Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
2	100	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
3	99.99	oe	ccsbBroad304_14242	MCCC2	-			
4	99.99	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
5	99.99	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
6	99.99	kd	CGS001-57804	POLD4	DNA polymerases			
7	99.97	oe	ccsbBroad304_01880	LAGE3	-			
8	99.97	oe	ccsbBroad304_03604	ENOSF1	-			
9	99.97	oe	ccsbBroad304_00464	DTNA	-			
10	99.97	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
11	99.97	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
12	99.97	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
13	99.97	oe	ccsbBroad304_01271	PPT1	-			
14	99.97	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
15	99.97	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
16	99.97	oe	ccsbBroad304_00809	HUS1	-			
17	99.97	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
18	99.97	oe	ccsbBroad304_06382	HMGCL	-			
19	99.97	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
20	99.97	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
21	99.97	oe	ccsbBroad304_07834	GGA2	-			
22	99.97	oe	ccsbBroad304_00644	GCLC	-			
23	99.97	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
24	99.97	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
25	99.97	oe	ccsbBroad304_02956	EHF	-			
26	99.97	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
27	99.97	oe	ccsbBroad304_00036	AFP	-			
28	99.97	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
29	99.97	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
30	99.97	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
31	99.97	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
32	99.97	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
33	99.97	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
34	99.97	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
35	99.97	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
36	99.97	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
37	99.97	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
38	99.97	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
39	99.97	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
40	99.97	kd	CGS001-22954	TRIM32	-			
41	99.97	kd	CGS001-10221	TRIB1	Trbl family			
42	99.97	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
43	99.97	kd	CGS001-10474	TADA3	-			
44	99.97	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
45	99.97	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
46	99.97	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
47	99.97	kd	CGS001-9404	LPXN	-			
48	99.97	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
49	99.97	kd	CGS001-2770	GNAI1	-			
50	99.97	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
51	99.97	kd	CGS001-1786	DNMT1	Methyltransferases			
52	99.97	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
53	99.96	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
54	99.96	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
55	99.96	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
56	99.96	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
57	99.96	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
58	99.96	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
59	99.96	oe	ccsbBroad304_02837	BHMT2	-			
60	99.96	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
61	99.96	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
62	99.96	kd	CGS001-23212	RRS1	-			
63	99.96	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
64	99.96	kd	CGS001-10465	PPIH	-			
65	99.96	kd	CGS001-1374	CPT1A	-			
66	99.96	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
67	99.96	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
68	99.96	kd	CGS001-10423	CDIPT	-			
69	99.96	kd	CGS001-84433	CARD11	-			
70	99.95	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
71	99.94	oe	ccsbBroad304_01651	TCF7L2	-			
72	99.94	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
73	99.94	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
74	99.94	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
75	99.94	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
76	99.94	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
77	99.94	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
78	99.94	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
79	99.94	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
80	99.94	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
81	99.94	kd	CGS001-7423	VEGFB	-			
82	99.94	kd	CGS001-8576	STK16	NAK family			
83	99.94	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
84	99.94	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
85	99.94	kd	CGS001-1606	DGKA	EF-hand domain containing			
86	99.93	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
87	99.93	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
88	99.93	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
89	99.93	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
90	99.93	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
91	99.93	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
92	99.93	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
93	99.93	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
94	99.93	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
95	99.93	kd	CGS001-4312	MMP1	Matrix metallopeptidase			
96	99.91	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
97	99.91	kd	CGS001-89882	TPD52L3	-			
98	99.91	kd	CGS001-391013	PLA2G2C	-			
99	99.91	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
100	99.91	kd	CGS001-60528	ELAC2	-			
101	99.91	kd	CGS001-23142	DCUN1D4	-			
102	99.9	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
103	99.9	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
104	99.9	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
105	99.9	oe	ccsbBroad304_04387	MKI67IP	-			
106	99.9	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
107	99.9	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
108	99.9	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
109	99.9	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
110	99.88	oe	ccsbBroad304_01618	STXBP1	-			
111	99.88	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
112	99.88	oe	ccsbBroad304_06695	PCK2	-			
113	99.88	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
114	99.88	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
115	99.88	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
116	99.88	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
117	99.88	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
118	99.88	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
119	99.88	kd	CGS001-2057	EPOR	Prolactin receptor family			
120	99.88	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
121	99.87	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
122	99.87	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
123	99.87	kd	CGS001-3032	HADHB	-			
124	99.85	oe	ccsbBroad304_00658	GNG5	-			
125	99.85	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
126	99.85	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
127	99.85	kd	CGS001-2752	GLUL	-			
128	99.85	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
129	99.85	kd	CGS001-9474	ATG5	-			
130	99.84	oe	ccsbBroad304_02843	FTSJ1	-			
131	99.84	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
132	99.84	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
133	99.84	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
134	99.84	kd	CGS001-4605	MYBL2	-			
135	99.83	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
136	99.82	oe	ccsbBroad304_02845	PRPF6	-			
137	99.82	kd	CGS001-64080	RBKS	-			
138	99.81	oe	ccsbBroad304_06665	OAT	-			
139	99.81	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
140	99.81	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
141	99.81	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
142	99.79	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
143	99.79	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
144	99.79	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
145	99.79	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
146	99.79	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
147	99.79	kd	CGS001-36	ACADSB	-			
148	99.78	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
149	99.78	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
150	99.78	oe	ccsbBroad304_05758	ACADSB	-			
151	99.78	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
152	99.76	oe	ccsbBroad304_02496	MTX2	-			
153	99.76	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
154	99.76	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
155	99.75	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
156	99.75	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
157	99.73	oe	ccsbBroad304_02875	BRP44	-			
158	99.73	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
159	99.73	kd	CGS001-2247	FGF2	Endogenous ligands			
160	99.73	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
161	99.72	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
162	99.71	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
163	99.71	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
164	99.69	oe	ccsbBroad304_00033	ADSS	-			
165	99.68	kd	CGS001-10190	TXNDC9	-			
166	99.66	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
167	99.66	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
168	99.65	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
169	99.65	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
170	99.65	kd	CGS001-337867	UBAC2	-			
171	99.65	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
172	99.62	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
173	99.61	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
174	99.6	oe	ccsbBroad304_03506	AURKAIP1	-			
175	99.6	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
176	99.6	kd	CGS001-9180	OSMR	IL-6 receptor family			
177	99.59	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
178	99.59	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
179	99.59	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
180	99.57	kd	CGS001-2152	F3	CD molecules			
181	99.56	oe	ccsbBroad304_00818	IDH3A	-			
182	99.56	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
183	99.56	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
184	99.56	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
185	99.56	kd	CGS001-4171	MCM2	-			
186	99.56	kd	CGS001-11129	CLASRP	-			
187	99.55	oe	ccsbBroad304_06458	IRF3	-			
188	99.55	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
189	99.55	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
190	99.55	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
191	99.54	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
192	99.54	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
193	99.54	kd	CGS001-2242	FES	Fer family			
194	99.53	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
195	99.53	kd	CGS001-351	APP	Endogenous ligands			
196	99.52	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
197	99.51	kd	CGS001-1725	DHPS	-			
198	99.5	kd	CGS001-9231	DLG5	-			
199	99.48	oe	ccsbBroad304_04619	GNG8	-			
200	99.48	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
201	99.48	kd	CGS001-9709	HERPUD1	-			
202	99.47	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
203	99.47	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
204	99.46	oe	ccsbBroad304_08266	PIPOX	-			
205	99.46	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
206	99.45	oe	ccsbBroad304_00116	ASS1	-			
207	99.45	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
208	99.44	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
209	99.44	oe	ccsbBroad304_00170	BNIP1	-			
210	99.44	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
211	99.44	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
212	99.39	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
213	99.38	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
214	99.37	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
215	99.37	kd	CGS001-91433	RCCD1	-			
216	99.35	kd	CGS001-10289	EIF1B	-			
217	99.34	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
218	99.34	kd	CGS001-1949	EFNB3	Ephrins			
219	99.33	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
220	99.32	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
221	99.32	kd	CGS001-2184	FAH	-			
222	99.31	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
223	99.31	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
224	99.31	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
225	99.31	kd	CGS001-4801	NFYB	-			
226	99.3	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
227	99.26	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
228	99.26	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
229	99.25	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
230	99.25	oe	ccsbBroad304_00515	ERH	-			
231	99.25	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
232	99.22	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
233	99.21	kd	CGS001-10253	SPRY2	-			
234	99.19	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
235	99.18	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
236	99.18	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
237	99.17	oe	ccsbBroad304_00709	GUK1	-			
238	99.15	kd	CGS001-84617	TUBB6	Tubulins			
239	99.15	kd	CGS001-4522	MTHFD1	-			
240	99.14	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
241	99.11	kd	CGS001-4610	MYCL1	-			
242	99.09	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
243	99.09	kd	CGS001-10973	ASCC3	-			
244	99.07	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
245	99.07	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
246	99.06	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
247	99.06	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
248	99.04	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
249	99.04	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
250	99.02	kd	CGS001-9943	OXSR1	FRAY subfamily			
251	99.01	oe	ccsbBroad304_02357	SSX3	-			
252	99.01	oe	ccsbBroad304_06291	GNAI1	-			
253	99.01	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
254	98.98	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
255	98.96	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
256	98.96	oe	ccsbBroad304_00221	CASP3	Caspases			
257	98.93	oe	ccsbBroad304_03268	GMPR2	-			
258	98.93	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
259	98.91	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
260	98.91	kd	CGS001-5428	POLG	DNA polymerases			
261	98.9	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
262	98.89	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
263	98.89	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
264	98.89	kd	CGS001-50813	COPS7A	-			
265	98.88	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
266	98.86	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
267	98.82	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
268	98.81	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
269	98.81	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
270	98.81	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
271	98.79	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
272	98.79	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
273	98.75	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
274	98.75	kd	CGS001-27241	BBS9	-			
275	98.73	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
276	98.73	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
277	98.72	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
278	98.71	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
279	98.69	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
280	98.67	oe	ccsbBroad304_06549	SMAD3	SMADs			
281	98.67	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
282	98.67	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
283	98.66	oe	ccsbBroad304_02231	USP6NL	-			
284	98.66	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
285	98.65	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
286	98.64	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
287	98.64	kd	CGS001-56654	NPDC1	-			
288	98.63	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
289	98.63	oe	ccsbBroad304_00003	ABAT	GABA turnover			
290	98.63	kd	CGS001-23223	RRP12	-			
291	98.6	kd	CGS001-4781	NFIB	-			
292	98.59	kd	CGS001-10398	MYL9	EF-hand domain containing			
293	98.58	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
294	98.58	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
295	98.57	oe	ccsbBroad304_06645	NQO2	-			
296	98.56	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
297	98.52	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
298	98.5	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
299	98.47	oe	ccsbBroad304_01208	PITPNA	-			
300	98.47	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
301	98.46	oe	ccsbBroad304_03237	LEF1	-			
302	98.44	oe	ccsbBroad304_02551	CPSF4	-			
303	98.44	kd	CGS001-4947	OAZ2	-			
304	98.42	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
305	98.42	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
306	98.42	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
307	98.42	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
308	98.42	kd	CGS001-5927	KDM5A	Histone demethylases			
309	98.4	kd	CGS001-5306	PITPNA	-			
310	98.39	oe	ccsbBroad304_00650	GNA11	-			
311	98.39	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
312	98.38	kd	CGS001-5579	PRKCB	Alpha subfamily			
313	98.38	kd	CGS001-9817	KEAP1	Kelch-like proteins			
314	98.33	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
315	98.32	oe	ccsbBroad304_03555	PANK4	-			
316	98.32	kd	CGS001-55837	EAPP	-			
317	98.31	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
318	98.3	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
319	98.28	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
320	98.27	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
321	98.26	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
322	98.26	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
323	98.26	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
324	98.25	kd	CGS001-79006	METRN	-			
325	98.24	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
326	98.24	kd	CGS001-5163	PDK1	-			
327	98.23	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
328	98.22	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
329	98.19	oe	ccsbBroad304_00833	IFNG	Interferons			
330	98.19	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
331	98.17	kd	CGS001-11179	ZNF277	-			
332	98.13	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
333	98.11	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
334	98.1	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
335	98.09	oe	ccsbBroad304_03173	TMED7	-			
336	98.08	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
337	98.07	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
338	98.06	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
339	98.05	kd	CGS001-10672	GNA13	-			
340	98.03	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
341	98	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
342	98	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
343	97.94	oe	ccsbBroad304_05547	TMEM110	-			
344	97.94	kd	CGS001-5092	PCBD1	-			
345	97.93	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
346	97.92	oe	ccsbBroad304_04153	PHF17	-			
347	97.9	kd	CGS001-29937	NENF	-			
348	97.9	kd	CGS001-717	C2	Complement system			
349	97.89	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
350	97.89	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
351	97.85	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
352	97.83	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
353	97.82	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
354	97.82	kd	CGS001-6282	S100A11	EF-hand domain containing			
355	97.82	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
356	97.8	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
357	97.77	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
358	97.77	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
359	97.76	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
360	97.74	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
361	97.73	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
362	97.72	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
363	97.71	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
364	97.69	oe	ccsbBroad304_12226	NAGK	-			
365	97.69	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
366	97.68	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
367	97.67	kd	CGS001-89910	UBE3B	-			
368	97.66	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
369	97.66	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
370	97.65	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
371	97.64	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
372	97.62	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
373	97.61	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
374	97.59	kd	CGS001-10670	RRAGA	-			
375	97.58	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
376	97.56	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
377	97.51	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
378	97.49	oe	ccsbBroad304_06255	LRRC32	-			
379	97.48	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
380	97.46	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
381	97.45	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
382	97.44	kd	CGS001-5446	PON3	Paraoxonases			
383	97.42	kd	CGS001-5091	PC	Carboxylases			
384	97.41	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
385	97.4	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
386	97.36	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
387	97.35	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
388	97.3	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
389	97.28	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
390	97.26	cc		IGF-1 inhibitor	-			
391	97.24	oe	ccsbBroad304_01002	METTL1	-			
392	97.23	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
393	97.23	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
394	97.21	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
395	97.2	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
396	97.19	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
397	97.17	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
398	97.16	kd	CGS001-3682	ITGAE	Integrins			
399	97.15	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
400	97.15	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
401	97.14	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
402	97.13	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
403	97.11	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
404	97.1	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
405	97.09	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
406	97.09	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
407	97.09	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
408	97.09	kd	CGS001-6603	SMARCD2	-			
409	97.06	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
410	97.06	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
411	97.05	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
412	97.04	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
413	97.04	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
414	97.03	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
415	96.99	oe	ccsbBroad304_07557	NAMPT	-			
416	96.98	kd	CGS001-7097	TLR2	Toll-like receptor family			
417	96.96	kd	CGS001-51002	TPRKB	-			
418	96.94	cc		X linked mental retardation group 2 LOF	-			
419	96.92	kd	CGS001-2212	FCGR2A	CD molecules			
420	96.91	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
421	96.9	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
422	96.89	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
423	96.89	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
424	96.86	oe	ccsbBroad304_01008	KITLG	-			
425	96.86	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
426	96.86	kd	CGS001-8295	TRRAP	TRRAP subfamily			
427	96.83	kd	CGS001-5359	PLSCR1	-			
428	96.78	kd	CGS001-6727	SRP14	-			
429	96.78	kd	CGS001-4255	MGMT	-			
430	96.76	oe	ccsbBroad304_01013	MIF	-			
431	96.75	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
432	96.72	kd	CGS001-64750	SMURF2	-			
433	96.71	oe	ccsbBroad304_03357	RASD1	-			
434	96.7	cc		Ubiquitin-specific peptidases LOF	-			
435	96.7	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
436	96.69	kd	CGS001-9232	PTTG1	-			
437	96.67	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
438	96.67	kd	CGS001-2079	ERH	-			
439	96.65	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
440	96.61	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
441	96.6	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
442	96.58	kd	CGS001-5966	REL	NFkappaB transcription factor family			
443	96.52	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
444	96.52	kd	CGS001-79947	DHDDS	-			
445	96.5	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
446	96.49	kd	CGS001-253430	IPMK	-			
447	96.4	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
448	96.38	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
449	96.37	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
450	96.3	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
451	96.22	kd	CGS001-5906	RAP1A	-			
452	96.19	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
453	96.16	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
454	96.15	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
455	96.1	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
456	96.08	kd	CGS001-3169	FOXA1	Forkhead boxes			
457	96.07	cc		BMP Signaling LOF	-			
458	96.06	kd	CGS001-230	ALDOC	-			
459	96.01	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
460	96	kd	CGS001-51070	NOSIP	-			
461	95.96	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
462	95.95	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
463	95.93	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
464	95.91	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
465	95.91	kd	CGS001-53340	SPA17	-			
466	95.9	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
467	95.9	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
468	95.89	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
469	95.87	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
470	95.8	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
471	95.77	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
472	95.76	oe	ccsbBroad304_07561	YAF2	-			
473	95.72	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
474	95.72	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
475	95.7	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
476	95.69	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
477	95.67	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
478	95.62	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
479	95.61	oe	ccsbBroad304_00532	F11	Chymotrypsin			
480	95.56	kd	CGS001-54915	YTHDF1	-			
481	95.51	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
482	95.51	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
483	95.49	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
484	95.47	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
485	95.46	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
486	95.45	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
487	95.44	kd	CGS001-3690	ITGB3	Integrins			
488	95.44	kd	CGS001-51727	CMPK1	-			
489	95.42	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
490	95.41	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
491	95.38	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
492	95.33	oe	ccsbBroad304_00615	GAPDH	-			
493	95.32	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
494	95.26	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
495	95.23	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
496	95.22	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
497	95.19	kd	CGS001-9124	PDLIM1	-			
498	95.19	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
499	95.16	kd	CGS001-10325	RRAGB	-			
500	95.12	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
501	95.12	kd	CGS001-1211	CLTA	-			
502	95.08	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
503	95.02	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
504	95	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
505	95	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
506	94.95	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
507	94.95	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
508	94.95	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
509	94.9	kd	CGS001-10434	LYPLA1	-			
510	94.85	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
511	94.82	oe	ccsbBroad304_00060	AMBP	Lipocalins			
512	94.81	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
513	94.81	kd	CGS001-6520	SLC3A2	SLC3 family			
514	94.81	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
515	94.79	oe	ccsbBroad304_07548	TSSC4	-			
516	94.79	kd	CGS001-9638	FEZ1	-			
517	94.77	kd	CGS001-51268	PIPOX	-			
518	94.75	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
519	94.65	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
520	94.59	oe	ccsbBroad304_03652	EXOC2	-			
521	94.57	cc		Homeobox Gene GOF	-			
522	94.56	oe	ccsbBroad304_06089	DDIT3	-			
523	94.54	oe	ccsbBroad304_02220	MTFR1	-			
524	94.53	oe	ccsbBroad304_01872	DGCR14	-			
525	94.49	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
526	94.46	oe	ccsbBroad304_07704	SUB1	-			
527	94.45	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
528	94.45	kd	CGS001-1534	CYB561	Cytochrome b genes			
529	94.44	oe	ccsbBroad304_00459	DPYD	-			
530	94.43	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
531	94.43	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
532	94.41	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
533	94.41	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
534	94.39	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
535	94.35	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
536	94.34	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
537	94.32	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
538	94.29	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
539	94.27	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
540	94.26	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
541	94.25	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
542	94.24	cc		Targets of VEGFR inhibitors GOF	-			
543	94.24	kd	CGS001-5653	KLK6	Chymotrypsin			
544	94.22	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
545	94.16	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
546	94.16	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
547	94.11	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
548	94.11	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
549	94.08	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
550	94.07	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
551	94.04	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
552	94.03	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
553	93.98	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
554	93.98	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
555	93.97	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
556	93.96	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
557	93.95	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
558	93.94	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
559	93.88	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
560	93.85	oe	ccsbBroad304_04544	RCCD1	-			
561	93.83	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
562	93.82	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
563	93.79	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
564	93.72	kd	CGS001-55810	FOXJ2	Forkhead boxes			
565	93.7	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
566	93.68	oe	ccsbBroad304_13891	LCK	Src family			
567	93.68	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
568	93.66	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
569	93.61	kd	CGS001-8453	CUL2	-			
570	93.58	kd	CGS001-1314	COPA	Endogenous ligands			
571	93.57	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
572	93.55	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
573	93.54	kd	CGS001-2882	GPX7	-			
574	93.53	oe	ccsbBroad304_02653	PRAF2	-			
575	93.5	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
576	93.48	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
577	93.48	kd	CGS001-8829	NRP1	CD molecules			
578	93.46	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
579	93.42	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
580	93.42	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
581	93.42	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
582	93.4	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
583	93.4	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
584	93.38	oe	ccsbBroad304_08346	COQ3	-			
585	93.35	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
586	93.34	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
587	93.32	kd	CGS001-5590	PRKCZ	Iota subfamily			
588	93.26	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
589	93.26	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
590	93.25	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
591	93.21	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
592	93.21	oe	ccsbBroad304_00020	ACY1	-			
593	93.21	kd	CGS001-9833	MELK	MELK subfamily			
594	93.2	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
595	93.13	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
596	93.1	oe	ccsbBroad304_06294	GNAZ	-			
597	93.07	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
598	93.04	oe	ccsbBroad304_03129	ERO1L	-			
599	93	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
600	92.92	kd	CGS001-185	AGTR1	Angiotensin receptors			
601	92.9	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
602	92.9	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
603	92.89	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
604	92.85	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
605	92.82	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
606	92.77	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
607	92.76	kd	CGS001-2956	MSH6	-			
608	92.73	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
609	92.66	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
610	92.65	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
611	92.63	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
612	92.62	oe	ccsbBroad304_07018	SUPT5H	-			
613	92.61	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
614	92.58	oe	ccsbBroad304_01701	TPI1	-			
615	92.57	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
616	92.57	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
617	92.54	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
618	92.51	kd	CGS001-64781	CERK	Ceramide kinase			
619	92.49	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
620	92.48	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
621	92.47	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
622	92.44	kd	CGS001-8720	MBTPS1	Subtilisin			
623	92.4	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
624	92.38	kd	CGS001-4282	MIF	-			
625	92.35	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
626	92.27	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
627	92.22	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
628	92.18	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
629	92.17	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
630	92.16	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
631	92.13	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
632	92.12	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
633	92.11	oe	ccsbBroad304_03269	CD320	CD molecules			
634	92.09	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
635	92.08	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
636	92.06	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
637	92.01	oe	ccsbBroad304_01413	RPA2	-			
638	91.99	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
639	91.95	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
640	91.9	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
641	91.88	kd	CGS001-6513	SLC2A1	Solute carriers			
642	91.85	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
643	91.82	oe	ccsbBroad304_01247	POU2AF1	-			
644	91.72	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
645	91.72	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
646	91.68	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
647	91.63	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
648	91.55	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
649	91.53	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
650	91.52	oe	ccsbBroad304_01203	PIM1	PIM family			
651	91.46	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
652	91.44	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
653	91.39	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
654	91.39	kd	CGS001-10084	PQBP1	-			
655	91.36	oe	ccsbBroad304_03853	LSM2	-			
656	91.36	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
657	91.36	kd	CGS001-2353	FOS	basic leucine zipper proteins			
658	91.32	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
659	91.31	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
660	91.31	kd	CGS001-57680	CHD8	-			
661	91.29	kd	CGS001-399664	MEX3D	Mex-3 homologs			
662	91.24	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
663	91.24	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
664	91.23	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
665	91.21	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
666	91.21	kd	CGS001-629	CFB	Complement system			
667	91.18	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
668	91.17	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
669	91.17	kd	CGS001-83440	ADPGK	-			
670	91.12	kd	CGS001-7405	UVRAG	-			
671	91.04	kd	CGS001-51292	GMPR2	-			
672	91.02	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
673	90.98	cp	BRD-K34508425	KUC103898N	-666			-666
674	90.95	oe	ccsbBroad304_01066	NDUFA4	-			
675	90.95	kd	CGS001-2639	GCDH	-			
676	90.92	kd	CGS001-23536	ADAT1	-			
677	90.89	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
678	90.86	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
679	90.86	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
680	90.83	oe	ccsbBroad304_00550	FDXR	-			
681	90.82	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
682	90.8	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
683	90.74	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
684	90.72	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
685	90.71	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
686	90.7	oe	ccsbBroad304_08511	RFK	-			
687	90.69	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
688	90.68	cc		Serine proteases GOF	-			
689	90.54	kd	CGS001-55604	LRRC16A	-			
690	90.49	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
691	90.48	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
692	90.47	oe	ccsbBroad304_09358	MAPK1IP1L	-			
693	90.46	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
694	90.45	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
695	90.34	oe	ccsbBroad304_02306	PQBP1	-			
696	90.23	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
697	90.23	kd	CGS001-5992	RFX4	-			
698	90.18	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
699	90.14	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
700	90.04	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
701	89.95	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
702	89.93	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
703	89.85	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
704	89.82	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
705	89.81	cc		MTOR inhibitor	-			
706	89.81	oe	ccsbBroad304_03772	CCNL1	-			
707	89.81	kd	CGS001-3956	LGALS1	Endogenous ligands			
708	89.6	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
709	89.59	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
710	89.57	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
711	89.56	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
712	89.55	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
713	89.55	kd	CGS001-6757	SSX2	-			
714	89.55	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
715	89.39	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
716	89.33	kd	CGS001-6778	STAT6	SH2 domain containing			
717	89.26	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
718	89.22	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
719	89.2	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
720	89.18	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
721	89.1	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
722	89.07	cc		Dihydrofolate reductase inhibitor	-			
723	89.07	kd	CGS001-2078	ERG	ETS Transcription Factors			
724	89.02	kd	CGS001-1892	ECHS1	-			
725	88.98	cc		Na-K-Cl transporter inhibitor	-			
726	88.91	kd	CGS001-253260	RICTOR	-			
727	88.9	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
728	88.86	kd	CGS001-10475	TRIM38	-			
729	88.85	kd	CGS001-55715	DOK4	Pleckstrin homology (PH) domain containing			
730	88.82	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
731	88.79	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
732	88.78	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
733	88.73	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
734	88.72	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
735	88.69	kd	CGS001-29763	PACSIN3	-			
736	88.68	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
737	88.61	kd	CGS001-6204	RPS10	S ribosomal proteins			
738	88.6	kd	CGS001-9787	DLGAP5	-			
739	88.59	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
740	88.55	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
741	88.51	cc		PI3K inhibitor	-			
742	88.5	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
743	88.48	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
744	88.45	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
745	88.38	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
746	88.38	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
747	88.37	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
748	88.37	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
749	88.34	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
750	88.24	oe	ccsbBroad304_00164	BLMH	-			
751	88.21	kd	CGS001-4016	LOXL1	-			
752	88.18	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
753	88.11	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
754	88.1	kd	CGS001-389421	LIN28B	-			
755	88.09	kd	CGS001-7525	YES1	Src family			
756	88.07	oe	ccsbBroad304_02737	JMJD6	-			
757	88.05	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
758	88.02	kd	CGS001-56616	DIABLO	-			
759	87.97	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
760	87.84	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
761	87.84	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
762	87.8	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
763	87.73	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
764	87.73	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
765	87.71	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
766	87.66	oe	ccsbBroad304_00652	GNAS	-			
767	87.63	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
768	87.54	kd	CGS001-4193	MDM2	-			
769	87.5	kd	CGS001-25942	SIN3A	-			
770	87.45	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
771	87.42	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
772	87.41	kd	CGS001-8896	BUD31	-			
773	87.39	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
774	87.37	kd	CGS001-3980	LIG3	-			
775	87.35	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
776	87.35	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
777	87.33	cc		Norepinephrine reuptake inhibitor	-			
778	87.33	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
779	87.31	kd	CGS001-26277	TINF2	-			
780	87.26	kd	CGS001-572	BAD	-			
781	87.24	oe	ccsbBroad304_00969	MAGEA10	-			
782	87.21	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
783	87.17	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
784	87.17	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
785	87.09	kd	CGS001-8535	CBX4	-			
786	87.04	oe	ccsbBroad304_00568	FHL2	-			
787	87.01	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
788	86.99	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
789	86.98	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
790	86.88	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
791	86.85	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
792	86.84	kd	CGS001-23463	ICMT	-			
793	86.82	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
794	86.78	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
795	86.69	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
796	86.69	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
797	86.68	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
798	86.67	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
799	86.65	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
800	86.62	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
801	86.61	oe	ccsbBroad304_08116	TBK1	IKK family			
802	86.6	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
803	86.59	cc		C2 domain containing protein kinases LOF	-			
804	86.59	cc		Leucine rich repeat kinase inhibitor	-			
805	86.59	oe	ccsbBroad304_06237	GAA	Glycosidases			
806	86.56	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
807	86.45	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
808	86.41	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
809	86.41	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
810	86.38	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
811	86.36	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
812	86.35	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
813	86.35	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
814	86.33	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
815	86.32	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
816	86.31	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
817	86.29	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
818	86.28	kd	CGS001-55802	DCP1A	-			
819	86.24	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
820	86.22	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
821	86.2	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
822	86.16	kd	CGS001-51380	CSAD	-			
823	86.14	kd	CGS001-51001	MTERFD1	-			
824	86.12	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
825	86.1	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
826	86.06	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
827	86.04	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
828	86.01	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
829	85.99	kd	CGS001-8864	PER2	-			
830	85.98	oe	ccsbBroad304_02432	IFI30	-			
831	85.97	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
832	85.95	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
833	85.95	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
834	85.89	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
835	85.86	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
836	85.75	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
837	85.69	kd	CGS001-9158	FIBP	-			
838	85.67	kd	CGS001-10007	GNPDA1	-			
839	85.61	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
840	85.58	oe	ccsbBroad304_00957	M6PR	-			
841	85.55	oe	ccsbBroad304_02686	COPZ1	-			
842	85.55	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
843	85.49	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
844	85.48	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
845	85.43	oe	ccsbBroad304_03874	UBL5	-			
846	85.41	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
847	85.39	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
848	85.39	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
849	85.34	kd	CGS001-23139	MAST2	MAST family			
850	85.34	kd	CGS001-1509	CTSD	Cathepsins			
851	85.29	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
852	85.27	kd	CGS001-3925	STMN1	-			
853	85.21	oe	ccsbBroad304_06098	DHCR24	-			
854	85.14	kd	CGS001-6050	RNH1	-			
855	85.1	kd	CGS001-11336	EXOC3	-			
856	85.05	oe	ccsbBroad304_12106	PXK	Slob family			
857	85.05	kd	CGS001-578	BAK1	-			
858	84.99	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
859	84.98	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
860	84.96	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
861	84.9	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
862	84.82	kd	CGS001-2538	G6PC	-			
863	84.8	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
864	84.77	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
865	84.69	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
866	84.68	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
867	84.6	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
868	84.59	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
869	84.58	oe	ccsbBroad304_02115	PTTG1	-			
870	84.43	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
871	84.34	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
872	84.33	kd	CGS001-3800	KIF5C	Kinesins			
873	84.26	oe	ccsbBroad304_01787	YES1	Src family			
874	84.25	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
875	84.18	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
876	84.15	kd	CGS001-56675	NRIP3	-			
877	84.14	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
878	84.11	oe	ccsbBroad304_03372	CAB39	-			
879	84.11	kd	CGS001-63948	DMRTB1	-			
880	84.02	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
881	83.99	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
882	83.92	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
883	83.91	kd	CGS001-6850	SYK	Syk family			
884	83.9	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
885	83.87	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
886	83.79	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
887	83.72	kd	CGS001-8848	TSC22D1	-			
888	83.64	kd	CGS001-3035	HARS	Aminoacyl tRNA synthetases / Class II			
889	83.58	oe	ccsbBroad304_05756	ACAA1	-			
890	83.58	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
