Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	99.95	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
2	99.95	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
3	99.95	kd	CGS001-9559	VPS26A	-			
4	99.95	kd	CGS001-7371	UCK2	-			
5	99.95	kd	CGS001-9375	TM9SF2	-			
6	99.95	kd	CGS001-8463	TEAD2	-			
7	99.95	kd	CGS001-64094	SMOC2	EF-hand domain containing			
8	99.95	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
9	99.95	kd	CGS001-22937	SCAP	WD repeat domain containing			
10	99.95	kd	CGS001-10921	RNPS1	RNA binding motif (RRM) containing			
11	99.95	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
12	99.95	kd	CGS001-5091	PC	Carboxylases			
13	99.95	kd	CGS001-7181	NR2C1	Testicular receptors			
14	99.95	kd	CGS001-25836	NIPBL	-			
15	99.95	kd	CGS001-3920	LAMP2	CD molecules			
16	99.95	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
17	99.95	kd	CGS001-10247	HRSP12	-			
18	99.95	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
19	99.95	kd	CGS001-2747	GLUD2	-			
20	99.95	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
21	99.95	kd	CGS001-79080	CCDC86	-			
22	99.95	kd	CGS001-51719	CAB39	-			
23	99.95	kd	CGS001-9184	BUB3	WD repeat domain containing			
24	99.95	kd	CGS001-10632	ATP5L	ATPases / F-type			
25	99.92	kd	CGS001-9412	MED21	-			
26	99.92	kd	CGS001-27297	CRCP	-			
27	99.92	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
28	99.92	kd	CGS001-83694	RPS6KL1	RSKL family			
29	99.92	kd	CGS001-5579	PRKCB	Alpha subfamily			
30	99.92	kd	CGS001-4927	NUP88	-			
31	99.92	kd	CGS001-26292	MYCBP	-			
32	99.92	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
33	99.92	kd	CGS001-3251	HPRT1	-			
34	99.92	kd	CGS001-2355	FOSL2	basic leucine zipper proteins			
35	99.92	kd	CGS001-11124	FAF1	UBX domain containing			
36	99.92	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
37	99.92	kd	CGS001-22794	CASC3	-			
38	99.91	oe	ccsbBroad304_00833	IFNG	Interferons			
39	99.91	oe	ccsbBroad304_08322	UFM1	-			
40	99.91	oe	ccsbBroad304_00880	IRF2	-			
41	99.91	oe	ccsbBroad304_00832	IFNB1	Interferons			
42	99.91	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
43	99.91	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
44	99.91	kd	CGS001-118738	ZNF488	Zinc fingers, C2H2-type			
45	99.91	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
46	99.91	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
47	99.91	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
48	99.91	oe	ccsbBroad304_08952	E2F8	-			
49	99.89	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
50	99.89	kd	CGS001-7106	TSPAN4	Tetraspanins			
51	99.89	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
52	99.89	kd	CGS001-56848	SPHK2	Sphingosine kinase			
53	99.89	kd	CGS001-9919	SEC16A	-			
54	99.89	kd	CGS001-10544	PROCR	CD molecules			
55	99.89	kd	CGS001-11188	NISCH	-			
56	99.89	kd	CGS001-4352	MPL	Prolactin receptor family			
57	99.89	kd	CGS001-3329	HSPD1	Heat Shock Proteins / Chaperonins			
58	99.89	kd	CGS001-55715	DOK4	Pleckstrin homology (PH) domain containing			
59	99.89	kd	CGS001-369	ARAF	RAF family			
60	99.89	kd	CGS001-18	ABAT	GABA turnover			
61	99.87	cc		C2 domain containing LOF	-			
62	99.87	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
63	99.87	kd	CGS001-6832	SUPV3L1	-			
64	99.87	kd	CGS001-6817	SULT1A1	Sulfotransferases, cytosolic			
65	99.87	kd	CGS001-5164	PDK2	PDHK family			
66	99.87	kd	CGS001-10651	MTX2	-			
67	99.87	kd	CGS001-81621	KAZALD1	Immunoglobulin superfamily / I-set domain containing			
68	99.87	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
69	99.87	kd	CGS001-2817	GPC1	Proteoglycans / Cell Surface : Glypicans			
70	99.87	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
71	99.87	kd	CGS001-545	ATR	ATR subfamily			
72	99.86	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
73	99.86	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
74	99.86	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
75	99.86	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
76	99.86	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
77	99.86	oe	ccsbBroad304_08797	FASTKD5	-			
78	99.84	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
79	99.84	kd	CGS001-7321	UBE2D1	Ubiquitin-conjugating enzymes E2			
80	99.84	kd	CGS001-6472	SHMT2	-			
81	99.84	kd	CGS001-3364	HUS1	-			
82	99.84	kd	CGS001-10691	GMEB1	-			
83	99.83	cc		IMPDH inhibitor	-			
84	99.82	kd	CGS001-5469	MED1	-			
85	99.82	kd	CGS001-8527	DGKD	Pleckstrin homology (PH) domain containing			
86	99.82	kd	CGS001-10153	CEBPZ	-			
87	99.81	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
88	99.81	oe	ccsbBroad304_05152	SSBP4	-			
89	99.8	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
90	99.79	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
91	99.79	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
92	99.79	kd	CGS001-9134	CCNE2	-			
93	99.79	kd	CGS001-55311	ZNF444	Zinc fingers, C2H2-type			
94	99.79	kd	CGS001-80351	TNKS2	Ankyrin repeat domain containing			
95	99.79	kd	CGS001-3717	JAK2	Janus kinase (JakA) family			
96	99.79	kd	CGS001-3481	IGF2	-			
97	99.79	kd	CGS001-1719	DHFR	Oxidoreductases			
98	99.79	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
99	99.79	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
100	99.77	oe	ccsbBroad304_02195	SPAG7	-			
101	99.77	kd	CGS001-286075	ZNF707	Zinc fingers, C2H2-type			
102	99.77	oe	ccsbBroad304_08553	STAP2	-			
103	99.77	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
104	99.76	kd	CGS001-8467	SMARCA5	-			
105	99.76	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
106	99.76	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
107	99.76	kd	CGS001-4047	LSS	Lanosterol biosynthesis pathway			
108	99.76	kd	CGS001-57406	ABHD6	Abhydrolase domain containing			
109	99.74	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
110	99.74	kd	CGS001-607	BCL9	-			
111	99.72	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
112	99.72	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
113	99.71	kd	CGS001-8848	TSC22D1	-			
114	99.71	kd	CGS001-25898	RCHY1	RING-type (C3HC4) zinc fingers			
115	99.71	kd	CGS001-5921	RASA1	Pleckstrin homology (PH) domain containing			
116	99.71	kd	CGS001-2523	FUT1	Fucosyltransferases			
117	99.68	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
118	99.68	kd	CGS001-25937	WWTR1	Hippo Signaling			
119	99.68	kd	CGS001-51271	UBAP1	-			
120	99.68	kd	CGS001-190	NR0B1	DAX-like receptors			
121	99.68	kd	CGS001-2168	FABP1	Fatty acid-binding proteins			
122	99.68	kd	CGS001-1499	CTNNB1	Catenins			
123	99.67	kd	CGS001-2261	FGFR3	Type V RTKs: FGF (fibroblast growth factor) receptor family			
124	99.66	cc		NFKB Activation GOF	-			
125	99.66	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
126	99.66	kd	CGS001-2786	GNG4	-			
127	99.66	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
128	99.66	kd	CGS001-629	CFB	Complement system			
129	99.66	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
130	99.64	kd	CGS001-8731	RNMT	-			
131	99.63	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
132	99.63	oe	ccsbBroad304_00118	ATIC	-			
133	99.63	kd	CGS001-3397	ID1	Basic helix-loop-helix proteins			
134	99.63	kd	CGS001-164091	PAQR7	-			
135	99.63	kd	CGS001-8318	CDC45	-			
136	99.63	kd	CGS001-25966	C2CD2	-			
137	99.63	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
138	99.63	oe	ccsbBroad304_00954	LYN	Src family			
139	99.61	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
140	99.61	kd	CGS001-10392	NOD1	Nucleotide-binding domain and leucine rich repeat containing			
141	99.61	kd	CGS001-2184	FAH	-			
142	99.61	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
143	99.58	kd	CGS001-51015	ISOC1	-			
144	99.58	kd	CGS001-9451	EIF2AK3	PEK subfamily			
145	99.58	kd	CGS001-55139	ANKZF1	Ankyrin repeat domain containing			
146	99.58	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
147	99.58	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
148	99.55	kd	CGS001-6461	SHB	SH2 domain containing			
149	99.55	kd	CGS001-9133	CCNB2	-			
150	99.55	kd	CGS001-83440	ADPGK	-			
151	99.55	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
152	99.53	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
153	99.53	kd	CGS001-23314	SATB2	Homeoboxes / CUT class			
154	99.53	kd	CGS001-11031	RAB31	RAB, member RAS oncogene			
155	99.53	kd	CGS001-84647	PLA2G12B	-			
156	99.53	kd	CGS001-2615	LRRC32	-			
157	99.52	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
158	99.51	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
159	99.49	cc		C2 domain containing protein kinases LOF	-			
160	99.49	oe	ccsbBroad304_06420	ICAM3	CD molecules			
161	99.48	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
162	99.47	kd	CGS001-7090	TLE3	WD repeat domain containing			
163	99.47	kd	CGS001-51097	SCCPDH	-			
164	99.45	kd	CGS001-28985	MCTS1	-			
165	99.45	kd	CGS001-9650	MTFR1	-			
166	99.44	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
167	99.42	cc		Homeobox Gene GOF	-			
168	99.42	kd	CGS001-5591	PRKDC	Other PIKK family kinases			
169	99.42	kd	CGS001-478	ATP1A3	ATPases / P-type			
170	99.4	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
171	99.4	oe	ccsbBroad304_01651	TCF7L2	-			
172	99.39	oe	ccsbBroad304_00212	CAMLG	-			
173	99.39	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
174	99.39	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
175	99.37	kd	CGS001-162699	TCEB3C	-			
176	99.37	kd	CGS001-84109	QRFPR	GPCR / Class A : RF amide peptide receptors			
177	99.37	kd	CGS001-51203	NUSAP1	-			
178	99.37	kd	CGS001-4190	MDH1	-			
179	99.35	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
180	99.35	oe	ccsbBroad304_01527	SGK1	SGK family			
181	99.35	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
182	99.35	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
183	99.35	oe	ccsbBroad304_07761	CORO1A	Coronins			
184	99.34	kd	CGS001-6675	UAP1	-			
185	99.34	kd	CGS001-55127	HEATR1	-			
186	99.34	kd	CGS001-2936	GSR	Oxidoreductases			
187	99.34	kd	CGS001-9212	AURKB	Aurora kinase			
188	99.32	kd	CGS001-5684	PSMA3	Proteasome subunits			
189	99.32	kd	CGS001-55837	EAPP	-			
190	99.3	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
191	99.3	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
192	99.29	kd	CGS001-83743	GRWD1	WD repeat domain containing			
193	99.26	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
194	99.26	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
195	99.26	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
196	99.26	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
197	99.26	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
198	99.26	kd	CGS001-8649	LAMTOR3	-			
199	99.26	kd	CGS001-8836	GGH	Gamma-glutamyl hydrolase			
200	99.26	kd	CGS001-1490	CTGF	-			
201	99.25	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
202	99.23	kd	CGS001-7727	ZNF174	Zinc fingers, C2H2-type			
203	99.22	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
204	99.21	kd	CGS001-10682	EBP	-			
205	99.21	oe	ccsbBroad304_08605	PBK	TOPK family			
206	99.21	oe	ccsbBroad304_12008	NLK	nmo subfamily			
207	99.19	kd	CGS001-5950	RBP4	Lipocalins			
208	99.19	kd	CGS001-9459	ARHGEF6	Rho guanine nucleotide exchange factors			
209	99.18	kd	CGS001-6652	SORD	-			
210	99.18	kd	CGS001-10589	DRAP1	-			
211	99.17	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
212	99.17	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
213	99.17	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
214	99.16	cc		Aldehyde dehydrogenases LOF	-			
215	99.16	kd	CGS001-9519	TBPL1	-			
216	99.15	cp	BRD-K44779798	miglitol	Glucosidase inhibitor		GAA, MGAM, GANAB, GANC, SLC5A4	Glucosidase inhibitor
217	99.14	kd	CGS001-8678	BECN1	-			
218	99.13	kd	CGS001-7405	UVRAG	-			
219	99.13	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
220	99.13	kd	CGS001-8531	CSDA	-			
221	99.12	kd	CGS001-51160	VPS28	-			
222	99.12	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
223	99.11	kd	CGS001-2852	GPER	-			
224	99.09	kd	CGS001-200081	TXLNA	-			
225	99.08	oe	ccsbBroad304_00032	ADSL	-			
226	99.08	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
227	99.07	cc		Targets of VEGFR inhibitors GOF	-			
228	99.07	oe	ccsbBroad304_02218	IKBKE	IKK family			
229	99.04	kd	CGS001-5357	PLS1	EF-hand domain containing			
230	99.04	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
231	99.03	kd	CGS001-65243	ZNF643	-			
232	99.03	kd	CGS001-2053	EPHX2	-			
233	99.03	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
234	99.01	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
235	99.01	kd	CGS001-51727	CMPK1	-			
236	99.01	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
237	99	kd	CGS001-9455	HOMER2	-			
238	98.98	kd	CGS001-84527	ZNF559	Zinc fingers, C2H2-type			
239	98.98	kd	CGS001-10845	CLPX	ATPases / AAA-type			
240	98.97	kd	CGS001-6259	RYK	Type XV RTKs: RYK			
241	98.97	kd	CGS001-5052	PRDX1	-			
242	98.97	kd	CGS001-55165	CEP55	-			
243	98.97	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
244	98.96	kd	CGS001-6727	SRP14	-			
245	98.95	kd	CGS001-26136	TES	-			
246	98.95	kd	CGS001-4067	LYN	Src family			
247	98.94	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
248	98.94	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
249	98.94	oe	ccsbBroad304_08093	DCPS	-			
250	98.92	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
251	98.92	kd	CGS001-6118	RPA2	-			
252	98.92	kd	CGS001-5355	PLP2	-			
253	98.92	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
254	98.92	kd	CGS001-5594	MAPK1	MAPK:ERK subfamily			
255	98.92	kd	CGS001-826	CAPNS1	EF-hand domain containing			
256	98.92	kd	CGS001-10241	CALCOCO2	-			
257	98.91	kd	CGS001-57215	THAP11	THAP (C2CH-type zinc finger) domain containing			
258	98.9	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
259	98.89	oe	ccsbBroad304_05528	TICAM2	-			
260	98.89	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
261	98.89	kd	CGS001-2683	B4GALT1	Beta 4-glycosyltransferases			
262	98.89	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
263	98.89	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
264	98.88	kd	CGS001-1027	CDKN1B	-			
265	98.87	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
266	98.87	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
267	98.87	kd	CGS001-171017	ZNF384	Zinc fingers, C2H2-type			
268	98.87	kd	CGS001-9891	NUAK1	NuaK subfamily			
269	98.86	oe	ccsbBroad304_00614	GAMT	-			
270	98.84	oe	ccsbBroad304_00420	DAP	-			
271	98.84	oe	ccsbBroad304_09396	TIRAP	-			
272	98.82	kd	CGS001-4144	MAT2A	-			
273	98.82	kd	CGS001-54566	EPB41L4B	-			
274	98.81	kd	CGS001-11073	TOPBP1	-			
275	98.8	oe	ccsbBroad304_07124	UROD	-			
276	98.8	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
277	98.79	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
278	98.78	cc		Mediator complex LOF	-			
279	98.76	cc		Topoisomerase inhibitor	-			
280	98.76	kd	CGS001-3778	KCNMA1	Calcium-activated potassium channels			
281	98.76	kd	CGS001-7184	HSP90B1	Heat shock proteins / HSPC			
282	98.75	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
283	98.74	kd	CGS001-183	AGT	Endogenous ligands			
284	98.73	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
285	98.73	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
286	98.72	kd	CGS001-185	AGTR1	Angiotensin receptors			
287	98.71	oe	ccsbBroad304_04616	ORMDL3	-			
288	98.7	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
289	98.7	kd	CGS001-873	CBR1	Prostaglandin synthases			
290	98.68	kd	CGS001-5660	PSAP	Endogenous ligands			
291	98.68	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
292	98.68	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
293	98.66	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
294	98.66	kd	CGS001-701	BUB1B	Bub family			
295	98.61	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
296	98.61	kd	CGS001-9695	EDEM1	-			
297	98.61	oe	ccsbBroad304_02843	FTSJ1	-			
298	98.59	kd	CGS001-7323	UBE2D3	Ubiquitin-conjugating enzymes E2			
299	98.58	kd	CGS001-6654	SOS1	Rho guanine nucleotide exchange factors			
300	98.58	kd	CGS001-8635	RNASET2	-			
301	98.58	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
302	98.57	kd	CGS001-7915	ALDH5A1	Aldehyde dehydrogenases			
303	98.55	kd	CGS001-6622	SNCA	Parkinson disease			
304	98.53	kd	CGS001-51071	DERA	-			
305	98.52	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
306	98.5	kd	CGS001-837	CASP4	Caspases			
307	98.49	kd	CGS001-546	ATRX	-			
308	98.48	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
309	98.46	kd	CGS001-58533	SNX6	Sorting nexins			
310	98.45	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
311	98.45	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
312	98.45	kd	CGS001-10987	COPS5	-			
313	98.44	kd	CGS001-8767	RIPK2	Receptor interacting protein kinase (RIPK) family			
314	98.43	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
315	98.41	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
316	98.38	kd	CGS001-22889	KIAA0907	-			
317	98.37	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
318	98.36	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
319	98.34	cc		CDK inhibitor	-			
320	98.34	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
321	98.34	kd	CGS001-116519	APOA5	Apolipoproteins			
322	98.34	kd	CGS001-51005	AMDHD2	-			
323	98.34	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
324	98.33	oe	ccsbBroad304_00147	BAG1	-			
325	98.31	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
326	98.3	cc		X linked mental retardation group 2 LOF	-			
327	98.29	oe	ccsbBroad304_06992	SRC	Src family			
328	98.29	kd	CGS001-6241	RRM2	Ribonucleoside-diphosphate reductases			
329	98.29	kd	CGS001-5985	RFC5	ATPases / AAA-type			
330	98.29	kd	CGS001-5693	PSMB5	Proteasome subunits			
331	98.29	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
332	98.28	kd	CGS001-9847	KIAA0528	-			
333	98.27	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
334	98.27	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
335	98.26	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
336	98.24	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
337	98.24	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
338	98.23	oe	ccsbBroad304_06278	GK	Glycerol kinases			
339	98.23	kd	CGS001-7099	TLR4	Toll-like receptor family			
340	98.22	kd	CGS001-6778	STAT6	SH2 domain containing			
341	98.21	kd	CGS001-4680	CEACAM6	CD molecules			
342	98.2	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
343	98.2	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
344	98.2	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
345	98.19	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
346	98.19	oe	ccsbBroad304_05823	ANXA2	Annexins			
347	98.18	kd	CGS001-23635	SSBP2	-			
348	98.18	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
349	98.17	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
350	98.13	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
351	98.13	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
352	98.12	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
353	98.11	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
354	98.07	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
355	98.06	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
356	98.06	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
357	98.06	kd	CGS001-57121	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
358	98.04	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
359	98.03	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
360	98.03	kd	CGS001-4088	SMAD3	SMADs			
361	97.99	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
362	97.96	oe	ccsbBroad304_02345	TXNDC9	-			
363	97.94	kd	CGS001-10608	MXD4	Basic helix-loop-helix proteins			
364	97.94	kd	CGS001-2057	EPOR	Prolactin receptor family			
365	97.92	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
366	97.92	kd	CGS001-9925	ZBTB5	BTB/POZ domain containing			
367	97.92	kd	CGS001-10413	YAP1	Hippo Signaling			
368	97.92	kd	CGS001-1429	CRYZ	-			
369	97.91	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
370	97.89	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
371	97.88	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
372	97.87	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
373	97.87	oe	ccsbBroad304_13939	MOK	RCK family			
374	97.84	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
375	97.84	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
376	97.83	kd	CGS001-3856	KRT8	Intermediate filaments type II, keratins (basic)			
377	97.82	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
378	97.82	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
379	97.8	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
380	97.79	kd	CGS001-10613	ERLIN1	-			
381	97.78	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
382	97.77	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
383	97.76	kd	CGS001-7132	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
384	97.76	kd	CGS001-10135	NAMPT	-			
385	97.75	kd	CGS001-6927	HNF1A	Homeoboxes / HNF class			
386	97.73	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
387	97.73	kd	CGS001-6434	TRA2B	RNA binding motif (RRM) containing			
388	97.69	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
389	97.68	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
390	97.67	kd	CGS001-79258	MMEL1	-			
391	97.65	kd	CGS001-7165	TPD52L2	-			
392	97.64	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
393	97.63	kd	CGS001-22	ABCB7	ATP binding cassette transporters / subfamily B			
394	97.62	kd	CGS001-4849	CNOT3	-			
395	97.61	kd	CGS001-7040	TGFB1	Endogenous ligands			
396	97.61	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
397	97.59	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
398	97.57	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
399	97.54	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
400	97.53	kd	CGS001-192286	HIGD2A	-			
401	97.5	oe	ccsbBroad304_01641	TAF13	-			
402	97.48	kd	CGS001-64080	RBKS	-			
403	97.46	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
404	97.45	kd	CGS001-2690	GHR	Prolactin receptor family			
405	97.43	kd	CGS001-58492	ZNF77	Zinc fingers, C2H2-type			
406	97.42	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
407	97.4	kd	CGS001-604	BCL6	BTB/POZ domain containing			
408	97.39	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
409	97.39	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
410	97.36	kd	CGS001-5727	PTCH1	-			
411	97.36	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
412	97.35	kd	CGS001-1031	CDKN2C	Ankyrin repeat domain containing			
413	97.33	kd	CGS001-55958	KLHL9	BTB/POZ domain containing			
414	97.32	kd	CGS001-2853	GPR31	GPCR / Class A : Orphans			
415	97.32	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
416	97.29	cc		HDAC inhibitor	-			
417	97.29	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
418	97.27	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
419	97.25	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
420	97.22	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
421	97.22	kd	CGS001-64783	RBM15	RNA binding motif (RRM) containing			
422	97.2	oe	ccsbBroad304_06174	ERCC1	-			
423	97.18	oe	ccsbBroad304_02048	BCL10	-			
424	97.18	kd	CGS001-89845	ABCC10	ATP binding cassette transporters / subfamily C			
425	97.15	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
426	97.15	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
427	97.11	kd	CGS001-114785	MBD6	-			
428	97.1	cc		Poly ADP ribose polymerases LOF	-			
429	97.1	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
430	97.08	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
431	97.08	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
432	97.08	kd	CGS001-55206	SBNO1	-			
433	97.06	kd	CGS001-5004	ORM1	Lipocalins			
434	97.05	kd	CGS001-8566	PDXK	-			
435	97.05	kd	CGS001-2356	FPGS	-			
436	97.03	kd	CGS001-8714	ABCC3	ATP binding cassette transporters / subfamily C			
437	97.01	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
438	96.99	oe	ccsbBroad304_02890	SYF2	-			
439	96.99	kd	CGS001-6469	SHH	-			
440	96.98	kd	CGS001-81894	SLC25A28	Miscellaneous SLC25 mitochondrial transporters			
441	96.97	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
442	96.93	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
443	96.92	kd	CGS001-10474	TADA3	-			
444	96.9	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
445	96.88	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
446	96.88	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
447	96.86	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
448	96.85	cp	BRD-A87125127	3-matida	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
449	96.82	oe	ccsbBroad304_06889	RPN2	-			
450	96.82	kd	CGS001-1806	DPYD	-			
451	96.8	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
452	96.79	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
453	96.78	kd	CGS001-642	BLMH	-			
454	96.76	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
455	96.76	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
456	96.74	oe	ccsbBroad304_13998	PDXK	-			
457	96.73	kd	CGS001-5217	PFN2	-			
458	96.72	kd	CGS001-50810	HDGFRP3	-			
459	96.69	cc		Cannabinoid receptor agonist	-			
460	96.69	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
461	96.68	cc		SRC inhibitor	-			
462	96.68	oe	ccsbBroad304_00447	DLD	-			
463	96.68	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
464	96.66	kd	CGS001-85480	TSLP	-			
465	96.65	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
466	96.65	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
467	96.65	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
468	96.63	kd	CGS001-8974	P4HA2	-			
469	96.62	oe	ccsbBroad304_03186	GMNN	-			
470	96.62	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
471	96.62	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
472	96.57	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
473	96.55	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
474	96.53	kd	CGS001-3162	HMOX1	Haem oxygenase			
475	96.52	kd	CGS001-5198	PFAS	-			
476	96.51	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
477	96.5	kd	CGS001-5236	PGM1	-			
478	96.5	kd	CGS001-2230	FDX1	-			
479	96.5	kd	CGS001-51181	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
480	96.48	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
481	96.48	kd	CGS001-161	AP2A2	-			
482	96.48	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
483	96.48	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
484	96.44	oe	ccsbBroad304_10846	GGT1	CD molecules			
485	96.43	cc		Mitogen activated protein kinases LOF	-			
486	96.43	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
487	96.43	kd	CGS001-5934	RBL2	-			
488	96.43	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
489	96.41	kd	CGS001-7534	YWHAZ	-			
490	96.41	kd	CGS001-7267	TTC3	RING-type (C3HC4) zinc fingers			
491	96.36	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
492	96.36	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
493	96.34	cp	BRD-K88701661	dimercaptosuccinic-acid	Chelating agent		DNMT1	Chelating agent
494	96.33	oe	ccsbBroad304_03121	NRBF2	-			
495	96.33	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
496	96.32	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
497	96.31	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
498	96.3	kd	CGS001-29916	SNX11	Sorting nexins			
499	96.29	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
500	96.26	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
501	96.23	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
502	96.23	kd	CGS001-51569	UFM1	-			
503	96.21	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
504	96.2	cc		FLT3 inhibitor	-			
505	96.2	kd	CGS001-4121	MAN1A1	-			
506	96.17	oe	ccsbBroad304_02443	HAX1	-			
507	96.17	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
508	96.14	oe	ccsbBroad304_07861	COBL	-			
509	96.07	cp	BRD-K59456551	methotrexate	Dihydrofolate reductase inhibitor		DHFR, AOX1, FOLR1, TYMS	Dihydrofolate reductase inhibitor
510	96.07	kd	CGS001-116832	RPL39L	L ribosomal proteins			
511	96.05	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
512	96.04	kd	CGS001-205564	SENP5	-			
513	96.03	kd	CGS001-1788	DNMT3A	Methyltransferases			
514	96.03	kd	CGS001-220	ALDH1A3	Aldehyde dehydrogenases			
515	96.02	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
516	96.02	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
517	95.98	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
518	95.94	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
519	95.94	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
520	95.93	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
521	95.91	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
522	95.89	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
523	95.88	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
524	95.87	kd	CGS001-9791	PTDSS1	-			
525	95.87	kd	CGS001-5451	POU2F1	Homeoboxes / POU class			
526	95.87	kd	CGS001-374291	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
527	95.84	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
528	95.83	oe	ccsbBroad304_07834	GGA2	-			
529	95.81	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
530	95.79	oe	ccsbBroad304_10207	ERLIN1	-			
531	95.76	kd	CGS001-10939	AFG3L2	ATPases / AAA-type			
532	95.73	kd	CGS001-57761	TRIB3	Trbl family			
533	95.73	kd	CGS001-9475	ROCK2	Pleckstrin homology (PH) domain containing			
534	95.7	cc		Proteasome Pathway LOF	-			
535	95.7	kd	CGS001-7175	TPR	-			
536	95.69	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
537	95.65	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
538	95.64	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
539	95.64	kd	CGS001-6990	DYNLT3	Cytoplasmic dyneins			
540	95.63	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
541	95.63	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
542	95.63	kd	CGS001-3693	ITGB5	Integrins			
543	95.57	kd	CGS001-9869	SETDB1	Histone methyltransferases (HMTs)			
544	95.54	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
545	95.51	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
546	95.5	kd	CGS001-25874	BRP44	-			
547	95.49	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
548	95.49	kd	CGS001-51684	SUFU	-			
549	95.47	oe	ccsbBroad304_00987	MCM3	-			
550	95.45	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
551	95.43	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
552	95.39	oe	ccsbBroad304_00268	CD81	CD molecules			
553	95.39	kd	CGS001-59343	SENP2	-			
554	95.38	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
555	95.37	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
556	95.33	cc		LIM class homeoboxes GOF	-			
557	95.31	oe	ccsbBroad304_03544	FAIM	-			
558	95.3	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
559	95.29	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
560	95.28	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
561	95.28	kd	CGS001-333929	SNAI3	Snail homologs			
562	95.27	oe	ccsbBroad304_00881	IRF5	-			
563	95.26	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
564	95.24	cp	BRD-K85503079	perospirone	Dopamine receptor antagonist		DRD2, HTR2A, DRD3, DRD4, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
565	95.24	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
566	95.22	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
567	95.21	oe	ccsbBroad304_02676	PHB2	-			
568	95.19	oe	ccsbBroad304_04153	PHF17	-			
569	95.16	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
570	95.15	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
571	95.12	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
572	95.1	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
573	95.09	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
574	95.09	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
575	95.09	oe	ccsbBroad304_01701	TPI1	-			
576	95.07	kd	CGS001-8428	STK24	YSK subfamily			
577	95.07	kd	CGS001-58478	ENOPH1	-			
578	95.05	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
579	95.05	kd	CGS001-56993	TOMM22	-			
580	95.03	cc		IGF-1 inhibitor	-			
581	95	kd	CGS001-718	C3	Endogenous ligands			
582	94.99	kd	CGS001-2581	GALC	-			
583	94.99	kd	CGS001-290	ANPEP	Aminopeptidase N			
584	94.98	kd	CGS001-9898	UBAP2L	-			
585	94.97	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
586	94.87	kd	CGS001-2167	FABP4	Fatty acid binding protein family			
587	94.86	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
588	94.82	oe	ccsbBroad304_00509	EPHX1	-			
589	94.81	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
590	94.79	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
591	94.77	cc		Cyclin dependent kinases LOF	-			
592	94.77	oe	ccsbBroad304_03232	VPS28	-			
593	94.76	kd	CGS001-6678	SPARC	-			
594	94.75	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
595	94.74	kd	CGS001-5327	PLAT	Chymotrypsin			
596	94.72	cp	BRD-K69650333	idarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
597	94.71	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
598	94.69	kd	CGS001-23	ABCF1	ATP binding cassette transporters / subfamily F			
599	94.68	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
600	94.67	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
601	94.66	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
602	94.65	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
603	94.6	kd	CGS001-833	CARS	Aminoacyl tRNA synthetases / Class I			
604	94.54	cp	BRD-K37798499	etoposide	Topoisomerase inhibitor		TOP2A, CYP2E1, CYP3A5, TOP2B	Topoisomerase inhibitor
605	94.53	kd	CGS001-10105	PPIF	-			
606	94.5	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
607	94.49	kd	CGS001-10971	YWHAQ	-			
608	94.49	oe	ccsbBroad304_04891	TMEM174	-			
609	94.48	oe	ccsbBroad304_02373	SPRY2	-			
610	94.48	kd	CGS001-2161	F12	Chymotrypsin			
611	94.46	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
612	94.46	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
613	94.46	kd	CGS001-53836	GPR87	GPCR / Class A : Orphans			
614	94.45	cc		MEK inhibitor	-			
615	94.45	kd	CGS001-4194	MDM4	-			
616	94.42	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
617	94.38	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
618	94.38	kd	CGS001-9587	MAD2L1BP	-			
619	94.37	kd	CGS001-10390	CEPT1	-			
620	94.36	kd	CGS001-23588	KLHDC2	-			
621	94.36	kd	CGS001-353345	GPR141	GPCR / Class A : Orphans			
622	94.33	kd	CGS001-29940	DSE	-			
623	94.27	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
624	94.26	kd	CGS001-8727	CTNNAL1	Catenins			
625	94.24	kd	CGS001-8480	RAE1	WD repeat domain containing			
626	94.22	oe	ccsbBroad304_02589	COPS5	-			
627	94.21	oe	ccsbBroad304_01186	PHB	-			
628	94.17	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
629	94.16	oe	ccsbBroad304_00964	SMAD7	SMADs			
630	94.14	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
631	94.12	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
632	94.12	oe	ccsbBroad304_01271	PPT1	-			
633	94.1	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
634	94.09	kd	CGS001-54957	TXNL4B	-			
635	94.09	kd	CGS001-54498	SMOX	-			
636	94.08	cp	BRD-K70358946	aripiprazole	Serotonin receptor agonist		DRD2, HTR1A, HTR2A, HRH1, HTR1B, HTR1D, HTR2C, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR1E, HTR3A, HTR6, HTR7	Serotonin receptor agonist, Serotonin receptor antagonist
637	94.05	cc		Cyclins LOF	-			
638	94.05	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
639	94.04	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
640	94.03	kd	CGS001-7298	TYMS	Methyltransferases			
641	94.02	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
642	94.01	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
643	93.99	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
644	93.98	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
645	93.96	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
646	93.95	kd	CGS001-3608	ILF2	-			
647	93.93	kd	CGS001-537	ATP6AP1	-			
648	93.92	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
649	93.9	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
650	93.89	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
651	93.88	kd	CGS001-4221	MEN1	-			
652	93.88	kd	CGS001-29880	ALG5	Glycosyltransferase family 2 domain containing			
653	93.87	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
654	93.86	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
655	93.85	kd	CGS001-8525	DGKZ	-			
656	93.85	oe	ccsbBroad304_02857	BAMBI	-			
657	93.81	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
658	93.77	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
659	93.76	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
660	93.76	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
661	93.75	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
662	93.74	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
663	93.7	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
664	93.69	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
665	93.68	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
666	93.68	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
667	93.68	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
668	93.65	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
669	93.65	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
670	93.63	kd	CGS001-10928	RALBP1	-			
671	93.63	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
672	93.61	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
673	93.61	kd	CGS001-1327	COX4I1	Mitochondrial respiratory chain complex			
674	93.59	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
675	93.58	kd	CGS001-9319	TRIP13	ATPases / AAA-type			
676	93.55	cc		Aurora kinase inhibitor	-			
677	93.55	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
678	93.55	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
679	93.55	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
680	93.53	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
681	93.53	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
682	93.52	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
683	93.51	kd	CGS001-2959	GTF2B	General transcription factors			
684	93.49	kd	CGS001-801	CALM1	EF-hand domain containing			
685	93.45	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
686	93.43	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
687	93.41	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
688	93.41	kd	CGS001-10138	YAF2	-			
689	93.4	cp	BRD-A42423104	benproperine	Antitussive			Antitussive
690	93.39	oe	ccsbBroad304_00471	E2F6	-			
691	93.38	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
692	93.34	kd	CGS001-10827	FAM114A2	-			
693	93.3	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
694	93.29	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
695	93.29	kd	CGS001-6196	RPS6KA2	RSK subfamily			
696	93.29	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
697	93.24	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
698	93.21	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
699	93.19	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
700	93.19	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
701	93.13	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
702	93.13	kd	CGS001-1457	CSNK2A1	Casein kinase 2 (CK2) family			
703	93.08	kd	CGS001-8548	BLZF1	-			
704	93.06	cp	BRD-K50866992	tropisetron	Serotonin receptor antagonist		HTR3A, GLRA1, GLRA2, GLRB, HTR4	Serotonin receptor antagonist
705	93.03	oe	ccsbBroad304_00397	CTSK	Cathepsins			
706	92.99	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
707	92.96	kd	CGS001-23386	NUDCD3	-			
708	92.95	kd	CGS001-5899	RALB	-			
709	92.95	kd	CGS001-1879	EBF1	-			
710	92.95	kd	CGS001-55832	CAND1	-			
711	92.91	kd	CGS001-9748	SLK	SLK subfamily			
712	92.86	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
713	92.83	oe	ccsbBroad304_08167	DNTTIP2	-			
714	92.82	kd	CGS001-9380	GRHPR	-			
715	92.8	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
716	92.8	oe	ccsbBroad304_07531	TANK	-			
717	92.79	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
718	92.76	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
719	92.74	kd	CGS001-7004	TEAD4	-			
720	92.74	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
721	92.73	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
722	92.73	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
723	92.72	kd	CGS001-2760	GM2A	-			
724	92.67	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
725	92.66	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
726	92.65	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
727	92.65	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
728	92.65	kd	CGS001-7508	XPC	-			
729	92.65	kd	CGS001-3612	IMPA1	Inositol monophosphatase			
730	92.65	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
731	92.64	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
732	92.61	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
733	92.54	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
734	92.54	kd	CGS001-7105	TSPAN6	Tetraspanins			
735	92.53	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
736	92.5	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
737	92.49	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
738	92.49	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
739	92.48	kd	CGS001-375318	AQP12A	Ion channels / Aquaporins			
740	92.47	kd	CGS001-27035	NOX1	-			
741	92.46	kd	CGS001-9807	IP6K1	-			
742	92.43	kd	CGS001-206358	SLC36A1	SLC36 family of proton-coupled amino acid transporters			
743	92.43	kd	CGS001-842	CASP9	Caspases			
744	92.42	kd	CGS001-399664	MEX3D	Mex-3 homologs			
745	92.4	kd	CGS001-29079	MED4	-			
746	92.39	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
747	92.38	kd	CGS001-8900	CCNA1	-			
748	92.35	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
749	92.34	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
750	92.33	kd	CGS001-79143	MBOAT7	-			
751	92.31	kd	CGS001-7292	TNFSF4	CD molecules			
752	92.3	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
753	92.25	kd	CGS001-2109	ETFB	-			
754	92.22	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
755	92.2	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
756	92.07	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
757	92.06	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
758	92.06	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
759	92.04	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
760	92.03	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
761	92.03	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
762	92.02	kd	CGS001-1022	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
763	92.01	kd	CGS001-55654	TMEM127	-			
764	92.01	kd	CGS001-2288	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
765	92	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
766	91.98	oe	ccsbBroad304_00865	ILF2	-			
767	91.96	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
768	91.92	kd	CGS001-9221	NOLC1	-			
769	91.9	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
770	91.9	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
771	91.9	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
772	91.9	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
773	91.85	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
774	91.82	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
775	91.79	kd	CGS001-55011	PIH1D1	-			
776	91.79	oe	ccsbBroad304_00564	FGR	Src family			
777	91.75	kd	CGS001-468	ATF4	basic leucine zipper proteins			
778	91.73	cp	BRD-K47780086	penciclovir	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor
779	91.71	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
780	91.7	cc		Ubiquitin-specific peptidases LOF	-			
781	91.67	kd	CGS001-10227	MFSD10	-			
782	91.64	oe	ccsbBroad304_01661	TFCP2	-			
783	91.62	kd	CGS001-6884	TAF13	-			
784	91.55	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
785	91.54	kd	CGS001-4485	MST1	-			
786	91.54	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
787	91.52	kd	CGS001-29965	C16ORF5	-			
788	91.52	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
789	91.5	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
790	91.49	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
791	91.46	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
792	91.42	oe	ccsbBroad304_03934	LEPRE1	-			
793	91.42	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
794	91.4	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
795	91.4	oe	ccsbBroad304_03237	LEF1	-			
796	91.38	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
797	91.33	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
798	91.33	oe	ccsbBroad304_03506	AURKAIP1	-			
799	91.28	oe	ccsbBroad304_07097	TRAF1	-			
800	91.25	kd	CGS001-10099	TSPAN3	Tetraspanins			
801	91.24	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
802	91.23	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
803	91.23	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
804	91.2	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
805	91.2	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
806	91.16	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
807	91.16	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
808	91.15	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
809	91.11	kd	CGS001-50813	COPS7A	-			
810	91.1	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
811	91.08	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
812	91.06	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
813	91.01	kd	CGS001-7480	WNT10B	Wingless-type MMTV integration sites			
814	91.01	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
815	91	kd	CGS001-7052	TGM2	Transglutaminases			
816	90.99	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
817	90.97	kd	CGS001-25885	POLR1A	RNA polymerase subunits			
818	90.96	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
819	90.95	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
820	90.94	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
821	90.88	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
822	90.88	kd	CGS001-140612	ZFP28	Zinc fingers, C2H2-type			
823	90.83	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
824	90.82	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
825	90.8	kd	CGS001-89882	TPD52L3	-			
826	90.79	kd	CGS001-5515	PPP2CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
827	90.77	oe	ccsbBroad304_07088	TP53	-			
828	90.77	kd	CGS001-7272	TTK	TTK family			
829	90.76	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
830	90.74	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
831	90.69	oe	ccsbBroad304_01532	SIAH1	-			
832	90.69	oe	ccsbBroad304_02633	LSM6	-			
833	90.64	kd	CGS001-9813	KIAA0494	-			
834	90.6	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
835	90.59	kd	CGS001-598	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
836	90.57	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
837	90.57	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
838	90.57	kd	CGS001-5682	PSMA1	Proteasome subunits			
839	90.56	cp	BRD-K85090592	pilocarpine	Acetylcholine receptor agonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor agonist
840	90.48	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
841	90.47	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
842	90.46	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
843	90.43	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
844	90.42	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
845	90.38	kd	CGS001-1020	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
846	90.37	kd	CGS001-5411	PNN	-			
847	90.37	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
848	90.29	kd	CGS001-5050	PAFAH1B3	-			
849	90.27	kd	CGS001-1844	DUSP2	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
850	90.26	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
851	90.24	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
852	90.22	kd	CGS001-9020	MAP3K14	MAPKKK:STE-unique family			
853	90.2	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
854	90.17	kd	CGS001-25819	CCRN4L	-			
855	90.15	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
856	90.14	kd	CGS001-4151	MB	-			
857	90.13	kd	CGS001-9231	DLG5	-			
858	90.12	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
859	90.12	kd	CGS001-4077	NBR1	-			
860	90.11	kd	CGS001-6258	RXRG	Retinoid X receptors			
861	90.07	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
862	90.07	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
863	90.05	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
864	90.01	kd	CGS001-64428	NARFL	-			
865	89.98	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
866	89.96	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
867	89.92	kd	CGS001-694	BTG1	-			
868	89.89	kd	CGS001-139760	GPR119	GPCR / Class A : Orphans			
869	89.88	kd	CGS001-57521	RPTOR	WD repeat domain containing			
870	89.88	kd	CGS001-5986	RFNG	Beta 3-glycosyltransferases			
871	89.83	cc		Supressors of cytokine signaling GOF	-			
872	89.81	kd	CGS001-10395	DLC1	Rho GTPase activating proteins			
873	89.78	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
874	89.75	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
875	89.74	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
876	89.72	kd	CGS001-4245	MGAT1	-			
877	89.71	kd	CGS001-55604	LRRC16A	-			
878	89.68	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
879	89.63	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
880	89.62	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
881	89.61	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
882	89.61	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
883	89.59	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
884	89.53	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
885	89.46	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
886	89.39	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
887	89.37	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
888	89.32	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
889	89.29	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
890	89.28	kd	CGS001-30836	DNTTIP2	-			
891	89.25	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
892	89.25	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
893	89.24	kd	CGS001-3957	LGALS2	Lectins, galactoside-binding			
894	89.22	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
895	89.21	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
896	89.2	kd	CGS001-2260	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
897	89.19	kd	CGS001-5092	PCBD1	-			
898	89.17	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
899	89.15	kd	CGS001-23464	GCAT	-			
900	89.13	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
901	89.12	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
902	89.1	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
903	89.1	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
904	89.1	kd	CGS001-5710	PSMD4	Proteasome (prosome, macropain) subunits			
905	89.09	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
906	89.09	kd	CGS001-22934	RPIA	-			
907	89.06	oe	ccsbBroad304_02446	TADA3	-			
908	89.02	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
909	88.92	kd	CGS001-7866	IFRD2	-			
910	88.92	oe	ccsbBroad304_07727	LIAS	-			
911	88.91	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
912	88.91	kd	CGS001-7159	TP53BP2	Ankyrin repeat domain containing			
913	88.91	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
914	88.9	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
915	88.83	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
916	88.75	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
917	88.74	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
918	88.74	oe	ccsbBroad304_06837	RAF1	RAF family			
919	88.73	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
920	88.72	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
921	88.69	kd	CGS001-5575	PRKAR1B	Protein kinase A			
922	88.67	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
923	88.62	kd	CGS001-23530	NNT	-			
924	88.61	oe	ccsbBroad304_03089	PACSIN3	-			
925	88.59	kd	CGS001-976	CD97	Adhesion Class GPCRs			
926	88.55	kd	CGS001-2071	ERCC3	General transcription factors			
927	88.53	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
928	88.5	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
929	88.49	kd	CGS001-1155	TBCB	-			
930	88.47	kd	CGS001-3171	FOXA3	Forkhead boxes			
931	88.45	kd	CGS001-6887	TAL2	Basic helix-loop-helix proteins			
932	88.43	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
933	88.4	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
934	88.4	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
935	88.38	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
936	88.38	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
