38	kd	CGS001-6822	SULT2A1	Sulfotransferases, cytosolic			
5447	-46.42	kd	CGS001-826	CAPNS1	EF-hand domain containing			
5448	-46.43	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5449	-46.43	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
5450	-46.47	kd	CGS001-5586	PKN2	Protein kinase N (PKN) family			
5451	-46.49	kd	CGS001-635	BHMT	-			
5452	-46.5	oe	ccsbBroad304_03268	GMPR2	-			
5453	-46.54	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
5454	-46.65	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5455	-46.66	cc		LIM class homeoboxes GOF	-			
5456	-46.66	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
5457	-46.7	cc		Androgen receptor modulator	-			
5458	-46.71	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
5459	-46.78	kd	CGS001-51441	YTHDF2	-			
5460	-46.82	oe	ccsbBroad304_13813	ARAF	RAF family			
5461	-46.86	oe	ccsbBroad304_03428	EXOSC4	-			
5462	-46.96	kd	CGS001-6622	SNCA	Parkinson disease			
5463	-46.96	kd	CGS001-533	ATP6V0B	ATPases / V-type			
5464	-47.05	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
5465	-47.05	kd	CGS001-79258	MMEL1	-			
5466	-47.06	kd	CGS001-83637	ZMIZ2	Zinc fingers, MIZ-type			
5467	-47.08	cc		Progesterone receptor antagonist	-			
5468	-47.08	kd	CGS001-375133	PI4KAP2	-			
5469	-47.13	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
5470	-47.19	kd	CGS001-310	ANXA7	Annexins			
5471	-47.2	kd	CGS001-9122	SLC16A4	SLC16 family of monocarboxylate transporters			
5472	-47.24	oe	ccsbBroad304_02276	MVP	-			
5473	-47.25	kd	CGS001-143187	VTI1A	-			
5474	-47.27	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
5475	-47.29	oe	ccsbBroad304_01632	SYPL1	-			
5476	-47.29	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
5477	-47.38	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
5478	-47.41	oe	ccsbBroad304_08536	PARL	-			
5479	-47.44	kd	CGS001-1950	EGF	-			
5480	-47.47	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
5481	-47.5	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
5482	-47.5	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
5483	-47.52	oe	ccsbBroad304_02884	POT1	-			
5484	-47.52	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
5485	-47.52	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5486	-47.52	kd	CGS001-2230	FDX1	-			
5487	-47.55	kd	CGS001-7431	VIM	Intermediate filaments type III			
5488	-47.6	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
5489	-47.63	oe	ccsbBroad304_03640	CEP72	-			
5490	-47.7	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
5491	-47.74	kd	CGS001-6514	SLC2A2	Solute carriers			
5492	-47.77	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
5493	-47.82	kd	CGS001-3161	HMMR	CD molecules			
5494	-47.83	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
5495	-47.86	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
5496	-47.96	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5497	-47.97	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
5498	-48.03	kd	CGS001-9612	NCOR2	-			
5499	-48.06	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
5500	-48.06	kd	CGS001-205	AK4	Adenylate kinases			
5501	-48.08	oe	ccsbBroad304_07029	TADA2A	-			
5502	-48.08	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
5503	-48.19	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
5504	-48.22	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
5505	-48.22	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
5506	-48.23	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5507	-48.3	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
5508	-48.31	kd	CGS001-10626	TRIM16	Tripartite motif containing			
5509	-48.35	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5510	-48.38	oe	ccsbBroad304_03080	C16ORF80	-			
5511	-48.41	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
5512	-48.42	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
5513	-48.45	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
5514	-48.45	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5515	-48.56	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
5516	-48.56	cp	BRD-K06817181	BRD-K06817181	JAK inhibitor		JAK2	JAK inhibitor
5517	-48.59	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
5518	-48.62	oe	ccsbBroad304_08898	TRAK2	-			
5519	-48.62	kd	CGS001-2878	GPX3	-			
5520	-48.65	kd	CGS001-293	SLC25A6	Mitochondrial nucleotide transporter subfamily			
5521	-48.66	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5522	-48.68	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
5523	-48.69	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5524	-48.76	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
5525	-48.76	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
5526	-48.81	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
5527	-48.81	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
5528	-48.84	kd	CGS001-351	APP	Endogenous ligands			
5529	-48.85	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
5530	-48.89	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
5531	-48.93	kd	CGS001-5663	PSEN1	Presenilin			
5532	-48.94	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
5533	-48.98	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
5534	-49	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
5535	-49.04	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
5536	-49.06	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
5537	-49.12	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
5538	-49.14	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
5539	-49.14	kd	CGS001-6926	TBX3	T-boxes			
5540	-49.18	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
5541	-49.26	kd	CGS001-51293	CD320	CD molecules			
5542	-49.29	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
5543	-49.29	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
5544	-49.29	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
5545	-49.46	oe	ccsbBroad304_00462	DR1	-			
5546	-49.64	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
5547	-49.64	kd	CGS001-84515	MCM8	-			
5548	-49.69	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
5549	-49.79	kd	CGS001-6513	SLC2A1	Solute carriers			
5550	-49.82	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
5551	-49.89	oe	ccsbBroad304_08045	NOX1	-			
5552	-49.89	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
5553	-49.89	kd	CGS001-2920	CXCL2	Endogenous ligands			
5554	-49.9	kd	CGS001-5255	PHKA1	-			
5555	-50.05	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
5556	-50.05	kd	CGS001-56005	C19ORF10	-			
5557	-50.07	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
5558	-50.1	kd	CGS001-85480	TSLP	-			
5559	-50.15	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
5560	-50.15	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
5561	-50.17	kd	CGS001-26149	ZNF658	Zinc fingers, C2H2-type			
5562	-50.17	kd	CGS001-9377	COX5A	Mitochondrial respiratory chain complex			
5563	-50.18	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
5564	-50.21	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
5565	-50.23	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
5566	-50.27	kd	CGS001-5188	PET112	-			
5567	-50.28	kd	CGS001-6443	SGCB	-			
5568	-50.34	oe	ccsbBroad304_00651	GNAI3	-			
5569	-50.37	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
5570	-50.4	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
5571	-50.53	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
5572	-50.55	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
5573	-50.58	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
5574	-50.59	cc		P38 MAPK inhibitor	-			
5575	-50.63	kd	CGS001-30836	DNTTIP2	-			
5576	-50.66	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
5577	-50.68	oe	ccsbBroad304_02484	PAICS	-			
5578	-50.72	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
5579	-50.75	oe	ccsbBroad304_03850	TRIB3	Trbl family			
5580	-50.76	oe	ccsbBroad304_01974	RNASET2	-			
5581	-50.81	kd	CGS001-89765	RSPH1	-			
5582	-50.87	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
5583	-50.89	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
5584	-51	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
5585	-51.02	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
5586	-51.02	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
5587	-51.08	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
5588	-51.15	kd	CGS001-55631	LRRC40	-			
5589	-51.16	kd	CGS001-54925	ZNF434	-			
5590	-51.16	kd	CGS001-51005	AMDHD2	-			
5591	-51.25	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
5592	-51.25	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
5593	-51.28	oe	ccsbBroad304_00490	EIF4EBP1	-			
5594	-51.29	kd	CGS001-57222	ERGIC1	-			
5595	-51.3	oe	ccsbBroad304_01222	PLP2	-			
5596	-51.38	kd	CGS001-51268	PIPOX	-			
5597	-51.43	oe	ccsbBroad304_07071	TKT	-			
5598	-51.5	kd	CGS001-873	CBR1	Prostaglandin synthases			
5599	-51.52	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
5600	-51.53	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
5601	-51.53	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
5602	-51.57	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
5603	-51.58	oe	ccsbBroad304_06462	ITGAE	Integrins			
5604	-51.59	kd	CGS001-5813	PURA	-			
5605	-51.6	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
5606	-51.63	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
5607	-51.64	kd	CGS001-54681	P4HTM	-			
5608	-51.65	oe	ccsbBroad304_06255	LRRC32	-			
5609	-51.65	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
5610	-51.67	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
5611	-51.68	cp	BRD-K49668410	clarithromycin	Bacterial 50S ribosomal subunit inhibitor		CYP2C19, CYP3A4, CYP3A5, CYP3A7	Bacterial 50S ribosomal subunit inhibitor
5612	-51.69	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
5613	-51.74	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
5614	-51.81	oe	ccsbBroad304_01880	LAGE3	-			
5615	-51.81	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
5616	-51.83	kd	CGS001-10423	CDIPT	-			
5617	-51.84	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
5618	-51.86	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
5619	-51.92	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
5620	-51.95	oe	ccsbBroad304_00472	EBF1	-			
5621	-51.96	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5622	-51.96	kd	CGS001-11212	PROSC	-			
5623	-52.01	cp	BRD-K44442813	pidotimod	Interferon receptor agonist			Interferon receptor agonist, Interleukin receptor agonist
5624	-52.1	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5625	-52.11	oe	ccsbBroad304_07632	PROCR	CD molecules			
5626	-52.11	kd	CGS001-8895	CPNE3	-			
5627	-52.15	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
5628	-52.15	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
5629	-52.16	kd	CGS001-10020	GNE	-			
5630	-52.21	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
5631	-52.22	kd	CGS001-7314	UBB	-			
5632	-52.23	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
5633	-52.23	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
5634	-52.28	kd	CGS001-23492	CBX7	-			
5635	-52.3	oe	ccsbBroad304_00570	FIGF	-			
5636	-52.33	kd	CGS001-4221	MEN1	-			
5637	-52.4	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
5638	-52.44	kd	CGS001-84930	MASTL	MAST family			
5639	-52.52	oe	ccsbBroad304_06094	DFFA	-			
5640	-52.52	oe	ccsbBroad304_01150	PCCB	Carboxylases			
5641	-52.53	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
5642	-52.55	cc		Zinc fingers RanBP2 type LOF	-			
5643	-52.55	kd	CGS001-5934	RBL2	-			
5644	-52.58	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
5645	-52.59	kd	CGS001-8797	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
5646	-52.61	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
5647	-52.76	oe	ccsbBroad304_03728	DIABLO	-			
5648	-52.77	kd	CGS001-821	CANX	-			
5649	-52.95	oe	ccsbBroad304_07374	PTPLA	-			
5650	-52.95	kd	CGS001-8575	PRKRA	-			
5651	-53	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
5652	-53	oe	ccsbBroad304_00020	ACY1	-			
5653	-53.05	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5654	-53.13	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
5655	-53.13	kd	CGS001-3998	LMAN1	-			
5656	-53.15	oe	ccsbBroad304_03812	PBXIP1	-			
5657	-53.16	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
5658	-53.16	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
5659	-53.19	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
5660	-53.19	kd	CGS001-35	ACADS	-			
5661	-53.25	oe	ccsbBroad304_02804	KLHDC2	-			
5662	-53.28	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
5663	-53.28	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
5664	-53.29	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
5665	-53.29	kd	CGS001-81577	GFOD2	-			
5666	-53.33	kd	CGS001-6307	MSMO1	Fatty acid hydroxylase domain containing			
5667	-53.45	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
5668	-53.46	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
5669	-53.48	kd	CGS001-63933	CCDC90A	-			
5670	-53.52	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
5671	-53.54	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
5672	-53.54	kd	CGS001-9589	WTAP	-			
5673	-53.57	kd	CGS001-9159	PCSK7	Subtilisin			
5674	-53.58	oe	ccsbBroad304_07798	EXOC3	-			
5675	-53.6	kd	CGS001-55746	NUP133	-			
5676	-53.6	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
5677	-53.61	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
5678	-53.63	kd	CGS001-5433	POLR2D	RNA polymerase subunits			
5679	-53.67	cc		Estrogen receptor agonist	-			
5680	-53.71	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
5681	-53.72	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
5682	-53.73	oe	ccsbBroad304_04675	ATG4A	-			
5683	-53.74	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
5684	-53.77	oe	ccsbBroad304_02772	ICMT	-			
5685	-53.82	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
5686	-53.84	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
5687	-53.87	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
5688	-53.91	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
5689	-53.92	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
5690	-53.94	kd	CGS001-7032	TFF2	-			
5691	-53.96	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
5692	-54	kd	CGS001-54957	TXNL4B	-			
5693	-54.06	cc		Tubulin inhibitor	-			
5694	-54.17	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
5695	-54.18	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
5696	-54.19	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
5697	-54.24	kd	CGS001-2244	FGB	Endogenous ligands			
5698	-54.27	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
5699	-54.3	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
5700	-54.3	oe	ccsbBroad304_01659	TERF1	-			
5701	-54.31	kd	CGS001-7027	TFDP1	-			
5702	-54.37	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
5703	-54.48	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
5704	-54.49	oe	ccsbBroad304_00397	CTSK	Cathepsins			
5705	-54.5	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
5706	-54.51	oe	ccsbBroad304_02287	GNPDA1	-			
5707	-54.54	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5708	-54.65	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
5709	-54.67	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
5710	-54.68	oe	ccsbBroad304_00661	GNGT2	-			
5711	-54.75	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
5712	-54.75	kd	CGS001-79080	CCDC86	-			
5713	-54.76	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
5714	-54.77	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
5715	-54.83	kd	CGS001-5184	PEPD	Methionyl aminopeptidase			
5716	-54.94	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
5717	-54.97	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
5718	-54.97	kd	CGS001-2629	GBA	-			
5719	-55	oe	ccsbBroad304_06783	LGMN	Legumain			
5720	-55.02	kd	CGS001-5914	RARA	Retinoic acid receptors			
5721	-55.03	kd	CGS001-54658	UGT1A1	UDP glucuronosyltransferases			
5722	-55.09	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
5723	-55.1	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
5724	-55.13	cp	BRD-K59753975	vindesine	Tubulin inhibitor		TUBB, TUBB1	Tubulin inhibitor
5725	-55.15	kd	CGS001-54821	ERCC6L	-			
5726	-55.26	kd	CGS001-2737	GLI3	Zinc fingers, C2H2-type			
5727	-55.26	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
5728	-55.28	oe	ccsbBroad304_00099	ARG2	Arginase			
5729	-55.29	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
5730	-55.32	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
5731	-55.35	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
5732	-55.44	kd	CGS001-11267	SNF8	-			
5733	-55.51	cp	BRD-K82109576	vincristine	Tubulin inhibitor		TUBB, TUBA4A	Tubulin inhibitor
5734	-55.53	oe	ccsbBroad304_05894	BLVRA	-			
5735	-55.6	kd	CGS001-7879	RAB7A	RAB, member RAS oncogene			
5736	-55.62	oe	ccsbBroad304_07490	SCRN1	-			
5737	-55.62	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
5738	-55.65	kd	CGS001-4200	ME2	-			
5739	-55.67	oe	ccsbBroad304_02864	PRDX5	-			
5740	-55.68	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
5741	-55.72	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
5742	-55.75	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5743	-55.77	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
5744	-55.78	kd	CGS001-9344	TAOK2	TAO subfamily			
5745	-55.84	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
5746	-55.85	kd	CGS001-2673	GFPT1	-			
5747	-55.88	cp	BRD-A79314293	cephalosporanic-acid	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5748	-55.97	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
5749	-56.01	kd	CGS001-5159	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5750	-56.07	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
5751	-56.09	kd	CGS001-5245	PHB	-			
5752	-56.12	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
5753	-56.16	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
5754	-56.18	kd	CGS001-440	ASNS	-			
5755	-56.21	cp	BRD-K50384076	7,4'-dihydroxyflavone	Opioid receptor antagonist		CYP19A1	Opioid receptor antagonist
5756	-56.22	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5757	-56.28	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
5758	-56.29	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
5759	-56.3	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
5760	-56.3	kd	CGS001-132	ADK	Adenosine turnover			
5761	-56.31	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
5762	-56.35	oe	ccsbBroad304_02443	HAX1	-			
5763	-56.36	oe	ccsbBroad304_01640	TAF12	-			
5764	-56.41	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
5765	-56.44	cc		EGFR inhibitor	-			
5766	-56.49	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
5767	-56.57	oe	ccsbBroad304_03264	UBAP1	-			
5768	-56.57	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
5769	-56.62	kd	CGS001-1020	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
5770	-56.63	oe	ccsbBroad304_02875	BRP44	-			
5771	-56.64	kd	CGS001-166793	ZBTB49	BTB/POZ domain containing			
5772	-56.65	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
5773	-56.67	kd	CGS001-5080	PAX6	Paired boxes			
5774	-56.71	cc		Baculoviral IAP repeat domain containing LOF	-			
5775	-56.72	kd	CGS001-8667	EIF3H	-			
5776	-56.77	kd	CGS001-5160	PDHA1	-			
5777	-56.83	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