891	83.53	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
892	83.53	kd	CGS001-538	ATP7A	ATPases / P-type			
893	83.46	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
894	83.46	kd	CGS001-1198	CLK3	CDC-like kinases			
895	83.4	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
896	83.37	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
897	83.34	oe	ccsbBroad304_06282	GLDC	-			
898	83.34	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
899	83.3	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
900	83.29	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
901	83.29	oe	ccsbBroad304_01623	SUPT4H1	-			
902	83.23	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
903	83.19	oe	ccsbBroad304_01054	GADD45B	-			
904	83.17	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
905	83.15	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
906	83.05	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
907	83.05	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
908	83.04	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
909	83.01	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
910	82.93	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
911	82.87	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
912	82.77	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
913	82.76	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
914	82.74	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
915	82.68	kd	CGS001-1659	DHX8	DEAH-boxes			
916	82.65	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
917	82.63	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
918	82.61	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
919	82.56	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
920	82.54	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
921	82.49	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
922	82.48	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
923	82.45	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
924	82.4	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
925	82.28	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
926	82.25	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
927	82.2	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
928	82.18	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
929	82.12	oe	ccsbBroad304_00933	LDHB	-			
930	82.05	kd	CGS001-1356	CP	-			
931	82.02	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
932	82	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
933	81.96	oe	ccsbBroad304_13939	MOK	RCK family			
934	81.96	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
935	81.87	kd	CGS001-10096	ACTR3	-			
936	81.86	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
937	81.85	oe	ccsbBroad304_06654	NPM1	-			
938	81.8	kd	CGS001-8895	CPNE3	-			
939	81.79	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
940	81.74	oe	ccsbBroad304_03072	GTPBP8	-			
941	81.72	oe	ccsbBroad304_06852	RBP4	Lipocalins			
942	81.71	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
943	81.7	oe	ccsbBroad304_03097	CNOT7	-			
944	81.69	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
945	81.67	kd	CGS001-328	APEX1	-			
946	81.65	kd	CGS001-24140	FTSJ1	-			
947	81.64	oe	ccsbBroad304_07920	NUP62	-			
948	81.62	oe	ccsbBroad304_00549	FDX1	-			
949	81.62	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
950	81.61	kd	CGS001-23678	SGK3	SGK family			
951	81.55	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
952	81.5	kd	CGS001-54442	KCTD5	-			
953	81.49	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
954	81.45	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
955	81.42	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
956	81.4	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
957	81.38	oe	ccsbBroad304_02741	PDS5A	-			
958	81.35	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
959	81.3	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
960	81.3	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
961	81.21	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
962	81.17	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
963	81.12	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
964	81.06	kd	CGS001-5144	PDE4D	Phosphodiesterases			
965	81.06	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
966	81.04	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
967	81.04	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
968	81.03	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
969	81.02	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
970	81.02	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
971	81	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
972	80.98	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
973	80.96	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
974	80.92	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
975	80.88	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
976	80.87	kd	CGS001-26298	EHF	-			
977	80.83	cc		VEGFR inhibitor	-			
978	80.78	kd	CGS001-4077	NBR1	-			
979	80.78	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
980	80.73	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
981	80.69	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
982	80.67	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
983	80.66	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
984	80.64	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
985	80.59	oe	ccsbBroad304_14174	CDKAL1	-			
986	80.57	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
987	80.53	kd	CGS001-151306	GPBAR1	Bile acid receptor			
988	80.43	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
989	80.42	oe	ccsbBroad304_08055	ATP5S	-			
990	80.4	kd	CGS001-2523	FUT1	Fucosyltransferases			
991	80.4	kd	CGS001-6347	CCL2	Chemokine ligands			
992	80.37	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
993	80.35	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
994	80.32	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
995	80.32	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
996	80.28	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
997	80.24	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
998	80.23	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
999	80.18	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
1000	80.09	kd	CGS001-55556	ENOSF1	-			
1001	79.99	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
1002	79.93	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
1003	79.84	kd	CGS001-8801	SUCLG2	-			
1004	79.81	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
1005	79.78	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
1006	79.77	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
1007	79.76	oe	ccsbBroad304_03405	CHRAC1	-			
1008	79.75	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
1009	79.68	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
1010	79.6	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
1011	79.56	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
1012	79.55	kd	CGS001-1195	CLK1	CDC-like kinases			
1013	79.52	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
1014	79.52	oe	ccsbBroad304_08825	LHPP	-			
1015	79.46	oe	ccsbBroad304_07094	TPMT	-			
1016	79.45	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
1017	79.45	kd	CGS001-965	CD58	CD molecules			
1018	79.41	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
1019	79.38	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
1020	79.31	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
1021	79.3	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
1022	79.28	kd	CGS001-64863	METTL4	-			
1023	79.25	oe	ccsbBroad304_01374	RAP1A	-			
1024	79.23	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
1025	79.22	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
1026	79.19	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
1027	79.13	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
1028	79.08	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
1029	78.91	oe	ccsbBroad304_02759	DICER1	-			
1030	78.85	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
1031	78.78	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
1032	78.7	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
1033	78.69	kd	CGS001-79109	MAPKAP1	-			
1034	78.68	cc		Beta-adrenergic receptor agonist	-			
1035	78.59	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
1036	78.59	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
1037	78.59	kd	CGS001-111	ADCY5	Adenylate cyclases			
1038	78.58	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
1039	78.53	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
1040	78.53	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
1041	78.5	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
1042	78.44	oe	ccsbBroad304_02578	EBNA1BP2	-			
1043	78.36	oe	ccsbBroad304_00359	CPT1A	-			
1044	78.2	kd	CGS001-340371	NRBP2	NRBP family			
1045	78.05	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
1046	78.02	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
1047	78.01	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
1048	77.9	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
1049	77.88	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
1050	77.88	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
1051	77.8	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
1052	77.79	oe	ccsbBroad304_02239	RASSF2	-			
1053	77.77	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
1054	77.73	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
1055	77.72	kd	CGS001-2109	ETFB	-			
1056	77.68	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
1057	77.58	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
1058	77.57	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1059	77.53	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
1060	77.52	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
1061	77.46	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
1062	77.46	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
1063	77.31	kd	CGS001-4616	GADD45B	-			
1064	77.29	kd	CGS001-2592	GALT	-			
1065	77.27	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
1066	77.23	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
1067	77.22	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
1068	77.2	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
1069	77.05	kd	CGS001-1072	CFL1	-			
1070	77.03	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
1071	77.02	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
1072	76.99	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
1073	76.96	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
1074	76.96	oe	ccsbBroad304_07798	EXOC3	-			
1075	76.92	oe	ccsbBroad304_01139	PA2G4	-			
1076	76.88	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
1077	76.84	kd	CGS001-506	ATP5B	ATPases / F-type			
1078	76.74	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
1079	76.72	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
1080	76.71	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
1081	76.68	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
1082	76.67	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
1083	76.66	kd	CGS001-388650	FAM69A	-			
1084	76.64	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
1085	76.61	kd	CGS001-10493	VAT1	-			
1086	76.6	oe	ccsbBroad304_13903	MTAP	-			
1087	76.58	oe	ccsbBroad304_13998	PDXK	-			
1088	76.56	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
1089	76.54	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
1090	76.52	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
1091	76.41	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
1092	76.38	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1093	76.36	kd	CGS001-103	ADAR	-			
1094	76.33	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
1095	76.33	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
1096	76.26	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
1097	76.25	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
1098	76.16	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
1099	76.16	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
1100	76.15	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
1101	76.15	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
1102	76.11	oe	ccsbBroad304_01061	NAB2	-			
1103	76.08	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
1104	75.98	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
1105	75.96	oe	ccsbBroad304_00424	DBI	-			
1106	75.94	oe	ccsbBroad304_14020	SH3BP5	-			
1107	75.93	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
1108	75.83	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
1109	75.78	oe	ccsbBroad304_03933	CARD9	-			
1110	75.73	kd	CGS001-79581	GPR172A	-			
1111	75.66	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
1112	75.64	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
1113	75.58	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
1114	75.54	oe	ccsbBroad304_07252	DGKZ	-			
1115	75.54	oe	ccsbBroad304_08104	MED4	-			
1116	75.53	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
1117	75.53	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
1118	75.52	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
1119	75.42	kd	CGS001-597	BCL2A1	-			
1120	75.38	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
1121	75.38	kd	CGS001-1119	CHKA	-			
1122	75.37	kd	CGS001-9170	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1123	75.34	kd	CGS001-8974	P4HA2	-			
1124	75.23	oe	ccsbBroad304_06349	HAGH	-			
1125	75.21	kd	CGS001-51271	UBAP1	-			
1126	75.08	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1127	75.07	cc		FGFR inhibitor	-			
1128	75.07	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
1129	75.07	kd	CGS001-4086	SMAD1	SMADs			
1130	75.06	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
1131	75.06	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
1132	75.06	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
1133	75	kd	CGS001-10329	TMEM5	-			
1134	74.99	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
1135	74.98	kd	CGS001-1376	CPT2	-			
1136	74.91	cc		Thymidylate synthase inhibitor	-			
1137	74.91	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
1138	74.9	oe	ccsbBroad304_02708	TRIM32	-			
1139	74.87	oe	ccsbBroad304_08426	TEX10	-			
1140	74.87	oe	ccsbBroad304_00098	ARG1	Arginase			
1141	74.86	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
1142	74.86	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
1143	74.84	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
1144	74.81	oe	ccsbBroad304_08452	PIH1D1	-			
1145	74.78	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
1146	74.77	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
1147	74.73	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
1148	74.67	oe	ccsbBroad304_07017	SUOX	-			
1149	74.66	kd	CGS001-63933	CCDC90A	-			
1150	74.61	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
1151	74.6	oe	ccsbBroad304_00570	FIGF	-			
1152	74.57	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
1153	74.53	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
1154	74.52	oe	ccsbBroad304_00001	NAT1	-			
1155	74.49	kd	CGS001-1948	EFNB2	Ephrins			
1156	74.47	kd	CGS001-5236	PGM1	-			
1157	74.46	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
1158	74.46	kd	CGS001-7917	BAG6	-			
1159	74.43	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
1160	74.43	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
1161	74.41	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1162	74.4	kd	CGS001-150094	SIK1	QIK subfamily			
1163	74.38	oe	ccsbBroad304_06264	GBP2	-			
1164	74.35	oe	ccsbBroad304_02804	KLHDC2	-			
1165	74.34	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
1166	74.3	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
1167	74.27	kd	CGS001-873	CBR1	Prostaglandin synthases			
1168	74.23	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
1169	74.21	cc		HIV protease inhibitor	-			
1170	74.2	kd	CGS001-57026	PDXP	-			
1171	74.18	kd	CGS001-6477	SIAH1	-			
1172	74.18	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
1173	74.1	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
1174	74.09	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
1175	74.07	cc		Retinoid receptor agonist	-			
1176	74.07	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
1177	74.07	kd	CGS001-9412	MED21	-			
1178	73.99	kd	CGS001-2768	GNA12	-			
1179	73.98	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
1180	73.97	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
1181	73.95	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
1182	73.92	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
1183	73.77	kd	CGS001-7374	UNG	-			
1184	73.74	kd	CGS001-7849	PAX8	Paired boxes			
1185	73.71	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
1186	73.71	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
1187	73.7	oe	ccsbBroad304_02566	MORF4L1	-			
1188	73.63	kd	CGS001-8805	TRIM24	TIF1 family			
1189	73.63	kd	CGS001-10928	RALBP1	-			
1190	73.6	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
1191	73.56	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
1192	73.55	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
1193	73.53	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
1194	73.53	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
1195	73.52	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1196	73.51	kd	CGS001-5105	PCK1	-			
1197	73.51	kd	CGS001-2335	FN1	Endogenous ligands			
1198	73.5	kd	CGS001-51097	SCCPDH	-			
1199	73.47	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
1200	73.39	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1201	73.37	kd	CGS001-2731	GLDC	-			
1202	73.34	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
1203	73.32	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
1204	73.31	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
1205	73.3	kd	CGS001-116832	RPL39L	L ribosomal proteins			
1206	73.29	oe	ccsbBroad304_01234	POLB	DNA polymerases			
1207	73.28	kd	CGS001-2159	F10	Chymotrypsin			
1208	73.18	kd	CGS001-7057	THBS1	-			
1209	73.17	kd	CGS001-5037	PEBP1	-			
1210	73.16	kd	CGS001-10452	TOMM40	-			
1211	73.09	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
1212	73.09	kd	CGS001-1676	DFFA	-			
1213	73.08	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
1214	73.06	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
1215	73.05	kd	CGS001-29978	UBQLN2	Ubiquilin family			
1216	73.03	kd	CGS001-3978	LIG1	-			
1217	73	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
1218	73	kd	CGS001-23530	NNT	-			
1219	72.99	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
1220	72.98	oe	ccsbBroad304_03848	METTL14	-			
1221	72.96	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
1222	72.95	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
1223	72.95	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1224	72.92	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
1225	72.88	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
1226	72.87	oe	ccsbBroad304_02287	GNPDA1	-			
1227	72.86	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
1228	72.85	kd	CGS001-3566	IL4R	IL-2 receptor family			
1229	72.79	oe	ccsbBroad304_06048	CRYZ	-			
1230	72.76	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
1231	72.68	oe	ccsbBroad304_07922	TRIM29	-			
1232	72.68	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
1233	72.67	oe	ccsbBroad304_06562	MAT1A	-			
1234	72.67	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
1235	72.66	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
1236	72.63	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
1237	72.62	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1238	72.62	kd	CGS001-3131	HLF	-			
1239	72.58	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
1240	72.56	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
1241	72.54	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
1242	72.48	kd	CGS001-8649	LAMTOR3	-			
1243	72.44	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
1244	72.4	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1245	72.39	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
1246	72.39	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
1247	72.32	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
1248	72.31	kd	CGS001-4121	MAN1A1	-			
1249	72.3	kd	CGS001-5050	PAFAH1B3	-			
1250	72.29	kd	CGS001-4151	MB	-			
1251	72.26	oe	ccsbBroad304_00370	CS	-			
1252	72.2	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
1253	72.2	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
1254	72.08	oe	ccsbBroad304_03266	ERGIC2	-			
1255	72.03	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1256	72.02	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
1257	72.01	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
1258	71.82	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
1259	71.81	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
1260	71.8	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
1261	71.73	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
1262	71.7	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
1263	71.65	oe	ccsbBroad304_02419	NDRG1	-			
1264	71.61	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
1265	71.56	kd	CGS001-11325	DDX42	DEAD-boxes			
1266	71.56	oe	ccsbBroad304_08045	NOX1	-			
1267	71.55	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
1268	71.51	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
1269	71.49	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
1270	71.46	kd	CGS001-55179	FAIM	-			
1271	71.42	kd	CGS001-30	ACAA1	-			
1272	71.4	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
1273	71.38	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
1274	71.35	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
1275	71.32	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
1276	71.32	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
1277	71.32	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
1278	71.24	kd	CGS001-4088	SMAD3	SMADs			
1279	71.23	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
1280	71.2	oe	ccsbBroad304_03878	SENP2	-			
1281	71.08	oe	ccsbBroad304_04786	CANT1	-			
1282	71	kd	CGS001-10904	BLCAP	-			
1283	71	kd	CGS001-367	AR	Nuclear hormone receptors			
1284	70.97	oe	ccsbBroad304_02756	RRP8	-			
1285	70.94	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
1286	70.93	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
1287	70.92	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
1288	70.88	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
1289	70.85	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
1290	70.85	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
1291	70.81	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
1292	70.81	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
1293	70.8	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
1294	70.79	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
1295	70.76	kd	CGS001-2475	MTOR	FRAP subfamily			
1296	70.74	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
1297	70.59	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
1298	70.5	kd	CGS001-5164	PDK2	PDHK family			
1299	70.42	oe	ccsbBroad304_00509	EPHX1	-			
1300	70.42	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
1301	70.41	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
1302	70.39	kd	CGS001-55176	SEC61A2	-			
1303	70.38	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
1304	70.29	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
1305	70.27	oe	ccsbBroad304_00150	BAX	-			
1306	70.25	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
1307	70.19	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
1308	70.11	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
1309	70.09	kd	CGS001-665	BNIP3L	-			
1310	70.05	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
1311	70.05	kd	CGS001-2023	ENO1	-			
1312	70.01	oe	ccsbBroad304_08167	DNTTIP2	-			
1313	70.01	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
1314	70.01	kd	CGS001-10972	TMED10	-			
1315	70.01	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
1316	69.92	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
1317	69.89	kd	CGS001-2961	GTF2E2	General transcription factors			
1318	69.88	oe	ccsbBroad304_07478	CCP110	-			
1319	69.86	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
1320	69.85	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
1321	69.85	kd	CGS001-23161	SNX13	Sorting nexins			
1322	69.84	oe	ccsbBroad304_02361	MFSD10	-			
1323	69.83	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
1324	69.78	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
1325	69.76	cc		PDGFR/KIT inhibitor	-			
1326	69.76	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
1327	69.76	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1328	69.71	kd	CGS001-4700	NDUFA6	LYR motif containing			
1329	69.64	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
1330	69.58	oe	ccsbBroad304_02604	B3GNT1	-			
1331	69.56	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
1332	69.31	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
1333	69.22	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
1334	69.22	kd	CGS001-8220	DGCR14	-			
1335	69.19	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
1336	69.14	oe	ccsbBroad304_03910	CCDC90A	-			
1337	69.13	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
1338	69.13	kd	CGS001-949	SCARB1	-			
1339	69.12	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1340	69.08	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
1341	69.01	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
1342	68.96	kd	CGS001-6832	SUPV3L1	-			
1343	68.91	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
1344	68.89	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
1345	68.88	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
1346	68.81	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
1347	68.77	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
1348	68.66	oe	ccsbBroad304_00006	ACADM	-			
1349	68.66	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
1350	68.63	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1351	68.63	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
1352	68.56	kd	CGS001-4734	NEDD4	-			
1353	68.52	kd	CGS001-64077	LHPP	-			
1354	68.51	oe	ccsbBroad304_03113	DSE	-			
1355	68.49	cc		IMPDH inhibitor	-			
1356	68.49	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
1357	68.4	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
1358	68.38	kd	CGS001-6723	SRM	-			
1359	68.28	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
1360	68.24	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
1361	68.19	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
1362	68.19	kd	CGS001-25874	BRP44	-			
1363	68.17	kd	CGS001-58472	SQRDL	-			
1364	68.15	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
1365	68.15	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
1366	68.1	kd	CGS001-26292	MYCBP	-			
1367	68.1	kd	CGS001-4144	MAT2A	-			
1368	68.07	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
1369	67.95	kd	CGS001-10513	APPBP2	-			
1370	67.85	kd	CGS001-255738	PCSK9	Subtilisin			
1371	67.84	kd	CGS001-9967	THRAP3	-			
1372	67.76	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
1373	67.72	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
1374	67.69	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
1375	67.67	oe	ccsbBroad304_02047	AP1S2	-			
1376	67.67	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
1377	67.67	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
1378	67.62	cc		MEK inhibitor	-			
1379	67.57	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
1380	67.54	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
1381	67.54	kd	CGS001-10810	WASF3	-			
1382	67.53	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
1383	67.52	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
1384	67.5	oe	ccsbBroad304_00423	DAXX	-			
1385	67.49	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
1386	67.43	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
1387	67.43	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
1388	67.42	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
1389	67.39	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
1390	67.38	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
1391	67.36	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
1392	67.34	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
1393	67.28	oe	ccsbBroad304_00836	IGF2	-			
1394	67.23	cc		FLT3 inhibitor	-			
1395	67.21	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
1396	67.15	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
1397	67.12	cc		Sigma receptor antagonist	-			
1398	67.08	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
1399	67.01	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
1400	66.94	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
1401	66.94	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
1402	66.93	kd	CGS001-5900	RALGDS	-			
1403	66.89	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
1404	66.88	kd	CGS001-7029	TFDP2	-			
1405	66.82	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
1406	66.81	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
1407	66.77	kd	CGS001-133690	CAPSL	EF-hand domain containing			
1408	66.7	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
1409	66.62	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
1410	66.61	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
1411	66.53	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
1412	66.51	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
1413	66.5	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
1414	66.35	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1415	66.28	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
1416	66.19	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
1417	66.18	oe	ccsbBroad304_00874	INS	-			
1418	66.15	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
1419	66.1	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
1420	66.09	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
1421	66.06	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
1422	66.04	oe	ccsbBroad304_06718	PFN2	-			
1423	66.04	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
1424	66.04	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
1425	66.01	kd	CGS001-57147	SCYL3	-			
1426	65.95	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
1427	65.89	kd	CGS001-7353	UFD1L	-			
1428	65.86	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
1429	65.84	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
1430	65.8	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
1431	65.76	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
1432	65.56	oe	ccsbBroad304_06172	EPS8	-			
1433	65.55	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
1434	65.52	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
1435	65.51	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
1436	65.46	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1437	65.43	kd	CGS001-9531	BAG3	-			
1438	65.37	oe	ccsbBroad304_07569	TRIB1	Trbl family			
1439	65.36	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
1440	65.35	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
1441	65.31	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
1442	65.29	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
1443	65.28	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
1444	65.27	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
1445	65.26	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
1446	65.14	kd	CGS001-8050	PDHX	-			
1447	65.11	kd	CGS001-7295	TXN	-			
1448	65.07	kd	CGS001-3676	ITGA4	Integrins			
1449	65.06	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
1450	65.05	oe	ccsbBroad304_05098	MAGEB6	-			
1451	65.02	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1452	65.01	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
1453	64.98	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
1454	64.91	kd	CGS001-378	ARF4	ADP-ribosylation factors			
1455	64.82	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
1456	64.8	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
1457	64.79	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
1458	64.77	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
1459	64.75	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
1460	64.68	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
1461	64.67	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
1462	64.64	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
1463	64.62	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
1464	64.61	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
1465	64.53	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
1466	64.45	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1467	64.44	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
1468	64.42	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
1469	64.33	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
1470	64.32	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1471	64.24	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
1472	64.23	oe	ccsbBroad304_02553	BLCAP	-			
1473	64.17	oe	ccsbBroad304_01398	RHEB	-			
1474	64.13	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
1475	64.12	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
1476	64.11	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
1477	64.09	kd	CGS001-11284	PNKP	-			
1478	64.06	kd	CGS001-10691	GMEB1	-			
1479	63.97	kd	CGS001-4221	MEN1	-			
1480	63.82	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
1481	63.8	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
1482	63.77	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
1483	63.74	oe	ccsbBroad304_00648	GLRX	-			
1484	63.72	oe	ccsbBroad304_00819	IDH3B	-			
1485	63.61	oe	ccsbBroad304_01114	NUP88	-			
1486	63.61	kd	CGS001-10447	FAM3C	-			
1487	63.6	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
1488	63.6	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
1489	63.55	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
1490	63.5	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
1491	63.49	oe	ccsbBroad304_02026	NRP1	CD molecules			
1492	63.48	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
1493	63.4	kd	CGS001-23585	TMEM50A	-			
1494	63.39	cc		Bromodomain Inhibitor	-			
1495	63.36	oe	ccsbBroad304_07890	CBX7	-			
1496	63.29	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
1497	63.25	oe	ccsbBroad304_06278	GK	Glycerol kinases			
1498	63.19	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
1499	63.17	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
1500	63.16	kd	CGS001-2113	ETS1	ETS Transcription Factors			
1501	63.05	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
1502	62.96	oe	ccsbBroad304_00876	INSIG1	-			
1503	62.96	oe	ccsbBroad304_04471	C5ORF62	-			
1504	62.95	kd	CGS001-6714	SRC	Src family			
1505	62.93	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
1506	62.92	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
1507	62.83	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
1508	62.81	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
1509	62.8	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
1510	62.8	kd	CGS001-4946	OAZ1	-			
1511	62.8	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
1512	62.75	kd	CGS001-2295	FOXF2	Forkhead boxes			
1513	62.74	kd	CGS001-8841	HDAC3	Histone deacetylases			
1514	62.72	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
1515	62.69	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
1516	62.62	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1517	62.53	oe	ccsbBroad304_07808	RAB11FIP2	-			
1518	62.52	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
1519	62.51	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
1520	62.48	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
1521	62.41	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
1522	62.41	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
1523	62.37	kd	CGS001-55612	FERMT1	Fermitins			
1524	62.35	kd	CGS001-1105	CHD1	-			
1525	62.34	oe	ccsbBroad304_04616	ORMDL3	-			
1526	62.34	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
1527	62.33	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
1528	62.29	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
1529	62.19	kd	CGS001-7292	TNFSF4	CD molecules			
1530	62.18	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
1531	62.17	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
1532	62.17	kd	CGS001-3033	HADH	-			
1533	62.15	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
1534	62.1	kd	CGS001-11151	CORO1A	Coronins			
1535	62.07	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
1536	62.07	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
1537	61.96	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
1538	61.91	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
1539	61.87	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
1540	61.82	kd	CGS001-9697	TRAM2	-			
1541	61.8	oe	ccsbBroad304_02922	TES	-			
1542	61.78	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
1543	61.72	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
1544	61.67	kd	CGS001-6884	TAF13	-			
1545	61.61	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
1546	61.6	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
1547	61.6	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
1548	61.56	kd	CGS001-32	ACACB	Carboxylases			
1549	61.54	kd	CGS001-4170	MCL1	-			
1550	61.53	oe	ccsbBroad304_01373	RAN	-			
1551	61.48	oe	ccsbBroad304_03808	ERGIC1	-			
1552	61.47	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
1553	61.46	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
1554	61.45	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
1555	61.43	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
1556	61.41	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
1557	61.39	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
1558	61.38	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
1559	61.38	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
1560	61.34	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
1561	61.33	cc		Topoisomerase inhibitor	-			
1562	61.26	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
1563	61.22	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
1564	61.2	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
1565	61.19	kd	CGS001-255877	BCL6B	BTB/POZ domain containing			
1566	61.16	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1567	61.03	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
1568	61.01	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
1569	61.01	kd	CGS001-23464	GCAT	-			
1570	60.99	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
1571	60.99	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
1572	60.89	cp	BRD-A71009679	KUC103420N	-666			-666
1573	60.84	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
1574	60.82	oe	ccsbBroad304_02452	NXF1	-			
1575	60.81	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
1576	60.8	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
1577	60.76	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
1578	60.75	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
1579	60.71	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
1580	60.7	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
1581	60.69	cc		C2 domain containing LOF	-			
1582	60.67	oe	ccsbBroad304_03232	VPS28	-			
1583	60.62	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
1584	60.6	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
1585	60.58	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
1586	60.53	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
1587	60.53	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1588	60.49	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
1589	60.47	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1590	60.45	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
1591	60.4	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
1592	60.34	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
1593	60.3	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
1594	60.28	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
1595	60.25	oe	ccsbBroad304_03640	CEP72	-			
1596	60.25	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
1597	60.13	kd	CGS001-161	AP2A2	-			
1598	60.11	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
1599	60.1	kd	CGS001-2745	GLRX	-			
1600	60.08	kd	CGS001-306	ANXA3	Annexins			
1601	60.03	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
1602	59.96	oe	ccsbBroad304_07766	RASSF1	-			
1603	59.96	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
1604	59.8	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
1605	59.76	oe	ccsbBroad304_14047	TACC3	-			
1606	59.76	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
1607	59.64	oe	ccsbBroad304_04788	OVCA2	-			
1608	59.64	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
1609	59.62	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
1610	59.54	oe	ccsbBroad304_00960	SMAD1	SMADs			
1611	59.47	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
1612	59.42	kd	CGS001-81848	SPRY4	-			
1613	59.41	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
1614	59.39	oe	ccsbBroad304_03118	NRBP1	NRBP family			
1615	59.3	cc		Interleukin receptors LOF	-			
1616	59.3	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
1617	59.27	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
1618	59.24	oe	ccsbBroad304_06569	MCM5	-			
1619	59.24	oe	ccsbBroad304_02398	LANCL1	-			
1620	59.17	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
1621	59.16	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
1622	59.13	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
1623	59.1	oe	ccsbBroad304_00100	RHOA	-			
1624	59.1	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
1625	59.08	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
1626	59.06	kd	CGS001-3927	LASP1	-			
1627	59.04	kd	CGS001-3098	HK1	-			
1628	58.99	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1629	58.96	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
1630	58.96	kd	CGS001-57787	MARK4	MARK subfamily			
1631	58.93	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1632	58.92	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
1633	58.9	kd	CGS001-205	AK4	Adenylate kinases			
1634	58.88	oe	ccsbBroad304_06870	RNH1	-			
1635	58.83	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
1636	58.82	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
1637	58.79	cc		HRH1 antagonist	-			
1638	58.73	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
1639	58.72	oe	ccsbBroad304_06739	PLOD1	-			
1640	58.62	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
1641	58.49	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
1642	58.49	kd	CGS001-54108	CHRAC1	-			
1643	58.41	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
1644	58.4	kd	CGS001-2037	EPB41L2	-			
1645	58.35	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
1646	58.29	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
1647	58.18	oe	ccsbBroad304_07238	STK24	YSK subfamily			
1648	58	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
1649	57.98	kd	CGS001-3659	IRF1	-			
1650	57.97	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
1651	57.93	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
1652	57.92	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
1653	57.87	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
1654	57.87	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
1655	57.87	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
1656	57.82	cc		SRY LOF	-			
1657	57.8	oe	ccsbBroad304_08339	CMPK1	-			
1658	57.8	kd	CGS001-587	BCAT2	-			
1659	57.79	kd	CGS001-84722	PSRC1	-			
1660	57.74	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
1661	57.73	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
1662	57.72	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
1663	57.72	kd	CGS001-9374	PPT2	-			
1664	57.71	kd	CGS001-2244	FGB	Endogenous ligands			
1665	57.7	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
1666	57.63	kd	CGS001-5373	PMM2	-			
1667	57.54	cc		PI3K Signaling LOF	-			
1668	57.54	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
1669	57.54	kd	CGS001-1497	CTNS	-			
1670	57.53	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
1671	57.49	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
1672	57.47	kd	CGS001-3481	IGF2	-			
1673	57.41	kd	CGS001-9128	PRPF4	WD repeat domain containing			
1674	57.41	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
1675	57.4	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
1676	57.39	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
1677	57.36	oe	ccsbBroad304_01163	PDHA1	-			
1678	57.35	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
1679	57.29	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
1680	57.27	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
1681	57.25	oe	ccsbBroad304_01150	PCCB	Carboxylases			
1682	57.23	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
1683	57.21	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
1684	57.15	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
1685	57.14	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
1686	57.07	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
1687	57.06	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
1688	57.03	kd	CGS001-1362	CPD	Carboxypeptidase A			
1689	57.02	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
1690	57.01	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
1691	56.93	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
1692	56.93	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
1693	56.92	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
1694	56.85	oe	ccsbBroad304_01754	UCK2	-			
1695	56.82	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
1696	56.82	oe	ccsbBroad304_08709	SCYL3	-			
1697	56.8	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
1698	56.77	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
1699	56.72	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
1700	56.7	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
1701	56.7	kd	CGS001-4811	NID1	-			
1702	56.63	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1703	56.63	kd	CGS001-1120	CHKB	-			
1704	56.62	oe	ccsbBroad304_00783	HPRT1	-			
1705	56.57	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
1706	56.55	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
1707	56.53	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
1708	56.5	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
1709	56.47	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1710	56.39	kd	CGS001-8835	SOCS2	SH2 domain containing			
1711	56.37	oe	ccsbBroad304_01143	PAFAH1B3	-			
1712	56.36	oe	ccsbBroad304_03182	GLOD4	-			
1713	56.34	cc		MDM inhibitor	-			
1714	56.33	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
1715	56.25	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
1716	56.24	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
1717	56.21	kd	CGS001-55437	STRADB	STLK subfamily			
1718	56.19	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
1719	56.12	oe	ccsbBroad304_02572	SERINC3	-			
1720	56.09	kd	CGS001-4176	MCM7	-			
1721	56.07	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
1722	56.01	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
1723	56	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1724	55.97	oe	ccsbBroad304_09035	COASY	-			
1725	55.97	kd	CGS001-10018	BCL2L11	-			
1726	55.95	kd	CGS001-56731	SLC2A4RG	-			
1727	55.91	cc		Cyclooxygenase inhibitor	-			
1728	55.74	cc		Vitamin D receptor agonist	-			
1729	55.71	kd	CGS001-1837	DTNA	-			
1730	55.62	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
1731	55.6	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
1732	55.55	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
1733	55.55	kd	CGS001-9447	AIM2	-			
1734	55.52	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
1735	55.52	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
1736	55.49	oe	ccsbBroad304_08386	SMOX	-			
1737	55.45	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
1738	55.44	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
1739	55.43	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
1740	55.42	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1741	55.36	kd	CGS001-2550	GABBR1	GABA receptors			
1742	55.24	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
1743	55.21	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
1744	55.2	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
1745	55.19	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
1746	55.13	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
1747	55.12	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
1748	55.11	cc		Tumor necrosis factor superfamily LOF	-			
1749	55.09	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
1750	55.08	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
1751	55.02	oe	ccsbBroad304_01841	BAG6	-			
1752	54.94	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
1753	54.92	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
1754	54.88	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1755	54.86	oe	ccsbBroad304_06720	PHYH	-			
1756	54.85	oe	ccsbBroad304_01855	NCOA4	-			
1757	54.82	kd	CGS001-308	ANXA5	Annexins			
1758	54.8	kd	CGS001-10198	MPHOSPH9	-			
1759	54.72	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
1760	54.7	kd	CGS001-7311	UBA52	L ribosomal proteins			
1761	54.65	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
1762	54.62	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
1763	54.58	oe	ccsbBroad304_06574	MDH2	-			
1764	54.57	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
1765	54.55	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
1766	54.52	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
1767	54.51	oe	ccsbBroad304_08536	PARL	-			
1768	54.48	oe	ccsbBroad304_02057	P4HA2	-			
1769	54.48	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
1770	54.48	kd	CGS001-80347	COASY	-			
1771	54.41	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
1772	54.41	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
1773	54.4	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
1774	54.39	kd	CGS001-4122	MAN2A2	-			