937	88.35	kd	CGS001-5962	RDX	-			
938	88.35	kd	CGS001-5686	PSMA5	Proteasome subunits			
939	88.34	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
940	88.3	kd	CGS001-2787	GNG5	-			
941	88.28	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
942	88.28	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
943	88.26	kd	CGS001-1488	CTBP2	-			
944	88.25	cp	BRD-K84566043	fenpiverinium	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
945	88.23	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
946	88.21	kd	CGS001-2335	FN1	Endogenous ligands			
947	88.2	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
948	88.2	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
949	88.2	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
950	88.19	cc		TGF beta receptor inhibitor	-			
951	88.19	kd	CGS001-3458	IFNG	Interferons			
952	88.18	kd	CGS001-51290	ERGIC2	-			
953	88.15	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
954	88.14	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
955	88.13	kd	CGS001-9903	KLHL21	BTB/POZ domain containing			
956	88.11	kd	CGS001-22954	TRIM32	-			
957	88.08	kd	CGS001-55500	ETNK1	-			
958	88.04	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
959	88.04	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
960	88.03	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
961	88.01	kd	CGS001-10180	RBM6	G patch domain containing			
962	88.01	oe	ccsbBroad304_02738	RRS1	-			
963	87.93	kd	CGS001-678	ZFP36L2	RING-type (C3HC4) zinc fingers			
964	87.92	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
965	87.91	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
966	87.9	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
967	87.9	cp	BRD-A79314293	cephalosporanic-acid	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
968	87.9	kd	CGS001-10412	NSA2	-			
969	87.88	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
970	87.88	kd	CGS001-5744	PTHLH	Endogenous ligands			
971	87.88	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
972	87.88	kd	CGS001-22850	ADNP2	Zinc fingers, C2H2-type			
973	87.81	kd	CGS001-440387	CTRB2	-			
974	87.79	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
975	87.78	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
976	87.78	kd	CGS001-2289	FKBP5	Tetratricopeptide (TTC) repeat domain containing			
977	87.78	kd	CGS001-1874	E2F4	-			
978	87.77	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
979	87.76	kd	CGS001-29982	NRBF2	-			
980	87.76	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
981	87.74	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
982	87.68	kd	CGS001-5160	PDHA1	-			
983	87.65	kd	CGS001-23378	RRP8	-			
984	87.63	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
985	87.59	oe	ccsbBroad304_00794	HSF1	-			
986	87.56	kd	CGS001-5245	PHB	-			
987	87.55	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
988	87.52	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
989	87.49	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
990	87.49	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
991	87.48	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
992	87.48	kd	CGS001-11112	HIBADH	-			
993	87.48	kd	CGS001-79071	ELOVL6	-			
994	87.42	kd	CGS001-1512	CTSH	Cathepsins			
995	87.41	oe	ccsbBroad304_10437	STMN1	-			
996	87.37	kd	CGS001-5583	PRKCH	Eta subfamily			
997	87.36	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
998	87.23	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
999	87.19	kd	CGS001-8435	SOAT2	-			
1000	87.15	kd	CGS001-5888	RAD51	-			
1001	87.12	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
1002	87.12	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
1003	87.1	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
1004	87.09	kd	CGS001-27333	GOLIM4	-			
1005	87.05	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
1006	87.04	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
1007	87.02	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
1008	87.02	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
1009	87.01	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
1010	86.97	kd	CGS001-4931	NVL	ATPases / AAA-type			
1011	86.96	oe	ccsbBroad304_06783	LGMN	Legumain			
1012	86.93	cp	BRD-K96471533	nitazoxanide	Pyruvate ferredoxin oxidoreductase inhibitor			Pyruvate ferredoxin oxidoreductase inhibitor
1013	86.9	kd	CGS001-929	CD14	CD molecules			
1014	86.89	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
1015	86.82	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
1016	86.82	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
1017	86.82	kd	CGS001-995	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1018	86.8	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
1019	86.76	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
1020	86.73	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
1021	86.62	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
1022	86.61	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
1023	86.59	kd	CGS001-3654	IRAK1	Interleukin-1 receptor-associated kinase (IRAK) family			
1024	86.59	kd	CGS001-21	ABCA3	ATP binding cassette transporters / subfamily A			
1025	86.59	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
1026	86.57	kd	CGS001-5689	PSMB1	Proteasome subunits			
1027	86.56	kd	CGS001-140685	ZBTB46	BTB/POZ domain containing			
1028	86.56	kd	CGS001-3800	KIF5C	Kinesins			
1029	86.56	kd	CGS001-2770	GNAI1	-			
1030	86.52	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
1031	86.51	kd	CGS001-111	ADCY5	Adenylate cyclases			
1032	86.49	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
1033	86.49	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
1034	86.47	kd	CGS001-2203	FBP1	-			
1035	86.45	kd	CGS001-1676	DFFA	-			
1036	86.45	kd	CGS001-811	CALR	-			
1037	86.41	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
1038	86.33	oe	ccsbBroad304_01880	LAGE3	-			
1039	86.33	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
1040	86.31	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
1041	86.3	kd	CGS001-7389	UROD	-			
1042	86.28	kd	CGS001-8804	CREG1	-			
1043	86.27	kd	CGS001-5708	PSMD2	Proteasome subunits			
1044	86.27	kd	CGS001-599	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1045	86.22	kd	CGS001-83448	PUS7L	-			
1046	86.22	kd	CGS001-64219	PJA1	RING-type (C3HC4) zinc fingers			
1047	86.2	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
1048	86.16	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
1049	86.14	kd	CGS001-1389	CREBL2	basic leucine zipper proteins			
1050	86.11	kd	CGS001-8536	CAMK1	CAMK1 family			
1051	86.09	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
1052	86.09	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
1053	86.09	kd	CGS001-79073	TMEM109	-			
1054	86.08	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
1055	86.07	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
1056	86.06	kd	CGS001-50846	DHH	-			
1057	86	kd	CGS001-435	ASL	-			
1058	85.99	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
1059	85.98	cp	BRD-K01649396	indatraline	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine transporter inhibitor
1060	85.97	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
1061	85.97	kd	CGS001-486	FXYD2	Ion transport regulator			
1062	85.95	cc		Bacterial 30S ribosomal subunit inhibitor	-			
1063	85.95	kd	CGS001-4143	MAT1A	-			
1064	85.93	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
1065	85.93	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
1066	85.91	kd	CGS001-2101	ESRRA	Estrogen-related receptors			
1067	85.91	oe	ccsbBroad304_01560	SNAPC1	-			
1068	85.9	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1069	85.87	kd	CGS001-23369	PUM2	-			
1070	85.86	oe	ccsbBroad304_00728	HBE1	-			
1071	85.85	kd	CGS001-213	ALB	-			
1072	85.83	oe	ccsbBroad304_07029	TADA2A	-			
1073	85.83	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
1074	85.82	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
1075	85.8	kd	CGS001-2212	FCGR2A	CD molecules			
1076	85.79	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
1077	85.77	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
1078	85.77	oe	ccsbBroad304_02922	TES	-			
1079	85.75	oe	ccsbBroad304_08825	LHPP	-			
1080	85.74	kd	CGS001-10252	SPRY1	-			
1081	85.67	kd	CGS001-4316	MMP7	Matrix metallopeptidase			
1082	85.67	kd	CGS001-83737	ITCH	-			
1083	85.64	kd	CGS001-5645	PRSS2	Serine peptidases			
1084	85.64	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
1085	85.64	kd	CGS001-1983	EIF5	-			
1086	85.58	kd	CGS001-11329	STK38	NDR family			
1087	85.57	cp	BRD-K96134740	kitasamycin	Protein synthesis inhibitor			Protein synthesis inhibitor
1088	85.56	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
1089	85.55	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
1090	85.55	kd	CGS001-9943	OXSR1	FRAY subfamily			
1091	85.55	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
1092	85.53	oe	ccsbBroad304_02497	YKT6	-			
1093	85.5	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
1094	85.48	kd	CGS001-1861	TOR1A	-			
1095	85.48	kd	CGS001-5688	PSMA7	Proteasome subunits			
1096	85.43	kd	CGS001-57222	ERGIC1	-			
1097	85.42	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
1098	85.4	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
1099	85.38	kd	CGS001-7474	WNT5A	Endogenous ligands			
1100	85.38	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
1101	85.36	oe	ccsbBroad304_03080	C16ORF80	-			
1102	85.3	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
1103	85.28	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
1104	85.26	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
1105	85.26	kd	CGS001-7917	BAG6	-			
1106	85.19	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
1107	85.18	oe	ccsbBroad304_00001	NAT1	-			
1108	85.17	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
1109	85.16	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1110	85.16	kd	CGS001-841	CASP8	Caspases			
1111	85.14	kd	CGS001-56731	SLC2A4RG	-			
1112	85.14	kd	CGS001-57680	CHD8	-			
1113	85.13	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
1114	85.12	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
1115	85.05	oe	ccsbBroad304_00690	GRN	-			
1116	85.03	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
1117	85.01	kd	CGS001-10813	UTP14A	-			
1118	84.96	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
1119	84.93	kd	CGS001-10906	TRAFD1	-			
1120	84.93	oe	ccsbBroad304_01102	NMT1	-			
1121	84.9	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
1122	84.89	kd	CGS001-55632	G2E3	Zinc fingers, PHD-type			
1123	84.88	kd	CGS001-8874	ARHGEF7	Rho guanine nucleotide exchange factors			
1124	84.85	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
1125	84.8	kd	CGS001-6253	RTN2	-			
1126	84.8	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
1127	84.78	cp	BRD-K10670311	sulfasalazine	Antirheumatic		PTGS1, PTGS2, ACAT1, ALOX5, CHUK, IKBKB, PLA2G1B, PPARG, SLC46A1, SLC7A11, TBXAS1	Antirheumatic, NFkB pathway inhibitor
1128	84.74	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
1129	84.71	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
1130	84.6	oe	ccsbBroad304_05758	ACADSB	-			
1131	84.59	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
1132	84.59	kd	CGS001-1820	ARID3A	-			
1133	84.56	kd	CGS001-23510	KCTD2	-			
1134	84.54	kd	CGS001-23786	BCL2L13	-			
1135	84.52	kd	CGS001-3476	IGBP1	-			
1136	84.51	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
1137	84.5	oe	ccsbBroad304_02502	GNA13	-			
1138	84.5	kd	CGS001-83933	HDAC10	Histone deacetylases			
1139	84.46	kd	CGS001-2882	GPX7	-			
1140	84.45	kd	CGS001-8864	PER2	-			
1141	84.41	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1142	84.39	cc		T-type calcium channel blocker	-			
1143	84.39	oe	ccsbBroad304_01143	PAFAH1B3	-			
1144	84.36	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
1145	84.33	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
1146	84.33	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
1147	84.32	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
1148	84.32	cp	BRD-K17705806	JTC-801	Opioid receptor antagonist		OPRL1	Opioid receptor antagonist
1149	84.32	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
1150	84.3	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1151	84.29	kd	CGS001-6611	SMS	-			
1152	84.27	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
1153	84.2	oe	ccsbBroad304_13813	ARAF	RAF family			
1154	84.09	kd	CGS001-3418	IDH2	-			
1155	84.07	cc		Imidazoline ligand	-			
1156	84.05	kd	CGS001-1349	COX7B	Mitochondrial respiratory chain complex			
1157	84.04	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
1158	84.03	kd	CGS001-9833	MELK	MELK subfamily			
1159	84.02	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
1160	83.94	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
1161	83.92	kd	CGS001-2037	EPB41L2	-			
1162	83.87	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
1163	83.85	kd	CGS001-10468	FST	-			
1164	83.82	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
1165	83.82	kd	CGS001-3488	IGFBP5	insulin-like growth factor (IGF) binding proteins			
1166	83.79	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
1167	83.76	oe	ccsbBroad304_07923	LSM5	-			
1168	83.69	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
1169	83.66	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
1170	83.65	kd	CGS001-22832	KIAA1009	-			
1171	83.64	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
1172	83.58	kd	CGS001-5336	PLCG2	Phosphoinositide-specific phospholipase C			
1173	83.54	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
1174	83.53	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
1175	83.52	kd	CGS001-7030	TFE3	Basic helix-loop-helix proteins			
1176	83.5	kd	CGS001-80777	CYB5B	-			
1177	83.49	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
1178	83.46	kd	CGS001-2160	F11	Chymotrypsin			
1179	83.41	kd	CGS001-4331	MNAT1	RING-type (C3HC4) zinc fingers			
1180	83.4	kd	CGS001-831	CAST	-			
1181	83.36	kd	CGS001-11319	ECD	-			
1182	83.34	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
1183	83.34	kd	CGS001-6541	SLC7A1	SLC7 family			
1184	83.33	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1185	83.32	kd	CGS001-6776	STAT5A	SH2 domain containing			
1186	83.32	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
1187	83.32	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
1188	83.31	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
1189	83.31	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
1190	83.3	kd	CGS001-10007	GNPDA1	-			
1191	83.28	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
1192	83.26	kd	CGS001-3199	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
1193	83.25	kd	CGS001-5590	PRKCZ	Iota subfamily			
1194	83.24	kd	CGS001-1855	DVL1	Dishevelled homologs			
1195	83.23	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
1196	83.2	kd	CGS001-6364	CCL20	Chemokine ligands			
1197	83.19	kd	CGS001-10681	GNB5	WD repeat domain containing			
1198	83.17	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
1199	83.14	kd	CGS001-7756	ZNF207	Zinc fingers, C2H2-type			
1200	83.1	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
1201	83.04	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
1202	83.03	cc		JAK inhibitor	-			
1203	82.99	kd	CGS001-7024	TFCP2	-			
1204	82.9	kd	CGS001-2099	ESR1	Estrogen receptors			
1205	82.86	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
1206	82.85	kd	CGS001-149233	IL23R	IL-12 receptor family			
1207	82.83	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1208	82.83	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
1209	82.76	kd	CGS001-5359	PLSCR1	-			
1210	82.76	kd	CGS001-10001	MED6	-			
1211	82.76	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
1212	82.73	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
1213	82.72	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
1214	82.69	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
1215	82.68	kd	CGS001-1386	ATF2	basic leucine zipper proteins			
1216	82.66	kd	CGS001-65263	PYCRL	-			
1217	82.66	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
1218	82.64	kd	CGS001-5226	PGD	-			
1219	82.59	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
1220	82.58	kd	CGS001-53340	SPA17	-			
1221	82.54	cc		PKC activator	-			
1222	82.53	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
1223	82.51	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
1224	82.49	oe	ccsbBroad304_01659	TERF1	-			
1225	82.45	kd	CGS001-1356	CP	-			
1226	82.43	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
1227	82.35	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
1228	82.35	oe	ccsbBroad304_06998	SRPK1	SRPK family			
1229	82.32	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
1230	82.31	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
1231	82.31	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1232	82.15	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
1233	82.14	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
1234	82.13	kd	CGS001-1500	CTNND1	Catenins			
1235	82.12	kd	CGS001-8738	CRADD	-			
1236	82.09	kd	CGS001-4671	NAIP	Inhibitors of apoptosis (IAP) protein family			
1237	82.04	kd	CGS001-10670	RRAGA	-			
1238	82.01	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
1239	82.01	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
1240	81.99	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
1241	81.98	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
1242	81.96	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
1243	81.93	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
1244	81.9	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
1245	81.89	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
1246	81.87	kd	CGS001-8192	CLPP	ATPases / AAA-type			
1247	81.82	kd	CGS001-54386	TERF2IP	-			
1248	81.81	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
1249	81.76	oe	ccsbBroad304_13633	PI4KAP2	-			
1250	81.76	kd	CGS001-7251	TSG101	-			
1251	81.76	kd	CGS001-1363	CPE	Carboxypeptidase A			
1252	81.71	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
1253	81.71	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
1254	81.7	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
1255	81.68	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
1256	81.67	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
1257	81.64	kd	CGS001-1978	EIF4EBP1	-			
1258	81.61	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
1259	81.6	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
1260	81.58	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
1261	81.58	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
1262	81.55	kd	CGS001-4781	NFIB	-			
1263	81.52	cc		Rho associated kinase inhibitor	-			
1264	81.51	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
1265	81.5	oe	ccsbBroad304_06133	TOR1A	-			
1266	81.49	kd	CGS001-5654	HTRA1	Serine peptidases / Serine peptidases			
1267	81.48	kd	CGS001-9851	KIAA0753	-			
1268	81.33	kd	CGS001-55818	KDM3A	Histone demethylases			
1269	81.31	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
1270	81.27	oe	ccsbBroad304_00392	CTLA4	CD molecules			
1271	81.26	kd	CGS001-51588	PIAS4	Zinc fingers, MIZ-type			
1272	81.21	kd	CGS001-4351	MPI	-			
1273	81.18	kd	CGS001-595	CCND1	-			
1274	81.13	oe	ccsbBroad304_00282	CDKN1A	-			
1275	81.13	kd	CGS001-10112	KIF20A	Kinesins			
1276	81.05	oe	ccsbBroad304_00738	HINT1	-			
1277	81.05	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
1278	81.05	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
1279	80.98	kd	CGS001-8431	NR0B2	DAX-like receptors			
1280	80.97	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
1281	80.97	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
1282	80.97	kd	CGS001-4522	MTHFD1	-			
1283	80.94	cc		Norepinephrine reuptake inhibitor	-			
1284	80.94	kd	CGS001-10059	DNM1L	-			
1285	80.94	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
1286	80.9	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
1287	80.89	cc		PKC inhibitor	-			
1288	80.88	kd	CGS001-8878	SQSTM1	-			
1289	80.85	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
1290	80.84	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
1291	80.83	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
1292	80.83	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
1293	80.8	oe	ccsbBroad304_00489	EHHADH	-			
1294	80.79	kd	CGS001-10641	NPRL2	-			
1295	80.74	kd	CGS001-9759	HDAC4	Histone deacetylases			
1296	80.61	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
1297	80.59	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
1298	80.53	kd	CGS001-80714	PBX4	Homeoboxes / TALE class			
1299	80.53	kd	CGS001-1659	DHX8	DEAH-boxes			
1300	80.5	kd	CGS001-22908	SACM1L	-			
1301	80.42	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
1302	80.42	kd	CGS001-2869	GRK5	GRK1/3 subfamily			
1303	80.36	kd	CGS001-6446	SGK1	SGK family			
1304	80.36	kd	CGS001-1974	EIF4A2	DEAD-boxes			
1305	80.35	kd	CGS001-4751	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
1306	80.31	kd	CGS001-57026	PDXP	-			
1307	80.27	kd	CGS001-5018	OXA1L	-			
1308	80.27	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
1309	80.24	cp	BRD-A80383043	BRD-A80383043	Glutamate receptor agonist		GRM1, GRM2	Glutamate receptor agonist, Glutamate receptor antagonist
1310	80.2	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
1311	80.19	kd	CGS001-79643	CHMP6	Charged multivesicular body proteins			
1312	80.18	kd	CGS001-2115	ETV1	ETS Transcription Factors			
1313	80.18	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1314	80.15	kd	CGS001-58477	SRPRB	-			
1315	80.14	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1316	80.13	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
1317	80.11	kd	CGS001-4830	NME1	-			
1318	80.11	kd	CGS001-3373	HYAL1	-			
1319	80.07	kd	CGS001-10769	PLK2	Polo-like kinase (PLK) family			
1320	80.06	kd	CGS001-57720	GPR107	GPCR / Unclassified : 7TM orphan receptors			
1321	80.03	kd	CGS001-9014	TAF1B	-			
1322	79.99	oe	ccsbBroad304_08452	PIH1D1	-			
1323	79.96	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
1324	79.92	oe	ccsbBroad304_01304	PSEN1	Presenilin			
1325	79.91	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
1326	79.9	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
1327	79.89	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
1328	79.85	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
1329	79.8	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
1330	79.78	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
1331	79.7	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
1332	79.69	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
1333	79.69	kd	CGS001-338	APOB	Apolipoproteins			
1334	79.68	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1335	79.63	oe	ccsbBroad304_01139	PA2G4	-			
1336	79.62	oe	ccsbBroad304_06301	GOT2	-			
1337	79.6	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
1338	79.59	kd	CGS001-211	ALAS1	-			
1339	79.58	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
1340	79.58	kd	CGS001-7010	TEK	Type XII RTKs: TIE family of angiopoietin receptors			
1341	79.56	oe	ccsbBroad304_02956	EHF	-			
1342	79.54	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1343	79.5	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
1344	79.39	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
1345	79.39	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
1346	79.37	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
1347	79.37	kd	CGS001-8022	LHX3	Homeoboxes / LIM class			
1348	79.34	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
1349	79.27	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1350	79.24	kd	CGS001-29083	GTPBP8	-			
1351	79.17	kd	CGS001-23659	PLA2G15	-			
1352	79.14	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
1353	79.04	oe	ccsbBroad304_07326	EIF2B2	-			
1354	79.04	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
1355	79.04	kd	CGS001-9263	STK17A	Death-associated kinase (DAPK) family			
1356	79.01	kd	CGS001-5588	PRKCQ	Delta subfamily			
1357	79	oe	ccsbBroad304_01699	TPD52L2	-			
1358	78.97	oe	ccsbBroad304_06458	IRF3	-			
1359	78.95	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
1360	78.95	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
1361	78.9	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
1362	78.84	oe	ccsbBroad304_00179	BTG1	-			
1363	78.82	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
1364	78.82	kd	CGS001-2781	GNAZ	-			
1365	78.8	oe	ccsbBroad304_11405	UBE3C	-			
1366	78.78	kd	CGS001-2961	GTF2E2	General transcription factors			
1367	78.7	kd	CGS001-2280	FKBP1A	Cis-trans-isomerases			
1368	78.69	kd	CGS001-55239	OGFOD1	-			
1369	78.68	cc		Wnt family LOF	-			
1370	78.64	kd	CGS001-29978	UBQLN2	Ubiquilin family			
1371	78.56	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
1372	78.55	oe	ccsbBroad304_08684	CXCR7	-			
1373	78.55	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
1374	78.54	kd	CGS001-7533	YWHAH	-			
1375	78.54	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
1376	78.53	kd	CGS001-10221	TRIB1	Trbl family			
1377	78.48	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
1378	78.48	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
1379	78.46	kd	CGS001-4968	OGG1	-			
1380	78.45	kd	CGS001-857	CAV1	-			
1381	78.44	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
1382	78.43	kd	CGS001-64167	ERAP2	Aminopeptidase N			
1383	78.38	oe	ccsbBroad304_01674	TIMP4	-			
1384	78.35	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
1385	78.34	kd	CGS001-10721	POLQ	DNA polymerases			
1386	78.34	kd	CGS001-9415	FADS2	Fatty acid desaturases			
1387	78.3	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
1388	78.29	oe	ccsbBroad304_06234	G6PC	-			
1389	78.27	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
1390	78.26	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
1391	78.24	oe	ccsbBroad304_01002	METTL1	-			
1392	78.17	cc		Estrogen receptor antagonist	-			
1393	78.16	kd	CGS001-3456	IFNB1	Interferons			
1394	78.15	kd	CGS001-1314	COPA	Endogenous ligands			
1395	78.08	oe	ccsbBroad304_01247	POU2AF1	-			
1396	78.05	kd	CGS001-2618	GART	Ribosyl transferases			
1397	78.02	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
1398	78.01	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
1399	77.99	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
1400	77.97	kd	CGS001-58497	PRUNE	-			
1401	77.97	kd	CGS001-54107	POLE3	DNA polymerases			
1402	77.96	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
1403	77.89	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
1404	77.85	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
1405	77.85	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
1406	77.82	kd	CGS001-6794	STK11	LKB subfamily			
1407	77.78	kd	CGS001-54106	TLR9	Toll-like receptor family			
1408	77.78	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
1409	77.76	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
1410	77.75	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
1411	77.67	kd	CGS001-324	APC	Armadillo repeat containing			
1412	77.66	kd	CGS001-3579	CXCR2	Chemokine receptors			
1413	77.66	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
1414	77.65	oe	ccsbBroad304_02287	GNPDA1	-			
1415	77.64	kd	CGS001-25793	FBXO7	F-boxes / other			
1416	77.62	kd	CGS001-5048	PAFAH1B1	WD repeat domain containing			
1417	77.61	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
1418	77.61	kd	CGS001-9052	GPRC5A	GPCR / Class C : Orphans			
1419	77.55	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
1420	77.54	oe	ccsbBroad304_02243	DLGAP5	-			
1421	77.53	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
1422	77.5	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
1423	77.5	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
1424	77.48	oe	ccsbBroad304_02845	PRPF6	-			
1425	77.47	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
1426	77.42	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
1427	77.41	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
1428	77.41	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
1429	77.39	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
1430	77.39	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
1431	77.38	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
1432	77.38	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
1433	77.35	oe	ccsbBroad304_01872	DGCR14	-			
1434	77.34	oe	ccsbBroad304_00120	ATOX1	-			
1435	77.28	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
1436	77.28	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
1437	77.28	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
1438	77.26	kd	CGS001-3755	KCNG1	Voltage-gated potassium channels			
1439	77.26	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
1440	77.25	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
1441	77.2	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
1442	77.2	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
1443	77.19	oe	ccsbBroad304_07704	SUB1	-			
1444	77.18	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
1445	77.12	kd	CGS001-122809	SOCS4	SH2 domain containing			
1446	77.11	cc		BMP Signaling LOF	-			
1447	77.08	cp	BRD-A37052580	physostigmine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Cholinesterase inhibitor
1448	77.05	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
1449	77.05	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1450	77.04	kd	CGS001-23038	WDTC1	DDB1 and CUL4 associated factors			
1451	77.04	kd	CGS001-64170	CARD9	-			
1452	77.02	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
1453	76.99	kd	CGS001-7076	TIMP1	-			
1454	76.98	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
1455	76.98	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
1456	76.97	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
1457	76.97	kd	CGS001-6477	SIAH1	-			
1458	76.97	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
1459	76.9	kd	CGS001-10254	STAM2	-			
1460	76.85	kd	CGS001-64121	RRAGC	-			
1461	76.84	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
1462	76.84	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
1463	76.8	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
1464	76.79	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
1465	76.76	kd	CGS001-11151	CORO1A	Coronins			
1466	76.7	kd	CGS001-2673	GFPT1	-			
1467	76.69	oe	ccsbBroad304_01066	NDUFA4	-			
1468	76.69	kd	CGS001-64175	LEPRE1	-			
1469	76.69	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
1470	76.67	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
1471	76.65	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
1472	76.6	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
1473	76.59	kd	CGS001-114112	TXNRD3	-			
1474	76.56	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
1475	76.56	kd	CGS001-8780	RIOK3	RIO3 subfamily			
1476	76.52	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
1477	76.47	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
1478	76.43	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
1479	76.41	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
1480	76.39	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
1481	76.39	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1482	76.39	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
1483	76.33	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
1484	76.33	kd	CGS001-6926	TBX3	T-boxes			
1485	76.32	oe	ccsbBroad304_02572	SERINC3	-			
1486	76.31	oe	ccsbBroad304_07094	TPMT	-			
1487	76.28	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
1488	76.28	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
1489	76.28	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
1490	76.23	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
1491	76.15	kd	CGS001-6895	TARBP2	-			
1492	76.09	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
1493	76.07	oe	ccsbBroad304_06518	LDHA	-			
1494	76.04	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1495	76.02	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
1496	76	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
1497	75.98	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
1498	75.98	kd	CGS001-4835	NQO2	-			
1499	75.96	kd	CGS001-255738	PCSK9	Subtilisin			
1500	75.92	kd	CGS001-65057	ACD	-			
1501	75.9	kd	CGS001-23523	CABIN1	-			
1502	75.83	kd	CGS001-7182	NR2C2	Testicular receptors			
1503	75.8	oe	ccsbBroad304_06525	LIPA	-			
1504	75.79	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1505	75.79	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
1506	75.69	kd	CGS001-5184	PEPD	Methionyl aminopeptidase			
1507	75.67	kd	CGS001-573	BAG1	-			
1508	75.66	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1509	75.62	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
1510	75.62	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
1511	75.59	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
1512	75.58	kd	CGS001-1951	CELSR3	Cadherins / Major cadherins			
1513	75.55	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
1514	75.49	kd	CGS001-4176	MCM7	-			
1515	75.46	cp	BRD-K34437622	BRD-K34437622	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
1516	75.46	oe	ccsbBroad304_00238	CCNE1	-			
1517	75.45	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
1518	75.44	kd	CGS001-7852	CXCR4	Chemokine receptors			
1519	75.43	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
1520	75.4	oe	ccsbBroad304_03640	CEP72	-			
1521	75.39	kd	CGS001-56834	GPR137	GPCR / Unclassified : 7TM orphan receptors			
1522	75.38	oe	ccsbBroad304_02276	MVP	-			
1523	75.31	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
1524	75.29	kd	CGS001-388677	NOTCH2NL	-			
1525	75.28	cp	BRD-K94887716	TFMPP	Serotonin receptor agonist			Serotonin receptor agonist, Serotonin receptor antagonist
1526	75.26	kd	CGS001-11154	AP4S1	-			
1527	75.24	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
1528	75.23	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
1529	75.18	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
1530	75.17	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
1531	75.15	kd	CGS001-11320	MGAT4A	-			
1532	75.13	kd	CGS001-23411	SIRT1	Histone deacetylases			
1533	75.13	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1534	75.01	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1535	74.98	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
1536	74.94	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
1537	74.84	kd	CGS001-8553	BHLHE40	Basic helix-loop-helix proteins			
1538	74.81	cc		Cell Cycle Inhibition GOF	-			
1539	74.8	kd	CGS001-9788	MTSS1	-			
1540	74.8	kd	CGS001-2768	GNA12	-			
1541	74.76	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
1542	74.73	kd	CGS001-23118	TAB2	-			
1543	74.71	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
1544	74.66	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
1545	74.62	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
1546	74.54	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
1547	74.54	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
1548	74.47	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
1549	74.45	kd	CGS001-4232	MEST	-			
1550	74.44	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
1551	74.43	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
1552	74.28	kd	CGS001-6917	TCEA1	General transcription factors			
1553	74.27	oe	ccsbBroad304_01327	PSPH	-			
1554	74.26	kd	CGS001-11198	SUPT16H	-			
1555	74.26	kd	CGS001-6347	CCL2	Chemokine ligands			
1556	74.24	oe	ccsbBroad304_04294	ATG10	-			
1557	74.22	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1558	74.22	oe	ccsbBroad304_03859	ENOPH1	-			
1559	74.2	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
1560	74.18	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
1561	74.18	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
1562	74.18	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
1563	74.1	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
1564	74.07	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
1565	74.05	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
1566	73.98	cc		Structural maintenance of chromosomes proteins LOF	-			
1567	73.96	kd	CGS001-5879	RAC1	Endogenous ligands			
1568	73.94	oe	ccsbBroad304_10758	CTBP2	-			
1569	73.93	kd	CGS001-5576	PRKAR2A	Protein kinase A			
1570	73.92	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
1571	73.87	kd	CGS001-4998	ORC1	ATPases / AAA-type			
1572	73.82	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
1573	73.78	cp	BRD-A71009679	KUC103420N	-666			-666
1574	73.69	kd	CGS001-54901	CDKAL1	-			
1575	73.68	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
1576	73.67	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
1577	73.67	kd	CGS001-1802	DPH2	-			
1578	73.63	kd	CGS001-4299	AFF1	-			
1579	73.6	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
1580	73.58	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
1581	73.57	kd	CGS001-1876	E2F6	-			
1582	73.56	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
1583	73.56	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
1584	73.5	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
1585	73.46	kd	CGS001-5906	RAP1A	-			
1586	73.41	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
1587	73.39	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
1588	73.38	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
1589	73.36	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
1590	73.35	kd	CGS001-5734	PTGER4	GPCR / Class A : Prostanoid receptors			
1591	73.33	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
1592	73.32	kd	CGS001-84159	ARID5B	-			
1593	73.25	kd	CGS001-9918	NCAPD2	-			
1594	73.24	oe	ccsbBroad304_01832	PAX8	Paired boxes			
1595	73.21	kd	CGS001-1045	CDX2	Homeoboxes / ANTP class : HOXL subclass			
1596	73.14	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
1597	73.07	kd	CGS001-8894	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1598	73.06	kd	CGS001-3976	LIF	-			
1599	73	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
1600	72.94	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
1601	72.94	kd	CGS001-10174	SORBS3	-			
1602	72.93	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
1603	72.93	kd	CGS001-9687	GREB1	-			
1604	72.87	oe	ccsbBroad304_00652	GNAS	-			
1605	72.84	kd	CGS001-5562	PRKAA1	AMPK subfamily			
1606	72.84	kd	CGS001-10491	CRTAP	-			
1607	72.79	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1608	72.73	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
1609	72.66	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
1610	72.65	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
1611	72.61	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
1612	72.55	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
1613	72.52	kd	CGS001-1677	DFFB	-			
1614	72.51	oe	ccsbBroad304_07662	NPRL2	-			
1615	72.51	kd	CGS001-5361	PLXNA1	Plexins			
1616	72.5	kd	CGS001-116535	MRGPRF	GPCR / Class A : Orphans			
1617	72.48	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
1618	72.45	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
1619	72.45	kd	CGS001-23743	BHMT2	-			
1620	72.41	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
1621	72.41	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
1622	72.39	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
1623	72.38	kd	CGS001-55509	BATF3	basic leucine zipper proteins			
1624	72.36	cp	BRD-A49172652	lansoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4, CYP3A5	ATPase inhibitor
1625	72.35	oe	ccsbBroad304_00617	GBA	-			
1626	72.33	kd	CGS001-5163	PDK1	-			
1627	72.29	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
1628	72.2	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
1629	72.17	kd	CGS001-2558	GABRA5	GABA receptors			
1630	72.16	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
1631	72.1	kd	CGS001-6204	RPS10	S ribosomal proteins			
1632	72.09	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
1633	72.05	cp	BRD-K32744045	disulfiram	Aldehyde dehydrogenase inhibitor		ALDH2, ALDH1A2, ALDH5A1, ALDH7A1, CYP2E1, DBH, DNMT1, TRPA1	Aldehyde dehydrogenase inhibitor, TRPV agonist, DNA methyltransferase inhibitor
1634	72	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
1635	71.99	kd	CGS001-23014	FBXO21	F-boxes / other			
1636	71.97	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
1637	71.97	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
1638	71.97	kd	CGS001-1810	DR1	-			
1639	71.96	cc		Histone deacetylases LOF	-			
1640	71.95	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
1641	71.91	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
1642	71.86	oe	ccsbBroad304_02801	CASP14	Caspases			
1643	71.84	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
1644	71.81	kd	CGS001-4023	LPL	-			
1645	71.79	cc		GPCR Subset GOF	-			
1646	71.78	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
1647	71.77	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
1648	71.76	kd	CGS001-5627	PROS1	-			
1649	71.76	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
1650	71.74	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
1651	71.72	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
1652	71.72	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
1653	71.71	kd	CGS001-64750	SMURF2	-			
1654	71.69	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
1655	71.65	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
1656	71.64	kd	CGS001-657	BMPR1A	Type I receptor serine/threonine kinases			
1657	71.63	kd	CGS001-9815	GIT2	Ankyrin repeat domain containing			
1658	71.59	kd	CGS001-587	BCAT2	-			
1659	71.57	kd	CGS001-5257	PHKB	-			
1660	71.55	oe	ccsbBroad304_01395	RFX5	-			
1661	71.54	kd	CGS001-8807	IL18RAP	CD molecules			
1662	71.5	kd	CGS001-7027	TFDP1	-			
1663	71.5	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
1664	71.47	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
1665	71.46	kd	CGS001-94235	GNG8	-			
1666	71.38	oe	ccsbBroad304_04626	EGLN3	-			
1667	71.35	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
1668	71.32	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
1669	71.32	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
1670	71.29	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
1671	71.28	oe	ccsbBroad304_04399	PGBD1	-			
1672	71.25	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
1673	71.17	kd	CGS001-8681	JMJD7-PLA2G4B	-			
1674	71.13	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1675	71.09	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
1676	71.08	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
1677	71.04	cp	BRD-K89708791	rifaximin	RNA synthesis inhibitor		NR1I2, CYP3A4	RNA synthesis inhibitor
1678	70.98	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
1679	70.97	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
1680	70.96	kd	CGS001-34	ACADM	-			
1681	70.95	oe	ccsbBroad304_09035	COASY	-			
1682	70.95	kd	CGS001-10287	RGS19	Regulators of G-protein signaling			
1683	70.94	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
1684	70.93	kd	CGS001-1062	CENPE	Kinesins			
1685	70.89	oe	ccsbBroad304_02569	BTG3	-			
1686	70.89	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
1687	70.88	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
1688	70.87	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
1689	70.85	kd	CGS001-115201	ATG4A	-			
1690	70.82	oe	ccsbBroad304_02875	BRP44	-			
1691	70.8	cc		Tricyclic antidepressant	-			
1692	70.8	oe	ccsbBroad304_01398	RHEB	-			
1693	70.78	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
1694	70.77	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
1695	70.76	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
1696	70.73	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
1697	70.72	kd	CGS001-10957	PNRC1	-			
1698	70.64	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
1699	70.64	oe	ccsbBroad304_02579	YWHAQ	-			
1700	70.63	kd	CGS001-3226	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
1701	70.62	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
1702	70.57	oe	ccsbBroad304_01008	KITLG	-			
1703	70.51	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
1704	70.48	kd	CGS001-154197	PNLDC1	-			
1705	70.47	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
1706	70.36	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
1707	70.35	kd	CGS001-10923	SUB1	-			
1708	70.31	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
1709	70.29	kd	CGS001-54499	TMCO1	-			
1710	70.29	kd	CGS001-665	BNIP3L	-			
1711	70.28	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
1712	70.26	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
1713	70.26	kd	CGS001-29984	RHOD	-			
1714	70.25	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
1715	70.24	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
1716	70.2	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
1717	70.18	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
1718	70.18	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
1719	70.18	kd	CGS001-4173	MCM4	-			
1720	70.15	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
1721	70.15	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
1722	70.12	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
1723	70.11	kd	CGS001-57192	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
1724	70.1	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
1725	70.09	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
1726	70.09	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
1727	70.03	kd	CGS001-3799	KIF5B	Kinesins			
1728	70	oe	ccsbBroad304_03118	NRBP1	NRBP family			
1729	69.97	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
1730	69.96	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
1731	69.92	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
1732	69.91	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
1733	69.88	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
1734	69.86	kd	CGS001-23710	GABARAPL1	-			
1735	69.86	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
1736	69.83	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
1737	69.82	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
1738	69.81	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
1739	69.78	kd	CGS001-634	CEACAM1	CD molecules			
1740	69.71	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
1741	69.68	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
1742	69.68	oe	ccsbBroad304_07754	FGFR1OP	-			
1743	69.66	cc		VEGFR inhibitor	-			
1744	69.66	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
1745	69.65	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
1746	69.62	kd	CGS001-10046	MAMLD1	-			
1747	69.61	kd	CGS001-283455	KSR2	RAF family			
1748	69.6	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
1749	69.6	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
1750	69.56	kd	CGS001-2512	FTL	-			
1751	69.55	oe	ccsbBroad304_03357	RASD1	-			
1752	69.54	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
1753	69.54	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
1754	69.48	kd	CGS001-55869	HDAC8	Histone deacetylases			
1755	69.45	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
1756	69.39	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
1757	69.33	kd	CGS001-84878	ZBTB45	BTB/POZ domain containing			
1758	69.33	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
1759	69.29	kd	CGS001-2629	GBA	-			
1760	69.27	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
1761	69.2	kd	CGS001-10010	TANK	-			
1762	69.15	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
1763	69.09	kd	CGS001-54805	CNNM2	-			
1764	69.06	kd	CGS001-8572	PDLIM4	-			
1765	69.06	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
1766	69.02	kd	CGS001-353	APRT	-			
1767	69.01	kd	CGS001-64343	AZI2	-			
1768	69	kd	CGS001-9360	PPIG	-			
1769	68.99	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
1770	68.98	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
1771	68.96	kd	CGS001-6827	SUPT4H1	-			
1772	68.95	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
1773	68.93	kd	CGS001-3776	KCNK2	Two-P potassium channels			
1774	68.9	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
1775	68.87	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
1776	68.86	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
1777	68.85	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
1778	68.83	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
1779	68.79	oe	ccsbBroad304_08802	ELAC2	-			
1780	68.77	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
1781	68.64	kd	CGS001-29928	TIMM22	-			
1782	68.62	kd	CGS001-5378	PMS1	-			
1783	68.62	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
1784	68.6	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
1785	68.55	oe	ccsbBroad304_07600	NSA2	-			
1786	68.54	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
1787	68.48	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
1788	68.47	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
1789	68.42	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
1790	68.41	kd	CGS001-7444	VRK2	Vaccina related kinase (VRK) family			
1791	68.41	kd	CGS001-1997	ELF1	ETS Transcription Factors			
1792	68.4	oe	ccsbBroad304_08292	IP6K2	-			
1793	68.4	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
1794	68.39	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
1795	68.36	kd	CGS001-6829	SUPT5H	-			
1796	68.34	kd	CGS001-4615	MYD88	-			
1797	68.31	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
1798	68.3	kd	CGS001-6387	CXCL12	Endogenous ligands			
1799	68.3	kd	CGS001-124583	CANT1	-			
1800	68.26	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
1801	68.24	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
1802	68.22	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
1803	68.22	kd	CGS001-5987	TRIM27	-			
1804	68.17	kd	CGS001-4482	MSRA	-			
1805	68.14	kd	CGS001-4267	CD99	CD molecules			
1806	68.1	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1807	68.07	kd	CGS001-818	CAMK2G	CAMK2 family			
1808	68.06	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
1809	68.05	oe	ccsbBroad304_02756	RRP8	-			
1810	68.05	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
1811	68.04	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
1812	68.04	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
1813	68.03	kd	CGS001-9541	CIR1	-			
1814	68.03	kd	CGS001-11142	PKIG	-			
1815	67.9	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
1816	67.89	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
1817	67.87	kd	CGS001-84923	FAM104A	-			
1818	67.86	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1819	67.84	kd	CGS001-3269	HRH1	Histamine receptors			
1820	67.83	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1821	67.7	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1822	67.69	kd	CGS001-7158	TP53BP1	-			
1823	67.63	kd	CGS001-11343	MGLL	Endocannabinoid turnover			
1824	67.62	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
1825	67.62	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
1826	67.61	kd	CGS001-3225	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
1827	67.61	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
1828	67.6	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
1829	67.57	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1830	67.57	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
1831	67.53	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
1832	67.5	cc		GATA Zinc finger domain containing LOF	-			
1833	67.5	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
1834	67.49	kd	CGS001-8576	STK16	NAK family			
1835	67.47	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1836	67.45	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
1837	67.42	cc		Lysine acetyltransferases LOF	-			
1838	67.39	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
1839	67.39	kd	CGS001-2919	CXCL1	Endogenous ligands			
1840	67.38	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
1841	67.36	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
1842	67.34	kd	CGS001-2145	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
1843	67.32	kd	CGS001-84290	CAPNS2	EF-hand domain containing			
1844	67.28	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
1845	67.23	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
1846	67.18	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
1847	67.16	kd	CGS001-10142	AKAP9	A-kinase anchor proteins			
1848	67.15	kd	CGS001-5695	PSMB7	Proteasome subunits			
1849	67.1	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
1850	67.08	kd	CGS001-55120	FANCL	Fanconi anemia, complementation groups			
1851	67.06	oe	ccsbBroad304_02367	CALCOCO2	-			
1852	67.05	kd	CGS001-5910	RAP1GDS1	Armadillo repeat containing			
1853	66.96	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