5778	-56.83	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
5779	-56.88	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
5780	-56.88	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
5781	-56.88	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
5782	-56.89	kd	CGS001-7474	WNT5A	Endogenous ligands			
5783	-56.95	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
5784	-56.96	kd	CGS001-7541	ZFP161	-			
5785	-56.99	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
5786	-57.12	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
5787	-57.12	kd	CGS001-27034	ACAD8	-			
5788	-57.15	cc		Serpin peptidase inhibitors LOF	-			
5789	-57.15	oe	ccsbBroad304_06449	ILF3	-			
5790	-57.16	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
5791	-57.2	kd	CGS001-8634	RTCD1	-			
5792	-57.21	kd	CGS001-2593	GAMT	-			
5793	-57.24	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
5794	-57.28	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
5795	-57.31	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
5796	-57.31	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
5797	-57.36	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
5798	-57.43	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
5799	-57.45	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
5800	-57.47	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
5801	-57.5	kd	CGS001-388677	NOTCH2NL	-			
5802	-57.5	kd	CGS001-10645	CAMKK2	Meta subfamily			
5803	-57.51	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
5804	-57.55	kd	CGS001-91949	COG7	Components of oligomeric golgi complex			
5805	-57.56	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
5806	-57.56	kd	CGS001-7165	TPD52L2	-			
5807	-57.58	cp	BRD-K51671335	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
5808	-57.59	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
5809	-57.66	kd	CGS001-7276	TTR	-			
5810	-57.7	oe	ccsbBroad304_02551	CPSF4	-			
5811	-57.72	oe	ccsbBroad304_10431	HADHB	-			
5812	-57.73	oe	ccsbBroad304_09281	TPD52L3	-			
5813	-57.81	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
5814	-57.83	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
5815	-57.85	oe	ccsbBroad304_10491	PFKL	-			
5816	-57.85	kd	CGS001-3479	IGF1	Endogenous ligands			
5817	-57.87	kd	CGS001-161	AP2A2	-			
5818	-57.96	oe	ccsbBroad304_00874	INS	-			
5819	-57.97	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
5820	-57.97	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
5821	-57.98	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
5822	-57.99	kd	CGS001-8837	CFLAR	Endogenous ligands			
5823	-58.01	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
5824	-58.03	kd	CGS001-10769	PLK2	Polo-like kinase (PLK) family			
5825	-58.04	oe	ccsbBroad304_07252	DGKZ	-			
5826	-58.04	oe	ccsbBroad304_05985	CFL1	-			
5827	-58.1	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
5828	-58.15	kd	CGS001-445	ASS1	-			
5829	-58.16	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
5830	-58.16	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
5831	-58.19	kd	CGS001-5345	SERPINF2	Serine (or cysteine) peptidase inhibitors			
5832	-58.2	oe	ccsbBroad304_00615	GAPDH	-			
5833	-58.22	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
5834	-58.24	kd	CGS001-5063	PAK3	PAKA subfamily			
5835	-58.25	kd	CGS001-5985	RFC5	ATPases / AAA-type			
5836	-58.27	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
5837	-58.32	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
5838	-58.34	oe	ccsbBroad304_06159	CTTN	-			
5839	-58.44	oe	ccsbBroad304_00614	GAMT	-			
5840	-58.55	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
5841	-58.56	kd	CGS001-1072	CFL1	-			
5842	-58.57	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
5843	-58.67	kd	CGS001-10933	MORF4L1	-			
5844	-58.7	cc		Protein synthesis inhibitor	-			
5845	-58.72	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
5846	-58.74	kd	CGS001-90655	TGIF2LY	Homeoboxes / TALE class			
5847	-58.76	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
5848	-58.76	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
5849	-58.79	kd	CGS001-6129	RPL7	L ribosomal proteins			
5850	-58.86	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
5851	-58.99	kd	CGS001-6723	SRM	-			
5852	-59.01	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
5853	-59.03	cp	BRD-K04710043	hexamethylenebisacetamide	AKT inhibitor			AKT inhibitor, Differentiation inducer, NFkB pathway inhibitor
5854	-59.04	oe	ccsbBroad304_00389	CTBP1	-			
5855	-59.05	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
5856	-59.09	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
5857	-59.11	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
5858	-59.11	kd	CGS001-47	ACLY	-			
5859	-59.12	oe	ccsbBroad304_04616	ORMDL3	-			
5860	-59.14	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
5861	-59.24	oe	ccsbBroad304_03311	EVL	-			
5862	-59.24	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
5863	-59.25	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
5864	-59.26	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
5865	-59.27	cp	BRD-K09471561	levofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
5866	-59.37	kd	CGS001-9512	PMPCB	-			
5867	-59.38	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
5868	-59.39	cc		Tricyclic antidepressant	-			
5869	-59.4	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
5870	-59.43	kd	CGS001-2643	GCH1	-			
5871	-59.46	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
5872	-59.46	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
5873	-59.48	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
5874	-59.49	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
5875	-59.52	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
5876	-59.58	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
5877	-59.62	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
5878	-59.63	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5879	-59.64	kd	CGS001-3725	JUN	basic leucine zipper proteins			
5880	-59.64	kd	CGS001-3313	HSPA9	Heat shock proteins / HSP70			
5881	-59.67	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
5882	-59.67	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5883	-59.68	oe	ccsbBroad304_08093	DCPS	-			
5884	-59.69	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
5885	-59.71	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
5886	-59.81	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
5887	-59.86	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
5888	-59.87	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
5889	-59.93	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
5890	-59.94	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
5891	-60.01	kd	CGS001-8731	RNMT	-			
5892	-60.02	kd	CGS001-8233	ZRSR2	RNA binding motif (RRM) containing			
5893	-60.07	kd	CGS001-8850	KAT2B	Histone acetyltransferases (HATs)			
5894	-60.08	kd	CGS001-4174	MCM5	-			
5895	-60.12	cp	BRD-A39172021	ampiroxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5896	-60.13	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
5897	-60.14	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5898	-60.16	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
5899	-60.16	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
5900	-60.17	oe	ccsbBroad304_00231	CBFB	-			
5901	-60.2	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
5902	-60.22	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
5903	-60.27	kd	CGS001-9404	LPXN	-			
5904	-60.28	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
5905	-60.3	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
5906	-60.33	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
5907	-60.34	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
5908	-60.35	oe	ccsbBroad304_07491	IP6K1	-			
5909	-60.47	kd	CGS001-25819	CCRN4L	-			
5910	-60.51	kd	CGS001-9531	BAG3	-			
5911	-60.55	kd	CGS001-896	CCND3	-			
5912	-60.59	kd	CGS001-9406	ZRANB2	Zinc fingers, RAN-binding domain containing			
5913	-60.65	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
5914	-60.67	kd	CGS001-169436	C9ORF96	-			
5915	-60.77	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
5916	-60.79	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
5917	-60.82	kd	CGS001-57804	POLD4	DNA polymerases			
5918	-60.88	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
5919	-60.93	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
5920	-61.01	cc		CDK inhibitor	-			
5921	-61.01	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
5922	-61.06	kd	CGS001-708	C1QBP	-			
5923	-61.15	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
5924	-61.16	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
5925	-61.17	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
5926	-61.21	kd	CGS001-133690	CAPSL	EF-hand domain containing			
5927	-61.23	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
5928	-61.27	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
5929	-61.31	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
5930	-61.31	kd	CGS001-10557	RPP38	-			
5931	-61.32	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
5932	-61.32	cp	BRD-A71009679	KUC103420N	-666			-666
5933	-61.37	kd	CGS001-55120	FANCL	Fanconi anemia, complementation groups			
5934	-61.39	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
5935	-61.39	kd	CGS001-5230	PGK1	-			
5936	-61.4	kd	CGS001-8874	ARHGEF7	Rho guanine nucleotide exchange factors			
5937	-61.46	oe	ccsbBroad304_07217	AXIN2	-			
5938	-61.61	oe	ccsbBroad304_06565	MB	-			
5939	-61.63	kd	CGS001-51282	SCAND1	-			
5940	-61.65	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5941	-61.65	kd	CGS001-55612	FERMT1	Fermitins			
5942	-61.71	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
5943	-61.74	kd	CGS001-7076	TIMP1	-			
5944	-61.75	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
5945	-61.8	kd	CGS001-6647	SOD1	-			
5946	-61.84	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
5947	-61.93	oe	ccsbBroad304_01105	PNP	-			
5948	-61.95	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
5949	-61.97	kd	CGS001-165082	GPR113	Adhesion Class GPCRs			
5950	-61.99	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
5951	-61.99	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
5952	-62	cp	BRD-K66412701	pazufloxacin	Topoisomerase inhibitor			Topoisomerase inhibitor
5953	-62.01	kd	CGS001-27097	TAF5L	WD repeat domain containing			
5954	-62.05	kd	CGS001-2678	GGT1	CD molecules			
5955	-62.07	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
5956	-62.09	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
5957	-62.11	oe	ccsbBroad304_03625	HIF1AN	-			
5958	-62.16	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
5959	-62.2	oe	ccsbBroad304_07101	TSC2	-			
5960	-62.22	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
5961	-62.22	kd	CGS001-84969	TOX2	-			
5962	-62.23	oe	ccsbBroad304_01483	SAT1	-			
5963	-62.26	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
5964	-62.26	kd	CGS001-2760	GM2A	-			
5965	-62.28	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
5966	-62.3	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
5967	-62.3	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
5968	-62.31	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
5969	-62.36	cp	BRD-K06388322	pramipexole	Dopamine receptor agonist		DRD3, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
5970	-62.4	cp	BRD-K63265447	docetaxel	Tubulin inhibitor		TUBB, BCL2, MAP2, MAP4, MAPT, NR1I2, TUBB1	Tubulin inhibitor
5971	-62.4	kd	CGS001-6391	SDHC	Mitochondrial respiratory chain complex / Complex II			
5972	-62.42	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
5973	-62.42	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
5974	-62.43	kd	CGS001-6493	SIM2	Basic helix-loop-helix proteins			
5975	-62.5	kd	CGS001-221188	GPR114	Adhesion Class GPCRs			
5976	-62.51	kd	CGS001-4704	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5977	-62.52	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
5978	-62.59	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
5979	-62.59	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
5980	-62.66	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
5981	-62.7	kd	CGS001-4718	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
5982	-62.71	oe	ccsbBroad304_07888	CBX6	-			
5983	-62.72	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
5984	-62.74	oe	ccsbBroad304_02801	CASP14	Caspases			
5985	-62.88	kd	CGS001-4092	SMAD7	SMADs			
5986	-62.9	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
5987	-62.95	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
5988	-63.01	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
5989	-63.07	oe	ccsbBroad304_02285	MED6	-			
5990	-63.07	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
5991	-63.12	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
5992	-63.15	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
5993	-63.2	kd	CGS001-1655	DDX5	DEAD-boxes			
5994	-63.21	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
5995	-63.22	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
5996	-63.25	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
5997	-63.37	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
5998	-63.39	kd	CGS001-4801	NFYB	-			
5999	-63.39	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
6000	-63.42	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
6001	-63.44	kd	CGS001-10544	PROCR	CD molecules			
6002	-63.45	kd	CGS001-5373	PMM2	-			
6003	-63.49	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
6004	-63.52	kd	CGS001-5538	PPT1	-			
6005	-63.54	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
6006	-63.55	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
6007	-63.55	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
6008	-63.55	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
6009	-63.58	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
6010	-63.61	kd	CGS001-57396	CLK4	CDC-like kinases			
6011	-63.74	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
6012	-63.78	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
6013	-63.81	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
6014	-63.82	oe	ccsbBroad304_08662	MCCC1	-			
6015	-63.82	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
6016	-63.83	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
6017	-63.86	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6018	-63.86	kd	CGS001-7270	TTF1	-			
6019	-63.9	cp	BRD-K54316499	tolterodine	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRM1, CHRM4, CHRM5	Acetylcholine receptor antagonist
6020	-63.95	kd	CGS001-7321	UBE2D1	Ubiquitin-conjugating enzymes E2			
6021	-63.99	kd	CGS001-7919	DDX39B	DEAD-boxes			
6022	-64	cp	BRD-A07395371	esmolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
6023	-64.01	kd	CGS001-9867	PJA2	RING-type (C3HC4) zinc fingers			
6024	-64.09	kd	CGS001-64080	RBKS	-			
6025	-64.11	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
6026	-64.21	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6027	-64.21	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
6028	-64.22	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
6029	-64.24	oe	ccsbBroad304_00152	BCAT2	-			
6030	-64.24	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
6031	-64.24	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
6032	-64.25	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
6033	-64.27	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
6034	-64.28	kd	CGS001-23118	TAB2	-			
6035	-64.32	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
6036	-64.34	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
6037	-64.37	cc		PPAR receptor agonist	-			
6038	-64.37	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
6039	-64.4	kd	CGS001-54749	EPDR1	-			
6040	-64.44	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
6041	-64.48	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
6042	-64.54	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
6043	-64.54	kd	CGS001-10813	UTP14A	-			
6044	-64.57	kd	CGS001-353345	GPR141	GPCR / Class A : Orphans			
6045	-64.67	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
6046	-64.67	kd	CGS001-28960	DCPS	-			
6047	-64.71	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
6048	-64.71	kd	CGS001-6502	SKP2	F-boxes / Leucine-rich repeats			
6049	-64.74	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
6050	-64.79	kd	CGS001-10298	PAK4	PAKB subfamily			
6051	-64.83	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
6052	-64.83	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6053	-64.84	oe	ccsbBroad304_07145	ZFP161	-			
6054	-64.88	kd	CGS001-8438	RAD54L	-			
6055	-64.9	oe	ccsbBroad304_05890	BHMT	-			
6056	-64.97	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
6057	-64.97	kd	CGS001-6654	SOS1	Rho guanine nucleotide exchange factors			
6058	-64.98	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
6059	-65.01	cp	BRD-K81855038	roxatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
6060	-65.05	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
6061	-65.05	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
6062	-65.05	kd	CGS001-472	ATM	Other PIKK family kinases			
6063	-65.06	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
6064	-65.08	cc		RNA Polymerase Enzymes LOF	-			
6065	-65.12	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6066	-65.15	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
6067	-65.22	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
6068	-65.26	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
6069	-65.26	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
6070	-65.32	kd	CGS001-84936	ZFYVE19	Zinc fingers, FYVE domain containing			
6071	-65.33	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
6072	-65.37	kd	CGS001-11112	HIBADH	-			
6073	-65.38	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
6074	-65.4	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
6075	-65.4	kd	CGS001-6722	SRF	-			
6076	-65.42	oe	ccsbBroad304_01061	NAB2	-			
6077	-65.43	kd	CGS001-5860	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
6078	-65.55	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
6079	-65.57	kd	CGS001-10383	TUBB2C	Tubulins			
6080	-65.6	kd	CGS001-7088	TLE1	WD repeat domain containing			
6081	-65.61	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
6082	-65.62	oe	ccsbBroad304_02671	ECD	-			
6083	-65.66	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
6084	-65.68	kd	CGS001-29888	STRN4	WD repeat domain containing			
6085	-65.68	kd	CGS001-5460	POU5F1	Homeoboxes / POU class			
6086	-65.69	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
6087	-65.69	kd	CGS001-2059	EPS8	-			
6088	-65.8	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
6089	-65.82	oe	ccsbBroad304_00398	CTSL2	-			
6090	-65.88	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
6091	-65.91	cc		Calmodulin antagonist	-			
6092	-65.94	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
6093	-65.95	cc		Cyclin dependent kinases LOF	-			
6094	-65.97	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
6095	-66	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
6096	-66.04	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
6097	-66.05	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
6098	-66.06	kd	CGS001-9797	TATDN2	-			