1775	54.37	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1776	54.37	kd	CGS001-1788	DNMT3A	Methyltransferases			
1777	54.35	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
1778	54.34	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
1779	54.32	kd	CGS001-624	BDKRB2	Bradykinin receptors			
1780	54.31	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
1781	54.25	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
1782	54.25	kd	CGS001-23014	FBXO21	F-boxes / other			
1783	54.2	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
1784	54.17	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
1785	54.12	kd	CGS001-161725	OTUD7A	OTU domain containing			
1786	54.1	kd	CGS001-7105	TSPAN6	Tetraspanins			
1787	54.1	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
1788	54.04	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
1789	54	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
1790	53.97	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
1791	53.94	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
1792	53.93	kd	CGS001-3664	IRF6	-			
1793	53.86	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
1794	53.86	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
1795	53.83	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
1796	53.79	oe	ccsbBroad304_07768	NISCH	-			
1797	53.79	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
1798	53.76	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
1799	53.72	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
1800	53.63	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
1801	53.63	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
1802	53.62	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
1803	53.59	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1804	53.58	oe	ccsbBroad304_05985	CFL1	-			
1805	53.57	oe	ccsbBroad304_01186	PHB	-			
1806	53.56	oe	ccsbBroad304_00120	ATOX1	-			
1807	53.55	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
1808	53.53	kd	CGS001-1605	DAG1	-			
1809	53.51	kd	CGS001-23636	NUP62	-			
1810	53.43	kd	CGS001-169841	ZNF169	Zinc fingers, C2H2-type			
1811	53.41	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
1812	53.32	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1813	53.3	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
1814	53.3	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
1815	53.28	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1816	53.21	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
1817	53.18	kd	CGS001-10298	PAK4	PAKB subfamily			
1818	53.14	kd	CGS001-29110	TBK1	IKK family			
1819	53.07	oe	ccsbBroad304_08684	CXCR7	-			
1820	53.06	kd	CGS001-25819	CCRN4L	-			
1821	53.05	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
1822	53.04	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1823	53	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
1824	52.95	oe	ccsbBroad304_07362	NMI	-			
1825	52.92	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
1826	52.84	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
1827	52.84	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
1828	52.8	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
1829	52.72	cc		Supressors of cytokine signaling GOF	-			
1830	52.72	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
1831	52.68	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
1832	52.67	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
1833	52.64	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
1834	52.63	kd	CGS001-3685	ITGAV	Integrins			
1835	52.62	oe	ccsbBroad304_07280	LAMTOR3	-			
1836	52.6	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
1837	52.56	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
1838	52.51	kd	CGS001-7919	DDX39B	DEAD-boxes			
1839	52.5	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
1840	52.49	cc		Akt Signaling GOF	-			
1841	52.36	kd	CGS001-11340	EXOSC8	-			
1842	52.34	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
1843	52.34	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
1844	52.3	kd	CGS001-4232	MEST	-			
1845	52.28	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
1846	52.22	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1847	52.09	kd	CGS001-435	ASL	-			
1848	52.04	oe	ccsbBroad304_02565	RALBP1	-			
1849	51.99	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
1850	51.98	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1851	51.98	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
1852	51.96	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
1853	51.86	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1854	51.85	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1855	51.85	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
1856	51.83	oe	ccsbBroad304_04379	LZIC	-			
1857	51.72	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
1858	51.7	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
1859	51.69	cc		TGF beta receptor inhibitor	-			
1860	51.69	oe	ccsbBroad304_01832	PAX8	Paired boxes			
1861	51.68	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
1862	51.65	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
1863	51.64	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1864	51.62	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
1865	51.61	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
1866	51.6	oe	ccsbBroad304_07140	XPC	-			
1867	51.6	kd	CGS001-5682	PSMA1	Proteasome subunits			
1868	51.54	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
1869	51.41	kd	CGS001-80349	WDR61	WD repeat domain containing			
1870	51.38	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
1871	51.36	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
1872	51.29	cc		SRC inhibitor	-			
1873	51.29	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
1874	51.28	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
1875	51.25	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
1876	51.21	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
1877	51.18	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
1878	51.16	kd	CGS001-6601	SMARCC2	-			
1879	51.13	kd	CGS001-1465	CSRP1	-			
1880	51.1	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
1881	51.09	oe	ccsbBroad304_07632	PROCR	CD molecules			
1882	51.08	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1883	51.06	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
1884	51.03	kd	CGS001-5053	PAH	Amino acid hydroxylases			
1885	50.95	oe	ccsbBroad304_04038	ELOVL6	-			
1886	50.95	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
1887	50.92	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
1888	50.9	oe	ccsbBroad304_01576	SOAT1	-			
1889	50.88	oe	ccsbBroad304_05823	ANXA2	Annexins			
1890	50.86	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
1891	50.84	kd	CGS001-6857	SYT1	Synaptotagmins			
1892	50.79	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
1893	50.72	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
1894	50.71	kd	CGS001-10284	SAP18	-			
1895	50.71	kd	CGS001-3418	IDH2	-			
1896	50.66	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
1897	50.62	kd	CGS001-56889	TM9SF3	-			
1898	50.54	oe	ccsbBroad304_01164	PDHB	-			
1899	50.5	oe	ccsbBroad304_06424	IFI16	-			
1900	50.49	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
1901	50.48	kd	CGS001-5883	RAD9A	-			
1902	50.47	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
1903	50.44	kd	CGS001-57222	ERGIC1	-			
1904	50.4	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
1905	50.38	oe	ccsbBroad304_02425	CDIPT	-			
1906	50.36	oe	ccsbBroad304_02002	RNMT	-			
1907	50.31	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1908	50.3	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
1909	50.29	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
1910	50.26	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
1911	50.23	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
1912	50.16	oe	ccsbBroad304_02955	MYCBP	-			
1913	50.13	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
1914	50.12	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
1915	50.07	cc		Vesicular Transport LOF	-			
1916	50.07	cc		Potassium channel blocker	-			
1917	49.94	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
1918	49.94	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
1919	49.92	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
1920	49.91	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
1921	49.9	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
1922	49.84	oe	ccsbBroad304_06040	CRY1	-			
1923	49.81	kd	CGS001-64094	SMOC2	EF-hand domain containing			
1924	49.8	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
1925	49.72	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
1926	49.67	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
1927	49.65	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1928	49.62	kd	CGS001-64943	NT5DC2	-			
1929	49.6	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
1930	49.51	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
1931	49.5	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1932	49.49	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
1933	49.44	kd	CGS001-6871	TADA2A	-			
1934	49.42	kd	CGS001-2771	GNAI2	-			
1935	49.42	kd	CGS001-701	BUB1B	Bub family			
1936	49.3	cc		Tachykinin antagonist	-			
1937	49.3	oe	ccsbBroad304_03428	EXOSC4	-			
1938	49.3	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
1939	49.26	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
1940	49.25	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
1941	49.24	kd	CGS001-3689	ITGB2	Integrins			
1942	49.23	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
1943	49.21	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
1944	49.2	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
1945	49.17	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
1946	49.17	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
1947	49.16	kd	CGS001-54899	PXK	Slob family			
1948	49.13	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
1949	49.11	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
1950	49.11	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
1951	49.1	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
1952	49.09	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
1953	49.06	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
1954	49.01	kd	CGS001-8872	CDC123	-			
1955	48.99	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
1956	48.99	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
1957	48.98	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
1958	48.98	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
1959	48.96	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
1960	48.85	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
1961	48.81	oe	ccsbBroad304_04399	PGBD1	-			
1962	48.76	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
1963	48.72	oe	ccsbBroad304_04404	TUBB6	Tubulins			
1964	48.71	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
1965	48.69	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
1966	48.68	kd	CGS001-26227	PHGDH	-			
1967	48.47	kd	CGS001-54623	PAF1	-			
1968	48.43	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1969	48.43	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
1970	48.43	kd	CGS001-3995	FADS3	Fatty acid desaturases			
1971	48.37	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
1972	48.36	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
1973	48.29	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
1974	48.28	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
1975	48.25	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
1976	48.24	kd	CGS001-5831	PYCR1	-			
1977	48.23	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
1978	48.23	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
1979	48.23	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1980	48.2	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
1981	48.2	kd	CGS001-5898	RALA	-			
1982	48.1	oe	ccsbBroad304_09615	LACC1	-			
1983	48.07	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
1984	48.05	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
1985	48.04	kd	CGS001-23658	LSM5	-			
1986	47.98	oe	ccsbBroad304_07515	GFPT2	-			
1987	47.98	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
1988	47.96	kd	CGS001-23650	TRIM29	-			
1989	47.92	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
1990	47.9	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
1991	47.86	kd	CGS001-2108	ETFA	-			
1992	47.84	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
1993	47.83	oe	ccsbBroad304_10431	HADHB	-			
1994	47.83	kd	CGS001-6598	SMARCB1	-			
1995	47.81	oe	ccsbBroad304_02633	LSM6	-			
1996	47.75	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
1997	47.71	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
1998	47.7	oe	ccsbBroad304_05152	SSBP4	-			
1999	47.67	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
2000	47.67	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
2001	47.67	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
2002	47.66	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
2003	47.64	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
2004	47.61	oe	ccsbBroad304_08662	MCCC1	-			
2005	47.57	kd	CGS001-4976	OPA1	-			
2006	47.5	kd	CGS001-23077	MYCBP2	-			
2007	47.5	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
2008	47.49	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
2009	47.44	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
2010	47.44	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
2011	47.24	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
2012	47.22	kd	CGS001-200734	SPRED2	-			
2013	47.18	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
2014	47.16	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
2015	47.15	oe	ccsbBroad304_03080	C16ORF80	-			
2016	47.1	kd	CGS001-8624	PSMG1	-			
2017	47.07	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
2018	47.05	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
2019	47.02	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
2020	47.02	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
2021	47.02	oe	ccsbBroad304_02052	KYNU	-			
2022	46.98	kd	CGS001-4299	AFF1	-			
2023	46.96	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
2024	46.93	oe	ccsbBroad304_02058	PLOD3	-			
2025	46.87	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
2026	46.86	oe	ccsbBroad304_08093	DCPS	-			
2027	46.85	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
2028	46.85	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
2029	46.85	kd	CGS001-3590	IL11RA	IL-6 receptor family			
2030	46.8	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
2031	46.71	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
2032	46.7	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
2033	46.7	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
2034	46.68	oe	ccsbBroad304_12008	NLK	nmo subfamily			
2035	46.67	kd	CGS001-2356	FPGS	-			
2036	46.66	oe	ccsbBroad304_01613	STK11	LKB subfamily			
2037	46.66	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
2038	46.64	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
2039	46.64	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
2040	46.64	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
2041	46.6	oe	ccsbBroad304_06287	GM2A	-			
2042	46.59	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
2043	46.49	kd	CGS001-27161	EIF2C2	-			
2044	46.48	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
2045	46.46	oe	ccsbBroad304_04465	RERG	-			
2046	46.44	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
2047	46.44	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
2048	46.43	oe	ccsbBroad304_02205	WTAP	-			
2049	46.4	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
2050	46.4	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
2051	46.4	kd	CGS001-896	CCND3	-			
2052	46.36	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
2053	46.32	kd	CGS001-1727	CYB5R3	-			
2054	46.31	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
2055	46.27	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
2056	46.25	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
2057	46.24	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
2058	46.24	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
2059	46.24	kd	CGS001-29940	DSE	-			
2060	46.19	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
2061	46.18	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
2062	46.14	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
2063	46.12	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2064	46.07	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
2065	46.06	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
2066	46.03	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
2067	45.97	oe	ccsbBroad304_03565	ADI1	-			
2068	45.92	kd	CGS001-571	BACH1	BTB/POZ domain containing			
2069	45.91	oe	ccsbBroad304_06140	EEF1D	-			
2070	45.87	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
2071	45.86	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
2072	45.85	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
2073	45.82	kd	CGS001-29083	GTPBP8	-			
2074	45.78	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
2075	45.75	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
2076	45.72	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
2077	45.71	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
2078	45.64	oe	ccsbBroad304_02485	STAMBP	-			
2079	45.64	kd	CGS001-9847	KIAA0528	-			
2080	45.64	kd	CGS001-149428	BNIPL	-			
2081	45.62	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
2082	45.58	kd	CGS001-10544	PROCR	CD molecules			
2083	45.58	kd	CGS001-1212	CLTB	-			
2084	45.56	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
2085	45.54	kd	CGS001-5018	OXA1L	-			
2086	45.54	kd	CGS001-27297	CRCP	-			
2087	45.53	kd	CGS001-4846	NOS3	Nitric oxide synthases			
2088	45.5	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
2089	45.49	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
2090	45.48	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
2091	45.47	oe	ccsbBroad304_07349	MAP7	-			
2092	45.46	oe	ccsbBroad304_09225	BUD13	-			
2093	45.44	kd	CGS001-7001	PRDX2	-			
2094	45.42	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
2095	45.42	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
2096	45.42	kd	CGS001-51071	DERA	-			
2097	45.41	kd	CGS001-481	ATP1B1	ATPases / P-type			
2098	45.33	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
2099	45.3	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
2100	45.26	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
2101	45.25	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
2102	45.24	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
2103	45.24	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
2104	45.24	kd	CGS001-1512	CTSH	Cathepsins			
2105	45.16	kd	CGS001-6732	SRPK1	SRPK family			
2106	45.11	oe	ccsbBroad304_02136	COPS2	-			
2107	45.1	cc		IL4 Pathway LOF	-			
2108	45.07	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
2109	45.06	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
2110	45.06	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
2111	45.01	kd	CGS001-1440	CSF3	Endogenous ligands			
2112	45	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
2113	44.99	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
2114	44.99	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
2115	44.97	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
2116	44.94	kd	CGS001-26128	KIAA1279	-			
2117	44.93	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
2118	44.89	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
2119	44.88	oe	ccsbBroad304_08605	PBK	TOPK family			
2120	44.8	kd	CGS001-1026	CDKN1A	-			
2121	44.77	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
2122	44.76	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
2123	44.73	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
2124	44.64	cc		Androgen receptor modulator	-			
2125	44.6	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
2126	44.58	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
2127	44.58	kd	CGS001-29105	C16ORF80	-			
2128	44.57	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
2129	44.46	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2130	44.41	kd	CGS001-661	POLR3D	RNA polymerase subunits			
2131	44.37	kd	CGS001-28511	NKIRAS2	-			
2132	44.34	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
2133	44.32	oe	ccsbBroad304_00101	RHOC	-			
2134	44.27	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
2135	44.22	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
2136	44.22	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
2137	44.14	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
2138	44.12	kd	CGS001-5891	MOK	RCK family			
2139	44.09	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
2140	44.09	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
2141	43.96	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
2142	43.95	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
2143	43.9	oe	ccsbBroad304_06159	CTTN	-			
2144	43.87	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2145	43.83	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
2146	43.83	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
2147	43.81	oe	ccsbBroad304_07053	TFPI	-			
2148	43.8	kd	CGS001-25793	FBXO7	F-boxes / other			
2149	43.78	oe	ccsbBroad304_01257	PPOX	-			
2150	43.78	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
2151	43.78	oe	ccsbBroad304_00964	SMAD7	SMADs			
2152	43.76	kd	CGS001-7157	TP53	-			
2153	43.73	kd	CGS001-7360	UGP2	-			
2154	43.68	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
2155	43.63	oe	ccsbBroad304_02045	BUD31	-			
2156	43.59	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
2157	43.54	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
2158	43.54	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
2159	43.54	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
2160	43.51	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2161	43.5	oe	ccsbBroad304_02446	TADA3	-			
2162	43.48	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
2163	43.47	kd	CGS001-58478	ENOPH1	-			
2164	43.46	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
2165	43.45	kd	CGS001-7298	TYMS	Methyltransferases			
2166	43.39	kd	CGS001-1128	CHRM1	Cholinergic receptors			
2167	43.38	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
2168	43.37	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
2169	43.31	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
2170	43.3	oe	ccsbBroad304_00418	CD55	CD molecules			
2171	43.25	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2172	43.25	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
2173	43.18	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
2174	43.17	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
2175	43.15	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
2176	43.1	oe	ccsbBroad304_08553	STAP2	-			
2177	42.9	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
2178	42.85	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
2179	42.84	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
2180	42.84	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
2181	42.83	kd	CGS001-51015	ISOC1	-			
2182	42.8	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
2183	42.8	kd	CGS001-3251	HPRT1	-			
2184	42.79	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
2185	42.78	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
2186	42.77	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
2187	42.77	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
2188	42.77	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
2189	42.76	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
2190	42.74	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
2191	42.73	kd	CGS001-2524	FUT2	Fucosyltransferases			
2192	42.71	kd	CGS001-55111	PLEKHJ1	Pleckstrin homology (PH) domain containing			
2193	42.7	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
2194	42.69	kd	CGS001-122402	TDRD9	Tudor domain containing			
2195	42.62	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
2196	42.51	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
2197	42.51	kd	CGS001-387	RHOA	-			
2198	42.44	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
2199	42.41	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
2200	42.39	kd	CGS001-818	CAMK2G	CAMK2 family			
2201	42.38	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
2202	42.36	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
2203	42.35	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
2204	42.29	oe	ccsbBroad304_05135	PARP15	-			
2205	42.25	oe	ccsbBroad304_06855	RDX	-			
2206	42.25	kd	CGS001-23588	KLHDC2	-			
2207	42.18	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
2208	42.16	oe	ccsbBroad304_04891	TMEM174	-			
2209	42.16	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
2210	42.13	oe	ccsbBroad304_02834	GABARAPL1	-			
2211	42.09	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
2212	42.09	oe	ccsbBroad304_06996	SRM	-			
2213	42.09	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
2214	42.06	oe	ccsbBroad304_01845	RDBP	-			
2215	42.06	kd	CGS001-1951	CELSR3	Cadherins / Major cadherins			
2216	42.05	cc		Bile acid	-			
2217	41.97	oe	ccsbBroad304_03308	YTHDF2	-			
2218	41.93	oe	ccsbBroad304_00738	HINT1	-			
2219	41.92	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
2220	41.92	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
2221	41.9	kd	CGS001-10969	EBNA1BP2	-			
2222	41.88	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
2223	41.86	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
2224	41.86	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
2225	41.85	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
2226	41.84	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
2227	41.8	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2228	41.78	kd	CGS001-6117	RPA1	-			
2229	41.76	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
2230	41.73	kd	CGS001-11212	PROSC	-			
2231	41.71	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
2232	41.69	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2233	41.69	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
2234	41.66	kd	CGS001-9443	MED7	-			
2235	41.61	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2236	41.56	kd	CGS001-5979	RET	Type XIV RTKs: RET			
2237	41.54	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
2238	41.54	kd	CGS001-6256	RXRA	Retinoid X receptors			
2239	41.5	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
2240	41.48	oe	ccsbBroad304_00614	GAMT	-			
2241	41.47	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
2242	41.41	oe	ccsbBroad304_07097	TRAF1	-			
2243	41.41	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
2244	41.34	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
2245	41.33	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
2246	41.32	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
2247	41.26	oe	ccsbBroad304_02500	RRAGA	-			
2248	41.26	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
2249	41.25	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
2250	41.2	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
2251	41.19	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
2252	41.13	oe	ccsbBroad304_03037	TMEM97	-			
2253	41.13	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
2254	41.04	oe	ccsbBroad304_01148	PCBD1	-			
2255	40.92	kd	CGS001-2067	ERCC1	-			
2256	40.92	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
2257	40.85	oe	ccsbBroad304_02298	DNM1L	-			
2258	40.82	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
2259	40.81	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
2260	40.81	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
2261	40.8	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
2262	40.78	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
2263	40.77	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
2264	40.76	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
2265	40.73	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
2266	40.72	oe	ccsbBroad304_06642	NIT1	-			
2267	40.69	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
2268	40.64	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
2269	40.62	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
2270	40.61	kd	CGS001-2645	GCK	Hexokinases			
2271	40.6	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
2272	40.59	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
2273	40.54	kd	CGS001-7728	ZNF175	Zinc fingers, C2H2-type			
2274	40.53	oe	ccsbBroad304_04202	MED28	-			
2275	40.53	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
2276	40.5	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
2277	40.48	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
2278	40.47	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
2279	40.44	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
2280	40.41	kd	CGS001-5223	PGAM1	-			
2281	40.38	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
2282	40.33	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
2283	40.32	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
2284	40.29	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
2285	40.25	oe	ccsbBroad304_02579	YWHAQ	-			
2286	40.24	kd	CGS001-10013	HDAC6	Histone deacetylases			
2287	40.22	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
2288	40.17	kd	CGS001-2717	GLA	-			
2289	40.15	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
2290	40.13	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
2291	40.11	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
2292	40.11	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
2293	40.04	kd	CGS001-26993	AKAP8L	-			
2294	40.01	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
2295	40	kd	CGS001-9767	PHF16	-			
2296	39.96	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
2297	39.92	kd	CGS001-6223	RPS19	S ribosomal proteins			
2298	39.92	kd	CGS001-5887	RAD23B	-			
2299	39.91	oe	ccsbBroad304_02501	DCTN6	-			
2300	39.84	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
2301	39.83	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
2302	39.8	kd	CGS001-593	BCKDHA	-			
2303	39.77	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
2304	39.77	kd	CGS001-9318	COPS2	-			
2305	39.75	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
2306	39.68	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
2307	39.65	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
2308	39.64	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
2309	39.63	kd	CGS001-79600	TCTN1	Tectonic proteins			
2310	39.62	oe	ccsbBroad304_00995	MECP2	-			
2311	39.61	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
2312	39.6	kd	CGS001-5073	PARN	-			
2313	39.55	cc		ATP synthase inhibitor	-			
2314	39.5	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2315	39.48	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
2316	39.42	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2317	39.42	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
2318	39.42	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
2319	39.41	kd	CGS001-901	CCNG2	-			
2320	39.4	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
2321	39.37	kd	CGS001-10671	DCTN6	-			
2322	39.35	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
2323	39.34	kd	CGS001-83448	PUS7L	-			
2324	39.31	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
2325	39.28	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
2326	39.23	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
2327	39.2	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
2328	39.14	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
2329	39.13	oe	ccsbBroad304_07080	TM7SF2	-			
2330	39.12	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
2331	39.12	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
2332	39.11	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
2333	39.08	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
2334	39.06	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
2335	39.05	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
2336	39.04	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
2337	38.99	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
2338	38.96	cc		JAK inhibitor	-			
2339	38.95	kd	CGS001-1488	CTBP2	-			
2340	38.92	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
2341	38.91	kd	CGS001-29984	RHOD	-			
2342	38.9	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2343	38.87	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
2344	38.87	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
2345	38.85	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
2346	38.84	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
2347	38.78	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
2348	38.78	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
2349	38.76	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
2350	38.71	oe	ccsbBroad304_05887	CFB	Complement system			
2351	38.71	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
2352	38.67	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
2353	38.65	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
2354	38.56	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
2355	38.55	kd	CGS001-6285	S100B	EF-hand domain containing			
2356	38.47	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
2357	38.45	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
2358	38.44	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2359	38.42	kd	CGS001-10645	CAMKK2	Meta subfamily			
2360	38.41	kd	CGS001-55644	OSGEP	-			
2361	38.3	cc		PKC inhibitor	-			
2362	38.3	kd	CGS001-5645	PRSS2	Serine peptidases			
2363	38.3	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
2364	38.28	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
2365	38.25	oe	ccsbBroad304_00390	CTGF	-			
2366	38.22	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
2367	38.21	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
2368	38.19	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
2369	38.17	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
2370	38.16	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
2371	38.1	oe	ccsbBroad304_06683	FURIN	Subtilisin			
2372	38.08	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
2373	38.08	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
2374	38.06	kd	CGS001-4190	MDH1	-			
2375	38.05	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
2376	38.05	kd	CGS001-2932	GSK3B	GSK subfamily			
2377	38.02	kd	CGS001-3034	HAL	-			
2378	38.01	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
2379	38.01	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
2380	37.95	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
2381	37.9	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
2382	37.86	kd	CGS001-8639	AOC3	Oxidoreductases			
2383	37.85	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
2384	37.84	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
2385	37.83	oe	ccsbBroad304_00961	SMAD2	SMADs			
2386	37.81	oe	ccsbBroad304_06670	OGG1	-			
2387	37.81	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
2388	37.8	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
2389	37.75	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
2390	37.75	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
2391	37.74	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2392	37.73	oe	ccsbBroad304_00469	DUT	-			
2393	37.73	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
2394	37.72	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
2395	37.72	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2396	37.69	oe	ccsbBroad304_02884	POT1	-			
2397	37.69	kd	CGS001-9870	KIAA0317	-			
2398	37.68	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2399	37.66	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
2400	37.64	kd	CGS001-1643	DDB2	WD repeat domain containing			
2401	37.63	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
2402	37.56	oe	ccsbBroad304_00392	CTLA4	CD molecules			
2403	37.56	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
2404	37.55	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
2405	37.54	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
2406	37.53	oe	ccsbBroad304_03191	NOSIP	-			
2407	37.49	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
2408	37.47	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
2409	37.45	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
2410	37.4	kd	CGS001-9156	EXO1	-			
2411	37.37	oe	ccsbBroad304_02270	FAM20B	-			
2412	37.36	oe	ccsbBroad304_02438	FAM3C	-			
2413	37.27	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
2414	37.21	cc		Progesterone receptor antagonist	-			
2415	37.21	kd	CGS001-51564	HDAC7	Histone deacetylases			
2416	37.19	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
2417	37.13	kd	CGS001-23047	PDS5B	-			
2418	37.09	kd	CGS001-900	CCNG1	-			
2419	37.04	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
2420	37.04	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
2421	37.03	kd	CGS001-5062	PAK2	PAKA subfamily			
2422	37.01	oe	ccsbBroad304_00268	CD81	CD molecules			
2423	36.98	kd	CGS001-944	TNFSF8	CD molecules			
2424	36.96	oe	ccsbBroad304_02674	STK38	NDR family			
2425	36.96	kd	CGS001-9670	IPO13	Importins			
2426	36.93	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
2427	36.88	oe	ccsbBroad304_04053	DERL1	-			
2428	36.87	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
2429	36.87	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
2430	36.87	kd	CGS001-9500	MAGED1	-			
2431	36.81	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
2432	36.78	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
2433	36.69	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
2434	36.68	kd	CGS001-22978	NT5C2	Adenosine turnover			
2435	36.61	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
2436	36.6	kd	CGS001-6652	SORD	-			
2437	36.59	oe	ccsbBroad304_03112	NENF	-			
2438	36.59	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
2439	36.59	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2440	36.58	kd	CGS001-55893	ZNF395	Zinc fingers, C2H2-type			
2441	36.55	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
2442	36.54	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
2443	36.53	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
2444	36.52	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
2445	36.52	kd	CGS001-7471	WNT1	Endogenous ligands			
2446	36.51	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
2447	36.47	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
2448	36.46	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
2449	36.46	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
2450	36.41	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
2451	36.39	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
2452	36.38	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
2453	36.36	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
2454	36.36	oe	ccsbBroad304_02702	MSRB2	-			
2455	36.35	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
2456	36.32	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
2457	36.32	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
2458	36.31	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
2459	36.29	cc		PPAR receptor agonist	-			
2460	36.29	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
2461	36.26	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
2462	36.22	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
2463	36.22	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
2464	36.18	kd	CGS001-7090	TLE3	WD repeat domain containing			
2465	36.15	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
2466	36.15	oe	ccsbBroad304_00617	GBA	-			
2467	36.03	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
2468	35.98	oe	ccsbBroad304_08292	IP6K2	-			
2469	35.98	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
2470	35.96	oe	ccsbBroad304_04775	NTAN1	-			
2471	35.91	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
2472	35.88	kd	CGS001-4482	MSRA	-			
2473	35.86	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
2474	35.86	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2475	35.83	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
2476	35.8	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
2477	35.73	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
2478	35.73	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
2479	35.73	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
2480	35.7	kd	CGS001-6443	SGCB	-			
2481	35.69	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
2482	35.64	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
2483	35.63	kd	CGS001-25836	NIPBL	-			
2484	35.6	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
2485	35.57	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2486	35.56	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2487	35.56	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
2488	35.56	kd	CGS001-116443	GRIN3A	Glutamate receptors			
2489	35.55	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
2490	35.48	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
2491	35.47	kd	CGS001-51441	YTHDF2	-			
2492	35.46	kd	CGS001-2309	FOXO3	Forkhead boxes			
2493	35.45	oe	ccsbBroad304_07287	HYAL2	-			
2494	35.42	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
2495	35.41	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
2496	35.41	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
2497	35.39	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
2498	35.39	kd	CGS001-8431	NR0B2	DAX-like receptors			
2499	35.37	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
2500	35.32	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
2501	35.32	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
2502	35.24	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2503	35.21	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
2504	35.21	kd	CGS001-670	BPHL	-			
2505	35.21	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
2506	35.14	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
2507	35.12	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
2508	35.11	kd	CGS001-22908	SACM1L	-			
2509	35.06	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
2510	35.03	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
2511	34.98	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
2512	34.95	oe	ccsbBroad304_01560	SNAPC1	-			
2513	34.93	oe	ccsbBroad304_02497	YKT6	-			
2514	34.93	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
2515	34.91	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
2516	34.88	oe	ccsbBroad304_00552	FEN1	-			
2517	34.87	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
2518	34.83	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
2519	34.83	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
2520	34.83	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
2521	34.82	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
2522	34.82	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
2523	34.81	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
2524	34.77	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
2525	34.77	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
2526	34.75	kd	CGS001-8802	SUCLG1	-			
2527	34.74	kd	CGS001-382	ARF6	ADP-ribosylation factors			
2528	34.71	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
2529	34.71	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
2530	34.66	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
2531	34.63	oe	ccsbBroad304_10437	STMN1	-			
2532	34.57	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
2533	34.56	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
2534	34.46	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
2535	34.46	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
2536	34.44	kd	CGS001-57157	PHTF2	-			
2537	34.43	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
2538	34.42	oe	ccsbBroad304_00986	MCM2	-			
2539	34.39	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
2540	34.38	kd	CGS001-51593	SRRT	-			
2541	34.36	kd	CGS001-3630	INS	-			
2542	34.34	kd	CGS001-6461	SHB	SH2 domain containing			
2543	34.34	kd	CGS001-2114	ETS2	ETS Transcription Factors			
2544	34.27	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
2545	34.25	kd	CGS001-115	ADCY9	Adenylyl cyclases			
2546	34.19	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2547	34.15	kd	CGS001-823	CAPN1	EF-hand domain containing			
2548	34.12	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
2549	34.12	kd	CGS001-801	CALM1	EF-hand domain containing			
2550	34.08	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
2551	34.08	kd	CGS001-4303	FOXO4	Forkhead boxes			
2552	34.07	kd	CGS001-51466	EVL	-			
2553	34.01	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
2554	33.98	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
2555	33.98	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
2556	33.95	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
2557	33.94	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
2558	33.93	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
2559	33.83	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2560	33.82	oe	ccsbBroad304_00881	IRF5	-			
2561	33.82	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
2562	33.81	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
2563	33.72	oe	ccsbBroad304_03934	LEPRE1	-			
2564	33.72	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
2565	33.71	oe	ccsbBroad304_02367	CALCOCO2	-			
2566	33.62	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
2567	33.62	kd	CGS001-2004	ELK3	ETS Transcription Factors			
2568	33.62	kd	CGS001-27034	ACAD8	-			
2569	33.58	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
2570	33.56	oe	ccsbBroad304_10230	STK19	G11 family			
2571	33.56	oe	ccsbBroad304_01624	SUPV3L1	-			
2572	33.55	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
2573	33.55	oe	ccsbBroad304_03641	ASF1B	-			
2574	33.46	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
2575	33.46	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
2576	33.46	kd	CGS001-11182	SLC2A6	Solute carriers			
2577	33.4	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
2578	33.36	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
2579	33.34	oe	ccsbBroad304_00099	ARG2	Arginase			
2580	33.28	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
2581	33.27	cc		Wnt family LOF	-			
2582	33.25	kd	CGS001-2588	GALNS	Arylsulfatase family			
2583	33.24	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
2584	33.23	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
2585	33.17	kd	CGS001-10613	ERLIN1	-			
2586	33.08	oe	ccsbBroad304_00053	ALDOA	-			
2587	33.03	oe	ccsbBroad304_06420	ICAM3	CD molecules			
2588	32.97	kd	CGS001-2877	GPX2	-			
2589	32.96	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
2590	32.93	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2591	32.92	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
2592	32.82	kd	CGS001-10247	HRSP12	-			
2593	32.78	oe	ccsbBroad304_00747	HLF	-			
2594	32.73	oe	ccsbBroad304_07012	STK3	MST subfamily			
2595	32.67	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
2596	32.64	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
2597	32.64	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
2598	32.63	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
2599	32.59	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
2600	32.58	oe	ccsbBroad304_07401	TXNL1	-			
2601	32.58	oe	ccsbBroad304_06828	PYCR1	-			
2602	32.58	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
2603	32.57	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
2604	32.57	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2605	32.56	kd	CGS001-10105	PPIF	-			
2606	32.53	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
2607	32.47	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
2608	32.46	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
2609	32.45	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
2610	32.37	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
2611	32.33	kd	CGS001-5664	PSEN2	Presenilin			
2612	32.31	kd	CGS001-835	CASP2	Caspases			
2613	32.3	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2614	32.27	kd	CGS001-54499	TMCO1	-			
2615	32.25	kd	CGS001-23344	ESYT1	Synaptotagmins			
2616	32.22	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
2617	32.19	oe	ccsbBroad304_07102	TSG101	-			
2618	32.19	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
2619	32.18	kd	CGS001-2534	FYN	Src family			
2620	32.12	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
2621	32.09	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
2622	32	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
2623	32	kd	CGS001-2931	GSK3A	GSK subfamily			
2624	31.93	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
2625	31.9	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
2626	31.86	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
2627	31.83	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
2628	31.81	kd	CGS001-10390	CEPT1	-			
2629	31.76	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
2630	31.64	kd	CGS001-29946	SERTAD3	-			
2631	31.59	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
2632	31.58	oe	ccsbBroad304_07754	FGFR1OP	-			
2633	31.57	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
2634	31.54	oe	ccsbBroad304_05821	ANXA1	Annexins			
2635	31.53	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
2636	31.5	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
2637	31.47	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
2638	31.42	kd	CGS001-1869	E2F1	-			
2639	31.4	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
2640	31.39	oe	ccsbBroad304_00620	GCDH	-			
2641	31.34	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
2642	31.33	oe	ccsbBroad304_06350	HAL	-			
2643	31.33	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
2644	31.2	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
2645	31.2	kd	CGS001-3066	HDAC2	Histone deacetylases			
2646	31.19	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
2647	31.18	oe	ccsbBroad304_04194	ELL3	-			
2648	31.18	kd	CGS001-79094	CHAC1	-			
2649	31.14	oe	ccsbBroad304_00210	CALR	-			
2650	31.14	kd	CGS001-8525	DGKZ	-			
2651	31.12	oe	ccsbBroad304_02175	MAGED1	-			
2652	31.1	oe	ccsbBroad304_00225	CAT	-			
2653	31.08	kd	CGS001-10400	PEMT	-			
2654	31.05	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