1854	66.95	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
1855	66.95	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
1856	66.94	kd	CGS001-7311	UBA52	L ribosomal proteins			
1857	66.89	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
1858	66.87	kd	CGS001-79187	FSD1	Fibronectin type III domain containing			
1859	66.85	cc		Interleukins GOF	-			
1860	66.85	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
1861	66.82	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
1862	66.82	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
1863	66.8	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
1864	66.71	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
1865	66.68	kd	CGS001-3553	IL1B	Interleukins and interleukin receptors			
1866	66.65	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
1867	66.61	kd	CGS001-3930	LBR	Tudor domain containing			
1868	66.53	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
1869	66.44	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1870	66.44	kd	CGS001-593	BCKDHA	-			
1871	66.43	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
1872	66.43	kd	CGS001-7078	TIMP3	-			
1873	66.38	kd	CGS001-55179	FAIM	-			
1874	66.3	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
1875	66.27	kd	CGS001-117581	TWIST2	Basic helix-loop-helix proteins			
1876	66.19	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
1877	66.17	kd	CGS001-6648	SOD2	-			
1878	66.17	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
1879	66.16	cc		MDM inhibitor	-			
1880	66.15	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
1881	66.14	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1882	66.13	kd	CGS001-56916	SMARCAD1	-			
1883	66.12	oe	ccsbBroad304_05937	CASP7	Caspases			
1884	66.1	kd	CGS001-28969	BZW2	-			
1885	66.09	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
1886	66.08	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
1887	66.07	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
1888	66.04	kd	CGS001-5159	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1889	66.03	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
1890	65.96	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
1891	65.95	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
1892	65.94	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
1893	65.91	kd	CGS001-84108	PCGF6	Polycomb group ring fingers			
1894	65.91	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
1895	65.86	oe	ccsbBroad304_00226	CAV1	-			
1896	65.86	kd	CGS001-1655	DDX5	DEAD-boxes			
1897	65.83	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
1898	65.83	kd	CGS001-4801	NFYB	-			
1899	65.83	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
1900	65.79	kd	CGS001-3417	IDH1	-			
1901	65.64	kd	CGS001-1950	EGF	-			
1902	65.61	oe	ccsbBroad304_00620	GCDH	-			
1903	65.6	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
1904	65.57	kd	CGS001-10810	WASF3	-			
1905	65.47	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1906	65.47	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
1907	65.46	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1908	65.44	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
1909	65.43	oe	ccsbBroad304_08840	KIF9	Kinesins			
1910	65.41	cc		Lipocalins GOF	-			
1911	65.41	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
1912	65.39	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
1913	65.39	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
1914	65.36	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
1915	65.36	kd	CGS001-9702	CEP57	-			
1916	65.36	oe	ccsbBroad304_01654	TCTA	-			
1917	65.35	kd	CGS001-2729	GCLC	-			
1918	65.33	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
1919	65.32	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
1920	65.29	cc		FOS transcription factor family GOF	-			
1921	65.28	kd	CGS001-4779	NFE2L1	basic leucine zipper proteins			
1922	65.27	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
1923	65.27	kd	CGS001-11340	EXOSC8	-			
1924	65.23	kd	CGS001-4094	MAF	-			
1925	65.23	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
1926	65.22	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
1927	65.2	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
1928	65.19	oe	ccsbBroad304_07374	PTPLA	-			
1929	65.12	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
1930	65.1	kd	CGS001-6009	RHEB	-			
1931	65.1	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
1932	65.06	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
1933	65.04	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
1934	65.03	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1935	65.02	kd	CGS001-57057	TBX20	T-boxes			
1936	64.99	kd	CGS001-3203	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
1937	64.99	kd	CGS001-84890	ADO	-			
1938	64.96	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
1939	64.95	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
1940	64.94	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
1941	64.88	cc		Toll like receptors LOF	-			
1942	64.88	kd	CGS001-9189	ZBED1	Pseudoautosomal regions / PAR1			
1943	64.88	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
1944	64.86	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
1945	64.83	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
1946	64.72	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1947	64.67	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
1948	64.67	kd	CGS001-822	CAPG	-			
1949	64.64	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
1950	64.64	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
1951	64.59	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
1952	64.57	kd	CGS001-5805	PTS	-			
1953	64.56	kd	CGS001-57157	PHTF2	-			
1954	64.53	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
1955	64.51	cc		HSP inhibitor	-			
1956	64.48	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
1957	64.46	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
1958	64.43	oe	ccsbBroad304_08104	MED4	-			
1959	64.41	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
1960	64.39	kd	CGS001-54881	TEX10	-			
1961	64.38	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
1962	64.36	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
1963	64.31	oe	ccsbBroad304_08461	CDCA4	-			
1964	64.31	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
1965	64.29	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
1966	64.29	kd	CGS001-1981	EIF4G1	Parkinson disease			
1967	64.27	kd	CGS001-3682	ITGAE	Integrins			
1968	64.22	kd	CGS001-182	JAG1	CD molecules			
1969	64.18	kd	CGS001-51347	TAOK3	TAO subfamily			
1970	64.17	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
1971	64.13	kd	CGS001-51564	HDAC7	Histone deacetylases			
1972	64.12	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
1973	64.11	kd	CGS001-509	ATP5C1	ATPases / F-type			
1974	64.09	kd	CGS001-25861	DFNB31	-			
1975	64.06	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
1976	63.95	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
1977	63.87	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
1978	63.84	cp	BRD-K81855038	roxatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
1979	63.82	cp	BRD-K37814297	acepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
1980	63.81	kd	CGS001-4869	NPM1	-			
1981	63.79	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
1982	63.78	oe	ccsbBroad304_01985	EIF3H	-			
1983	63.77	oe	ccsbBroad304_00063	AMPD2	-			
1984	63.73	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
1985	63.66	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
1986	63.66	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
1987	63.63	kd	CGS001-9929	JOSD1	-			
1988	63.59	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1989	63.57	kd	CGS001-30	ACAA1	-			
1990	63.56	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
1991	63.5	oe	ccsbBroad304_02884	POT1	-			
1992	63.49	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
1993	63.45	cp	BRD-K15519488	CS-110266	Dopamine receptor agonist		SLC6A3	Dopamine receptor agonist
1994	63.45	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
1995	63.44	kd	CGS001-125950	RAVER1	RNA binding motif (RRM) containing			
1996	63.41	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
1997	63.36	oe	ccsbBroad304_09225	BUD13	-			
1998	63.34	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
1999	63.33	kd	CGS001-1515	CTSL2	-			
2000	63.32	kd	CGS001-79850	FAM57A	-			
2001	63.27	cc		Cyclooxygenase inhibitor	-			
2002	63.27	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
2003	63.27	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
2004	63.26	kd	CGS001-80349	WDR61	WD repeat domain containing			
2005	63.25	oe	ccsbBroad304_02398	LANCL1	-			
2006	63.22	kd	CGS001-9531	BAG3	-			
2007	63.2	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
2008	63.18	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
2009	63.14	kd	CGS001-835	CASP2	Caspases			
2010	63.12	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
2011	63.12	kd	CGS001-94103	ORMDL3	-			
2012	63.11	kd	CGS001-112812	FDX1L	-			
2013	63.1	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
2014	63.1	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
2015	63.09	kd	CGS001-6491	STIL	-			
2016	63.07	kd	CGS001-351	APP	Endogenous ligands			
2017	63.03	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
2018	62.99	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
2019	62.97	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
2020	62.92	oe	ccsbBroad304_06237	GAA	Glycosidases			
2021	62.92	kd	CGS001-57326	PBXIP1	-			
2022	62.9	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
2023	62.89	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
2024	62.88	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
2025	62.85	kd	CGS001-2247	FGF2	Endogenous ligands			
2026	62.84	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
2027	62.84	kd	CGS001-91137	SLC25A46	Miscellaneous SLC25 mitochondrial transporters			
2028	62.82	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
2029	62.81	oe	ccsbBroad304_02052	KYNU	-			
2030	62.81	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
2031	62.78	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
2032	62.75	kd	CGS001-65123	INTS3	-			
2033	62.72	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
2034	62.69	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
2035	62.68	kd	CGS001-3664	IRF6	-			
2036	62.63	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
2037	62.59	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
2038	62.59	kd	CGS001-9616	RNF7	RING-type (C3HC4) zinc fingers			
2039	62.55	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
2040	62.55	oe	ccsbBroad304_06282	GLDC	-			
2041	62.51	oe	ccsbBroad304_02163	MED7	-			
2042	62.46	kd	CGS001-253260	RICTOR	-			
2043	62.46	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
2044	62.44	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
2045	62.43	kd	CGS001-5193	PEX12	-			
2046	62.42	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
2047	62.41	kd	CGS001-7247	TSN	-			
2048	62.39	kd	CGS001-23405	DICER1	-			
2049	62.35	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
2050	62.32	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
2051	62.31	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
2052	62.27	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
2053	62.18	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
2054	62.16	kd	CGS001-10284	SAP18	-			
2055	62.16	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
2056	62.14	kd	CGS001-115727	RASGRP4	EF-hand domain containing			
2057	62.08	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
2058	62.02	kd	CGS001-4312	MMP1	Matrix metallopeptidase			
2059	62.01	kd	CGS001-4602	MYB	-			
2060	61.98	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
2061	61.96	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
2062	61.92	kd	CGS001-50808	AK3	-			
2063	61.9	oe	ccsbBroad304_01577	SOD1	-			
2064	61.87	oe	ccsbBroad304_02485	STAMBP	-			
2065	61.85	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
2066	61.85	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
2067	61.82	kd	CGS001-29998	GLTSCR1	-			
2068	61.8	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
2069	61.8	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
2070	61.78	kd	CGS001-10308	ZNF267	Zinc fingers, C2H2-type			
2071	61.77	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2072	61.77	kd	CGS001-57167	SALL4	Zinc fingers, C2H2-type			
2073	61.72	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
2074	61.7	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
2075	61.69	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
2076	61.67	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
2077	61.66	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
2078	61.63	kd	CGS001-5743	PTGS2	Cyclooxygenase			
2079	61.6	kd	CGS001-11157	LSM6	-			
2080	61.59	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
2081	61.57	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
2082	61.56	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
2083	61.55	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
2084	61.55	kd	CGS001-10161	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2085	61.49	oe	ccsbBroad304_01371	RALA	-			
2086	61.44	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
2087	61.43	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
2088	61.42	kd	CGS001-2539	G6PD	-			
2089	61.38	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
2090	61.32	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
2091	61.27	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
2092	61.27	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
2093	61.27	kd	CGS001-149428	BNIPL	-			
2094	61.23	kd	CGS001-7465	WEE1	WEE family			
2095	61.23	kd	CGS001-2730	GCLM	-			
2096	61.21	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
2097	61.2	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
2098	61.16	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
2099	61.13	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
2100	61.09	cc		CCK receptor antagonist	-			
2101	61.09	kd	CGS001-9887	SMG7	-			
2102	61.08	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
2103	61.08	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
2104	61.03	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
2105	61.03	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
2106	61.02	kd	CGS001-7353	UFD1L	-			
2107	61	kd	CGS001-57154	SMURF1	-			
2108	60.99	oe	ccsbBroad304_06642	NIT1	-			
2109	60.97	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2110	60.92	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
2111	60.85	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
2112	60.77	kd	CGS001-7484	WNT9B	Wingless-type MMTV integration sites			
2113	60.75	kd	CGS001-7103	TSPAN8	Tetraspanins			
2114	60.71	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
2115	60.66	oe	ccsbBroad304_05907	BUB1B	Bub family			
2116	60.63	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
2117	60.63	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
2118	60.62	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
2119	60.59	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2120	60.56	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
2121	60.56	kd	CGS001-81620	CDT1	-			
2122	60.5	kd	CGS001-9488	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
2123	60.5	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
2124	60.47	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
2125	60.42	oe	ccsbBroad304_07766	RASSF1	-			
2126	60.4	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
2127	60.36	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
2128	60.34	kd	CGS001-5891	MOK	RCK family			
2129	60.34	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
2130	60.28	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
2131	60.21	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
2132	60.15	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
2133	60.15	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
2134	60.13	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
2135	60.1	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
2136	60.09	kd	CGS001-8834	TMEM11	-			
2137	60.08	kd	CGS001-57149	LYRM1	LYR motif containing			
2138	59.99	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
2139	59.99	kd	CGS001-1036	CDO1	-			
2140	59.9	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
2141	59.89	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
2142	59.89	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
2143	59.88	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2144	59.84	oe	ccsbBroad304_09095	PUS7L	-			
2145	59.76	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2146	59.75	oe	ccsbBroad304_00036	AFP	-			
2147	59.75	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
2148	59.72	oe	ccsbBroad304_08839	IFIH1	-			
2149	59.69	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
2150	59.66	kd	CGS001-8334	HIST1H2AC	Histones / Replication-dependent			
2151	59.64	kd	CGS001-5045	FURIN	Subtilisin			
2152	59.63	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
2153	59.61	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
2154	59.61	oe	ccsbBroad304_03420	TOLLIP	-			
2155	59.57	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
2156	59.56	kd	CGS001-9797	TATDN2	-			
2157	59.54	oe	ccsbBroad304_00510	EPHX2	-			
2158	59.54	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2159	59.48	kd	CGS001-1154	CISH	SH2 domain containing			
2160	59.45	kd	CGS001-6857	SYT1	Synaptotagmins			
2161	59.44	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
2162	59.44	oe	ccsbBroad304_00102	RND3	-			
2163	59.43	kd	CGS001-7035	TFPI	-			
2164	59.43	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
2165	59.37	kd	CGS001-5445	PON2	Paraoxonases			
2166	59.35	cp	BRD-A95696820	acadesine	AMPK activator			AMPK activator
2167	59.35	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
2168	59.31	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
2169	59.29	kd	CGS001-4199	ME1	-			
2170	59.17	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
2171	59.17	kd	CGS001-3589	IL11	Endogenous ligands			
2172	59.17	oe	ccsbBroad304_14011	PAPSS1	-			
2173	59.16	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
2174	59.16	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
2175	59.14	kd	CGS001-56616	DIABLO	-			
2176	59.09	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
2177	59.09	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
2178	59.06	kd	CGS001-8837	CFLAR	Endogenous ligands			
2179	58.88	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
2180	58.83	kd	CGS001-161725	OTUD7A	OTU domain containing			
2181	58.83	kd	CGS001-2149	F2R	Protease activated receptors			
2182	58.74	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
2183	58.73	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
2184	58.72	cc		PI3K Signaling LOF	-			
2185	58.72	kd	CGS001-4798	NFRKB	INO80 complex subunits			
2186	58.67	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
2187	58.63	kd	CGS001-3614	IMPDH1	Oxidoreductases			
2188	58.62	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
2189	58.61	kd	CGS001-27113	BBC3	-			
2190	58.6	cc		Angiotensin receptor antagonist	-			
2191	58.57	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
2192	58.51	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
2193	58.49	oe	ccsbBroad304_00747	HLF	-			
2194	58.47	kd	CGS001-9928	KIF14	Kinesins			
2195	58.45	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
2196	58.45	kd	CGS001-6598	SMARCB1	-			
2197	58.41	kd	CGS001-10051	SMC4	Structural maintenance of chromosomes proteins			
2198	58.41	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
2199	58.38	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
2200	58.38	kd	CGS001-64333	ARHGAP9	Rho GTPase activating proteins			
2201	58.28	cp	BRD-K13664374	dichloroacetic-acid	Pyruvate dehydrogenase kinase inhibitor		PDK1	Pyruvate dehydrogenase kinase inhibitor
2202	58.28	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
2203	58.28	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
2204	58.25	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
2205	58.23	cp	BRD-K66412701	pazufloxacin	Topoisomerase inhibitor			Topoisomerase inhibitor
2206	58.16	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
2207	58.15	oe	ccsbBroad304_05931	CAPG	-			
2208	58.15	oe	ccsbBroad304_07219	CDC7	CDC7 family			
2209	58.14	oe	ccsbBroad304_06435	RBPJ	-			
2210	58.13	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
2211	58.12	kd	CGS001-64781	CERK	Ceramide kinase			
2212	58.1	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
2213	58.08	kd	CGS001-8193	DPF1	Zinc fingers, PHD-type			
2214	58.07	kd	CGS001-80135	RPF1	-			
2215	58.07	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
2216	58.06	kd	CGS001-23509	POFUT1	Fucosyltransferases			
2217	57.99	kd	CGS001-8801	SUCLG2	-			
2218	57.93	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
2219	57.91	kd	CGS001-1407	CRY1	-			
2220	57.91	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
2221	57.89	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
2222	57.86	kd	CGS001-5933	RBL1	-			
2223	57.86	oe	ccsbBroad304_04649	ADC	-			
2224	57.82	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
2225	57.81	kd	CGS001-147179	WIPF2	-			
2226	57.79	kd	CGS001-51380	CSAD	-			
2227	57.77	oe	ccsbBroad304_04544	RCCD1	-			
2228	57.68	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
2229	57.65	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
2230	57.64	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
2231	57.61	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
2232	57.6	kd	CGS001-3109	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
2233	57.58	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
2234	57.57	kd	CGS001-55620	STAP2	-			
2235	57.57	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
2236	57.52	kd	CGS001-5584	PRKCI	Iota subfamily			
2237	57.52	kd	CGS001-5427	POLE2	DNA polymerases			
2238	57.47	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
2239	57.45	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2240	57.44	kd	CGS001-586	BCAT1	-			
2241	57.4	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
2242	57.4	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
2243	57.39	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
2244	57.39	kd	CGS001-23657	SLC7A11	Solute carriers			
2245	57.38	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
2246	57.35	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
2247	57.34	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
2248	57.34	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
2249	57.34	kd	CGS001-10645	CAMKK2	Meta subfamily			
2250	57.33	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
2251	57.29	kd	CGS001-23149	FCHO1	-			
2252	57.29	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
2253	57.23	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
2254	57.22	kd	CGS001-3516	RBPJ	-			
2255	57.2	kd	CGS001-57504	MTA3	GATA zinc finger domain containing			
2256	57.15	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
2257	57.13	kd	CGS001-3032	HADHB	-			
2258	57.1	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
2259	57.07	kd	CGS001-388	RHOB	-			
2260	57.06	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
2261	57.06	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
2262	57.01	cc		Calmodulin antagonist	-			
2263	56.99	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
2264	56.96	oe	ccsbBroad304_05547	TMEM110	-			
2265	56.94	kd	CGS001-7840	ALMS1	-			
2266	56.91	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
2267	56.89	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
2268	56.88	oe	ccsbBroad304_09006	RPF1	-			
2269	56.88	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
2270	56.88	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2271	56.86	kd	CGS001-81611	ANP32E	ANP32 acidic nuclear phosphoproteins			
2272	56.84	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
2273	56.84	kd	CGS001-3939	LDHA	-			
2274	56.83	kd	CGS001-9917	FAM20B	-			
2275	56.82	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
2276	56.81	oe	ccsbBroad304_02012	FADD	-			
2277	56.8	kd	CGS001-5566	PRKACA	Protein kinase A			
2278	56.79	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
2279	56.78	cp	BRD-K83144676	olmesartan	Angiotensin antagonist		AGTR1	Angiotensin antagonist
2280	56.77	kd	CGS001-109	ADCY3	Adenylyl cyclases			
2281	56.76	kd	CGS001-55577	NAGK	-			
2282	56.73	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
2283	56.72	oe	ccsbBroad304_07491	IP6K1	-			
2284	56.7	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
2285	56.69	kd	CGS001-1645	AKR1C1	Aldo-keto reductases			
2286	56.68	kd	CGS001-11315	PARK7	Parkinson disease			
2287	56.67	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
2288	56.67	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
2289	56.66	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2290	56.6	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
2291	56.57	oe	ccsbBroad304_01061	NAB2	-			
2292	56.53	kd	CGS001-23678	SGK3	SGK family			
2293	56.52	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
2294	56.49	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
2295	56.49	kd	CGS001-5105	PCK1	-			
2296	56.46	oe	ccsbBroad304_02626	PKIG	-			
2297	56.46	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
2298	56.44	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
2299	56.42	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
2300	56.4	kd	CGS001-8313	AXIN2	-			
2301	56.4	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
2302	56.33	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
2303	56.32	kd	CGS001-54623	PAF1	-			
2304	56.31	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
2305	56.28	kd	CGS001-9867	PJA2	RING-type (C3HC4) zinc fingers			
2306	56.28	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
2307	56.27	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
2308	56.24	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
2309	56.21	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
2310	56.21	kd	CGS001-5446	PON3	Paraoxonases			
2311	56.21	kd	CGS001-140690	CTCFL	Zinc fingers, C2H2-type			
2312	56.16	kd	CGS001-10914	PAPOLA	-			
2313	56.14	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
2314	56.12	oe	ccsbBroad304_07411	LPXN	-			
2315	56.1	kd	CGS001-6821	SUOX	-			
2316	56.09	kd	CGS001-10362	HMG20B	High mobility group / Non-canonical			
2317	56.04	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2318	56.04	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
2319	56.02	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2320	56.02	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
2321	56.01	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
2322	55.99	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
2323	55.94	oe	ccsbBroad304_09615	LACC1	-			
2324	55.93	kd	CGS001-1387	CREBBP	Chromatin-modifying enzymes / K-acetyltransferases			
2325	55.88	kd	CGS001-6421	SFPQ	RNA binding motif (RRM) containing			
2326	55.85	kd	CGS001-1445	CSK	Csk family			
2327	55.84	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
2328	55.84	kd	CGS001-2885	GRB2	SH2 domain containing			
2329	55.84	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
2330	55.83	kd	CGS001-949	SCARB1	-			
2331	55.81	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
2332	55.81	kd	CGS001-6713	SQLE	Lanosterol biosynthesis pathway			
2333	55.81	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
2334	55.78	oe	ccsbBroad304_05194	LIPH	-			
2335	55.74	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
2336	55.71	kd	CGS001-27336	HTATSF1	RNA binding motif (RRM) containing			
2337	55.7	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
2338	55.64	cp	BRD-K49481516	galantamine	Acetylcholinesterase inhibitor		ACHE, BCHE, CHRNA1, CHRNA10, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNA9, CHRNB1, CHRNB2, CHRNB3, CHRNB4, CHRND, CHRNE, CHRNG	Acetylcholinesterase inhibitor
2339	55.63	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
2340	55.63	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
2341	55.51	oe	ccsbBroad304_00006	ACADM	-			
2342	55.51	kd	CGS001-51027	BOLA1	-			
2343	55.5	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
2344	55.46	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
2345	55.45	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
2346	55.45	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
2347	55.43	kd	CGS001-80212	CCDC92	-			
2348	55.42	oe	ccsbBroad304_04292	INHBE	-			
2349	55.41	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
2350	55.38	kd	CGS001-56889	TM9SF3	-			
2351	55.36	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
2352	55.35	oe	ccsbBroad304_02432	IFI30	-			
2353	55.33	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
2354	55.18	oe	ccsbBroad304_06048	CRYZ	-			
2355	55.15	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
2356	55.15	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
2357	55.14	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
2358	55.13	kd	CGS001-84811	BUD13	-			
2359	55.09	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
2360	55.08	kd	CGS001-8522	GAS7	-			
2361	55.05	kd	CGS001-4191	MDH2	-			
2362	55.04	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
2363	55.03	kd	CGS001-10084	PQBP1	-			
2364	55.02	oe	ccsbBroad304_07557	NAMPT	-			
2365	54.99	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
2366	54.95	kd	CGS001-5641	LGMN	Legumain			
2367	54.95	kd	CGS001-2548	GAA	Glycosidases			
2368	54.94	kd	CGS001-10383	TUBB2C	Tubulins			
2369	54.93	oe	ccsbBroad304_00550	FDXR	-			
2370	54.87	kd	CGS001-1616	DAXX	-			
2371	54.81	oe	ccsbBroad304_07890	CBX7	-			
2372	54.78	oe	ccsbBroad304_06538	LSP1	-			
2373	54.76	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
2374	54.75	kd	CGS001-9967	THRAP3	-			
2375	54.74	kd	CGS001-5447	POR	-			
2376	54.73	kd	CGS001-9868	TOMM70A	Tetratricopeptide (TTC) repeat domain containing			
2377	54.69	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2378	54.69	oe	ccsbBroad304_08392	EXOC6	-			
2379	54.68	kd	CGS001-10401	PIAS3	Zinc fingers, MIZ-type			
2380	54.66	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
2381	54.64	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
2382	54.61	cc		Retinoid receptor agonist	-			
2383	54.61	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
2384	54.6	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
2385	54.57	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
2386	54.56	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
2387	54.49	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
2388	54.49	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
2389	54.49	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
2390	54.45	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
2391	54.45	kd	CGS001-6871	TADA2A	-			
2392	54.42	kd	CGS001-7528	YY1	INO80 complex subunits			
2393	54.42	kd	CGS001-9817	KEAP1	Kelch-like proteins			
2394	54.37	oe	ccsbBroad304_07808	RAB11FIP2	-			
2395	54.37	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
2396	54.36	kd	CGS001-64943	NT5DC2	-			
2397	54.36	kd	CGS001-57396	CLK4	CDC-like kinases			
2398	54.28	kd	CGS001-3638	INSIG1	-			
2399	54.26	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
2400	54.24	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
2401	54.22	oe	ccsbBroad304_07197	PDHX	-			
2402	54.22	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
2403	54.21	cp	BRD-K04710043	hexamethylenebisacetamide	AKT inhibitor			AKT inhibitor, Differentiation inducer, NFkB pathway inhibitor
2404	54.21	kd	CGS001-79947	DHDDS	-			
2405	54.21	kd	CGS001-11214	AKAP13	A-kinase anchor proteins			
2406	54.2	cc		Dopamine receptor antagonist	-			
2407	54.19	kd	CGS001-23013	SPEN	RNA binding motif (RRM) containing			
2408	54.16	oe	ccsbBroad304_02402	TMEM5	-			
2409	54.16	kd	CGS001-1675	CFD	Complement system			
2410	54.14	kd	CGS001-10626	TRIM16	Tripartite motif containing			
2411	54.14	kd	CGS001-23081	KDM4C	Histone demethylases			
2412	54.12	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
2413	54.11	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
2414	54.11	kd	CGS001-2793	GNGT2	-			
2415	54.1	oe	ccsbBroad304_02496	MTX2	-			
2416	54.09	kd	CGS001-1910	EDNRB	Endothelin receptors			
2417	54.07	kd	CGS001-54899	PXK	Slob family			
2418	54.07	oe	ccsbBroad304_05894	BLVRA	-			
2419	54.03	kd	CGS001-4329	ALDH6A1	Aldehyde dehydrogenases			
2420	54.02	kd	CGS001-10013	HDAC6	Histone deacetylases			
2421	54	kd	CGS001-5663	PSEN1	Presenilin			
2422	53.91	cp	BRD-A15914070	4-hydroxy-2-nonenal	Cytotoxic lipid peroxidation product		IKBKB	Cytotoxic lipid peroxidation product
2423	53.88	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
2424	53.88	oe	ccsbBroad304_04387	MKI67IP	-			
2425	53.85	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2426	53.84	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
2427	53.83	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
2428	53.78	cc		Bromodomain Inhibitor	-			
2429	53.78	kd	CGS001-9784	SNX17	Sorting nexins			
2430	53.76	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
2431	53.74	oe	ccsbBroad304_08152	PSAT1	-			
2432	53.74	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2433	53.74	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
2434	53.73	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
2435	53.72	oe	ccsbBroad304_06292	GNAI2	-			
2436	53.72	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
2437	53.63	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
2438	53.63	kd	CGS001-23621	BACE1	Pepsin			
2439	53.61	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
2440	53.58	kd	CGS001-2806	GOT2	-			
2441	53.57	oe	ccsbBroad304_09281	TPD52L3	-			
2442	53.51	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
2443	53.43	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
2444	53.43	kd	CGS001-3630	INS	-			
2445	53.43	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
2446	53.42	kd	CGS001-54205	CYCS	-			
2447	53.42	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
2448	53.4	kd	CGS001-6285	S100B	EF-hand domain containing			
2449	53.36	kd	CGS001-6514	SLC2A2	Solute carriers			
2450	53.34	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
2451	53.34	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
2452	53.32	kd	CGS001-10991	SLC38A3	System N-like transporters			
2453	53.31	kd	CGS001-26064	RAI14	Ankyrin repeat domain containing			
2454	53.3	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
2455	53.28	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
2456	53.25	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
2457	53.23	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
2458	53.23	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
2459	53.22	kd	CGS001-6856	SYPL1	-			
2460	53.22	kd	CGS001-55163	PNPO	-			
2461	53.21	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
2462	53.2	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
2463	53.18	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
2464	53.18	kd	CGS001-3615	IMPDH2	Oxidoreductases			
2465	53.16	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
2466	53.15	cc		Wnt family GOF	-			
2467	53.13	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
2468	53.11	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
2469	53.08	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
2470	53.08	kd	CGS001-23576	DDAH1	Dimethylarginine dimethylaminohydrolases			
2471	53.07	kd	CGS001-3460	IFNGR2	Interferon receptor family			
2472	53.07	oe	ccsbBroad304_07217	AXIN2	-			
2473	53.05	kd	CGS001-9270	ITGB1BP1	-			
2474	53.04	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
2475	53.04	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
2476	53.02	kd	CGS001-23536	ADAT1	-			
2477	53	oe	ccsbBroad304_03113	DSE	-			
2478	52.92	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2479	52.88	kd	CGS001-3676	ITGA4	Integrins			
2480	52.87	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
2481	52.87	kd	CGS001-117154	DACH2	-			
2482	52.86	kd	CGS001-8639	AOC3	Oxidoreductases			
2483	52.75	oe	ccsbBroad304_06103	DMD	-			
2484	52.74	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
2485	52.72	kd	CGS001-578	BAK1	-			
2486	52.68	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
2487	52.68	kd	CGS001-9337	CNOT8	-			
2488	52.66	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
2489	52.66	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
2490	52.63	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
2491	52.63	oe	ccsbBroad304_02018	SUCLA2	-			
2492	52.6	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
2493	52.59	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
2494	52.57	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
2495	52.56	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
2496	52.53	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
2497	52.52	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
2498	52.44	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
2499	52.43	oe	ccsbBroad304_00171	BNIP3L	-			
2500	52.43	kd	CGS001-93134	ZNF561	Zinc fingers, C2H2-type			
2501	52.4	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
2502	52.38	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
2503	52.32	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
2504	52.31	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
2505	52.29	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
2506	52.27	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
2507	52.26	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
2508	52.24	kd	CGS001-8942	KYNU	-			
2509	52.24	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
2510	52.21	kd	CGS001-55176	SEC61A2	-			
2511	52.18	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
2512	52.05	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
2513	52.04	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
2514	52.03	kd	CGS001-808	CALM3	EF-hand domain containing			
2515	51.98	kd	CGS001-2172	FABP6	Fatty acid binding protein family			
2516	51.97	oe	ccsbBroad304_03951	NARFL	-			
2517	51.89	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
2518	51.87	kd	CGS001-4090	SMAD5	SMADs			
2519	51.85	kd	CGS001-5338	PLD2	Hydrolases			
2520	51.83	kd	CGS001-1072	CFL1	-			
2521	51.82	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
2522	51.82	kd	CGS001-6502	SKP2	F-boxes / Leucine-rich repeats			
2523	51.81	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
2524	51.77	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
2525	51.77	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
2526	51.76	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
2527	51.72	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
2528	51.71	cp	BRD-K63265447	docetaxel	Tubulin inhibitor		TUBB, BCL2, MAP2, MAP4, MAPT, NR1I2, TUBB1	Tubulin inhibitor
2529	51.71	oe	ccsbBroad304_05821	ANXA1	Annexins			
2530	51.68	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
2531	51.57	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
2532	51.56	kd	CGS001-5690	PSMB2	Proteasome subunits			
2533	51.56	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
2534	51.55	cp	BRD-K41903098	diphenoxylate	Opioid receptor agonist		OPRM1, OPRD1	Opioid receptor agonist
2535	51.55	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
2536	51.53	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
2537	51.52	kd	CGS001-23463	ICMT	-			
2538	51.52	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
2539	51.51	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
2540	51.49	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
2541	51.46	kd	CGS001-5966	REL	NFkappaB transcription factor family			
2542	51.45	kd	CGS001-80274	SCUBE1	-			
2543	51.42	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
2544	51.39	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
2545	51.38	kd	CGS001-4594	MUT	-			
2546	51.36	oe	ccsbBroad304_07280	LAMTOR3	-			
2547	51.34	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
2548	51.34	kd	CGS001-10482	NXF1	-			
2549	51.32	kd	CGS001-55082	ARGLU1	-			
2550	51.32	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
2551	51.32	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
2552	51.31	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
2553	51.3	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
2554	51.3	kd	CGS001-8453	CUL2	-			
2555	51.23	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
2556	51.22	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
2557	51.2	kd	CGS001-1305	COL13A1	Collagens			
2558	51.19	kd	CGS001-9183	ZW10	-			
2559	51.19	kd	CGS001-23076	RRP1B	-			
2560	51.18	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
2561	51.16	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
2562	51.14	kd	CGS001-3675	ITGA3	Integrins			
2563	51.13	kd	CGS001-10765	KDM5B	Histone demethylases			
2564	51.12	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
2565	51.06	cc		Glucocorticoid receptor agonist	-			
2566	51.03	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
2567	50.99	oe	ccsbBroad304_00423	DAXX	-			
2568	50.98	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
2569	50.94	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
2570	50.92	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
2571	50.91	oe	ccsbBroad304_03072	GTPBP8	-			
2572	50.89	cc		HIF activator	-			
2573	50.87	oe	ccsbBroad304_01205	PIN1	-			
2574	50.77	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
2575	50.75	oe	ccsbBroad304_06535	LPL	-			
2576	50.74	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
2577	50.64	kd	CGS001-10901	DHRS4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2578	50.64	kd	CGS001-688	KLF5	Kruppel-like transcription factors			
2579	50.63	kd	CGS001-4363	ABCC1	ATP binding cassette transporters / subfamily C			
2580	50.49	kd	CGS001-22891	ZNF365	Zinc fingers, C2H2-type			
2581	50.47	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
2582	50.45	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
2583	50.42	kd	CGS001-3980	LIG3	-			
2584	50.37	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
2585	50.33	kd	CGS001-55437	STRADB	STLK subfamily			
2586	50.32	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
2587	50.3	kd	CGS001-3601	IL15RA	IL-2 receptor family			
2588	50.27	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
2589	50.27	kd	CGS001-1635	DCTD	-			
2590	50.26	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
2591	50.26	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
2592	50.24	oe	ccsbBroad304_08645	BCCIP	-			
2593	50.2	kd	CGS001-51720	UIMC1	-			
2594	50.19	kd	CGS001-5062	PAK2	PAKA subfamily			
2595	50.17	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
2596	50.17	kd	CGS001-581	BAX	-			
2597	50.14	oe	ccsbBroad304_01787	YES1	Src family			
2598	50.11	kd	CGS001-6925	TCF4	Basic helix-loop-helix proteins			
2599	50.1	oe	ccsbBroad304_01257	PPOX	-			
2600	50.05	kd	CGS001-5564	PRKAB1	AMPK subfamily			
2601	49.98	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
2602	49.96	kd	CGS001-5373	PMM2	-			
2603	49.94	oe	ccsbBroad304_06665	OAT	-			
2604	49.94	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
2605	49.94	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
2606	49.93	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
2607	49.92	kd	CGS001-10475	TRIM38	-			
2608	49.91	oe	ccsbBroad304_03047	BZW2	-			
2609	49.91	kd	CGS001-9638	FEZ1	-			
2610	49.86	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
2611	49.85	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
2612	49.84	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
2613	49.82	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
2614	49.77	kd	CGS001-10452	TOMM40	-			
2615	49.76	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
2616	49.73	kd	CGS001-1211	CLTA	-			
2617	49.72	kd	CGS001-7168	TPM1	Tropomyosins			
2618	49.65	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
2619	49.65	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
2620	49.57	kd	CGS001-6720	SREBF1	Basic helix-loop-helix proteins			
2621	49.57	kd	CGS001-10489	LRRC41	-			
2622	49.53	kd	CGS001-10477	UBE2E3	Ubiquitin-conjugating enzymes E2			
2623	49.52	oe	ccsbBroad304_00648	GLRX	-			
2624	49.5	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
2625	49.46	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
2626	49.38	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
2627	49.36	kd	CGS001-9252	RPS6KA5	MSK subfamily			
2628	49.34	oe	ccsbBroad304_04788	OVCA2	-			
2629	49.31	kd	CGS001-7013	TERF1	-			
2630	49.28	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2631	49.27	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
2632	49.21	kd	CGS001-6723	SRM	-			
2633	49.2	kd	CGS001-1854	DUT	-			
2634	49.19	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
2635	49.18	cc		MTOR inhibitor	-			
2636	49.15	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
2637	49.13	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
2638	49.13	kd	CGS001-283450	C12ORF51	-			
2639	49.09	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
2640	49.07	oe	ccsbBroad304_00985	MCL1	-			
2641	49.05	kd	CGS001-55193	PBRM1	Non-enzymatic BRD containing proteins			
2642	49.02	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
2643	48.97	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
2644	48.96	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
2645	48.94	kd	CGS001-8870	IER3	-			
2646	48.94	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
2647	48.94	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
2648	48.93	oe	ccsbBroad304_03444	PAF1	-			
2649	48.93	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
2650	48.93	kd	CGS001-3419	IDH3A	-			
2651	48.92	oe	ccsbBroad304_05590	NOTCH2NL	-			
2652	48.92	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
2653	48.89	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
2654	48.79	kd	CGS001-9710	KIAA0355	-			
2655	48.77	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
2656	48.76	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
2657	48.74	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
2658	48.73	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
2659	48.72	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
2660	48.72	kd	CGS001-150094	SIK1	QIK subfamily			
2661	48.63	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
2662	48.62	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
2663	48.6	kd	CGS001-89765	RSPH1	-			
2664	48.57	kd	CGS001-2098	ESD	-			
2665	48.56	kd	CGS001-337867	UBAC2	-			
2666	48.41	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
2667	48.37	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
2668	48.37	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
2669	48.37	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
2670	48.33	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
2671	48.32	oe	ccsbBroad304_06324	GPX7	-			
2672	48.29	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
2673	48.28	kd	CGS001-7155	TOP2B	DNA Topoisomerases			
2674	48.24	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
2675	48.24	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
2676	48.23	oe	ccsbBroad304_02399	TNIP1	-			
2677	48.21	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
2678	48.2	kd	CGS001-7020	TFAP2A	-			
2679	48.19	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
2680	48.16	oe	ccsbBroad304_02002	RNMT	-			
2681	48.07	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
2682	48.06	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
2683	48.06	oe	ccsbBroad304_00112	ASNA1	-			
2684	48.01	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
2685	48	kd	CGS001-3065	HDAC1	Histone deacetylases			
2686	47.95	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
2687	47.93	kd	CGS001-56654	NPDC1	-			
2688	47.91	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
2689	47.91	kd	CGS001-1717	DHCR7	-			
2690	47.89	kd	CGS001-975	CD81	CD molecules			
2691	47.86	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
2692	47.83	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
2693	47.81	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2694	47.77	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
2695	47.76	kd	CGS001-23192	ATG4B	Aut2 peptidase			
2696	47.66	kd	CGS001-56882	CDC42SE1	-			
2697	47.66	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
2698	47.65	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2699	47.63	cp	BRD-K82147103	lofepramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
2700	47.56	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
2701	47.53	kd	CGS001-6788	STK3	MST subfamily			
2702	47.49	kd	CGS001-664	BNIP3	-			
2703	47.48	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
2704	47.45	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
2705	47.42	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
2706	47.38	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
2707	47.35	kd	CGS001-8233	ZRSR2	RNA binding motif (RRM) containing			
2708	47.35	kd	CGS001-1837	DTNA	-			
2709	47.34	cp	BRD-K82795137	loratadine	Histamine receptor antagonist		HRH1, CYP2C19, CYP3A5	Histamine receptor antagonist
2710	47.32	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
2711	47.28	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
2712	47.21	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
2713	47.19	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
2714	47.19	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
2715	47.18	kd	CGS001-2920	CXCL2	Endogenous ligands			
2716	47.13	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
2717	47.11	kd	CGS001-775	CACNA1C	Calcium channel subunits			
2718	47.1	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
2719	47.08	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
2720	47.03	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
2721	47	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
2722	46.99	kd	CGS001-29899	GPSM2	Tetratricopeptide (TTC) repeat domain containing			
2723	46.97	kd	CGS001-84333	PCGF5	Polycomb group ring fingers			
2724	46.95	oe	ccsbBroad304_01211	PKM2	-			
2725	46.95	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
2726	46.93	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
2727	46.93	kd	CGS001-9709	HERPUD1	-			
2728	46.92	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
2729	46.9	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
2730	46.86	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
2731	46.83	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
2732	46.8	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
2733	46.76	kd	CGS001-56139	PCDHA10	Cadherins / Protocadherins : Clustered			
2734	46.75	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
2735	46.74	kd	CGS001-210	ALAD	-			
2736	46.72	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
2737	46.68	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
2738	46.64	kd	CGS001-1869	E2F1	-			
2739	46.6	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
2740	46.59	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
2741	46.54	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
2742	46.47	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
2743	46.47	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
2744	46.44	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
2745	46.38	kd	CGS001-4172	MCM3	-			
2746	46.37	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
2747	46.35	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2748	46.34	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
2749	46.34	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
2750	46.3	kd	CGS001-10841	FTCD	-			
2751	46.29	kd	CGS001-23670	TMEM2	-			
2752	46.27	kd	CGS001-8495	PPFIBP2	Sterile alpha motif (SAM) domain containing			
2753	46.27	kd	CGS001-79581	GPR172A	-			
2754	46.25	kd	CGS001-5777	PTPN6	Protein tyrosine phosphatases			
2755	46.23	kd	CGS001-2876	GPX1	-			
2756	46.2	cp	BRD-K92870997	pterostilbene	Cyclooxygenase inhibitor		FAAH, PPARA, PTGS1, PTGS2	Cyclooxygenase inhibitor, PPAR receptor agonist
2757	46.19	oe	ccsbBroad304_06013	CLPTM1	-			
2758	46.19	kd	CGS001-11004	KIF2C	Kinesins			
2759	46.19	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
2760	46.14	kd	CGS001-8853	ASAP2	Ankyrin repeat domain containing			
2761	46.08	cp	BRD-A62890442	3-methyl-GABA	GABA aminotransferase activator			GABA aminotransferase activator
2762	46.04	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
2763	46.03	kd	CGS001-80306	MED28	-			