6099	-66.07	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
6100	-66.17	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6101	-66.18	kd	CGS001-382	ARF6	ADP-ribosylation factors			
6102	-66.24	cc		Aromatase inhibitor	-			
6103	-66.37	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
6104	-66.4	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
6105	-66.46	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6106	-66.49	kd	CGS001-3661	IRF3	-			
6107	-66.52	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
6108	-66.54	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
6109	-66.6	kd	CGS001-4835	NQO2	-			
6110	-66.65	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
6111	-66.71	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
6112	-66.75	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
6113	-66.78	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
6114	-66.79	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
6115	-66.8	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
6116	-66.9	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
6117	-66.94	kd	CGS001-10452	TOMM40	-			
6118	-66.95	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
6119	-66.98	kd	CGS001-257397	TAB3	-			
6120	-67.04	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
6121	-67.05	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
6122	-67.08	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
6123	-67.12	kd	CGS001-5320	PLA2G2A	Hydrolases			
6124	-67.13	cp	BRD-K21806131	tegaserod	Serotonin receptor partial agonist		HTR4, HTR2B, HTR2A, HTR2C	Serotonin receptor partial agonist
6125	-67.14	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
6126	-67.16	oe	ccsbBroad304_01034	MSH2	-			
6127	-67.24	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
6128	-67.3	kd	CGS001-2224	FDPS	Lanosterol biosynthesis pathway			
6129	-67.33	oe	ccsbBroad304_01147	PC	Carboxylases			
6130	-67.35	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
6131	-67.37	kd	CGS001-5471	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
6132	-67.4	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
6133	-67.42	oe	ccsbBroad304_13891	LCK	Src family			
6134	-67.48	cp	BRD-K63784565	BRD-K63784565	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
6135	-67.48	kd	CGS001-8824	CES2	Carboxylesterases			
6136	-67.53	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
6137	-67.58	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6138	-67.61	kd	CGS001-9180	OSMR	IL-6 receptor family			
6139	-67.67	cp	BRD-K39391626	ethylestrenol	Progesterone receptor agonist		AR	Progesterone receptor agonist
6140	-67.68	kd	CGS001-7295	TXN	-			
6141	-67.7	cc		ATPase inhibitor	-			
6142	-67.77	oe	ccsbBroad304_00957	M6PR	-			
6143	-67.79	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
6144	-67.89	kd	CGS001-64167	ERAP2	Aminopeptidase N			
6145	-67.93	oe	ccsbBroad304_07337	TAF1B	-			
6146	-67.97	kd	CGS001-8803	SUCLA2	-			
6147	-67.97	kd	CGS001-9978	RBX1	RING-type (C3HC4) zinc fingers			
6148	-68	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
6149	-68.01	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
6150	-68.02	kd	CGS001-9695	EDEM1	-			
6151	-68.03	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
6152	-68.07	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
6153	-68.08	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
6154	-68.11	cp	BRD-K92413528	thiazolidinecarboxylic-acid	Reducing agent			Reducing agent
6155	-68.12	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
6156	-68.27	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6157	-68.27	kd	CGS001-7849	PAX8	Paired boxes			
6158	-68.28	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6159	-68.28	kd	CGS001-6793	STK10	SLK subfamily			
6160	-68.29	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
6161	-68.29	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
6162	-68.32	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6163	-68.33	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
6164	-68.33	kd	CGS001-27076	LYPD3	-			
6165	-68.39	kd	CGS001-9443	MED7	-			
6166	-68.4	kd	CGS001-5613	PRKX	Protein kinase A			
6167	-68.48	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
6168	-68.48	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
6169	-68.51	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6170	-68.52	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
6171	-68.55	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
6172	-68.57	kd	CGS001-57616	TSHZ3	Teashirt zinc fingers			
6173	-68.57	kd	CGS001-5306	PITPNA	-			
6174	-68.57	kd	CGS001-2735	GLI1	Zinc fingers, C2H2-type			
6175	-68.58	cp	BRD-K97752965	nicorandil	Nitric oxide donor		ABCC9, KCNJ11, KCNJ8	Nitric oxide donor, Potassium channel activator
6176	-68.59	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
6177	-68.61	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
6178	-68.65	kd	CGS001-5355	PLP2	-			
6179	-68.77	oe	ccsbBroad304_07119	UGP2	-			
6180	-68.8	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
6181	-68.81	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
6182	-68.88	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
6183	-68.9	kd	CGS001-5595	MAPK3	MAPK:ERK subfamily			
6184	-68.91	oe	ccsbBroad304_00072	ANXA7	Annexins			
6185	-68.95	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
6186	-69.04	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
6187	-69.05	cc		Gamma secretase inhibitor	-			
6188	-69.09	oe	ccsbBroad304_05528	TICAM2	-			
6189	-69.2	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
6190	-69.25	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
6191	-69.27	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
6192	-69.29	cc		Integrin subunits beta LOF	-			
6193	-69.29	kd	CGS001-9807	IP6K1	-			
6194	-69.33	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
6195	-69.33	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
6196	-69.36	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
6197	-69.41	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
6198	-69.45	kd	CGS001-5025	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
6199	-69.56	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6200	-69.57	kd	CGS001-51070	NOSIP	-			
6201	-69.63	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
6202	-69.7	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
6203	-69.71	oe	ccsbBroad304_02497	YKT6	-			
6204	-69.71	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
6205	-69.76	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
6206	-69.77	kd	CGS001-5033	P4HA1	-			
6207	-69.82	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
6208	-69.84	kd	CGS001-290	ANPEP	Aminopeptidase N			
6209	-69.87	oe	ccsbBroad304_05098	MAGEB6	-			
6210	-69.9	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
6211	-69.9	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
6212	-69.91	kd	CGS001-54811	ZNF562	Zinc fingers, C2H2-type			
6213	-69.94	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
6214	-70.01	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
6215	-70.04	oe	ccsbBroad304_08511	RFK	-			
6216	-70.08	oe	ccsbBroad304_07124	UROD	-			
6217	-70.09	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
6218	-70.12	oe	ccsbBroad304_00222	CASP6	Caspases			
6219	-70.12	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6220	-70.14	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
6221	-70.16	kd	CGS001-3575	IL7R	IL-2 receptor family			
6222	-70.16	kd	CGS001-50604	IL20	Interleukins and interleukin receptors			
6223	-70.2	kd	CGS001-6446	SGK1	SGK family			
6224	-70.21	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
6225	-70.23	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
6226	-70.27	kd	CGS001-23196	FAM120A	-			
6227	-70.3	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
6228	-70.3	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
6229	-70.3	kd	CGS001-369	ARAF	RAF family			
6230	-70.33	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
6231	-70.34	kd	CGS001-55163	PNPO	-			
6232	-70.43	oe	ccsbBroad304_07548	TSSC4	-			
6233	-70.43	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
6234	-70.44	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
6235	-70.47	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
6236	-70.54	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
6237	-70.59	kd	CGS001-4436	MSH2	-			
6238	-70.61	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6239	-70.64	oe	ccsbBroad304_00210	CALR	-			
6240	-70.66	kd	CGS001-5744	PTHLH	Endogenous ligands			
6241	-70.78	oe	ccsbBroad304_07080	TM7SF2	-			
6242	-70.79	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
6243	-70.9	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
6244	-70.9	kd	CGS001-55206	SBNO1	-			
6245	-70.92	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
6246	-70.93	oe	ccsbBroad304_02218	IKBKE	IKK family			
6247	-70.94	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
6248	-70.97	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
6249	-71.04	oe	ccsbBroad304_03570	QRSL1	-			
6250	-71.09	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
6251	-71.11	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
6252	-71.13	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
6253	-71.13	kd	CGS001-9761	MLEC	-			
6254	-71.16	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
6255	-71.18	oe	ccsbBroad304_01654	TCTA	-			
6256	-71.18	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
6257	-71.26	kd	CGS001-2872	MKNK2	MKN subfamily			
6258	-71.27	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6259	-71.31	kd	CGS001-1198	CLK3	CDC-like kinases			
6260	-71.39	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
6261	-71.42	kd	CGS001-3033	HADH	-			
6262	-71.47	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
6263	-71.47	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
6264	-71.47	kd	CGS001-50813	COPS7A	-			
6265	-71.52	kd	CGS001-7172	TPMT	-			
6266	-71.56	oe	ccsbBroad304_00961	SMAD2	SMADs			
6267	-71.56	oe	ccsbBroad304_06287	GM2A	-			
6268	-71.6	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
6269	-71.65	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
6270	-71.66	kd	CGS001-1859	DYRK1A	Dyrk1 subfamily			
6271	-71.68	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
6272	-71.73	oe	ccsbBroad304_00510	EPHX2	-			
6273	-71.73	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
6274	-71.76	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
6275	-71.76	oe	ccsbBroad304_00491	EIF4EBP2	-			
6276	-71.78	kd	CGS001-602	BCL3	Ankyrin repeat domain containing			
6277	-71.85	kd	CGS001-4926	NUMA1	-			
6278	-71.86	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
6279	-71.91	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6280	-71.91	kd	CGS001-6886	TAL1	Basic helix-loop-helix proteins			
6281	-72.03	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
6282	-72.04	oe	ccsbBroad304_06133	TOR1A	-			
6283	-72.05	oe	ccsbBroad304_10230	STK19	G11 family			
6284	-72.07	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
6285	-72.11	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
6286	-72.14	kd	CGS001-51460	SFMBT1	Sterile alpha motif (SAM) domain containing			
6287	-72.15	oe	ccsbBroad304_00549	FDX1	-			
6288	-72.18	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6289	-72.22	kd	CGS001-124626	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6290	-72.26	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
6291	-72.26	kd	CGS001-8027	STAM	-			
6292	-72.34	kd	CGS001-847	CAT	-			
6293	-72.37	kd	CGS001-5810	RAD1	-			
6294	-72.37	kd	CGS001-121549	ASCL4	Basic helix-loop-helix proteins			
6295	-72.38	cc		Proteasome inhibitor	-			
6296	-72.38	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6297	-72.43	oe	ccsbBroad304_02175	MAGED1	-			
6298	-72.43	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
6299	-72.46	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
6300	-72.55	cc		Supressors of cytokine signaling GOF	-			
6301	-72.55	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6302	-72.62	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
6303	-72.67	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
6304	-72.67	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
6305	-72.68	kd	CGS001-51174	TUBD1	Tubulins			
6306	-72.72	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
6307	-72.72	kd	CGS001-23081	KDM4C	Histone demethylases			
6308	-72.76	kd	CGS001-2274	FHL2	-			
6309	-72.79	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
6310	-72.82	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
6311	-72.83	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
6312	-72.88	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
6313	-72.91	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
6314	-72.93	oe	ccsbBroad304_02955	MYCBP	-			
6315	-72.93	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
6316	-72.93	kd	CGS001-11044	PAPD7	-			
6317	-72.96	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6318	-73	kd	CGS001-10888	GPR83	GPCR / Class A : Orphans			
6319	-73	kd	CGS001-1147	CHUK	IKK family			
6320	-73.01	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
6321	-73.08	kd	CGS001-116931	MED12L	-			
6322	-73.14	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
6323	-73.15	oe	ccsbBroad304_05887	CFB	Complement system			
6324	-73.17	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
6325	-73.18	cc		Integrin subunits alpha LOF	-			
6326	-73.23	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
6327	-73.24	kd	CGS001-3559	IL2RA	IL-2 receptor family			
6328	-73.35	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
6329	-73.37	kd	CGS001-23338	PHF15	-			
6330	-73.37	oe	ccsbBroad304_05936	CASP2	Caspases			
6331	-73.38	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
6332	-73.42	kd	CGS001-111	ADCY5	Adenylate cyclases			
6333	-73.44	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
6334	-73.44	kd	CGS001-1376	CPT2	-			
6335	-73.46	oe	ccsbBroad304_02677	PDAP1	-			
6336	-73.47	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
6337	-73.48	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
6338	-73.51	kd	CGS001-9851	KIAA0753	-			
6339	-73.57	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
6340	-73.59	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
6341	-73.6	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
6342	-73.6	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
6343	-73.71	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
6344	-73.74	oe	ccsbBroad304_05821	ANXA1	Annexins			
6345	-73.77	cp	BRD-K41051431	mecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6346	-73.81	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
6347	-73.84	kd	CGS001-7247	TSN	-			
6348	-73.85	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
6349	-73.86	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
6350	-73.91	oe	ccsbBroad304_01930	CUL2	-			
6351	-73.95	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
6352	-73.95	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
6353	-73.99	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6354	-73.99	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
6355	-74.01	kd	CGS001-2115	ETV1	ETS Transcription Factors			
6356	-74.03	oe	ccsbBroad304_00652	GNAS	-			
6357	-74.03	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
6358	-74.09	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
6359	-74.1	oe	ccsbBroad304_05980	CDKN1B	-			
6360	-74.1	kd	CGS001-775	CACNA1C	Calcium channel subunits			
6361	-74.12	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
6362	-74.15	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
6363	-74.15	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
6364	-74.22	kd	CGS001-1675	CFD	Complement system			
6365	-74.3	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
6366	-74.34	oe	ccsbBroad304_03554	NAT10	-			
6367	-74.34	kd	CGS001-2849	GPR26	GPCR / Class A : Orphans			
6368	-74.36	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
6369	-74.41	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
6370	-74.42	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
6371	-74.46	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6372	-74.5	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
6373	-74.51	cp	BRD-K23369905	oxiconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6374	-74.54	oe	ccsbBroad304_02569	BTG3	-			
6375	-74.61	kd	CGS001-80237	ELL3	-			
6376	-74.67	kd	CGS001-966	CD59	CD molecules			
6377	-74.68	kd	CGS001-4522	MTHFD1	-			
6378	-74.72	cc		Kruppel like transcription factors LOF	-			
6379	-74.73	oe	ccsbBroad304_06103	DMD	-			
6380	-74.74	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
6381	-74.75	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
6382	-74.8	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
6383	-74.8	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
6384	-74.83	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
6385	-74.88	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
6386	-74.9	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
6387	-74.97	oe	ccsbBroad304_06639	NFYB	-			
6388	-74.98	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
6389	-75.01	kd	CGS001-8714	ABCC3	ATP binding cassette transporters / subfamily C			
6390	-75.03	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
6391	-75.06	oe	ccsbBroad304_06066	CTSL1	-			
6392	-75.07	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
6393	-75.11	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
6394	-75.12	kd	CGS001-3673	ITGA2	Integrins			
6395	-75.14	oe	ccsbBroad304_02298	DNM1L	-			
6396	-75.2	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
6397	-75.2	kd	CGS001-79109	MAPKAP1	-			
6398	-75.22	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
6399	-75.22	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6400	-75.23	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
6401	-75.23	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
6402	-75.26	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
6403	-75.3	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
6404	-75.31	kd	CGS001-2863	GPR39	GPCR / Class A : Orphans			
6405	-75.32	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
6406	-75.34	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
6407	-75.34	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
6408	-75.34	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
6409	-75.37	kd	CGS001-114609	TIRAP	-			
6410	-75.38	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
6411	-75.46	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
6412	-75.46	kd	CGS001-663	BNIP2	-			
6413	-75.47	oe	ccsbBroad304_01184	PGK1	-			
6414	-75.47	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
6415	-75.48	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6416	-75.53	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
6417	-75.55	kd	CGS001-10857	PGRMC1	-			
6418	-75.59	kd	CGS001-400	ARL1	ADP-ribosylation factors			
6419	-75.62	kd	CGS001-23365	ARHGEF12	Rho guanine nucleotide exchange factors			
6420	-75.79	oe	ccsbBroad304_01351	PEX19	-			
6421	-75.8	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
6422	-75.86	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
6423	-75.87	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