2655	31.01	oe	ccsbBroad304_00966	MAFG	-			
2656	30.98	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
2657	30.94	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
2658	30.9	kd	CGS001-55620	STAP2	-			
2659	30.87	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
2660	30.87	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
2661	30.8	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
2662	30.73	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
2663	30.73	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
2664	30.71	kd	CGS001-9788	MTSS1	-			
2665	30.69	oe	ccsbBroad304_02506	EBP	-			
2666	30.69	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
2667	30.66	oe	ccsbBroad304_01152	PCNA	-			
2668	30.65	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
2669	30.63	oe	ccsbBroad304_02092	SYNGR3	-			
2670	30.63	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
2671	30.63	kd	CGS001-5588	PRKCQ	Delta subfamily			
2672	30.58	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
2673	30.56	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2674	30.55	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
2675	30.51	kd	CGS001-644	BLVRA	-			
2676	30.49	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
2677	30.48	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
2678	30.45	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
2679	30.42	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
2680	30.42	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
2681	30.41	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2682	30.37	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
2683	30.37	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
2684	30.36	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
2685	30.32	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
2686	30.28	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
2687	30.28	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
2688	30.17	kd	CGS001-29883	CNOT7	-			
2689	30.04	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2690	30.04	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
2691	30	kd	CGS001-5933	RBL1	-			
2692	29.98	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
2693	29.93	kd	CGS001-4048	LTA4H	Hydrolases			
2694	29.92	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
2695	29.89	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
2696	29.89	kd	CGS001-2017	CTTN	-			
2697	29.88	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
2698	29.86	oe	ccsbBroad304_07320	SQSTM1	-			
2699	29.85	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
2700	29.83	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2701	29.83	kd	CGS001-7852	CXCR4	Chemokine receptors			
2702	29.75	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
2703	29.71	kd	CGS001-10412	NSA2	-			
2704	29.66	oe	ccsbBroad304_09095	PUS7L	-			
2705	29.61	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
2706	29.57	kd	CGS001-4864	NPC1	-			
2707	29.53	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2708	29.5	kd	CGS001-388	RHOB	-			
2709	29.44	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
2710	29.36	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
2711	29.35	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
2712	29.35	oe	ccsbBroad304_00162	BIK	-			
2713	29.29	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
2714	29.29	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
2715	29.24	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
2716	29.23	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
2717	29.23	kd	CGS001-353	APRT	-			
2718	29.21	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
2719	29.2	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
2720	29.16	kd	CGS001-4172	MCM3	-			
2721	29.11	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
2722	29.08	kd	CGS001-4507	MTAP	-			
2723	29.04	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
2724	29.03	oe	ccsbBroad304_06535	LPL	-			
2725	29.02	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
2726	28.94	kd	CGS001-3456	IFNB1	Interferons			
2727	28.93	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
2728	28.92	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
2729	28.9	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
2730	28.85	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
2731	28.81	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
2732	28.75	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
2733	28.74	oe	ccsbBroad304_00212	CAMLG	-			
2734	28.74	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
2735	28.73	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
2736	28.73	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
2737	28.72	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
2738	28.71	kd	CGS001-11116	FGFR1OP	-			
2739	28.66	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
2740	28.66	kd	CGS001-94234	FOXQ1	Forkhead boxes			
2741	28.58	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
2742	28.54	kd	CGS001-5004	ORM1	Lipocalins			
2743	28.51	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
2744	28.49	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
2745	28.45	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
2746	28.39	kd	CGS001-8089	YEATS4	-			
2747	28.38	oe	ccsbBroad304_07923	LSM5	-			
2748	28.33	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
2749	28.29	oe	ccsbBroad304_03119	C16ORF5	-			
2750	28.29	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
2751	28.29	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
2752	28.28	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
2753	28.26	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
2754	28.22	kd	CGS001-58528	RRAGD	-			
2755	28.21	kd	CGS001-116931	MED12L	-			
2756	28.18	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2757	28.14	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
2758	28.12	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
2759	28.11	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
2760	28.11	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
2761	27.89	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
2762	27.85	kd	CGS001-8634	RTCD1	-			
2763	27.83	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
2764	27.82	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
2765	27.82	kd	CGS001-25913	POT1	-			
2766	27.71	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
2767	27.68	kd	CGS001-22794	CASC3	-			
2768	27.67	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
2769	27.64	oe	ccsbBroad304_08325	LIPT1	-			
2770	27.64	oe	ccsbBroad304_06765	PRCC	-			
2771	27.63	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
2772	27.62	kd	CGS001-1950	EGF	-			
2773	27.49	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
2774	27.39	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
2775	27.38	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
2776	27.34	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
2777	27.31	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
2778	27.28	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
2779	27.2	kd	CGS001-1312	COMT	Catecholamine turnover			
2780	27.14	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
2781	27.12	oe	ccsbBroad304_07267	PDLIM4	-			
2782	27.11	kd	CGS001-89766	UMODL1	-			
2783	27.09	kd	CGS001-861	RUNX1	-			
2784	27.08	kd	CGS001-55968	NSFL1C	UBX domain containing			
2785	26.94	kd	CGS001-64135	IFIH1	-			
2786	26.92	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
2787	26.91	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
2788	26.89	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
2789	26.86	kd	CGS001-9807	IP6K1	-			
2790	26.83	kd	CGS001-57819	LSM2	-			
2791	26.72	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
2792	26.71	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
2793	26.7	kd	CGS001-23492	CBX7	-			
2794	26.69	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
2795	26.66	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
2796	26.64	oe	ccsbBroad304_03311	EVL	-			
2797	26.6	kd	CGS001-11136	SLC7A9	SLC7 family			
2798	26.41	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
2799	26.37	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
2800	26.35	oe	ccsbBroad304_06837	RAF1	RAF family			
2801	26.34	kd	CGS001-3939	LDHA	-			
2802	26.23	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2803	26.14	kd	CGS001-5934	RBL2	-			
2804	26.04	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
2805	25.98	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
2806	25.95	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2807	25.93	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
2808	25.88	oe	ccsbBroad304_13880	IDH3G	-			
2809	25.85	kd	CGS001-117154	DACH2	-			
2810	25.84	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
2811	25.78	kd	CGS001-116519	APOA5	Apolipoproteins			
2812	25.7	kd	CGS001-4837	NNMT	-			
2813	25.7	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
2814	25.62	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
2815	25.5	kd	CGS001-7020	TFAP2A	-			
2816	25.49	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
2817	25.39	kd	CGS001-23192	ATG4B	Aut2 peptidase			
2818	25.38	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2819	25.32	oe	ccsbBroad304_06462	ITGAE	Integrins			
2820	25.3	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
2821	25.29	oe	ccsbBroad304_01485	SC5DL	-			
2822	25.2	oe	ccsbBroad304_06180	ESD	-			
2823	25.2	kd	CGS001-8837	CFLAR	Endogenous ligands			
2824	25.19	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
2825	25.16	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
2826	25.1	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
2827	25.1	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
2828	25.02	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
2829	25	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
2830	24.97	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
2831	24.92	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
2832	24.77	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
2833	24.71	oe	ccsbBroad304_03618	OSGEP	-			
2834	24.62	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
2835	24.58	cc		ATPase inhibitor	-			
2836	24.56	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
2837	24.55	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
2838	24.47	kd	CGS001-5167	ENPP1	-			
2839	24.45	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
2840	24.44	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
2841	24.44	kd	CGS001-5338	PLD2	Hydrolases			
2842	24.34	kd	CGS001-662	BNIP1	-			
2843	24.33	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
2844	24.28	kd	CGS001-7078	TIMP3	-			
2845	24.23	cc		DNA synthesis inhibitor	-			
2846	24.11	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
2847	24.1	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
2848	24.07	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
2849	24.05	kd	CGS001-4067	LYN	Src family			
2850	23.92	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
2851	23.85	oe	ccsbBroad304_05907	BUB1B	Bub family			
2852	23.85	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
2853	23.8	kd	CGS001-7185	TRAF1	-			
2854	23.79	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
2855	23.77	kd	CGS001-2099	ESR1	Estrogen receptors			
2856	23.73	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
2857	23.66	kd	CGS001-4860	PNP	-			
2858	23.65	oe	ccsbBroad304_06976	SMARCE1	-			
2859	23.61	kd	CGS001-54407	SLC38A2	System A-like transporters			
2860	23.57	kd	CGS001-23509	POFUT1	Fucosyltransferases			
2861	23.52	kd	CGS001-7477	WNT7B	Endogenous ligands			
2862	23.41	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
2863	23.32	kd	CGS001-10214	SSX3	-			
2864	23.31	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
2865	23.3	kd	CGS001-8192	CLPP	ATPases / AAA-type			
2866	23.2	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
2867	23.11	oe	ccsbBroad304_02086	PDLIM1	-			
2868	22.99	kd	CGS001-9612	NCOR2	-			
2869	22.9	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
2870	22.89	oe	ccsbBroad304_04649	ADC	-			
2871	22.84	kd	CGS001-1736	DKC1	-			
2872	22.8	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
2873	22.77	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
2874	22.76	oe	ccsbBroad304_05745	CD24	CD molecules			
2875	22.68	kd	CGS001-271	AMPD2	-			
2876	22.64	oe	ccsbBroad304_02133	CD83	CD molecules			
2877	22.63	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
2878	22.61	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
2879	22.54	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
2880	22.48	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
2881	22.45	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
2882	22.39	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
2883	22.3	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
2884	22.24	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
2885	22.16	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
2886	22.13	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
2887	22.13	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
2888	22.08	kd	CGS001-513	ATP5D	ATPases / F-type			
2889	21.7	kd	CGS001-7013	TERF1	-			
2890	21.69	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
2891	21.62	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
2892	21.62	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
2893	21.54	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
2894	21.52	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2895	21.32	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
2896	21.31	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
2897	21.29	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
2898	21.2	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
2899	21.19	kd	CGS001-10078	TSSC4	-			
2900	21.15	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
2901	21.12	oe	ccsbBroad304_03444	PAF1	-			
2902	21.12	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
2903	21.06	kd	CGS001-3608	ILF2	-			
2904	21.02	kd	CGS001-144811	LACC1	-			
2905	20.97	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
2906	20.94	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
2907	20.73	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
2908	20.57	kd	CGS001-1981	EIF4G1	Parkinson disease			
2909	20.52	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
2910	20.34	kd	CGS001-8826	IQGAP1	-			
2911	20.31	kd	CGS001-388677	NOTCH2NL	-			
2912	20.3	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
2913	20.23	kd	CGS001-10914	PAPOLA	-			
2914	20	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
2915	19.93	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
2916	19.79	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
2917	19.63	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2918	19.55	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
2919	19.52	kd	CGS001-2203	FBP1	-			
2920	19.45	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
2921	19.38	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
2922	19.37	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
2923	19.2	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
2924	19.09	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
2925	19.05	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
2926	19.02	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
2927	18.94	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2928	18.72	cc		Phospholipases LOF	-			
2929	18.69	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
2930	18.63	oe	ccsbBroad304_04292	INHBE	-			
2931	18.63	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
2932	18.6	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
2933	18.58	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
2934	18.56	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
2935	18.25	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
2936	18.08	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
2937	18.04	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
2938	18.04	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
2939	17.95	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
2940	17.89	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
2941	17.78	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
2942	17.75	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
2943	17.67	oe	ccsbBroad304_00626	GDI1	-			
2944	17.41	kd	CGS001-966	CD59	CD molecules			
2945	17.29	oe	ccsbBroad304_04534	HN1L	-			
2946	17.18	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
2947	17.1	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
2948	16.83	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
2949	16.78	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
2950	16.75	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
2951	16.65	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2952	16.49	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
2953	16.42	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
2954	16.4	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
2955	16.24	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
2956	16.13	oe	ccsbBroad304_01483	SAT1	-			
2957	15.66	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2958	15.55	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
2959	15.49	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
2960	15.46	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
2961	15.32	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
2962	14.52	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
2963	14.39	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
2964	14.33	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
2965	14.28	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
2966	14.1	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
2967	14.09	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
2968	13.45	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2969	13.31	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
2970	12.77	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
2971	12.76	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
2972	12.73	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
2973	12.55	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
2974	11.75	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
2975	11.38	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
2976	11.26	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
2977	11.25	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
2978	11.07	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
2979	10.69	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
2980	10.1	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
2981	9.59	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
2982	9.34	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
2983	9.14	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2984	8.67	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
2985	8.17	cc		Mediator complex LOF	-			
2986	7.67	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
2987	6.37	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
2988	6.14	cc		Mitogen activated protein kinases LOF	-			
2989	-4.79	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
2990	-6.59	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
2991	-7.85	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
2992	-8.17	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
2993	-8.87	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
2994	-9.17	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2995	-10.13	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
2996	-10.89	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
2997	-11.35	cc		RNA Polymerase Enzymes LOF	-			
2998	-11.65	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
2999	-11.66	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
3000	-11.67	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
3001	-11.86	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
3002	-11.87	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
3003	-12.27	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
3004	-12.43	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
3005	-12.49	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
3006	-12.72	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
3007	-12.87	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
3008	-13.03	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
3009	-13.25	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
3010	-13.71	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
3011	-14.01	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
3012	-14.18	kd	CGS001-65243	ZNF643	-			
3013	-14.4	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
3014	-14.4	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
3015	-14.57	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
3016	-14.78	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3017	-14.84	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
3018	-14.85	kd	CGS001-2288	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
3019	-14.88	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
3020	-14.91	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
3021	-15.37	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
3022	-15.52	kd	CGS001-9541	CIR1	-			
3023	-15.58	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
3024	-15.71	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
3025	-15.99	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
3026	-16.13	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3027	-16.5	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
3028	-16.57	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
3029	-16.73	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
3030	-16.73	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
3031	-16.76	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3032	-16.78	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
3033	-16.78	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
3034	-16.91	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
3035	-16.97	kd	CGS001-7965	AIMP2	-			
3036	-17.02	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
3037	-17.02	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3038	-17.05	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
3039	-17.14	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
3040	-17.16	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
3041	-17.16	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3042	-17.2	cc		HOXL subclass homeoboxes LOF	-			
3043	-17.48	cc		Tricyclic antidepressant	-			
3044	-17.5	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
3045	-17.6	cc		GPCR Subset GOF	-			
3046	-17.64	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
3047	-17.77	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
3048	-18.07	kd	CGS001-11344	TWF2	Twinfilin subfamily			
3049	-18.2	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
3050	-18.33	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
3051	-18.77	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3052	-18.83	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
3053	-18.98	kd	CGS001-7016	TESK1	TESK subfamily			
3054	-19.01	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
3055	-19.1	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
3056	-19.15	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3057	-19.21	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
3058	-19.24	kd	CGS001-472	ATM	Other PIKK family kinases			
3059	-19.36	kd	CGS001-6776	STAT5A	SH2 domain containing			
3060	-19.46	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
3061	-19.48	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
3062	-19.53	kd	CGS001-1997	ELF1	ETS Transcription Factors			
3063	-19.63	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
3064	-19.72	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
3065	-19.86	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3066	-19.87	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
3067	-19.91	kd	CGS001-4758	NEU1	-			
3068	-19.92	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
3069	-19.96	kd	CGS001-2919	CXCL1	Endogenous ligands			
3070	-20.06	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
3071	-20.1	oe	ccsbBroad304_00975	MAT2A	-			
3072	-20.13	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
3073	-20.26	kd	CGS001-283150	FOXR1	Forkhead boxes			
3074	-20.28	kd	CGS001-84890	ADO	-			
3075	-20.29	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
3076	-20.34	kd	CGS001-1036	CDO1	-			
3077	-20.37	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
3078	-20.41	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
3079	-20.43	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
3080	-20.45	kd	CGS001-65123	INTS3	-			
3081	-20.49	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
3082	-20.53	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
3083	-20.69	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
3084	-20.7	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
3085	-20.74	oe	ccsbBroad304_09833	SENP5	-			
3086	-20.79	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
3087	-20.84	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
3088	-20.89	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
3089	-20.94	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
3090	-20.98	kd	CGS001-7088	TLE1	WD repeat domain containing			
3091	-21.17	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
3092	-21.18	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
3093	-21.25	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
3094	-21.26	oe	ccsbBroad304_07490	SCRN1	-			
3095	-21.26	kd	CGS001-4069	LYZ	-			
3096	-21.34	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
3097	-21.35	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
3098	-21.36	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3099	-21.36	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
3100	-21.4	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
3101	-21.45	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
3102	-21.46	kd	CGS001-399694	SHC4	SH2 domain containing			
3103	-21.51	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
3104	-21.62	kd	CGS001-23647	ARFIP2	-			
3105	-21.67	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
3106	-21.68	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
3107	-21.79	kd	CGS001-23196	FAM120A	-			
3108	-21.8	kd	CGS001-3242	HPD	Oxidoreductases			
3109	-21.81	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
3110	-21.84	kd	CGS001-4245	MGAT1	-			
3111	-22.01	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
3112	-22.05	oe	ccsbBroad304_06234	G6PC	-			
3113	-22.06	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
3114	-22.08	kd	CGS001-84923	FAM104A	-			
3115	-22.09	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
3116	-22.11	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
3117	-22.24	oe	ccsbBroad304_01527	SGK1	SGK family			
3118	-22.27	kd	CGS001-55191	NADSYN1	-			
3119	-22.32	oe	ccsbBroad304_02416	TUBB4B	-			
3120	-22.35	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
3121	-22.38	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3122	-22.39	kd	CGS001-9131	AIFM1	-			
3123	-22.42	oe	ccsbBroad304_02318	KIF20A	Kinesins			
3124	-22.42	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
3125	-22.44	kd	CGS001-5663	PSEN1	Presenilin			
3126	-22.48	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
3127	-22.62	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
3128	-22.65	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
3129	-22.65	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
3130	-22.71	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
3131	-22.73	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
3132	-22.74	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
3133	-22.75	oe	ccsbBroad304_06367	HK1	-			
3134	-22.76	oe	ccsbBroad304_02345	TXNDC9	-			
3135	-22.78	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
3136	-22.79	kd	CGS001-5894	RAF1	RAF family			
3137	-22.8	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
3138	-22.82	kd	CGS001-8313	AXIN2	-			
3139	-22.83	kd	CGS001-4637	MYL6	EF-hand domain containing			
3140	-22.91	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
3141	-22.92	cc		G2 M Checkpoint LOF	-			
3142	-22.92	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
3143	-22.92	kd	CGS001-100	ADA	Adenosine turnover			
3144	-22.95	cc		PKC activator	-			
3145	-23.11	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
3146	-23.13	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
3147	-23.15	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
3148	-23.17	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
3149	-23.22	oe	ccsbBroad304_01605	SSX2	-			
3150	-23.26	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
3151	-23.27	kd	CGS001-10923	SUB1	-			
3152	-23.32	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
3153	-23.32	kd	CGS001-7018	TF	-			
3154	-23.33	kd	CGS001-10312	TCIRG1	ATPases / V-type			
3155	-23.39	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
3156	-23.41	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
3157	-23.41	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
3158	-23.46	kd	CGS001-8743	TNFSF10	CD molecules			
3159	-23.47	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
3160	-23.52	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
3161	-23.53	cc		Reverse transcriptase inhibitor	-			
3162	-23.61	oe	ccsbBroad304_00949	LRPAP1	-			
3163	-23.72	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3164	-23.74	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
3165	-23.74	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
3166	-23.74	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
3167	-23.8	oe	ccsbBroad304_07045	TEAD4	-			
3168	-23.83	kd	CGS001-1514	CTSL1	-			
3169	-23.85	oe	ccsbBroad304_02509	GMEB1	-			
3170	-23.87	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
3171	-23.96	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
3172	-23.97	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
3173	-24	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
3174	-24.01	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3175	-24.02	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
3176	-24.09	oe	ccsbBroad304_00865	ILF2	-			
3177	-24.14	kd	CGS001-5562	PRKAA1	AMPK subfamily			
3178	-24.18	kd	CGS001-317705	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
3179	-24.19	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
3180	-24.23	kd	CGS001-6446	SGK1	SGK family			
3181	-24.27	kd	CGS001-50808	AK3	-			
3182	-24.28	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
3183	-24.31	kd	CGS001-25824	PRDX5	-			
3184	-24.34	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
3185	-24.4	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
3186	-24.41	kd	CGS001-4697	NDUFA4	-			
3187	-24.48	kd	CGS001-4287	ATXN3	Ataxins			
3188	-24.49	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
3189	-24.52	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
3190	-24.53	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
3191	-24.54	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
3192	-24.64	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
3193	-24.66	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
3194	-24.71	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
3195	-24.72	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
3196	-24.75	oe	ccsbBroad304_07024	SYK	Syk family			
3197	-24.75	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
3198	-24.78	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
3199	-24.78	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
3200	-24.8	kd	CGS001-5355	PLP2	-			
3201	-24.81	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
3202	-24.81	kd	CGS001-1499	CTNNB1	Catenins			
3203	-24.83	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
3204	-24.88	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
3205	-24.92	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
3206	-24.93	oe	ccsbBroad304_06648	CNOT3	-			
3207	-24.96	kd	CGS001-80314	EPC1	-			
3208	-24.97	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
3209	-24.98	kd	CGS001-5170	PDPK1	PDK1 family			
3210	-24.99	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
3211	-25.01	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
3212	-25.01	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3213	-25.06	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
3214	-25.06	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
3215	-25.07	kd	CGS001-22889	KIAA0907	-			
3216	-25.11	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
3217	-25.19	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
3218	-25.23	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
3219	-25.24	kd	CGS001-91304	C19ORF6	-			
3220	-25.27	kd	CGS001-1763	DNA2	-			
3221	-25.32	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
3222	-25.32	oe	ccsbBroad304_00991	MDH1	-			
3223	-25.33	oe	ccsbBroad304_00054	ALDOC	-			
3224	-25.34	kd	CGS001-1737	DLAT	-			
3225	-25.36	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
3226	-25.39	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
3227	-25.43	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3228	-25.43	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3229	-25.45	kd	CGS001-822	CAPG	-			
3230	-25.46	oe	ccsbBroad304_06820	PTS	-			
3231	-25.46	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
3232	-25.48	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
3233	-25.52	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
3234	-25.59	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
3235	-25.65	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
3236	-25.73	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
3237	-25.74	kd	CGS001-3821	KLRC1	CD molecules			
3238	-25.81	oe	ccsbBroad304_06174	ERCC1	-			
3239	-25.81	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
3240	-25.84	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
3241	-25.86	kd	CGS001-10001	MED6	-			
3242	-25.88	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
3243	-25.88	kd	CGS001-83729	INHBE	-			
3244	-25.89	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
3245	-25.9	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
3246	-25.95	cc		Estrogen receptor antagonist	-			
3247	-25.97	kd	CGS001-10468	FST	-			
3248	-25.99	kd	CGS001-3988	LIPA	-			
3249	-26.01	oe	ccsbBroad304_03767	TOMM22	-			
3250	-26.08	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
3251	-26.09	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
3252	-26.09	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
3253	-26.09	kd	CGS001-545	ATR	ATR subfamily			
3254	-26.1	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
3255	-26.12	kd	CGS001-11044	PAPD7	-			
3256	-26.14	oe	ccsbBroad304_00472	EBF1	-			
3257	-26.17	oe	ccsbBroad304_07887	GCAT	-			
3258	-26.17	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
3259	-26.18	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
3260	-26.19	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
3261	-26.21	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
3262	-26.22	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
3263	-26.22	kd	CGS001-8800	PEX11A	-			
3264	-26.23	oe	ccsbBroad304_00070	ANXA5	Annexins			
3265	-26.3	kd	CGS001-9275	BCL7B	-			
3266	-26.38	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
3267	-26.41	kd	CGS001-11200	CHEK2	CHK1 subfamily			
3268	-26.45	kd	CGS001-11164	NUDT5	Nudix motif containing			
3269	-26.48	cc		DNA Replication LOF	-			
3270	-26.48	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
3271	-26.56	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
3272	-26.57	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
3273	-26.63	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
3274	-26.63	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
3275	-26.71	oe	ccsbBroad304_01001	MEST	-			
3276	-26.72	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
3277	-26.73	oe	ccsbBroad304_03858	SRPRB	-			
3278	-26.75	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
3279	-26.75	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
3280	-26.77	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
3281	-26.8	kd	CGS001-10111	RAD50	-			
3282	-26.92	kd	CGS001-64786	TBC1D15	-			
3283	-26.93	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
3284	-27.01	oe	ccsbBroad304_07843	FCHO1	-			
3285	-27.01	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
3286	-27.04	kd	CGS001-55379	LRRC59	-			
3287	-27.08	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
3288	-27.09	kd	CGS001-2000	ELF4	ETS Transcription Factors			
3289	-27.2	kd	CGS001-10494	STK25	YSK subfamily			
3290	-27.2	oe	ccsbBroad304_05981	CDO1	-			
3291	-27.24	oe	ccsbBroad304_00941	LIG3	-			
3292	-27.25	kd	CGS001-6196	RPS6KA2	RSK subfamily			
3293	-27.3	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
3294	-27.37	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
3295	-27.41	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
3296	-27.48	kd	CGS001-2783	GNB2	WD repeat domain containing			
3297	-27.52	cc		Zinc fingers RanBP2 type LOF	-			
3298	-27.56	kd	CGS001-7040	TGFB1	Endogenous ligands			
3299	-27.58	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
3300	-27.62	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
3301	-27.63	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
3302	-27.66	kd	CGS001-23075	SWAP70	EF-hand domain containing			
3303	-27.68	kd	CGS001-6774	STAT3	SH2 domain containing			
3304	-27.71	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
3305	-27.71	kd	CGS001-10046	MAMLD1	-			
3306	-27.76	kd	CGS001-8669	EIF3J	-			
3307	-27.8	kd	CGS001-10657	KHDRBS1	-			
3308	-27.83	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
3309	-27.84	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
3310	-27.85	kd	CGS001-5427	POLE2	DNA polymerases			
3311	-27.94	kd	CGS001-51720	UIMC1	-			
3312	-27.96	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
3313	-27.96	kd	CGS001-5194	PEX13	-			
3314	-27.97	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
3315	-27.98	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
3316	-27.98	kd	CGS001-8833	GMPS	-			
3317	-28.03	oe	ccsbBroad304_01052	MYB	-			
3318	-28.04	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
3319	-28.04	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
3320	-28.05	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
3321	-28.07	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
3322	-28.08	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
3323	-28.1	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
3324	-28.1	kd	CGS001-4664	NAB1	-			
3325	-28.12	oe	ccsbBroad304_06134	ECH1	-			
3326	-28.13	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
3327	-28.14	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
3328	-28.19	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
3329	-28.19	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
3330	-28.24	kd	CGS001-23030	KDM4B	Histone demethylases			
3331	-28.25	kd	CGS001-2885	GRB2	SH2 domain containing			
3332	-28.26	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
3333	-28.27	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
3334	-28.28	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
3335	-28.28	kd	CGS001-3476	IGBP1	-			
3336	-28.3	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
3337	-28.31	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
3338	-28.33	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
3339	-28.34	oe	ccsbBroad304_00725	HADHA	-			
3340	-28.35	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
3341	-28.38	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
3342	-28.39	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
3343	-28.41	oe	ccsbBroad304_01675	TK1	-			
3344	-28.41	kd	CGS001-283	ANG	Ribonucleases, RNase A			
3345	-28.44	kd	CGS001-1647	GADD45A	-			
3346	-28.45	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
3347	-28.46	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
3348	-28.48	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
3349	-28.48	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
3350	-28.48	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
3351	-28.5	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
3352	-28.5	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
3353	-28.56	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
3354	-28.57	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
3355	-28.6	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
3356	-28.61	oe	ccsbBroad304_07827	STK38L	NDR family			
3357	-28.61	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
3358	-28.61	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
3359	-28.65	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
3360	-28.72	kd	CGS001-2161	F12	Chymotrypsin			
3361	-28.73	kd	CGS001-345611	IRGM	-			
3362	-28.74	kd	CGS001-1111	CHEK1	CHK1 subfamily			
3363	-28.79	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
3364	-28.79	kd	CGS001-4125	MAN2B1	-			
3365	-28.81	cc		Purinergic receptors P2Y GOF	-			
3366	-28.81	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
3367	-28.82	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
3368	-28.85	cc		Akt Signaling LOF	-			
3369	-28.87	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
3370	-28.88	kd	CGS001-4931	NVL	ATPases / AAA-type			
3371	-28.91	oe	ccsbBroad304_03235	TUBD1	Tubulins			
3372	-28.92	kd	CGS001-375133	PI4KAP2	-			
3373	-28.94	kd	CGS001-9759	HDAC4	Histone deacetylases			
3374	-28.98	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
3375	-28.99	oe	ccsbBroad304_00447	DLD	-			
3376	-28.99	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
3377	-29.05	kd	CGS001-7504	XK	Blood group antigens			
3378	-29.05	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
3379	-29.09	oe	ccsbBroad304_04655	TRIM9	-			
3380	-29.09	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
3381	-29.09	kd	CGS001-7270	TTF1	-			
3382	-29.12	kd	CGS001-29102	DROSHA	-			
3383	-29.18	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
3384	-29.2	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
3385	-29.21	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
3386	-29.26	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
3387	-29.29	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
3388	-29.29	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
3389	-29.3	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
3390	-29.34	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
3391	-29.36	oe	ccsbBroad304_02738	RRS1	-			
3392	-29.36	oe	ccsbBroad304_02596	KDELR3	-			
3393	-29.38	kd	CGS001-63892	THADA	-			
3394	-29.39	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
3395	-29.41	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
3396	-29.45	kd	CGS001-6829	SUPT5H	-			
3397	-29.47	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
3398	-29.49	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
3399	-29.56	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
3400	-29.57	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
3401	-29.6	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
3402	-29.65	kd	CGS001-2782	GNB1	WD repeat domain containing			
3403	-29.67	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
3404	-29.67	kd	CGS001-57149	LYRM1	LYR motif containing			
3405	-29.68	kd	CGS001-3416	IDE	Pitrilysin			
3406	-29.69	oe	ccsbBroad304_13813	ARAF	RAF family			
3407	-29.74	oe	ccsbBroad304_01401	RIT1	-			
3408	-29.75	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
3409	-29.76	kd	CGS001-664	BNIP3	-			
3410	-29.78	kd	CGS001-9354	UBE4A	U-box domain containing			
3411	-29.84	kd	CGS001-9791	PTDSS1	-			
3412	-29.85	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
3413	-29.87	cc		Non Homologous End Joining LOF	-			
3414	-29.87	cc		HSP inhibitor	-			
3415	-29.88	oe	ccsbBroad304_02831	SGK3	SGK family			
3416	-29.89	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
3417	-29.89	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
3418	-29.91	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
3419	-29.92	oe	ccsbBroad304_07219	CDC7	CDC7 family			
3420	-29.93	kd	CGS001-29888	STRN4	WD repeat domain containing			
3421	-29.98	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3422	-30	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
3423	-30.01	kd	CGS001-169436	C9ORF96	-			
3424	-30.02	kd	CGS001-7263	TST	-			
3425	-30.04	kd	CGS001-80135	RPF1	-			
3426	-30.05	kd	CGS001-6185	RPN2	-			
3427	-30.05	kd	CGS001-890	CCNA2	-			
3428	-30.07	kd	CGS001-7039	TGFA	-			
3429	-30.13	kd	CGS001-9270	ITGB1BP1	-			
3430	-30.14	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
3431	-30.2	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3432	-30.23	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
3433	-30.23	kd	CGS001-2010	EMD	-			
3434	-30.24	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
3435	-30.25	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
3436	-30.27	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
3437	-30.31	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
3438	-30.34	kd	CGS001-7128	TNFAIP3	OTU domain containing			
3439	-30.38	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
3440	-30.4	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
3441	-30.4	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
3442	-30.42	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
3443	-30.43	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
3444	-30.45	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
3445	-30.45	kd	CGS001-1827	RCAN1	-			
3446	-30.45	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
3447	-30.46	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
3448	-30.48	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
3449	-30.48	kd	CGS001-23102	TBC1D2B	-			
3450	-30.55	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
3451	-30.58	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
3452	-30.58	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
3453	-30.59	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
3454	-30.6	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
3455	-30.6	oe	ccsbBroad304_03812	PBXIP1	-			
3456	-30.66	kd	CGS001-2987	GUK1	-			
3457	-30.67	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
3458	-30.7	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3459	-30.7	kd	CGS001-64223	MLST8	WD repeat domain containing			
3460	-30.72	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
3461	-30.73	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
3462	-30.73	kd	CGS001-5357	PLS1	EF-hand domain containing			
3463	-30.74	kd	CGS001-9375	TM9SF2	-			
3464	-30.76	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
3465	-30.76	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
3466	-30.77	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
3467	-30.79	kd	CGS001-6632	SNRPD1	-			
3468	-30.81	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
3469	-30.83	kd	CGS001-9140	ATG12	-			
3470	-30.87	kd	CGS001-9797	TATDN2	-			
3471	-30.9	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
3472	-30.92	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
3473	-30.92	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
3474	-30.94	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
3475	-30.94	kd	CGS001-53343	NUDT9	Nudix motif containing			
3476	-31.01	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3477	-31.06	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
3478	-31.07	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
3479	-31.09	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
3480	-31.12	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
3481	-31.13	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
3482	-31.13	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
3483	-31.15	kd	CGS001-5188	PET112	-			
3484	-31.16	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
3485	-31.18	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3486	-31.21	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
3487	-31.23	kd	CGS001-23028	KDM1A	Histone demethylase			
3488	-31.24	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
3489	-31.24	kd	CGS001-29116	MYLIP	-			
3490	-31.26	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
3491	-31.29	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
3492	-31.35	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
3493	-31.36	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
3494	-31.38	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
3495	-31.39	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
3496	-31.41	oe	ccsbBroad304_00486	EFNB2	Ephrins			
3497	-31.45	kd	CGS001-345	APOC3	Apolipoproteins			
3498	-31.46	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3499	-31.49	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
3500	-31.5	kd	CGS001-6119	RPA3	-			
3501	-31.52	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3502	-31.54	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
3503	-31.55	oe	ccsbBroad304_10846	GGT1	CD molecules			
3504	-31.57	kd	CGS001-6895	TARBP2	-			
3505	-31.6	kd	CGS001-11198	SUPT16H	-			
3506	-31.61	kd	CGS001-9926	LPGAT1	-			
3507	-31.61	oe	ccsbBroad304_14011	PAPSS1	-			
3508	-31.62	cc		HMGCR inhibitor	-			
3509	-31.62	kd	CGS001-84971	ATG4D	-			
3510	-31.67	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
3511	-31.67	kd	CGS001-708	C1QBP	-			
3512	-31.7	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
3513	-31.73	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
3514	-31.75	oe	ccsbBroad304_03047	BZW2	-			
3515	-31.77	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
3516	-31.78	kd	CGS001-23451	SF3B1	-			
3517	-31.79	kd	CGS001-57057	TBX20	T-boxes			
3518	-31.81	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
3519	-31.82	oe	ccsbBroad304_01930	CUL2	-			
3520	-31.89	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
3521	-31.9	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
3522	-31.9	kd	CGS001-6514	SLC2A2	Solute carriers			
3523	-31.93	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