2764	46.03	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
2765	45.92	kd	CGS001-6197	RPS6KA3	RSK subfamily			
2766	45.92	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2767	45.91	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
2768	45.9	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
2769	45.87	kd	CGS001-7597	ZBTB25	BTB/POZ domain containing			
2770	45.85	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
2771	45.82	kd	CGS001-26039	SS18L1	-			
2772	45.78	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2773	45.76	kd	CGS001-6625	SNRNP70	RNA binding motif (RRM) containing			
2774	45.76	kd	CGS001-8624	PSMG1	-			
2775	45.75	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
2776	45.75	kd	CGS001-5108	PCM1	-			
2777	45.71	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
2778	45.71	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
2779	45.7	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
2780	45.69	kd	CGS001-661	POLR3D	RNA polymerase subunits			
2781	45.68	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
2782	45.68	kd	CGS001-5230	PGK1	-			
2783	45.66	kd	CGS001-10196	PRMT3	Protein arginine N-methyltransferases			
2784	45.63	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
2785	45.61	kd	CGS001-5571	PRKAG1	AMPK subfamily			
2786	45.59	cc		Sterol demethylase inhibitor	-			
2787	45.54	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
2788	45.52	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
2789	45.47	kd	CGS001-9643	MORF4L2	-			
2790	45.42	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
2791	45.37	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
2792	45.33	oe	ccsbBroad304_00430	GADD45A	-			
2793	45.33	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
2794	45.31	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
2795	45.3	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2796	45.28	kd	CGS001-285267	ZNF619	Zinc fingers, C2H2-type			
2797	45.28	kd	CGS001-25942	SIN3A	-			
2798	45.26	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
2799	45.25	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
2800	45.24	kd	CGS001-36	ACADSB	-			
2801	45.21	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2802	45.21	kd	CGS001-9500	MAGED1	-			
2803	45.2	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
2804	45.19	kd	CGS001-51222	ZNF219	Zinc fingers, C2H2-type			
2805	45.18	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
2806	45.18	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
2807	45.17	cp	BRD-K19462402	buflomedil	Adrenergic receptor antagonist		CACNA1C	Adrenergic receptor antagonist, Calcium channel blocker
2808	45.12	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
2809	45.04	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
2810	45.04	kd	CGS001-7263	TST	-			
2811	45.04	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
2812	45	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
2813	44.99	kd	CGS001-4129	MAOB	Catecholamine turnover			
2814	44.97	cp	BRD-K99063460	didanosine	Nucleoside reverse transcriptase inhibitor		PNP	Nucleoside reverse transcriptase inhibitor
2815	44.96	cp	BRD-K33312228	halometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2816	44.94	cc		AHSP Pathway LOF	-			
2817	44.94	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
2818	44.91	kd	CGS001-1066	CES1	Carboxylesterases			
2819	44.8	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
2820	44.78	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
2821	44.75	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
2822	44.73	oe	ccsbBroad304_07490	SCRN1	-			
2823	44.71	kd	CGS001-9589	WTAP	-			
2824	44.68	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
2825	44.66	kd	CGS001-5194	PEX13	-			
2826	44.63	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
2827	44.62	kd	CGS001-840	CASP7	Caspases			
2828	44.58	oe	ccsbBroad304_05135	PARP15	-			
2829	44.58	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
2830	44.51	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
2831	44.51	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
2832	44.44	kd	CGS001-10617	STAMBP	-			
2833	44.4	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
2834	44.4	kd	CGS001-54659	UGT1A3	UDP glucuronosyltransferases			
2835	44.39	oe	ccsbBroad304_05890	BHMT	-			
2836	44.38	oe	ccsbBroad304_06985	SORD	-			
2837	44.33	kd	CGS001-5567	PRKACB	Protein kinase A			
2838	44.3	kd	CGS001-6050	RNH1	-			
2839	44.21	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
2840	44.21	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
2841	44.21	oe	ccsbBroad304_13903	MTAP	-			
2842	44.2	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
2843	44.16	cp	BRD-K57930253	nitrazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, SCN1A	Benzodiazepine receptor agonist
2844	44.15	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
2845	44.15	oe	ccsbBroad304_02110	VAPB	-			
2846	44.14	kd	CGS001-472	ATM	Other PIKK family kinases			
2847	44.14	kd	CGS001-572	BAD	-			
2848	44.13	kd	CGS001-2072	ERCC4	-			
2849	44.07	kd	CGS001-7846	TUBA1A	Tubulins			
2850	43.99	cc		Kinase anchoring proteins LOF	-			
2851	43.99	cp	BRD-K93618743	ipriflavone	Bone resorption inhibitor			Bone resorption inhibitor
2852	43.98	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
2853	43.94	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
2854	43.85	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
2855	43.83	kd	CGS001-24138	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
2856	43.81	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
2857	43.79	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
2858	43.79	kd	CGS001-64710	NUCKS1	-			
2859	43.76	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
2860	43.75	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
2861	43.75	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
2862	43.73	kd	CGS001-3177	SLC29A2	SLC29 family			
2863	43.72	kd	CGS001-8464	SUPT3H	-			
2864	43.69	kd	CGS001-9612	NCOR2	-			
2865	43.69	kd	CGS001-1605	DAG1	-			
2866	43.67	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
2867	43.65	kd	CGS001-8797	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
2868	43.58	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
2869	43.57	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2870	43.56	kd	CGS001-328	APEX1	-			
2871	43.51	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
2872	43.45	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
2873	43.44	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
2874	43.41	oe	ccsbBroad304_01632	SYPL1	-			
2875	43.37	kd	CGS001-9738	CCP110	-			
2876	43.37	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
2877	43.35	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
2878	43.35	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
2879	43.34	kd	CGS001-83439	TCF7L1	-			
2880	43.32	kd	CGS001-4947	OAZ2	-			
2881	43.29	kd	CGS001-133522	PPARGC1B	RNA binding motif (RRM) containing			
2882	43.23	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
2883	43.17	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
2884	43.15	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
2885	43.15	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
2886	43.11	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
2887	43.1	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
2888	43.1	kd	CGS001-6988	TCTA	-			
2889	43.06	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
2890	43.04	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
2891	43.03	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
2892	43.03	kd	CGS001-23636	NUP62	-			
2893	42.99	kd	CGS001-5875	RABGGTA	Prenyltransferase alpha subunit repeat containing			
2894	42.98	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
2895	42.97	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
2896	42.91	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
2897	42.85	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
2898	42.84	oe	ccsbBroad304_06711	PFAS	-			
2899	42.82	cc		PARP inhibitor	-			
2900	42.8	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
2901	42.8	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
2902	42.79	kd	CGS001-8850	KAT2B	Histone acetyltransferases (HATs)			
2903	42.78	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
2904	42.78	oe	ccsbBroad304_03604	ENOSF1	-			
2905	42.77	oe	ccsbBroad304_02057	P4HA2	-			
2906	42.77	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
2907	42.74	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
2908	42.74	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
2909	42.72	kd	CGS001-1001	CDH3	Cadherins / Major cadherins			
2910	42.72	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
2911	42.67	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
2912	42.65	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
2913	42.61	kd	CGS001-3560	IL2RB	IL-2 receptor family			
2914	42.52	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
2915	42.5	kd	CGS001-6464	SHC1	SH2 domain containing			
2916	42.49	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
2917	42.44	cc		Dihydrofolate reductase inhibitor	-			
2918	42.43	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
2919	42.38	oe	ccsbBroad304_07688	FAM114A2	-			
2920	42.35	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
2921	42.35	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
2922	42.31	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2923	42.3	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
2924	42.29	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
2925	42.18	kd	CGS001-7345	UCHL1	Ubiquitin C-terminal hydrolase			
2926	42.15	cp	BRD-A23637604	oxymetholone	Androgen receptor agonist		AR	Androgen receptor agonist
2927	42.13	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
2928	42.12	kd	CGS001-8061	FOSL1	basic leucine zipper proteins			
2929	42.1	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
2930	42.04	cc		RAF inhibitor	-			
2931	42.03	kd	CGS001-2710	GK	Glycerol kinases			
2932	42.01	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
2933	41.99	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2934	41.96	kd	CGS001-81577	GFOD2	-			
2935	41.94	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
2936	41.94	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
2937	41.94	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
2938	41.91	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
2939	41.88	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
2940	41.87	kd	CGS001-10202	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2941	41.82	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
2942	41.81	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
2943	41.8	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
2944	41.8	oe	ccsbBroad304_01019	MLH1	-			
2945	41.76	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2946	41.74	kd	CGS001-10538	BATF	basic leucine zipper proteins			
2947	41.68	cp	BRD-K34508425	KUC103898N	-666			-666
2948	41.68	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
2949	41.66	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
2950	41.64	kd	CGS001-7360	UGP2	-			
2951	41.63	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
2952	41.63	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
2953	41.62	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
2954	41.57	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
2955	41.56	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
2956	41.53	kd	CGS001-124535	HSF5	-			
2957	41.51	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
2958	41.5	cc		Leucine rich repeat kinase inhibitor	-			
2959	41.48	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
2960	41.46	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
2961	41.42	kd	CGS001-54681	P4HTM	-			
2962	41.4	kd	CGS001-5993	RFX5	-			
2963	41.37	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
2964	41.35	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
2965	41.34	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
2966	41.34	kd	CGS001-10257	ABCC4	ATP binding cassette transporters / subfamily C			
2967	41.33	oe	ccsbBroad304_09833	SENP5	-			
2968	41.31	oe	ccsbBroad304_03773	CIAPIN1	-			
2969	41.3	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
2970	41.28	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
2971	41.27	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
2972	41.26	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
2973	41.23	oe	ccsbBroad304_02270	FAM20B	-			
2974	41.23	kd	CGS001-10014	HDAC5	Histone deacetylases			
2975	41.17	kd	CGS001-4200	ME2	-			
2976	41.17	kd	CGS001-2077	ERF	ETS Transcription Factors			
2977	41.16	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
2978	41.15	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
2979	41.15	kd	CGS001-4712	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
2980	41.14	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
2981	41.12	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
2982	41.08	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
2983	41.06	kd	CGS001-6714	SRC	Src family			
2984	41.05	kd	CGS001-3998	LMAN1	-			
2985	41.01	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
2986	41.01	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
2987	41	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
2988	40.97	kd	CGS001-4548	MTR	-			
2989	40.96	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
2990	40.95	oe	ccsbBroad304_00221	CASP3	Caspases			
2991	40.91	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
2992	40.89	kd	CGS001-54512	EXOSC4	-			
2993	40.89	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
2994	40.85	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
2995	40.84	cc		Nucleoside reverse transcriptase inhibitor	-			
2996	40.84	kd	CGS001-1643	DDB2	WD repeat domain containing			
2997	40.81	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
2998	40.79	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
2999	40.74	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3000	40.72	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
3001	40.7	kd	CGS001-22949	PTGR1	-			
3002	40.67	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
3003	40.58	kd	CGS001-2565	GABRG1	GABA receptors			
3004	40.58	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
3005	40.55	kd	CGS001-64319	FBRS	-			
3006	40.54	kd	CGS001-7276	TTR	-			
3007	40.52	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
3008	40.5	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
3009	40.48	kd	CGS001-5054	SERPINE1	Serine (or cysteine) peptidase inhibitors			
3010	40.46	oe	ccsbBroad304_06140	EEF1D	-			
3011	40.45	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
3012	40.41	oe	ccsbBroad304_02086	PDLIM1	-			
3013	40.39	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
3014	40.35	kd	CGS001-10494	STK25	YSK subfamily			
3015	40.32	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
3016	40.31	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
3017	40.31	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
3018	40.3	cp	BRD-K85030058	benactyzine	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
3019	40.16	oe	ccsbBroad304_00709	GUK1	-			
3020	40.16	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
3021	40.16	kd	CGS001-11162	NUDT6	Nudix motif containing			
3022	40.14	cp	BRD-K55034111	pefloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
3023	40.08	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
3024	40.07	kd	CGS001-2639	GCDH	-			
3025	40.01	kd	CGS001-53834	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
3026	39.96	kd	CGS001-7862	BRPF1	Non-enzymatic BRD containing proteins			
3027	39.9	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
3028	39.9	kd	CGS001-7295	TXN	-			
3029	39.9	kd	CGS001-2023	ENO1	-			
3030	39.85	kd	CGS001-54732	TMED9	-			
3031	39.83	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
3032	39.79	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
3033	39.78	oe	ccsbBroad304_08116	TBK1	IKK family			
3034	39.76	kd	CGS001-3169	FOXA1	Forkhead boxes			
3035	39.74	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
3036	39.74	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3037	39.7	kd	CGS001-2963	GTF2F2	General transcription factors			
3038	39.69	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
3039	39.67	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
3040	39.66	kd	CGS001-5053	PAH	Amino acid hydroxylases			
3041	39.61	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
3042	39.61	kd	CGS001-4893	NRAS	RAS subfamily			
3043	39.59	kd	CGS001-4122	MAN2A2	-			
3044	39.58	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
3045	39.58	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
3046	39.53	cp	BRD-K73991644	isoquercetin	Aldose reductase inhibitor		AKR1B1, ACE	Aldose reductase inhibitor
3047	39.52	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
3048	39.51	kd	CGS001-5306	PITPNA	-			
3049	39.51	oe	ccsbBroad304_00650	GNA11	-			
3050	39.46	kd	CGS001-2731	GLDC	-			
3051	39.42	kd	CGS001-51495	PTPLAD1	-			
3052	39.41	oe	ccsbBroad304_14242	MCCC2	-			
3053	39.34	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
3054	39.32	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
3055	39.32	oe	ccsbBroad304_00359	CPT1A	-			
3056	39.31	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
3057	39.3	oe	ccsbBroad304_02534	UTP14A	-			
3058	39.3	kd	CGS001-3034	HAL	-			
3059	39.28	cc		DNA Replication LOF	-			
3060	39.27	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
3061	39.25	kd	CGS001-9552	SPAG7	-			
3062	39.24	kd	CGS001-8312	AXIN1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3063	39.23	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
3064	39.21	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
3065	39.2	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
3066	39.19	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
3067	39.19	kd	CGS001-5909	RAP1GAP	-			
3068	39.15	oe	ccsbBroad304_08346	COQ3	-			
3069	39.12	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
3070	39.11	cc		Progesterone receptor agonist	-			
3071	39.11	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
3072	39.08	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
3073	39.08	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
3074	39.08	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
3075	39.03	oe	ccsbBroad304_03164	MTERFD1	-			
3076	38.98	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3077	38.97	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
3078	38.92	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
3079	38.9	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
3080	38.9	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
3081	38.89	kd	CGS001-26227	PHGDH	-			
3082	38.84	cp	BRD-K06878038	deferiprone	Chelating agent		CYP4F2	Chelating agent
3083	38.82	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
3084	38.81	kd	CGS001-23344	ESYT1	Synaptotagmins			
3085	38.81	kd	CGS001-22905	EPN2	-			
3086	38.81	kd	CGS001-102	ADAM10	ADAM metallopeptidase domain containing			
3087	38.65	oe	ccsbBroad304_08775	SQRDL	-			
3088	38.61	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
3089	38.61	kd	CGS001-26128	KIAA1279	-			
3090	38.56	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
3091	38.55	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
3092	38.52	kd	CGS001-3609	ILF3	-			
3093	38.5	kd	CGS001-63948	DMRTB1	-			
3094	38.48	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3095	38.47	kd	CGS001-84617	TUBB6	Tubulins			
3096	38.45	cp	BRD-A20589515	dihydroxyphenylglycine	Glutamate receptor agonist		GRM1	Glutamate receptor agonist
3097	38.44	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
3098	38.4	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
3099	38.38	cp	BRD-K48932581	cetraxate	Mucus protecting agent		GAST	Mucus protecting agent
3100	38.38	kd	CGS001-1633	DCK	-			
3101	38.36	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
3102	38.36	kd	CGS001-388650	FAM69A	-			
3103	38.34	kd	CGS001-80758	PRR7	-			
3104	38.32	kd	CGS001-1725	DHPS	-			
3105	38.31	kd	CGS001-54677	CROT	-			
3106	38.3	kd	CGS001-121599	SPIC	ETS Transcription Factors			
3107	38.29	oe	ccsbBroad304_06382	HMGCL	-			
3108	38.22	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
3109	38.21	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
3110	38.21	kd	CGS001-9900	SV2A	Major facilitator superfamily (MFS) of transporters			
3111	38.17	kd	CGS001-9512	PMPCB	-			
3112	38.16	kd	CGS001-10253	SPRY2	-			
3113	38.16	kd	CGS001-8505	PARG	-			
3114	38.16	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
3115	38.12	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
3116	38.1	kd	CGS001-29890	RBM15B	RNA binding motif (RRM) containing			
3117	38.08	oe	ccsbBroad304_00469	DUT	-			
3118	38.06	oe	ccsbBroad304_04257	SPRY4	-			
3119	38.06	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
3120	38.06	kd	CGS001-527	ATP6V0C	ATPases / V-type			
3121	38.05	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
3122	38.04	kd	CGS001-9156	EXO1	-			
3123	38.01	kd	CGS001-64376	IKZF5	IKAROS zinc fingers			
3124	37.97	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
3125	37.96	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
3126	37.83	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
3127	37.82	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
3128	37.82	kd	CGS001-11168	PSIP1	-			
3129	37.78	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
3130	37.74	oe	ccsbBroad304_01519	SET	-			
3131	37.72	oe	ccsbBroad304_03878	SENP2	-			
3132	37.72	oe	ccsbBroad304_00101	RHOC	-			
3133	37.68	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
3134	37.62	cc		Gamma secretase inhibitor	-			
3135	37.61	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
3136	37.46	cc		Beta-adrenergic receptor agonist	-			
3137	37.41	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
3138	37.37	oe	ccsbBroad304_00376	CSK	Csk family			
3139	37.35	kd	CGS001-126208	ZNF787	Zinc fingers, C2H2-type			
3140	37.33	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
3141	37.31	kd	CGS001-9181	ARHGEF2	Rho guanine nucleotide exchange factors			
3142	37.29	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
3143	37.28	oe	ccsbBroad304_07017	SUOX	-			
3144	37.23	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
3145	37.23	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
3146	37.2	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
3147	37.17	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
3148	37.15	kd	CGS001-9232	PTTG1	-			
3149	37.15	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
3150	37.11	kd	CGS001-9326	ZNHIT3	Zinc fingers, HIT-type			
3151	37.1	kd	CGS001-10020	GNE	-			
3152	37.07	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
3153	37.06	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
3154	37.06	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3155	37.05	kd	CGS001-1465	CSRP1	-			
3156	37.03	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
3157	37.03	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3158	37.02	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
3159	36.97	kd	CGS001-4282	MIF	-			
3160	36.94	kd	CGS001-23067	SETD1B	Histone methyltransferases (HMTs)			
3161	36.93	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
3162	36.89	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
3163	36.84	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
3164	36.82	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
3165	36.79	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
3166	36.76	cp	BRD-A52282606	lacidipine	Calcium channel blocker		CACNA1C	Calcium channel blocker
3167	36.76	kd	CGS001-5577	PRKAR2B	Protein kinase A			
3168	36.74	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
3169	36.72	kd	CGS001-439	ASNA1	-			
3170	36.71	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
3171	36.68	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
3172	36.67	kd	CGS001-8720	MBTPS1	Subtilisin			
3173	36.67	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
3174	36.66	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
3175	36.65	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
3176	36.65	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
3177	36.63	kd	CGS001-28512	NKIRAS1	-			
3178	36.62	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
3179	36.61	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
3180	36.6	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
3181	36.6	kd	CGS001-10795	ZNF268	Zinc fingers, C2H2-type			
3182	36.58	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
3183	36.56	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
3184	36.55	oe	ccsbBroad304_02425	CDIPT	-			
3185	36.55	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
3186	36.47	kd	CGS001-7029	TFDP2	-			
3187	36.44	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
3188	36.44	kd	CGS001-805	CALM2	EF-hand domain containing			
3189	36.43	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
3190	36.41	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
3191	36.4	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
3192	36.4	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
3193	36.34	cc		HRH1 antagonist	-			
3194	36.34	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
3195	36.32	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
3196	36.31	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
3197	36.26	cp	BRD-K44353683	nateglinide	Insulin secretagogue		ABCC8, KCNJ11, CYP3A4, INS, KCNJ10, PPARG	Insulin secretagogue
3198	36.22	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
3199	36.22	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
3200	36.22	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
3201	36.2	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
3202	36.18	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
3203	36.15	oe	ccsbBroad304_04471	C5ORF62	-			
3204	36.11	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
3205	36.08	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
3206	36.05	oe	ccsbBroad304_00532	F11	Chymotrypsin			
3207	36.05	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
3208	36.03	kd	CGS001-28511	NKIRAS2	-			
3209	36	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
3210	35.99	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
3211	35.98	kd	CGS001-2932	GSK3B	GSK subfamily			
3212	35.97	oe	ccsbBroad304_06820	PTS	-			
3213	35.94	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
3214	35.92	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
3215	35.92	oe	ccsbBroad304_02026	NRP1	CD molecules			
3216	35.91	oe	ccsbBroad304_08898	TRAK2	-			
3217	35.82	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3218	35.8	kd	CGS001-8644	AKR1C3	Prostaglandin synthases			
3219	35.79	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
3220	35.79	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
3221	35.77	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
3222	35.7	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
3223	35.7	kd	CGS001-6304	SATB1	Homeoboxes / CUT class			
3224	35.66	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
3225	35.64	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
3226	35.61	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
3227	35.61	kd	CGS001-467	ATF3	basic leucine zipper proteins			
3228	35.58	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
3229	35.58	kd	CGS001-6924	TCEB3	-			
3230	35.58	kd	CGS001-29959	NRBP1	NRBP family			
3231	35.55	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
3232	35.5	kd	CGS001-7108	TM7SF2	-			
3233	35.47	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
3234	35.44	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
3235	35.41	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
3236	35.31	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
3237	35.31	kd	CGS001-1984	EIF5A	-			
3238	35.26	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
3239	35.22	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
3240	35.21	kd	CGS001-11257	TP53TG1	-			
3241	35.17	oe	ccsbBroad304_03565	ADI1	-			
3242	35.14	kd	CGS001-8896	BUD31	-			
3243	35.13	kd	CGS001-389421	LIN28B	-			
3244	35.12	kd	CGS001-10444	ZER1	ZYG11 cell cycle regulator family			
3245	35.11	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
3246	35.11	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
3247	35.1	kd	CGS001-5550	PREP	Prolyl oligopeptidase			
3248	35.03	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
3249	35.02	kd	CGS001-6207	RPS13	S ribosomal proteins			
3250	35.01	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
3251	35.01	kd	CGS001-27125	AFF4	-			
3252	35	kd	CGS001-9897	KIAA0196	-			
3253	34.98	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
3254	34.97	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
3255	34.95	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
3256	34.94	kd	CGS001-1606	DGKA	EF-hand domain containing			
3257	34.9	kd	CGS001-1051	CEBPB	basic leucine zipper proteins			
3258	34.86	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
3259	34.82	kd	CGS001-1737	DLAT	-			
3260	34.71	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
3261	34.7	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
3262	34.7	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
3263	34.66	cc		IKK inhibitor	-			
3264	34.65	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
3265	34.64	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
3266	34.64	kd	CGS001-2931	GSK3A	GSK subfamily			
3267	34.63	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
3268	34.63	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3269	34.61	cc		BCL inhibitor	-			
3270	34.6	kd	CGS001-2048	EPHB2	Type XIII RTKs: Ephrin receptor family			
3271	34.57	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
3272	34.56	kd	CGS001-25925	ZNF521	Zinc fingers, C2H2-type			
3273	34.52	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
3274	34.51	kd	CGS001-51520	LARS	Aminoacyl tRNA synthetases / Class I			
3275	34.49	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
3276	34.47	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
3277	34.44	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
3278	34.43	kd	CGS001-8503	PIK3R3	Phosphatidylinositol kinases			
3279	34.43	kd	CGS001-1460	CSNK2B	Casein kinase 2 (CK2) family			
3280	34.42	kd	CGS001-9770	RASSF2	-			
3281	34.39	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
3282	34.37	oe	ccsbBroad304_01976	EIF4EBP3	-			
3283	34.31	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
3284	34.3	oe	ccsbBroad304_00183	C1S	Complement system			
3285	34.29	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
3286	34.22	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
3287	34.15	kd	CGS001-8826	IQGAP1	-			
3288	34.14	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
3289	34.12	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
3290	34.12	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
3291	34.12	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
3292	34.07	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
3293	34.06	kd	CGS001-10919	EHMT2	Histone methyltransferases			
3294	34.06	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
3295	34.04	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
3296	34.02	kd	CGS001-7374	UNG	-			
3297	34.01	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
3298	34	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
3299	34	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
3300	33.94	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
3301	33.91	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
3302	33.83	kd	CGS001-5019	OXCT1	-			
3303	33.83	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
3304	33.78	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
3305	33.76	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
3306	33.74	kd	CGS001-2015	EMR1	Adhesion Class GPCRs			
3307	33.74	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
3308	33.69	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
3309	33.66	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
3310	33.65	kd	CGS001-23239	PHLPP1	Pleckstrin homology (PH) domain containing			
3311	33.64	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3312	33.58	kd	CGS001-7832	BTG2	-			
3313	33.57	oe	ccsbBroad304_03056	MCTS1	-			
3314	33.56	oe	ccsbBroad304_02653	PRAF2	-			
3315	33.54	kd	CGS001-6822	SULT2A1	Sulfotransferases, cytosolic			
3316	33.51	kd	CGS001-635	BHMT	-			
3317	33.49	oe	ccsbBroad304_07080	TM7SF2	-			
3318	33.42	kd	CGS001-3053	SERPIND1	Serine (or cysteine) peptidase inhibitors			
3319	33.4	kd	CGS001-2235	FECH	-			
3320	33.38	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
3321	33.36	kd	CGS001-148103	ZNF599	Zinc fingers, C2H2-type			
3322	33.34	kd	CGS001-3149	HMGB3	High-mobility group / Canonical			
3323	33.28	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
3324	33.28	kd	CGS001-203	AK1	Adenylate kinases			
3325	33.26	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
3326	33.23	kd	CGS001-817	CAMK2D	CAMK2 family			
3327	33.14	kd	CGS001-6709	SPTAN1	EF-hand domain containing			
3328	33.09	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
3329	33.08	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
3330	33.08	kd	CGS001-84775	ZNF607	Zinc fingers, C2H2-type			
3331	33.08	kd	CGS001-4773	NFATC2	Nuclear factor of activated T-cells			
3332	33.07	oe	ccsbBroad304_01150	PCCB	Carboxylases			
3333	33.06	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
3334	33.06	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
3335	33.04	kd	CGS001-3123	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
3336	33.02	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3337	32.99	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
3338	32.99	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
3339	32.99	kd	CGS001-6885	MAP3K7	MAPKKK:TAK1 subfamily			
3340	32.99	kd	CGS001-51026	GOLT1B	-			
3341	32.98	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
3342	32.97	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
3343	32.96	kd	CGS001-55191	NADSYN1	-			
3344	32.95	kd	CGS001-8895	CPNE3	-			
3345	32.91	kd	CGS001-80237	ELL3	-			
3346	32.91	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
3347	32.9	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
3348	32.87	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
3349	32.86	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
3350	32.85	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
3351	32.73	kd	CGS001-10891	PPARGC1A	RNA binding motif (RRM) containing			
3352	32.7	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
3353	32.7	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
3354	32.62	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
3355	32.61	kd	CGS001-4012	LNPEP	Aminopeptidase N			
3356	32.6	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
3357	32.59	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3358	32.56	kd	CGS001-93594	WDR67	-			
3359	32.55	kd	CGS001-8655	DYNLL1	Cytoplasmic dyneins			
3360	32.54	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3361	32.53	kd	CGS001-22894	DIS3	-			
3362	32.53	oe	ccsbBroad304_07920	NUP62	-			
3363	32.49	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
3364	32.43	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
3365	32.4	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
3366	32.39	kd	CGS001-5618	PRLR	Prolactin receptor family			
3367	32.38	kd	CGS001-9143	SYNGR3	-			
3368	32.36	kd	CGS001-558	AXL	Fibronectin type III domain containing			
3369	32.33	oe	ccsbBroad304_00626	GDI1	-			
3370	32.33	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
3371	32.32	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3372	32.3	cp	BRD-A35519318	benidipine	Calcium channel blocker		CACNA1C, CACNA1G, CYP3A5	Calcium channel blocker
3373	32.3	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
3374	32.28	kd	CGS001-169792	GLIS3	Zinc fingers, C2H2-type			
3375	32.27	kd	CGS001-5914	RARA	Retinoic acid receptors			
3376	32.24	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
3377	32.23	kd	CGS001-4638	MYLK	Myosin Light Chain Kinase (MLCK) family			
3378	32.17	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
3379	32.17	kd	CGS001-5901	RAN	-			
3380	32.12	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
3381	32.11	kd	CGS001-7077	TIMP2	-			
3382	32.11	oe	ccsbBroad304_00174	BRAF	RAF family			
3383	32.09	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
3384	32.07	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
3385	32.07	kd	CGS001-4074	M6PR	-			
3386	32.07	kd	CGS001-25948	KBTBD2	BTB/POZ domain containing			
3387	32.04	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
3388	32.03	kd	CGS001-10312	TCIRG1	ATPases / V-type			
3389	32.03	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
3390	32.03	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
3391	32.02	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
3392	32.02	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
3393	32	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
3394	31.99	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
3395	31.96	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
3396	31.93	oe	ccsbBroad304_00644	GCLC	-			
3397	31.89	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
3398	31.89	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
3399	31.83	cp	BRD-K46435977	valaciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
3400	31.81	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
3401	31.79	oe	ccsbBroad304_01672	TIMP2	-			
3402	31.77	oe	ccsbBroad304_03311	EVL	-			
3403	31.75	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
3404	31.71	cp	BRD-K44094599	tacrolimus	Calcineurin inhibitor		FKBP1A, CYP3A5, CYP3A7	Calcineurin inhibitor
3405	31.69	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
3406	31.65	kd	CGS001-5860	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
3407	31.59	kd	CGS001-54556	ING3	Zinc fingers, PHD-type			
3408	31.59	kd	CGS001-9034	CCRL2	Chemokine receptors			
3409	31.58	kd	CGS001-2495	FTH1	-			
3410	31.57	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
3411	31.56	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
3412	31.55	kd	CGS001-1119	CHKA	-			
3413	31.55	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
3414	31.52	oe	ccsbBroad304_05887	CFB	Complement system			
3415	31.5	kd	CGS001-1173	AP2M1	-			
3416	31.49	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
3417	31.48	kd	CGS001-57019	CIAPIN1	-			
3418	31.46	oe	ccsbBroad304_06975	SMARCC2	-			
3419	31.44	oe	ccsbBroad304_12226	NAGK	-			
3420	31.4	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
3421	31.37	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
3422	31.36	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
3423	31.36	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
3424	31.35	kd	CGS001-7001	PRDX2	-			
3425	31.33	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
3426	31.32	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
3427	31.28	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
3428	31.28	cp	BRD-A64297288	amlodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, ABCG2, CA1, CACNA1B, CACNA1S, CACNA2D3, CACNB1, CACNB2, SMPD1	Calcium channel blocker
3429	31.24	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
3430	31.18	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
3431	31.15	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
3432	31.14	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
3433	31.13	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
3434	31.1	kd	CGS001-29763	PACSIN3	-			
3435	31.09	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
3436	31.08	oe	ccsbBroad304_00164	BLMH	-			
3437	31.04	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
3438	31.02	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
3439	31.02	cp	BRD-K88304388	dextrorphan	Glutamate receptor antagonist		OPRM1, OPRK1, OPRD1, GRIN1, HTR1A, SLC6A2	Glutamate receptor antagonist
3440	31.01	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3441	31	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
3442	30.99	kd	CGS001-6757	SSX2	-			
3443	30.94	kd	CGS001-27347	STK39	FRAY subfamily			
3444	30.92	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
3445	30.91	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
3446	30.91	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
3447	30.91	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
3448	30.89	oe	ccsbBroad304_05980	CDKN1B	-			
3449	30.87	cc		NFkB pathway inhibitor	-			
3450	30.86	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
3451	30.85	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
3452	30.85	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
3453	30.84	oe	ccsbBroad304_01052	MYB	-			
3454	30.84	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
3455	30.82	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
3456	30.8	kd	CGS001-670	BPHL	-			
3457	30.79	kd	CGS001-23210	JMJD6	-			
3458	30.77	cc		Non Homologous End Joining LOF	-			
3459	30.72	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
3460	30.71	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
3461	30.7	kd	CGS001-3131	HLF	-			
3462	30.65	kd	CGS001-51547	SIRT7	Histone deacetylases (HDACs)			
3463	30.64	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
3464	30.63	kd	CGS001-285676	ZNF454	Zinc fingers, C2H2-type			
3465	30.59	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
3466	30.57	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
3467	30.57	kd	CGS001-4864	NPC1	-			
3468	30.55	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
3469	30.54	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
3470	30.5	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
3471	30.48	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
3472	30.46	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
3473	30.46	oe	ccsbBroad304_06523	LIG1	-			
3474	30.44	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
3475	30.44	kd	CGS001-1376	CPT2	-			
3476	30.42	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
3477	30.39	kd	CGS001-6591	SNAI2	Snail homologs			
3478	30.37	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
3479	30.37	kd	CGS001-10493	VAT1	-			
3480	30.37	kd	CGS001-79135	APOO	Apolipoproteins			
3481	30.33	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
3482	30.32	kd	CGS001-257397	TAB3	-			
3483	30.31	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
3484	30.31	kd	CGS001-57657	HCN3	Cyclic nucleotide-regulated channels			
3485	30.3	kd	CGS001-23650	TRIM29	-			
3486	30.28	kd	CGS001-91949	COG7	Components of oligomeric golgi complex			
3487	30.26	oe	ccsbBroad304_03848	METTL14	-			
3488	30.26	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
3489	30.22	oe	ccsbBroad304_00632	GGCX	Carboxylases			
3490	30.19	kd	CGS001-125919	ZNF543	Zinc fingers, C2H2-type			
3491	30.19	oe	ccsbBroad304_02205	WTAP	-			
3492	30.11	kd	CGS001-2079	ERH	-			
3493	30.08	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
3494	30.05	kd	CGS001-3485	IGFBP2	insulin-like growth factor (IGF) binding proteins			
3495	30.03	kd	CGS001-2254	FGF9	Endogenous ligands			
3496	30.02	kd	CGS001-114609	TIRAP	-			
3497	30	kd	CGS001-597	BCL2A1	-			
3498	30	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
3499	29.98	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
3500	29.95	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
3501	29.93	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
3502	29.9	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
3503	29.89	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
3504	29.89	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
3505	29.88	kd	CGS001-25989	ULK3	Unc-51-like kinase (ULK) family			
3506	29.88	kd	CGS001-23271	CAMSAP2	-			
3507	29.85	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
3508	29.82	cp	BRD-K15916496	clotrimazole	Cytochrome P450 inhibitor		KCNN4, CYP3A4, CYP51A1, NR1I2, NR1I3, TRPM2, TRPM4, TRPM8	Cytochrome P450 inhibitor, Imidazoline receptor ligand
3509	29.76	kd	CGS001-6621	SNAPC4	-			
3510	29.72	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
3511	29.71	oe	ccsbBroad304_06565	MB	-			
3512	29.71	kd	CGS001-7039	TGFA	-			
3513	29.7	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
3514	29.66	oe	ccsbBroad304_07178	ZFP112	-			
3515	29.65	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
3516	29.65	kd	CGS001-57007	CXCR7	-			
3517	29.64	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
3518	29.64	oe	ccsbBroad304_02990	LYPD3	-			
3519	29.63	kd	CGS001-9290	GPR55	GPCR / Class A : Orphans			
3520	29.58	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
3521	29.55	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3522	29.55	kd	CGS001-54442	KCTD5	-			
3523	29.52	kd	CGS001-3281	HSBP1	-			
3524	29.51	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
3525	29.5	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
3526	29.49	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
3527	29.49	kd	CGS001-1827	RCAN1	-			
3528	29.49	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
3529	29.49	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3530	29.48	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
3531	29.46	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
3532	29.44	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
3533	29.39	kd	CGS001-51031	GLOD4	-			
3534	29.39	kd	CGS001-1209	CLPTM1	-			
3535	29.38	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
3536	29.33	kd	CGS001-6282	S100A11	EF-hand domain containing			
3537	29.31	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
3538	29.28	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
3539	29.25	oe	ccsbBroad304_01576	SOAT1	-			
3540	29.24	kd	CGS001-51182	HSPA14	Heat shock proteins / HSP70			
3541	29.23	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
3542	29.23	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
3543	29.21	kd	CGS001-4175	MCM6	-			
3544	29.19	kd	CGS001-8833	GMPS	-			
3545	29.16	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
3546	29.13	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
3547	29.12	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
3548	29.09	kd	CGS001-5467	PPARD	Nuclear hormone receptors			
3549	29.08	kd	CGS001-27109	ATP5S	-			
3550	29.04	kd	CGS001-6608	SMO	GPCR / Class F : Frizzled receptors			
3551	29.01	kd	CGS001-9688	NUP93	-			
3552	29.01	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
3553	29	kd	CGS001-727	C5	Endogenous ligands			
3554	28.99	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
3555	28.94	kd	CGS001-55662	HIF1AN	-			
3556	28.93	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
3557	28.93	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
3558	28.92	kd	CGS001-9767	PHF16	-			
3559	28.91	kd	CGS001-5581	PRKCE	Eta subfamily			
3560	28.89	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
3561	28.83	oe	ccsbBroad304_00854	IL8	-			
3562	28.83	kd	CGS001-5134	PDCD2	Zinc fingers, MYND-type			
3563	28.79	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
3564	28.77	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3565	28.77	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
3566	28.69	kd	CGS001-11331	PHB2	-			
3567	28.69	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
3568	28.67	oe	ccsbBroad304_02313	ACTR3	-			
3569	28.6	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
3570	28.59	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
3571	28.57	kd	CGS001-3566	IL4R	IL-2 receptor family			
3572	28.54	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
3573	28.47	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
3574	28.46	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
3575	28.45	kd	CGS001-2887	GRB10	Pleckstrin homology (PH) domain containing			
3576	28.43	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
3577	28.43	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
3578	28.42	kd	CGS001-55129	ANO10	Calcium activated chloride channel			
3579	28.41	cp	BRD-K90733503	cefalexin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3580	28.4	kd	CGS001-11129	CLASRP	-			
3581	28.4	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3582	28.39	oe	ccsbBroad304_00239	CCNG1	-			
3583	28.37	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
3584	28.36	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
3585	28.33	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3586	28.32	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
3587	28.3	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
3588	28.25	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
3589	28.25	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
3590	28.24	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
3591	28.23	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
3592	28.22	kd	CGS001-64858	DCLRE1B	-			
3593	28.19	kd	CGS001-84515	MCM8	-			
3594	28.19	kd	CGS001-8535	CBX4	-			
3595	28.16	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
3596	28.14	oe	ccsbBroad304_00795	HSF2	-			
3597	28.13	kd	CGS001-5664	PSEN2	Presenilin			
3598	28.11	kd	CGS001-2773	GNAI3	-			
3599	28.1	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
3600	28.09	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
3601	28.06	kd	CGS001-57787	MARK4	MARK subfamily			
3602	28.06	kd	CGS001-2674	GFRA1	GDNF receptor family			
3603	28.03	oe	ccsbBroad304_00222	CASP6	Caspases			
3604	28	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
3605	27.98	kd	CGS001-2147	F2	Endogenous ligands			
3606	27.97	oe	ccsbBroad304_00963	SMAD5	SMADs			
3607	27.97	kd	CGS001-11164	NUDT5	Nudix motif containing			
3608	27.95	kd	CGS001-51053	GMNN	-			
3609	27.94	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
3610	27.92	kd	CGS001-8772	FADD	-			
3611	27.92	kd	CGS001-717	C2	Complement system			
3612	27.9	kd	CGS001-6715	SRD5A1	-			
3613	27.87	kd	CGS001-5997	RGS2	Endogenous ligands			
3614	27.84	oe	ccsbBroad304_06235	G6PD	-			
3615	27.84	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
3616	27.83	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
3617	27.81	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
3618	27.8	kd	CGS001-7421	VDR	Vitamin D receptors			
3619	27.8	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
3620	27.77	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
3621	27.76	cc		Thromboxane receptor antagonist	-			
3622	27.76	kd	CGS001-890	CCNA2	-			
3623	27.75	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
3624	27.69	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
3625	27.68	kd	CGS001-84722	PSRC1	-			
3626	27.62	oe	ccsbBroad304_07252	DGKZ	-			
3627	27.62	kd	CGS001-11212	PROSC	-			
3628	27.61	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3629	27.59	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
3630	27.59	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
3631	27.58	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
3632	27.58	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
3633	27.56	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
3634	27.53	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
3635	27.53	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
3636	27.51	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
3637	27.49	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
3638	27.47	oe	ccsbBroad304_00424	DBI	-			
3639	27.46	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
3640	27.45	oe	ccsbBroad304_04675	ATG4A	-			
3641	27.44	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
3642	27.43	cp	BRD-K00532621	midazolam	Benzodiazepine receptor agonist		CYP3A5, CYP3A7, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3	Benzodiazepine receptor agonist
3643	27.4	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
3644	27.32	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
3645	27.3	oe	ccsbBroad304_04404	TUBB6	Tubulins			
3646	27.3	kd	CGS001-5894	RAF1	RAF family			
3647	27.28	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
3648	27.22	kd	CGS001-139135	PASD1	-			
3649	27.2	kd	CGS001-54658	UGT1A1	UDP glucuronosyltransferases			
3650	27.16	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
3651	27.15	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
3652	27.12	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
3653	27.1	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
3654	27.09	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
3655	27.05	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