6424	-75.92	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
6425	-75.94	cp	BRD-A02189320	met-leu-phe	-666			-666
6426	-75.95	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6427	-76.02	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6428	-76.04	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
6429	-76.1	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
6430	-76.12	kd	CGS001-3281	HSBP1	-			
6431	-76.13	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
6432	-76.13	kd	CGS001-9143	SYNGR3	-			
6433	-76.17	kd	CGS001-54536	EXOC6	-			
6434	-76.21	kd	CGS001-7477	WNT7B	Endogenous ligands			
6435	-76.24	kd	CGS001-6857	SYT1	Synaptotagmins			
6436	-76.29	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
6437	-76.32	kd	CGS001-7913	DEK	-			
6438	-76.33	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
6439	-76.34	kd	CGS001-54490	UGT2B28	UDP glucuronosyltransferases			
6440	-76.35	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
6441	-76.43	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
6442	-76.45	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
6443	-76.5	oe	ccsbBroad304_04752	IKBIP	-			
6444	-76.59	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
6445	-76.6	kd	CGS001-6387	CXCL12	Endogenous ligands			
6446	-76.64	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
6447	-76.65	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
6448	-76.67	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
6449	-76.72	kd	CGS001-8942	KYNU	-			
6450	-76.73	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
6451	-76.77	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
6452	-76.79	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
6453	-76.79	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
6454	-76.88	oe	ccsbBroad304_00237	CCND3	-			
6455	-76.92	kd	CGS001-22832	KIAA1009	-			
6456	-76.93	kd	CGS001-11157	LSM6	-			
6457	-76.95	cp	BRD-K49481516	galantamine	Acetylcholinesterase inhibitor		ACHE, BCHE, CHRNA1, CHRNA10, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNA9, CHRNB1, CHRNB2, CHRNB3, CHRNB4, CHRND, CHRNE, CHRNG	Acetylcholinesterase inhibitor
6458	-76.95	kd	CGS001-387	RHOA	-			
6459	-76.96	cc		PARP inhibitor	-			
6460	-76.98	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
6461	-77	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
6462	-77.03	oe	ccsbBroad304_07320	SQSTM1	-			
6463	-77.07	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
6464	-77.24	kd	CGS001-475	ATOX1	-			
6465	-77.26	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
6466	-77.27	oe	ccsbBroad304_09578	PASD1	-			
6467	-77.28	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
6468	-77.28	oe	ccsbBroad304_04465	RERG	-			
6469	-77.32	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
6470	-77.33	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
6471	-77.33	oe	ccsbBroad304_00817	IDH2	-			
6472	-77.38	kd	CGS001-4637	MYL6	EF-hand domain containing			
6473	-77.42	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
6474	-77.44	oe	ccsbBroad304_08137	HOOK2	-			
6475	-77.48	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
6476	-77.61	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
6477	-77.66	kd	CGS001-7358	UGDH	-			
6478	-77.75	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
6479	-77.78	cp	BRD-K98493452	honokiol	AKT inhibitor		ALOX5, PTGS1, PTGS2	AKT inhibitor
6480	-77.78	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
6481	-77.78	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
6482	-77.83	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
6483	-77.84	oe	ccsbBroad304_07466	VGLL4	-			
6484	-77.88	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
6485	-77.89	kd	CGS001-6271	S100A1	EF-hand domain containing			
6486	-77.91	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
6487	-77.91	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6488	-77.93	oe	ccsbBroad304_06172	EPS8	-			
6489	-77.94	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
6490	-77.96	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
6491	-78	kd	CGS001-340371	NRBP2	NRBP family			
6492	-78.04	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
6493	-78.04	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
6494	-78.1	cp	BRD-A68888262	azelastine	Histamine receptor antagonist		HRH1, CYP2C19	Histamine receptor antagonist
6495	-78.19	oe	ccsbBroad304_03732	NPDC1	-			
6496	-78.37	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
6497	-78.38	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
6498	-78.41	oe	ccsbBroad304_05439	O3FAR1	-			
6499	-78.43	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
6500	-78.43	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
6501	-78.55	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6502	-78.59	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
6503	-78.61	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6504	-78.63	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
6505	-78.7	kd	CGS001-3149	HMGB3	High-mobility group / Canonical			
6506	-78.71	oe	ccsbBroad304_01152	PCNA	-			
6507	-78.77	oe	ccsbBroad304_01166	PDK2	PDHK family			
6508	-78.79	kd	CGS001-1855	DVL1	Dishevelled homologs			
6509	-78.84	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
6510	-78.86	cp	BRD-A80383043	BRD-A80383043	Glutamate receptor agonist		GRM1, GRM2	Glutamate receptor agonist, Glutamate receptor antagonist
6511	-78.88	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
6512	-78.88	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
6513	-78.91	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
6514	-78.94	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
6515	-78.94	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
6516	-78.97	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
6517	-79.03	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
6518	-79.03	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
6519	-79.11	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
6520	-79.11	kd	CGS001-57167	SALL4	Zinc fingers, C2H2-type			
6521	-79.18	kd	CGS001-6670	SP3	Specificity protein transcription factors			
6522	-79.2	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
6523	-79.24	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
6524	-79.26	oe	ccsbBroad304_02838	SDF2L1	-			
6525	-79.3	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6526	-79.35	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
6527	-79.38	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
6528	-79.39	kd	CGS001-6646	SOAT1	-			
6529	-79.45	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6530	-79.46	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
6531	-79.47	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
6532	-79.5	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
6533	-79.55	cc		Cyclooxygenase inhibitor	-			
6534	-79.58	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
6535	-79.61	kd	CGS001-6421	SFPQ	RNA binding motif (RRM) containing			
6536	-79.64	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
6537	-79.68	kd	CGS001-23075	SWAP70	EF-hand domain containing			
6538	-79.7	kd	CGS001-6272	SORT1	-			
6539	-79.72	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
6540	-79.76	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
6541	-79.78	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
6542	-79.83	oe	ccsbBroad304_07923	LSM5	-			
6543	-79.86	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
6544	-79.87	cp	BRD-K19462402	buflomedil	Adrenergic receptor antagonist		CACNA1C	Adrenergic receptor antagonist, Calcium channel blocker
6545	-79.87	kd	CGS001-64786	TBC1D15	-			
6546	-79.87	kd	CGS001-3988	LIPA	-			
6547	-79.93	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
6548	-80.03	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6549	-80.05	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
6550	-80.06	kd	CGS001-677	ZFP36L1	RING-type (C3HC4) zinc fingers			
6551	-80.08	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
6552	-80.15	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
6553	-80.19	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
6554	-80.26	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
6555	-80.28	kd	CGS001-10437	IFI30	-			
6556	-80.3	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
6557	-80.3	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
6558	-80.33	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
6559	-80.35	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
6560	-80.39	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
6561	-80.48	oe	ccsbBroad304_01845	RDBP	-			
6562	-80.52	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
6563	-80.57	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
6564	-80.59	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
6565	-80.69	oe	ccsbBroad304_00854	IL8	-			
6566	-80.71	kd	CGS001-433	ASGR2	C-type lectin domain containing			
6567	-80.73	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
6568	-80.73	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
6569	-80.75	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
6570	-80.76	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6571	-80.77	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
6572	-80.78	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
6573	-80.78	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6574	-80.8	kd	CGS001-25989	ULK3	Unc-51-like kinase (ULK) family			
6575	-80.82	kd	CGS001-3832	KIF11	Kinesins			
6576	-80.84	kd	CGS001-122618	PLD4	-			
6577	-80.84	kd	CGS001-57721	METTL14	-			
6578	-80.9	kd	CGS001-10460	TACC3	-			
6579	-80.93	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
6580	-80.98	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
6581	-81.04	kd	CGS001-6774	STAT3	SH2 domain containing			
6582	-81.05	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
6583	-81.08	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
6584	-81.08	kd	CGS001-112812	FDX1L	-			
6585	-81.1	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
6586	-81.11	kd	CGS001-25824	PRDX5	-			
6587	-81.13	kd	CGS001-301	ANXA1	Annexins			
6588	-81.14	kd	CGS001-22	ABCB7	ATP binding cassette transporters / subfamily B			
6589	-81.16	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
6590	-81.19	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
6591	-81.19	oe	ccsbBroad304_01052	MYB	-			
6592	-81.25	kd	CGS001-9337	CNOT8	-			
6593	-81.3	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
6594	-81.34	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
6595	-81.34	kd	CGS001-55379	LRRC59	-			
6596	-81.35	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
6597	-81.37	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
6598	-81.37	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
6599	-81.39	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
6600	-81.41	cc		Angiotensin receptor antagonist	-			
6601	-81.42	oe	ccsbBroad304_00492	EIF5A	-			
6602	-81.45	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
6603	-81.5	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
6604	-81.5	kd	CGS001-1399	CRKL	SH2 domain containing			
6605	-81.51	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
6606	-81.53	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
6607	-81.53	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
6608	-81.79	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
6609	-81.82	kd	CGS001-9641	IKBKE	IKK family			
6610	-81.85	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
6611	-81.87	kd	CGS001-8893	EIF2B5	-			
6612	-81.88	kd	CGS001-7292	TNFSF4	CD molecules			
6613	-81.98	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
6614	-82.06	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
6615	-82.08	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6616	-82.09	kd	CGS001-31	ACACA	Carboxylases			
6617	-82.18	kd	CGS001-572	BAD	-			
6618	-82.19	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
6619	-82.2	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
6620	-82.32	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
6621	-82.33	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
6622	-82.35	kd	CGS001-8678	BECN1	-			
6623	-82.38	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
6624	-82.44	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
6625	-82.46	kd	CGS001-3992	FADS1	Fatty acid desaturases			
6626	-82.49	cc		Imidazoline ligand	-			
6627	-82.49	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
6628	-82.49	kd	CGS001-29947	DNMT3L	-			
6629	-82.51	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
6630	-82.52	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
6631	-82.55	kd	CGS001-125950	RAVER1	RNA binding motif (RRM) containing			
6632	-82.57	kd	CGS001-4967	OGDH	-			
6633	-82.61	cp	BRD-A88254928	salbutamol	Adrenergic receptor agonist		ADRB2, ADRB1	Adrenergic receptor agonist
6634	-82.66	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
6635	-82.69	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
6636	-82.71	oe	ccsbBroad304_02919	KIAA1279	-			
6637	-82.71	oe	ccsbBroad304_00645	GCLM	-			
6638	-82.72	oe	ccsbBroad304_07887	GCAT	-			
6639	-82.74	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6640	-82.76	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
6641	-82.77	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
6642	-82.78	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
6643	-82.78	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
6644	-82.81	kd	CGS001-151306	GPBAR1	Bile acid receptor			
6645	-82.83	cp	BRD-K10961822	latanoprost	Prostanoid receptor agonist		PTGFR	Prostanoid receptor agonist
6646	-82.83	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
6647	-82.86	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
6648	-82.87	kd	CGS001-130497	OSR1	Zinc fingers, C2H2-type			
6649	-82.9	cp	BRD-K86887724	dofetilide	Potassium channel blocker		KCNH2, KCNH1, KCNJ12, KCNK2	Potassium channel blocker
6650	-82.91	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
6651	-82.97	kd	CGS001-7251	TSG101	-			
6652	-83	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
6653	-83.01	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
6654	-83.03	kd	CGS001-9467	SH3BP5	-			
6655	-83.05	kd	CGS001-6303	SAT1	-			
6656	-83.06	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
6657	-83.08	oe	ccsbBroad304_00987	MCM3	-			
6658	-83.09	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
6659	-83.09	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
6660	-83.09	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
6661	-83.11	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
6662	-83.16	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
6663	-83.18	kd	CGS001-11230	PRAF2	-			
6664	-83.19	oe	ccsbBroad304_04202	MED28	-			
6665	-83.2	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
6666	-83.23	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
6667	-83.31	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
6668	-83.35	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
6669	-83.44	kd	CGS001-2931	GSK3A	GSK subfamily			
6670	-83.46	cp	BRD-K90733503	cefalexin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6671	-83.48	oe	ccsbBroad304_13998	PDXK	-			
6672	-83.48	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6673	-83.5	kd	CGS001-8935	SKAP2	Pleckstrin homology (PH) domain containing			
6674	-83.51	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
6675	-83.51	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
6676	-83.58	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
6677	-83.59	oe	ccsbBroad304_00116	ASS1	-			
6678	-83.59	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
6679	-83.62	kd	CGS001-7764	ZNF217	Zinc fingers, C2H2-type			
6680	-83.63	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
6681	-83.65	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
6682	-83.67	kd	CGS001-7466	WFS1	-			
6683	-83.7	kd	CGS001-29775	CARD10	-			
6684	-83.75	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6685	-83.77	kd	CGS001-26271	FBXO5	F-boxes / other			
6686	-83.82	kd	CGS001-831	CAST	-			
6687	-83.83	kd	CGS001-90861	HN1L	-			
6688	-83.86	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
6689	-83.87	kd	CGS001-26227	PHGDH	-			
6690	-83.9	oe	ccsbBroad304_02956	EHF	-			
6691	-83.91	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
6692	-83.93	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
6693	-83.93	kd	CGS001-26191	PTPN22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6694	-83.93	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
6695	-83.97	kd	CGS001-1119	CHKA	-			
6696	-83.98	kd	CGS001-64223	MLST8	WD repeat domain containing			
6697	-84.02	cc		Bacterial 30S ribosomal subunit inhibitor	-			
6698	-84.07	kd	CGS001-3476	IGBP1	-			
6699	-84.09	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
6700	-84.13	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
6701	-84.15	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
6702	-84.25	kd	CGS001-6491	STIL	-			
6703	-84.27	cp	BRD-K46435977	valaciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
6704	-84.27	kd	CGS001-57215	THAP11	THAP (C2CH-type zinc finger) domain containing			
6705	-84.29	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
6706	-84.32	cp	BRD-K65910366	KUC103904N	-666			-666
6707	-84.33	kd	CGS001-64422	ATG3	-			
6708	-84.34	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
6709	-84.38	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6710	-84.4	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
6711	-84.43	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
6712	-84.44	kd	CGS001-4709	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6713	-84.45	kd	CGS001-6520	SLC3A2	SLC3 family			
6714	-84.46	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
6715	-84.55	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
6716	-84.56	kd	CGS001-1027	CDKN1B	-			
6717	-84.57	kd	CGS001-8914	TIMELESS	-			
6718	-84.59	oe	ccsbBroad304_02458	STK25	YSK subfamily			
6719	-84.6	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
6720	-84.6	kd	CGS001-2781	GNAZ	-			
6721	-84.62	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
6722	-84.66	oe	ccsbBroad304_00249	CD14	CD molecules			
6723	-84.68	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6724	-84.7	kd	CGS001-324	APC	Armadillo repeat containing			
6725	-84.73	kd	CGS001-3420	IDH3B	-			
6726	-84.79	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
6727	-84.8	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
6728	-84.8	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
6729	-84.81	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
6730	-84.91	kd	CGS001-4931	NVL	ATPases / AAA-type			
6731	-84.92	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
6732	-84.93	kd	CGS001-114785	MBD6	-			
6733	-84.93	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
6734	-84.94	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
6735	-84.96	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
6736	-84.98	oe	ccsbBroad304_03119	C16ORF5	-			
6737	-85.01	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
6738	-85.07	kd	CGS001-9929	JOSD1	-			
6739	-85.08	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
6740	-85.08	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6741	-85.09	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