3524	-31.93	oe	ccsbBroad304_02857	BAMBI	-			
3525	-31.94	kd	CGS001-11004	KIF2C	Kinesins			
3526	-31.97	kd	CGS001-5498	PPOX	-			
3527	-31.98	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
3528	-31.98	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
3529	-31.99	kd	CGS001-147179	WIPF2	-			
3530	-32	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
3531	-32.03	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
3532	-32.06	kd	CGS001-8435	SOAT2	-			
3533	-32.11	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
3534	-32.15	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
3535	-32.15	kd	CGS001-6500	SKP1	-			
3536	-32.16	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
3537	-32.18	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
3538	-32.21	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
3539	-32.23	kd	CGS001-3420	IDH3B	-			
3540	-32.25	kd	CGS001-7982	ST7	-			
3541	-32.27	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
3542	-32.28	kd	CGS001-4905	NSF	ATPases / AAA-type			
3543	-32.3	kd	CGS001-6258	RXRG	Retinoid X receptors			
3544	-32.32	kd	CGS001-7276	TTR	-			
3545	-32.37	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
3546	-32.38	kd	CGS001-4683	NBN	-			
3547	-32.41	kd	CGS001-29916	SNX11	Sorting nexins			
3548	-32.44	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
3549	-32.44	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
3550	-32.46	kd	CGS001-1384	CRAT	-			
3551	-32.47	oe	ccsbBroad304_05936	CASP2	Caspases			
3552	-32.54	kd	CGS001-10827	FAM114A2	-			
3553	-32.56	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
3554	-32.57	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
3555	-32.58	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
3556	-32.59	oe	ccsbBroad304_02368	TIMM17B	-			
3557	-32.61	cc		Protein phosphatase catalytic subunits LOF	-			
3558	-32.61	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
3559	-32.61	kd	CGS001-4194	MDM4	-			
3560	-32.64	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3561	-32.65	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
3562	-32.7	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
3563	-32.7	kd	CGS001-2621	GAS6	-			
3564	-32.72	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
3565	-32.75	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
3566	-32.77	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
3567	-32.77	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
3568	-32.84	oe	ccsbBroad304_06136	ECHS1	-			
3569	-32.85	kd	CGS001-22887	FOXJ3	Forkhead boxes			
3570	-32.86	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
3571	-32.91	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
3572	-32.92	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
3573	-32.92	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3574	-32.96	oe	ccsbBroad304_08660	SMARCAD1	-			
3575	-32.97	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
3576	-32.97	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
3577	-32.97	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
3578	-32.97	oe	ccsbBroad304_07688	FAM114A2	-			
3579	-32.99	kd	CGS001-58533	SNX6	Sorting nexins			
3580	-33	oe	ccsbBroad304_03859	ENOPH1	-			
3581	-33.05	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
3582	-33.06	kd	CGS001-93594	WDR67	-			
3583	-33.07	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
3584	-33.11	oe	ccsbBroad304_08898	TRAK2	-			
3585	-33.15	oe	ccsbBroad304_06952	SKP1	-			
3586	-33.15	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
3587	-33.16	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
3588	-33.16	kd	CGS001-4267	CD99	CD molecules			
3589	-33.2	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
3590	-33.22	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3591	-33.22	kd	CGS001-10797	MTHFD2	-			
3592	-33.26	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
3593	-33.27	kd	CGS001-121599	SPIC	ETS Transcription Factors			
3594	-33.34	kd	CGS001-5575	PRKAR1B	Protein kinase A			
3595	-33.37	oe	ccsbBroad304_00063	AMPD2	-			
3596	-33.4	kd	CGS001-50846	DHH	-			
3597	-33.41	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
3598	-33.43	kd	CGS001-2072	ERCC4	-			
3599	-33.44	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
3600	-33.46	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
3601	-33.46	kd	CGS001-3579	CXCR2	Chemokine receptors			
3602	-33.47	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
3603	-33.48	oe	ccsbBroad304_06004	CKB	-			
3604	-33.51	kd	CGS001-375449	MAST4	MAST family			
3605	-33.56	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
3606	-33.56	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
3607	-33.56	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
3608	-33.56	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
3609	-33.57	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
3610	-33.59	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
3611	-33.6	oe	ccsbBroad304_00880	IRF2	-			
3612	-33.61	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
3613	-33.64	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
3614	-33.66	kd	CGS001-59343	SENP2	-			
3615	-33.7	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
3616	-33.73	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
3617	-33.75	kd	CGS001-59286	UBL5	-			
3618	-33.8	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
3619	-33.84	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
3620	-33.85	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
3621	-33.86	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
3622	-33.87	oe	ccsbBroad304_03121	NRBF2	-			
3623	-33.88	oe	ccsbBroad304_06783	LGMN	Legumain			
3624	-33.88	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
3625	-33.89	kd	CGS001-2773	GNAI3	-			
3626	-33.91	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
3627	-33.94	oe	ccsbBroad304_01142	PAFAH1B2	-			
3628	-33.96	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
3629	-33.96	oe	ccsbBroad304_02668	PNKP	-			
3630	-33.98	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
3631	-34.01	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
3632	-34.02	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
3633	-34.02	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
3634	-34.03	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
3635	-34.05	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
3636	-34.05	kd	CGS001-5566	PRKACA	Protein kinase A			
3637	-34.06	oe	ccsbBroad304_14143	NUSAP1	-			
3638	-34.06	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
3639	-34.08	oe	ccsbBroad304_02110	VAPB	-			
3640	-34.09	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
3641	-34.09	oe	ccsbBroad304_06292	GNAI2	-			
3642	-34.09	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
3643	-34.11	kd	CGS001-4173	MCM4	-			
3644	-34.12	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3645	-34.12	kd	CGS001-23475	QPRT	-			
3646	-34.13	kd	CGS001-35	ACADS	-			
3647	-34.14	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3648	-34.16	kd	CGS001-6788	STK3	MST subfamily			
3649	-34.19	oe	ccsbBroad304_02458	STK25	YSK subfamily			
3650	-34.2	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
3651	-34.21	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
3652	-34.24	kd	CGS001-10174	SORBS3	-			
3653	-34.27	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
3654	-34.3	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
3655	-34.32	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
3656	-34.35	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
3657	-34.35	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
3658	-34.35	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
3659	-34.38	kd	CGS001-9276	COPB2	WD repeat domain containing			
3660	-34.42	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
3661	-34.43	oe	ccsbBroad304_00651	GNAI3	-			
3662	-34.45	kd	CGS001-8531	CSDA	-			
3663	-34.47	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
3664	-34.51	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
3665	-34.54	oe	ccsbBroad304_03591	ETNK1	-			
3666	-34.55	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
3667	-34.56	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3668	-34.57	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
3669	-34.62	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
3670	-34.63	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
3671	-34.64	kd	CGS001-23118	TAB2	-			
3672	-34.64	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
3673	-34.67	kd	CGS001-10614	HEXIM1	-			
3674	-34.68	kd	CGS001-56922	MCCC1	-			
3675	-34.69	kd	CGS001-5538	PPT1	-			
3676	-34.7	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
3677	-34.71	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
3678	-34.71	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
3679	-34.72	oe	ccsbBroad304_07374	PTPLA	-			
3680	-34.73	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
3681	-34.74	kd	CGS001-55082	ARGLU1	-			
3682	-34.76	kd	CGS001-4665	NAB2	-			
3683	-34.76	kd	CGS001-813	CALU	EF-hand domain containing			
3684	-34.78	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
3685	-34.8	kd	CGS001-10250	SRRM1	-			
3686	-34.81	oe	ccsbBroad304_00222	CASP6	Caspases			
3687	-34.82	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
3688	-34.86	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
3689	-34.87	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
3690	-34.91	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
3691	-34.92	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
3692	-34.94	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
3693	-34.95	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
3694	-34.97	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
3695	-34.98	oe	ccsbBroad304_07888	CBX6	-			
3696	-34.98	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
3697	-35.01	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
3698	-35.02	oe	ccsbBroad304_03040	NKIRAS2	-			
3699	-35.03	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
3700	-35.04	oe	ccsbBroad304_00789	HSBP1	-			
3701	-35.04	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
3702	-35.05	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
3703	-35.06	oe	ccsbBroad304_06318	GPER	-			
3704	-35.06	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
3705	-35.06	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
3706	-35.07	kd	CGS001-3030	HADHA	-			
3707	-35.07	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
3708	-35.08	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
3709	-35.08	kd	CGS001-663	BNIP2	-			
3710	-35.08	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
3711	-35.09	oe	ccsbBroad304_02671	ECD	-			
3712	-35.1	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
3713	-35.1	kd	CGS001-6643	SNX2	Sorting nexins			
3714	-35.12	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
3715	-35.16	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
3716	-35.18	kd	CGS001-1495	CTNNA1	Catenins			
3717	-35.19	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
3718	-35.19	kd	CGS001-29775	CARD10	-			
3719	-35.21	oe	ccsbBroad304_03186	GMNN	-			
3720	-35.21	kd	CGS001-84515	MCM8	-			
3721	-35.22	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
3722	-35.22	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
3723	-35.23	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
3724	-35.23	kd	CGS001-6647	SOD1	-			
3725	-35.25	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
3726	-35.27	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
3727	-35.29	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
3728	-35.34	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
3729	-35.38	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
3730	-35.41	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
3731	-35.42	kd	CGS001-3660	IRF2	-			
3732	-35.45	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
3733	-35.47	kd	CGS001-53632	PRKAG3	AMPK subfamily			
3734	-35.48	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
3735	-35.49	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
3736	-35.5	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
3737	-35.51	oe	ccsbBroad304_00492	EIF5A	-			
3738	-35.52	oe	ccsbBroad304_06178	ERCC5	-			
3739	-35.54	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
3740	-35.54	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
3741	-35.61	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
3742	-35.62	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
3743	-35.63	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
3744	-35.63	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
3745	-35.65	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3746	-35.66	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
3747	-35.66	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
3748	-35.67	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
3749	-35.69	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
3750	-35.7	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
3751	-35.7	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
3752	-35.71	cc		Angiotensin receptor antagonist	-			
3753	-35.71	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
3754	-35.76	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
3755	-35.76	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
3756	-35.77	oe	ccsbBroad304_07088	TP53	-			
3757	-35.77	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
3758	-35.79	kd	CGS001-64858	DCLRE1B	-			
3759	-35.81	oe	ccsbBroad304_09503	KLHDC9	-			
3760	-35.85	cc		Structural maintenance of chromosomes proteins LOF	-			
3761	-35.86	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
3762	-35.86	kd	CGS001-5708	PSMD2	Proteasome subunits			
3763	-35.87	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
3764	-35.9	kd	CGS001-23076	RRP1B	-			
3765	-35.97	kd	CGS001-57521	RPTOR	WD repeat domain containing			
3766	-35.98	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
3767	-36	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
3768	-36.01	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
3769	-36.01	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
3770	-36.03	kd	CGS001-4907	NT5E	Adenosine turnover			
3771	-36.03	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
3772	-36.04	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
3773	-36.06	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3774	-36.11	kd	CGS001-6722	SRF	-			
3775	-36.11	kd	CGS001-9988	DMTF1	-			
3776	-36.11	kd	CGS001-283450	C12ORF51	-			
3777	-36.12	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
3778	-36.14	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
3779	-36.16	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
3780	-36.18	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
3781	-36.19	oe	ccsbBroad304_07528	DMTF1	-			
3782	-36.22	kd	CGS001-5982	RFC2	ATPases / AAA-type			
3783	-36.22	kd	CGS001-439	ASNA1	-			
3784	-36.25	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
3785	-36.26	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
3786	-36.27	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
3787	-36.29	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
3788	-36.29	kd	CGS001-11142	PKIG	-			
3789	-36.31	kd	CGS001-56647	BCCIP	-			
3790	-36.37	oe	ccsbBroad304_00085	APRT	-			
3791	-36.38	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
3792	-36.38	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3793	-36.39	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
3794	-36.39	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
3795	-36.44	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
3796	-36.51	oe	ccsbBroad304_01035	MSH5	-			
3797	-36.52	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
3798	-36.52	kd	CGS001-4547	MTTP	-			
3799	-36.56	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
3800	-36.56	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
3801	-36.57	kd	CGS001-2597	GAPDH	-			
3802	-36.57	kd	CGS001-1840	DTX1	-			
3803	-36.58	kd	CGS001-18	ABAT	GABA turnover			
3804	-36.6	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
3805	-36.64	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
3806	-36.66	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
3807	-36.66	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
3808	-36.69	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
3809	-36.73	oe	ccsbBroad304_03415	GFOD1	-			
3810	-36.74	oe	ccsbBroad304_02862	CCRN4L	-			
3811	-36.75	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
3812	-36.75	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
3813	-36.76	kd	CGS001-2664	GDI1	-			
3814	-36.77	kd	CGS001-7035	TFPI	-			
3815	-36.81	cc		Serotonin receptor antagonist	-			
3816	-36.81	kd	CGS001-2957	GTF2A1	General transcription factors			
3817	-36.86	oe	ccsbBroad304_06523	LIG1	-			
3818	-36.86	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
3819	-36.87	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
3820	-36.89	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
3821	-36.9	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
3822	-36.9	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
3823	-36.9	kd	CGS001-790	CAD	-			
3824	-36.92	oe	ccsbBroad304_03773	CIAPIN1	-			
3825	-36.92	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
3826	-36.94	kd	CGS001-80274	SCUBE1	-			
3827	-37.01	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
3828	-37.01	oe	ccsbBroad304_00657	GNG4	-			
3829	-37.01	kd	CGS001-257397	TAB3	-			
3830	-37.01	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3831	-37.04	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3832	-37.06	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
3833	-37.07	cc		Progesterone receptor agonist	-			
3834	-37.1	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
3835	-37.13	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
3836	-37.14	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
3837	-37.14	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
3838	-37.15	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
3839	-37.16	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
3840	-37.17	kd	CGS001-9322	TRIP10	-			
3841	-37.18	kd	CGS001-384	ARG2	Arginase			
3842	-37.2	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
3843	-37.24	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
3844	-37.26	oe	ccsbBroad304_02502	GNA13	-			
3845	-37.26	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
3846	-37.28	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
3847	-37.29	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
3848	-37.29	kd	CGS001-2073	ERCC5	-			
3849	-37.3	oe	ccsbBroad304_02157	MED21	-			
3850	-37.3	kd	CGS001-8914	TIMELESS	-			
3851	-37.32	oe	ccsbBroad304_05194	LIPH	-			
3852	-37.35	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3853	-37.36	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
3854	-37.36	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
3855	-37.36	kd	CGS001-154197	PNLDC1	-			
3856	-37.38	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
3857	-37.4	oe	ccsbBroad304_08888	ACD	-			
3858	-37.4	kd	CGS001-6827	SUPT4H1	-			
3859	-37.4	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
3860	-37.44	oe	ccsbBroad304_02716	NMNAT2	-			
3861	-37.45	oe	ccsbBroad304_06518	LDHA	-			
3862	-37.45	kd	CGS001-5378	PMS1	-			
3863	-37.45	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
3864	-37.46	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
3865	-37.48	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
3866	-37.48	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
3867	-37.52	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
3868	-37.52	kd	CGS001-2230	FDX1	-			
3869	-37.53	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
3870	-37.53	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
3871	-37.56	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3872	-37.57	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
3873	-37.57	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
3874	-37.59	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
3875	-37.6	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
3876	-37.62	oe	ccsbBroad304_07466	VGLL4	-			
3877	-37.62	oe	ccsbBroad304_03164	MTERFD1	-			
3878	-37.62	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
3879	-37.63	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
3880	-37.65	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
3881	-37.65	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
3882	-37.66	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
3883	-37.68	kd	CGS001-57721	METTL14	-			
3884	-37.7	kd	CGS001-1955	MEGF9	-			
3885	-37.72	kd	CGS001-1962	EHHADH	-			
3886	-37.75	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
3887	-37.76	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
3888	-37.76	kd	CGS001-11014	KDELR2	-			
3889	-37.77	kd	CGS001-79073	TMEM109	-			
3890	-37.78	kd	CGS001-5920	RARRES3	-			
3891	-37.79	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
3892	-37.83	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
3893	-37.84	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
3894	-37.86	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
3895	-37.86	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
3896	-37.9	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
3897	-37.97	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
3898	-37.97	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
3899	-37.97	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
3900	-38.06	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
3901	-38.11	oe	ccsbBroad304_05749	A2M	-			
3902	-38.11	oe	ccsbBroad304_04626	EGLN3	-			
3903	-38.12	cc		LIM class homeoboxes GOF	-			
3904	-38.16	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
3905	-38.19	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
3906	-38.22	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
3907	-38.22	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
3908	-38.24	kd	CGS001-1611	DAP	-			
3909	-38.24	kd	CGS001-1604	CD55	CD molecules			
3910	-38.25	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
3911	-38.27	kd	CGS001-11243	PMF1	-			
3912	-38.28	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
3913	-38.3	oe	ccsbBroad304_03023	CRCP	-			
3914	-38.33	oe	ccsbBroad304_06565	MB	-			
3915	-38.36	oe	ccsbBroad304_02229	TRAM2	-			
3916	-38.36	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
3917	-38.36	kd	CGS001-6499	SKIV2L	-			
3918	-38.38	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
3919	-38.4	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3920	-38.41	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
3921	-38.42	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
3922	-38.46	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
3923	-38.47	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
3924	-38.48	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
3925	-38.49	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
3926	-38.55	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
3927	-38.56	oe	ccsbBroad304_00795	HSF2	-			
3928	-38.56	kd	CGS001-523	ATP6V1A	ATPases / V-type			
3929	-38.57	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
3930	-38.59	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3931	-38.59	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
3932	-38.6	oe	ccsbBroad304_00728	HBE1	-			
3933	-38.71	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
3934	-38.72	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
3935	-38.75	kd	CGS001-31	ACACA	Carboxylases			
3936	-38.76	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
3937	-38.77	oe	ccsbBroad304_06226	FTL	-			
3938	-38.78	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
3939	-38.79	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
3940	-38.79	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3941	-38.8	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3942	-38.81	oe	ccsbBroad304_06975	SMARCC2	-			
3943	-38.87	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
3944	-38.9	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
3945	-38.92	kd	CGS001-54205	CYCS	-			
3946	-38.93	cc		Lysine acetyltransferases LOF	-			
3947	-38.94	kd	CGS001-1655	DDX5	DEAD-boxes			
3948	-38.95	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
3949	-39.03	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
3950	-39.04	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
3951	-39.04	oe	ccsbBroad304_01641	TAF13	-			
3952	-39.06	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
3953	-39.1	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
3954	-39.11	oe	ccsbBroad304_00710	GUSB	-			
3955	-39.12	oe	ccsbBroad304_06998	SRPK1	SRPK family			
3956	-39.13	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
3957	-39.15	oe	ccsbBroad304_01962	STK16	NAK family			
3958	-39.15	oe	ccsbBroad304_03625	HIF1AN	-			
3959	-39.16	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
3960	-39.17	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
3961	-39.23	oe	ccsbBroad304_10758	CTBP2	-			
3962	-39.26	oe	ccsbBroad304_03155	DHH	-			
3963	-39.31	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
3964	-39.4	oe	ccsbBroad304_01699	TPD52L2	-			
3965	-39.41	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
3966	-39.42	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
3967	-39.45	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
3968	-39.46	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
3969	-39.46	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
3970	-39.46	kd	CGS001-25966	C2CD2	-			
3971	-39.47	oe	ccsbBroad304_06188	F10	Chymotrypsin			
3972	-39.47	kd	CGS001-1029	CDKN2A	-			
3973	-39.5	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
3974	-39.56	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
3975	-39.58	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
3976	-39.6	kd	CGS001-2852	GPER	-			
3977	-39.64	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
3978	-39.7	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
3979	-39.7	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
3980	-39.71	oe	ccsbBroad304_01304	PSEN1	Presenilin			
3981	-39.77	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
3982	-39.81	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
3983	-39.83	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
3984	-39.86	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
3985	-39.86	kd	CGS001-1841	DTYMK	-			
3986	-39.87	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
3987	-39.89	oe	ccsbBroad304_13633	PI4KAP2	-			
3988	-39.92	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
3989	-39.95	oe	ccsbBroad304_07616	ZNF238	-			
3990	-39.98	kd	CGS001-7086	TKT	-			
3991	-39.98	oe	ccsbBroad304_03950	ATG3	-			
3992	-39.99	oe	ccsbBroad304_01659	TERF1	-			
3993	-39.99	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
3994	-40	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3995	-40.01	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
3996	-40.06	oe	ccsbBroad304_02487	TXNIP	-			
3997	-40.06	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
3998	-40.08	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
3999	-40.09	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
4000	-40.19	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4001	-40.22	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
4002	-40.22	kd	CGS001-10252	SPRY1	-			
4003	-40.24	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
4004	-40.24	kd	CGS001-54805	CNNM2	-			
4005	-40.25	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
4006	-40.25	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
4007	-40.28	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
4008	-40.29	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
4009	-40.3	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
4010	-40.35	oe	ccsbBroad304_05948	CCND2	-			
4011	-40.4	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
4012	-40.43	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
4013	-40.44	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
4014	-40.44	oe	ccsbBroad304_00661	GNGT2	-			
4015	-40.44	kd	CGS001-2030	SLC29A1	SLC29 family			
4016	-40.46	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
4017	-40.47	oe	ccsbBroad304_06985	SORD	-			
4018	-40.47	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
4019	-40.48	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
4020	-40.48	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
4021	-40.49	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
4022	-40.5	kd	CGS001-5621	PRNP	CD molecules			
4023	-40.51	kd	CGS001-23210	JMJD6	-			
4024	-40.53	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
4025	-40.54	cc		Rho associated kinase inhibitor	-			
4026	-40.55	oe	ccsbBroad304_04064	PRR15L	-			
4027	-40.57	kd	CGS001-8731	RNMT	-			
4028	-40.6	oe	ccsbBroad304_03573	BRF2	-			
4029	-40.6	kd	CGS001-1490	CTGF	-			
4030	-40.61	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
4031	-40.68	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
4032	-40.68	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
4033	-40.68	kd	CGS001-6519	SLC3A1	SLC3 family			
4034	-40.69	oe	ccsbBroad304_00510	EPHX2	-			
4035	-40.7	oe	ccsbBroad304_00854	IL8	-			
4036	-40.7	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
4037	-40.7	kd	CGS001-10482	NXF1	-			
4038	-40.72	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
4039	-40.72	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
4040	-40.75	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
4041	-40.76	kd	CGS001-6469	SHH	-			
4042	-40.78	oe	ccsbBroad304_02869	ASF1A	-			
4043	-40.8	cc		Canonical high mobility group proteins LOF	-			
4044	-40.83	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
4045	-40.83	kd	CGS001-87	ACTN1	EF-hand domain containing			
4046	-40.86	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
4047	-40.87	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
4048	-40.87	kd	CGS001-348	APOE	Apolipoproteins			
4049	-40.88	cc		HDAC inhibitor	-			
4050	-40.88	kd	CGS001-170463	SSBP4	-			
4051	-40.88	kd	CGS001-6210	RPS15A	S ribosomal proteins			
4052	-40.91	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
4053	-40.98	kd	CGS001-22921	MSRB2	-			
4054	-40.99	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
4055	-41.02	oe	ccsbBroad304_06711	PFAS	-			
4056	-41.03	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
4057	-41.04	oe	ccsbBroad304_03798	PHTF2	-			
4058	-41.04	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4059	-41.06	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
4060	-41.08	kd	CGS001-3663	IRF5	-			
4061	-41.11	kd	CGS001-8428	STK24	YSK subfamily			
4062	-41.12	kd	CGS001-30836	DNTTIP2	-			
4063	-41.14	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
4064	-41.14	kd	CGS001-57018	CCNL1	-			
4065	-41.15	kd	CGS001-60493	FASTKD5	-			
4066	-41.16	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
4067	-41.16	kd	CGS001-642	BLMH	-			
4068	-41.18	oe	ccsbBroad304_07884	RYBP	-			
4069	-41.19	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
4070	-41.19	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
4071	-41.21	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
4072	-41.23	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4073	-41.24	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
4074	-41.25	kd	CGS001-5411	PNN	-			
4075	-41.26	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
4076	-41.29	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
4077	-41.32	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
4078	-41.32	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
4079	-41.33	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
4080	-41.33	kd	CGS001-3161	HMMR	CD molecules			
4081	-41.34	oe	ccsbBroad304_02203	MAD2L1BP	-			
4082	-41.34	kd	CGS001-2197	FAU	S ribosomal proteins			
4083	-41.35	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
4084	-41.35	oe	ccsbBroad304_01640	TAF12	-			
4085	-41.35	oe	ccsbBroad304_02109	XPR1	-			
4086	-41.38	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
4087	-41.42	oe	ccsbBroad304_02589	COPS5	-			
4088	-41.45	kd	CGS001-4836	NMT1	-			
4089	-41.48	kd	CGS001-3845	KRAS	RAS subfamily			
4090	-41.49	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
4091	-41.51	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
4092	-41.51	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
4093	-41.51	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
4094	-41.52	kd	CGS001-397	ARHGDIB	Endogenous ligands			
4095	-41.56	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
4096	-41.58	kd	CGS001-2155	F7	Chymotrypsin			
4097	-41.6	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
4098	-41.61	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
4099	-41.64	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
4100	-41.66	kd	CGS001-7099	TLR4	Toll-like receptor family			
4101	-41.72	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4102	-41.72	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
4103	-41.73	kd	CGS001-4200	ME2	-			
4104	-41.76	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
4105	-41.81	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
4106	-41.82	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
4107	-41.82	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
4108	-41.84	oe	ccsbBroad304_09354	IGSF8	CD molecules			
4109	-41.87	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
4110	-41.88	cc		Aurora kinase inhibitor	-			
4111	-41.88	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
4112	-41.9	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
4113	-41.97	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
4114	-42.01	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
4115	-42.02	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
4116	-42.04	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
4117	-42.05	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
4118	-42.06	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
4119	-42.08	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
4120	-42.08	kd	CGS001-85004	RERG	-			
4121	-42.09	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
4122	-42.13	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
4123	-42.14	kd	CGS001-3029	HAGH	-			
4124	-42.19	oe	ccsbBroad304_01661	TFCP2	-			
4125	-42.19	kd	CGS001-634	CEACAM1	CD molecules			
4126	-42.21	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
4127	-42.21	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
4128	-42.21	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
4129	-42.22	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
4130	-42.24	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
4131	-42.26	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
4132	-42.28	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4133	-42.32	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
4134	-42.35	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
4135	-42.36	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
4136	-42.41	oe	ccsbBroad304_06663	OAS1	-			
4137	-42.42	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
4138	-42.48	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
4139	-42.49	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
4140	-42.49	kd	CGS001-9218	VAPA	-			
4141	-42.53	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
4142	-42.56	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
4143	-42.58	oe	ccsbBroad304_10207	ERLIN1	-			
4144	-42.64	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
4145	-42.66	oe	ccsbBroad304_01716	TSN	-			
4146	-42.66	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
4147	-42.68	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
4148	-42.79	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
4149	-42.8	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
4150	-42.81	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
4151	-42.83	oe	ccsbBroad304_01019	MLH1	-			
4152	-42.86	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
4153	-42.86	oe	ccsbBroad304_02285	MED6	-			
4154	-42.86	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
4155	-42.86	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
4156	-42.88	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
4157	-42.92	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
4158	-42.93	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
4159	-42.93	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
4160	-42.93	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
4161	-42.96	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4162	-42.97	oe	ccsbBroad304_04490	RSPH1	-			
4163	-43	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
4164	-43	kd	CGS001-150280	HORMAD2	-			
4165	-43.09	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
4166	-43.1	kd	CGS001-7389	UROD	-			
4167	-43.12	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
4168	-43.15	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
4169	-43.18	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
4170	-43.19	oe	ccsbBroad304_09281	TPD52L3	-			
4171	-43.21	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4172	-43.22	oe	ccsbBroad304_08879	CASD1	-			
4173	-43.25	oe	ccsbBroad304_06386	HNMT	-			
4174	-43.26	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
4175	-43.27	oe	ccsbBroad304_01723	TTK	TTK family			
4176	-43.28	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
4177	-43.31	oe	ccsbBroad304_06008	AP2M1	-			
4178	-43.31	kd	CGS001-11157	LSM6	-			
4179	-43.31	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
4180	-43.32	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
4181	-43.33	kd	CGS001-7248	TSC1	-			
4182	-43.34	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
4183	-43.36	kd	CGS001-6646	SOAT1	-			
4184	-43.36	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
4185	-43.37	oe	ccsbBroad304_06324	GPX7	-			
4186	-43.4	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
4187	-43.4	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
4188	-43.43	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
4189	-43.44	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
4190	-43.44	kd	CGS001-5480	PPIC	-			
4191	-43.46	oe	ccsbBroad304_00954	LYN	Src family			
4192	-43.47	kd	CGS001-2747	GLUD2	-			
4193	-43.49	oe	ccsbBroad304_02576	MLLT11	-			
4194	-43.53	oe	ccsbBroad304_08322	UFM1	-			
4195	-43.53	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4196	-43.54	oe	ccsbBroad304_06253	GALT	-			
4197	-43.56	kd	CGS001-6772	STAT1	SH2 domain containing			
4198	-43.57	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
4199	-43.58	oe	ccsbBroad304_00572	FKBP3	-			
4200	-43.61	oe	ccsbBroad304_07875	SPECC1L	-			
4201	-43.63	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
4202	-43.64	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
4203	-43.66	kd	CGS001-4300	MLLT3	-			
4204	-43.68	kd	CGS001-5045	FURIN	Subtilisin			
4205	-43.72	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
4206	-43.73	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
4207	-43.76	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
4208	-43.81	kd	CGS001-8692	HYAL2	-			
4209	-43.84	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
4210	-43.84	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
4211	-43.86	kd	CGS001-9455	HOMER2	-			
4212	-43.87	kd	CGS001-3065	HDAC1	Histone deacetylases			
4213	-43.9	kd	CGS001-3725	JUN	basic leucine zipper proteins			
4214	-43.94	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
4215	-43.95	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
4216	-43.95	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
4217	-44	kd	CGS001-6491	STIL	-			
4218	-44.02	kd	CGS001-2963	GTF2F2	General transcription factors			
4219	-44.06	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
4220	-44.07	kd	CGS001-1155	TBCB	-			
4221	-44.09	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4222	-44.09	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
4223	-44.14	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
4224	-44.15	kd	CGS001-7296	TXNRD1	-			
4225	-44.17	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
4226	-44.18	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
4227	-44.2	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
4228	-44.23	kd	CGS001-55165	CEP55	-			
4229	-44.3	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
4230	-44.37	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
4231	-44.4	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
4232	-44.44	oe	ccsbBroad304_05937	CASP7	Caspases			
4233	-44.44	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
4234	-44.54	kd	CGS001-8678	BECN1	-			
4235	-44.55	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4236	-44.58	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
4237	-44.59	oe	ccsbBroad304_01395	RFX5	-			
4238	-44.62	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
4239	-44.62	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
4240	-44.62	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
4241	-44.63	oe	ccsbBroad304_00794	HSF1	-			
4242	-44.69	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4243	-44.71	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4244	-44.73	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
4245	-44.74	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
4246	-44.75	kd	CGS001-10523	CHERP	G patch domain containing			
4247	-44.78	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
4248	-44.8	kd	CGS001-10681	GNB5	WD repeat domain containing			
4249	-44.81	kd	CGS001-2548	GAA	Glycosidases			
4250	-44.82	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
4251	-44.85	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
4252	-44.88	kd	CGS001-400	ARL1	ADP-ribosylation factors			
4253	-44.88	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
4254	-44.89	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
4255	-44.93	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
4256	-44.98	oe	ccsbBroad304_00397	CTSK	Cathepsins			
4257	-45	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
4258	-45.08	oe	ccsbBroad304_08802	ELAC2	-			
4259	-45.08	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4260	-45.08	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
4261	-45.14	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
4262	-45.15	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
4263	-45.2	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
4264	-45.21	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
4265	-45.22	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
4266	-45.22	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
4267	-45.22	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
4268	-45.22	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
4269	-45.24	kd	CGS001-347736	NME9	-			
4270	-45.25	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
4271	-45.26	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
4272	-45.29	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
4273	-45.29	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
4274	-45.31	oe	ccsbBroad304_01577	SOD1	-			
4275	-45.33	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
4276	-45.35	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
4277	-45.39	kd	CGS001-57048	PLSCR3	-			
4278	-45.4	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
4279	-45.42	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
4280	-45.42	kd	CGS001-27113	BBC3	-			
4281	-45.43	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
4282	-45.45	cc		BCL inhibitor	-			
4283	-45.46	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
4284	-45.47	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
4285	-45.51	cc		Calmodulin antagonist	-			
4286	-45.52	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
4287	-45.53	oe	ccsbBroad304_01101	NME1	-			
4288	-45.55	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
4289	-45.59	oe	ccsbBroad304_06235	G6PD	-			
4290	-45.6	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
4291	-45.61	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
4292	-45.67	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
4293	-45.68	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
4294	-45.74	oe	ccsbBroad304_06094	DFFA	-			
4295	-45.74	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
4296	-45.76	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
4297	-45.78	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
4298	-45.79	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
4299	-45.79	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
4300	-45.82	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
4301	-45.83	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
4302	-45.85	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
4303	-45.88	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4304	-45.89	kd	CGS001-51805	COQ3	-			
4305	-45.92	oe	ccsbBroad304_07277	RTCD1	-			
4306	-45.92	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
4307	-45.93	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
4308	-45.94	cc		EGFR inhibitor	-			
4309	-45.96	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
4310	-45.99	oe	ccsbBroad304_00542	FBP1	-			
4311	-45.99	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
4312	-46.02	oe	ccsbBroad304_05439	O3FAR1	-			
4313	-46.03	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
4314	-46.04	cc		Cyclin dependent kinases LOF	-			
4315	-46.08	cc		Tubulin inhibitor	-			
4316	-46.09	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4317	-46.09	kd	CGS001-5366	PMAIP1	-			
4318	-46.1	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
4319	-46.12	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
4320	-46.15	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
4321	-46.15	kd	CGS001-3669	ISG20	-			
4322	-46.2	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
4323	-46.21	kd	CGS001-8464	SUPT3H	-			
4324	-46.21	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
4325	-46.24	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
4326	-46.25	oe	ccsbBroad304_00237	CCND3	-			
4327	-46.28	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
4328	-46.3	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4329	-46.33	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
4330	-46.35	oe	ccsbBroad304_01166	PDK2	PDHK family			
4331	-46.36	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
4332	-46.42	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
4333	-46.44	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
4334	-46.45	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
4335	-46.51	oe	ccsbBroad304_04675	ATG4A	-			
4336	-46.51	kd	CGS001-8467	SMARCA5	-			
4337	-46.55	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
4338	-46.55	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
4339	-46.56	kd	CGS001-64428	NARFL	-			
4340	-46.57	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
4341	-46.59	oe	ccsbBroad304_00810	HYAL1	-			
4342	-46.59	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
4343	-46.59	kd	CGS001-4668	NAGA	-			
4344	-46.62	kd	CGS001-5660	PSAP	Endogenous ligands			
4345	-46.63	cc		P38 MAPK inhibitor	-			
4346	-46.64	kd	CGS001-4087	SMAD2	SMADs			
4347	-46.66	kd	CGS001-350	APOH	Apolipoproteins			
4348	-46.71	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
4349	-46.74	kd	CGS001-23386	NUDCD3	-			
4350	-46.76	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
4351	-46.79	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
4352	-46.8	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
4353	-46.81	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
4354	-46.81	kd	CGS001-403	ARL3	ADP-ribosylation factors			
4355	-46.84	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
4356	-46.91	kd	CGS001-51160	VPS28	-			
4357	-46.94	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
4358	-46.94	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
4359	-47.01	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4360	-47.02	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
4361	-47.03	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4362	-47.06	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
4363	-47.06	kd	CGS001-3932	LCK	Src family			
4364	-47.07	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
4365	-47.08	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
4366	-47.09	cc		CDK inhibitor	-			
4367	-47.09	oe	ccsbBroad304_02822	ARFIP2	-			
4368	-47.12	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
4369	-47.13	kd	CGS001-9415	FADS2	Fatty acid desaturases			
4370	-47.17	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
4371	-47.21	oe	ccsbBroad304_03544	FAIM	-			
4372	-47.23	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
4373	-47.27	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
4374	-47.27	kd	CGS001-3575	IL7R	IL-2 receptor family			
4375	-47.33	oe	ccsbBroad304_01091	NFIB	-			
4376	-47.35	oe	ccsbBroad304_06095	DFFB	-			
4377	-47.35	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
4378	-47.44	oe	ccsbBroad304_07861	COBL	-			
4379	-47.44	kd	CGS001-54861	SNRK	SNRK subfamily			
4380	-47.46	kd	CGS001-8985	PLOD3	-			
4381	-47.48	oe	ccsbBroad304_02219	MORF4L2	-			
4382	-47.48	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
4383	-47.49	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
4384	-47.52	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
4385	-47.53	kd	CGS001-8569	MKNK1	MKN subfamily			
4386	-47.54	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
4387	-47.61	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
4388	-47.61	oe	ccsbBroad304_06290	GNA15	-			
4389	-47.61	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4390	-47.63	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
4391	-47.64	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
4392	-47.66	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
4393	-47.66	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
4394	-47.67	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
4395	-47.68	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
4396	-47.73	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
4397	-47.74	kd	CGS001-7832	BTG2	-			
4398	-47.79	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
4399	-47.82	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