3656	27.03	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
3657	27.03	kd	CGS001-10943	MSL3	-			
3658	27.01	oe	ccsbBroad304_07827	STK38L	NDR family			
3659	26.98	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
3660	26.97	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3661	26.95	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
3662	26.93	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
3663	26.92	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
3664	26.92	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
3665	26.89	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
3666	26.87	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
3667	26.84	kd	CGS001-115650	TNFRSF13C	Tumour necrosis factor (TNF) receptor family			
3668	26.82	kd	CGS001-2159	F10	Chymotrypsin			
3669	26.78	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
3670	26.78	oe	ccsbBroad304_07050	TFAP2A	-			
3671	26.77	oe	ccsbBroad304_00931	LCN2	Lipocalins			
3672	26.77	oe	ccsbBroad304_02553	BLCAP	-			
3673	26.77	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
3674	26.75	kd	CGS001-5538	PPT1	-			
3675	26.72	oe	ccsbBroad304_03933	CARD9	-			
3676	26.72	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
3677	26.64	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
3678	26.64	kd	CGS001-6337	SCNN1A	Epithelial sodium channels (ENaC)			
3679	26.64	kd	CGS001-63933	CCDC90A	-			
3680	26.63	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
3681	26.62	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
3682	26.62	kd	CGS001-204	AK2	Adenylate kinases			
3683	26.6	kd	CGS001-151126	ZNF385B	-			
3684	26.6	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
3685	26.54	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
3686	26.53	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
3687	26.53	kd	CGS001-2990	GUSB	-			
3688	26.52	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
3689	26.52	kd	CGS001-8569	MKNK1	MKN subfamily			
3690	26.51	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
3691	26.5	kd	CGS001-6897	TARS	Aminoacyl tRNA synthetases / Class II			
3692	26.47	kd	CGS001-25824	PRDX5	-			
3693	26.45	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
3694	26.44	cc		PI3K inhibitor	-			
3695	26.41	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
3696	26.41	kd	CGS001-5827	PXMP2	-			
3697	26.4	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
3698	26.39	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
3699	26.38	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
3700	26.37	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
3701	26.37	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
3702	26.31	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
3703	26.3	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
3704	26.29	kd	CGS001-3176	HNMT	-			
3705	26.29	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
3706	26.29	kd	CGS001-2	A2M	-			
3707	26.28	kd	CGS001-7057	THBS1	-			
3708	26.25	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
3709	26.21	kd	CGS001-9686	VGLL4	-			
3710	26.21	oe	ccsbBroad304_08480	PNPO	-			
3711	26.2	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
3712	26.19	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3713	26.12	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
3714	26.1	kd	CGS001-54749	EPDR1	-			
3715	26.09	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3716	26.08	kd	CGS001-23429	RYBP	-			
3717	26.07	kd	CGS001-55770	EXOC2	-			
3718	26.05	kd	CGS001-1105	CHD1	-			
3719	26.01	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
3720	26	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3721	26	kd	CGS001-10023	FRAT1	-			
3722	25.99	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
3723	25.98	kd	CGS001-5255	PHKA1	-			
3724	25.97	kd	CGS001-7764	ZNF217	Zinc fingers, C2H2-type			
3725	25.94	oe	ccsbBroad304_03405	CHRAC1	-			
3726	25.93	kd	CGS001-23499	MACF1	EF-hand domain containing			
3727	25.91	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
3728	25.88	kd	CGS001-4860	PNP	-			
3729	25.86	kd	CGS001-306	ANXA3	Annexins			
3730	25.84	kd	CGS001-148327	CREB3L4	basic leucine zipper proteins			
3731	25.82	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
3732	25.79	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3733	25.75	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
3734	25.75	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
3735	25.7	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
3736	25.7	kd	CGS001-10128	LRPPRC	-			
3737	25.69	oe	ccsbBroad304_07884	RYBP	-			
3738	25.69	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3739	25.66	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
3740	25.59	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
3741	25.56	kd	CGS001-2937	GSS	-			
3742	25.54	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
3743	25.54	kd	CGS001-6595	SMARCA2	Non-enzymatic BRD containing proteins			
3744	25.54	kd	CGS001-350	APOH	Apolipoproteins			
3745	25.52	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
3746	25.52	oe	ccsbBroad304_07208	NRIP1	-			
3747	25.49	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
3748	25.49	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
3749	25.49	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
3750	25.41	kd	CGS001-29937	NENF	-			
3751	25.4	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
3752	25.39	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3753	25.39	kd	CGS001-7185	TRAF1	-			
3754	25.37	oe	ccsbBroad304_02416	TUBB4B	-			
3755	25.33	oe	ccsbBroad304_03428	EXOSC4	-			
3756	25.31	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
3757	25.29	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
3758	25.26	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3759	25.26	kd	CGS001-3576	IL8	-			
3760	25.25	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
3761	25.24	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
3762	25.23	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
3763	25.2	kd	CGS001-83637	ZMIZ2	Zinc fingers, MIZ-type			
3764	25.16	kd	CGS001-2909	ARHGAP35	Rho GTPase activating proteins			
3765	25.15	cp	BRD-K84955386	hyperoside	Glucosidase inhibitor		ACE, AKR1B1, GAA	Glucosidase inhibitor
3766	25.15	kd	CGS001-6303	SAT1	-			
3767	25.15	kd	CGS001-51422	PRKAG2	AMPK subfamily			
3768	25.14	kd	CGS001-51441	YTHDF2	-			
3769	25.11	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
3770	25.11	kd	CGS001-10972	TMED10	-			
3771	25.09	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
3772	25.08	kd	CGS001-204851	HIPK1	HIPK subfamily			
3773	25.04	kd	CGS001-5586	PKN2	Protein kinase N (PKN) family			
3774	25.02	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
3775	25	kd	CGS001-3932	LCK	Src family			
3776	24.98	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
3777	24.97	oe	ccsbBroad304_02452	NXF1	-			
3778	24.94	kd	CGS001-83593	RASSF5	-			
3779	24.94	oe	ccsbBroad304_07598	PEMT	-			
3780	24.93	kd	CGS001-4791	NFKB2	NFkappaB transcription factor family			
3781	24.84	kd	CGS001-3978	LIG1	-			
3782	24.83	cc		Sodium channel blocker	-			
3783	24.8	oe	ccsbBroad304_03112	NENF	-			
3784	24.8	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3785	24.76	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
3786	24.76	kd	CGS001-19	ABCA1	ATP binding cassette transporters / subfamily A			
3787	24.75	oe	ccsbBroad304_00515	ERH	-			
3788	24.71	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
3789	24.71	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
3790	24.67	kd	CGS001-9318	COPS2	-			
3791	24.64	kd	CGS001-51593	SRRT	-			
3792	24.63	kd	CGS001-397	ARHGDIB	Endogenous ligands			
3793	24.62	kd	CGS001-1948	EFNB2	Ephrins			
3794	24.6	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
3795	24.58	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
3796	24.57	kd	CGS001-10214	SSX3	-			
3797	24.57	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
3798	24.56	kd	CGS001-22938	SNW1	-			
3799	24.55	kd	CGS001-6286	S100P	EF-hand domain containing			
3800	24.54	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
3801	24.54	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
3802	24.47	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
3803	24.46	cc		Benzodiazepine receptor agonist	-			
3804	24.44	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
3805	24.36	cc		Zinc fingers RanBP2 type LOF	-			
3806	24.35	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
3807	24.32	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
3808	24.29	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
3809	24.28	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
3810	24.26	oe	ccsbBroad304_01618	STXBP1	-			
3811	24.24	oe	ccsbBroad304_06255	LRRC32	-			
3812	24.21	kd	CGS001-94234	FOXQ1	Forkhead boxes			
3813	24.18	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
3814	24.17	kd	CGS001-5925	RB1	Endogenous ligands			
3815	24.16	kd	CGS001-5621	PRNP	CD molecules			
3816	24.13	kd	CGS001-25797	QPCT	Aminopeptidase Y			
3817	24.12	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
3818	24.09	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
3819	24.09	kd	CGS001-7082	TJP1	-			
3820	24.09	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
3821	24.02	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
3822	24.01	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3823	23.91	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
3824	23.91	kd	CGS001-3487	IGFBP4	insulin-like growth factor (IGF) binding proteins			
3825	23.86	kd	CGS001-63892	THADA	-			
3826	23.85	cc		Sirtuins GOF	-			
3827	23.82	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
3828	23.81	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
3829	23.81	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
3830	23.76	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
3831	23.76	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
3832	23.72	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
3833	23.68	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
3834	23.63	kd	CGS001-8651	SOCS1	SH2 domain containing			
3835	23.62	kd	CGS001-3845	KRAS	RAS subfamily			
3836	23.61	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
3837	23.6	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
3838	23.58	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3839	23.58	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
3840	23.57	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
3841	23.56	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
3842	23.54	kd	CGS001-2767	GNA11	-			
3843	23.53	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
3844	23.46	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
3845	23.46	oe	ccsbBroad304_03310	LCMT1	-			
3846	23.4	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
3847	23.39	oe	ccsbBroad304_03858	SRPRB	-			
3848	23.38	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
3849	23.38	kd	CGS001-5432	POLR2C	RNA polymerase subunits			
3850	23.38	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
3851	23.35	cp	BRD-K82143716	flucytosine	Antifungal		DNMT1	Antifungal
3852	23.34	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
3853	23.34	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
3854	23.33	kd	CGS001-1662	DDX10	DEAD-boxes			
3855	23.3	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
3856	23.28	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
3857	23.28	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
3858	23.28	kd	CGS001-11186	RASSF1	-			
3859	23.26	kd	CGS001-54815	GATAD2A	GATA zinc finger domain containing			
3860	23.24	kd	CGS001-9258	MFHAS1	-			
3861	23.22	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
3862	23.22	cp	BRD-K60160658	tiagabine	GABA uptake inhibitor		SLC6A1, CYP2C19	GABA uptake inhibitor
3863	23.2	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3864	23.2	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
3865	23.19	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
3866	23.18	cp	BRD-K39621635	artemether	Antimalarial		ATP1A1, CYP2B6, CYP2C19, CYP3A5	Antimalarial
3867	23.18	cp	BRD-K94144010	cotinine	Nicotine metabolite			Nicotine metabolite
3868	23.16	kd	CGS001-3074	HEXB	-			
3869	23.13	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3870	23.08	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
3871	23.04	oe	ccsbBroad304_06718	PFN2	-			
3872	23.04	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3873	23.03	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
3874	22.99	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
3875	22.99	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
3876	22.98	oe	ccsbBroad304_06855	RDX	-			
3877	22.97	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
3878	22.97	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
3879	22.92	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
3880	22.92	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
3881	22.9	oe	ccsbBroad304_06765	PRCC	-			
3882	22.89	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
3883	22.86	oe	ccsbBroad304_01658	PRDX2	-			
3884	22.79	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
3885	22.76	kd	CGS001-6787	NEK4	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3886	22.76	kd	CGS001-3956	LGALS1	Endogenous ligands			
3887	22.72	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
3888	22.72	kd	CGS001-1184	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
3889	22.69	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
3890	22.68	oe	ccsbBroad304_03308	YTHDF2	-			
3891	22.68	kd	CGS001-4439	MSH5	-			
3892	22.68	oe	ccsbBroad304_03658	DCP1A	-			
3893	22.66	kd	CGS001-51022	GLRX2	-			
3894	22.66	kd	CGS001-32	ACACB	Carboxylases			
3895	22.64	cp	BRD-K98493452	honokiol	AKT inhibitor		ALOX5, PTGS1, PTGS2	AKT inhibitor
3896	22.64	kd	CGS001-2138	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
3897	22.63	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
3898	22.63	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
3899	22.62	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
3900	22.59	oe	ccsbBroad304_09284	UBE3B	-			
3901	22.58	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
3902	22.52	kd	CGS001-10797	MTHFD2	-			
3903	22.51	kd	CGS001-5292	PIM1	PIM family			
3904	22.47	kd	CGS001-3297	HSF1	-			
3905	22.46	oe	ccsbBroad304_00113	ASNS	-			
3906	22.46	kd	CGS001-2242	FES	Fer family			
3907	22.45	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3908	22.43	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
3909	22.42	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
3910	22.4	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
3911	22.39	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
3912	22.39	oe	ccsbBroad304_02554	TRAFD1	-			
3913	22.34	kd	CGS001-3054	HCFC1	-			
3914	22.33	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
3915	22.33	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
3916	22.31	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
3917	22.27	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
3918	22.25	kd	CGS001-6773	STAT2	SH2 domain containing			
3919	22.23	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
3920	22.17	kd	CGS001-199704	ZNF585A	Zinc fingers, C2H2-type			
3921	22.14	oe	ccsbBroad304_01724	TTR	-			
3922	22.12	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
3923	22.1	kd	CGS001-6804	STX1A	-			
3924	22.1	kd	CGS001-3775	KCNK1	Two-P potassium channels			
3925	22.06	oe	ccsbBroad304_07363	AIFM1	-			
3926	22.03	kd	CGS001-23647	ARFIP2	-			
3927	22.02	oe	ccsbBroad304_02298	DNM1L	-			
3928	22.01	kd	CGS001-662	BNIP1	-			
3929	21.96	oe	ccsbBroad304_01923	UXT	-			
3930	21.95	oe	ccsbBroad304_03615	ZNF673	-			
3931	21.94	kd	CGS001-10097	ACTR2	-			
3932	21.92	kd	CGS001-79960	PHF17	-			
3933	21.89	kd	CGS001-6185	RPN2	-			
3934	21.88	oe	ccsbBroad304_02017	PEX11A	-			
3935	21.83	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
3936	21.83	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
3937	21.83	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
3938	21.8	oe	ccsbBroad304_07506	UBAP2L	-			
3939	21.75	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
3940	21.74	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
3941	21.73	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
3942	21.72	kd	CGS001-7486	WRN	-			
3943	21.71	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
3944	21.7	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
3945	21.69	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
3946	21.68	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3947	21.66	oe	ccsbBroad304_09503	KLHDC9	-			
3948	21.58	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
3949	21.57	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
3950	21.51	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
3951	21.5	kd	CGS001-4837	NNMT	-			
3952	21.48	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
3953	21.45	oe	ccsbBroad304_10230	STK19	G11 family			
3954	21.44	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
3955	21.44	kd	CGS001-375133	PI4KAP2	-			
3956	21.42	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
3957	21.41	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
3958	21.4	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
3959	21.39	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3960	21.39	oe	ccsbBroad304_07875	SPECC1L	-			
3961	21.36	kd	CGS001-1528	CYB5A	Cytochrome b genes			
3962	21.3	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
3963	21.29	kd	CGS001-1030	CDKN2B	-			
3964	21.29	oe	ccsbBroad304_07569	TRIB1	Trbl family			
3965	21.27	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
3966	21.25	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
3967	21.25	kd	CGS001-9871	SEC24D	-			
3968	21.22	oe	ccsbBroad304_00665	GOT1	-			
3969	21.21	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
3970	21.21	kd	CGS001-50604	IL20	Interleukins and interleukin receptors			
3971	21.15	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
3972	21.13	cc		ATP synthase inhibitor	-			
3973	21.11	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
3974	21.09	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
3975	21.08	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
3976	21.07	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
3977	21.07	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
3978	21.05	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
3979	21.04	cp	BRD-K99447003	enalaprilat	ACE inhibitor		ACE	ACE inhibitor
3980	20.95	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
3981	20.95	kd	CGS001-170591	S100Z	EF-hand domain containing			
3982	20.95	kd	CGS001-302	ANXA2	Annexins			
3983	20.9	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
3984	20.9	kd	CGS001-5979	RET	Type XIV RTKs: RET			
3985	20.88	cp	BRD-K22227508	targinine	Nitric oxide synthase inhibitor		NOS2, NOS3	Nitric oxide synthase inhibitor
3986	20.87	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
3987	20.86	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
3988	20.86	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
3989	20.86	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
3990	20.82	kd	CGS001-3685	ITGAV	Integrins			
3991	20.78	oe	ccsbBroad304_03928	RRAGC	-			
3992	20.78	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
3993	20.73	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3994	20.7	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
3995	20.66	kd	CGS001-4287	ATXN3	Ataxins			
3996	20.65	oe	ccsbBroad304_09195	MCM8	-			
3997	20.63	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
3998	20.62	oe	ccsbBroad304_02772	ICMT	-			
3999	20.62	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
4000	20.62	kd	CGS001-861	RUNX1	-			
4001	20.62	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
4002	20.61	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
4003	20.61	kd	CGS001-55290	BRF2	-			
4004	20.57	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
4005	20.57	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
4006	20.57	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
4007	20.57	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
4008	20.53	cc		Integrin subunits alpha LOF	-			
4009	20.5	cc		Protein phosphatase catalytic subunits LOF	-			
4010	20.49	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
4011	20.49	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
4012	20.48	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4013	20.48	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
4014	20.46	kd	CGS001-319100	TAAR6	GPCR / Class A : Trace amine associated receptors			
4015	20.45	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
4016	20.44	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
4017	20.43	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
4018	20.43	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
4019	20.41	kd	CGS001-839	CASP6	Caspases			
4020	20.41	oe	ccsbBroad304_14174	CDKAL1	-			
4021	20.37	kd	CGS001-27241	BBS9	-			
4022	20.36	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
4023	20.35	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
4024	20.34	kd	CGS001-1384	CRAT	-			
4025	20.33	kd	CGS001-25801	GCA	EF-hand domain containing			
4026	20.31	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
4027	20.31	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
4028	20.24	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
4029	20.23	kd	CGS001-3660	IRF2	-			
4030	20.22	oe	ccsbBroad304_08596	EAPP	-			
4031	20.2	oe	ccsbBroad304_03415	GFOD1	-			
4032	20.14	oe	ccsbBroad304_02789	ADAT1	-			
4033	20.14	kd	CGS001-203523	ZNF449	Zinc fingers, C2H2-type			
4034	20.12	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
4035	20.1	oe	ccsbBroad304_01723	TTK	TTK family			
4036	20.06	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
4037	20	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
4038	19.98	kd	CGS001-275	AMT	-			
4039	19.93	kd	CGS001-2266	FGG	Endogenous ligands			
4040	19.88	kd	CGS001-201799	TMEM154	-			
4041	19.87	kd	CGS001-147686	ZNF418	Zinc fingers, C2H2-type			
4042	19.87	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
4043	19.86	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
4044	19.84	kd	CGS001-23066	CAND2	-			
4045	19.83	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
4046	19.82	kd	CGS001-79006	METRN	-			
4047	19.82	kd	CGS001-2182	ACSL4	Acyl-CoA synthetase family			
4048	19.8	oe	ccsbBroad304_07466	VGLL4	-			
4049	19.78	cc		Phospholipases GOF	-			
4050	19.76	kd	CGS001-25842	ASF1A	-			
4051	19.73	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
4052	19.73	kd	CGS001-896	CCND3	-			
4053	19.68	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
4054	19.63	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
4055	19.62	oe	ccsbBroad304_02804	KLHDC2	-			
4056	19.61	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
4057	19.6	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
4058	19.58	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
4059	19.58	kd	CGS001-10096	ACTR3	-			
4060	19.57	oe	ccsbBroad304_07528	DMTF1	-			
4061	19.57	kd	CGS001-1955	MEGF9	-			
4062	19.52	oe	ccsbBroad304_00572	FKBP3	-			
4063	19.51	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4064	19.5	kd	CGS001-1859	DYRK1A	Dyrk1 subfamily			
4065	19.48	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
4066	19.46	kd	CGS001-6119	RPA3	-			
4067	19.44	kd	CGS001-23761	PISD	Decarboxylases			
4068	19.41	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
4069	19.4	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
4070	19.33	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
4071	19.33	kd	CGS001-51548	SIRT6	Histone deacetylases (HDACs)			
4072	19.33	kd	CGS001-51451	LCMT1	-			
4073	19.3	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
4074	19.3	kd	CGS001-10400	PEMT	-			
4075	19.29	kd	CGS001-1756	DMD	-			
4076	19.26	oe	ccsbBroad304_01960	CASK	CASK family			
4077	19.24	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
4078	19.22	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
4079	19.2	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
4080	19.19	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
4081	19.17	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
4082	19.13	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
4083	19.13	kd	CGS001-79733	E2F8	-			
4084	19.13	kd	CGS001-55214	LEPREL1	-			
4085	19.12	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
4086	19.09	kd	CGS001-776	CACNA1D	Calcium channel subunits			
4087	19.08	oe	ccsbBroad304_06720	PHYH	-			
4088	19.06	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
4089	19.06	kd	CGS001-7316	UBC	-			
4090	19.06	kd	CGS001-5723	PSPH	-			
4091	19.05	oe	ccsbBroad304_02361	MFSD10	-			
4092	19.05	kd	CGS001-8050	PDHX	-			
4093	19.03	kd	CGS001-10111	RAD50	-			
4094	19	oe	ccsbBroad304_03961	SMURF2	-			
4095	18.96	kd	CGS001-10329	TMEM5	-			
4096	18.93	oe	ccsbBroad304_02834	GABARAPL1	-			
4097	18.92	kd	CGS001-375	ARF1	ADP-ribosylation factors			
4098	18.89	cc		S100 calcium binding proteins LOF	-			
4099	18.89	oe	ccsbBroad304_10487	BPHL	-			
4100	18.88	oe	ccsbBroad304_03386	SPA17	-			
4101	18.88	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
4102	18.84	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
4103	18.83	kd	CGS001-5037	PEBP1	-			
4104	18.82	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
4105	18.82	kd	CGS001-29888	STRN4	WD repeat domain containing			
4106	18.79	cc		Bile acid	-			
4107	18.78	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
4108	18.78	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
4109	18.77	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
4110	18.74	kd	CGS001-55644	OSGEP	-			
4111	18.73	kd	CGS001-5110	PCMT1	-			
4112	18.71	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
4113	18.71	kd	CGS001-28964	GIT1	Ankyrin repeat domain containing			
4114	18.66	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
4115	18.65	cp	BRD-A68888262	azelastine	Histamine receptor antagonist		HRH1, CYP2C19	Histamine receptor antagonist
4116	18.59	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
4117	18.59	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
4118	18.59	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
4119	18.56	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
4120	18.53	kd	CGS001-8089	YEATS4	-			
4121	18.45	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
4122	18.42	kd	CGS001-5624	PROC	Endogenous ligands			
4123	18.38	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
4124	18.36	oe	ccsbBroad304_01392	TRIM27	-			
4125	18.36	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
4126	18.31	kd	CGS001-6271	S100A1	EF-hand domain containing			
4127	18.3	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
4128	18.3	kd	CGS001-10955	SERINC3	-			
4129	18.23	kd	CGS001-4734	NEDD4	-			
4130	18.22	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
4131	18.2	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
4132	18.2	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
4133	18.19	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4134	18.17	kd	CGS001-2295	FOXF2	Forkhead boxes			
4135	18.16	kd	CGS001-6397	SEC14L1	-			
4136	18.13	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
4137	18.13	kd	CGS001-60493	FASTKD5	-			
4138	18.12	kd	CGS001-5763	PTMS	-			
4139	18.1	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
4140	18.09	kd	CGS001-51750	RTEL1	-			
4141	18.09	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
4142	18.06	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
4143	18.04	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
4144	18.04	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
4145	18.03	kd	CGS001-23274	CLEC16A	C-type lectin domain containing			
4146	18.02	kd	CGS001-47	ACLY	-			
4147	18.02	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
4148	18.01	oe	ccsbBroad304_06098	DHCR24	-			
4149	18.01	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
4150	17.99	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
4151	17.97	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
4152	17.96	oe	ccsbBroad304_02340	SORBS3	-			
4153	17.94	kd	CGS001-8634	RTCD1	-			
4154	17.94	kd	CGS001-8204	NRIP1	-			
4155	17.89	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
4156	17.89	kd	CGS001-58528	RRAGD	-			
4157	17.88	cp	BRD-K53220666	trimetozine	Sedative			Sedative
4158	17.83	oe	ccsbBroad304_02133	CD83	CD molecules			
4159	17.81	oe	ccsbBroad304_07362	NMI	-			
4160	17.81	kd	CGS001-26149	ZNF658	Zinc fingers, C2H2-type			
4161	17.79	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
4162	17.75	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
4163	17.73	oe	ccsbBroad304_02094	FIBP	-			
4164	17.72	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
4165	17.7	kd	CGS001-255877	BCL6B	BTB/POZ domain containing			
4166	17.67	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
4167	17.66	kd	CGS001-2957	GTF2A1	General transcription factors			
4168	17.62	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
4169	17.6	kd	CGS001-9218	VAPA	-			
4170	17.54	kd	CGS001-6601	SMARCC2	-			
4171	17.5	kd	CGS001-481	ATP1B1	ATPases / P-type			
4172	17.48	kd	CGS001-8835	SOCS2	SH2 domain containing			
4173	17.47	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
4174	17.43	kd	CGS001-57721	METTL14	-			
4175	17.4	kd	CGS001-10476	ATP5H	ATPases / F-type			
4176	17.38	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
4177	17.36	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
4178	17.36	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
4179	17.35	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
4180	17.34	kd	CGS001-54438	GFOD1	-			
4181	17.31	kd	CGS001-283	ANG	Ribonucleases, RNase A			
4182	17.29	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
4183	17.28	oe	ccsbBroad304_02759	DICER1	-			
4184	17.26	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
4185	17.24	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
4186	17.24	kd	CGS001-54884	RETSAT	-			
4187	17.24	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
4188	17.23	kd	CGS001-79139	DERL1	-			
4189	17.22	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
4190	17.21	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
4191	17.2	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
4192	17.19	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
4193	17.18	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
4194	17.14	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
4195	17.09	cp	BRD-K10961822	latanoprost	Prostanoid receptor agonist		PTGFR	Prostanoid receptor agonist
4196	17.09	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
4197	17.08	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
4198	17.07	kd	CGS001-8650	NUMB	-			
4199	17.05	kd	CGS001-79885	HDAC11	Histone deacetylases			
4200	17.05	kd	CGS001-1763	DNA2	-			
4201	17.03	kd	CGS001-7097	TLR2	Toll-like receptor family			
4202	17	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
4203	16.99	cc		PRD class homeoboxes and psudogenes LOF	-			
4204	16.99	kd	CGS001-652	BMP4	Bone morphogenetic proteins			
4205	16.98	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
4206	16.97	kd	CGS001-7088	TLE1	WD repeat domain containing			
4207	16.96	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
4208	16.95	oe	ccsbBroad304_02414	IRF9	-			
4209	16.94	kd	CGS001-23266	LPHN2	Adhesion Class GPCRs			
4210	16.93	kd	CGS001-2287	FKBP3	-			
4211	16.92	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
4212	16.88	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
4213	16.88	kd	CGS001-5144	PDE4D	Phosphodiesterases			
4214	16.83	cp	BRD-K47278471	diphenhydramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4215	16.82	kd	CGS001-399694	SHC4	SH2 domain containing			
4216	16.81	kd	CGS001-644	BLVRA	-			
4217	16.81	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
4218	16.77	kd	CGS001-59286	UBL5	-			
4219	16.77	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
4220	16.76	kd	CGS001-26086	GPSM1	Tetratricopeptide (TTC) repeat domain containing			
4221	16.73	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
4222	16.72	kd	CGS001-51586	MED15	-			
4223	16.7	kd	CGS001-3665	IRF7	-			
4224	16.68	oe	ccsbBroad304_01613	STK11	LKB subfamily			
4225	16.67	kd	CGS001-10460	TACC3	-			
4226	16.64	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
4227	16.63	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
4228	16.63	oe	ccsbBroad304_06180	ESD	-			
4229	16.59	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
4230	16.58	kd	CGS001-7003	TEAD1	-			
4231	16.53	kd	CGS001-5696	PSMB8	Proteasome (prosome, macropain) subunits			
4232	16.5	oe	ccsbBroad304_01605	SSX2	-			
4233	16.5	oe	ccsbBroad304_08662	MCCC1	-			
4234	16.46	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
4235	16.46	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
4236	16.46	kd	CGS001-2864	FFAR1	Fatty acid receptors			
4237	16.45	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
4238	16.44	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
4239	16.43	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
4240	16.43	kd	CGS001-134187	POU5F2	Homeoboxes / POU class			
4241	16.43	kd	CGS001-3572	IL6ST	IL-6 receptor family			
4242	16.42	oe	ccsbBroad304_09054	EGFL8	-			
4243	16.41	kd	CGS001-25949	SYF2	-			
4244	16.37	oe	ccsbBroad304_00519	ETFB	-			
4245	16.36	kd	CGS001-1644	DDC	Catecholamine turnover			
4246	16.34	kd	CGS001-1284	COL4A2	Collagens			
4247	16.28	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
4248	16.27	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
4249	16.26	kd	CGS001-85004	RERG	-			
4250	16.22	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
4251	16.16	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
4252	16.16	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
4253	16.15	kd	CGS001-4605	MYBL2	-			
4254	16.12	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
4255	16.1	kd	CGS001-51070	NOSIP	-			
4256	16.09	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
4257	16.04	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
4258	16.03	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
4259	16.01	kd	CGS001-29915	HCFC2	-			
4260	16.01	oe	ccsbBroad304_01142	PAFAH1B2	-			
4261	15.99	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
4262	15.99	kd	CGS001-2717	GLA	-			
4263	15.99	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
4264	15.94	kd	CGS001-3383	ICAM1	CD molecules			
4265	15.93	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
4266	15.92	cc		Reverse transcriptase inhibitor	-			
4267	15.89	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
4268	15.83	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
4269	15.83	kd	CGS001-4170	MCL1	-			
4270	15.83	kd	CGS001-1514	CTSL1	-			
4271	15.8	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
4272	15.79	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
4273	15.78	oe	ccsbBroad304_00054	ALDOC	-			
4274	15.78	kd	CGS001-2100	ESR2	Estrogen receptors			
4275	15.75	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
4276	15.74	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
4277	15.74	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
4278	15.7	kd	CGS001-403	ARL3	ADP-ribosylation factors			
4279	15.69	oe	ccsbBroad304_03554	NAT10	-			
4280	15.67	cp	BRD-K04196797	oxcarbazepine	Sodium channel blocker		CYP2C19, CYP3A4, CYP3A5, SCN1A, SCN3A, SCN5A	Sodium channel blocker
4281	15.67	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
4282	15.66	kd	CGS001-2634	GBP2	-			
4283	15.65	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
4284	15.65	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
4285	15.6	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
4286	15.6	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
4287	15.56	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
4288	15.52	oe	ccsbBroad304_03264	UBAP1	-			
4289	15.51	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
4290	15.5	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
4291	15.48	kd	CGS001-56647	BCCIP	-			
4292	15.47	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
4293	15.47	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
4294	15.46	kd	CGS001-54998	AURKAIP1	-			
4295	15.45	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
4296	15.42	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
4297	15.41	kd	CGS001-222	ALDH3B2	Aldehyde dehydrogenases			
4298	15.4	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
4299	15.38	kd	CGS001-3690	ITGB3	Integrins			
4300	15.38	kd	CGS001-9131	AIFM1	-			
4301	15.37	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
4302	15.34	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
4303	15.32	kd	CGS001-27	ABL2	Abl family			
4304	15.28	kd	CGS001-4976	OPA1	-			
4305	15.25	oe	ccsbBroad304_02708	TRIM32	-			
4306	15.24	kd	CGS001-28960	DCPS	-			
4307	15.22	kd	CGS001-9180	OSMR	IL-6 receptor family			
4308	15.21	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
4309	15.21	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
4310	15.19	kd	CGS001-54505	DHX29	DEAH-boxes			
4311	15.19	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
4312	15.18	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
4313	15.17	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
4314	15.17	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
4315	15.16	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
4316	15.11	kd	CGS001-2967	GTF2H3	General transcription factors			
4317	15.1	oe	ccsbBroad304_06645	NQO2	-			
4318	15.08	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
4319	15.07	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
4320	15.07	kd	CGS001-6193	RPS5	S ribosomal proteins			
4321	15.05	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
4322	15.04	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
4323	15.04	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
4324	15.01	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
4325	15.01	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
4326	15.01	kd	CGS001-2224	FDPS	Lanosterol biosynthesis pathway			
4327	14.99	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
4328	14.99	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
4329	14.98	kd	CGS001-9978	RBX1	RING-type (C3HC4) zinc fingers			
4330	14.98	oe	ccsbBroad304_06264	GBP2	-			
4331	14.96	kd	CGS001-115	ADCY9	Adenylyl cyclases			
4332	14.9	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
4333	14.87	kd	CGS001-5610	EIF2AK2	Other PEK family kinases			
4334	14.82	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
4335	14.82	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
4336	14.81	kd	CGS001-7905	REEP5	Receptor accessory proteins			
4337	14.79	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
4338	14.78	kd	CGS001-8226	HDHD1	-			
4339	14.77	oe	ccsbBroad304_00552	FEN1	-			
4340	14.77	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
4341	14.77	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
4342	14.75	kd	CGS001-378	ARF4	ADP-ribosylation factors			
4343	14.74	oe	ccsbBroad304_10431	HADHB	-			
4344	14.7	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
4345	14.7	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
4346	14.68	kd	CGS001-23475	QPRT	-			
4347	14.68	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
4348	14.67	kd	CGS001-3416	IDE	Pitrilysin			
4349	14.64	oe	ccsbBroad304_06745	PNN	-			
4350	14.63	kd	CGS001-8795	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
4351	14.62	kd	CGS001-2181	ACSL3	Acyl-CoA synthetase family			
4352	14.62	oe	ccsbBroad304_07267	PDLIM4	-			
4353	14.61	oe	ccsbBroad304_01662	TFDP2	-			
4354	14.6	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
4355	14.58	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
4356	14.56	kd	CGS001-383	ARG1	Arginase			
4357	14.51	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
4358	14.5	oe	ccsbBroad304_09354	IGSF8	CD molecules			
4359	14.43	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
4360	14.42	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4361	14.42	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
4362	14.42	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
4363	14.4	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
4364	14.38	kd	CGS001-9341	VAMP3	Vesicle-associated membrane proteins			
4365	14.34	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
4366	14.34	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
4367	14.34	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
4368	14.32	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
4369	14.28	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
4370	14.27	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
4371	14.27	cp	BRD-K18523449	mestanolone	Androgenic steroid			Androgenic steroid
4372	14.25	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
4373	14.25	kd	CGS001-7913	DEK	-			
4374	14.25	kd	CGS001-384	ARG2	Arginase			
4375	14.2	kd	CGS001-7511	XPNPEP1	Methionyl aminopeptidase			
4376	14.16	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
4377	14.14	kd	CGS001-7415	VCP	ATPases / AAA-type			
4378	14.09	oe	ccsbBroad304_02506	EBP	-			
4379	14.09	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
4380	14.07	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
4381	14.06	oe	ccsbBroad304_01208	PITPNA	-			
4382	14.04	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4383	14.03	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
4384	14.03	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
4385	14.01	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
4386	13.97	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
4387	13.84	kd	CGS001-2593	GAMT	-			
4388	13.81	kd	CGS001-166793	ZBTB49	BTB/POZ domain containing			
4389	13.81	kd	CGS001-54915	YTHDF1	-			
4390	13.81	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
4391	13.73	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
4392	13.69	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
4393	13.67	kd	CGS001-55107	ANO1	Calcium activated chloride channel			
4394	13.67	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
4395	13.67	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
4396	13.65	oe	ccsbBroad304_08511	RFK	-			
4397	13.64	oe	ccsbBroad304_06085	DCK	-			
4398	13.64	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
4399	13.63	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
4400	13.56	kd	CGS001-9958	USP15	Ubiquitin-specific peptidases			
4401	13.56	kd	CGS001-89766	UMODL1	-			
4402	13.56	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
4403	13.53	kd	CGS001-6850	SYK	Syk family			
4404	13.52	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
4405	13.51	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
4406	13.51	oe	ccsbBroad304_06976	SMARCE1	-			
4407	13.49	kd	CGS001-2030	SLC29A1	SLC29 family			
4408	13.48	kd	CGS001-84669	USP32	EF-hand domain containing			
4409	13.47	kd	CGS001-6617	SNAPC1	-			
4410	13.45	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
4411	13.41	oe	ccsbBroad304_07401	TXNL1	-			
4412	13.41	kd	CGS001-4905	NSF	ATPases / AAA-type			
4413	13.41	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
4414	13.4	kd	CGS001-367	AR	Nuclear hormone receptors			
4415	13.4	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
4416	13.35	kd	CGS001-9404	LPXN	-			
4417	13.33	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
4418	13.31	kd	CGS001-4817	NIT1	-			
4419	13.28	kd	CGS001-6658	SOX3	SRY (sex determining region Y)-boxes			
4420	13.28	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
4421	13.21	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
4422	13.2	kd	CGS001-112858	TP53RK	Bud32 family			
4423	13.19	kd	CGS001-6790	AURKA	Aurora kinase			
4424	13.18	cp	BRD-A24381660	zeranol	Estrogen receptor agonist			Estrogen receptor agonist
4425	13.18	oe	ccsbBroad304_10212	GRHL3	-			
4426	13.15	oe	ccsbBroad304_01584	SPARC	-			
4427	13.14	kd	CGS001-54490	UGT2B28	UDP glucuronosyltransferases			
4428	13.1	kd	CGS001-2966	GTF2H2	General transcription factors			
4429	13.09	oe	ccsbBroad304_00459	DPYD	-			
4430	13.07	kd	CGS001-10888	GPR83	GPCR / Class A : Orphans			
4431	13.05	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
4432	13.01	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
4433	12.99	kd	CGS001-55278	QRSL1	-			
4434	12.98	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
4435	12.9	cc		DNA polymerase inhibitor	-			
4436	12.9	kd	CGS001-10587	TXNRD2	-			
4437	12.89	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
4438	12.85	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
4439	12.83	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
4440	12.78	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
4441	12.75	kd	CGS001-6418	SET	-			
4442	12.75	kd	CGS001-5025	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
4443	12.74	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
4444	12.67	oe	ccsbBroad304_02596	KDELR3	-			
4445	12.67	kd	CGS001-84936	ZFYVE19	Zinc fingers, FYVE domain containing			
4446	12.66	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
4447	12.65	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
4448	12.6	kd	CGS001-3551	IKBKB	IKK family			
4449	12.6	kd	CGS001-4089	SMAD4	SMADs			
4450	12.59	kd	CGS001-51174	TUBD1	Tubulins			
4451	12.59	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
4452	12.58	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
4453	12.53	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
4454	12.5	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4455	12.48	oe	ccsbBroad304_00966	MAFG	-			
4456	12.46	oe	ccsbBroad304_02032	TSC22D1	-			
4457	12.46	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
4458	12.46	kd	CGS001-4833	NME4	-			
4459	12.46	kd	CGS001-10423	CDIPT	-			
4460	12.43	oe	ccsbBroad304_03177	FIS1	-			
4461	12.43	kd	CGS001-10381	TUBB3	Tubulins			
4462	12.42	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4463	12.42	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
4464	12.38	kd	CGS001-4072	EPCAM	CD molecules			
4465	12.32	kd	CGS001-8764	TNFRSF14	Tumour necrosis factor (TNF) receptor family			
4466	12.31	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
4467	12.3	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4468	12.29	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
4469	12.29	cp	BRD-K82357231	desloratadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4470	12.25	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
4471	12.22	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
4472	12.21	oe	ccsbBroad304_08339	CMPK1	-			
4473	12.21	oe	ccsbBroad304_06008	AP2M1	-			
4474	12.2	kd	CGS001-81539	SLC38A1	System A-like transporters			
4475	12.18	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
4476	12.18	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4477	12.17	kd	CGS001-3670	ISL1	Homeoboxes / LIM class			
4478	12.17	oe	ccsbBroad304_00038	AGL	-			
4479	12.16	kd	CGS001-124641	OVCA2	-			
4480	12.13	cp	BRD-K16336526	capsaicin	TRPV agonist		TRPV1, CFTR, ENOX2	TRPV agonist
4481	12.1	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
4482	12.09	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
4483	12.08	kd	CGS001-3895	KTN1	-			
4484	12.07	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
4485	12.04	kd	CGS001-226	ALDOA	-			
4486	12.03	kd	CGS001-677	ZFP36L1	RING-type (C3HC4) zinc fingers			
4487	12.03	kd	CGS001-7249	TSC2	-			
4488	11.98	oe	ccsbBroad304_02217	FEZ1	-			
4489	11.96	kd	CGS001-3066	HDAC2	Histone deacetylases			
4490	11.91	kd	CGS001-427	ASAH1	Acid ceramidase			
4491	11.9	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
4492	11.9	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
4493	11.89	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
4494	11.88	kd	CGS001-10975	UQCR11	Mitochondrial respiratory chain complex / Complex III			
4495	11.88	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
4496	11.87	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
4497	11.86	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
4498	11.85	kd	CGS001-2837	UTS2R	Urotensin receptor			
4499	11.85	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
4500	11.81	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
4501	11.8	cc		SMAD family LOF	-			
4502	11.8	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
4503	11.8	oe	ccsbBroad304_08365	CYCS	-			
4504	11.78	kd	CGS001-205	AK4	Adenylate kinases			
4505	11.76	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
4506	11.75	kd	CGS001-58472	SQRDL	-			
4507	11.73	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
4508	11.68	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
4509	11.66	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
4510	11.6	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
4511	11.6	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
4512	11.59	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
4513	11.58	kd	CGS001-7431	VIM	Intermediate filaments type III			
4514	11.56	kd	CGS001-1128	CHRM1	Cholinergic receptors			
4515	11.55	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
4516	11.49	oe	ccsbBroad304_00949	LRPAP1	-			
4517	11.48	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
4518	11.43	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
4519	11.4	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4520	11.4	kd	CGS001-488	ATP2A2	Calcium-ATPases			
4521	11.39	kd	CGS001-5253	PHF2	Histone demethylases			
4522	11.38	kd	CGS001-515	ATP5F1	ATPases / F-type			
4523	11.37	kd	CGS001-2879	GPX4	-			
4524	11.34	kd	CGS001-221895	JAZF1	Zinc fingers, C2H2-type			
4525	11.34	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4526	11.32	kd	CGS001-2782	GNB1	WD repeat domain containing			
4527	11.31	kd	CGS001-7086	TKT	-			
4528	11.3	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
4529	11.29	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
4530	11.28	kd	CGS001-26523	EIF2C1	-			
4531	11.27	kd	CGS001-637	BID	Endogenous ligands			
4532	11.26	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
4533	11.25	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
4534	11.24	cc		Purinergic receptors P2Y GOF	-			
4535	11.23	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
4536	11.18	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
4537	11.17	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
4538	11.16	oe	ccsbBroad304_00329	CLTA	-			
4539	11.11	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
4540	11.09	kd	CGS001-4436	MSH2	-			
4541	11.06	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
4542	11.02	cp	BRD-A39172021	ampiroxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4543	10.96	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
4544	10.96	oe	ccsbBroad304_02837	BHMT2	-			
4545	10.94	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
4546	10.87	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
4547	10.87	oe	ccsbBroad304_06383	HMMR	CD molecules			
4548	10.86	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
4549	10.85	cc		General transcription factors group 2 LOF	-			
4550	10.83	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
4551	10.83	oe	ccsbBroad304_04379	LZIC	-			
4552	10.82	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
4553	10.8	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
4554	10.78	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
4555	10.76	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
4556	10.66	kd	CGS001-3827	KNG1	Endogenous ligands			
4557	10.62	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
4558	10.61	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
4559	10.6	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
4560	10.56	kd	CGS001-7477	WNT7B	Endogenous ligands			
4561	10.56	kd	CGS001-27346	TMEM97	-			
4562	10.55	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
4563	10.49	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
4564	10.48	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4565	10.47	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
4566	10.46	cp	BRD-K00673382	famotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
4567	10.46	oe	ccsbBroad304_01593	SRP14	-			
4568	10.43	kd	CGS001-10673	TNFSF13B	CD molecules			
4569	10.42	cc		Na-K-Cl transporter inhibitor	-			
4570	10.42	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
4571	10.4	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
4572	10.39	oe	ccsbBroad304_07511	KIF14	Kinesins			
4573	10.38	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
4574	10.34	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
4575	10.34	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
4576	10.34	kd	CGS001-51292	GMPR2	-			