6742	-85.11	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
6743	-85.13	oe	ccsbBroad304_01618	STXBP1	-			
6744	-85.14	kd	CGS001-3242	HPD	Oxidoreductases			
6745	-85.15	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
6746	-85.17	kd	CGS001-23549	DNPEP	Aminopeptidase I			
6747	-85.2	oe	ccsbBroad304_01855	NCOA4	-			
6748	-85.23	kd	CGS001-5901	RAN	-			
6749	-85.25	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
6750	-85.27	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
6751	-85.28	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
6752	-85.31	kd	CGS001-2023	ENO1	-			
6753	-85.33	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
6754	-85.34	oe	ccsbBroad304_03798	PHTF2	-			
6755	-85.34	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
6756	-85.37	kd	CGS001-5054	SERPINE1	Serine (or cysteine) peptidase inhibitors			
6757	-85.39	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6758	-85.4	kd	CGS001-5927	KDM5A	Histone demethylases			
6759	-85.44	oe	ccsbBroad304_02370	HRSP12	-			
6760	-85.49	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
6761	-85.5	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
6762	-85.51	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
6763	-85.53	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
6764	-85.53	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
6765	-85.59	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
6766	-85.59	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
6767	-85.61	oe	ccsbBroad304_00518	ETFA	-			
6768	-85.7	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
6769	-85.73	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
6770	-85.75	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
6771	-85.76	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
6772	-85.77	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
6773	-85.77	kd	CGS001-5073	PARN	-			
6774	-85.79	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
6775	-85.8	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
6776	-85.81	oe	ccsbBroad304_01658	PRDX2	-			
6777	-85.83	cc		HIF activator	-			
6778	-85.83	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
6779	-85.83	kd	CGS001-50846	DHH	-			
6780	-85.84	kd	CGS001-5879	RAC1	Endogenous ligands			
6781	-85.84	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
6782	-85.86	oe	ccsbBroad304_06178	ERCC5	-			
6783	-85.89	cc		Phospholipases LOF	-			
6784	-85.9	kd	CGS001-3298	HSF2	-			
6785	-85.93	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
6786	-85.96	kd	CGS001-6767	ST13	Tetratricopeptide (TTC) repeat domain containing			
6787	-86	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
6788	-86.01	kd	CGS001-79073	TMEM109	-			
6789	-86.03	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
6790	-86.03	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
6791	-86.06	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
6792	-86.09	kd	CGS001-1026	CDKN1A	-			
6793	-86.1	kd	CGS001-991	CDC20	WD repeat domain containing			
6794	-86.12	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
6795	-86.12	kd	CGS001-3572	IL6ST	IL-6 receptor family			
6796	-86.13	cc		Structural maintenance of chromosomes proteins LOF	-			
6797	-86.13	oe	ccsbBroad304_01593	SRP14	-			
6798	-86.15	oe	ccsbBroad304_07922	TRIM29	-			
6799	-86.15	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
6800	-86.24	oe	ccsbBroad304_06126	TSC22D3	-			
6801	-86.25	kd	CGS001-5932	RBBP8	-			
6802	-86.25	kd	CGS001-4552	MTRR	-			
6803	-86.27	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
6804	-86.29	kd	CGS001-84890	ADO	-			
6805	-86.31	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
6806	-86.32	oe	ccsbBroad304_00100	RHOA	-			
6807	-86.33	kd	CGS001-199704	ZNF585A	Zinc fingers, C2H2-type			
6808	-86.35	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
6809	-86.37	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
6810	-86.37	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
6811	-86.37	kd	CGS001-899	CCNF	F-boxes / other			
6812	-86.38	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
6813	-86.4	kd	CGS001-9020	MAP3K14	MAPKKK:STE-unique family			
6814	-86.41	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
6815	-86.43	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
6816	-86.43	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
6817	-86.47	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
6818	-86.49	kd	CGS001-2172	FABP6	Fatty acid binding protein family			
6819	-86.58	kd	CGS001-955	ENTPD6	-			
6820	-86.61	kd	CGS001-7052	TGM2	Transglutaminases			
6821	-86.65	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
6822	-86.68	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
6823	-86.68	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
6824	-86.7	oe	ccsbBroad304_01748	UFD1L	-			
6825	-86.7	kd	CGS001-9712	USP6NL	-			
6826	-86.78	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
6827	-86.79	kd	CGS001-8220	DGCR14	-			
6828	-86.82	oe	ccsbBroad304_00250	CD19	CD molecules			
6829	-86.82	kd	CGS001-1875	E2F5	-			
6830	-86.84	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
6831	-86.85	kd	CGS001-4610	MYCL1	-			
6832	-86.92	cp	BRD-K92870997	pterostilbene	Cyclooxygenase inhibitor		FAAH, PPARA, PTGS1, PTGS2	Cyclooxygenase inhibitor, PPAR receptor agonist
6833	-86.92	kd	CGS001-57048	PLSCR3	-			
6834	-87	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
6835	-87	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
6836	-87.07	kd	CGS001-10131	TRAP1	Heat shock proteins / HSPC			
6837	-87.13	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
6838	-87.13	kd	CGS001-11182	SLC2A6	Solute carriers			
6839	-87.17	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
6840	-87.18	cp	BRD-K88701661	dimercaptosuccinic-acid	Chelating agent		DNMT1	Chelating agent
6841	-87.2	cp	BRD-K66206289	lobeline	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist
6842	-87.27	cp	BRD-A00520476	otenzepad	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6843	-87.29	oe	ccsbBroad304_07861	COBL	-			
6844	-87.29	oe	ccsbBroad304_00600	FYN	Src family			
6845	-87.29	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
6846	-87.3	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6847	-87.31	oe	ccsbBroad304_00515	ERH	-			
6848	-87.34	oe	ccsbBroad304_07800	EXOSC8	-			
6849	-87.37	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
6850	-87.39	kd	CGS001-29946	SERTAD3	-			
6851	-87.43	kd	CGS001-10174	SORBS3	-			
6852	-87.47	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6853	-87.48	oe	ccsbBroad304_07834	GGA2	-			
6854	-87.5	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
6855	-87.57	kd	CGS001-51053	GMNN	-			
6856	-87.59	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
6857	-87.63	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
6858	-87.65	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6859	-87.69	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
6860	-87.7	kd	CGS001-5111	PCNA	-			
6861	-87.74	cp	BRD-K39621635	artemether	Antimalarial		ATP1A1, CYP2B6, CYP2C19, CYP3A5	Antimalarial
6862	-87.76	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
6863	-87.8	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
6864	-87.81	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
6865	-87.82	kd	CGS001-5144	PDE4D	Phosphodiesterases			
6866	-87.82	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
6867	-87.87	oe	ccsbBroad304_00551	FECH	-			
6868	-87.89	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
6869	-87.9	kd	CGS001-5576	PRKAR2A	Protein kinase A			
6870	-87.92	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
6871	-87.92	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
6872	-87.96	kd	CGS001-2944	GSTM1	Glutathione S-transferases / Soluble			
6873	-87.98	oe	ccsbBroad304_00174	BRAF	RAF family			
6874	-88.04	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
6875	-88.05	oe	ccsbBroad304_00648	GLRX	-			
6876	-88.06	kd	CGS001-94103	ORMDL3	-			
6877	-88.07	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
6878	-88.1	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
6879	-88.12	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
6880	-88.12	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6881	-88.15	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
6882	-88.15	kd	CGS001-54584	GNB1L	WD repeat domain containing			
6883	-88.16	kd	CGS001-678	ZFP36L2	RING-type (C3HC4) zinc fingers			
6884	-88.22	cc		Canonical high mobility group proteins LOF	-			
6885	-88.27	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
6886	-88.27	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
6887	-88.29	kd	CGS001-9308	CD83	CD molecules			
6888	-88.33	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
6889	-88.34	kd	CGS001-9805	SCRN1	-			
6890	-88.37	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
6891	-88.41	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
6892	-88.42	kd	CGS001-4439	MSH5	-			
6893	-88.46	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
6894	-88.46	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
6895	-88.47	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
6896	-88.49	kd	CGS001-55620	STAP2	-			
6897	-88.52	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6898	-88.54	oe	ccsbBroad304_03232	VPS28	-			
6899	-88.54	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
6900	-88.56	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
6901	-88.56	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
6902	-88.59	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
6903	-88.63	kd	CGS001-8334	HIST1H2AC	Histones / Replication-dependent			
6904	-88.64	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
6905	-88.67	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
6906	-88.67	kd	CGS001-7444	VRK2	Vaccina related kinase (VRK) family			
6907	-88.69	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
6908	-88.71	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6909	-88.71	kd	CGS001-6741	SSB	La ribonucleoprotein domain containing			
6910	-88.78	oe	ccsbBroad304_00832	IFNB1	Interferons			
6911	-88.78	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
6912	-88.78	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
6913	-88.85	kd	CGS001-23102	TBC1D2B	-			
6914	-88.86	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
6915	-88.87	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
6916	-88.88	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
6917	-88.88	kd	CGS001-673	BRAF	RAF family			
6918	-88.92	oe	ccsbBroad304_06739	PLOD1	-			
6919	-88.92	kd	CGS001-345611	IRGM	-			
6920	-88.97	kd	CGS001-3685	ITGAV	Integrins			
6921	-89	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6922	-89.06	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
6923	-89.06	kd	CGS001-51466	EVL	-			
6924	-89.07	kd	CGS001-54861	SNRK	SNRK subfamily			
6925	-89.14	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
6926	-89.21	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
6927	-89.23	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
6928	-89.24	oe	ccsbBroad304_07889	QPRT	-			
6929	-89.24	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
6930	-89.24	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
6931	-89.25	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
6932	-89.29	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
6933	-89.29	cp	BRD-K13800121	parecoxib	Cyclooxygenase inhibitor		LTF, PTGS2	Cyclooxygenase inhibitor
6934	-89.31	kd	CGS001-3034	HAL	-			
6935	-89.32	cc		IKK inhibitor	-			
6936	-89.33	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
6937	-89.33	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
6938	-89.33	kd	CGS001-79921	TCEAL4	-			
6939	-89.36	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
6940	-89.37	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6941	-89.38	kd	CGS001-6721	SREBF2	Basic helix-loop-helix proteins			
6942	-89.39	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6943	-89.42	kd	CGS001-4087	SMAD2	SMADs			
6944	-89.43	oe	ccsbBroad304_01327	PSPH	-			
6945	-89.49	cp	BRD-K22947005	dexbrompheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6946	-89.49	kd	CGS001-5723	PSPH	-			
6947	-89.5	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
6948	-89.51	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6949	-89.53	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
6950	-89.55	oe	ccsbBroad304_09095	PUS7L	-			
6951	-89.57	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
6952	-89.64	kd	CGS001-5105	PCK1	-			
6953	-89.64	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
6954	-89.7	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
6955	-89.78	kd	CGS001-8741	TNFSF13	CD molecules			
6956	-89.78	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
6957	-89.83	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
6958	-89.84	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
6959	-89.85	kd	CGS001-9252	RPS6KA5	MSK subfamily			
6960	-89.93	kd	CGS001-5796	PTPRK	Receptor tyrosine phosphatases (RTP)			
6961	-89.96	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
6962	-89.97	kd	CGS001-226	ALDOA	-			
6963	-89.99	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
6964	-89.99	kd	CGS001-513	ATP5D	ATPases / F-type			
6965	-90.01	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
6966	-90.05	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
6967	-90.08	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
6968	-90.08	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
6969	-90.12	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
6970	-90.14	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
6971	-90.16	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
6972	-90.18	kd	CGS001-2182	ACSL4	Acyl-CoA synthetase family			
6973	-90.19	kd	CGS001-5422	POLA1	DNA polymerases			
6974	-90.2	kd	CGS001-2768	GNA12	-			
6975	-90.24	oe	ccsbBroad304_00789	HSBP1	-			
6976	-90.29	cc		T-type calcium channel blocker	-			
6977	-90.31	oe	ccsbBroad304_00212	CAMLG	-			
6978	-90.31	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
6979	-90.32	oe	ccsbBroad304_07511	KIF14	Kinesins			
6980	-90.33	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
6981	-90.33	kd	CGS001-55256	ADI1	-			
6982	-90.34	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
6983	-90.36	cp	BRD-K33312228	halometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6984	-90.38	kd	CGS001-10827	FAM114A2	-			
6985	-90.39	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
6986	-90.39	kd	CGS001-23678	SGK3	SGK family			
6987	-90.41	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
6988	-90.43	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
6989	-90.48	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
6990	-90.49	kd	CGS001-1488	CTBP2	-			
6991	-90.54	kd	CGS001-7128	TNFAIP3	OTU domain containing			
6992	-90.56	cp	BRD-K88304388	dextrorphan	Glutamate receptor antagonist		OPRM1, OPRK1, OPRD1, GRIN1, HTR1A, SLC6A2	Glutamate receptor antagonist
6993	-90.6	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
6994	-90.62	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
6995	-90.65	kd	CGS001-9813	KIAA0494	-			
6996	-90.66	kd	CGS001-1155	TBCB	-			
6997	-90.73	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
6998	-90.73	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
6999	-90.75	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
7000	-90.76	kd	CGS001-6909	TBX2	T-boxes			
7001	-90.77	kd	CGS001-51734	SEPX1	-			
7002	-90.77	kd	CGS001-283	ANG	Ribonucleases, RNase A			
7003	-90.78	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
7004	-90.79	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
7005	-90.8	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
7006	-90.82	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
7007	-90.85	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
7008	-90.89	kd	CGS001-330	BIRC3	Inhibitors of apoptosis (IAP) protein family			
7009	-90.9	kd	CGS001-6595	SMARCA2	Non-enzymatic BRD containing proteins			
7010	-90.91	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
7011	-91.02	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
7012	-91.03	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
7013	-91.05	cc		PKA inhibitor	-			
7014	-91.1	kd	CGS001-55176	SEC61A2	-			
7015	-91.13	oe	ccsbBroad304_08452	PIH1D1	-			
7016	-91.15	cp	BRD-K83144676	olmesartan	Angiotensin antagonist		AGTR1	Angiotensin antagonist
7017	-91.19	oe	ccsbBroad304_10240	CROT	-			
7018	-91.19	kd	CGS001-5696	PSMB8	Proteasome (prosome, macropain) subunits			
7019	-91.19	kd	CGS001-4077	NBR1	-			
7020	-91.2	oe	ccsbBroad304_06996	SRM	-			
7021	-91.21	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
7022	-91.22	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
7023	-91.23	kd	CGS001-2885	GRB2	SH2 domain containing			
7024	-91.31	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
7025	-91.35	kd	CGS001-1508	CTSB	Cathepsins			
7026	-91.36	kd	CGS001-55718	POLR3E	RNA polymerase subunits			
7027	-91.38	cc		Adenosine receptor agonist	-			
7028	-91.4	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
7029	-91.41	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
7030	-91.43	oe	ccsbBroad304_08152	PSAT1	-			
7031	-91.44	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
7032	-91.45	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
7033	-91.48	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
7034	-91.5	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
7035	-91.57	kd	CGS001-10447	FAM3C	-			
7036	-91.58	cc		NFkB pathway inhibitor	-			
7037	-91.61	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
7038	-91.62	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
7039	-91.67	kd	CGS001-10285	SMNDC1	Tudor domain containing			
7040	-91.67	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
7041	-91.71	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
7042	-91.72	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
7043	-91.72	kd	CGS001-51752	ERAP1	Aminopeptidase N			
7044	-91.73	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
7045	-91.75	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
7046	-91.75	kd	CGS001-2597	GAPDH	-			
7047	-91.79	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
7048	-91.8	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
7049	-91.83	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
7050	-91.83	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
7051	-91.85	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
7052	-91.86	kd	CGS001-9341	VAMP3	Vesicle-associated membrane proteins			
7053	-91.87	oe	ccsbBroad304_07178	ZFP112	-			
7054	-91.91	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
7055	-91.95	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
7056	-91.98	oe	ccsbBroad304_06538	LSP1	-			
7057	-92.02	cc		Purinergic receptors P2Y GOF	-			
7058	-92.06	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7059	-92.08	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
7060	-92.1	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
7061	-92.1	kd	CGS001-64858	DCLRE1B	-			
7062	-92.11	kd	CGS001-11136	SLC7A9	SLC7 family			
7063	-92.12	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
7064	-92.13	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
7065	-92.15	kd	CGS001-4938	OAS1	-			