4400	-47.84	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
4401	-47.86	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
4402	-47.89	kd	CGS001-29911	HOOK2	-			
4403	-47.94	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
4404	-47.97	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
4405	-47.99	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
4406	-48.01	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
4407	-48.03	oe	ccsbBroad304_03917	RBKS	-			
4408	-48.06	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
4409	-48.13	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4410	-48.13	kd	CGS001-23499	MACF1	EF-hand domain containing			
4411	-48.15	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
4412	-48.16	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
4413	-48.17	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
4414	-48.2	kd	CGS001-51128	SAR1B	-			
4415	-48.22	oe	ccsbBroad304_03615	ZNF673	-			
4416	-48.24	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
4417	-48.24	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
4418	-48.25	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
4419	-48.26	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
4420	-48.27	kd	CGS001-819	CAMLG	-			
4421	-48.28	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
4422	-48.35	cc		Aminoacyl tRNA synthetases class II LOF	-			
4423	-48.35	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4424	-48.35	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
4425	-48.39	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
4426	-48.4	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
4427	-48.53	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
4428	-48.54	oe	ccsbBroad304_01674	TIMP4	-			
4429	-48.56	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
4430	-48.61	kd	CGS001-727	C5	Endogenous ligands			
4431	-48.65	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
4432	-48.67	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
4433	-48.71	kd	CGS001-1154	CISH	SH2 domain containing			
4434	-48.71	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
4435	-48.73	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
4436	-48.74	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
4437	-48.77	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
4438	-48.78	oe	ccsbBroad304_08023	EIF2C1	-			
4439	-48.78	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
4440	-48.81	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
4441	-48.82	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4442	-48.91	kd	CGS001-3479	IGF1	Endogenous ligands			
4443	-48.94	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
4444	-48.98	oe	ccsbBroad304_09821	TMEM154	-			
4445	-49.01	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
4446	-49.02	oe	ccsbBroad304_03310	LCMT1	-			
4447	-49.02	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
4448	-49.08	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
4449	-49.14	oe	ccsbBroad304_09254	PAQR8	-			
4450	-49.15	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4451	-49.18	oe	ccsbBroad304_01654	TCTA	-			
4452	-49.19	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
4453	-49.2	kd	CGS001-4817	NIT1	-			
4454	-49.21	kd	CGS001-55577	NAGK	-			
4455	-49.25	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
4456	-49.26	cc		Bacterial cell wall synthesis inhibitor	-			
4457	-49.27	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
4458	-49.29	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
4459	-49.29	kd	CGS001-475	ATOX1	-			
4460	-49.34	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
4461	-49.37	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4462	-49.37	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
4463	-49.38	oe	ccsbBroad304_08694	TBX20	T-boxes			
4464	-49.4	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
4465	-49.4	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
4466	-49.41	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
4467	-49.42	kd	CGS001-174	AFP	-			
4468	-49.46	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
4469	-49.47	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
4470	-49.47	kd	CGS001-10617	STAMBP	-			
4471	-49.47	kd	CGS001-4292	MLH1	-			
4472	-49.53	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
4473	-49.54	kd	CGS001-6622	SNCA	Parkinson disease			
4474	-49.55	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4475	-49.6	oe	ccsbBroad304_02012	FADD	-			
4476	-49.61	oe	ccsbBroad304_03928	RRAGC	-			
4477	-49.64	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4478	-49.65	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
4479	-49.66	oe	ccsbBroad304_10212	GRHL3	-			
4480	-49.7	kd	CGS001-56005	C19ORF10	-			
4481	-49.71	cc		NFKB Activation GOF	-			
4482	-49.74	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
4483	-49.76	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
4484	-49.76	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
4485	-49.81	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
4486	-49.84	oe	ccsbBroad304_03264	UBAP1	-			
4487	-49.86	cc		Interleukins GOF	-			
4488	-49.87	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
4489	-49.89	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
4490	-49.94	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
4491	-49.94	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
4492	-49.95	kd	CGS001-58477	SRPRB	-			
4493	-50	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
4494	-50.01	kd	CGS001-56993	TOMM22	-			
4495	-50.02	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
4496	-50.07	kd	CGS001-498	ATP5A1	ATPases / F-type			
4497	-50.09	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4498	-50.1	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
4499	-50.11	oe	ccsbBroad304_01205	PIN1	-			
4500	-50.11	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
4501	-50.13	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
4502	-50.22	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
4503	-50.27	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
4504	-50.28	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
4505	-50.3	oe	ccsbBroad304_08839	IFIH1	-			
4506	-50.3	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
4507	-50.35	oe	ccsbBroad304_01372	RALB	-			
4508	-50.36	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
4509	-50.36	kd	CGS001-64422	ATG3	-			
4510	-50.37	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
4511	-50.4	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
4512	-50.43	kd	CGS001-5573	PRKAR1A	Protein kinase A			
4513	-50.43	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
4514	-50.45	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
4515	-50.47	oe	ccsbBroad304_02443	HAX1	-			
4516	-50.49	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
4517	-50.49	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
4518	-50.5	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
4519	-50.5	kd	CGS001-1070	CETN3	EF-hand domain containing			
4520	-50.55	kd	CGS001-2115	ETV1	ETS Transcription Factors			
4521	-50.55	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
4522	-50.58	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
4523	-50.6	kd	CGS001-51290	ERGIC2	-			
4524	-50.64	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
4525	-50.66	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
4526	-50.68	cc		Histone deacetylases LOF	-			
4527	-50.73	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
4528	-50.74	cp	BRD-K15842202	eudesmic-acid	-666			-666
4529	-50.77	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
4530	-50.77	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
4531	-50.79	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
4532	-50.82	cc		Gamma secretase inhibitor	-			
4533	-50.85	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4534	-50.91	kd	CGS001-7251	TSG101	-			
4535	-50.92	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
4536	-50.99	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
4537	-51.06	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
4538	-51.13	oe	ccsbBroad304_06225	FTH1	-			
4539	-51.15	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
4540	-51.16	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
4541	-51.16	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
4542	-51.18	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4543	-51.22	kd	CGS001-5743	PTGS2	Cyclooxygenase			
4544	-51.24	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
4545	-51.25	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
4546	-51.26	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
4547	-51.26	kd	CGS001-178	AGL	-			
4548	-51.29	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
4549	-51.31	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
4550	-51.34	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
4551	-51.38	oe	ccsbBroad304_07326	EIF2B2	-			
4552	-51.4	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
4553	-51.41	kd	CGS001-3909	LAMA3	Laminins			
4554	-51.43	oe	ccsbBroad304_02048	BCL10	-			
4555	-51.44	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
4556	-51.47	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
4557	-51.49	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
4558	-51.52	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
4559	-51.54	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
4560	-51.54	kd	CGS001-427	ASAH1	Acid ceramidase			
4561	-51.55	oe	ccsbBroad304_02772	ICMT	-			
4562	-51.56	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
4563	-51.57	kd	CGS001-5110	PCMT1	-			
4564	-51.58	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
4565	-51.59	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
4566	-51.6	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
4567	-51.6	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
4568	-51.61	kd	CGS001-3827	KNG1	Endogenous ligands			
4569	-51.71	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
4570	-51.74	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
4571	-51.77	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
4572	-51.8	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
4573	-51.8	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4574	-51.81	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4575	-51.82	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
4576	-51.82	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
4577	-51.85	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
4578	-51.86	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
4579	-51.92	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
4580	-51.96	oe	ccsbBroad304_09578	PASD1	-			
4581	-51.99	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4582	-52	oe	ccsbBroad304_00231	CBFB	-			
4583	-52.11	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
4584	-52.12	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
4585	-52.14	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
4586	-52.15	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
4587	-52.15	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
4588	-52.16	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
4589	-52.17	kd	CGS001-5925	RB1	Endogenous ligands			
4590	-52.18	kd	CGS001-11168	PSIP1	-			
4591	-52.2	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
4592	-52.25	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
4593	-52.29	kd	CGS001-5997	RGS2	Endogenous ligands			
4594	-52.31	cc		Sterol demethylase inhibitor	-			
4595	-52.35	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
4596	-52.37	oe	ccsbBroad304_05763	ACTB	-			
4597	-52.4	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
4598	-52.4	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
4599	-52.41	kd	CGS001-183	AGT	Endogenous ligands			
4600	-52.42	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
4601	-52.42	oe	ccsbBroad304_06013	CLPTM1	-			
4602	-52.42	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
4603	-52.43	oe	ccsbBroad304_02626	PKIG	-			
4604	-52.45	kd	CGS001-10476	ATP5H	ATPases / F-type			
4605	-52.51	oe	ccsbBroad304_09881	RFX6	-			
4606	-52.62	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
4607	-52.62	kd	CGS001-3171	FOXA3	Forkhead boxes			
4608	-52.63	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
4609	-52.66	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
4610	-52.67	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
4611	-52.69	oe	ccsbBroad304_00250	CD19	CD molecules			
4612	-52.7	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
4613	-52.7	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
4614	-52.75	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
4615	-52.77	oe	ccsbBroad304_01933	TEAD2	-			
4616	-52.81	oe	ccsbBroad304_00471	E2F6	-			
4617	-52.82	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
4618	-52.82	kd	CGS001-1633	DCK	-			
4619	-52.84	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
4620	-52.85	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
4621	-52.87	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
4622	-52.91	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
4623	-52.91	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
4624	-52.91	kd	CGS001-23621	BACE1	Pepsin			
4625	-52.94	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
4626	-52.97	oe	ccsbBroad304_02919	KIAA1279	-			
4627	-53	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
4628	-53.02	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
4629	-53.03	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
4630	-53.07	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
4631	-53.09	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
4632	-53.11	kd	CGS001-54386	TERF2IP	-			
4633	-53.13	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
4634	-53.16	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4635	-53.16	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
4636	-53.2	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
4637	-53.22	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
4638	-53.23	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
4639	-53.23	kd	CGS001-3551	IKBKB	IKK family			
4640	-53.23	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
4641	-53.24	oe	ccsbBroad304_07178	ZFP112	-			
4642	-53.27	kd	CGS001-5909	RAP1GAP	-			
4643	-53.36	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
4644	-53.37	kd	CGS001-7187	TRAF3	-			
4645	-53.38	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
4646	-53.41	kd	CGS001-27125	AFF4	-			
4647	-53.45	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
4648	-53.46	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
4649	-53.47	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
4650	-53.48	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
4651	-53.5	kd	CGS001-5230	PGK1	-			
4652	-53.51	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
4653	-53.52	oe	ccsbBroad304_08596	EAPP	-			
4654	-53.58	oe	ccsbBroad304_03554	NAT10	-			
4655	-53.59	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
4656	-53.6	oe	ccsbBroad304_08645	BCCIP	-			
4657	-53.61	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
4658	-53.69	oe	ccsbBroad304_00430	GADD45A	-			
4659	-53.7	kd	CGS001-8996	NOL3	-			
4660	-53.71	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
4661	-53.71	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
4662	-53.72	kd	CGS001-11124	FAF1	UBX domain containing			
4663	-53.73	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
4664	-53.77	cc		FXR antagonist	-			
4665	-53.77	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
4666	-53.81	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
4667	-53.82	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
4668	-53.84	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
4669	-53.89	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
4670	-53.91	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
4671	-53.93	oe	ccsbBroad304_05192	SPRED2	-			
4672	-53.93	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
4673	-53.93	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
4674	-53.96	cc		Imidazoline ligand	-			
4675	-53.96	kd	CGS001-5624	PROC	Endogenous ligands			
4676	-53.99	kd	CGS001-56916	SMARCAD1	-			
4677	-53.99	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
4678	-54.02	oe	ccsbBroad304_07851	FAM120A	-			
4679	-54.05	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
4680	-54.13	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
4681	-54.15	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
4682	-54.15	kd	CGS001-6118	RPA2	-			
4683	-54.22	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
4684	-54.23	oe	ccsbBroad304_00811	ICAM1	CD molecules			
4685	-54.26	oe	ccsbBroad304_07761	CORO1A	Coronins			
4686	-54.31	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
4687	-54.32	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4688	-54.32	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
4689	-54.33	oe	ccsbBroad304_03433	DDIT4	-			
4690	-54.36	kd	CGS001-226	ALDOA	-			
4691	-54.37	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
4692	-54.43	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
4693	-54.43	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
4694	-54.44	oe	ccsbBroad304_07511	KIF14	Kinesins			
4695	-54.46	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
4696	-54.53	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
4697	-54.55	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
4698	-54.55	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
4699	-54.57	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
4700	-54.58	kd	CGS001-8772	FADD	-			
4701	-54.65	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
4702	-54.68	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
4703	-54.7	oe	ccsbBroad304_03089	PACSIN3	-			
4704	-54.71	kd	CGS001-5581	PRKCE	Eta subfamily			
4705	-54.71	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
4706	-54.76	cc		Aromatase inhibitor	-			
4707	-54.76	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
4708	-54.76	kd	CGS001-3482	IGF2R	CD molecules			
4709	-54.76	kd	CGS001-11007	CCDC85B	-			
4710	-54.77	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
4711	-54.79	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
4712	-54.79	oe	ccsbBroad304_02890	SYF2	-			
4713	-54.81	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
4714	-54.82	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
4715	-54.85	oe	ccsbBroad304_00987	MCM3	-			
4716	-54.86	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
4717	-54.87	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
4718	-54.88	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
4719	-54.9	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
4720	-54.96	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4721	-55.01	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
4722	-55.06	cc		IKK inhibitor	-			
4723	-55.07	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4724	-55.07	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4725	-55.15	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
4726	-55.21	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
4727	-55.24	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
4728	-55.29	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
4729	-55.29	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
4730	-55.3	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
4731	-55.31	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
4732	-55.32	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
4733	-55.34	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
4734	-55.35	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
4735	-55.35	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
4736	-55.36	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
4737	-55.36	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
4738	-55.37	oe	ccsbBroad304_08481	CEP55	-			
4739	-55.38	oe	ccsbBroad304_02032	TSC22D1	-			
4740	-55.38	oe	ccsbBroad304_02313	ACTR3	-			
4741	-55.39	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
4742	-55.39	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
4743	-55.39	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
4744	-55.4	kd	CGS001-2077	ERF	ETS Transcription Factors			
4745	-55.43	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
4746	-55.44	kd	CGS001-9552	SPAG7	-			
4747	-55.46	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
4748	-55.51	oe	ccsbBroad304_01617	STX4	-			
4749	-55.52	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
4750	-55.53	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
4751	-55.53	kd	CGS001-7771	ZFP112	-			
4752	-55.57	kd	CGS001-182	JAG1	CD molecules			
4753	-55.62	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4754	-55.67	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
4755	-55.67	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
4756	-55.69	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
4757	-55.69	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
4758	-55.71	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
4759	-55.71	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
4760	-55.72	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
4761	-55.76	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
4762	-55.85	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
4763	-55.85	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
4764	-55.86	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
4765	-55.86	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
4766	-55.88	kd	CGS001-3930	LBR	Tudor domain containing			
4767	-55.9	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
4768	-55.94	oe	ccsbBroad304_00171	BNIP3L	-			
4769	-55.97	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
4770	-55.97	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
4771	-55.98	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
4772	-56.01	kd	CGS001-3155	HMGCL	-			
4773	-56.03	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
4774	-56.03	kd	CGS001-6275	S100A4	EF-hand domain containing			
4775	-56.05	oe	ccsbBroad304_00034	AES	-			
4776	-56.05	kd	CGS001-7913	DEK	-			
4777	-56.07	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4778	-56.13	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
4779	-56.14	kd	CGS001-23131	GPATCH8	G patch domain containing			
4780	-56.15	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
4781	-56.17	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
4782	-56.25	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
4783	-56.26	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
4784	-56.26	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
4785	-56.29	kd	CGS001-4795	NFKBIL1	-			
4786	-56.31	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
4787	-56.31	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
4788	-56.36	kd	CGS001-327	APEH	Prolyl oligopeptidase			
4789	-56.37	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
4790	-56.39	oe	ccsbBroad304_00841	IKBKB	IKK family			
4791	-56.4	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
4792	-56.43	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
4793	-56.44	oe	ccsbBroad304_07800	EXOSC8	-			
4794	-56.49	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
4795	-56.52	oe	ccsbBroad304_00183	C1S	Complement system			
4796	-56.54	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
4797	-56.55	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
4798	-56.57	oe	ccsbBroad304_01392	TRIM27	-			
4799	-56.6	kd	CGS001-51734	SEPX1	-			
4800	-56.62	oe	ccsbBroad304_10491	PFKL	-			
4801	-56.63	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
4802	-56.66	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
4803	-56.7	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
4804	-56.75	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
4805	-56.75	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
4806	-56.76	oe	ccsbBroad304_02386	EIF1B	-			
4807	-56.85	cc		Sodium channel blocker	-			
4808	-56.87	kd	CGS001-5361	PLXNA1	Plexins			
4809	-56.92	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
4810	-56.97	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
4811	-56.98	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
4812	-56.98	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
4813	-57.03	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
4814	-57.04	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
4815	-57.04	kd	CGS001-433	ASGR2	C-type lectin domain containing			
4816	-57.15	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4817	-57.17	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
4818	-57.19	kd	CGS001-8870	IER3	-			
4819	-57.2	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
4820	-57.28	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
4821	-57.33	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
4822	-57.42	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4823	-57.42	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4824	-57.44	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
4825	-57.46	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
4826	-57.49	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
4827	-57.5	oe	ccsbBroad304_02864	PRDX5	-			
4828	-57.53	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
4829	-57.54	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
4830	-57.54	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
4831	-57.58	kd	CGS001-3248	HPGD	Prostaglandin synthases			
4832	-57.59	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
4833	-57.64	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
4834	-57.66	kd	CGS001-335	APOA1	Apolipoproteins			
4835	-57.73	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
4836	-57.77	oe	ccsbBroad304_01664	TGFA	-			
4837	-57.78	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
4838	-57.8	oe	ccsbBroad304_07598	PEMT	-			
4839	-57.82	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
4840	-57.82	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
4841	-57.85	kd	CGS001-64121	RRAGC	-			
4842	-57.86	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
4843	-57.87	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
4844	-57.91	kd	CGS001-6611	SMS	-			
4845	-57.92	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
4846	-57.95	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
4847	-57.97	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
4848	-58.03	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
4849	-58.06	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
4850	-58.08	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
4851	-58.08	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
4852	-58.12	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
4853	-58.17	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
4854	-58.24	oe	ccsbBroad304_00501	EMD	-			
4855	-58.24	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4856	-58.29	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
4857	-58.33	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
4858	-58.34	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
4859	-58.36	oe	ccsbBroad304_01371	RALA	-			
4860	-58.36	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
4861	-58.38	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
4862	-58.38	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
4863	-58.39	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4864	-58.4	cc		Toll like receptors LOF	-			
4865	-58.41	oe	ccsbBroad304_07217	AXIN2	-			
4866	-58.43	kd	CGS001-2002	ELK1	ETS Transcription Factors			
4867	-58.44	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
4868	-58.44	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
4869	-58.49	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
4870	-58.5	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
4871	-58.51	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
4872	-58.52	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
4873	-58.52	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
4874	-58.53	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
4875	-58.57	kd	CGS001-54512	EXOSC4	-			
4876	-58.58	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
4877	-58.59	oe	ccsbBroad304_01394	RFX4	-			
4878	-58.61	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
4879	-58.63	oe	ccsbBroad304_00282	CDKN1A	-			
4880	-58.67	kd	CGS001-10652	YKT6	-			
4881	-58.68	kd	CGS001-5253	PHF2	Histone demethylases			
4882	-58.69	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
4883	-58.73	kd	CGS001-2864	FFAR1	Fatty acid receptors			
4884	-58.75	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
4885	-58.75	kd	CGS001-9688	NUP93	-			
4886	-58.81	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4887	-58.83	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
4888	-58.88	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
4889	-58.96	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
4890	-58.97	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
4891	-58.99	kd	CGS001-85442	KNDC1	-			
4892	-59	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
4893	-59.01	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
4894	-59.08	kd	CGS001-2673	GFPT1	-			
4895	-59.11	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
4896	-59.15	oe	ccsbBroad304_08461	CDCA4	-			
4897	-59.2	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
4898	-59.24	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
4899	-59.32	kd	CGS001-5827	PXMP2	-			
4900	-59.33	cc		Wnt family GOF	-			
4901	-59.37	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
4902	-59.41	oe	ccsbBroad304_02533	NOXA1	-			
4903	-59.41	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
4904	-59.48	kd	CGS001-54505	DHX29	DEAH-boxes			
4905	-59.51	oe	ccsbBroad304_01180	PFKFB3	-			
4906	-59.52	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
4907	-59.53	oe	ccsbBroad304_07727	LIAS	-			
4908	-59.54	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
4909	-59.58	kd	CGS001-55526	DHTKD1	-			
4910	-59.59	oe	ccsbBroad304_06651	NOV	-			
4911	-59.6	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
4912	-59.61	kd	CGS001-51586	MED15	-			
4913	-59.63	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
4914	-59.65	oe	ccsbBroad304_06671	OPA1	-			
4915	-59.67	oe	ccsbBroad304_02838	SDF2L1	-			
4916	-59.73	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
4917	-59.78	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
4918	-59.78	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
4919	-59.85	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
4920	-59.89	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4921	-59.9	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
4922	-59.92	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
4923	-59.94	cc		Dopamine receptor antagonist	-			
4924	-59.95	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
4925	-59.96	oe	ccsbBroad304_13499	KSR2	RAF family			
4926	-60	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
4927	-60.06	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
4928	-60.1	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
4929	-60.11	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
4930	-60.11	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
4931	-60.15	kd	CGS001-2760	GM2A	-			
4932	-60.18	oe	ccsbBroad304_07889	QPRT	-			
4933	-60.19	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
4934	-60.2	kd	CGS001-8575	PRKRA	-			
4935	-60.23	cc		NFkB pathway inhibitor	-			
4936	-60.23	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
4937	-60.27	oe	ccsbBroad304_01131	OXCT1	-			
4938	-60.27	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
4939	-60.39	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
4940	-60.45	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
4941	-60.46	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
4942	-60.48	kd	CGS001-776	CACNA1D	Calcium channel subunits			
4943	-60.53	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
4944	-60.55	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
4945	-60.58	kd	CGS001-23378	RRP8	-			
4946	-60.69	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
4947	-60.71	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
4948	-60.72	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4949	-60.77	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
4950	-60.77	kd	CGS001-83593	RASSF5	-			
4951	-60.8	kd	CGS001-51655	RASD1	-			
4952	-60.81	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
4953	-60.82	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
4954	-60.85	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
4955	-60.86	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
4956	-60.89	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
4957	-60.9	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
4958	-60.91	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
4959	-60.96	kd	CGS001-22930	RAB3GAP1	-			
4960	-60.97	oe	ccsbBroad304_06085	DCK	-			
4961	-60.97	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
4962	-61	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
4963	-61.03	kd	CGS001-1999	ELF3	ETS Transcription Factors			
4964	-61.05	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
4965	-61.06	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
4966	-61.09	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
4967	-61.12	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
4968	-61.13	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
4969	-61.18	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
4970	-61.18	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
4971	-61.19	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
4972	-61.2	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
4973	-61.22	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
4974	-61.24	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
4975	-61.3	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
4976	-61.33	oe	ccsbBroad304_07101	TSC2	-			
4977	-61.35	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
4978	-61.38	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
4979	-61.39	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
4980	-61.44	kd	CGS001-2098	ESD	-			
4981	-61.46	kd	CGS001-8480	RAE1	WD repeat domain containing			
4982	-61.47	oe	ccsbBroad304_02163	MED7	-			
4983	-61.5	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
4984	-61.52	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
4985	-61.62	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
4986	-61.67	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
4987	-61.76	kd	CGS001-55536	CDCA7L	-			
4988	-61.79	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
4989	-61.8	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
4990	-61.84	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
4991	-61.86	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
4992	-61.87	kd	CGS001-3638	INSIG1	-			
4993	-61.92	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
4994	-61.92	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
4995	-61.94	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
4996	-61.95	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
4997	-62	kd	CGS001-826	CAPNS1	EF-hand domain containing			
4998	-62.19	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
4999	-62.2	oe	ccsbBroad304_07491	IP6K1	-			
5000	-62.23	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
5001	-62.27	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
5002	-62.3	oe	ccsbBroad304_00600	FYN	Src family			
5003	-62.31	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
5004	-62.32	oe	ccsbBroad304_00238	CCNE1	-			
5005	-62.36	oe	ccsbBroad304_00564	FGR	Src family			
5006	-62.4	oe	ccsbBroad304_03980	DCLRE1B	-			
5007	-62.4	kd	CGS001-122809	SOCS4	SH2 domain containing			
5008	-62.5	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
5009	-62.51	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
5010	-62.61	oe	ccsbBroad304_10487	BPHL	-			
5011	-62.69	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
5012	-62.71	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
5013	-62.71	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
5014	-62.72	oe	ccsbBroad304_01951	BLZF1	-			
5015	-62.91	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
5016	-63	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
5017	-63.01	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
5018	-63.1	kd	CGS001-8804	CREG1	-			
5019	-63.12	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
5020	-63.14	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
5021	-63.18	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
5022	-63.2	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5023	-63.23	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
5024	-63.23	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
5025	-63.26	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
5026	-63.29	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
5027	-63.3	cc		PKA inhibitor	-			
5028	-63.38	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
5029	-63.39	kd	CGS001-9738	CCP110	-			
5030	-63.44	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
5031	-63.45	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
5032	-63.46	oe	ccsbBroad304_02964	TIMM9	-			
5033	-63.5	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
5034	-63.51	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
5035	-63.55	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
5036	-63.56	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
5037	-63.58	oe	ccsbBroad304_00102	RND3	-			
5038	-63.6	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
5039	-63.66	oe	ccsbBroad304_01748	UFD1L	-			
5040	-63.67	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5041	-63.71	oe	ccsbBroad304_02218	IKBKE	IKK family			
5042	-63.71	kd	CGS001-5618	PRLR	Prolactin receptor family			
5043	-63.71	oe	ccsbBroad304_08797	FASTKD5	-			
5044	-63.72	cp	BRD-K53220666	trimetozine	Sedative			Sedative
5045	-63.73	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
5046	-63.74	oe	ccsbBroad304_00249	CD14	CD molecules			
5047	-63.77	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5048	-63.78	oe	ccsbBroad304_05757	ACADS	-			
5049	-63.78	oe	ccsbBroad304_00883	ISG20	-			
5050	-63.81	kd	CGS001-3560	IL2RB	IL-2 receptor family			
5051	-63.83	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
5052	-63.85	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
5053	-63.85	kd	CGS001-9221	NOLC1	-			
5054	-63.89	oe	ccsbBroad304_00376	CSK	Csk family			
5055	-63.97	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
5056	-64.01	kd	CGS001-54584	GNB1L	WD repeat domain containing			
5057	-64.07	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
5058	-64.09	kd	CGS001-5300	PIN1	-			
5059	-64.1	kd	CGS001-5209	PFKFB3	-			
5060	-64.2	oe	ccsbBroad304_02094	FIBP	-			
5061	-64.24	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
5062	-64.28	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
5063	-64.35	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
5064	-64.38	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
5065	-64.43	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
5066	-64.48	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5067	-64.59	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
5068	-64.6	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
5069	-64.65	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
5070	-64.69	oe	ccsbBroad304_01673	TIMP3	-			
5071	-64.69	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
5072	-64.79	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
5073	-64.87	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
5074	-64.93	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
5075	-64.93	kd	CGS001-23581	CASP14	Caspases			
5076	-65.01	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
5077	-65.04	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
5078	-65.04	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
5079	-65.05	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
5080	-65.1	oe	ccsbBroad304_03961	SMURF2	-			
5081	-65.14	kd	CGS001-124583	CANT1	-			
5082	-65.15	kd	CGS001-84647	PLA2G12B	-			
5083	-65.22	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
5084	-65.26	kd	CGS001-1131	CHRM3	Cholinergic receptors			
5085	-65.27	oe	ccsbBroad304_00239	CCNG1	-			
5086	-65.33	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
5087	-65.36	oe	ccsbBroad304_02018	SUCLA2	-			
5088	-65.36	kd	CGS001-930	CD19	CD molecules			
5089	-65.41	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5090	-65.43	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
5091	-65.46	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
5092	-65.47	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
5093	-65.48	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
5094	-65.5	oe	ccsbBroad304_05528	TICAM2	-			
5095	-65.53	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
5096	-65.58	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
5097	-65.6	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
5098	-65.64	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
5099	-65.67	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
5100	-65.69	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
5101	-65.72	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
5102	-65.73	kd	CGS001-10427	SEC24B	-			
5103	-65.8	kd	CGS001-24148	PRPF6	-			
5104	-65.81	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
5105	-65.85	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
5106	-65.87	oe	ccsbBroad304_06916	SCP2	-			
5107	-65.97	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
5108	-65.98	oe	ccsbBroad304_00690	GRN	-			
5109	-66	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
5110	-66.09	oe	ccsbBroad304_02554	TRAFD1	-			
5111	-66.13	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
5112	-66.18	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
5113	-66.23	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
5114	-66.27	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
5115	-66.32	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
5116	-66.37	kd	CGS001-9380	GRHPR	-			
5117	-66.4	kd	CGS001-4594	MUT	-			
5118	-66.44	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
5119	-66.56	kd	CGS001-4179	CD46	CD molecules			
5120	-66.57	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
5121	-66.59	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
5122	-66.62	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
5123	-66.62	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
5124	-66.65	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
5125	-66.68	kd	CGS001-836	CASP3	Caspases			
5126	-66.76	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
5127	-66.81	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5128	-66.86	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
5129	-66.88	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
5130	-66.89	kd	CGS001-527	ATP6V0C	ATPases / V-type			
5131	-66.93	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
5132	-66.94	kd	CGS001-47	ACLY	-			
5133	-66.97	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
5134	-67.09	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
5135	-67.1	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
5136	-67.11	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
5137	-67.12	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
5138	-67.17	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
5139	-67.27	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
5140	-67.27	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
5141	-67.28	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
5142	-67.34	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
5143	-67.44	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5144	-67.51	kd	CGS001-1662	DDX10	DEAD-boxes			
5145	-67.52	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
5146	-67.52	kd	CGS001-6397	SEC14L1	-			
5147	-67.53	kd	CGS001-5962	RDX	-			
5148	-67.6	oe	ccsbBroad304_06383	HMMR	CD molecules			
5149	-67.64	oe	ccsbBroad304_07662	NPRL2	-			
5150	-67.66	oe	ccsbBroad304_06888	RPN1	-			
5151	-67.69	kd	CGS001-216	ALDH1A1	Aldehyde dehydrogenases			
5152	-67.7	cp	BRD-K65910366	KUC103904N	-666			-666
5153	-67.7	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
5154	-67.71	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
5155	-67.76	kd	CGS001-1196	CLK2	CDC-like kinases			
5156	-67.82	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5157	-67.86	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
5158	-67.89	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
5159	-67.92	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
5160	-67.95	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
5161	-67.97	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
5162	-68.01	kd	CGS001-10538	BATF	basic leucine zipper proteins			
5163	-68.02	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
5164	-68.07	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
5165	-68.08	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
5166	-68.12	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
5167	-68.13	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
5168	-68.15	kd	CGS001-1398	CRK	SH2 domain containing			
5169	-68.16	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
5170	-68.2	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
5171	-68.23	kd	CGS001-955	ENTPD6	-			
5172	-68.24	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
5173	-68.27	kd	CGS001-28960	DCPS	-			
5174	-68.28	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
5175	-68.3	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
5176	-68.33	kd	CGS001-11180	WDR6	WD repeat domain containing			
5177	-68.37	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
5178	-68.37	kd	CGS001-25987	TSKU	-			
5179	-68.41	kd	CGS001-5106	PCK2	-			
5180	-68.47	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
5181	-68.49	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
5182	-68.57	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
5183	-68.57	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
5184	-68.65	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
5185	-68.66	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
5186	-68.74	oe	ccsbBroad304_00993	MDM4	-			
5187	-68.79	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
5188	-68.8	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
5189	-68.84	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
5190	-68.87	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
5191	-68.88	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
5192	-68.9	oe	ccsbBroad304_07411	LPXN	-			
5193	-68.94	kd	CGS001-10285	SMNDC1	Tudor domain containing			
5194	-68.99	kd	CGS001-1399	CRKL	SH2 domain containing			
5195	-69.03	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
5196	-69.05	cc		Bacterial 30S ribosomal subunit inhibitor	-			
5197	-69.06	kd	CGS001-6342	SCP2	-			
5198	-69.08	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
5199	-69.1	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
5200	-69.14	oe	ccsbBroad304_08217	SCCPDH	-			
5201	-69.16	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
5202	-69.19	kd	CGS001-4849	CNOT3	-			
5203	-69.2	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
5204	-69.2	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
5205	-69.21	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
5206	-69.3	oe	ccsbBroad304_01174	PEX13	-			
5207	-69.32	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
5208	-69.33	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
5209	-69.36	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5210	-69.39	oe	ccsbBroad304_06889	RPN2	-			
5211	-69.39	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
5212	-69.4	kd	CGS001-5245	PHB	-			
5213	-69.44	kd	CGS001-1879	EBF1	-			
5214	-69.48	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
5215	-69.49	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
5216	-69.49	oe	ccsbBroad304_02349	MPHOSPH9	-			
5217	-69.54	oe	ccsbBroad304_01379	RBBP6	-			
5218	-69.57	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
5219	-69.59	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
5220	-69.59	kd	CGS001-7486	WRN	-			
5221	-69.63	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
5222	-69.66	kd	CGS001-51741	WWOX	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5223	-69.67	kd	CGS001-11232	POLG2	DNA polymerases			
5224	-69.73	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
5225	-69.76	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
5226	-69.8	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
5227	-69.82	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
5228	-69.86	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
5229	-69.86	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
5230	-69.86	kd	CGS001-7158	TP53BP1	-			
5231	-69.91	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
5232	-69.92	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
5233	-69.96	kd	CGS001-23753	SDF2L1	-			
5234	-69.97	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
5235	-70.06	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
5236	-70.1	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
5237	-70.11	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
5238	-70.15	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
5239	-70.17	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
5240	-70.17	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
5241	-70.17	kd	CGS001-2053	EPHX2	-			
5242	-70.18	kd	CGS001-30001	ERO1L	-			
5243	-70.2	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
5244	-70.26	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
5245	-70.31	cc		Cannabinoid receptor agonist	-			
5246	-70.35	kd	CGS001-3572	IL6ST	IL-6 receptor family			
5247	-70.36	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
5248	-70.37	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
5249	-70.37	kd	CGS001-54884	RETSAT	-			
5250	-70.37	kd	CGS001-54555	DDX49	DEAD-boxes			
5251	-70.38	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