4577	10.33	oe	ccsbBroad304_00486	EFNB2	Ephrins			
4578	10.32	kd	CGS001-27034	ACAD8	-			
4579	10.31	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
4580	10.31	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
4581	10.3	kd	CGS001-6493	SIM2	Basic helix-loop-helix proteins			
4582	10.23	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
4583	10.21	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
4584	10.2	oe	ccsbBroad304_04457	TOX2	-			
4585	10.18	kd	CGS001-9354	UBE4A	U-box domain containing			
4586	10.14	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
4587	10.13	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
4588	10.13	kd	CGS001-6217	RPS16	S ribosomal proteins			
4589	10.1	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
4590	10.1	kd	CGS001-51268	PIPOX	-			
4591	10.08	kd	CGS001-5501	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4592	10.05	oe	ccsbBroad304_00956	LYZ	-			
4593	10.03	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
4594	10.02	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
4595	10.02	kd	CGS001-2118	ETV4	ETS Transcription Factors			
4596	10.01	kd	CGS001-1906	EDN1	Endogenous ligands			
4597	9.98	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
4598	9.98	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
4599	9.97	kd	CGS001-23512	SUZ12	Zinc fingers, C2H2-type			
4600	9.97	kd	CGS001-7849	PAX8	Paired boxes			
4601	9.96	oe	ccsbBroad304_08266	PIPOX	-			
4602	9.96	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
4603	9.91	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
4604	9.9	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4605	9.87	oe	ccsbBroad304_10240	CROT	-			
4606	9.87	kd	CGS001-293	SLC25A6	Mitochondrial nucleotide transporter subfamily			
4607	9.83	cc		FXR antagonist	-			
4608	9.78	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
4609	9.75	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
4610	9.69	kd	CGS001-1399	CRKL	SH2 domain containing			
4611	9.68	kd	CGS001-129685	TAF8	-			
4612	9.68	kd	CGS001-3708	ITPR1	Ion channels / Inositol triphosphate receptors			
4613	9.65	kd	CGS001-55802	DCP1A	-			
4614	9.62	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
4615	9.61	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
4616	9.6	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
4617	9.58	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4618	9.58	kd	CGS001-55612	FERMT1	Fermitins			
4619	9.57	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
4620	9.56	kd	CGS001-22796	COG2	Components of oligomeric golgi complex			
4621	9.55	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
4622	9.52	oe	ccsbBroad304_13499	KSR2	RAF family			
4623	9.52	kd	CGS001-3242	HPD	Oxidoreductases			
4624	9.51	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
4625	9.51	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
4626	9.5	kd	CGS001-5170	PDPK1	PDK1 family			
4627	9.47	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
4628	9.46	kd	CGS001-57661	PHRF1	Zinc fingers, PHD-type			
4629	9.45	kd	CGS001-408	ARRB1	-			
4630	9.44	kd	CGS001-54541	DDIT4	-			
4631	9.41	oe	ccsbBroad304_01054	GADD45B	-			
4632	9.37	cc		PDGFR/KIT inhibitor	-			
4633	9.37	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
4634	9.36	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
4635	9.35	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
4636	9.35	kd	CGS001-5387	PMS2P3	-			
4637	9.33	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
4638	9.33	kd	CGS001-84875	PARP10	Poly (ADP-ribose) polymerases			
4639	9.31	kd	CGS001-79109	MAPKAP1	-			
4640	9.28	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
4641	9.26	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
4642	9.25	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
4643	9.25	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
4644	9.22	cc		Interleukin receptors LOF	-			
4645	9.22	kd	CGS001-998	CDC42	-			
4646	9.21	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
4647	9.18	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
4648	9.17	oe	ccsbBroad304_01373	RAN	-			
4649	9.13	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
4650	9.09	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4651	9.08	kd	CGS001-4323	MMP14	Matrix metallopeptidase			
4652	9.07	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
4653	9.06	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
4654	9.05	kd	CGS001-121549	ASCL4	Basic helix-loop-helix proteins			
4655	9.01	oe	ccsbBroad304_01841	BAG6	-			
4656	8.98	oe	ccsbBroad304_00370	CS	-			
4657	8.97	kd	CGS001-8935	SKAP2	Pleckstrin homology (PH) domain containing			
4658	8.96	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
4659	8.96	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
4660	8.92	oe	ccsbBroad304_03950	ATG3	-			
4661	8.9	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
4662	8.9	kd	CGS001-29102	DROSHA	-			
4663	8.88	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
4664	8.85	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4665	8.84	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
4666	8.82	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
4667	8.75	kd	CGS001-415116	PIM3	PIM family			
4668	8.75	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
4669	8.7	cc		MCM family LOF	-			
4670	8.7	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
4671	8.67	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
4672	8.66	cc		EGFR inhibitor	-			
4673	8.65	cp	BRD-K02227374	milnacipran	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Serotonin reuptake inhibitor
4674	8.63	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
4675	8.6	kd	CGS001-123803	NTAN1	-			
4676	8.53	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
4677	8.52	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
4678	8.5	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
4679	8.47	kd	CGS001-22887	FOXJ3	Forkhead boxes			
4680	8.45	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
4681	8.43	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
4682	8.42	cp	BRD-K88679075	methandriol	Androgenic steroid			Androgenic steroid
4683	8.41	kd	CGS001-55536	CDCA7L	-			
4684	8.29	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
4685	8.25	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
4686	8.21	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
4687	8.2	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
4688	8.16	kd	CGS001-2810	SFN	-			
4689	8.15	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
4690	8.15	oe	ccsbBroad304_00789	HSBP1	-			
4691	8.1	oe	ccsbBroad304_02370	HRSP12	-			
4692	8.09	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
4693	8.09	kd	CGS001-347736	NME9	-			
4694	8.08	oe	ccsbBroad304_06287	GM2A	-			
4695	8.01	kd	CGS001-5223	PGAM1	-			
4696	7.99	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
4697	7.96	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4698	7.93	oe	ccsbBroad304_01379	RBBP6	-			
4699	7.89	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
4700	7.88	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
4701	7.88	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
4702	7.87	kd	CGS001-4836	NMT1	-			
4703	7.83	oe	ccsbBroad304_03129	ERO1L	-			
4704	7.78	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
4705	7.76	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
4706	7.75	oe	ccsbBroad304_09578	PASD1	-			
4707	7.73	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
4708	7.69	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
4709	7.64	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
4710	7.62	kd	CGS001-3992	FADS1	Fatty acid desaturases			
4711	7.61	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
4712	7.61	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
4713	7.61	oe	ccsbBroad304_03808	ERGIC1	-			
4714	7.59	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
4715	7.57	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
4716	7.56	cp	BRD-K97752965	nicorandil	Nitric oxide donor		ABCC9, KCNJ11, KCNJ8	Nitric oxide donor, Potassium channel activator
4717	7.5	oe	ccsbBroad304_00472	EBF1	-			
4718	7.49	oe	ccsbBroad304_02372	SPRY1	-			
4719	7.48	kd	CGS001-5920	RARRES3	-			
4720	7.45	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
4721	7.41	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
4722	7.35	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
4723	7.34	oe	ccsbBroad304_05745	CD24	CD molecules			
4724	7.31	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
4725	7.31	oe	ccsbBroad304_01034	MSH2	-			
4726	7.3	kd	CGS001-5883	RAD9A	-			
4727	7.17	kd	CGS001-11019	LIAS	-			
4728	7.15	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
4729	7.13	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
4730	7.13	kd	CGS001-256281	NUDT14	Nudix motif containing			
4731	7.12	kd	CGS001-65975	STK33	CAMK-unique family			
4732	7.09	kd	CGS001-10078	TSSC4	-			
4733	7.08	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
4734	7.08	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
4735	7.07	kd	CGS001-4683	NBN	-			
4736	7.04	oe	ccsbBroad304_02136	COPS2	-			
4737	7.03	kd	CGS001-9641	IKBKE	IKK family			
4738	7.01	cp	BRD-A70083328	secnidazole	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Microtubule inhibitor, Antiprotozoal
4739	7	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
4740	6.94	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
4741	6.94	kd	CGS001-54555	DDX49	DEAD-boxes			
4742	6.93	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
4743	6.92	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
4744	6.92	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
4745	6.9	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
4746	6.86	kd	CGS001-2277	FIGF	-			
4747	6.84	oe	ccsbBroad304_02349	MPHOSPH9	-			
4748	6.83	kd	CGS001-54861	SNRK	SNRK subfamily			
4749	6.81	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
4750	6.81	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
4751	6.81	kd	CGS001-7423	VEGFB	-			
4752	6.79	kd	CGS001-5033	P4HA1	-			
4753	6.76	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
4754	6.75	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
4755	6.72	cp	BRD-K65910366	KUC103904N	-666			-666
4756	6.71	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
4757	6.7	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
4758	6.69	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
4759	6.69	kd	CGS001-5580	PRKCD	Delta subfamily			
4760	6.69	oe	ccsbBroad304_00962	SMAD4	SMADs			
4761	6.66	kd	CGS001-2821	GPI	-			
4762	6.64	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
4763	6.61	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
4764	6.57	oe	ccsbBroad304_00836	IGF2	-			
4765	6.55	kd	CGS001-444	ASPH	-			
4766	6.53	oe	ccsbBroad304_06424	IFI16	-			
4767	6.53	oe	ccsbBroad304_00809	HUS1	-			
4768	6.5	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
4769	6.47	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
4770	6.46	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
4771	6.43	kd	CGS001-1875	E2F5	-			
4772	6.39	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
4773	6.37	oe	ccsbBroad304_01084	NEU1	-			
4774	6.31	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
4775	6.27	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
4776	6.23	kd	CGS001-3832	KIF11	Kinesins			
4777	6.22	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
4778	6.2	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
4779	6.17	kd	CGS001-836	CASP3	Caspases			
4780	6.16	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
4781	6.12	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4782	6.11	kd	CGS001-2475	MTOR	FRAP subfamily			
4783	6.05	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
4784	6.03	kd	CGS001-10421	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4785	6.02	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
4786	6.01	kd	CGS001-10873	ME3	-			
4787	5.97	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
4788	5.97	oe	ccsbBroad304_00152	BCAT2	-			
4789	5.95	kd	CGS001-892	CCNC	-			
4790	5.89	oe	ccsbBroad304_00398	CTSL2	-			
4791	5.88	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
4792	5.88	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
4793	5.87	kd	CGS001-51734	SEPX1	-			
4794	5.8	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
4795	5.79	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
4796	5.79	oe	ccsbBroad304_07478	CCP110	-			
4797	5.79	oe	ccsbBroad304_07012	STK3	MST subfamily			
4798	5.76	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
4799	5.75	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
4800	5.74	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
4801	5.67	oe	ccsbBroad304_01347	RAD1	-			
4802	5.67	oe	ccsbBroad304_07277	RTCD1	-			
4803	5.66	oe	ccsbBroad304_06952	SKP1	-			
4804	5.66	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
4805	5.63	kd	CGS001-310	ANXA7	Annexins			
4806	5.6	oe	ccsbBroad304_01184	PGK1	-			
4807	5.57	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
4808	5.56	kd	CGS001-865	CBFB	-			
4809	5.51	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
4810	5.5	cc		Potassium channel activator	-			
4811	5.47	kd	CGS001-4097	MAFG	-			
4812	5.45	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
4813	5.4	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
4814	5.37	oe	ccsbBroad304_01372	RALB	-			
4815	5.36	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
4816	5.33	kd	CGS001-7525	YES1	Src family			
4817	5.29	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
4818	5.29	kd	CGS001-4664	NAB1	-			
4819	5.28	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
4820	5.27	oe	ccsbBroad304_01105	PNP	-			
4821	5.25	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
4822	5.17	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4823	5.05	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
4824	5	kd	CGS001-64223	MLST8	WD repeat domain containing			
4825	4.95	oe	ccsbBroad304_06134	ECH1	-			
4826	4.93	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
4827	4.9	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
4828	4.84	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
4829	4.79	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
4830	4.7	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
4831	4.69	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
4832	4.62	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
4833	4.58	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
4834	4.53	kd	CGS001-4668	NAGA	-			
4835	4.5	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
4836	4.44	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
4837	4.44	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
4838	4.39	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
4839	4.33	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
4840	4.32	kd	CGS001-55699	IARS2	Aminoacyl tRNA synthetases / Class I			
4841	4.31	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
4842	4.26	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
4843	4.26	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
4844	4.23	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4845	4.23	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
4846	4.21	oe	ccsbBroad304_00570	FIGF	-			
4847	4.13	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
4848	4.12	oe	ccsbBroad304_06144	EFNB3	Ephrins			
4849	4.12	kd	CGS001-5573	PRKAR1A	Protein kinase A			
4850	4.08	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
4851	4.07	cc		Canonical high mobility group proteins LOF	-			
4852	4	kd	CGS001-169436	C9ORF96	-			
4853	3.97	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
4854	3.95	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
4855	3.94	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
4856	3.93	oe	ccsbBroad304_02580	TMED10	-			
4857	3.93	oe	ccsbBroad304_01166	PDK2	PDHK family			
4858	3.92	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
4859	3.84	oe	ccsbBroad304_06916	SCP2	-			
4860	3.79	cp	BRD-K28849549	mesalazine	Cyclooxygenase inhibitor		PTGS1, PPARG, PTGS2, ALOX5, CHUK, CTNNB1, IKBKB, MPO, NAT1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor, Prostanoid receptor antagonist
4861	3.63	oe	ccsbBroad304_00661	GNGT2	-			
4862	3.57	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
4863	3.52	cc		KCNJ11 modulator	-			
4864	3.52	kd	CGS001-11200	CHEK2	CHK1 subfamily			
4865	3.52	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
4866	3.52	oe	ccsbBroad304_01035	MSH5	-			
4867	3.49	cc		IL4 Pathway LOF	-			
4868	3.38	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
4869	3.34	cc		G2 M Checkpoint LOF	-			
4870	3.24	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
4871	3.23	oe	ccsbBroad304_07800	EXOSC8	-			
4872	3.21	cp	BRD-K29530284	amlexanox	Histamine receptor modulator		FGF1, IL3, S100A12, S100A13	Histamine receptor modulator
4873	3.19	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
4874	3.19	cp	BRD-K30563334	rifabutin	Protein synthesis inhibitor		CYP3A4, HSP90AA1, HSP90B1	Protein synthesis inhibitor
4875	3.15	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
4876	3.1	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
4877	2.95	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
4878	2.75	cc		HMGCR inhibitor	-			
4879	2.5	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
4880	2.45	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
4881	2.41	cc		Akt Signaling LOF	-			
4882	2.23	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
4883	2.17	cc		SRY LOF	-			
4884	2.13	oe	ccsbBroad304_02487	TXNIP	-			
4885	2.04	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
4886	1.97	kd	CGS001-31	ACACA	Carboxylases			
4887	1.9	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
4888	1.85	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
4889	1.71	oe	ccsbBroad304_06178	ERCC5	-			
4890	1.4	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
4891	1.3	oe	ccsbBroad304_00009	ACLY	-			
4892	1.2	oe	ccsbBroad304_06852	RBP4	Lipocalins			
4893	1.09	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
4894	0.26	kd	CGS001-1111	CHEK1	CHK1 subfamily			
4895	-0.89	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
4896	-1.13	cc		Calcium channel blocker	-			
4897	-1.55	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
4898	-1.67	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
4899	-1.8	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
4900	-1.83	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
4901	-1.87	cc		Progesterone receptor antagonist	-			
4902	-2.27	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
4903	-2.31	oe	ccsbBroad304_06004	CKB	-			
4904	-2.36	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
4905	-2.39	cc		Androgen receptor modulator	-			
4906	-2.45	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
4907	-2.49	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
4908	-2.64	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
4909	-2.69	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
4910	-2.78	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4911	-2.83	kd	CGS001-501	ALDH7A1	Aldehyde dehydrogenases			
4912	-2.93	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
4913	-2.99	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
4914	-3.1	oe	ccsbBroad304_01091	NFIB	-			
4915	-3.15	oe	ccsbBroad304_01556	SMARCB1	-			
4916	-3.33	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
4917	-3.47	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
4918	-3.51	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
4919	-3.52	oe	ccsbBroad304_03191	NOSIP	-			
4920	-3.56	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
4921	-3.56	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
4922	-3.56	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
4923	-3.61	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
4924	-3.66	oe	ccsbBroad304_07768	NISCH	-			
4925	-3.7	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
4926	-3.74	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
4927	-3.76	kd	CGS001-1632	ECI1	-			
4928	-4.06	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
4929	-4.07	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
4930	-4.1	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
4931	-4.11	kd	CGS001-708	C1QBP	-			
4932	-4.12	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
4933	-4.18	cc		Vitamin D receptor agonist	-			
4934	-4.29	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
4935	-4.4	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
4936	-4.43	cc		Rho GTPase activating proteins LOF	-			
4937	-4.43	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
4938	-4.58	cp	BRD-K86887724	dofetilide	Potassium channel blocker		KCNH2, KCNH1, KCNJ12, KCNK2	Potassium channel blocker
4939	-4.58	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
4940	-4.61	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
4941	-4.63	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
4942	-4.7	kd	CGS001-83999	KREMEN1	-			
4943	-4.72	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4944	-4.75	cp	BRD-K10065684	dantron	Laxative			Laxative
4945	-4.77	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
4946	-4.91	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4947	-4.94	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
4948	-4.95	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
4949	-4.95	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
4950	-4.99	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
4951	-5.01	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
4952	-5.04	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
4953	-5.05	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
4954	-5.1	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
4955	-5.19	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
4956	-5.19	oe	ccsbBroad304_03182	GLOD4	-			
4957	-5.19	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
4958	-5.21	oe	ccsbBroad304_03652	EXOC2	-			
4959	-5.23	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
4960	-5.24	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
4961	-5.28	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
4962	-5.29	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
4963	-5.35	oe	ccsbBroad304_07724	KDELR2	-			
4964	-5.37	oe	ccsbBroad304_06089	DDIT3	-			
4965	-5.39	oe	ccsbBroad304_02306	PQBP1	-			
4966	-5.46	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
4967	-5.46	oe	ccsbBroad304_02197	VPS26A	-			
4968	-5.47	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
4969	-5.49	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
4970	-5.49	oe	ccsbBroad304_06671	OPA1	-			
4971	-5.52	oe	ccsbBroad304_06569	MCM5	-			
4972	-5.57	oe	ccsbBroad304_13891	LCK	Src family			
4973	-5.67	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
4974	-5.67	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
4975	-5.71	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
4976	-5.74	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
4977	-5.76	oe	ccsbBroad304_03767	TOMM22	-			
4978	-5.79	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
4979	-5.81	oe	ccsbBroad304_04775	NTAN1	-			
4980	-5.82	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
4981	-5.9	oe	ccsbBroad304_00969	MAGEA10	-			
4982	-5.92	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
4983	-5.97	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
4984	-5.98	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
4985	-5.98	kd	CGS001-433	ASGR2	C-type lectin domain containing			
4986	-6	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
4987	-6	kd	CGS001-900	CCNG1	-			
4988	-6.02	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
4989	-6.05	kd	CGS001-5202	PFDN2	-			
4990	-6.07	kd	CGS001-7280	TUBB2A	Tubulins			
4991	-6.12	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
4992	-6.15	kd	CGS001-8702	B4GALT4	Beta 4-glycosyltransferases			
4993	-6.16	kd	CGS001-2664	GDI1	-			
4994	-6.2	oe	ccsbBroad304_06845	RARRES3	-			
4995	-6.21	kd	CGS001-116113	FOXP4	Forkhead boxes			
4996	-6.27	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
4997	-6.29	kd	CGS001-4758	NEU1	-			
4998	-6.3	kd	CGS001-7771	ZFP112	-			
4999	-6.31	oe	ccsbBroad304_01147	PC	Carboxylases			
5000	-6.36	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
5001	-6.37	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
5002	-6.38	kd	CGS001-8408	ULK1	Unc-51-like kinase (ULK) family			
5003	-6.47	oe	ccsbBroad304_08217	SCCPDH	-			
5004	-6.49	kd	CGS001-54108	CHRAC1	-			
5005	-6.67	oe	ccsbBroad304_04194	ELL3	-			
5006	-6.67	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
5007	-6.69	oe	ccsbBroad304_00162	BIK	-			
5008	-6.71	kd	CGS001-29105	C16ORF80	-			
5009	-6.78	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
5010	-6.79	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
5011	-6.97	kd	CGS001-1649	DDIT3	-			
5012	-6.99	cc		Potassium channel blocker	-			
5013	-7.03	oe	ccsbBroad304_06095	DFFB	-			
5014	-7.08	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
5015	-7.1	kd	CGS001-638	BIK	-			
5016	-7.15	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
5017	-7.16	kd	CGS001-10048	RANBP9	-			
5018	-7.17	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
5019	-7.18	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
5020	-7.18	kd	CGS001-7089	TLE2	WD repeat domain containing			
5021	-7.25	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
5022	-7.31	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
5023	-7.33	kd	CGS001-3673	ITGA2	Integrins			
5024	-7.36	oe	ccsbBroad304_01664	TGFA	-			
5025	-7.4	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
5026	-7.42	kd	CGS001-10465	PPIH	-			
5027	-7.47	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
5028	-7.5	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
5029	-7.54	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
5030	-7.54	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
5031	-7.56	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
5032	-7.61	cp	BRD-K66896231	BRD-K66896231	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5033	-7.62	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
5034	-7.63	kd	CGS001-6210	RPS15A	S ribosomal proteins			
5035	-7.63	kd	CGS001-2863	GPR39	GPCR / Class A : Orphans			
5036	-7.64	oe	ccsbBroad304_02157	MED21	-			
5037	-7.65	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
5038	-7.65	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
5039	-7.66	kd	CGS001-3565	IL4	Interleukins and interleukin receptors			
5040	-7.73	kd	CGS001-5211	PFKL	-			
5041	-7.77	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
5042	-7.77	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
5043	-7.78	cc		HOXL subclass homeoboxes LOF	-			
5044	-7.84	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
5045	-7.84	kd	CGS001-308	ANXA5	Annexins			
5046	-7.86	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
5047	-7.86	kd	CGS001-4665	NAB2	-			
5048	-7.87	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
5049	-7.89	kd	CGS001-10165	SLC25A13	Mitochondrial amino acid transporter subfamily			
5050	-7.93	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
5051	-7.93	kd	CGS001-6934	TCF7L2	-			
5052	-7.95	kd	CGS001-51776	ZAK	MLK subfamily			
5053	-7.96	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5054	-7.98	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
5055	-8.08	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
5056	-8.11	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
5057	-8.13	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
5058	-8.14	cc		Glycogen synthase kinase inhibitor	-			
5059	-8.15	oe	ccsbBroad304_08709	SCYL3	-			
5060	-8.16	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
5061	-8.22	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
5062	-8.24	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
5063	-8.25	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
5064	-8.27	oe	ccsbBroad304_02862	CCRN4L	-			
5065	-8.29	kd	CGS001-22930	RAB3GAP1	-			
5066	-8.37	oe	ccsbBroad304_03235	TUBD1	Tubulins			
5067	-8.41	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
5068	-8.43	kd	CGS001-7471	WNT1	Endogenous ligands			
5069	-8.45	cc		Ribonucleotide reductase inhibitor	-			
5070	-8.49	kd	CGS001-10616	RBCK1	RING-type (C3HC4) zinc fingers			
5071	-8.51	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
5072	-8.52	cc		Serotonin receptor antagonist	-			
5073	-8.52	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
5074	-8.52	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
5075	-8.54	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
5076	-8.58	kd	CGS001-3669	ISG20	-			
5077	-8.61	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
5078	-8.61	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
5079	-8.63	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
5080	-8.66	kd	CGS001-2155	F7	Chymotrypsin			
5081	-8.68	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
5082	-8.74	kd	CGS001-22978	NT5C2	Adenosine turnover			
5083	-8.77	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
5084	-8.77	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
5085	-8.79	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
5086	-8.8	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5087	-8.81	kd	CGS001-284119	PTRF	-			
5088	-8.83	kd	CGS001-29883	CNOT7	-			
5089	-8.83	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
5090	-8.88	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
5091	-8.89	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
5092	-8.92	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
5093	-8.94	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
5094	-8.95	oe	ccsbBroad304_07119	UGP2	-			
5095	-9	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
5096	-9.04	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
5097	-9.07	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
5098	-9.07	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
5099	-9.13	oe	ccsbBroad304_10491	PFKL	-			
5100	-9.17	kd	CGS001-716	C1S	Complement system			
5101	-9.18	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5102	-9.18	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
5103	-9.19	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
5104	-9.21	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
5105	-9.21	kd	CGS001-2872	MKNK2	MKN subfamily			
5106	-9.24	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
5107	-9.24	oe	ccsbBroad304_00462	DR1	-			
5108	-9.26	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
5109	-9.38	oe	ccsbBroad304_02919	KIAA1279	-			
5110	-9.44	kd	CGS001-6721	SREBF2	Basic helix-loop-helix proteins			
5111	-9.5	oe	ccsbBroad304_02239	RASSF2	-			
5112	-9.58	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
5113	-9.59	cp	BRD-A96107863	nisoldipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNB2, CYP3A5	Calcium channel blocker
5114	-9.6	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
5115	-9.61	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
5116	-9.67	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
5117	-9.7	oe	ccsbBroad304_02318	KIF20A	Kinesins			
5118	-9.7	oe	ccsbBroad304_00615	GAPDH	-			
5119	-9.73	oe	ccsbBroad304_02271	LPGAT1	-			
5120	-9.78	kd	CGS001-8802	SUCLG1	-			
5121	-9.78	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
5122	-9.79	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
5123	-9.82	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
5124	-9.87	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
5125	-9.91	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
5126	-10.05	oe	ccsbBroad304_07337	TAF1B	-			
5127	-10.05	kd	CGS001-3161	HMMR	CD molecules			
5128	-10.08	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
5129	-10.08	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
5130	-10.11	cc		PPAR receptor agonist	-			
5131	-10.14	kd	CGS001-8872	CDC123	-			
5132	-10.18	kd	CGS001-3725	JUN	basic leucine zipper proteins			
5133	-10.18	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
5134	-10.19	kd	CGS001-7100	TLR5	Toll-like receptor family			
5135	-10.19	kd	CGS001-7879	RAB7A	RAB, member RAS oncogene			
5136	-10.24	cp	BRD-K33106058	cytarabine	Ribonucleotide reductase inhibitor		POLB, POLA1	Ribonucleotide reductase inhibitor
5137	-10.25	cp	BRD-A24543851	nornicotine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
5138	-10.27	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5139	-10.28	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
5140	-10.29	cp	BRD-K07237224	moclobemide	Monoamine oxidase inhibitor		MAOA, CYP2C19, MAOB	Monoamine oxidase inhibitor
5141	-10.32	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
5142	-10.32	oe	ccsbBroad304_00883	ISG20	-			
5143	-10.36	kd	CGS001-1856	DVL2	Dishevelled homologs			
5144	-10.38	cp	BRD-K39391626	ethylestrenol	Progesterone receptor agonist		AR	Progesterone receptor agonist
5145	-10.42	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
5146	-10.49	oe	ccsbBroad304_06349	HAGH	-			
5147	-10.5	kd	CGS001-11336	EXOC3	-			
5148	-10.5	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
5149	-10.51	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5150	-10.52	oe	ccsbBroad304_03798	PHTF2	-			
5151	-10.53	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
5152	-10.53	cp	BRD-K62858456	lomerizine	Calcium channel blocker		ABCB1, CACNA1B, SCN5A	Calcium channel blocker
5153	-10.57	cp	BRD-K54316499	tolterodine	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRM1, CHRM4, CHRM5	Acetylcholine receptor antagonist
5154	-10.57	kd	CGS001-6932	TCF7	-			
5155	-10.62	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
5156	-10.71	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
5157	-10.73	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
5158	-10.78	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
5159	-10.85	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
5160	-10.87	kd	CGS001-1840	DTX1	-			
5161	-10.95	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
5162	-10.96	kd	CGS001-387	RHOA	-			
5163	-10.99	oe	ccsbBroad304_01623	SUPT4H1	-			
5164	-10.99	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
5165	-10.99	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
5166	-11	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
5167	-11	oe	ccsbBroad304_07118	UGDH	-			
5168	-11.01	kd	CGS001-10969	EBNA1BP2	-			
5169	-11.02	kd	CGS001-85442	KNDC1	-			
5170	-11.11	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
5171	-11.12	oe	ccsbBroad304_07798	EXOC3	-			
5172	-11.13	kd	CGS001-771	CA12	Carbonic anhydrases			
5173	-11.19	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
5174	-11.2	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
5175	-11.22	kd	CGS001-150280	HORMAD2	-			
5176	-11.28	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
5177	-11.28	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
5178	-11.29	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
5179	-11.36	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
5180	-11.37	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
5181	-11.38	kd	CGS001-4087	SMAD2	SMADs			
5182	-11.39	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
5183	-11.4	oe	ccsbBroad304_04202	MED28	-			
5184	-11.41	kd	CGS001-641	BLM	-			
5185	-11.44	kd	CGS001-3248	HPGD	Prostaglandin synthases			
5186	-11.46	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
5187	-11.46	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
5188	-11.48	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
5189	-11.49	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
5190	-11.52	oe	ccsbBroad304_00658	GNG5	-			
5191	-11.56	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
5192	-11.58	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
5193	-11.58	kd	CGS001-100	ADA	Adenosine turnover			
5194	-11.59	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
5195	-11.62	kd	CGS001-4300	MLLT3	-			
5196	-11.64	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
5197	-11.68	kd	CGS001-51545	ZNF581	Zinc fingers, C2H2-type			
5198	-11.68	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
5199	-11.7	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
5200	-11.7	kd	CGS001-9441	MED26	-			
5201	-11.71	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
5202	-11.73	kd	CGS001-9122	SLC16A4	SLC16 family of monocarboxylate transporters			
5203	-11.8	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
5204	-11.89	kd	CGS001-1028	CDKN1C	-			
5205	-11.91	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5206	-11.93	kd	CGS001-327	APEH	Prolyl oligopeptidase			
5207	-11.98	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
5208	-11.98	kd	CGS001-3596	IL13	Interleukins and interleukin receptors			
5209	-12.04	oe	ccsbBroad304_03618	OSGEP	-			
5210	-12.06	oe	ccsbBroad304_02500	RRAGA	-			
5211	-12.07	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
5212	-12.11	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
5213	-12.12	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
5214	-12.13	kd	CGS001-3265	HRAS	RAS subfamily			
5215	-12.14	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
5216	-12.18	kd	CGS001-7150	TOP1	DNA Topoisomerases			
5217	-12.18	kd	CGS001-3119	HLA-DQB1	Immunoglobulin superfamily / C1-set domain containing			
5218	-12.24	kd	CGS001-1152	CKB	-			
5219	-12.26	kd	CGS001-7342	UBP1	-			
5220	-12.3	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
5221	-12.3	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
5222	-12.37	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
5223	-12.38	kd	CGS001-8031	NCOA4	-			
5224	-12.43	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
5225	-12.44	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
5226	-12.46	oe	ccsbBroad304_02686	COPZ1	-			
5227	-12.47	oe	ccsbBroad304_06663	OAS1	-			
5228	-12.5	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5229	-12.52	cp	BRD-A16444946	acarbose	Glucosidase inhibitor		GAA, MGAM, AMY2A, SI	Glucosidase inhibitor
5230	-12.52	kd	CGS001-539	ATP5O	ATPases / F-type			
5231	-12.53	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
5232	-12.56	kd	CGS001-51176	LEF1	-			
5233	-12.7	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
5234	-12.7	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
5235	-12.71	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
5236	-12.75	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
5237	-12.76	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
5238	-12.77	cc		DNA synthesis inhibitor	-			
5239	-12.77	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
5240	-12.8	cc		DNA dependent protein kinase inhibitor	-			
5241	-12.9	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
5242	-12.91	kd	CGS001-7054	TH	Amino acid hydroxylases			
5243	-12.92	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
5244	-13	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
5245	-13.01	oe	ccsbBroad304_03372	CAB39	-			
5246	-13.01	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
5247	-13.02	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
5248	-13.06	oe	ccsbBroad304_00161	BID	Endogenous ligands			
5249	-13.06	cp	BRD-K52080565	rilmenidine	Imidazoline receptor agonist		NISCH	Imidazoline receptor agonist
5250	-13.07	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
5251	-13.08	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
5252	-13.08	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
5253	-13.14	kd	CGS001-4254	KITLG	-			
5254	-13.15	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
5255	-13.2	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
5256	-13.2	kd	CGS001-6663	SOX10	SRY (sex determining region Y)-boxes			
5257	-13.23	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5258	-13.24	kd	CGS001-55054	ATG16L1	WD repeat domain containing			
5259	-13.25	oe	ccsbBroad304_02115	PTTG1	-			
5260	-13.3	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
5261	-13.3	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
5262	-13.43	oe	ccsbBroad304_00390	CTGF	-			
5263	-13.54	kd	CGS001-9690	UBE3C	-			
5264	-13.56	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
5265	-13.6	kd	CGS001-5264	PHYH	-			
5266	-13.6	kd	CGS001-1786	DNMT1	Methyltransferases			
5267	-13.63	oe	ccsbBroad304_06040	CRY1	-			
5268	-13.66	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
5269	-13.67	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
5270	-13.67	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
5271	-13.7	kd	CGS001-1495	CTNNA1	Catenins			
5272	-13.74	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
5273	-13.75	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
5274	-13.75	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
5275	-13.75	oe	ccsbBroad304_03739	NRIP3	-			
5276	-13.77	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
5277	-13.81	oe	ccsbBroad304_04038	ELOVL6	-			
5278	-13.82	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
5279	-13.83	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
5280	-13.84	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
5281	-13.85	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
5282	-13.87	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
5283	-13.89	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
5284	-13.9	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
5285	-13.95	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
5286	-13.96	kd	CGS001-200879	LIPH	-			
5287	-13.99	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
5288	-14	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
5289	-14.07	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
5290	-14.1	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
5291	-14.11	cp	BRD-K56450366	NSC-94258	Antineoplastic		AKR1B1, CYP19A1, HSD17B1	Antineoplastic
5292	-14.11	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
5293	-14.19	kd	CGS001-4552	MTRR	-			
5294	-14.21	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
5295	-14.28	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
5296	-14.29	kd	CGS001-84759	PCGF1	Polycomb group ring fingers			
5297	-14.3	kd	CGS001-25	ABL1	Abl family			
5298	-14.33	kd	CGS001-6775	STAT4	SH2 domain containing			
5299	-14.33	kd	CGS001-5900	RALGDS	-			
5300	-14.36	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
5301	-14.42	kd	CGS001-58508	MLL3	-			
5302	-14.43	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
5303	-14.45	oe	ccsbBroad304_03850	TRIB3	Trbl family			
5304	-14.46	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
5305	-14.48	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
5306	-14.49	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
5307	-14.49	kd	CGS001-7248	TSC1	-			
5308	-14.51	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
5309	-14.51	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
5310	-14.54	kd	CGS001-5565	PRKAB2	AMPK subfamily			
5311	-14.55	oe	ccsbBroad304_07128	VHL	-			
5312	-14.56	cp	BRD-K51671335	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
5313	-14.57	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
5314	-14.61	kd	CGS001-1647	GADD45A	-			
5315	-14.64	kd	CGS001-29968	PSAT1	-			
5316	-14.64	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5317	-14.65	kd	CGS001-51752	ERAP1	Aminopeptidase N			
5318	-14.72	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
5319	-14.8	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5320	-14.82	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
5321	-14.82	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5322	-14.83	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
5323	-14.84	kd	CGS001-3170	FOXA2	Forkhead boxes			
5324	-14.87	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
5325	-14.91	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
5326	-14.92	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
5327	-14.92	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
5328	-14.96	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
5329	-14.97	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
5330	-15	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
5331	-15.03	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
5332	-15.04	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
5333	-15.06	oe	ccsbBroad304_03119	C16ORF5	-			
5334	-15.12	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
5335	-15.22	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
5336	-15.27	kd	CGS001-891	CCNB1	-			
5337	-15.34	cp	BRD-K25310650	ormetoprim	Bacterial antifolate			Bacterial antifolate
5338	-15.34	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
5339	-15.36	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
5340	-15.36	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
5341	-15.38	cp	BRD-A88254928	salbutamol	Adrenergic receptor agonist		ADRB2, ADRB1	Adrenergic receptor agonist
5342	-15.39	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
5343	-15.46	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
5344	-15.46	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
5345	-15.47	kd	CGS001-158	ADSL	-			
5346	-15.48	kd	CGS001-3163	HMOX2	Haem oxygenase			
5347	-15.51	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
5348	-15.51	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
5349	-15.52	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5350	-15.53	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
5351	-15.57	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
5352	-15.58	oe	ccsbBroad304_01769	VEGFB	-			
5353	-15.58	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
5354	-15.59	oe	ccsbBroad304_06172	EPS8	-			
5355	-15.62	kd	CGS001-4700	NDUFA6	LYR motif containing			
5356	-15.65	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
5357	-15.73	kd	CGS001-4711	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
5358	-15.73	kd	CGS001-10285	SMNDC1	Tudor domain containing			
5359	-15.73	kd	CGS001-6277	S100A6	EF-hand domain containing			
5360	-15.75	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
5361	-15.75	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
5362	-15.76	oe	ccsbBroad304_06350	HAL	-			
5363	-15.79	oe	ccsbBroad304_02840	PISD	Decarboxylases			
5364	-15.79	oe	ccsbBroad304_01152	PCNA	-			
5365	-15.82	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
5366	-15.82	kd	CGS001-23102	TBC1D2B	-			
5367	-15.84	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
5368	-15.86	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
5369	-15.88	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
5370	-16.02	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
5371	-16.03	kd	CGS001-1493	CTLA4	CD molecules			
5372	-16.04	oe	ccsbBroad304_03853	LSM2	-			
5373	-16.04	oe	ccsbBroad304_03591	ETNK1	-			
5374	-16.07	kd	CGS001-51284	TLR7	Toll-like receptor family			
5375	-16.1	oe	ccsbBroad304_02143	CNOT8	-			
5376	-16.11	kd	CGS001-151742	PPM1L	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
5377	-16.16	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
5378	-16.17	kd	CGS001-3718	JAK3	Janus kinase (JakA) family			
5379	-16.19	oe	ccsbBroad304_07238	STK24	YSK subfamily			
5380	-16.2	oe	ccsbBroad304_00072	ANXA7	Annexins			
5381	-16.24	kd	CGS001-55631	LRRC40	-			
5382	-16.29	oe	ccsbBroad304_14291	GDPD5	-			
5383	-16.33	kd	CGS001-23566	LPAR3	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
5384	-16.37	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
5385	-16.37	kd	CGS001-25888	ZNF473	Zinc fingers, C2H2-type			
5386	-16.39	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
5387	-16.39	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
5388	-16.4	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
5389	-16.42	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
5390	-16.43	oe	ccsbBroad304_03155	DHH	-			
5391	-16.44	oe	ccsbBroad304_04406	PLA2G12B	-			
5392	-16.46	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5393	-16.47	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
5394	-16.5	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
5395	-16.5	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
5396	-16.5	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
5397	-16.51	cp	BRD-K06817181	BRD-K06817181	JAK inhibitor		JAK2	JAK inhibitor
5398	-16.51	cp	BRD-A79903587	tegafur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
5399	-16.58	kd	CGS001-11284	PNKP	-			
5400	-16.59	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
5401	-16.63	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
5402	-16.66	cp	BRD-K94649603	taxifolin	Opioid receptor antagonist		APOB, APP, HMGCR	Opioid receptor antagonist
5403	-16.74	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
5404	-16.76	kd	CGS001-2263	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
5405	-16.77	oe	ccsbBroad304_06549	SMAD3	SMADs			
5406	-16.79	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
5407	-16.79	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
5408	-16.83	kd	CGS001-64863	METTL4	-			
5409	-16.86	oe	ccsbBroad304_01222	PLP2	-			
5410	-16.89	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
5411	-16.89	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
5412	-16.89	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
5413	-16.93	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
5414	-16.96	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
5415	-17	kd	CGS001-10451	VAV3	Rho guanine nucleotide exchange factors			
5416	-17.01	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
5417	-17.01	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
5418	-17.02	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
5419	-17.04	oe	ccsbBroad304_00394	CTSD	Cathepsins			
5420	-17.07	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
5421	-17.08	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
5422	-17.09	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
5423	-17.09	oe	ccsbBroad304_00783	HPRT1	-			
5424	-17.1	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
5425	-17.13	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
5426	-17.14	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
5427	-17.18	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
5428	-17.2	kd	CGS001-9700	ESPL1	-			
5429	-17.22	kd	CGS001-6184	RPN1	-			
5430	-17.26	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
5431	-17.27	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
5432	-17.28	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
5433	-17.28	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
5434	-17.3	kd	CGS001-7572	ZNF24	Zinc fingers, C2H2-type			
5435	-17.33	oe	ccsbBroad304_09708	PNLDC1	-			
5436	-17.33	cp	BRD-A23359898	sibutramine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, CYP2B6, CYP2C19, CYP3A5	Serotonin reuptake inhibitor
5437	-17.34	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
5438	-17.39	cc		P38 MAPK inhibitor	-			
5439	-17.39	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
5440	-17.48	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
5441	-17.51	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
5442	-17.54	kd	CGS001-7037	TFRC	CD molecules			
5443	-17.57	kd	CGS001-2678	GGT1	CD molecules			
5444	-17.59	oe	ccsbBroad304_00077	APEX1	-			
5445	-17.59	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
5446	-17.63	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
5447	-17.68	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
5448	-17.68	kd	CGS001-513	ATP5D	ATPases / F-type			
5449	-17.68	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
5450	-17.69	kd	CGS001-7083	TK1	-			
5451	-17.7	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
5452	-17.72	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
5453	-17.72	cp	BRD-K73196317	urapidil	Adrenergic receptor antagonist		HTR1A	Adrenergic receptor antagonist
5454	-17.77	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
5455	-17.82	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
5456	-17.83	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
5457	-17.84	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
5458	-17.87	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
5459	-17.88	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
5460	-17.89	kd	CGS001-4704	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5461	-17.9	cp	BRD-K51730347	diphencyprone	Immunostimulant			Immunostimulant
5462	-17.95	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
5463	-17.95	kd	CGS001-85377	MICALL1	-			
5464	-18.03	oe	ccsbBroad304_02702	MSRB2	-			
5465	-18.05	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
5466	-18.08	oe	ccsbBroad304_06094	DFFA	-			