7066	-92.2	kd	CGS001-6919	TCEA2	-			
7067	-92.23	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
7068	-92.25	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
7069	-92.25	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
7070	-92.27	cp	BRD-K84955386	hyperoside	Glucosidase inhibitor		ACE, AKR1B1, GAA	Glucosidase inhibitor
7071	-92.32	kd	CGS001-7480	WNT10B	Wingless-type MMTV integration sites			
7072	-92.34	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
7073	-92.34	kd	CGS001-4968	OGG1	-			
7074	-92.34	kd	CGS001-5608	MAP2K6	MAPKK:STE7 family			
7075	-92.35	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
7076	-92.36	oe	ccsbBroad304_02626	PKIG	-			
7077	-92.38	oe	ccsbBroad304_01933	TEAD2	-			
7078	-92.41	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
7079	-92.42	kd	CGS001-2961	GTF2E2	General transcription factors			
7080	-92.43	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
7081	-92.47	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
7082	-92.51	cp	BRD-A95696820	acadesine	AMPK activator			AMPK activator
7083	-92.52	oe	ccsbBroad304_09035	COASY	-			
7084	-92.53	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
7085	-92.54	cp	BRD-K96471533	nitazoxanide	Pyruvate ferredoxin oxidoreductase inhibitor			Pyruvate ferredoxin oxidoreductase inhibitor
7086	-92.55	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
7087	-92.56	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
7088	-92.57	oe	ccsbBroad304_02163	MED7	-			
7089	-92.61	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
7090	-92.62	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
7091	-92.65	kd	CGS001-5217	PFN2	-			
7092	-92.66	kd	CGS001-7345	UCHL1	Ubiquitin C-terminal hydrolase			
7093	-92.67	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
7094	-92.7	oe	ccsbBroad304_07018	SUPT5H	-			
7095	-92.71	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
7096	-92.71	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
7097	-92.72	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
7098	-92.73	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
7099	-92.74	cp	BRD-A16934955	nalbuphine	Opioid receptor agonist		OPRD1, OPRK1, OPRM1	Opioid receptor agonist, Opioid receptor antagonist
7100	-92.79	kd	CGS001-1949	EFNB3	Ephrins			
7101	-92.8	kd	CGS001-2752	GLUL	-			
7102	-92.82	kd	CGS001-23046	KIF21B	Kinesins			
7103	-92.85	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
7104	-92.86	kd	CGS001-6203	RPS9	S ribosomal proteins			
7105	-92.87	oe	ccsbBroad304_00841	IKBKB	IKK family			
7106	-92.87	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
7107	-92.87	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
7108	-92.88	cc		Glucocorticoid receptor agonist	-			
7109	-92.9	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
7110	-92.92	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
7111	-92.93	kd	CGS001-3329	HSPD1	Heat Shock Proteins / Chaperonins			
7112	-92.96	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
7113	-92.96	kd	CGS001-6418	SET	-			
7114	-92.96	kd	CGS001-6193	RPS5	S ribosomal proteins			
7115	-92.98	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
7116	-93.03	kd	CGS001-8891	EIF2B3	-			
7117	-93.05	kd	CGS001-1312	COMT	Catecholamine turnover			
7118	-93.09	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
7119	-93.09	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
7120	-93.1	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
7121	-93.11	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
7122	-93.12	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
7123	-93.12	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
7124	-93.13	kd	CGS001-5891	MOK	RCK family			
7125	-93.15	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
7126	-93.18	oe	ccsbBroad304_01577	SOD1	-			
7127	-93.19	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
7128	-93.2	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
7129	-93.2	kd	CGS001-2821	GPI	-			
7130	-93.25	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
7131	-93.25	kd	CGS001-3821	KLRC1	CD molecules			
7132	-93.33	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
7133	-93.33	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
7134	-93.34	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
7135	-93.35	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
7136	-93.37	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
7137	-93.37	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
7138	-93.38	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
7139	-93.39	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
7140	-93.39	kd	CGS001-10046	MAMLD1	-			
7141	-93.41	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
7142	-93.43	kd	CGS001-23211	ZC3H4	Zinc fingers, CCCH-type domain containing			
7143	-93.46	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
7144	-93.46	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
7145	-93.46	kd	CGS001-3066	HDAC2	Histone deacetylases			
7146	-93.49	kd	CGS001-1213	CLTC	-			
7147	-93.51	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
7148	-93.51	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
7149	-93.52	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
7150	-93.53	kd	CGS001-94234	FOXQ1	Forkhead boxes			
7151	-93.54	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
7152	-93.57	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
7153	-93.57	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
7154	-93.57	kd	CGS001-25937	WWTR1	Hippo Signaling			
7155	-93.58	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
7156	-93.6	cp	BRD-K88679075	methandriol	Androgenic steroid			Androgenic steroid
7157	-93.61	kd	CGS001-4664	NAB1	-			
7158	-93.63	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
7159	-93.64	kd	CGS001-8431	NR0B2	DAX-like receptors			
7160	-93.65	cc		Interleukins GOF	-			
7161	-93.65	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
7162	-93.67	kd	CGS001-65263	PYCRL	-			
7163	-93.68	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
7164	-93.7	kd	CGS001-390980	ZNF805	Zinc fingers, C2H2-type			
7165	-93.75	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
7166	-93.79	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
7167	-93.79	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
7168	-93.81	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
7169	-93.83	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
7170	-93.83	kd	CGS001-6591	SNAI2	Snail homologs			
7171	-93.84	kd	CGS001-112858	TP53RK	Bud32 family			
7172	-93.84	kd	CGS001-253260	RICTOR	-			
7173	-93.84	kd	CGS001-5515	PPP2CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
7174	-93.85	kd	CGS001-813	CALU	EF-hand domain containing			
7175	-93.91	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
7176	-93.92	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
7177	-93.92	kd	CGS001-2030	SLC29A1	SLC29 family			
7178	-93.94	kd	CGS001-2114	ETS2	ETS Transcription Factors			
7179	-93.95	oe	ccsbBroad304_00262	CD59	CD molecules			
7180	-93.96	kd	CGS001-1725	DHPS	-			
7181	-93.98	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
7182	-93.98	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
7183	-94.01	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
7184	-94.01	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
7185	-94.03	kd	CGS001-54915	YTHDF1	-			
7186	-94.04	kd	CGS001-5829	PXN	-			
7187	-94.05	kd	CGS001-79581	GPR172A	-			
7188	-94.06	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
7189	-94.07	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
7190	-94.08	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
7191	-94.12	kd	CGS001-5058	PAK1	PAKA subfamily			
7192	-94.13	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
7193	-94.15	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
7194	-94.15	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
7195	-94.16	kd	CGS001-3693	ITGB5	Integrins			
7196	-94.2	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
7197	-94.24	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
7198	-94.34	kd	CGS001-1727	CYB5R3	-			
7199	-94.35	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
7200	-94.35	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
7201	-94.36	cp	BRD-M41783010	acamprosate	Glutamate receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B, GRM5	Glutamate receptor antagonist
7202	-94.37	kd	CGS001-6256	RXRA	Retinoid X receptors			
7203	-94.38	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
7204	-94.4	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
7205	-94.42	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
7206	-94.43	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
7207	-94.43	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
7208	-94.44	kd	CGS001-10671	DCTN6	-			
7209	-94.49	cc		Serine proteases GOF	-			
7210	-94.49	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
7211	-94.49	kd	CGS001-10969	EBNA1BP2	-			
7212	-94.51	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
7213	-94.53	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
7214	-94.55	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
7215	-94.55	kd	CGS001-8826	IQGAP1	-			
7216	-94.56	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
7217	-94.56	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
7218	-94.61	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
7219	-94.62	kd	CGS001-55486	PARL	-			
7220	-94.63	kd	CGS001-6894	TARBP1	-			
7221	-94.63	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
7222	-94.64	kd	CGS001-7018	TF	-			
7223	-94.65	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
7224	-94.68	kd	CGS001-960	CD44	CD molecules			
7225	-94.71	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
7226	-94.77	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
7227	-94.8	oe	ccsbBroad304_04379	LZIC	-			
7228	-94.85	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
7229	-94.89	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
7230	-94.91	kd	CGS001-25888	ZNF473	Zinc fingers, C2H2-type			
7231	-94.92	kd	CGS001-55556	ENOSF1	-			
7232	-94.93	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
7233	-94.93	kd	CGS001-4043	LRPAP1	-			
7234	-95.02	kd	CGS001-84159	ARID5B	-			
7235	-95.03	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
7236	-95.03	kd	CGS001-10051	SMC4	Structural maintenance of chromosomes proteins			
7237	-95.04	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
7238	-95.04	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
7239	-95.05	oe	ccsbBroad304_04775	NTAN1	-			
7240	-95.09	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
7241	-95.1	kd	CGS001-10616	RBCK1	RING-type (C3HC4) zinc fingers			
7242	-95.1	kd	CGS001-4953	ODC1	Decarboxylases			
7243	-95.11	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
7244	-95.14	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
7245	-95.15	cp	BRD-K94649603	taxifolin	Opioid receptor antagonist		APOB, APP, HMGCR	Opioid receptor antagonist
7246	-95.17	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
7247	-95.17	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
7248	-95.18	oe	ccsbBroad304_08292	IP6K2	-			
7249	-95.19	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
7250	-95.19	kd	CGS001-2153	F5	Blood coagulation components			
7251	-95.25	kd	CGS001-2348	FOLR1	-			
7252	-95.27	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
7253	-95.28	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
7254	-95.28	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
7255	-95.3	kd	CGS001-3615	IMPDH2	Oxidoreductases			
7256	-95.31	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
7257	-95.31	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
7258	-95.33	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
7259	-95.34	oe	ccsbBroad304_06464	ITGB2	Integrins			
7260	-95.36	oe	ccsbBroad304_07401	TXNL1	-			
7261	-95.38	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
7262	-95.41	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
7263	-95.47	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
7264	-95.48	oe	ccsbBroad304_07754	FGFR1OP	-			
7265	-95.51	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
7266	-95.51	kd	CGS001-50	ACO2	-			
7267	-95.53	kd	CGS001-39	ACAT2	Lanosterol biosynthesis pathway			
7268	-95.54	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
7269	-95.56	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
7270	-95.56	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
7271	-95.57	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
7272	-95.57	kd	CGS001-2057	EPOR	Prolactin receptor family			
7273	-95.58	kd	CGS001-10254	STAM2	-			
7274	-95.59	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
7275	-95.59	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
7276	-95.59	kd	CGS001-22818	COPZ1	-			
7277	-95.61	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
7278	-95.63	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
7279	-95.64	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
7280	-95.64	kd	CGS001-79094	CHAC1	-			
7281	-95.65	kd	CGS001-23244	PDS5A	-			
7282	-95.66	kd	CGS001-805	CALM2	EF-hand domain containing			
7283	-95.68	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
7284	-95.68	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
7285	-95.68	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
7286	-95.69	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
7287	-95.69	cp	BRD-A12560204	nitrendipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1H, CACNA1S, CACNA2D2, CACNB2, CACNG1, KCNN4	Calcium channel blocker
7288	-95.69	kd	CGS001-6772	STAT1	SH2 domain containing			
7289	-95.71	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
7290	-95.71	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
7291	-95.71	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
7292	-95.72	kd	CGS001-116113	FOXP4	Forkhead boxes			
7293	-95.74	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
7294	-95.78	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
7295	-95.78	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
7296	-95.79	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
7297	-95.79	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
7298	-95.81	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
7299	-95.81	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
7300	-95.82	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
7301	-95.82	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
7302	-95.82	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
7303	-95.83	kd	CGS001-378	ARF4	ADP-ribosylation factors			
7304	-95.84	kd	CGS001-3226	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
7305	-95.85	kd	CGS001-8915	BCL10	-			
7306	-95.86	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
7307	-95.86	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
7308	-95.87	kd	CGS001-10950	BTG3	-			
7309	-95.88	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
7310	-95.91	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
7311	-95.92	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
7312	-95.92	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
7313	-95.94	cp	BRD-K60160658	tiagabine	GABA uptake inhibitor		SLC6A1, CYP2C19	GABA uptake inhibitor
7314	-95.94	kd	CGS001-2067	ERCC1	-			
7315	-95.94	kd	CGS001-818	CAMK2G	CAMK2 family			
7316	-95.95	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
7317	-95.98	kd	CGS001-11142	PKIG	-			
7318	-95.99	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
7319	-96	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
7320	-96	oe	ccsbBroad304_04534	HN1L	-			
7321	-96.01	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
7322	-96.01	cp	BRD-A75935363	atracurium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
7323	-96.01	kd	CGS001-4927	NUP88	-			
7324	-96.02	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
7325	-96.02	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
7326	-96.04	kd	CGS001-9697	TRAM2	-			
7327	-96.1	kd	CGS001-7832	BTG2	-			
7328	-96.11	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
7329	-96.11	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
7330	-96.12	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
7331	-96.12	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
7332	-96.13	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
7333	-96.14	kd	CGS001-4907	NT5E	Adenosine turnover			
7334	-96.15	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
7335	-96.15	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
7336	-96.17	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7337	-96.19	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
7338	-96.19	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
7339	-96.2	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
7340	-96.21	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
7341	-96.23	kd	CGS001-5096	PCCB	Carboxylases			
7342	-96.24	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
7343	-96.24	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
7344	-96.28	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
7345	-96.29	kd	CGS001-136	ADORA2B	GPCR / Class A : Adenosine receptors			
7346	-96.35	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
7347	-96.35	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7348	-96.39	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
7349	-96.42	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
7350	-96.42	cp	BRD-K73196317	urapidil	Adrenergic receptor antagonist		HTR1A	Adrenergic receptor antagonist
7351	-96.42	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
7352	-96.43	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
7353	-96.43	kd	CGS001-11333	PDAP1	-			
7354	-96.45	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
7355	-96.46	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
7356	-96.46	kd	CGS001-388	RHOB	-			
7357	-96.47	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
7358	-96.47	kd	CGS001-8313	AXIN2	-			
7359	-96.48	cp	BRD-K15519488	CS-110266	Dopamine receptor agonist		SLC6A3	Dopamine receptor agonist
7360	-96.49	kd	CGS001-23566	LPAR3	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7361	-96.5	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
7362	-96.51	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
7363	-96.52	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
7364	-96.56	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
7365	-96.57	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
7366	-96.58	kd	CGS001-5498	PPOX	-			
7367	-96.58	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
7368	-96.59	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7369	-96.61	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
7370	-96.61	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
7371	-96.62	oe	ccsbBroad304_02115	PTTG1	-			
7372	-96.62	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
7373	-96.63	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
7374	-96.63	kd	CGS001-9988	DMTF1	-			
7375	-96.64	cp	BRD-K22227508	targinine	Nitric oxide synthase inhibitor		NOS2, NOS3	Nitric oxide synthase inhibitor
7376	-96.65	oe	ccsbBroad304_01001	MEST	-			
7377	-96.65	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
7378	-96.65	kd	CGS001-23786	BCL2L13	-			
7379	-96.66	kd	CGS001-2634	GBP2	-			