5252	-70.44	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
5253	-70.45	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
5254	-70.5	kd	CGS001-55038	CDCA4	-			
5255	-70.55	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
5256	-70.56	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
5257	-70.58	oe	ccsbBroad304_11405	UBE3C	-			
5258	-70.59	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
5259	-70.61	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
5260	-70.66	oe	ccsbBroad304_10240	CROT	-			
5261	-70.71	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
5262	-70.71	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
5263	-70.75	oe	ccsbBroad304_02373	SPRY2	-			
5264	-70.75	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
5265	-70.75	kd	CGS001-23369	PUM2	-			
5266	-70.79	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
5267	-70.81	oe	ccsbBroad304_00816	IDE	Pitrilysin			
5268	-70.83	oe	ccsbBroad304_06745	PNN	-			
5269	-70.93	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
5270	-70.96	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
5271	-70.98	cc		CCK receptor antagonist	-			
5272	-71	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
5273	-71.05	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
5274	-71.08	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
5275	-71.09	oe	ccsbBroad304_01351	PEX19	-			
5276	-71.09	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
5277	-71.11	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
5278	-71.12	kd	CGS001-1028	CDKN1C	-			
5279	-71.14	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
5280	-71.14	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5281	-71.16	cc		Cell Cycle Inhibition GOF	-			
5282	-71.17	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
5283	-71.2	oe	ccsbBroad304_01034	MSH2	-			
5284	-71.25	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
5285	-71.25	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
5286	-71.25	kd	CGS001-5580	PRKCD	Delta subfamily			
5287	-71.25	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
5288	-71.26	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
5289	-71.34	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
5290	-71.34	kd	CGS001-7485	WRB	-			
5291	-71.36	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
5292	-71.36	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
5293	-71.39	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
5294	-71.39	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
5295	-71.39	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
5296	-71.39	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
5297	-71.43	kd	CGS001-23510	KCTD2	-			
5298	-71.47	kd	CGS001-3176	HNMT	-			
5299	-71.54	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
5300	-71.59	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
5301	-71.59	oe	ccsbBroad304_08392	EXOC6	-			
5302	-71.62	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
5303	-71.64	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
5304	-71.65	oe	ccsbBroad304_06090	DDOST	-			
5305	-71.7	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5306	-71.7	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
5307	-71.72	oe	ccsbBroad304_00518	ETFA	-			
5308	-71.73	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5309	-71.74	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
5310	-71.75	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
5311	-71.77	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
5312	-71.8	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
5313	-71.85	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5314	-71.87	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
5315	-71.9	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
5316	-71.94	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
5317	-71.95	kd	CGS001-7358	UGDH	-			
5318	-71.98	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
5319	-71.99	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
5320	-72.02	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
5321	-72.02	kd	CGS001-5202	PFDN2	-			
5322	-72.04	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
5323	-72.05	oe	ccsbBroad304_07208	NRIP1	-			
5324	-72.05	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
5325	-72.07	kd	CGS001-2781	GNAZ	-			
5326	-72.1	oe	ccsbBroad304_06449	ILF3	-			
5327	-72.1	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5328	-72.14	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
5329	-72.15	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
5330	-72.16	oe	ccsbBroad304_06639	NFYB	-			
5331	-72.16	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
5332	-72.17	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5333	-72.2	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
5334	-72.21	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
5335	-72.23	kd	CGS001-55486	PARL	-			
5336	-72.27	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
5337	-72.31	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
5338	-72.32	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
5339	-72.37	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
5340	-72.39	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
5341	-72.39	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
5342	-72.44	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
5343	-72.49	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
5344	-72.53	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
5345	-72.55	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
5346	-72.56	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
5347	-72.61	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
5348	-72.62	kd	CGS001-11040	PIM2	PIM family			
5349	-72.66	kd	CGS001-1738	DLD	-			
5350	-72.72	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
5351	-72.75	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
5352	-72.79	oe	ccsbBroad304_00963	SMAD5	SMADs			
5353	-72.8	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
5354	-72.83	oe	ccsbBroad304_00155	CCND1	-			
5355	-72.89	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
5356	-73.01	oe	ccsbBroad304_02340	SORBS3	-			
5357	-73.01	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
5358	-73.02	kd	CGS001-3992	FADS1	Fatty acid desaturases			
5359	-73.08	oe	ccsbBroad304_07128	VHL	-			
5360	-73.11	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
5361	-73.11	kd	CGS001-6201	RPS7	S ribosomal proteins			
5362	-73.11	kd	CGS001-149233	IL23R	IL-12 receptor family			
5363	-73.13	kd	CGS001-54957	TXNL4B	-			
5364	-73.16	oe	ccsbBroad304_07071	TKT	-			
5365	-73.17	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
5366	-73.24	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
5367	-73.27	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
5368	-73.3	oe	ccsbBroad304_02484	PAICS	-			
5369	-73.3	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
5370	-73.3	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
5371	-73.34	oe	ccsbBroad304_04257	SPRY4	-			
5372	-73.37	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
5373	-73.37	kd	CGS001-2266	FGG	Endogenous ligands			
5374	-73.38	kd	CGS001-8226	HDHD1	-			
5375	-73.45	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
5376	-73.5	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
5377	-73.52	oe	ccsbBroad304_02249	KIAA0494	-			
5378	-73.53	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
5379	-73.58	kd	CGS001-112858	TP53RK	Bud32 family			
5380	-73.59	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
5381	-73.59	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
5382	-73.6	oe	ccsbBroad304_01183	PGD	-			
5383	-73.61	kd	CGS001-25797	QPCT	Aminopeptidase Y			
5384	-73.67	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
5385	-73.68	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
5386	-73.69	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
5387	-73.7	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
5388	-73.71	kd	CGS001-4925	NUCB2	EF-hand domain containing			
5389	-73.72	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
5390	-73.72	kd	CGS001-7056	THBD	CD molecules			
5391	-73.75	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
5392	-73.76	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5393	-73.78	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
5394	-73.79	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5395	-73.86	kd	CGS001-857	CAV1	-			
5396	-73.91	oe	ccsbBroad304_00161	BID	Endogenous ligands			
5397	-73.94	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
5398	-73.96	kd	CGS001-90861	HN1L	-			
5399	-73.97	oe	ccsbBroad304_01532	SIAH1	-			
5400	-73.97	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
5401	-73.98	kd	CGS001-4833	NME4	-			
5402	-73.99	oe	ccsbBroad304_06144	EFNB3	Ephrins			
5403	-74.02	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
5404	-74.03	oe	ccsbBroad304_07605	LYPLA1	-			
5405	-74.04	kd	CGS001-11319	ECD	-			
5406	-74.06	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
5407	-74.06	kd	CGS001-7054	TH	Amino acid hydroxylases			
5408	-74.08	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
5409	-74.08	oe	ccsbBroad304_07600	NSA2	-			
5410	-74.09	oe	ccsbBroad304_01724	TTR	-			
5411	-74.11	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
5412	-74.14	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
5413	-74.14	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
5414	-74.17	oe	ccsbBroad304_07124	UROD	-			
5415	-74.17	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
5416	-74.17	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
5417	-74.21	kd	CGS001-23242	COBL	-			
5418	-74.23	kd	CGS001-9784	SNX17	Sorting nexins			
5419	-74.24	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
5420	-74.25	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
5421	-74.27	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
5422	-74.32	oe	ccsbBroad304_07220	CDC45	-			
5423	-74.33	kd	CGS001-8667	EIF3H	-			
5424	-74.37	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
5425	-74.37	kd	CGS001-9159	PCSK7	Subtilisin			
5426	-74.39	oe	ccsbBroad304_02276	MVP	-			
5427	-74.39	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
5428	-74.39	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
5429	-74.4	kd	CGS001-1066	CES1	Carboxylesterases			
5430	-74.41	kd	CGS001-8741	TNFSF13	CD molecules			
5431	-74.5	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
5432	-74.5	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
5433	-74.51	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
5434	-74.52	kd	CGS001-22938	SNW1	-			
5435	-74.53	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
5436	-74.54	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
5437	-74.55	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
5438	-74.61	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
5439	-74.64	kd	CGS001-10497	UNC13B	-			
5440	-74.66	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
5441	-74.66	kd	CGS001-10318	TNIP1	-			
5442	-74.69	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
5443	-74.73	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
5444	-74.75	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
5445	-74.76	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
5446	-74.76	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
5447	-74.8	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
5448	-74.8	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
5449	-74.87	oe	ccsbBroad304_00113	ASNS	-			
5450	-74.88	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
5451	-74.9	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
5452	-74.93	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
5453	-74.95	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
5454	-74.97	kd	CGS001-5198	PFAS	-			
5455	-74.98	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
5456	-75.02	kd	CGS001-190	NR0B1	DAX-like receptors			
5457	-75.02	kd	CGS001-10314	LANCL1	-			
5458	-75.03	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
5459	-75.04	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
5460	-75.2	oe	ccsbBroad304_05590	NOTCH2NL	-			
5461	-75.2	oe	ccsbBroad304_06538	LSP1	-			
5462	-75.22	kd	CGS001-151126	ZNF385B	-			
5463	-75.28	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
5464	-75.28	kd	CGS001-4439	MSH5	-			
5465	-75.33	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
5466	-75.38	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
5467	-75.44	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
5468	-75.44	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
5469	-75.45	kd	CGS001-22933	SIRT2	Histone deacetylases			
5470	-75.5	oe	ccsbBroad304_03479	YTHDF1	-			
5471	-75.57	cc		FOS transcription factor family GOF	-			
5472	-75.58	oe	ccsbBroad304_00645	GCLM	-			
5473	-75.58	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5474	-75.63	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
5475	-75.63	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
5476	-75.64	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
5477	-75.64	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
5478	-75.65	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
5479	-75.78	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
5480	-75.8	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
5481	-75.82	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
5482	-75.83	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
5483	-75.84	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
5484	-75.84	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
5485	-75.85	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
5486	-75.88	oe	ccsbBroad304_01769	VEGFB	-			
5487	-75.92	oe	ccsbBroad304_02372	SPRY1	-			
5488	-75.92	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
5489	-75.95	kd	CGS001-5264	PHYH	-			
5490	-75.96	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
5491	-75.99	oe	ccsbBroad304_02569	BTG3	-			
5492	-76.01	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
5493	-76.02	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
5494	-76.14	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
5495	-76.2	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
5496	-76.21	kd	CGS001-10673	TNFSF13B	CD molecules			
5497	-76.26	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5498	-76.27	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
5499	-76.28	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
5500	-76.34	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
5501	-76.34	kd	CGS001-1632	ECI1	-			
5502	-76.36	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
5503	-76.39	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
5504	-76.39	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
5505	-76.44	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
5506	-76.45	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
5507	-76.46	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
5508	-76.47	oe	ccsbBroad304_02789	ADAT1	-			
5509	-76.53	oe	ccsbBroad304_00985	MCL1	-			
5510	-76.53	kd	CGS001-84547	PGBD1	-			
5511	-76.54	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
5512	-76.55	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
5513	-76.57	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
5514	-76.6	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
5515	-76.62	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
5516	-76.64	cc		GATA Zinc finger domain containing LOF	-			
5517	-76.64	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
5518	-76.65	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
5519	-76.67	oe	ccsbBroad304_01658	PRDX2	-			
5520	-76.67	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
5521	-76.68	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
5522	-76.69	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5523	-76.7	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
5524	-76.71	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
5525	-76.74	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5526	-76.76	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
5527	-76.77	kd	CGS001-9871	SEC24D	-			
5528	-76.81	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5529	-76.82	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
5530	-76.83	kd	CGS001-54681	P4HTM	-			
5531	-76.9	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
5532	-76.9	kd	CGS001-6217	RPS16	S ribosomal proteins			
5533	-76.91	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
5534	-76.92	oe	ccsbBroad304_01222	PLP2	-			
5535	-76.98	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
5536	-76.98	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
5537	-76.98	kd	CGS001-23710	GABARAPL1	-			
5538	-76.99	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
5539	-77.02	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
5540	-77.04	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
5541	-77.11	oe	ccsbBroad304_04752	IKBIP	-			
5542	-77.11	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5543	-77.13	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
5544	-77.13	oe	ccsbBroad304_02990	LYPD3	-			
5545	-77.18	cc		Glucocorticoid receptor agonist	-			
5546	-77.18	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
5547	-77.21	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
5548	-77.27	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
5549	-77.27	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
5550	-77.29	oe	ccsbBroad304_05947	CCNC	-			
5551	-77.37	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
5552	-77.37	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
5553	-77.38	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
5554	-77.39	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
5555	-77.43	oe	ccsbBroad304_03386	SPA17	-			
5556	-77.43	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
5557	-77.45	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
5558	-77.49	cc		Nucleophosmin inhibitor	-			
5559	-77.5	oe	ccsbBroad304_00313	TBCB	-			
5560	-77.51	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5561	-77.56	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
5562	-77.59	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
5563	-77.59	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
5564	-77.6	cc		Bacterial DNA gyrase inhibitor	-			
5565	-77.61	oe	ccsbBroad304_00489	EHHADH	-			
5566	-77.69	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
5567	-77.81	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
5568	-77.82	oe	ccsbBroad304_02534	UTP14A	-			
5569	-77.82	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
5570	-77.86	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
5571	-77.88	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
5572	-77.91	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
5573	-77.93	kd	CGS001-1069	CETN2	EF-hand domain containing			
5574	-77.95	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
5575	-77.96	kd	CGS001-55278	QRSL1	-			
5576	-77.99	kd	CGS001-2313	FLI1	ETS Transcription Factors			
5577	-78.08	kd	CGS001-4436	MSH2	-			
5578	-78.1	kd	CGS001-64343	AZI2	-			
5579	-78.14	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
5580	-78.23	oe	ccsbBroad304_01147	PC	Carboxylases			
5581	-78.23	kd	CGS001-27244	SESN1	-			
5582	-78.29	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
5583	-78.3	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
5584	-78.32	oe	ccsbBroad304_02677	PDAP1	-			
5585	-78.36	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
5586	-78.36	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
5587	-78.45	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5588	-78.49	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5589	-78.51	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
5590	-78.55	kd	CGS001-2810	SFN	-			
5591	-78.61	oe	ccsbBroad304_01146	PARN	-			
5592	-78.61	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
5593	-78.64	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
5594	-78.67	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
5595	-78.72	oe	ccsbBroad304_02399	TNIP1	-			
5596	-78.73	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
5597	-78.75	kd	CGS001-11267	SNF8	-			
5598	-78.77	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
5599	-78.78	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
5600	-78.82	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
5601	-78.85	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
5602	-78.85	kd	CGS001-2232	FDXR	-			
5603	-78.85	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
5604	-78.88	kd	CGS001-5479	PPIB	-			
5605	-78.91	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
5606	-78.91	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
5607	-79.01	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
5608	-79.07	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
5609	-79.07	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
5610	-79.08	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5611	-79.1	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
5612	-79.15	kd	CGS001-6009	RHEB	-			
5613	-79.16	oe	ccsbBroad304_00962	SMAD4	SMADs			
5614	-79.19	kd	CGS001-11315	PARK7	Parkinson disease			
5615	-79.21	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
5616	-79.24	oe	ccsbBroad304_06301	GOT2	-			
5617	-79.24	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
5618	-79.24	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5619	-79.26	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
5620	-79.3	kd	CGS001-839	CASP6	Caspases			
5621	-79.33	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
5622	-79.34	kd	CGS001-139135	PASD1	-			
5623	-79.37	oe	ccsbBroad304_01327	PSPH	-			
5624	-79.38	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
5625	-79.45	oe	ccsbBroad304_07197	PDHX	-			
5626	-79.45	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
5627	-79.47	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
5628	-79.5	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
5629	-79.51	cc		Serotonin receptor agonist	-			
5630	-79.51	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
5631	-79.55	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5632	-79.56	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
5633	-79.56	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
5634	-79.57	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
5635	-79.59	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
5636	-79.6	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
5637	-79.61	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
5638	-79.64	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
5639	-79.72	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
5640	-79.73	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
5641	-79.75	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
5642	-79.81	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
5643	-79.82	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
5644	-79.87	kd	CGS001-3985	LIMK2	LIMK subfamily			
5645	-79.89	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
5646	-79.94	oe	ccsbBroad304_00072	ANXA7	Annexins			
5647	-79.97	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
5648	-80.03	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
5649	-80.05	oe	ccsbBroad304_09396	TIRAP	-			
5650	-80.1	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
5651	-80.11	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
5652	-80.13	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
5653	-80.15	oe	ccsbBroad304_02017	PEX11A	-			
5654	-80.15	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
5655	-80.15	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
5656	-80.16	oe	ccsbBroad304_09708	PNLDC1	-			
5657	-80.16	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5658	-80.16	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
5659	-80.17	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
5660	-80.18	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
5661	-80.19	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
5662	-80.24	oe	ccsbBroad304_02676	PHB2	-			
5663	-80.24	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
5664	-80.24	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
5665	-80.25	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
5666	-80.3	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
5667	-80.32	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
5668	-80.4	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
5669	-80.4	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
5670	-80.41	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
5671	-80.46	oe	ccsbBroad304_06777	PRNP	CD molecules			
5672	-80.46	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
5673	-80.49	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
5674	-80.52	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
5675	-80.55	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
5676	-80.6	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
5677	-80.65	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
5678	-80.66	kd	CGS001-694	BTG1	-			
5679	-80.7	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
5680	-80.7	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5681	-80.71	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
5682	-80.75	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
5683	-80.77	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5684	-80.82	oe	ccsbBroad304_00147	BAG1	-			
5685	-80.83	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
5686	-80.85	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
5687	-80.9	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
5688	-80.91	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
5689	-80.92	oe	ccsbBroad304_02415	TUBB3	Tubulins			
5690	-80.93	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
5691	-80.95	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
5692	-80.96	oe	ccsbBroad304_00262	CD59	CD molecules			
5693	-80.96	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
5694	-81.03	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5695	-81.04	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
5696	-81.05	oe	ccsbBroad304_01215	PLAUR	CD molecules			
5697	-81.09	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5698	-81.09	kd	CGS001-3281	HSBP1	-			
5699	-81.12	oe	ccsbBroad304_02243	DLGAP5	-			
5700	-81.17	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
5701	-81.24	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
5702	-81.27	kd	CGS001-50943	FOXP3	Forkhead boxes			
5703	-81.28	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
5704	-81.29	oe	ccsbBroad304_07820	SNW1	-			
5705	-81.33	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
5706	-81.38	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
5707	-81.39	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5708	-81.4	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
5709	-81.43	kd	CGS001-5162	PDHB	-			
5710	-81.45	oe	ccsbBroad304_13598	NRBP2	NRBP family			
5711	-81.48	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
5712	-81.48	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
5713	-81.5	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
5714	-81.51	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
5715	-81.61	cc		AHSP Pathway LOF	-			
5716	-81.72	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
5717	-81.72	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
5718	-81.72	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5719	-81.73	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
5720	-81.74	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
5721	-81.78	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
5722	-81.8	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
5723	-82.01	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
5724	-82.02	oe	ccsbBroad304_02292	BCL2L11	-			
5725	-82.04	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
5726	-82.05	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
5727	-82.07	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
5728	-82.11	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
5729	-82.13	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
5730	-82.13	oe	ccsbBroad304_00009	ACLY	-			
5731	-82.14	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
5732	-82.16	kd	CGS001-54438	GFOD1	-			
5733	-82.2	oe	ccsbBroad304_03746	CDC42SE1	-			
5734	-82.2	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
5735	-82.24	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
5736	-82.24	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
5737	-82.26	oe	ccsbBroad304_01632	SYPL1	-			
5738	-82.3	oe	ccsbBroad304_00329	CLTA	-			
5739	-82.32	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
5740	-82.33	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
5741	-82.34	oe	ccsbBroad304_06133	TOR1A	-			
5742	-82.36	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
5743	-82.38	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
5744	-82.39	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
5745	-82.41	kd	CGS001-5690	PSMB2	Proteasome subunits			
5746	-82.42	cc		Lipocalins GOF	-			
5747	-82.42	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
5748	-82.43	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
5749	-82.43	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5750	-82.48	oe	ccsbBroad304_08993	DHDDS	-			
5751	-82.54	oe	ccsbBroad304_14291	GDPD5	-			
5752	-82.54	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
5753	-82.58	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
5754	-82.58	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
5755	-82.6	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5756	-82.61	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
5757	-82.64	cc		Trace amine receptors LOF	-			
5758	-82.66	kd	CGS001-5881	RAC3	Endogenous ligands			
5759	-82.66	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
5760	-82.67	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
5761	-82.73	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
5762	-82.79	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
5763	-82.81	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5764	-82.86	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
5765	-82.92	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
5766	-82.94	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
5767	-82.95	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
5768	-82.95	kd	CGS001-1201	CLN3	-			
5769	-82.96	kd	CGS001-7077	TIMP2	-			
5770	-82.98	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
5771	-83.1	oe	ccsbBroad304_06525	LIPA	-			
5772	-83.2	oe	ccsbBroad304_02788	PRAME	-			
5773	-83.21	kd	CGS001-124535	HSF5	-			
5774	-83.21	oe	ccsbBroad304_01974	RNASET2	-			
5775	-83.22	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
5776	-83.24	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
5777	-83.24	kd	CGS001-23670	TMEM2	-			
5778	-83.27	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
5779	-83.29	oe	ccsbBroad304_02581	ASCC3	-			
5780	-83.29	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
5781	-83.35	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
5782	-83.46	kd	CGS001-3421	IDH3G	-			
5783	-83.48	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
5784	-83.49	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
5785	-83.51	oe	ccsbBroad304_08137	HOOK2	-			
5786	-83.53	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
5787	-83.57	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
5788	-83.61	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
5789	-83.65	kd	CGS001-1284	COL4A2	Collagens			
5790	-83.69	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
5791	-83.7	cc		DNA dependent protein kinase inhibitor	-			
5792	-83.71	oe	ccsbBroad304_02217	FEZ1	-			
5793	-83.72	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
5794	-83.8	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
5795	-83.8	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
5796	-83.83	kd	CGS001-4089	SMAD4	SMADs			
5797	-83.87	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
5798	-83.87	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
5799	-83.87	kd	CGS001-83933	HDAC10	Histone deacetylases			
5800	-83.91	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
5801	-83.92	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
5802	-83.93	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
5803	-83.95	cp	BRD-K10065684	dantron	Laxative			Laxative
5804	-83.96	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
5805	-83.98	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
5806	-83.99	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
5807	-84	oe	ccsbBroad304_05980	CDKN1B	-			
5808	-84.03	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5809	-84.06	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
5810	-84.13	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
5811	-84.16	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
5812	-84.16	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
5813	-84.2	kd	CGS001-7466	WFS1	-			
5814	-84.25	kd	CGS001-2615	LRRC32	-			
5815	-84.25	kd	CGS001-2821	GPI	-			
5816	-84.28	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
5817	-84.34	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
5818	-84.39	kd	CGS001-7100	TLR5	Toll-like receptor family			
5819	-84.43	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
5820	-84.44	kd	CGS001-2277	FIGF	-			
5821	-84.44	kd	CGS001-10682	EBP	-			
5822	-84.51	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
5823	-84.52	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
5824	-84.53	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
5825	-84.54	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
5826	-84.55	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
5827	-84.57	oe	ccsbBroad304_00462	DR1	-			
5828	-84.57	oe	ccsbBroad304_02173	ATG5	-			
5829	-84.59	oe	ccsbBroad304_05894	BLVRA	-			
5830	-84.61	oe	ccsbBroad304_00956	LYZ	-			
5831	-84.62	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
5832	-84.62	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
5833	-84.64	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
5834	-84.66	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
5835	-84.66	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
5836	-84.68	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
5837	-84.69	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5838	-84.73	kd	CGS001-5914	RARA	Retinoic acid receptors			
5839	-84.74	oe	ccsbBroad304_04294	ATG10	-			
5840	-84.76	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
5841	-84.78	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
5842	-84.84	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
5843	-84.87	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
5844	-84.88	kd	CGS001-10775	POP4	-			
5845	-84.92	cc		General transcription factors group 2 LOF	-			
5846	-84.92	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
5847	-84.93	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
5848	-84.96	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
5849	-84.96	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
5850	-84.97	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
5851	-85.03	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
5852	-85.04	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
5853	-85.04	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
5854	-85.04	kd	CGS001-85480	TSLP	-			
5855	-85.04	kd	CGS001-9813	KIAA0494	-			
5856	-85.06	kd	CGS001-1756	DMD	-			
5857	-85.08	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
5858	-85.12	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
5859	-85.13	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
5860	-85.13	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
5861	-85.13	kd	CGS001-55206	SBNO1	-			
5862	-85.16	oe	ccsbBroad304_00174	BRAF	RAF family			
5863	-85.16	kd	CGS001-6856	SYPL1	-			
5864	-85.19	kd	CGS001-8807	IL18RAP	CD molecules			
5865	-85.3	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
5866	-85.42	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
5867	-85.46	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
5868	-85.49	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
5869	-85.49	oe	ccsbBroad304_06286	GLUL	-			
5870	-85.49	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5871	-85.51	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
5872	-85.52	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
5873	-85.54	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
5874	-85.59	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
5875	-85.59	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
5876	-85.61	oe	ccsbBroad304_08480	PNPO	-			
5877	-85.61	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
5878	-85.62	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
5879	-85.62	kd	CGS001-122618	PLD4	-			
5880	-85.65	kd	CGS001-5257	PHKB	-			
5881	-85.66	kd	CGS001-3269	HRH1	Histamine receptors			
5882	-85.66	kd	CGS001-8536	CAMK1	CAMK1 family			
5883	-85.68	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
5884	-85.74	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
5885	-85.76	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
5886	-85.76	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
5887	-85.79	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
5888	-85.79	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5889	-85.79	kd	CGS001-11329	STK38	NDR family			
5890	-85.83	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
5891	-85.87	kd	CGS001-11041	B3GNT1	-			
5892	-85.88	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
5893	-85.88	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
5894	-85.91	kd	CGS001-6944	VPS72	-			
5895	-85.93	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
5896	-85.94	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
5897	-85.98	kd	CGS001-1854	DUT	-			
5898	-86	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
5899	-86.02	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
5900	-86.06	kd	CGS001-3516	RBPJ	-			
5901	-86.07	kd	CGS001-1287	COL4A5	Collagens			
5902	-86.12	oe	ccsbBroad304_00316	CKS1B	-			
5903	-86.14	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
5904	-86.15	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
5905	-86.15	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
5906	-86.17	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
5907	-86.18	kd	CGS001-54106	TLR9	Toll-like receptor family			
5908	-86.22	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
5909	-86.22	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
5910	-86.25	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
5911	-86.28	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
5912	-86.34	cc		Apolipoproteins LOF	-			
5913	-86.36	kd	CGS001-3895	KTN1	-			
5914	-86.37	cc		HIF activator	-			
5915	-86.39	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
5916	-86.4	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
5917	-86.43	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
5918	-86.45	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
5919	-86.46	cc		S100 calcium binding proteins LOF	-			
5920	-86.46	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
5921	-86.5	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
5922	-86.53	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5923	-86.55	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
5924	-86.55	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
5925	-86.56	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
5926	-86.59	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
5927	-86.63	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
5928	-86.63	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
5929	-86.63	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
5930	-86.65	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
5931	-86.68	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
5932	-86.71	oe	ccsbBroad304_00038	AGL	-			
5933	-86.73	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
5934	-86.75	oe	ccsbBroad304_01105	PNP	-			
5935	-86.76	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
5936	-86.76	kd	CGS001-64333	ARHGAP9	Rho GTPase activating proteins			
5937	-86.79	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
5938	-86.82	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
5939	-86.82	kd	CGS001-375	ARF1	ADP-ribosylation factors			
5940	-86.83	kd	CGS001-3460	IFNGR2	Interferon receptor family			
5941	-86.89	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
5942	-86.9	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
5943	-86.93	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
5944	-86.96	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
5945	-86.96	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
5946	-86.99	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
5947	-87	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
5948	-87	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
5949	-87.02	oe	ccsbBroad304_09756	PAQR7	-			
5950	-87.02	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
5951	-87.05	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
5952	-87.11	kd	CGS001-1445	CSK	Csk family			
5953	-87.15	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
5954	-87.17	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
5955	-87.2	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
5956	-87.21	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
5957	-87.26	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
5958	-87.27	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
5959	-87.32	kd	CGS001-1528	CYB5A	Cytochrome b genes			
5960	-87.36	kd	CGS001-54881	TEX10	-			
5961	-87.37	oe	ccsbBroad304_01038	MSRA	-			
5962	-87.46	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
5963	-87.46	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
5964	-87.51	oe	ccsbBroad304_01663	TFF2	-			
5965	-87.51	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
5966	-87.59	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5967	-87.65	oe	ccsbBroad304_05902	BNIP3	-			
5968	-87.67	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
5969	-87.69	kd	CGS001-3383	ICAM1	CD molecules			
5970	-87.71	oe	ccsbBroad304_03570	QRSL1	-			
5971	-87.74	oe	ccsbBroad304_01948	GAS7	-			
5972	-87.76	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
5973	-87.77	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
5974	-87.79	oe	ccsbBroad304_07119	UGP2	-			
5975	-87.8	kd	CGS001-2767	GNA11	-			
5976	-87.81	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
5977	-87.89	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
5978	-87.89	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
5979	-87.94	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
5980	-87.97	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
5981	-88	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
5982	-88.01	cc		Glycogen synthase kinase inhibitor	-			
5983	-88.06	kd	CGS001-51447	IP6K2	-			
5984	-88.07	kd	CGS001-338	APOB	Apolipoproteins			
5985	-88.11	oe	ccsbBroad304_09954	PTRF	-			
5986	-88.11	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
5987	-88.2	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
5988	-88.23	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
5989	-88.23	kd	CGS001-9200	PTPLA	-			
5990	-88.25	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
5991	-88.26	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
5992	-88.26	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
5993	-88.28	oe	ccsbBroad304_01211	PKM2	-			
5994	-88.28	kd	CGS001-9441	MED26	-			
5995	-88.3	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
5996	-88.31	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
5997	-88.34	kd	CGS001-6184	RPN1	-			
5998	-88.34	kd	CGS001-10491	CRTAP	-			
5999	-88.35	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
6000	-88.36	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
6001	-88.39	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
6002	-88.42	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
6003	-88.49	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
6004	-88.52	kd	CGS001-5684	PSMA3	Proteasome subunits			
6005	-88.58	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
6006	-88.62	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
6007	-88.62	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
6008	-88.64	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
6009	-88.65	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
6010	-88.65	kd	CGS001-6793	STK10	SLK subfamily			
6011	-88.67	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
6012	-88.68	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
6013	-88.69	oe	ccsbBroad304_00931	LCN2	Lipocalins			
6014	-88.7	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
6015	-88.72	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
6016	-88.72	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
6017	-88.76	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
6018	-88.79	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
6019	-88.83	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
6020	-88.83	kd	CGS001-9655	SOCS5	SH2 domain containing			
6021	-88.84	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
6022	-88.85	kd	CGS001-4998	ORC1	ATPases / AAA-type			
6023	-88.91	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
6024	-88.94	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
6025	-88.94	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
6026	-88.96	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
6027	-88.96	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
6028	-88.97	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
6029	-88.98	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
6030	-89	kd	CGS001-1503	CTPS	-			
6031	-89.02	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
6032	-89.02	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
6033	-89.02	kd	CGS001-3672	ITGA1	Integrins			
6034	-89.06	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
6035	-89.13	kd	CGS001-9111	NMI	-			
6036	-89.19	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
6037	-89.23	kd	CGS001-8727	CTNNAL1	Catenins			
6038	-89.25	kd	CGS001-4351	MPI	-			
6039	-89.26	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
6040	-89.26	kd	CGS001-84669	USP32	EF-hand domain containing			
6041	-89.28	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
6042	-89.32	oe	ccsbBroad304_03850	TRIB3	Trbl family			
6043	-89.32	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
6044	-89.32	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
6045	-89.33	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
6046	-89.33	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
6047	-89.36	oe	ccsbBroad304_01347	RAD1	-			
6048	-89.42	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
6049	-89.44	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
6050	-89.47	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
6051	-89.5	oe	ccsbBroad304_01469	RSU1	-			
6052	-89.58	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
6053	-89.58	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
6054	-89.59	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
6055	-89.6	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
6056	-89.6	kd	CGS001-9695	EDEM1	-			
6057	-89.61	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
6058	-89.62	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
6059	-89.66	kd	CGS001-10841	FTCD	-			
6060	-89.67	cc		RAF inhibitor	-			
6061	-89.69	oe	ccsbBroad304_08365	CYCS	-			
6062	-89.72	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
6063	-89.72	kd	CGS001-2966	GTF2H2	General transcription factors			
6064	-89.83	kd	CGS001-65263	PYCRL	-			
6065	-89.86	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
6066	-89.87	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
6067	-89.87	kd	CGS001-1062	CENPE	Kinesins			
6068	-89.89	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
6069	-89.91	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
6070	-89.92	kd	CGS001-23149	FCHO1	-			
6071	-89.95	kd	CGS001-27035	NOX1	-			
6072	-89.96	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
6073	-89.97	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
6074	-89.99	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
6075	-90	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
6076	-90	kd	CGS001-10755	GIPC1	-			
6077	-90.01	kd	CGS001-7083	TK1	-			
6078	-90.01	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
6079	-90.04	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
6080	-90.05	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
6081	-90.07	oe	ccsbBroad304_02405	TFG	-			
6082	-90.08	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
6083	-90.09	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
6084	-90.1	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
6085	-90.1	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
6086	-90.12	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6087	-90.13	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
6088	-90.15	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
6089	-90.18	kd	CGS001-51293	CD320	CD molecules			
6090	-90.25	oe	ccsbBroad304_06435	RBPJ	-			
6091	-90.28	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
6092	-90.3	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
6093	-90.31	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
6094	-90.35	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
6095	-90.41	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
6096	-90.42	kd	CGS001-5019	OXCT1	-			
6097	-90.44	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6098	-90.45	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
6099	-90.45	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6100	-90.48	kd	CGS001-2678	GGT1	CD molecules			
6101	-90.54	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
6102	-90.56	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
6103	-90.56	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
6104	-90.58	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