5467	-18.09	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
5468	-18.1	oe	ccsbBroad304_01148	PCBD1	-			
5469	-18.11	kd	CGS001-79618	HMBOX1	Homeoboxes / HNF class			
5470	-18.14	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
5471	-18.15	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
5472	-18.2	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
5473	-18.21	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
5474	-18.23	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
5475	-18.24	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
5476	-18.28	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
5477	-18.31	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
5478	-18.31	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
5479	-18.32	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
5480	-18.33	kd	CGS001-5471	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
5481	-18.34	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
5482	-18.38	kd	CGS001-132	ADK	Adenosine turnover			
5483	-18.48	oe	ccsbBroad304_00941	LIG3	-			
5484	-18.48	cp	BRD-A92630576	trimebutine	Opioid receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Opioid receptor agonist
5485	-18.48	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
5486	-18.49	kd	CGS001-2877	GPX2	-			
5487	-18.51	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
5488	-18.52	kd	CGS001-163688	CALML6	EF-hand domain containing			
5489	-18.55	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
5490	-18.57	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
5491	-18.57	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
5492	-18.57	kd	CGS001-563	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
5493	-18.58	kd	CGS001-81848	SPRY4	-			
5494	-18.58	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
5495	-18.66	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
5496	-18.69	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
5497	-18.74	kd	CGS001-1468	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
5498	-18.76	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5499	-18.79	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
5500	-18.79	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
5501	-18.81	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
5502	-18.82	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
5503	-18.82	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
5504	-18.85	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5505	-18.86	cp	BRD-K40758068	efavirenz	HIV protease inhibitor		CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5	HIV protease inhibitor
5506	-18.87	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
5507	-18.87	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
5508	-18.87	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
5509	-18.89	kd	CGS001-29947	DNMT3L	-			
5510	-18.93	oe	ccsbBroad304_02203	MAD2L1BP	-			
5511	-18.95	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
5512	-18.97	kd	CGS001-6189	RPS3A	S ribosomal proteins			
5513	-19.02	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5514	-19.09	kd	CGS001-55746	NUP133	-			
5515	-19.16	kd	CGS001-2878	GPX3	-			
5516	-19.21	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
5517	-19.21	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
5518	-19.28	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
5519	-19.37	kd	CGS001-11041	B3GNT1	-			
5520	-19.38	oe	ccsbBroad304_02815	SSBP2	-			
5521	-19.41	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
5522	-19.43	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
5523	-19.45	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
5524	-19.48	kd	CGS001-84930	MASTL	MAST family			
5525	-19.53	oe	ccsbBroad304_02737	JMJD6	-			
5526	-19.58	cp	BRD-K32311154	nifekalant	Potassium channel blocker			Potassium channel blocker
5527	-19.6	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5528	-19.62	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
5529	-19.63	kd	CGS001-262	AMD1	Decarboxylases			
5530	-19.69	kd	CGS001-23046	KIF21B	Kinesins			
5531	-19.7	kd	CGS001-11113	CIT	Other DMPK family kinases			
5532	-19.76	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
5533	-19.79	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
5534	-19.84	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
5535	-19.88	kd	CGS001-27148	STK36	Unc-51-like kinase (ULK) family			
5536	-19.91	kd	CGS001-4205	MEF2A	Myocyte enhancer factors			
5537	-19.92	kd	CGS001-7296	TXNRD1	-			
5538	-19.93	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
5539	-19.96	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
5540	-19.96	kd	CGS001-506	ATP5B	ATPases / F-type			
5541	-19.98	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
5542	-20.02	kd	CGS001-126823	KLHDC9	-			
5543	-20.03	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
5544	-20.04	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
5545	-20.05	kd	CGS001-54821	ERCC6L	-			
5546	-20.09	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
5547	-20.12	kd	CGS001-23466	CBX6	-			
5548	-20.14	kd	CGS001-10695	CNPY3	Trinucleotide (CAG) repeat containing			
5549	-20.19	kd	CGS001-2309	FOXO3	Forkhead boxes			
5550	-20.22	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5551	-20.24	kd	CGS001-10554	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
5552	-20.25	kd	CGS001-5612	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
5553	-20.25	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
5554	-20.25	kd	CGS001-392	ARHGAP1	Rho GTPase activating proteins			
5555	-20.25	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
5556	-20.27	kd	CGS001-10437	IFI30	-			
5557	-20.28	kd	CGS001-23057	NMNAT2	-			
5558	-20.3	oe	ccsbBroad304_06449	ILF3	-			
5559	-20.31	kd	CGS001-23355	VPS8	-			
5560	-20.32	oe	ccsbBroad304_08386	SMOX	-			
5561	-20.37	oe	ccsbBroad304_00223	CASP9	Caspases			
5562	-20.4	kd	CGS001-5111	PCNA	-			
5563	-20.43	kd	CGS001-375449	MAST4	MAST family			
5564	-20.47	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
5565	-20.5	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
5566	-20.51	kd	CGS001-165082	GPR113	Adhesion Class GPCRs			
5567	-20.51	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
5568	-20.51	oe	ccsbBroad304_05936	CASP2	Caspases			
5569	-20.52	kd	CGS001-80314	EPC1	-			
5570	-20.55	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
5571	-20.58	kd	CGS001-9703	KIAA0100	-			
5572	-20.63	kd	CGS001-8477	GPR65	GPCR / Class A : Orphans			
5573	-20.65	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
5574	-20.68	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
5575	-20.72	kd	CGS001-7337	UBE3A	-			
5576	-20.73	kd	CGS001-2243	FGA	Endogenous ligands			
5577	-20.74	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
5578	-20.81	kd	CGS001-7056	THBD	CD molecules			
5579	-20.82	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
5580	-20.84	kd	CGS001-1196	CLK2	CDC-like kinases			
5581	-20.86	oe	ccsbBroad304_03268	GMPR2	-			
5582	-20.86	kd	CGS001-7172	TPMT	-			
5583	-20.87	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
5584	-21.01	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
5585	-21.01	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
5586	-21.02	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
5587	-21.07	kd	CGS001-26277	TINF2	-			
5588	-21.08	oe	ccsbBroad304_00933	LDHB	-			
5589	-21.09	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
5590	-21.1	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
5591	-21.11	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
5592	-21.13	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5593	-21.15	oe	ccsbBroad304_00225	CAT	-			
5594	-21.18	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
5595	-21.19	oe	ccsbBroad304_02526	POP4	-			
5596	-21.22	oe	ccsbBroad304_06226	FTL	-			
5597	-21.23	kd	CGS001-4255	MGMT	-			
5598	-21.24	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
5599	-21.25	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
5600	-21.26	oe	ccsbBroad304_06789	PSEN2	Presenilin			
5601	-21.27	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
5602	-21.28	kd	CGS001-2588	GALNS	Arylsulfatase family			
5603	-21.32	oe	ccsbBroad304_06291	GNAI1	-			
5604	-21.33	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
5605	-21.34	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
5606	-21.34	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5607	-21.35	oe	ccsbBroad304_08660	SMARCAD1	-			
5608	-21.38	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
5609	-21.39	kd	CGS001-4507	MTAP	-			
5610	-21.41	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
5611	-21.43	oe	ccsbBroad304_01164	PDHB	-			
5612	-21.44	kd	CGS001-9443	MED7	-			
5613	-21.46	oe	ccsbBroad304_00115	ASPH	-			
5614	-21.49	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
5615	-21.52	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
5616	-21.53	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
5617	-21.54	oe	ccsbBroad304_06494	KLRC1	CD molecules			
5618	-21.56	cp	BRD-K41051431	mecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5619	-21.57	oe	ccsbBroad304_02415	TUBB3	Tubulins			
5620	-21.62	kd	CGS001-8692	HYAL2	-			
5621	-21.65	kd	CGS001-11136	SLC7A9	SLC7 family			
5622	-21.66	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
5623	-21.69	oe	ccsbBroad304_03179	BOLA1	-			
5624	-21.71	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
5625	-21.73	kd	CGS001-7919	DDX39B	DEAD-boxes			
5626	-21.78	kd	CGS001-11040	PIM2	PIM family			
5627	-21.79	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
5628	-21.79	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
5629	-21.8	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
5630	-21.8	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
5631	-21.8	oe	ccsbBroad304_06695	PCK2	-			
5632	-21.81	oe	ccsbBroad304_03450	TMED9	-			
5633	-21.82	oe	ccsbBroad304_00210	CALR	-			
5634	-21.83	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
5635	-21.84	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
5636	-21.88	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
5637	-21.91	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
5638	-21.93	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
5639	-21.97	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
5640	-21.98	kd	CGS001-54851	ANKRD49	Ankyrin repeat domain containing			
5641	-22	cc		Tachykinin antagonist	-			
5642	-22	kd	CGS001-8220	DGCR14	-			
5643	-22	oe	ccsbBroad304_04064	PRR15L	-			
5644	-22.01	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
5645	-22.04	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
5646	-22.04	kd	CGS001-4926	NUMA1	-			
5647	-22.05	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
5648	-22.06	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
5649	-22.06	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5650	-22.08	kd	CGS001-53347	UBASH3A	-			
5651	-22.1	oe	ccsbBroad304_06318	GPER	-			
5652	-22.11	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
5653	-22.11	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
5654	-22.12	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
5655	-22.14	kd	CGS001-113451	ADC	-			
5656	-22.15	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
5657	-22.18	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
5658	-22.19	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
5659	-22.19	kd	CGS001-23043	TNIK	MSN subfamily			
5660	-22.23	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
5661	-22.23	oe	ccsbBroad304_02605	PAPD7	-			
5662	-22.23	oe	ccsbBroad304_00841	IKBKB	IKK family			
5663	-22.27	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
5664	-22.32	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
5665	-22.39	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
5666	-22.44	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
5667	-22.55	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
5668	-22.56	kd	CGS001-9568	GABBR2	GABA receptors			
5669	-22.57	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
5670	-22.58	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5671	-22.62	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
5672	-22.66	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
5673	-22.8	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
5674	-22.82	kd	CGS001-10607	TBL3	WD repeat domain containing			
5675	-22.82	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
5676	-22.83	kd	CGS001-10314	LANCL1	-			
5677	-22.87	kd	CGS001-4929	NR4A2	Nerve growth factor IB-like receptors			
5678	-22.87	kd	CGS001-9275	BCL7B	-			
5679	-22.9	kd	CGS001-55234	SMU1	WD repeat domain containing			
5680	-22.97	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
5681	-23	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
5682	-23.01	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
5683	-23.03	kd	CGS001-6016	RIT1	-			
5684	-23.04	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
5685	-23.07	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
5686	-23.08	cc		FGFR inhibitor	-			
5687	-23.11	kd	CGS001-6194	RPS6	S ribosomal proteins			
5688	-23.13	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
5689	-23.15	oe	ccsbBroad304_03097	CNOT7	-			
5690	-23.2	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
5691	-23.22	kd	CGS001-2834	PRLHR	GPCR / Class A : RF amide peptide receptors			
5692	-23.28	cp	BRD-K81169441	cerivastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A5	HMGCR inhibitor
5693	-23.28	oe	ccsbBroad304_13880	IDH3G	-			
5694	-23.29	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
5695	-23.3	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
5696	-23.32	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
5697	-23.35	oe	ccsbBroad304_01962	STK16	NAK family			
5698	-23.35	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
5699	-23.35	kd	CGS001-336	APOA2	Apolipoproteins			
5700	-23.35	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
5701	-23.37	kd	CGS001-4610	MYCL1	-			
5702	-23.39	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
5703	-23.43	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5704	-23.44	kd	CGS001-23387	SIK3	QIK subfamily			
5705	-23.45	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
5706	-23.46	cp	BRD-A68589262	troxipide	Glucosamine synthetase stimulant			Glucosamine synthetase stimulant
5707	-23.47	kd	CGS001-3586	IL10	Interleukins and interleukin receptors			
5708	-23.49	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
5709	-23.5	kd	CGS001-3925	STMN1	-			
5710	-23.51	oe	ccsbBroad304_07843	FCHO1	-			
5711	-23.52	oe	ccsbBroad304_02671	ECD	-			
5712	-23.54	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
5713	-23.58	oe	ccsbBroad304_07102	TSG101	-			
5714	-23.6	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
5715	-23.61	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
5716	-23.64	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
5717	-23.66	oe	ccsbBroad304_02438	FAM3C	-			
5718	-23.66	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
5719	-23.69	kd	CGS001-23244	PDS5A	-			
5720	-23.69	oe	ccsbBroad304_04053	DERL1	-			
5721	-23.71	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
5722	-23.72	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
5723	-23.77	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
5724	-23.78	kd	CGS001-5931	RBBP7	WD repeat domain containing			
5725	-23.83	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
5726	-23.83	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5727	-23.84	kd	CGS001-5329	PLAUR	CD molecules			
5728	-23.87	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
5729	-23.88	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
5730	-23.91	kd	CGS001-84328	LZIC	-			
5731	-23.94	oe	ccsbBroad304_06188	F10	Chymotrypsin			
5732	-23.94	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
5733	-23.97	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
5734	-23.99	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
5735	-24.02	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
5736	-24.04	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
5737	-24.11	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
5738	-24.14	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
5739	-24.14	kd	CGS001-8543	LMO4	-			
5740	-24.19	kd	CGS001-3127	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
5741	-24.21	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
5742	-24.23	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
5743	-24.24	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
5744	-24.25	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
5745	-24.25	oe	ccsbBroad304_03122	RHOD	-			
5746	-24.3	oe	ccsbBroad304_06462	ITGAE	Integrins			
5747	-24.31	cp	BRD-K09471561	levofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
5748	-24.33	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
5749	-24.33	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
5750	-24.36	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
5751	-24.37	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
5752	-24.37	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
5753	-24.37	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
5754	-24.41	cc		Protein synthesis inhibitor	-			
5755	-24.42	kd	CGS001-847	CAT	-			
5756	-24.44	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
5757	-24.44	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
5758	-24.46	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
5759	-24.54	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
5760	-24.56	kd	CGS001-5535	PPP3R2	EF-hand domain containing			
5761	-24.58	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
5762	-24.61	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
5763	-24.62	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
5764	-24.63	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
5765	-24.63	kd	CGS001-1398	CRK	SH2 domain containing			
5766	-24.68	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
5767	-24.68	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
5768	-24.69	kd	CGS001-8741	TNFSF13	CD molecules			
5769	-24.7	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
5770	-24.7	kd	CGS001-9697	TRAM2	-			
5771	-24.78	oe	ccsbBroad304_05192	SPRED2	-			
5772	-24.94	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
5773	-24.96	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
5774	-25	kd	CGS001-2153	F5	Blood coagulation components			
5775	-25.02	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
5776	-25.05	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
5777	-25.1	kd	CGS001-1112	FOXN3	Forkhead boxes			
5778	-25.2	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5779	-25.21	kd	CGS001-4708	NDUFB2	Mitochondrial respiratory chain complex / Complex I			
5780	-25.24	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
5781	-25.24	kd	CGS001-178	AGL	-			
5782	-25.31	oe	ccsbBroad304_02045	BUD31	-			
5783	-25.32	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
5784	-25.35	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
5785	-25.36	kd	CGS001-57048	PLSCR3	-			
5786	-25.37	kd	CGS001-1374	CPT1A	-			
5787	-25.38	kd	CGS001-7187	TRAF3	-			
5788	-25.4	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
5789	-25.41	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
5790	-25.42	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
5791	-25.49	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
5792	-25.5	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
5793	-25.52	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
5794	-25.58	kd	CGS001-405	ARNT	Basic helix-loop-helix proteins			
5795	-25.66	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
5796	-25.71	kd	CGS001-64425	POLR1E	RNA polymerase subunits			
5797	-25.73	kd	CGS001-5817	PVR	Immunoglobulin superfamily / C2-set domain containing			
5798	-25.75	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
5799	-25.76	oe	ccsbBroad304_06286	GLUL	-			
5800	-25.76	kd	CGS001-3030	HADHA	-			
5801	-25.78	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
5802	-25.81	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
5803	-25.82	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
5804	-25.82	oe	ccsbBroad304_06836	RAD23B	-			
5805	-25.83	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
5806	-25.89	kd	CGS001-55226	NAT10	-			
5807	-25.94	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
5808	-25.99	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
5809	-26.05	cc		Estrogen receptor agonist	-			
5810	-26.07	kd	CGS001-11116	FGFR1OP	-			
5811	-26.08	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
5812	-26.09	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
5813	-26.17	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
5814	-26.2	oe	ccsbBroad304_05038	HORMAD2	-			
5815	-26.2	kd	CGS001-54788	DNAJB12	Heat shock proteins / DNAJ (HSP40)			
5816	-26.21	kd	CGS001-9158	FIBP	-			
5817	-26.21	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
5818	-26.22	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
5819	-26.25	kd	CGS001-2119	ETV5	ETS Transcription Factors			
5820	-26.26	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
5821	-26.29	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
5822	-26.32	kd	CGS001-7016	TESK1	TESK subfamily			
5823	-26.37	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
5824	-26.38	oe	ccsbBroad304_00876	INSIG1	-			
5825	-26.4	kd	CGS001-317705	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
5826	-26.43	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
5827	-26.46	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
5828	-26.47	kd	CGS001-221188	GPR114	Adhesion Class GPCRs			
5829	-26.49	kd	CGS001-991	CDC20	WD repeat domain containing			
5830	-26.51	oe	ccsbBroad304_07561	YAF2	-			
5831	-26.52	oe	ccsbBroad304_00710	GUSB	-			
5832	-26.54	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
5833	-26.54	kd	CGS001-7982	ST7	-			
5834	-26.55	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
5835	-26.56	kd	CGS001-200734	SPRED2	-			
5836	-26.58	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
5837	-26.68	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
5838	-26.69	kd	CGS001-84539	MCHR2	GPCR / Class A : MCH receptors			
5839	-26.71	kd	CGS001-1195	CLK1	CDC-like kinases			
5840	-26.73	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
5841	-26.86	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
5842	-26.96	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
5843	-26.97	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
5844	-26.99	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
5845	-26.99	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
5846	-27.01	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
5847	-27.01	kd	CGS001-4048	LTA4H	Hydrolases			
5848	-27.07	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
5849	-27.08	kd	CGS001-55810	FOXJ2	Forkhead boxes			
5850	-27.09	oe	ccsbBroad304_13598	NRBP2	NRBP family			
5851	-27.1	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
5852	-27.14	oe	ccsbBroad304_07287	HYAL2	-			
5853	-27.19	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
5854	-27.26	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
5855	-27.29	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
5856	-27.31	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
5857	-27.31	kd	CGS001-2348	FOLR1	-			
5858	-27.32	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
5859	-27.32	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
5860	-27.33	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
5861	-27.33	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
5862	-27.38	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
5863	-27.4	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5864	-27.42	oe	ccsbBroad304_00262	CD59	CD molecules			
5865	-27.44	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
5866	-27.46	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
5867	-27.47	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
5868	-27.49	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
5869	-27.53	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
5870	-27.53	oe	ccsbBroad304_12106	PXK	Slob family			
5871	-27.53	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
5872	-27.55	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
5873	-27.57	oe	ccsbBroad304_00033	ADSS	-			
5874	-27.61	kd	CGS001-7018	TF	-			
5875	-27.62	oe	ccsbBroad304_00099	ARG2	Arginase			
5876	-27.63	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
5877	-27.63	kd	CGS001-8669	EIF3J	-			
5878	-27.64	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
5879	-27.64	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
5880	-27.67	cp	BRD-K15842202	eudesmic-acid	-666			-666
5881	-27.69	kd	CGS001-93487	MAPK1IP1L	-			
5882	-27.71	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
5883	-27.72	oe	ccsbBroad304_03037	TMEM97	-			
5884	-27.73	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
5885	-27.74	kd	CGS001-284	ANGPT1	Fibrinogen C domain containing			
5886	-27.76	kd	CGS001-5881	RAC3	Endogenous ligands			
5887	-27.83	kd	CGS001-7485	WRB	-			
5888	-27.83	kd	CGS001-498	ATP5A1	ATPases / F-type			
5889	-27.87	kd	CGS001-5328	PLAU	Chymotrypsin			
5890	-27.88	cc		ATPase inhibitor	-			
5891	-27.9	oe	ccsbBroad304_01114	NUP88	-			
5892	-27.93	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
5893	-27.93	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
5894	-27.96	kd	CGS001-2735	GLI1	Zinc fingers, C2H2-type			
5895	-27.98	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
5896	-28.09	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
5897	-28.1	kd	CGS001-10497	UNC13B	-			
5898	-28.11	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
5899	-28.11	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
5900	-28.16	kd	CGS001-54811	ZNF562	Zinc fingers, C2H2-type			
5901	-28.18	oe	ccsbBroad304_02047	AP1S2	-			
5902	-28.2	kd	CGS001-2073	ERCC5	-			
5903	-28.21	oe	ccsbBroad304_08993	DHDDS	-			
5904	-28.24	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
5905	-28.28	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
5906	-28.28	kd	CGS001-1736	DKC1	-			
5907	-28.29	oe	ccsbBroad304_04655	TRIM9	-			
5908	-28.3	oe	ccsbBroad304_08481	CEP55	-			
5909	-28.34	kd	CGS001-51135	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
5910	-28.38	oe	ccsbBroad304_08137	HOOK2	-			
5911	-28.38	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
5912	-28.38	kd	CGS001-4946	OAZ1	-			
5913	-28.4	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
5914	-28.43	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
5915	-28.45	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
5916	-28.46	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
5917	-28.47	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
5918	-28.53	oe	ccsbBroad304_05902	BNIP3	-			
5919	-28.56	oe	ccsbBroad304_08536	PARL	-			
5920	-28.58	kd	CGS001-345	APOC3	Apolipoproteins			
5921	-28.61	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
5922	-28.63	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
5923	-28.63	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
5924	-28.64	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
5925	-28.65	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
5926	-28.68	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
5927	-28.7	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
5928	-28.71	kd	CGS001-965	CD58	CD molecules			
5929	-28.73	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
5930	-28.77	kd	CGS001-9374	PPT2	-			
5931	-28.77	kd	CGS001-10094	ARPC3	Actin related protein 2/3 complex subunits			
5932	-28.77	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
5933	-28.79	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
5934	-28.8	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
5935	-28.83	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
5936	-29	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
5937	-29	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
5938	-29.06	kd	CGS001-5036	PA2G4	-			
5939	-29.09	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
5940	-29.1	kd	CGS001-5362	PLXNA2	Plexins			
5941	-29.1	kd	CGS001-1069	CETN2	EF-hand domain containing			
5942	-29.14	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
5943	-29.16	kd	CGS001-23534	TNPO3	Importins			
5944	-29.2	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
5945	-29.21	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
5946	-29.26	kd	CGS001-7079	TIMP4	-			
5947	-29.27	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
5948	-29.28	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
5949	-29.3	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
5950	-29.3	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
5951	-29.3	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
5952	-29.33	kd	CGS001-55526	DHTKD1	-			
5953	-29.34	oe	ccsbBroad304_07515	GFPT2	-			
5954	-29.38	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
5955	-29.38	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
5956	-29.39	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
5957	-29.49	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
5958	-29.51	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
5959	-29.51	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
5960	-29.52	cc		Trace amine receptors LOF	-			
5961	-29.58	kd	CGS001-51079	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
5962	-29.6	kd	CGS001-5423	POLB	DNA polymerases			
5963	-29.6	kd	CGS001-5106	PCK2	-			
5964	-29.62	kd	CGS001-6098	ROS1	Type XVII RTKs: ROS receptors			
5965	-29.67	kd	CGS001-6696	SPP1	Endogenous ligands			
5966	-29.69	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
5967	-29.7	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
5968	-29.77	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
5969	-29.8	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
5970	-29.85	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
5971	-29.91	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
5972	-29.92	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
5973	-29.93	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
5974	-29.94	kd	CGS001-135	ADORA2A	GPCR / Class A : Adenosine receptors			
5975	-29.98	oe	ccsbBroad304_06386	HNMT	-			
5976	-29.98	oe	ccsbBroad304_03433	DDIT4	-			
5977	-30.03	kd	CGS001-1029	CDKN2A	-			
5978	-30.04	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
5979	-30.04	kd	CGS001-55324	ABCF3	ATP binding cassette transporters / subfamily F			
5980	-30.08	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
5981	-30.1	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
5982	-30.19	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
5983	-30.21	kd	CGS001-91304	C19ORF6	-			
5984	-30.24	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
5985	-30.27	kd	CGS001-3482	IGF2R	CD molecules			
5986	-30.28	oe	ccsbBroad304_03269	CD320	CD molecules			
5987	-30.29	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
5988	-30.31	cc		Heat shock 70kDa proteins LOF	-			
5989	-30.34	oe	ccsbBroad304_06651	NOV	-			
5990	-30.34	kd	CGS001-9945	GFPT2	-			
5991	-30.36	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
5992	-30.36	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
5993	-30.38	oe	ccsbBroad304_00492	EIF5A	-			
5994	-30.39	oe	ccsbBroad304_07220	CDC45	-			
5995	-30.41	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
5996	-30.45	kd	CGS001-147837	ZNF563	Zinc fingers, C2H2-type			
5997	-30.53	kd	CGS001-6513	SLC2A1	Solute carriers			
5998	-30.53	kd	CGS001-55937	APOM	Apolipoproteins			
5999	-30.57	kd	CGS001-4179	CD46	CD molecules			
6000	-30.58	cc		Akt Signaling GOF	-			
6001	-30.59	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
6002	-30.6	kd	CGS001-1962	EHHADH	-			
6003	-30.61	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
6004	-30.62	kd	CGS001-169841	ZNF169	Zinc fingers, C2H2-type			
6005	-30.63	kd	CGS001-26298	EHF	-			
6006	-30.66	kd	CGS001-64147	KIF9	Kinesins			
6007	-30.68	oe	ccsbBroad304_01131	OXCT1	-			
6008	-30.68	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
6009	-30.73	oe	ccsbBroad304_03746	CDC42SE1	-			
6010	-30.75	kd	CGS001-2950	GSTP1	Glutathione S-transferases			
6011	-30.76	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
6012	-30.79	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
6013	-30.81	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
6014	-30.83	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
6015	-30.85	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
6016	-30.87	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
6017	-30.95	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
6018	-30.98	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
6019	-31.04	kd	CGS001-5707	PSMD1	Proteasome subunits			
6020	-31.04	kd	CGS001-5613	PRKX	Protein kinase A			
6021	-31.04	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
6022	-31.06	oe	ccsbBroad304_01930	CUL2	-			
6023	-31.09	kd	CGS001-1070	CETN3	EF-hand domain containing			
6024	-31.11	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
6025	-31.11	kd	CGS001-6908	TBP	General transcription factors			
6026	-31.18	kd	CGS001-10525	HYOU1	Heat shock proteins / HSP70			
6027	-31.19	kd	CGS001-3094	HINT1	-			
6028	-31.26	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
6029	-31.27	cc		Thymidylate synthase inhibitor	-			
6030	-31.28	kd	CGS001-4193	MDM2	-			
6031	-31.28	oe	ccsbBroad304_01163	PDHA1	-			
6032	-31.32	kd	CGS001-4174	MCM5	-			
6033	-31.4	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
6034	-31.42	kd	CGS001-55423	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
6035	-31.46	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
6036	-31.46	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
6037	-31.51	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
6038	-31.53	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
6039	-31.56	kd	CGS001-9146	HGS	Zinc fingers, FYVE domain containing			
6040	-31.65	kd	CGS001-342926	ZNF677	Zinc fingers, C2H2-type			
6041	-31.67	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
6042	-31.73	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
6043	-31.76	kd	CGS001-26191	PTPN22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6044	-31.77	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
6045	-31.78	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
6046	-31.86	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
6047	-31.92	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
6048	-31.96	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
6049	-31.96	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6050	-31.98	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
6051	-32.01	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6052	-32.03	kd	CGS001-160	AP2A1	-			
6053	-32.05	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
6054	-32.09	kd	CGS001-53343	NUDT9	Nudix motif containing			
6055	-32.15	cp	BRD-K46742498	alosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
6056	-32.15	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
6057	-32.15	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
6058	-32.2	cp	BRD-A16934955	nalbuphine	Opioid receptor agonist		OPRD1, OPRK1, OPRM1	Opioid receptor agonist, Opioid receptor antagonist
6059	-32.23	oe	ccsbBroad304_07053	TFPI	-			
6060	-32.26	kd	CGS001-55723	ASF1B	-			
6061	-32.27	kd	CGS001-823	CAPN1	EF-hand domain containing			
6062	-32.28	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
6063	-32.29	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
6064	-32.3	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
6065	-32.35	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
6066	-32.35	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
6067	-32.35	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
6068	-32.37	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
6069	-32.39	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
6070	-32.39	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
6071	-32.41	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
6072	-32.44	kd	CGS001-4069	LYZ	-			
6073	-32.52	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
6074	-32.52	kd	CGS001-8446	DUSP11	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6075	-32.58	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
6076	-32.6	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
6077	-32.61	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
6078	-32.66	kd	CGS001-140465	MYL6B	EF-hand domain containing			
6079	-32.68	cc		Serotonin receptor agonist	-			
6080	-32.7	kd	CGS001-8449	DHX16	DEAH-boxes			
6081	-32.71	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
6082	-32.72	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
6083	-32.73	kd	CGS001-3593	IL12B	Interleukins and interleukin receptors			
6084	-32.78	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
6085	-32.79	oe	ccsbBroad304_05749	A2M	-			
6086	-32.79	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
6087	-32.81	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
6088	-32.82	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
6089	-32.84	kd	CGS001-55312	RFK	-			
6090	-32.86	kd	CGS001-5320	PLA2G2A	Hydrolases			
6091	-32.86	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
6092	-32.89	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
6093	-32.9	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
6094	-32.94	kd	CGS001-10250	SRRM1	-			
6095	-32.99	oe	ccsbBroad304_02565	RALBP1	-			
6096	-33	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6097	-33.03	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
6098	-33.08	cc		Adenosine receptor agonist	-			
6099	-33.1	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
6100	-33.1	kd	CGS001-7167	TPI1	-			
6101	-33.1	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
6102	-33.17	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
6103	-33.17	kd	CGS001-286380	FOXD4L3	-			
6104	-33.17	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
6105	-33.19	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
6106	-33.22	kd	CGS001-22921	MSRB2	-			
6107	-33.24	kd	CGS001-2550	GABBR1	GABA receptors			
6108	-33.25	kd	CGS001-57147	SCYL3	-			
6109	-33.26	kd	CGS001-259	AMBP	Lipocalins			
6110	-33.28	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
6111	-33.3	oe	ccsbBroad304_03479	YTHDF1	-			
6112	-33.33	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
6113	-33.34	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
6114	-33.34	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
6115	-33.36	kd	CGS001-26036	ZNF451	Zinc fingers, C2H2-type			
6116	-33.4	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
6117	-33.41	kd	CGS001-55328	RNLS	-			
6118	-33.44	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
6119	-33.45	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
6120	-33.54	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
6121	-33.56	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
6122	-33.57	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
6123	-33.59	kd	CGS001-2976	GTF3C2	General transcription factors			
6124	-33.6	oe	ccsbBroad304_01038	MSRA	-			
6125	-33.66	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
6126	-33.67	oe	ccsbBroad304_08325	LIPT1	-			
6127	-33.7	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
6128	-33.74	kd	CGS001-54407	SLC38A2	System A-like transporters			
6129	-33.77	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
6130	-33.78	oe	ccsbBroad304_00874	INS	-			
6131	-33.84	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
6132	-33.87	kd	CGS001-624	BDKRB2	Bradykinin receptors			
6133	-33.92	cc		Minor histocompatibility antigens LOF	-			
6134	-33.93	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
6135	-33.94	kd	CGS001-7357	UGCG	Glycosyltransferase family 2 domain containing			
6136	-33.97	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
6137	-34.05	kd	CGS001-5066	PAM	-			
6138	-34.12	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
6139	-34.13	kd	CGS001-2237	FEN1	-			
6140	-34.15	kd	CGS001-9787	DLGAP5	-			
6141	-34.17	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
6142	-34.2	kd	CGS001-116931	MED12L	-			
6143	-34.21	kd	CGS001-26993	AKAP8L	-			
6144	-34.22	kd	CGS001-23028	KDM1A	Histone demethylase			
6145	-34.34	kd	CGS001-79174	CRELD2	-			
6146	-34.36	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
6147	-34.37	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
6148	-34.39	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
6149	-34.41	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
6150	-34.41	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
6151	-34.42	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
6152	-34.44	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
6153	-34.47	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6154	-34.47	cp	BRD-K32398298	alprazolam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, CYP3A5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
6155	-34.5	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6156	-34.53	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
6157	-34.55	oe	ccsbBroad304_01469	RSU1	-			
6158	-34.57	kd	CGS001-6936	C2ORF3	-			
6159	-34.58	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
6160	-34.6	kd	CGS001-1431	CS	-			
6161	-34.66	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
6162	-34.66	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
6163	-34.66	kd	CGS001-63874	ABHD4	Abhydrolase domain containing			
6164	-34.67	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
6165	-34.69	kd	CGS001-1936	EEF1D	-			
6166	-34.71	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
6167	-34.76	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
6168	-34.78	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6169	-34.82	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
6170	-34.85	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
6171	-34.86	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6172	-34.86	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
6173	-34.93	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
6174	-35.01	kd	CGS001-9447	AIM2	-			
6175	-35.06	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
6176	-35.1	kd	CGS001-699	BUB1	Bub family			
6177	-35.19	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
6178	-35.24	kd	CGS001-3313	HSPA9	Heat shock proteins / HSP70			
6179	-35.25	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
6180	-35.32	oe	ccsbBroad304_00070	ANXA5	Annexins			
6181	-35.36	kd	CGS001-819	CAMLG	-			
6182	-35.42	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
6183	-35.43	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
6184	-35.46	kd	CGS001-966	CD59	CD molecules			
6185	-35.46	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
6186	-35.52	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
6187	-35.53	kd	CGS001-650	BMP2	Bone morphogenetic proteins			
6188	-35.56	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6189	-35.58	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
6190	-35.66	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
6191	-35.69	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
6192	-35.72	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
6193	-35.73	kd	CGS001-10237	SLC35B1	SLC35 family of nucleotide sugar transporters			
6194	-35.76	kd	CGS001-7965	AIMP2	-			
6195	-35.77	kd	CGS001-23062	GGA2	-			
6196	-35.82	kd	CGS001-6603	SMARCD2	-			
6197	-35.84	kd	CGS001-79145	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
6198	-35.89	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
6199	-35.95	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
6200	-35.95	kd	CGS001-390980	ZNF805	Zinc fingers, C2H2-type			
6201	-35.98	kd	CGS001-9124	PDLIM1	-			
6202	-36.02	kd	CGS001-10775	POP4	-			
6203	-36.06	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
6204	-36.1	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
6205	-36.11	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
6206	-36.11	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
6207	-36.15	cc		NADH ubiquinone oxidoreductase supernumerary subunits LOF	-			
6208	-36.15	oe	ccsbBroad304_01234	POLB	DNA polymerases			
6209	-36.22	oe	ccsbBroad304_00106	ARRB1	-			
6210	-36.25	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
6211	-36.25	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
6212	-36.27	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
6213	-36.27	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
6214	-36.28	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
6215	-36.29	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
6216	-36.32	oe	ccsbBroad304_04786	CANT1	-			
6217	-36.33	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6218	-36.4	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
6219	-36.46	kd	CGS001-224	ALDH3A2	Aldehyde dehydrogenases			
6220	-36.46	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
6221	-36.49	oe	ccsbBroad304_06290	GNA15	-			
6222	-36.49	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
6223	-36.51	kd	CGS001-3880	KRT19	Intermediate filaments type I, keratins (acidic)			
6224	-36.51	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
6225	-36.52	oe	ccsbBroad304_06777	PRNP	CD molecules			
6226	-36.56	kd	CGS001-22933	SIRT2	Histone deacetylases			
6227	-36.62	cp	BRD-K27184429	levocetirizine	Histamine receptor antagonist		HRH1, CXCL8	Histamine receptor antagonist
6228	-36.66	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
6229	-36.74	oe	ccsbBroad304_02788	PRAME	-			
6230	-36.76	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
6231	-36.8	kd	CGS001-2562	GABRB3	GABA receptors			
6232	-36.8	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
6233	-36.82	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
6234	-36.83	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
6235	-36.84	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
6236	-36.85	kd	CGS001-5653	KLK6	Chymotrypsin			
6237	-36.87	kd	CGS001-6772	STAT1	SH2 domain containing			
6238	-36.89	kd	CGS001-301	ANXA1	Annexins			
6239	-36.89	kd	CGS001-25913	POT1	-			
6240	-36.91	oe	ccsbBroad304_02285	MED6	-			
6241	-36.92	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6242	-36.95	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
6243	-37.09	cc		GABA receptor antagonist	-			
6244	-37.1	oe	ccsbBroad304_03732	NPDC1	-			
6245	-37.13	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
6246	-37.15	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
6247	-37.16	kd	CGS001-51601	LIPT1	-			
6248	-37.19	kd	CGS001-11230	PRAF2	-			
6249	-37.21	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
6250	-37.22	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
6251	-37.33	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
6252	-37.34	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
6253	-37.35	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
6254	-37.38	kd	CGS001-6810	STX4	-			
6255	-37.38	oe	ccsbBroad304_05439	O3FAR1	-			
6256	-37.44	kd	CGS001-64077	LHPP	-			
6257	-37.46	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
6258	-37.47	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
6259	-37.48	kd	CGS001-23408	SIRT5	Histone deacetylases			
6260	-37.48	kd	CGS001-3098	HK1	-			
6261	-37.5	kd	CGS001-4292	MLH1	-			
6262	-37.51	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
6263	-37.54	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
6264	-37.55	oe	ccsbBroad304_07632	PROCR	CD molecules			
6265	-37.57	oe	ccsbBroad304_02964	TIMM9	-			
6266	-37.63	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
6267	-37.63	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6268	-37.65	cp	BRD-K06388322	pramipexole	Dopamine receptor agonist		DRD3, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
6269	-37.66	kd	CGS001-85315	PAQR8	-			
6270	-37.66	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6271	-37.66	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
6272	-37.69	kd	CGS001-10553	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
6273	-37.7	oe	ccsbBroad304_00993	MDM4	-			
6274	-37.77	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
6275	-37.8	cp	BRD-K63784565	BRD-K63784565	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
6276	-37.85	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
6277	-37.87	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
6278	-37.88	kd	CGS001-27244	SESN1	-			
6279	-37.88	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
6280	-37.92	kd	CGS001-1212	CLTB	-			
6281	-37.94	oe	ccsbBroad304_06294	GNAZ	-			
6282	-37.95	oe	ccsbBroad304_07045	TEAD4	-			
6283	-37.99	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6284	-38.01	kd	CGS001-813	CALU	EF-hand domain containing			
6285	-38.04	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
6286	-38.16	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
6287	-38.16	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
6288	-38.18	kd	CGS001-406	ARNTL	Basic helix-loop-helix proteins			
6289	-38.2	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6290	-38.22	kd	CGS001-7468	WHSC1	Zinc fingers, PHD-type			
6291	-38.26	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
6292	-38.26	kd	CGS001-57616	TSHZ3	Teashirt zinc fingers			
6293	-38.26	kd	CGS001-10018	BCL2L11	-			
6294	-38.27	kd	CGS001-6195	RPS6KA1	RSK subfamily			
6295	-38.31	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
6296	-38.33	oe	ccsbBroad304_01748	UFD1L	-			
6297	-38.33	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
6298	-38.34	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
6299	-38.35	kd	CGS001-11140	CDC37	-			
6300	-38.44	kd	CGS001-3692	EIF6	-			
6301	-38.46	kd	CGS001-5058	PAK1	PAKA subfamily			
6302	-38.47	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
6303	-38.48	oe	ccsbBroad304_02278	THRAP3	-			
6304	-38.48	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
6305	-38.5	kd	CGS001-5915	RARB	Retinoic acid receptors			
6306	-38.51	kd	CGS001-7535	ZAP70	Syk family			
6307	-38.52	kd	CGS001-91392	ZNF502	Zinc fingers, C2H2-type			
6308	-38.53	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
6309	-38.53	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6310	-38.58	oe	ccsbBroad304_00961	SMAD2	SMADs			
6311	-38.59	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
6312	-38.59	kd	CGS001-5293	PIK3CD	Phosphatidylinositol kinases			
6313	-38.65	kd	CGS001-11267	SNF8	-			
6314	-38.68	kd	CGS001-4724	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
6315	-38.72	kd	CGS001-7025	NR2F1	COUP-TF-like receptors			
6316	-38.94	kd	CGS001-2021	ENDOG	-			
6317	-38.98	oe	ccsbBroad304_07018	SUPT5H	-			
6318	-39.01	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
6319	-39.02	cp	BRD-K21806131	tegaserod	Serotonin receptor partial agonist		HTR4, HTR2B, HTR2A, HTR2C	Serotonin receptor partial agonist
6320	-39.02	cp	BRD-M47937986	cefatrizine	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6321	-39.1	cc		Apolipoproteins LOF	-			
6322	-39.14	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
6323	-39.16	oe	ccsbBroad304_01675	TK1	-			
6324	-39.18	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6325	-39.22	kd	CGS001-5928	RBBP4	WD repeat domain containing			
6326	-39.24	cp	BRD-K81916719	triclabendazole	Microtubule inhibitor		DNMT1	Microtubule inhibitor
6327	-39.24	oe	ccsbBroad304_06996	SRM	-			
6328	-39.25	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
6329	-39.28	kd	CGS001-1362	CPD	Carboxypeptidase A			
6330	-39.29	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
6331	-39.42	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
6332	-39.45	oe	ccsbBroad304_08055	ATP5S	-			
6333	-39.45	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
6334	-39.47	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
6335	-39.49	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
6336	-39.52	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6337	-39.52	kd	CGS001-3035	HARS	Aminoacyl tRNA synthetases / Class II			
6338	-39.55	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
6339	-39.57	cc		Proteasome inhibitor	-			
6340	-39.57	kd	CGS001-23030	KDM4B	Histone demethylases			
6341	-39.61	oe	ccsbBroad304_06670	OGG1	-			
6342	-39.63	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
6343	-39.64	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
6344	-39.64	oe	ccsbBroad304_06654	NPM1	-			
6345	-39.65	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