7380	-96.68	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
7381	-96.73	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
7382	-96.73	kd	CGS001-6599	SMARCC1	-			
7383	-96.73	kd	CGS001-81544	GDPD5	-			
7384	-96.75	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
7385	-96.78	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
7386	-96.79	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
7387	-96.79	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
7388	-96.79	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
7389	-96.8	kd	CGS001-5986	RFNG	Beta 3-glycosyltransferases			
7390	-96.8	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
7391	-96.84	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7392	-96.86	oe	ccsbBroad304_02109	XPR1	-			
7393	-96.86	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
7394	-96.86	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
7395	-96.87	kd	CGS001-5092	PCBD1	-			
7396	-96.91	kd	CGS001-8834	TMEM11	-			
7397	-96.92	kd	CGS001-2588	GALNS	Arylsulfatase family			
7398	-96.93	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
7399	-96.94	oe	ccsbBroad304_08684	CXCR7	-			
7400	-96.94	kd	CGS001-51465	UBE2J1	Ubiquitin-conjugating enzymes E2			
7401	-96.94	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
7402	-96.95	kd	CGS001-8624	PSMG1	-			
7403	-97	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
7404	-97	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
7405	-97.02	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
7406	-97.04	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
7407	-97.05	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
7408	-97.06	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
7409	-97.06	kd	CGS001-83448	PUS7L	-			
7410	-97.07	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
7411	-97.07	kd	CGS001-9833	MELK	MELK subfamily			
7412	-97.1	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
7413	-97.11	oe	ccsbBroad304_00238	CCNE1	-			
7414	-97.12	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
7415	-97.15	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
7416	-97.15	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
7417	-97.16	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
7418	-97.17	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
7419	-97.18	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7420	-97.21	oe	ccsbBroad304_06386	HNMT	-			
7421	-97.25	kd	CGS001-6337	SCNN1A	Epithelial sodium channels (ENaC)			
7422	-97.26	cp	BRD-K81169441	cerivastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A5	HMGCR inhibitor
7423	-97.28	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
7424	-97.29	kd	CGS001-51593	SRRT	-			
7425	-97.31	kd	CGS001-79711	IPO4	Importins			
7426	-97.31	kd	CGS001-54438	GFOD1	-			
7427	-97.32	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7428	-97.33	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
7429	-97.33	kd	CGS001-8717	TRADD	-			
7430	-97.34	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
7431	-97.34	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
7432	-97.36	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
7433	-97.36	oe	ccsbBroad304_05763	ACTB	-			
7434	-97.39	oe	ccsbBroad304_06976	SMARCE1	-			
7435	-97.39	oe	ccsbBroad304_03772	CCNL1	-			
7436	-97.39	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
7437	-97.39	kd	CGS001-28969	BZW2	-			
7438	-97.4	cc		Benzodiazepine receptor agonist	-			
7439	-97.41	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
7440	-97.42	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
7441	-97.42	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
7442	-97.44	oe	ccsbBroad304_00809	HUS1	-			
7443	-97.45	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
7444	-97.47	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
7445	-97.47	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
7446	-97.47	kd	CGS001-259	AMBP	Lipocalins			
7447	-97.49	cp	BRD-K37798499	etoposide	Topoisomerase inhibitor		TOP2A, CYP2E1, CYP3A5, TOP2B	Topoisomerase inhibitor
7448	-97.5	kd	CGS001-10111	RAD50	-			
7449	-97.53	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
7450	-97.54	cp	BRD-K13664374	dichloroacetic-acid	Pyruvate dehydrogenase kinase inhibitor		PDK1	Pyruvate dehydrogenase kinase inhibitor
7451	-97.54	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
7452	-97.55	oe	ccsbBroad304_06292	GNAI2	-			
7453	-97.55	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
7454	-97.55	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
7455	-97.57	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
7456	-97.58	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
7457	-97.58	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
7458	-97.59	oe	ccsbBroad304_04292	INHBE	-			
7459	-97.6	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
7460	-97.61	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
7461	-97.62	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
7462	-97.64	kd	CGS001-5610	EIF2AK2	Other PEK family kinases			
7463	-97.67	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
7464	-97.68	kd	CGS001-10975	UQCR11	Mitochondrial respiratory chain complex / Complex III			
7465	-97.68	kd	CGS001-1212	CLTB	-			
7466	-97.69	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
7467	-97.7	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
7468	-97.72	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
7469	-97.72	kd	CGS001-1616	DAXX	-			
7470	-97.73	oe	ccsbBroad304_00833	IFNG	Interferons			
7471	-97.73	oe	ccsbBroad304_01395	RFX5	-			
7472	-97.74	kd	CGS001-6258	RXRG	Retinoid X receptors			
7473	-97.75	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
7474	-97.76	oe	ccsbBroad304_02045	BUD31	-			
7475	-97.76	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
7476	-97.77	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
7477	-97.77	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
7478	-97.77	kd	CGS001-406	ARNTL	Basic helix-loop-helix proteins			
7479	-97.78	cc		DNA polymerase inhibitor	-			
7480	-97.78	oe	ccsbBroad304_08266	PIPOX	-			
7481	-97.78	oe	ccsbBroad304_03652	EXOC2	-			
7482	-97.78	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
7483	-97.8	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
7484	-97.8	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
7485	-97.81	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
7486	-97.81	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
7487	-97.83	kd	CGS001-415116	PIM3	PIM family			
7488	-97.84	oe	ccsbBroad304_01164	PDHB	-			
7489	-97.84	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
7490	-97.84	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
7491	-97.86	cp	BRD-K15916496	clotrimazole	Cytochrome P450 inhibitor		KCNN4, CYP3A4, CYP51A1, NR1I2, NR1I3, TRPM2, TRPM4, TRPM8	Cytochrome P450 inhibitor, Imidazoline receptor ligand
7492	-97.87	cp	BRD-A20589515	dihydroxyphenylglycine	Glutamate receptor agonist		GRM1	Glutamate receptor agonist
7493	-97.87	kd	CGS001-10142	AKAP9	A-kinase anchor proteins			
7494	-97.88	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
7495	-97.89	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
7496	-97.9	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
7497	-97.91	oe	ccsbBroad304_06985	SORD	-			
7498	-97.91	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
7499	-97.91	kd	CGS001-219333	USP12	Ubiquitin-specific peptidases			
7500	-97.91	kd	CGS001-5387	PMS2P3	-			
7501	-97.91	kd	CGS001-2558	GABRA5	GABA receptors			
7502	-97.93	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
7503	-97.93	kd	CGS001-7037	TFRC	CD molecules			
7504	-97.93	kd	CGS001-10651	MTX2	-			
7505	-97.93	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
7506	-97.93	kd	CGS001-9945	GFPT2	-			
7507	-97.94	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
7508	-97.95	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
7509	-97.95	kd	CGS001-7267	TTC3	RING-type (C3HC4) zinc fingers			
7510	-97.95	kd	CGS001-5900	RALGDS	-			
7511	-97.96	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
7512	-97.96	oe	ccsbBroad304_07102	TSG101	-			
7513	-97.97	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
7514	-97.97	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
7515	-97.98	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
7516	-97.98	kd	CGS001-55781	RIOK2	RIO2 subfamily			
7517	-98	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
7518	-98.01	oe	ccsbBroad304_06569	MCM5	-			
7519	-98.02	oe	ccsbBroad304_06040	CRY1	-			
7520	-98.03	kd	CGS001-2235	FECH	-			
7521	-98.03	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
7522	-98.04	oe	ccsbBroad304_00960	SMAD1	SMADs			
7523	-98.04	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
7524	-98.04	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
7525	-98.05	kd	CGS001-55107	ANO1	Calcium activated chloride channel			
7526	-98.06	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
7527	-98.06	kd	CGS001-100	ADA	Adenosine turnover			
7528	-98.07	oe	ccsbBroad304_02789	ADAT1	-			
7529	-98.08	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
7530	-98.1	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
7531	-98.1	kd	CGS001-2079	ERH	-			
7532	-98.11	kd	CGS001-9213	XPR1	-			
7533	-98.11	kd	CGS001-10923	SUB1	-			
7534	-98.12	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
7535	-98.12	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
7536	-98.13	oe	ccsbBroad304_06234	G6PC	-			
7537	-98.13	kd	CGS001-5335	PLCG1	Phosphoinositide-specific phospholipase C			
7538	-98.14	kd	CGS001-3569	IL6	Interferons			
7539	-98.16	kd	CGS001-6632	SNRPD1	-			
7540	-98.16	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
7541	-98.17	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
7542	-98.18	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
7543	-98.18	kd	CGS001-3692	EIF6	-			
7544	-98.18	kd	CGS001-665	BNIP3L	-			
7545	-98.19	kd	CGS001-50814	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7546	-98.19	oe	ccsbBroad304_06663	OAS1	-			
7547	-98.2	oe	ccsbBroad304_06523	LIG1	-			
7548	-98.2	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
7549	-98.2	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
7550	-98.21	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
7551	-98.21	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
7552	-98.24	oe	ccsbBroad304_03767	TOMM22	-			
7553	-98.24	kd	CGS001-11325	DDX42	DEAD-boxes			
7554	-98.27	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
7555	-98.27	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
7556	-98.27	kd	CGS001-65243	ZNF643	-			
7557	-98.28	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
7558	-98.3	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
7559	-98.3	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
7560	-98.3	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
7561	-98.31	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7562	-98.32	kd	CGS001-6204	RPS10	S ribosomal proteins			
7563	-98.32	kd	CGS001-1728	NQO1	-			
7564	-98.34	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
7565	-98.34	kd	CGS001-22796	COG2	Components of oligomeric golgi complex			
7566	-98.36	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
7567	-98.36	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
7568	-98.37	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
7569	-98.39	oe	ccsbBroad304_00115	ASPH	-			
7570	-98.39	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
7571	-98.42	kd	CGS001-4708	NDUFB2	Mitochondrial respiratory chain complex / Complex I			
7572	-98.43	kd	CGS001-23761	PISD	Decarboxylases			
7573	-98.43	kd	CGS001-23239	PHLPP1	Pleckstrin homology (PH) domain containing			
7574	-98.45	oe	ccsbBroad304_03961	SMURF2	-			
7575	-98.45	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
7576	-98.45	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
7577	-98.46	kd	CGS001-5916	RARG	Retinoic acid receptors			
7578	-98.46	kd	CGS001-8446	DUSP11	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7579	-98.46	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
7580	-98.47	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
7581	-98.47	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
7582	-98.48	oe	ccsbBroad304_14047	TACC3	-			
7583	-98.48	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
7584	-98.48	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
7585	-98.48	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
7586	-98.49	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
7587	-98.5	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
7588	-98.5	kd	CGS001-2621	GAS6	-			
7589	-98.51	oe	ccsbBroad304_01413	RPA2	-			
7590	-98.51	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
7591	-98.51	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
7592	-98.51	kd	CGS001-9688	NUP93	-			
7593	-98.52	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
7594	-98.54	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
7595	-98.54	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
7596	-98.58	kd	CGS001-10112	KIF20A	Kinesins			
7597	-98.59	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
7598	-98.59	oe	ccsbBroad304_02565	RALBP1	-			
7599	-98.59	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7600	-98.6	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
7601	-98.63	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7602	-98.66	kd	CGS001-55239	OGFOD1	-			
7603	-98.66	kd	CGS001-2539	G6PD	-			
7604	-98.67	kd	CGS001-27161	EIF2C2	-			
7605	-98.67	kd	CGS001-1662	DDX10	DEAD-boxes			
7606	-98.69	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
7607	-98.69	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
7608	-98.7	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
7609	-98.7	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
7610	-98.7	kd	CGS001-5315	PKM2	-			
7611	-98.7	kd	CGS001-11215	AKAP11	A-kinase anchor proteins			
7612	-98.71	cp	BRD-A41450521	tosufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
7613	-98.71	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
7614	-98.74	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7615	-98.75	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
7616	-98.75	kd	CGS001-80025	PANK2	-			
7617	-98.76	oe	ccsbBroad304_00101	RHOC	-			
7618	-98.76	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
7619	-98.77	oe	ccsbBroad304_09284	UBE3B	-			
7620	-98.77	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
7621	-98.78	kd	CGS001-8772	FADD	-			
7622	-98.79	oe	ccsbBroad304_02357	SSX3	-			
7623	-98.79	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
7624	-98.79	kd	CGS001-9451	EIF2AK3	PEK subfamily			
7625	-98.8	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
7626	-98.8	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
7627	-98.81	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
7628	-98.81	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
7629	-98.82	kd	CGS001-5781	PTPN11	Protein tyrosine phosphatases			
7630	-98.83	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
7631	-98.84	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
7632	-98.86	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7633	-98.87	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
7634	-98.87	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
7635	-98.88	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
7636	-98.88	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
7637	-98.88	kd	CGS001-7185	TRAF1	-			
7638	-98.88	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
7639	-98.89	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
7640	-98.89	kd	CGS001-84619	ZGPAT	G patch domain containing			
7641	-98.89	kd	CGS001-6208	RPS14	S ribosomal proteins			
7642	-98.9	oe	ccsbBroad304_03928	RRAGC	-			
7643	-98.9	oe	ccsbBroad304_00113	ASNS	-			
7644	-98.9	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
7645	-98.91	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
7646	-98.91	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
7647	-98.91	kd	CGS001-5366	PMAIP1	-			
7648	-98.91	kd	CGS001-3248	HPGD	Prostaglandin synthases			
7649	-98.92	kd	CGS001-6194	RPS6	S ribosomal proteins			
7650	-98.92	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
7651	-98.93	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
7652	-98.93	kd	CGS001-6625	SNRNP70	RNA binding motif (RRM) containing			
7653	-98.93	kd	CGS001-10775	POP4	-			
7654	-98.94	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
7655	-98.95	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
7656	-98.95	oe	ccsbBroad304_00085	APRT	-			
7657	-98.95	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
7658	-98.96	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
7659	-98.97	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
7660	-98.98	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
7661	-98.98	kd	CGS001-55765	C1ORF106	-			
7662	-98.99	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
7663	-98.99	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
7664	-98.99	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
7665	-99	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
7666	-99	kd	CGS001-51586	MED15	-			
7667	-99	kd	CGS001-760	CA2	Carbonic anhydrases			
7668	-99.02	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
7669	-99.02	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
7670	-99.03	kd	CGS001-661	POLR3D	RNA polymerase subunits			
7671	-99.04	kd	CGS001-2966	GTF2H2	General transcription factors			
7672	-99.05	kd	CGS001-59286	UBL5	-			
7673	-99.05	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
7674	-99.05	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
7675	-99.06	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
7676	-99.06	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
7677	-99.08	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
7678	-99.09	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
7679	-99.1	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
7680	-99.11	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
7681	-99.12	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
7682	-99.12	kd	CGS001-11040	PIM2	PIM family			
7683	-99.13	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
7684	-99.13	kd	CGS001-2037	EPB41L2	-			
7685	-99.14	cc		Kinase anchoring proteins LOF	-			
7686	-99.15	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
7687	-99.15	kd	CGS001-9124	PDLIM1	-			
7688	-99.16	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
7689	-99.16	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
7690	-99.16	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
7691	-99.16	kd	CGS001-6871	TADA2A	-			
7692	-99.17	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
7693	-99.17	kd	CGS001-203523	ZNF449	Zinc fingers, C2H2-type			
7694	-99.18	kd	CGS001-10797	MTHFD2	-			
7695	-99.18	kd	CGS001-54788	DNAJB12	Heat shock proteins / DNAJ (HSP40)			
7696	-99.19	kd	CGS001-11254	SLC6A14	Glycine transporter subfamily			
7697	-99.19	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
7698	-99.2	kd	CGS001-1936	EEF1D	-			
7699	-99.21	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
7700	-99.22	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
7701	-99.22	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