6105	-90.66	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
6106	-90.69	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6107	-90.7	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
6108	-90.72	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6109	-90.72	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
6110	-90.73	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
6111	-90.75	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
6112	-90.75	kd	CGS001-83999	KREMEN1	-			
6113	-90.78	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
6114	-90.81	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
6115	-90.83	oe	ccsbBroad304_07029	TADA2A	-			
6116	-90.88	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
6117	-90.9	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
6118	-90.93	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
6119	-90.94	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6120	-90.98	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6121	-90.99	kd	CGS001-5292	PIM1	PIM family			
6122	-91	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6123	-91.05	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
6124	-91.06	oe	ccsbBroad304_00394	CTSD	Cathepsins			
6125	-91.07	oe	ccsbBroad304_01960	CASK	CASK family			
6126	-91.08	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
6127	-91.12	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
6128	-91.18	oe	ccsbBroad304_01084	NEU1	-			
6129	-91.19	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
6130	-91.24	oe	ccsbBroad304_03732	NPDC1	-			
6131	-91.27	kd	CGS001-2160	F11	Chymotrypsin			
6132	-91.28	oe	ccsbBroad304_09284	UBE3B	-			
6133	-91.34	kd	CGS001-54498	SMOX	-			
6134	-91.36	kd	CGS001-5362	PLXNA2	Plexins			
6135	-91.38	kd	CGS001-204851	HIPK1	HIPK subfamily			
6136	-91.42	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
6137	-91.45	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
6138	-91.46	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
6139	-91.57	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
6140	-91.59	oe	ccsbBroad304_02138	TRIP10	-			
6141	-91.61	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
6142	-91.64	oe	ccsbBroad304_00389	CTBP1	-			
6143	-91.64	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
6144	-91.65	oe	ccsbBroad304_00832	IFNB1	Interferons			
6145	-91.65	kd	CGS001-2729	GCLC	-			
6146	-91.72	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
6147	-91.75	cc		PRD class homeoboxes and psudogenes LOF	-			
6148	-91.76	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
6149	-91.76	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
6150	-91.77	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
6151	-91.78	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
6152	-91.79	oe	ccsbBroad304_00420	DAP	-			
6153	-91.79	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
6154	-91.79	kd	CGS001-25842	ASF1A	-			
6155	-91.8	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
6156	-91.81	oe	ccsbBroad304_08152	PSAT1	-			
6157	-91.82	kd	CGS001-11019	LIAS	-			
6158	-91.82	kd	CGS001-51053	GMNN	-			
6159	-91.83	kd	CGS001-114785	MBD6	-			
6160	-91.86	kd	CGS001-1152	CKB	-			
6161	-91.87	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
6162	-91.87	kd	CGS001-7165	TPD52L2	-			
6163	-91.87	kd	CGS001-718	C3	Endogenous ligands			
6164	-91.88	kd	CGS001-3569	IL6	Interferons			
6165	-91.89	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
6166	-91.91	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
6167	-91.94	kd	CGS001-51022	GLRX2	-			
6168	-91.96	oe	ccsbBroad304_00490	EIF4EBP1	-			
6169	-91.97	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
6170	-92.08	kd	CGS001-3998	LMAN1	-			
6171	-92.11	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
6172	-92.11	oe	ccsbBroad304_00152	BCAT2	-			
6173	-92.12	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
6174	-92.17	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
6175	-92.17	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
6176	-92.18	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
6177	-92.2	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
6178	-92.21	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
6179	-92.23	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
6180	-92.24	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
6181	-92.27	kd	CGS001-6197	RPS6KA3	RSK subfamily			
6182	-92.3	cc		Minor histocompatibility antigens LOF	-			
6183	-92.31	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
6184	-92.33	kd	CGS001-5565	PRKAB2	AMPK subfamily			
6185	-92.36	kd	CGS001-27097	TAF5L	WD repeat domain containing			
6186	-92.42	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
6187	-92.43	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
6188	-92.44	kd	CGS001-9451	EIF2AK3	PEK subfamily			
6189	-92.47	oe	ccsbBroad304_02840	PISD	Decarboxylases			
6190	-92.48	kd	CGS001-11230	PRAF2	-			
6191	-92.51	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
6192	-92.54	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
6193	-92.55	kd	CGS001-7003	TEAD1	-			
6194	-92.56	oe	ccsbBroad304_07832	XPO7	Exportins			
6195	-92.57	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
6196	-92.58	cc		Estrogen receptor agonist	-			
6197	-92.6	kd	CGS001-9512	PMPCB	-			
6198	-92.61	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
6199	-92.62	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
6200	-92.64	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
6201	-92.7	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
6202	-92.72	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
6203	-92.72	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
6204	-92.77	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
6205	-92.78	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
6206	-92.78	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
6207	-92.78	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
6208	-92.79	cc		Potassium channel activator	-			
6209	-92.81	kd	CGS001-54541	DDIT4	-			
6210	-92.83	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
6211	-92.86	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
6212	-92.87	kd	CGS001-10587	TXNRD2	-			
6213	-92.9	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
6214	-92.91	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
6215	-92.92	oe	ccsbBroad304_00888	ITPK1	-			
6216	-92.92	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
6217	-92.95	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
6218	-92.96	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
6219	-92.98	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
6220	-93	oe	ccsbBroad304_07337	TAF1B	-			
6221	-93	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
6222	-93	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
6223	-93.02	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
6224	-93.04	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
6225	-93.15	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
6226	-93.18	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
6227	-93.21	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
6228	-93.21	kd	CGS001-7079	TIMP4	-			
6229	-93.22	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
6230	-93.26	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
6231	-93.28	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
6232	-93.3	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
6233	-93.32	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
6234	-93.33	kd	CGS001-5160	PDHA1	-			
6235	-93.42	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
6236	-93.43	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
6237	-93.43	kd	CGS001-4046	LSP1	-			
6238	-93.45	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
6239	-93.48	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
6240	-93.49	kd	CGS001-10606	PAICS	-			
6241	-93.49	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
6242	-93.5	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
6243	-93.55	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
6244	-93.56	kd	CGS001-79733	E2F8	-			
6245	-93.57	oe	ccsbBroad304_00398	CTSL2	-			
6246	-93.62	kd	CGS001-5613	PRKX	Protein kinase A			
6247	-93.64	kd	CGS001-10020	GNE	-			
6248	-93.66	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
6249	-93.68	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
6250	-93.68	kd	CGS001-9467	SH3BP5	-			
6251	-93.69	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
6252	-93.69	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
6253	-93.72	kd	CGS001-3046	HBE1	-			
6254	-93.74	kd	CGS001-10943	MSL3	-			
6255	-93.75	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
6256	-93.75	kd	CGS001-3832	KIF11	Kinesins			
6257	-93.75	kd	CGS001-11140	CDC37	-			
6258	-93.76	oe	ccsbBroad304_01584	SPARC	-			
6259	-93.78	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
6260	-93.8	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
6261	-93.8	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
6262	-93.81	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
6263	-93.83	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
6264	-93.83	kd	CGS001-275	AMT	-			
6265	-93.87	oe	ccsbBroad304_04457	TOX2	-			
6266	-93.88	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
6267	-93.89	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
6268	-93.9	kd	CGS001-8780	RIOK3	RIO3 subfamily			
6269	-93.91	oe	ccsbBroad304_02592	KIF2C	Kinesins			
6270	-93.92	oe	ccsbBroad304_07531	TANK	-			
6271	-93.95	oe	ccsbBroad304_01184	PGK1	-			
6272	-93.97	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
6273	-93.99	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6274	-94	kd	CGS001-9637	FEZ2	-			
6275	-94.04	oe	ccsbBroad304_00817	IDH2	-			
6276	-94.04	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
6277	-94.06	oe	ccsbBroad304_02801	CASP14	Caspases			
6278	-94.06	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6279	-94.07	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
6280	-94.08	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
6281	-94.09	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6282	-94.09	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
6283	-94.1	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
6284	-94.1	oe	ccsbBroad304_00491	EIF4EBP2	-			
6285	-94.1	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
6286	-94.1	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
6287	-94.12	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
6288	-94.12	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
6289	-94.13	oe	ccsbBroad304_00226	CAV1	-			
6290	-94.14	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
6291	-94.14	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
6292	-94.15	oe	ccsbBroad304_03122	RHOD	-			
6293	-94.15	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
6294	-94.16	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
6295	-94.17	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
6296	-94.17	kd	CGS001-1493	CTLA4	CD molecules			
6297	-94.19	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
6298	-94.23	kd	CGS001-6696	SPP1	Endogenous ligands			
6299	-94.26	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
6300	-94.26	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
6301	-94.32	oe	ccsbBroad304_02143	CNOT8	-			
6302	-94.33	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
6303	-94.35	oe	ccsbBroad304_09195	MCM8	-			
6304	-94.36	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
6305	-94.36	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
6306	-94.38	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
6307	-94.38	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
6308	-94.39	kd	CGS001-162699	TCEB3C	-			
6309	-94.41	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
6310	-94.45	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
6311	-94.45	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
6312	-94.45	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
6313	-94.49	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
6314	-94.55	kd	CGS001-10765	KDM5B	Histone demethylases			
6315	-94.55	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
6316	-94.58	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
6317	-94.61	kd	CGS001-2896	GRN	-			
6318	-94.61	kd	CGS001-595	CCND1	-			
6319	-94.62	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
6320	-94.64	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
6321	-94.65	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
6322	-94.68	kd	CGS001-126823	KLHDC9	-			
6323	-94.68	oe	ccsbBroad304_06464	ITGB2	Integrins			
6324	-94.74	oe	ccsbBroad304_07145	ZFP161	-			
6325	-94.74	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
6326	-94.76	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
6327	-94.77	oe	ccsbBroad304_08840	KIF9	Kinesins			
6328	-94.79	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
6329	-94.79	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
6330	-94.8	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
6331	-94.85	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
6332	-94.85	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
6333	-94.86	kd	CGS001-637	BID	Endogenous ligands			
6334	-94.88	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
6335	-94.9	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
6336	-94.93	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
6337	-94.97	oe	ccsbBroad304_06862	RGS3	-			
6338	-94.97	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
6339	-95	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6340	-95.06	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
6341	-95.08	oe	ccsbBroad304_02580	TMED10	-			
6342	-95.08	kd	CGS001-10472	ZNF238	-			
6343	-95.16	kd	CGS001-6387	CXCL12	Endogenous ligands			
6344	-95.18	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
6345	-95.18	kd	CGS001-1429	CRYZ	-			
6346	-95.19	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
6347	-95.21	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
6348	-95.21	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
6349	-95.22	oe	ccsbBroad304_00519	ETFB	-			
6350	-95.22	oe	ccsbBroad304_05931	CAPG	-			
6351	-95.22	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
6352	-95.22	kd	CGS001-9710	KIAA0355	-			
6353	-95.22	kd	CGS001-9641	IKBKE	IKK family			
6354	-95.23	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
6355	-95.26	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
6356	-95.27	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6357	-95.28	oe	ccsbBroad304_07724	KDELR2	-			
6358	-95.29	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
6359	-95.33	oe	ccsbBroad304_06066	CTSL1	-			
6360	-95.35	kd	CGS001-843	CASP10	Caspases			
6361	-95.37	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
6362	-95.38	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
6363	-95.38	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
6364	-95.39	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
6365	-95.4	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
6366	-95.41	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
6367	-95.42	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
6368	-95.44	cc		T-type calcium channel blocker	-			
6369	-95.46	kd	CGS001-23244	PDS5A	-			
6370	-95.49	cc		GABA receptor antagonist	-			
6371	-95.5	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
6372	-95.51	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
6373	-95.53	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
6374	-95.57	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
6375	-95.58	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
6376	-95.59	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
6377	-95.6	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
6378	-95.6	kd	CGS001-9687	GREB1	-			
6379	-95.62	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
6380	-95.62	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
6381	-95.63	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
6382	-95.64	oe	ccsbBroad304_00665	GOT1	-			
6383	-95.64	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6384	-95.65	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
6385	-95.67	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6386	-95.68	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
6387	-95.7	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
6388	-95.71	oe	ccsbBroad304_01593	SRP14	-			
6389	-95.71	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
6390	-95.71	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
6391	-95.71	kd	CGS001-4175	MCM6	-			
6392	-95.73	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
6393	-95.73	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
6394	-95.74	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
6395	-95.76	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
6396	-95.77	oe	ccsbBroad304_04190	CCDC92	-			
6397	-95.79	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
6398	-95.8	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
6399	-95.8	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
6400	-95.81	kd	CGS001-533	ATP6V0B	ATPases / V-type			
6401	-95.82	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
6402	-95.84	oe	ccsbBroad304_04406	PLA2G12B	-			
6403	-95.89	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
6404	-95.89	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
6405	-95.9	oe	ccsbBroad304_05038	HORMAD2	-			
6406	-95.91	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
6407	-95.91	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
6408	-95.91	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
6409	-95.92	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
6410	-95.92	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
6411	-95.93	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6412	-95.93	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
6413	-95.96	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
6414	-95.99	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6415	-96.01	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
6416	-96.04	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
6417	-96.04	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
6418	-96.04	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
6419	-96.06	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
6420	-96.1	kd	CGS001-10607	TBL3	WD repeat domain containing			
6421	-96.14	oe	ccsbBroad304_01519	SET	-			
6422	-96.16	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
6423	-96.17	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
6424	-96.19	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
6425	-96.19	kd	CGS001-4199	ME1	-			
6426	-96.2	oe	ccsbBroad304_00112	ASNA1	-			
6427	-96.21	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
6428	-96.24	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
6429	-96.28	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
6430	-96.3	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
6431	-96.32	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
6432	-96.33	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
6433	-96.35	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
6434	-96.37	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
6435	-96.42	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
6436	-96.42	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
6437	-96.42	kd	CGS001-2147	F2	Endogenous ligands			
6438	-96.44	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
6439	-96.46	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
6440	-96.5	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6441	-96.5	kd	CGS001-23743	BHMT2	-			
6442	-96.51	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
6443	-96.51	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
6444	-96.52	cc		Proteasome inhibitor	-			
6445	-96.52	kd	CGS001-5727	PTCH1	-			
6446	-96.54	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
6447	-96.54	kd	CGS001-3265	HRAS	RAS subfamily			
6448	-96.55	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
6449	-96.57	oe	ccsbBroad304_02195	SPAG7	-			
6450	-96.61	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
6451	-96.61	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
6452	-96.63	kd	CGS001-6277	S100A6	EF-hand domain containing			
6453	-96.66	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
6454	-96.67	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
6455	-96.68	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
6456	-96.7	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
6457	-96.72	kd	CGS001-8900	CCNA1	-			
6458	-96.73	kd	CGS001-26511	CHIC2	-			
6459	-96.74	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6460	-96.75	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
6461	-96.75	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
6462	-96.76	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
6463	-96.76	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
6464	-96.8	kd	CGS001-284119	PTRF	-			
6465	-96.8	kd	CGS001-256281	NUDT14	Nudix motif containing			
6466	-96.8	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
6467	-96.81	cc		SMAD family LOF	-			
6468	-96.86	kd	CGS001-2100	ESR2	Estrogen receptors			
6469	-96.9	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
6470	-96.92	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
6471	-96.96	cc		Kruppel like transcription factors LOF	-			
6472	-96.96	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
6473	-96.96	kd	CGS001-2697	GJA1	Ion channels / Gap junction proteins (connexins)			
6474	-96.97	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
6475	-96.98	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
6476	-97	kd	CGS001-84365	MKI67IP	-			
6477	-97.02	kd	CGS001-56882	CDC42SE1	-			
6478	-97.03	kd	CGS001-5387	PMS2P3	-			
6479	-97.03	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
6480	-97.04	oe	ccsbBroad304_08952	E2F8	-			
6481	-97.04	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
6482	-97.05	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
6483	-97.06	oe	ccsbBroad304_06126	TSC22D3	-			
6484	-97.06	oe	ccsbBroad304_06993	SRD5A1	-			
6485	-97.06	oe	ccsbBroad304_08775	SQRDL	-			
6486	-97.06	oe	ccsbBroad304_00624	GCK	Hexokinases			
6487	-97.06	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
6488	-97.06	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
6489	-97.09	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6490	-97.1	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
6491	-97.1	oe	ccsbBroad304_06103	DMD	-			
6492	-97.1	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6493	-97.11	oe	ccsbBroad304_00077	APEX1	-			
6494	-97.11	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
6495	-97.11	kd	CGS001-9183	ZW10	-			
6496	-97.13	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
6497	-97.13	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
6498	-97.14	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6499	-97.15	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
6500	-97.15	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6501	-97.18	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
6502	-97.2	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
6503	-97.21	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
6504	-97.23	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
6505	-97.25	oe	ccsbBroad304_03728	DIABLO	-			
6506	-97.27	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
6507	-97.29	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
6508	-97.29	kd	CGS001-7316	UBC	-			
6509	-97.3	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
6510	-97.3	kd	CGS001-10180	RBM6	G patch domain containing			
6511	-97.34	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
6512	-97.35	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
6513	-97.36	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
6514	-97.37	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
6515	-97.37	oe	ccsbBroad304_01923	UXT	-			
6516	-97.38	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
6517	-97.38	kd	CGS001-29982	NRBF2	-			
6518	-97.4	cc		Phospholipases GOF	-			
6519	-97.43	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
6520	-97.46	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
6521	-97.47	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
6522	-97.49	oe	ccsbBroad304_00115	ASPH	-			
6523	-97.53	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6524	-97.54	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
6525	-97.54	oe	ccsbBroad304_01985	EIF3H	-			
6526	-97.54	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6527	-97.55	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
6528	-97.55	kd	CGS001-2581	GALC	-			
6529	-97.55	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
6530	-97.57	oe	ccsbBroad304_07651	HEXIM1	-			
6531	-97.61	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
6532	-97.61	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
6533	-97.61	kd	CGS001-6195	RPS6KA1	RSK subfamily			
6534	-97.62	kd	CGS001-80212	CCDC92	-			
6535	-97.63	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
6536	-97.64	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
6537	-97.65	cc		V type ATPases LOF	-			
6538	-97.65	oe	ccsbBroad304_03179	BOLA1	-			
6539	-97.66	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
6540	-97.67	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
6541	-97.68	kd	CGS001-10641	NPRL2	-			
6542	-97.73	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
6543	-97.74	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
6544	-97.8	oe	ccsbBroad304_07118	UGDH	-			
6545	-97.8	kd	CGS001-10873	ME3	-			
6546	-97.8	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
6547	-97.81	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
6548	-97.81	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
6549	-97.83	oe	ccsbBroad304_02197	VPS26A	-			
6550	-97.84	kd	CGS001-1831	TSC22D3	-			
6551	-97.88	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
6552	-97.88	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
6553	-97.88	kd	CGS001-4830	NME1	-			
6554	-97.88	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
6555	-97.89	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6556	-97.91	oe	ccsbBroad304_03450	TMED9	-			
6557	-97.91	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
6558	-97.91	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
6559	-97.92	oe	ccsbBroad304_02230	HERPUD1	-			
6560	-97.92	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
6561	-97.95	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
6562	-97.95	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
6563	-97.99	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
6564	-98	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
6565	-98	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
6566	-98.03	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
6567	-98.05	cc		DNA polymerase inhibitor	-			
6568	-98.05	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
6569	-98.07	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
6570	-98.08	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
6571	-98.1	kd	CGS001-3920	LAMP2	CD molecules			
6572	-98.11	cc		PARP inhibitor	-			
6573	-98.12	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
6574	-98.12	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
6575	-98.14	kd	CGS001-55746	NUP133	-			
6576	-98.15	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
6577	-98.15	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
6578	-98.18	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
6579	-98.19	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6580	-98.19	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
6581	-98.2	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
6582	-98.23	kd	CGS001-2274	FHL2	-			
6583	-98.24	kd	CGS001-5824	PEX19	-			
6584	-98.25	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
6585	-98.26	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
6586	-98.27	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
6587	-98.29	kd	CGS001-84619	ZGPAT	G patch domain containing			
6588	-98.31	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
6589	-98.31	kd	CGS001-3163	HMOX2	Haem oxygenase			
6590	-98.34	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6591	-98.35	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
6592	-98.35	kd	CGS001-57019	CIAPIN1	-			
6593	-98.37	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
6594	-98.38	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
6595	-98.38	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
6596	-98.38	kd	CGS001-771	CA12	Carbonic anhydrases			
6597	-98.39	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
6598	-98.4	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
6599	-98.46	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
6600	-98.47	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
6601	-98.48	kd	CGS001-7431	VIM	Intermediate filaments type III			
6602	-98.49	kd	CGS001-55662	HIF1AN	-			
6603	-98.51	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
6604	-98.52	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
6605	-98.53	oe	ccsbBroad304_01862	YEATS4	-			
6606	-98.53	oe	ccsbBroad304_03497	TXNL4B	-			
6607	-98.53	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
6608	-98.53	kd	CGS001-2967	GTF2H3	General transcription factors			
6609	-98.54	cc		Serpin peptidase inhibitors LOF	-			
6610	-98.55	oe	ccsbBroad304_02526	POP4	-			
6611	-98.56	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
6612	-98.58	oe	ccsbBroad304_03951	NARFL	-			
6613	-98.58	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
6614	-98.58	kd	CGS001-54821	ERCC6L	-			
6615	-98.58	kd	CGS001-213	ALB	-			
6616	-98.6	kd	CGS001-6364	CCL20	Chemokine ligands			
6617	-98.61	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
6618	-98.61	oe	ccsbBroad304_00032	ADSL	-			
6619	-98.63	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
6620	-98.64	cc		Ribonucleotide reductase inhibitor	-			
6621	-98.64	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6622	-98.64	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
6623	-98.67	oe	ccsbBroad304_02278	THRAP3	-			
6624	-98.68	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
6625	-98.69	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
6626	-98.7	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6627	-98.72	oe	ccsbBroad304_04170	PANK2	-			
6628	-98.73	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
6629	-98.74	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
6630	-98.74	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
6631	-98.75	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
6632	-98.76	kd	CGS001-93185	IGSF8	CD molecules			
6633	-98.77	oe	ccsbBroad304_01102	NMT1	-			
6634	-98.77	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
6635	-98.78	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
6636	-98.79	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
6637	-98.81	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6638	-98.81	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
6639	-98.81	kd	CGS001-51172	NAGPA	-			
6640	-98.82	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
6641	-98.82	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
6642	-98.83	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
6643	-98.84	oe	ccsbBroad304_07050	TFAP2A	-			
6644	-98.84	oe	ccsbBroad304_07814	SACM1L	-			
6645	-98.84	kd	CGS001-55214	LEPREL1	-			
6646	-98.87	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
6647	-98.89	oe	ccsbBroad304_06836	RAD23B	-			
6648	-98.9	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
6649	-98.91	oe	ccsbBroad304_07275	PSMG1	-			
6650	-98.91	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
6651	-98.91	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
6652	-98.91	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
6653	-98.91	kd	CGS001-79071	ELOVL6	-			
6654	-98.91	kd	CGS001-1504	CTRB1	-			
6655	-98.91	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
6656	-98.92	kd	CGS001-6189	RPS3A	S ribosomal proteins			
6657	-98.94	oe	ccsbBroad304_13952	SHMT2	-			
6658	-98.95	oe	ccsbBroad304_00446	DKC1	-			
6659	-98.95	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
6660	-98.97	kd	CGS001-55163	PNPO	-			
6661	-98.99	oe	ccsbBroad304_03696	C19ORF10	-			
6662	-99	cc		Nucleoporin LOF	-			
6663	-99	cc		Protein synthesis inhibitor	-			
6664	-99	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
6665	-99	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
6666	-99	kd	CGS001-8681	JMJD7-PLA2G4B	-			
6667	-99.01	cp	BRD-A02189320	met-leu-phe	-666			-666
6668	-99.01	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
6669	-99.03	oe	ccsbBroad304_00632	GGCX	Carboxylases			
6670	-99.03	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
6671	-99.03	kd	CGS001-79139	DERL1	-			
6672	-99.04	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
6673	-99.04	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
6674	-99.06	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
6675	-99.07	kd	CGS001-55793	FAM63A	-			
6676	-99.08	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
6677	-99.08	kd	CGS001-23081	KDM4C	Histone demethylases			
6678	-99.09	cc		Cyclins LOF	-			
6679	-99.1	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
6680	-99.1	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
6681	-99.1	kd	CGS001-29915	HCFC2	-			
6682	-99.1	oe	ccsbBroad304_00551	FECH	-			
6683	-99.11	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
6684	-99.12	kd	CGS001-2235	FECH	-			
6685	-99.14	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
6686	-99.16	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
6687	-99.16	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6688	-99.16	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
6689	-99.17	oe	ccsbBroad304_00118	ATIC	-			
6690	-99.17	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
6691	-99.17	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
6692	-99.18	cc		Adenosine receptor agonist	-			
6693	-99.18	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
6694	-99.18	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
6695	-99.19	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
6696	-99.23	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6697	-99.23	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
6698	-99.23	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
6699	-99.24	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
6700	-99.24	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
6701	-99.25	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
6702	-99.25	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
6703	-99.25	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
6704	-99.26	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
6705	-99.29	oe	ccsbBroad304_01662	TFDP2	-			
6706	-99.31	oe	ccsbBroad304_09006	RPF1	-			
6707	-99.31	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
6708	-99.31	kd	CGS001-286380	FOXD4L3	-			
6709	-99.31	kd	CGS001-125965	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
6710	-99.32	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
6711	-99.32	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6712	-99.32	kd	CGS001-4074	M6PR	-			
6713	-99.35	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
6714	-99.35	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
6715	-99.35	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
6716	-99.37	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
6717	-99.37	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
6718	-99.38	kd	CGS001-4782	NFIC	-			
6719	-99.38	kd	CGS001-81533	ITFG1	-			
6720	-99.4	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
6721	-99.4	kd	CGS001-7082	TJP1	-			
6722	-99.41	kd	CGS001-5829	PXN	-			
6723	-99.41	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
6724	-99.42	oe	ccsbBroad304_00184	C2	Complement system			
6725	-99.43	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
6726	-99.44	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
6727	-99.44	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6728	-99.45	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6729	-99.45	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
6730	-99.45	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
6731	-99.45	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
6732	-99.45	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
6733	-99.45	kd	CGS001-5763	PTMS	-			
6734	-99.47	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
6735	-99.47	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
6736	-99.47	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
6737	-99.48	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
6738	-99.48	oe	ccsbBroad304_07592	CEPT1	-			
6739	-99.48	kd	CGS001-847	CAT	-			
6740	-99.48	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
6741	-99.49	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
6742	-99.49	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
6743	-99.5	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
6744	-99.5	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
6745	-99.51	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
6746	-99.51	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
6747	-99.51	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
6748	-99.52	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
6749	-99.52	kd	CGS001-4090	SMAD5	SMADs			
6750	-99.52	kd	CGS001-5688	PSMA7	Proteasome subunits			
6751	-99.53	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
6752	-99.54	oe	ccsbBroad304_00223	CASP9	Caspases			
6753	-99.54	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
6754	-99.54	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
6755	-99.54	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
6756	-99.54	kd	CGS001-2287	FKBP3	-			
6757	-99.55	kd	CGS001-64170	CARD9	-			
6758	-99.56	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6759	-99.56	kd	CGS001-5108	PCM1	-			
6760	-99.56	kd	CGS001-79902	NUP85	-			
6761	-99.57	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
6762	-99.57	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
6763	-99.57	kd	CGS001-114609	TIRAP	-			
6764	-99.57	oe	ccsbBroad304_02605	PAPD7	-			
6765	-99.58	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
6766	-99.58	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
6767	-99.59	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6768	-99.59	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
6769	-99.59	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
6770	-99.6	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
6771	-99.6	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
6772	-99.6	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
6773	-99.6	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
6774	-99.6	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
6775	-99.62	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
6776	-99.62	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
6777	-99.62	kd	CGS001-4602	MYB	-			
6778	-99.62	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
6779	-99.62	kd	CGS001-113451	ADC	-			
6780	-99.63	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
6781	-99.63	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
6782	-99.63	kd	CGS001-842	CASP9	Caspases			
6783	-99.64	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
6784	-99.64	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
6785	-99.65	oe	ccsbBroad304_02815	SSBP2	-			
6786	-99.65	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
6787	-99.65	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
6788	-99.66	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
6789	-99.67	oe	ccsbBroad304_01556	SMARCB1	-			
6790	-99.67	kd	CGS001-6016	RIT1	-			
6791	-99.68	cc		KCNJ11 modulator	-			
6792	-99.68	oe	ccsbBroad304_06992	SRC	Src family			
6793	-99.68	kd	CGS001-6810	STX4	-			
6794	-99.69	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
6795	-99.69	kd	CGS001-222546	RFX6	-			
6796	-99.71	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6797	-99.71	oe	ccsbBroad304_03658	DCP1A	-			
6798	-99.71	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
6799	-99.71	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
6800	-99.71	kd	CGS001-5686	PSMA5	Proteasome subunits			
6801	-99.72	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
6802	-99.72	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
6803	-99.73	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6804	-99.73	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
6805	-99.73	kd	CGS001-5423	POLB	DNA polymerases			
6806	-99.73	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
6807	-99.73	kd	CGS001-2878	GPX3	-			
6808	-99.73	kd	CGS001-302	ANXA2	Annexins			
6809	-99.73	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
6810	-99.74	kd	CGS001-10898	CPSF4	-			
6811	-99.75	oe	ccsbBroad304_05183	TXLNA	-			
6812	-99.75	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
6813	-99.75	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
6814	-99.75	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
6815	-99.75	kd	CGS001-6193	RPS5	S ribosomal proteins			
6816	-99.75	kd	CGS001-310	ANXA7	Annexins			
6817	-99.75	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
6818	-99.76	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
6819	-99.76	oe	ccsbBroad304_09054	EGFL8	-			
6820	-99.76	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
6821	-99.76	kd	CGS001-840	CASP7	Caspases			
6822	-99.76	kd	CGS001-158	ADSL	-			
6823	-99.77	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
6824	-99.78	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
6825	-99.78	oe	ccsbBroad304_01976	EIF4EBP3	-			
6826	-99.78	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6827	-99.78	kd	CGS001-6599	SMARCC1	-			
6828	-99.78	kd	CGS001-5033	P4HA1	-			
6829	-99.78	kd	CGS001-25	ABL1	Abl family			
6830	-99.79	oe	ccsbBroad304_00529	F3	CD molecules			
6831	-99.79	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
6832	-99.79	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
6833	-99.79	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
6834	-99.79	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
6835	-99.8	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
6836	-99.81	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
6837	-99.81	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
6838	-99.81	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
6839	-99.81	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
6840	-99.82	oe	ccsbBroad304_01165	PDK1	-			
6841	-99.82	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
6842	-99.82	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
6843	-99.82	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
6844	-99.82	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
6845	-99.82	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
6846	-99.82	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
6847	-99.82	kd	CGS001-5255	PHKA1	-			
6848	-99.82	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
6849	-99.84	oe	ccsbBroad304_06494	KLRC1	CD molecules			
6850	-99.84	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
6851	-99.84	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
6852	-99.84	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
6853	-99.85	oe	ccsbBroad304_08878	METTL4	-			
6854	-99.85	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
6855	-99.85	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
6856	-99.85	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6857	-99.86	oe	ccsbBroad304_00179	BTG1	-			
6858	-99.87	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
6859	-99.87	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
6860	-99.88	oe	ccsbBroad304_02402	TMEM5	-			
6861	-99.88	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
6862	-99.88	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
6863	-99.88	oe	ccsbBroad304_05890	BHMT	-			
6864	-99.88	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
6865	-99.88	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
6866	-99.88	kd	CGS001-9	NAT1	-			
6867	-99.88	kd	CGS001-673	BRAF	RAF family			
6868	-99.9	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
6869	-99.9	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
6870	-99.9	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
6871	-99.9	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
6872	-99.91	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
6873	-99.91	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
6874	-99.91	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
6875	-99.91	kd	CGS001-81539	SLC38A1	System A-like transporters			
6876	-99.91	kd	CGS001-5932	RBBP8	-			
6877	-99.91	kd	CGS001-9133	CCNB2	-			
6878	-99.91	kd	CGS001-7840	ALMS1	-			
6879	-99.93	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
6880	-99.93	oe	ccsbBroad304_02271	LPGAT1	-			
6881	-99.93	oe	ccsbBroad304_02414	IRF9	-			
6882	-99.93	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
6883	-99.93	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
6884	-99.93	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6885	-99.93	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
6886	-99.93	kd	CGS001-25885	POLR1A	RNA polymerase subunits			
6887	-99.93	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
6888	-99.93	kd	CGS001-2879	GPX4	-			
6889	-99.93	kd	CGS001-383	ARG1	Arginase			
6890	-99.94	cc		Thromboxane receptor antagonist	-			
6891	-99.94	oe	ccsbBroad304_03420	TOLLIP	-			
6892	-99.94	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
6893	-99.94	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
6894	-99.94	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
6895	-99.94	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
6896	-99.94	oe	ccsbBroad304_03739	NRIP3	-			
6897	-99.94	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
6898	-99.94	oe	ccsbBroad304_03533	CDCA8	-			
6899	-99.94	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
6900	-99.94	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
6901	-99.94	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
6902	-99.94	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
6903	-99.94	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
6904	-99.94	kd	CGS001-9805	SCRN1	-			
6905	-99.94	kd	CGS001-6233	RPS27A	S ribosomal proteins			
6906	-99.94	kd	CGS001-4174	MCM5	-			
6907	-99.94	kd	CGS001-10128	LRPPRC	-			
6908	-99.94	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
6909	-99.96	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
6910	-99.96	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
6911	-99.96	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
6912	-99.96	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
6913	-99.96	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
6914	-99.96	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
6915	-99.96	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
6916	-99.96	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
6917	-99.96	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6918	-99.96	kd	CGS001-55634	ZNF673	-			
6919	-99.96	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
6920	-99.96	kd	CGS001-51014	TMED7	-			
6921	-99.96	kd	CGS001-6194	RPS6	S ribosomal proteins			
6922	-99.96	kd	CGS001-6188	RPS3	S ribosomal proteins			
6923	-99.96	kd	CGS001-6208	RPS14	S ribosomal proteins			
6924	-99.96	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
6925	-99.96	oe	ccsbBroad304_05963	CD44	CD molecules			
6926	-99.97	cc		Ribosomal 40s Subunit LOF	-			
6927	-99.97	cc		Proteasome Pathway LOF	-			
6928	-99.97	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
6929	-99.97	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6930	-99.97	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
6931	-99.97	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
6932	-99.97	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6933	-99.97	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6934	-99.97	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
6935	-99.97	oe	ccsbBroad304_07363	AIFM1	-			
6936	-99.97	oe	ccsbBroad304_07506	UBAP2L	-			
6937	-99.97	oe	ccsbBroad304_01672	TIMP2	-			
6938	-99.97	oe	ccsbBroad304_06845	RARRES3	-			
6939	-99.97	oe	ccsbBroad304_06789	PSEN2	Presenilin			
6940	-99.97	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
6941	-99.97	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
6942	-99.97	oe	ccsbBroad304_03056	MCTS1	-			
6943	-99.97	oe	ccsbBroad304_02370	HRSP12	-			
6944	-99.97	oe	ccsbBroad304_03177	FIS1	-			
6945	-99.97	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
6946	-99.97	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
6947	-99.97	oe	ccsbBroad304_00146	BAD	-			
6948	-99.97	oe	ccsbBroad304_00106	ARRB1	-			
6949	-99.97	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
6950	-99.97	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
6951	-99.97	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
6952	-99.97	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
6953	-99.97	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
6954	-99.97	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
6955	-99.97	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6956	-99.97	kd	CGS001-6464	SHC1	SH2 domain containing			
6957	-99.97	kd	CGS001-7089	TLE2	WD repeat domain containing			
6958	-99.97	kd	CGS001-51750	RTEL1	-			
6959	-99.97	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
6960	-99.97	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
6961	-99.97	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
6962	-99.97	kd	CGS001-4893	NRAS	RAS subfamily			
6963	-99.97	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
6964	-99.97	kd	CGS001-8508	NIPSNAP1	-			
6965	-99.97	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
6966	-99.97	kd	CGS001-1163	CKS1B	-			
6967	-99.97	kd	CGS001-638	BIK	-			
6968	-100	cc		Sirtuins GOF	-			
6969	-100	cc		MCM family LOF	-			
6970	-100	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
6971	-100	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
6972	-100	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