7702	-99.23	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
7703	-99.23	oe	ccsbBroad304_08023	EIF2C1	-			
7704	-99.24	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
7705	-99.25	cc		Ubiquitin-specific peptidases LOF	-			
7706	-99.25	oe	ccsbBroad304_01862	YEATS4	-			
7707	-99.25	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
7708	-99.25	kd	CGS001-10342	TFG	-			
7709	-99.25	kd	CGS001-6794	STK11	LKB subfamily			
7710	-99.26	cc		Non Homologous End Joining LOF	-			
7711	-99.27	oe	ccsbBroad304_00810	HYAL1	-			
7712	-99.27	oe	ccsbBroad304_08365	CYCS	-			
7713	-99.27	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
7714	-99.27	kd	CGS001-5566	PRKACA	Protein kinase A			
7715	-99.27	kd	CGS001-191	AHCY	Adenosine turnover			
7716	-99.28	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
7717	-99.28	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
7718	-99.29	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
7719	-99.29	oe	ccsbBroad304_02138	TRIP10	-			
7720	-99.3	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
7721	-99.3	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
7722	-99.3	kd	CGS001-1962	EHHADH	-			
7723	-99.31	oe	ccsbBroad304_02398	LANCL1	-			
7724	-99.31	kd	CGS001-1831	TSC22D3	-			
7725	-99.31	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
7726	-99.32	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
7727	-99.32	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
7728	-99.32	kd	CGS001-8503	PIK3R3	Phosphatidylinositol kinases			
7729	-99.32	kd	CGS001-929	CD14	CD molecules			
7730	-99.32	kd	CGS001-6936	C2ORF3	-			
7731	-99.33	cc		Nucleoporin LOF	-			
7732	-99.33	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
7733	-99.33	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
7734	-99.33	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7735	-99.33	kd	CGS001-63892	THADA	-			
7736	-99.33	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
7737	-99.34	oe	ccsbBroad304_06525	LIPA	-			
7738	-99.35	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
7739	-99.35	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
7740	-99.36	oe	ccsbBroad304_00657	GNG4	-			
7741	-99.36	oe	ccsbBroad304_00542	FBP1	-			
7742	-99.36	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
7743	-99.36	kd	CGS001-2197	FAU	S ribosomal proteins			
7744	-99.37	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
7745	-99.37	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
7746	-99.37	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
7747	-99.37	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
7748	-99.37	cp	BRD-K48932581	cetraxate	Mucus protecting agent		GAST	Mucus protecting agent
7749	-99.37	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
7750	-99.38	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
7751	-99.38	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
7752	-99.4	oe	ccsbBroad304_13598	NRBP2	NRBP family			
7753	-99.4	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
7754	-99.4	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
7755	-99.41	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
7756	-99.41	kd	CGS001-27	ABL2	Abl family			
7757	-99.42	oe	ccsbBroad304_06136	ECHS1	-			
7758	-99.42	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
7759	-99.42	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
7760	-99.43	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
7761	-99.43	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
7762	-99.44	oe	ccsbBroad304_06888	RPN1	-			
7763	-99.44	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
7764	-99.44	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
7765	-99.44	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
7766	-99.45	oe	ccsbBroad304_01165	PDK1	-			
7767	-99.45	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
7768	-99.45	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
7769	-99.45	kd	CGS001-1717	DHCR7	-			
7770	-99.47	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
7771	-99.47	kd	CGS001-6201	RPS7	S ribosomal proteins			
7772	-99.47	kd	CGS001-29915	HCFC2	-			
7773	-99.48	oe	ccsbBroad304_14291	GDPD5	-			
7774	-99.48	oe	ccsbBroad304_00568	FHL2	-			
7775	-99.48	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
7776	-99.49	cc		Ribosomal 40s Subunit LOF	-			
7777	-99.49	kd	CGS001-6223	RPS19	S ribosomal proteins			
7778	-99.49	kd	CGS001-23475	QPRT	-			
7779	-99.49	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
7780	-99.49	kd	CGS001-23658	LSM5	-			
7781	-99.49	kd	CGS001-94239	H2AFV	Histones / Replication-independent			
7782	-99.5	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
7783	-99.5	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
7784	-99.5	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
7785	-99.5	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
7786	-99.5	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
7787	-99.5	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
7788	-99.5	kd	CGS001-5209	PFKFB3	-			
7789	-99.51	oe	ccsbBroad304_09881	RFX6	-			
7790	-99.51	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
7791	-99.51	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
7792	-99.51	kd	CGS001-9958	USP15	Ubiquitin-specific peptidases			
7793	-99.52	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
7794	-99.52	kd	CGS001-2021	ENDOG	-			
7795	-99.53	oe	ccsbBroad304_09833	SENP5	-			
7796	-99.53	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
7797	-99.53	kd	CGS001-3588	IL10RB	IL-10 receptor family			
7798	-99.53	kd	CGS001-230	ALDOC	-			
7799	-99.54	kd	CGS001-64921	CASD1	-			
7800	-99.54	kd	CGS001-652	BMP4	Bone morphogenetic proteins			
7801	-99.55	oe	ccsbBroad304_02219	MORF4L2	-			
7802	-99.56	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
7803	-99.56	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
7804	-99.57	oe	ccsbBroad304_00963	SMAD5	SMADs			
7805	-99.57	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
7806	-99.57	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
7807	-99.59	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
7808	-99.59	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
7809	-99.59	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
7810	-99.59	kd	CGS001-3109	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
7811	-99.6	oe	ccsbBroad304_02405	TFG	-			
7812	-99.6	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
7813	-99.61	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
7814	-99.61	kd	CGS001-6621	SNAPC4	-			
7815	-99.62	oe	ccsbBroad304_01234	POLB	DNA polymerases			
7816	-99.62	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
7817	-99.62	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
7818	-99.64	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
7819	-99.64	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
7820	-99.64	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
7821	-99.65	oe	ccsbBroad304_06562	MAT1A	-			
7822	-99.65	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
7823	-99.65	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
7824	-99.65	kd	CGS001-56998	CTNNBIP1	Catenins			
7825	-99.65	kd	CGS001-55872	PBK	TOPK family			
7826	-99.66	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
7827	-99.66	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
7828	-99.66	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
7829	-99.66	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
7830	-99.67	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
7831	-99.67	oe	ccsbBroad304_06718	PFN2	-			
7832	-99.67	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
7833	-99.67	oe	ccsbBroad304_00423	DAXX	-			
7834	-99.67	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
7835	-99.67	kd	CGS001-93134	ZNF561	Zinc fingers, C2H2-type			
7836	-99.68	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
7837	-99.68	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
7838	-99.68	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
7839	-99.68	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
7840	-99.68	kd	CGS001-57147	SCYL3	-			
7841	-99.68	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
7842	-99.68	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
7843	-99.68	kd	CGS001-2353	FOS	basic leucine zipper proteins			
7844	-99.7	oe	ccsbBroad304_01663	TFF2	-			
7845	-99.7	oe	ccsbBroad304_01951	BLZF1	-			
7846	-99.7	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
7847	-99.7	kd	CGS001-8644	AKR1C3	Prostaglandin synthases			
7848	-99.71	oe	ccsbBroad304_01271	PPT1	-			
7849	-99.71	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
7850	-99.71	kd	CGS001-5636	PRPSAP2	-			
7851	-99.71	kd	CGS001-1362	CPD	Carboxypeptidase A			
7852	-99.72	cp	BRD-A11990600	lorazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, TSPO	Benzodiazepine receptor agonist
7853	-99.73	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
7854	-99.73	kd	CGS001-5664	PSEN2	Presenilin			
7855	-99.74	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
7856	-99.74	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
7857	-99.74	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
7858	-99.74	kd	CGS001-1062	CENPE	Kinesins			
7859	-99.75	kd	CGS001-2568	GABRP	GABA receptors			
7860	-99.76	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
7861	-99.76	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
7862	-99.77	kd	CGS001-5565	PRKAB2	AMPK subfamily			
7863	-99.77	kd	CGS001-1844	DUSP2	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
7864	-99.77	oe	ccsbBroad304_00969	MAGEA10	-			
7865	-99.78	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
7866	-99.78	oe	ccsbBroad304_00070	ANXA5	Annexins			
7867	-99.78	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
7868	-99.78	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
7869	-99.78	cp	BRD-A43082555	loxoprofen	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
7870	-99.78	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
7871	-99.78	kd	CGS001-80777	CYB5B	-			
7872	-99.79	oe	ccsbBroad304_00991	MDH1	-			
7873	-99.79	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
7874	-99.79	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
7875	-99.79	kd	CGS001-51096	UTP18	WD repeat domain containing			
7876	-99.79	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
7877	-99.81	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
7878	-99.81	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
7879	-99.81	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
7880	-99.81	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
7881	-99.81	kd	CGS001-5763	PTMS	-			
7882	-99.81	kd	CGS001-5351	PLOD1	-			
7883	-99.81	kd	CGS001-4234	METTL1	-			
7884	-99.82	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
7885	-99.82	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
7886	-99.82	kd	CGS001-10190	TXNDC9	-			
7887	-99.82	kd	CGS001-6777	STAT5B	SH2 domain containing			
7888	-99.82	oe	ccsbBroad304_06253	GALT	-			
7889	-99.83	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
7890	-99.83	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
7891	-99.83	kd	CGS001-5480	PPIC	-			
7892	-99.84	oe	ccsbBroad304_06574	MDH2	-			
7893	-99.84	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
7894	-99.84	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
7895	-99.84	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
7896	-99.84	kd	CGS001-6207	RPS13	S ribosomal proteins			
7897	-99.85	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
7898	-99.85	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
7899	-99.85	kd	CGS001-10915	TCERG1	-			
7900	-99.85	kd	CGS001-56654	NPDC1	-			
7901	-99.85	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
7902	-99.85	kd	CGS001-54205	CYCS	-			
7903	-99.87	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
7904	-99.87	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
7905	-99.87	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
7906	-99.87	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
7907	-99.87	kd	CGS001-7357	UGCG	Glycosyltransferase family 2 domain containing			
7908	-99.87	kd	CGS001-5211	PFKL	-			
7909	-99.87	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
7910	-99.87	kd	CGS001-9275	BCL7B	-			
7911	-99.87	kd	CGS001-350	APOH	Apolipoproteins			
7912	-99.88	oe	ccsbBroad304_03555	PANK4	-			
7913	-99.88	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
7914	-99.88	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
7915	-99.88	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
7916	-99.88	kd	CGS001-6188	RPS3	S ribosomal proteins			
7917	-99.88	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
7918	-99.88	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
7919	-99.88	kd	CGS001-51024	FIS1	-			
7920	-99.89	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
7921	-99.89	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
7922	-99.89	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7923	-99.89	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
7924	-99.89	kd	CGS001-5930	RBBP6	-			
7925	-99.89	kd	CGS001-3775	KCNK1	Two-P potassium channels			
7926	-99.89	kd	CGS001-9270	ITGB1BP1	-			
7927	-99.9	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
7928	-99.9	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
7929	-99.9	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
7930	-99.9	kd	CGS001-10497	UNC13B	-			
7931	-99.91	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
7932	-99.91	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
7933	-99.91	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
7934	-99.91	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
7935	-99.91	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
7936	-99.91	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
7937	-99.91	oe	ccsbBroad304_02452	NXF1	-			
7938	-99.92	cc		SMAD family LOF	-			
7939	-99.92	kd	CGS001-5777	PTPN6	Protein tyrosine phosphatases			
7940	-99.93	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
7941	-99.93	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
7942	-99.93	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
7943	-99.93	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
7944	-99.93	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
7945	-99.93	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
7946	-99.93	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
7947	-99.94	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
7948	-99.94	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
7949	-99.94	kd	CGS001-4811	NID1	-			
7950	-99.94	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
7951	-99.95	oe	ccsbBroad304_08879	CASD1	-			
7952	-99.95	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
7953	-99.95	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
7954	-99.95	kd	CGS001-206358	SLC36A1	SLC36 family of proton-coupled amino acid transporters			
7955	-99.95	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
7956	-99.95	kd	CGS001-2771	GNAI2	-			
7957	-99.95	kd	CGS001-9453	GGPS1	Lanosterol biosynthesis pathway			
7958	-99.95	kd	CGS001-54555	DDX49	DEAD-boxes			
7959	-99.96	cc		Bacterial cell wall synthesis inhibitor	-			
7960	-99.96	oe	ccsbBroad304_01723	TTK	TTK family			
7961	-99.96	oe	ccsbBroad304_00888	ITPK1	-			
7962	-99.96	oe	ccsbBroad304_00170	BNIP1	-			
7963	-99.96	oe	ccsbBroad304_08888	ACD	-			
7964	-99.96	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
7965	-99.96	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
7966	-99.96	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
7967	-99.96	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
7968	-99.96	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
7969	-99.96	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
7970	-99.96	kd	CGS001-79862	ZNF669	Zinc fingers, C2H2-type			
7971	-99.96	kd	CGS001-6477	SIAH1	-			
7972	-99.96	kd	CGS001-9871	SEC24D	-			
7973	-99.96	kd	CGS001-5293	PIK3CD	Phosphatidylinositol kinases			
7974	-99.96	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
7975	-99.96	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
7976	-99.96	kd	CGS001-8639	AOC3	Oxidoreductases			
7977	-99.96	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
7978	-99.98	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
7979	-99.98	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
7980	-99.98	oe	ccsbBroad304_07832	XPO7	Exportins			
7981	-99.98	oe	ccsbBroad304_07814	SACM1L	-			
7982	-99.98	oe	ccsbBroad304_14143	NUSAP1	-			
7983	-99.98	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
7984	-99.98	oe	ccsbBroad304_06535	LPL	-			
7985	-99.98	oe	ccsbBroad304_06350	HAL	-			
7986	-99.98	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
7987	-99.98	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
7988	-99.98	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
7989	-99.98	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
7990	-99.98	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
7991	-99.98	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
7992	-99.98	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
7993	-99.98	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
7994	-99.98	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
7995	-99.98	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
7996	-99.98	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
7997	-99.98	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
7998	-99.98	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
7999	-99.98	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
8000	-99.98	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
8001	-99.98	cp	BRD-K07237224	moclobemide	Monoamine oxidase inhibitor		MAOA, CYP2C19, MAOB	Monoamine oxidase inhibitor
8002	-99.98	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
8003	-99.98	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
8004	-99.98	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
8005	-99.98	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
8006	-99.98	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
8007	-99.98	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
8008	-99.98	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
8009	-99.98	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
8010	-99.98	kd	CGS001-147948	ZNF582	Zinc fingers, C2H2-type			
8011	-99.98	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
8012	-99.98	kd	CGS001-3431	SP110	Non-enzymatic BRD containing proteins			
8013	-99.98	kd	CGS001-4089	SMAD4	SMADs			
8014	-99.98	kd	CGS001-5371	PML	RING-type (C3HC4) zinc fingers			
8015	-99.98	kd	CGS001-4485	MST1	-			
8016	-99.98	kd	CGS001-85442	KNDC1	-			
8017	-99.98	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
8018	-99.98	kd	CGS001-84634	KISS1R	GPCR / Class A : RF amide peptide receptors			
8019	-99.98	kd	CGS001-23325	KIAA1033	-			
8020	-99.98	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
8021	-99.98	kd	CGS001-3672	ITGA1	Integrins			
8022	-99.98	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
8023	-99.98	kd	CGS001-79187	FSD1	Fibronectin type III domain containing			
8024	-99.98	kd	CGS001-1806	DPYD	-			
8025	-99.98	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
8026	-99.98	kd	CGS001-10898	CPSF4	-			
8027	-99.98	kd	CGS001-55832	CAND1	-			
8028	-99.98	kd	CGS001-95	ACY1	-			