6346	-39.69	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
6347	-39.7	kd	CGS001-253430	IPMK	-			
6348	-39.72	kd	CGS001-4707	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
6349	-39.76	oe	ccsbBroad304_08694	TBX20	T-boxes			
6350	-39.77	kd	CGS001-10318	TNIP1	-			
6351	-39.8	kd	CGS001-9170	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6352	-39.84	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
6353	-39.89	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
6354	-39.92	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
6355	-39.93	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
6356	-39.98	oe	ccsbBroad304_00645	GCLM	-			
6357	-40	kd	CGS001-55012	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
6358	-40.01	kd	CGS001-1440	CSF3	Endogenous ligands			
6359	-40.07	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
6360	-40.09	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
6361	-40.12	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
6362	-40.16	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
6363	-40.18	oe	ccsbBroad304_03772	CCNL1	-			
6364	-40.18	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
6365	-40.18	kd	CGS001-3590	IL11RA	IL-6 receptor family			
6366	-40.2	oe	ccsbBroad304_04170	PANK2	-			
6367	-40.22	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
6368	-40.25	kd	CGS001-5479	PPIB	-			
6369	-40.34	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
6370	-40.37	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
6371	-40.37	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6372	-40.38	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
6373	-40.41	kd	CGS001-344	APOC2	Apolipoproteins			
6374	-40.49	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
6375	-40.52	kd	CGS001-4763	NF1	-			
6376	-40.52	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6377	-40.53	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
6378	-40.55	kd	CGS001-23753	SDF2L1	-			
6379	-40.6	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
6380	-40.6	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
6381	-40.62	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
6382	-40.65	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
6383	-40.67	kd	CGS001-2744	GLS	Ankyrin repeat domain containing			
6384	-40.67	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
6385	-40.67	oe	ccsbBroad304_03040	NKIRAS2	-			
6386	-40.69	kd	CGS001-1163	CKS1B	-			
6387	-40.69	oe	ccsbBroad304_02566	MORF4L1	-			
6388	-40.72	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
6389	-40.72	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
6390	-40.74	kd	CGS001-283150	FOXR1	Forkhead boxes			
6391	-40.81	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
6392	-40.84	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
6393	-40.91	kd	CGS001-1513	CTSK	Cathepsins			
6394	-40.93	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
6395	-40.96	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
6396	-41.01	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
6397	-41.05	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
6398	-41.07	cp	BRD-K11630072	carmofur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
6399	-41.12	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
6400	-41.12	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
6401	-41.13	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
6402	-41.22	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
6403	-41.26	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6404	-41.26	kd	CGS001-9276	COPB2	WD repeat domain containing			
6405	-41.32	kd	CGS001-216	ALDH1A1	Aldehyde dehydrogenases			
6406	-41.33	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
6407	-41.35	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
6408	-41.41	kd	CGS001-152	ADRA2C	GPCR / Class A : Adrenoceptors : alpha			
6409	-41.43	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
6410	-41.45	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
6411	-41.5	kd	CGS001-476	ATP1A1	ATPases / P-type			
6412	-41.52	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
6413	-41.53	kd	CGS001-55486	PARL	-			
6414	-41.55	kd	CGS001-79712	GTDC1	Glycosyltransferase group 1 domain containing			
6415	-41.56	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
6416	-41.56	kd	CGS001-3029	HAGH	-			
6417	-41.62	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
6418	-41.65	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
6419	-41.66	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
6420	-41.69	kd	CGS001-8829	NRP1	CD molecules			
6421	-41.78	kd	CGS001-5927	KDM5A	Histone demethylases			
6422	-41.81	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
6423	-41.84	oe	ccsbBroad304_03497	TXNL4B	-			
6424	-41.84	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
6425	-41.84	kd	CGS001-4907	NT5E	Adenosine turnover			
6426	-41.86	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
6427	-41.9	kd	CGS001-8805	TRIM24	TIF1 family			
6428	-41.93	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
6429	-41.95	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
6430	-41.96	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
6431	-42.03	kd	CGS001-790	CAD	-			
6432	-42.04	kd	CGS001-901	CCNG2	-			
6433	-42.07	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
6434	-42.17	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6435	-42.21	kd	CGS001-3958	LGALS3	Endogenous ligands			
6436	-42.21	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
6437	-42.22	cc		Aromatase inhibitor	-			
6438	-42.26	kd	CGS001-474354	LRRC18	-			
6439	-42.29	kd	CGS001-5294	PIK3CG	Phosphatidylinositol kinases			
6440	-42.37	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
6441	-42.46	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
6442	-42.5	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
6443	-42.5	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
6444	-42.5	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
6445	-42.51	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
6446	-42.51	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
6447	-42.51	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
6448	-42.52	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
6449	-42.52	kd	CGS001-23252	OTUD3	OTU domain containing			
6450	-42.55	cp	BRD-A80928489	1-monopalmitin	P-glycoprotein inhibitor		ABCB1	P-glycoprotein inhibitor
6451	-42.64	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
6452	-42.71	oe	ccsbBroad304_00003	ABAT	GABA turnover			
6453	-42.73	oe	ccsbBroad304_07320	SQSTM1	-			
6454	-42.74	kd	CGS001-9670	IPO13	Importins			
6455	-42.75	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
6456	-42.88	oe	ccsbBroad304_02458	STK25	YSK subfamily			
6457	-42.9	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
6458	-42.92	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
6459	-42.95	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
6460	-43	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
6461	-43	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
6462	-43.05	cp	BRD-K60690191	MPEP	Glutamate receptor antagonist		GRM5, GRM1, GRM4	Glutamate receptor antagonist
6463	-43.08	kd	CGS001-6233	RPS27A	S ribosomal proteins			
6464	-43.1	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
6465	-43.11	kd	CGS001-7428	VHL	-			
6466	-43.15	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
6467	-43.21	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
6468	-43.22	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
6469	-43.22	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
6470	-43.23	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
6471	-43.28	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
6472	-43.29	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
6473	-43.33	kd	CGS001-2956	MSH6	-			
6474	-43.35	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
6475	-43.35	kd	CGS001-1131	CHRM3	Cholinergic receptors			
6476	-43.36	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
6477	-43.36	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
6478	-43.45	oe	ccsbBroad304_05947	CCNC	-			
6479	-43.52	oe	ccsbBroad304_00316	CKS1B	-			
6480	-43.56	oe	ccsbBroad304_02219	MORF4L2	-			
6481	-43.56	cp	BRD-K23369905	oxiconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6482	-43.57	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
6483	-43.59	kd	CGS001-29116	MYLIP	-			
6484	-43.62	kd	CGS001-10131	TRAP1	Heat shock proteins / HSPC			
6485	-43.62	kd	CGS001-8945	BTRC	F-boxes / WD-40 domains			
6486	-43.64	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
6487	-43.65	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
6488	-43.65	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
6489	-43.67	cp	BRD-K85925969	zalcitabine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
6490	-43.69	kd	CGS001-9926	LPGAT1	-			
6491	-43.7	kd	CGS001-79722	ANKRD55	Ankyrin repeat domain containing			
6492	-43.94	kd	CGS001-55718	POLR3E	RNA polymerase subunits			
6493	-43.95	kd	CGS001-90861	HN1L	-			
6494	-43.95	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
6495	-43.97	kd	CGS001-10725	NFAT5	Nuclear factor of activated T-cells			
6496	-43.97	kd	CGS001-23401	FRAT2	-			
6497	-44.01	oe	ccsbBroad304_01146	PARN	-			
6498	-44.06	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
6499	-44.07	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
6500	-44.11	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
6501	-44.16	kd	CGS001-899	CCNF	F-boxes / other			
6502	-44.18	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
6503	-44.18	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
6504	-44.22	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
6505	-44.22	kd	CGS001-23361	ZNF629	Zinc fingers, C2H2-type			
6506	-44.23	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
6507	-44.31	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
6508	-44.31	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
6509	-44.32	oe	ccsbBroad304_05757	ACADS	-			
6510	-44.36	oe	ccsbBroad304_01624	SUPV3L1	-			
6511	-44.39	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
6512	-44.41	kd	CGS001-8409	UXT	-			
6513	-44.46	kd	CGS001-6198	RPS6KB1	p70 subfamily			
6514	-44.47	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
6515	-44.49	oe	ccsbBroad304_07922	TRIM29	-			
6516	-44.49	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
6517	-44.51	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
6518	-44.65	kd	CGS001-2010	EMD	-			
6519	-44.69	oe	ccsbBroad304_07071	TKT	-			
6520	-44.69	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
6521	-44.7	oe	ccsbBroad304_00231	CBFB	-			
6522	-44.73	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
6523	-44.75	kd	CGS001-5829	PXN	-			
6524	-44.76	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
6525	-44.78	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
6526	-44.79	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
6527	-44.83	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
6528	-44.89	oe	ccsbBroad304_02869	ASF1A	-			
6529	-44.93	kd	CGS001-2778	GNAS	-			
6530	-44.93	kd	CGS001-1622	DBI	-			
6531	-44.99	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
6532	-45	oe	ccsbBroad304_00146	BAD	-			
6533	-45.08	kd	CGS001-51465	UBE2J1	Ubiquitin-conjugating enzymes E2			
6534	-45.1	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
6535	-45.12	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
6536	-45.13	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
6537	-45.17	kd	CGS001-10671	DCTN6	-			
6538	-45.19	oe	ccsbBroad304_00446	DKC1	-			
6539	-45.2	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
6540	-45.21	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
6541	-45.24	kd	CGS001-1999	ELF3	ETS Transcription Factors			
6542	-45.33	kd	CGS001-6500	SKP1	-			
6543	-45.37	kd	CGS001-4091	SMAD6	SMADs			
6544	-45.38	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
6545	-45.4	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
6546	-45.44	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
6547	-45.45	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
6548	-45.46	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
6549	-45.48	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
6550	-45.51	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
6551	-45.51	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
6552	-45.52	kd	CGS001-1120	CHKB	-			
6553	-45.58	kd	CGS001-3927	LASP1	-			
6554	-45.63	oe	ccsbBroad304_03910	CCDC90A	-			
6555	-45.71	kd	CGS001-5366	PMAIP1	-			
6556	-45.72	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
6557	-45.73	kd	CGS001-50	ACO2	-			
6558	-45.75	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
6559	-45.78	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
6560	-45.79	kd	CGS001-4841	NONO	RNA binding motif (RRM) containing			
6561	-45.79	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6562	-45.82	kd	CGS001-57819	LSM2	-			
6563	-45.88	cc		Vesicular Transport LOF	-			
6564	-45.88	kd	CGS001-8803	SUCLA2	-			
6565	-45.88	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
6566	-45.89	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
6567	-45.89	kd	CGS001-5087	PBX1	Homeoboxes / TALE class			
6568	-45.89	kd	CGS001-84365	MKI67IP	-			
6569	-45.94	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
6570	-45.98	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
6571	-46.02	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
6572	-46.17	kd	CGS001-5796	PTPRK	Receptor tyrosine phosphatases (RTP)			
6573	-46.17	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
6574	-46.18	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
6575	-46.23	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
6576	-46.24	kd	CGS001-35	ACADS	-			
6577	-46.26	kd	CGS001-1903	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
6578	-46.28	kd	CGS001-81533	ITFG1	-			
6579	-46.28	oe	ccsbBroad304_00549	FDX1	-			
6580	-46.38	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
6581	-46.42	kd	CGS001-56675	NRIP3	-			
6582	-46.42	kd	CGS001-2353	FOS	basic leucine zipper proteins			
6583	-46.43	oe	ccsbBroad304_02109	XPR1	-			
6584	-46.47	kd	CGS001-4208	MEF2C	Myocyte enhancer factors			
6585	-46.49	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
6586	-46.51	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
6587	-46.56	kd	CGS001-6519	SLC3A1	SLC3 family			
6588	-46.61	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
6589	-46.61	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
6590	-46.62	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
6591	-46.69	kd	CGS001-5916	RARG	Retinoic acid receptors			
6592	-46.69	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
6593	-46.7	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
6594	-46.71	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
6595	-46.77	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
6596	-46.83	kd	CGS001-475	ATOX1	-			
6597	-46.85	kd	CGS001-2776	GNAQ	-			
6598	-46.88	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
6599	-46.93	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
6600	-46.98	kd	CGS001-54536	EXOC6	-			
6601	-47.01	cc		Serpin peptidase inhibitors LOF	-			
6602	-47.01	kd	CGS001-11243	PMF1	-			
6603	-47.04	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
6604	-47.09	kd	CGS001-221391	OPN5	GPCR / Class A : Opsin receptors			
6605	-47.1	kd	CGS001-9	NAT1	-			
6606	-47.11	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
6607	-47.11	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6608	-47.14	kd	CGS001-230	ALDOC	-			
6609	-47.18	cp	BRD-A00520476	otenzepad	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6610	-47.21	kd	CGS001-83729	INHBE	-			
6611	-47.23	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
6612	-47.27	kd	CGS001-11137	PWP1	WD repeat domain containing			
6613	-47.28	oe	ccsbBroad304_00098	ARG1	Arginase			
6614	-47.33	kd	CGS001-95	ACY1	-			
6615	-47.37	kd	CGS001-6929	TCF3	Basic helix-loop-helix proteins			
6616	-47.46	kd	CGS001-9261	MAPKAPK2	MAPKAPK subfamily			
6617	-47.48	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
6618	-47.49	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
6619	-47.51	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
6620	-47.55	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
6621	-47.58	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
6622	-47.7	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
6623	-47.74	kd	CGS001-27102	EIF2AK1	Other PEK family kinases			
6624	-47.77	oe	ccsbBroad304_03641	ASF1B	-			
6625	-47.78	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
6626	-47.83	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
6627	-47.88	kd	CGS001-10019	SH2B3	Pleckstrin homology (PH) domain containing			
6628	-47.89	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
6629	-47.9	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
6630	-47.93	oe	ccsbBroad304_00975	MAT2A	-			
6631	-48	oe	ccsbBroad304_02231	USP6NL	-			
6632	-48.05	kd	CGS001-170463	SSBP4	-			
6633	-48.06	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
6634	-48.07	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
6635	-48.1	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
6636	-48.19	kd	CGS001-462	SERPINC1	Serine (or cysteine) peptidase inhibitors			
6637	-48.21	kd	CGS001-1050	CEBPA	basic leucine zipper proteins			
6638	-48.23	kd	CGS001-10973	ASCC3	-			
6639	-48.27	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
6640	-48.31	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
6641	-48.32	oe	ccsbBroad304_00491	EIF4EBP2	-			
6642	-48.33	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
6643	-48.35	kd	CGS001-6223	RPS19	S ribosomal proteins			
6644	-48.37	kd	CGS001-1604	CD55	CD molecules			
6645	-48.38	cp	BRD-A75935363	atracurium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
6646	-48.39	cc		Nucleoporin LOF	-			
6647	-48.4	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
6648	-48.41	oe	ccsbBroad304_07275	PSMG1	-			
6649	-48.44	kd	CGS001-2244	FGB	Endogenous ligands			
6650	-48.47	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
6651	-48.47	kd	CGS001-3385	ICAM3	CD molecules			
6652	-48.54	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
6653	-48.58	kd	CGS001-4086	SMAD1	SMADs			
6654	-48.59	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
6655	-48.65	kd	CGS001-10058	ABCB6	ATP binding cassette transporters / subfamily B			
6656	-48.67	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6657	-48.68	kd	CGS001-222546	RFX6	-			
6658	-48.76	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
6659	-48.76	oe	ccsbBroad304_03728	DIABLO	-			
6660	-48.78	kd	CGS001-10289	EIF1B	-			
6661	-48.79	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
6662	-48.8	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
6663	-48.84	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
6664	-48.86	oe	ccsbBroad304_01401	RIT1	-			
6665	-48.88	kd	CGS001-1345	COX6C	Mitochondrial respiratory chain complex			
6666	-48.91	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
6667	-48.93	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
6668	-48.97	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
6669	-49	oe	ccsbBroad304_06367	HK1	-			
6670	-49.02	kd	CGS001-54584	GNB1L	WD repeat domain containing			
6671	-49.04	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6672	-49.06	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
6673	-49.09	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
6674	-49.09	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
6675	-49.25	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6676	-49.26	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
6677	-49.28	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
6678	-49.31	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
6679	-49.34	oe	ccsbBroad304_03533	CDCA8	-			
6680	-49.34	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
6681	-49.38	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6682	-49.41	kd	CGS001-79600	TCTN1	Tectonic proteins			
6683	-49.41	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
6684	-49.43	kd	CGS001-3651	PDX1	Homeoboxes / ANTP class : HOXL subclass			
6685	-49.43	kd	CGS001-10513	APPBP2	-			
6686	-49.45	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
6687	-49.46	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6688	-49.47	kd	CGS001-445	ASS1	-			
6689	-49.48	kd	CGS001-57459	GATAD2B	GATA zinc finger domain containing			
6690	-49.49	kd	CGS001-11015	KDELR3	-			
6691	-49.57	cp	BRD-K18895904	olanzapine	Dopamine receptor antagonist		DRD2, HTR2A, HTR2C, DRD1, DRD3, DRD4, HRH1, HTR1A, HTR1B, HTR1D, HTR1E, HTR6, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C8, DRD5, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH2, HRH4, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
6692	-49.62	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
6693	-49.62	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
6694	-49.63	kd	CGS001-64241	ABCG8	ATP binding cassette transporters / subfamily G			
6695	-49.67	kd	CGS001-2645	GCK	Hexokinases			
6696	-49.67	kd	CGS001-2232	FDXR	-			
6697	-49.69	oe	ccsbBroad304_03266	ERGIC2	-			
6698	-49.73	kd	CGS001-6117	RPA1	-			
6699	-49.74	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6700	-49.75	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
6701	-49.77	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
6702	-49.84	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
6703	-49.88	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
6704	-49.88	oe	ccsbBroad304_07140	XPC	-			
6705	-49.9	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
6706	-49.91	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
6707	-49.94	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6708	-49.96	cp	BRD-A84134924	pancuronium	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRNA1, CHRNA2	Acetylcholine receptor antagonist
6709	-49.97	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
6710	-50.02	kd	CGS001-8841	HDAC3	Histone deacetylases			
6711	-50.08	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6712	-50.09	kd	CGS001-55256	ADI1	-			
6713	-50.12	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
6714	-50.14	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
6715	-50.17	cc		Ribosomal 40s Subunit LOF	-			
6716	-50.2	kd	CGS001-84969	TOX2	-			
6717	-50.21	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
6718	-50.26	kd	CGS001-222894	FERD3L	Basic helix-loop-helix proteins			
6719	-50.3	kd	CGS001-2113	ETS1	ETS Transcription Factors			
6720	-50.32	oe	ccsbBroad304_02220	MTFR1	-			
6721	-50.32	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
6722	-50.34	oe	ccsbBroad304_03812	PBXIP1	-			
6723	-50.35	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
6724	-50.35	cp	BRD-K62374253	rufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6725	-50.47	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
6726	-50.48	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
6727	-50.48	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
6728	-50.5	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
6729	-50.5	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
6730	-50.52	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6731	-50.55	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
6732	-50.65	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6733	-50.72	cp	BRD-K22009844	phenprobamate	Muscle relaxant			Muscle relaxant
6734	-50.73	kd	CGS001-7693	ZNF134	Zinc fingers, C2H2-type			
6735	-50.74	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
6736	-50.75	oe	ccsbBroad304_01948	GAS7	-			
6737	-50.76	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
6738	-50.77	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6739	-50.79	oe	ccsbBroad304_05963	CD44	CD molecules			
6740	-50.81	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
6741	-50.82	kd	CGS001-382	ARF6	ADP-ribosylation factors			
6742	-50.83	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
6743	-50.87	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
6744	-50.9	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
6745	-50.91	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
6746	-50.91	oe	ccsbBroad304_07820	SNW1	-			
6747	-50.93	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
6748	-50.96	kd	CGS001-8915	BCL10	-			
6749	-51.02	oe	ccsbBroad304_00624	GCK	Hexokinases			
6750	-51.03	cc		Serine proteases GOF	-			
6751	-51.04	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
6752	-51.05	kd	CGS001-1504	CTRB1	-			
6753	-51.06	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6754	-51.12	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
6755	-51.12	kd	CGS001-84634	KISS1R	GPCR / Class A : RF amide peptide receptors			
6756	-51.15	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
6757	-51.22	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
6758	-51.27	kd	CGS001-1287	COL4A5	Collagens			
6759	-51.28	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
6760	-51.31	kd	CGS001-9429	ABCG2	ATP binding cassette transporters / subfamily G			
6761	-51.37	kd	CGS001-57804	POLD4	DNA polymerases			
6762	-51.38	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
6763	-51.39	kd	CGS001-55876	GSDMB	-			
6764	-51.46	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
6765	-51.53	kd	CGS001-144811	LACC1	-			
6766	-51.56	kd	CGS001-23335	WDR7	WD repeat domain containing			
6767	-51.56	kd	CGS001-10950	BTG3	-			
6768	-51.57	kd	CGS001-3486	IGFBP3	insulin-like growth factor (IGF) binding proteins			
6769	-51.58	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
6770	-51.6	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
6771	-51.66	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
6772	-51.66	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
6773	-51.68	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6774	-51.72	cc		Integrin subunits beta LOF	-			
6775	-51.75	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
6776	-51.76	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6777	-51.77	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
6778	-51.78	kd	CGS001-5162	PDHB	-			
6779	-51.78	oe	ccsbBroad304_09254	PAQR8	-			
6780	-51.81	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
6781	-51.83	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
6782	-51.83	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
6783	-51.96	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
6784	-51.98	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
6785	-51.99	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
6786	-52.05	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
6787	-52.06	kd	CGS001-898	CCNE1	-			
6788	-52.12	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
6789	-52.12	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
6790	-52.21	kd	CGS001-390212	GPR152	GPCR / Class A : Orphans			
6791	-52.24	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
6792	-52.28	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6793	-52.29	oe	ccsbBroad304_03696	C19ORF10	-			
6794	-52.29	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
6795	-52.29	kd	CGS001-1508	CTSB	Cathepsins			
6796	-52.32	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
6797	-52.34	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6798	-52.34	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
6799	-52.4	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
6800	-52.45	kd	CGS001-8573	CASK	CASK family			
6801	-52.46	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
6802	-52.52	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
6803	-52.52	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
6804	-52.54	kd	CGS001-53632	PRKAG3	AMPK subfamily			
6805	-52.55	oe	ccsbBroad304_01180	PFKFB3	-			
6806	-52.56	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
6807	-52.59	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
6808	-52.64	kd	CGS001-79921	TCEAL4	-			
6809	-52.67	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
6810	-52.72	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
6811	-52.77	kd	CGS001-55968	NSFL1C	UBX domain containing			
6812	-52.81	oe	ccsbBroad304_01013	MIF	-			
6813	-52.81	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
6814	-52.82	kd	CGS001-2987	GUK1	-			
6815	-52.84	kd	CGS001-2308	FOXO1	Forkhead boxes			
6816	-52.85	kd	CGS001-3912	LAMB1	Laminins			
6817	-52.85	oe	ccsbBroad304_07616	ZNF238	-			
6818	-52.85	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
6819	-52.86	kd	CGS001-23131	GPATCH8	G patch domain containing			
6820	-52.89	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
6821	-52.9	oe	ccsbBroad304_03570	QRSL1	-			
6822	-52.9	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
6823	-52.92	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
6824	-52.94	oe	ccsbBroad304_00551	FECH	-			
6825	-52.97	kd	CGS001-51741	WWOX	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6826	-53.15	kd	CGS001-516	ATP5G1	ATPases / F-type			
6827	-53.16	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6828	-53.2	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
6829	-53.21	kd	CGS001-4925	NUCB2	EF-hand domain containing			
6830	-53.22	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
6831	-53.23	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
6832	-53.25	kd	CGS001-5352	PLOD2	-			
6833	-53.41	kd	CGS001-2769	GNA15	-			
6834	-53.42	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
6835	-53.43	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
6836	-53.45	kd	CGS001-4718	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
6837	-53.5	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
6838	-53.51	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
6839	-53.57	oe	ccsbBroad304_01933	TEAD2	-			
6840	-53.59	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
6841	-53.65	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
6842	-53.71	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
6843	-53.72	oe	ccsbBroad304_05756	ACAA1	-			
6844	-53.8	kd	CGS001-673	BRAF	RAF family			
6845	-53.83	kd	CGS001-3688	ITGB1	Integrins			
6846	-53.84	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
6847	-53.86	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
6848	-53.87	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
6849	-53.87	kd	CGS001-930	CD19	CD molecules			
6850	-53.87	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
6851	-53.88	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
6852	-53.92	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
6853	-53.99	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
6854	-54	kd	CGS001-23240	KIAA0922	-			
6855	-54.01	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
6856	-54.04	oe	ccsbBroad304_00957	M6PR	-			
6857	-54.06	kd	CGS001-11007	CCDC85B	-			
6858	-54.08	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
6859	-54.1	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
6860	-54.2	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
6861	-54.21	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
6862	-54.22	kd	CGS001-3309	HSPA5	Heat shock proteins / HSP70			
6863	-54.23	kd	CGS001-1503	CTPS	-			
6864	-54.26	kd	CGS001-323	APBB2	-			
6865	-54.29	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
6866	-54.4	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
6867	-54.42	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
6868	-54.44	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
6869	-54.44	kd	CGS001-1534	CYB561	Cytochrome b genes			
6870	-54.54	kd	CGS001-8726	EED	Neutral sphingomyelinase coupling factors			
6871	-54.56	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
6872	-54.63	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
6873	-54.72	kd	CGS001-4856	NOV	-			
6874	-54.73	kd	CGS001-3689	ITGB2	Integrins			
6875	-54.81	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
6876	-54.82	kd	CGS001-23492	CBX7	-			
6877	-54.84	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
6878	-54.87	kd	CGS001-6443	SGCB	-			
6879	-54.91	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
6880	-54.92	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
6881	-54.97	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
6882	-55.04	oe	ccsbBroad304_01165	PDK1	-			
6883	-55.06	kd	CGS001-9842	PLEKHM1	Pleckstrin homology (PH) domain containing			
6884	-55.12	kd	CGS001-133690	CAPSL	EF-hand domain containing			
6885	-55.16	kd	CGS001-5228	PGF	-			
6886	-55.16	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
6887	-55.17	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
6888	-55.22	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
6889	-55.25	kd	CGS001-11254	SLC6A14	Glycine transporter subfamily			
6890	-55.26	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
6891	-55.26	kd	CGS001-3431	SP110	Non-enzymatic BRD containing proteins			
6892	-55.26	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
6893	-55.27	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
6894	-55.27	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
6895	-55.31	oe	ccsbBroad304_02058	PLOD3	-			
6896	-55.41	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
6897	-55.45	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
6898	-55.47	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
6899	-55.47	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
6900	-55.52	kd	CGS001-4043	LRPAP1	-			
6901	-55.61	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
6902	-55.66	oe	ccsbBroad304_06993	SRD5A1	-			
6903	-55.66	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
6904	-55.67	kd	CGS001-23451	SF3B1	-			
6905	-55.72	kd	CGS001-2000	ELF4	ETS Transcription Factors			
6906	-55.74	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
6907	-55.77	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
6908	-55.78	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
6909	-55.82	kd	CGS001-8575	PRKRA	-			
6910	-55.84	cp	BRD-K52020312	metronidazole	DNA inhibitor		CYP2C8, CYP2E1, CYP3A5, CYP3A7	DNA inhibitor, Antiprotozoal
6911	-55.84	kd	CGS001-2538	G6PC	-			
6912	-55.86	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
6913	-55.89	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
6914	-55.89	kd	CGS001-6201	RPS7	S ribosomal proteins			
6915	-55.97	oe	ccsbBroad304_06739	PLOD1	-			
6916	-56.04	cp	BRD-A12560204	nitrendipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1H, CACNA1S, CACNA2D2, CACNB2, CACNG1, KCNN4	Calcium channel blocker
6917	-56.04	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
6918	-56.05	cp	BRD-A48261811	argatroban	Thrombin inhibitor		F2, CYP3A5	Thrombin inhibitor
6919	-56.07	oe	ccsbBroad304_02386	EIF1B	-			
6920	-56.14	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
6921	-56.14	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
6922	-56.17	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
6923	-56.19	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
6924	-56.25	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
6925	-56.25	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
6926	-56.34	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
6927	-56.35	kd	CGS001-3783	KCNN4	Calcium-activated potassium channels			
6928	-56.37	kd	CGS001-4697	NDUFA4	-			
6929	-56.38	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
6930	-56.38	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
6931	-56.41	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
6932	-56.42	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6933	-56.47	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
6934	-56.47	kd	CGS001-51001	MTERFD1	-			
6935	-56.5	cp	BRD-K05350981	oligomycin-c	ATPase inhibitor		ATP5A1	ATPase inhibitor, ATP synthase inhibitor
6936	-56.63	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
6937	-56.64	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
6938	-56.79	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6939	-56.82	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
6940	-56.82	oe	ccsbBroad304_09756	PAQR7	-			
6941	-56.82	kd	CGS001-84433	CARD11	-			
6942	-56.83	kd	CGS001-11232	POLG2	DNA polymerases			
6943	-56.83	kd	CGS001-3945	LDHB	-			
6944	-56.84	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6945	-56.85	oe	ccsbBroad304_03173	TMED7	-			
6946	-56.85	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
6947	-56.92	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
6948	-56.97	oe	ccsbBroad304_07814	SACM1L	-			
6949	-56.99	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
6950	-57	kd	CGS001-6256	RXRA	Retinoid X receptors			
6951	-57.07	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
6952	-57.07	kd	CGS001-10295	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
6953	-57.07	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
6954	-57.08	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6955	-57.18	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
6956	-57.26	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
6957	-57.32	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6958	-57.43	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
6959	-57.49	kd	CGS001-760	CA2	Carbonic anhydrases			
6960	-57.54	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
6961	-57.61	kd	CGS001-2313	FLI1	ETS Transcription Factors			
6962	-57.63	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
6963	-57.63	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
6964	-57.73	kd	CGS001-9761	MLEC	-			
6965	-57.75	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
6966	-57.77	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
6967	-57.83	kd	CGS001-2737	GLI3	Zinc fingers, C2H2-type			
6968	-57.88	kd	CGS001-7504	XK	Blood group antigens			
6969	-57.92	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
6970	-57.94	kd	CGS001-23597	ACOT9	Acyl CoA thioesterases			
6971	-57.95	cp	BRD-K37516142	idebenone	Calcium channel modulator			Calcium channel modulator
6972	-58.01	kd	CGS001-1891	ECH1	-			
6973	-58.09	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
6974	-58.1	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
6975	-58.12	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
6976	-58.12	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6977	-58.13	oe	ccsbBroad304_01101	NME1	-			
6978	-58.2	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
6979	-58.21	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
6980	-58.26	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
6981	-58.34	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
6982	-58.34	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
6983	-58.37	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6984	-58.37	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
6985	-58.4	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
6986	-58.43	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
6987	-58.46	oe	ccsbBroad304_02509	GMEB1	-			
6988	-58.47	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
6989	-58.58	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
6990	-58.62	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
6991	-58.65	kd	CGS001-9217	VAPB	-			
6992	-58.67	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6993	-58.69	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
6994	-58.7	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
6995	-58.72	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
6996	-58.79	kd	CGS001-3691	ITGB4	Integrins			
6997	-58.8	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6998	-58.81	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
6999	-59	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
7000	-59.01	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
7001	-59.01	kd	CGS001-10628	TXNIP	-			
7002	-59.04	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
7003	-59.07	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
7004	-59.07	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
7005	-59.08	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
7006	-59.1	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
7007	-59.12	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
7008	-59.15	kd	CGS001-10481	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
7009	-59.16	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
7010	-59.2	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
7011	-59.21	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
7012	-59.26	kd	CGS001-10614	HEXIM1	-			
7013	-59.28	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
7014	-59.32	kd	CGS001-2568	GABRP	GABA receptors			
7015	-59.34	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
7016	-59.34	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
7017	-59.36	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
7018	-59.37	kd	CGS001-9111	NMI	-			
7019	-59.38	kd	CGS001-5428	POLG	DNA polymerases			
7020	-59.39	oe	ccsbBroad304_02501	DCTN6	-			
7021	-59.43	kd	CGS001-1545	CYP1B1	Cytochrome P450s			
7022	-59.54	kd	CGS001-339403	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
7023	-59.56	cp	BRD-K29653726	topiramate	Carbonic anhydrase inhibitor		CA2, CA4, GRIK1, CA1, CA12, CA7, CYP2C19, CYP3A4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA1, SCN1A, SCN5A	Carbonic anhydrase inhibitor, Glutamate receptor antagonist, Kainate receptor antagonist
7024	-59.66	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
7025	-59.67	kd	CGS001-7358	UGDH	-			
7026	-59.71	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
7027	-59.72	kd	CGS001-81550	TDRD3	Tudor domain containing			
7028	-59.74	kd	CGS001-2746	GLUD1	-			
7029	-59.76	kd	CGS001-10397	NDRG1	-			
7030	-59.79	kd	CGS001-55556	ENOSF1	-			
7031	-59.8	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
7032	-59.82	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
7033	-59.9	oe	ccsbBroad304_07592	CEPT1	-			
7034	-59.97	oe	ccsbBroad304_01673	TIMP3	-			
7035	-60.03	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
7036	-60.04	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
7037	-60.18	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
7038	-60.21	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
7039	-60.21	cp	BRD-K13800121	parecoxib	Cyclooxygenase inhibitor		LTF, PTGS2	Cyclooxygenase inhibitor
7040	-60.23	kd	CGS001-23658	LSM5	-			
7041	-60.26	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
7042	-60.32	kd	CGS001-1871	E2F3	-			
7043	-60.36	oe	ccsbBroad304_00250	CD19	CD molecules			
7044	-60.39	kd	CGS001-91975	ZNF300	Zinc fingers, C2H2-type			
7045	-60.39	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
7046	-60.41	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
7047	-60.42	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
7048	-60.48	oe	ccsbBroad304_00085	APRT	-			
7049	-60.53	oe	ccsbBroad304_02551	CPSF4	-			
7050	-60.54	oe	ccsbBroad304_03874	UBL5	-			
7051	-60.57	kd	CGS001-7936	RDBP	-			
7052	-60.57	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
7053	-60.67	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
7054	-60.69	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7055	-60.75	cc		PKA inhibitor	-			
7056	-60.75	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
7057	-60.75	kd	CGS001-6722	SRF	-			
7058	-60.76	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
7059	-60.79	cp	BRD-K96740444	itopride	Dopamine receptor antagonist		DRD2, ACHE, CHRM3	Dopamine receptor antagonist
7060	-60.8	oe	ccsbBroad304_08045	NOX1	-			
7061	-60.91	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
7062	-60.91	kd	CGS001-26205	GMEB2	-			
7063	-60.94	oe	ccsbBroad304_02581	ASCC3	-			
7064	-61	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
7065	-61.04	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
7066	-61.07	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
7067	-61.08	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
7068	-61.12	oe	ccsbBroad304_04534	HN1L	-			
7069	-61.13	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
7070	-61.15	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
7071	-61.2	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
7072	-61.26	kd	CGS001-64422	ATG3	-			
7073	-61.33	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
7074	-61.41	kd	CGS001-271	AMPD2	-			
7075	-61.42	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
7076	-61.44	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
7077	-61.44	kd	CGS001-23224	SYNE2	-			
7078	-61.55	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
7079	-61.62	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
7080	-61.67	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
7081	-61.68	kd	CGS001-338557	O3FAR1	-			
7082	-61.75	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
7083	-61.78	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
7084	-61.79	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
7085	-61.81	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
7086	-61.84	kd	CGS001-8800	PEX11A	-			
7087	-61.86	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
7088	-61.93	cp	BRD-K43236057	piceid	ICAM1 inhibitor		GAA, XDH	ICAM1 inhibitor
7089	-61.94	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
7090	-61.95	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
7091	-62.05	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
7092	-62.15	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
7093	-62.16	kd	CGS001-978	CDA	-			
7094	-62.17	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
7095	-62.24	kd	CGS001-571	BACH1	BTB/POZ domain containing			
7096	-62.31	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
7097	-62.4	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
7098	-62.44	cc		Nucleophosmin inhibitor	-			
7099	-62.44	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
7100	-62.46	oe	ccsbBroad304_00995	MECP2	-			
7101	-62.47	kd	CGS001-5824	PEX19	-			
7102	-62.48	oe	ccsbBroad304_02175	MAGED1	-			
7103	-62.6	kd	CGS001-84971	ATG4D	-			
7104	-62.6	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
7105	-62.65	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
7106	-62.69	kd	CGS001-23212	RRS1	-			
7107	-62.75	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
7108	-62.77	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
7109	-62.77	oe	ccsbBroad304_02484	PAICS	-			
7110	-62.83	kd	CGS001-57665	RDH14	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
7111	-62.85	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
7112	-62.85	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
7113	-62.87	kd	CGS001-1841	DTYMK	-			
7114	-62.94	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
7115	-62.99	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
7116	-63.01	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
7117	-63.05	kd	CGS001-4846	NOS3	Nitric oxide synthases			
7118	-63.06	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
7119	-63.18	kd	CGS001-22818	COPZ1	-			
7120	-63.18	kd	CGS001-400	ARL1	ADP-ribosylation factors			
7121	-63.19	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
7122	-63.21	kd	CGS001-64135	IFIH1	-			
7123	-63.22	kd	CGS001-64786	TBC1D15	-			
7124	-63.25	kd	CGS001-238	ALK	Leukocyte tyrosine kinase (LTK) receptor family			
7125	-63.28	kd	CGS001-9453	GGPS1	Lanosterol biosynthesis pathway			
7126	-63.35	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
7127	-63.36	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
7128	-63.44	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
7129	-63.45	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
7130	-63.5	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
7131	-63.54	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
7132	-63.57	oe	ccsbBroad304_02677	PDAP1	-			
7133	-63.6	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
7134	-63.61	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
7135	-63.68	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
7136	-63.69	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
7137	-63.73	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
7138	-63.73	kd	CGS001-51024	FIS1	-			
7139	-63.78	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
7140	-63.79	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
7141	-63.8	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
7142	-63.85	oe	ccsbBroad304_13952	SHMT2	-			
7143	-63.85	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
7144	-63.87	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
7145	-63.88	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
7146	-63.93	oe	ccsbBroad304_01001	MEST	-			
7147	-63.95	kd	CGS001-8148	TAF15	RNA binding motif (RRM) containing			
7148	-63.96	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
7149	-63.98	kd	CGS001-10915	TCERG1	-			
7150	-63.98	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
7151	-64.02	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
7152	-64.03	kd	CGS001-7424	VEGFC	-			
7153	-64.05	cc		EMSY complex LOF	-			
7154	-64.06	kd	CGS001-3588	IL10RB	IL-10 receptor family			
7155	-64.16	cp	BRD-K39983086	loteprednol	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Phospholipase inhibitor
7156	-64.16	cp	BRD-A94543220	bifonazole	Sterol demethylase inhibitor		CYP2B6	Sterol demethylase inhibitor
7157	-64.17	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
7158	-64.21	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
7159	-64.21	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
7160	-64.3	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
7161	-64.33	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
7162	-64.33	kd	CGS001-30001	ERO1L	-			
7163	-64.34	kd	CGS001-7343	UBTF	-			
7164	-64.42	oe	ccsbBroad304_01845	RDBP	-			
7165	-64.43	cp	BRD-K50384076	7,4'-dihydroxyflavone	Opioid receptor antagonist		CYP19A1	Opioid receptor antagonist
7166	-64.47	kd	CGS001-1026	CDKN1A	-			
7167	-64.5	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
7168	-64.5	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
7169	-64.53	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
7170	-64.58	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
7171	-64.6	kd	CGS001-11044	PAPD7	-			
7172	-64.67	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
7173	-64.76	oe	ccsbBroad304_00464	DTNA	-			
7174	-64.79	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
7175	-64.83	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
7176	-64.84	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
7177	-64.86	cc		Sigma receptor antagonist	-			
7178	-64.86	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
7179	-64.87	kd	CGS001-4942	OAT	-			
7180	-64.9	kd	CGS001-84288	EFCAB2	EF-hand domain containing			
7181	-64.93	cp	BRD-K33483813	actarit	Interleukin receptor agonist			Interleukin receptor agonist
7182	-65.03	kd	CGS001-1213	CLTC	-			
7183	-65.04	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
7184	-65.08	kd	CGS001-51172	NAGPA	-			
7185	-65.09	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
7186	-65.1	kd	CGS001-4637	MYL6	EF-hand domain containing			
7187	-65.17	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
7188	-65.2	kd	CGS001-8985	PLOD3	-			
7189	-65.21	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
7190	-65.27	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
7191	-65.33	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
7192	-65.34	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
7193	-65.36	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
7194	-65.37	kd	CGS001-2805	GOT1	-			
7195	-65.42	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
7196	-65.43	kd	CGS001-26271	FBXO5	F-boxes / other			
7197	-65.44	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
7198	-65.46	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
7199	-65.53	kd	CGS001-3559	IL2RA	IL-2 receptor family			
7200	-65.55	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
7201	-65.55	kd	CGS001-6453	ITSN1	Rho guanine nucleotide exchange factors			
7202	-65.56	kd	CGS001-326	AIRE	Zinc fingers, PHD-type			
7203	-65.59	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
7204	-65.59	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
7205	-65.68	kd	CGS001-10427	SEC24B	-			
7206	-65.69	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
7207	-65.75	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
7208	-65.76	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
7209	-65.76	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
7210	-65.78	kd	CGS001-7541	ZFP161	-			
7211	-65.78	kd	CGS001-51096	UTP18	WD repeat domain containing			
7212	-65.87	kd	CGS001-11215	AKAP11	A-kinase anchor proteins			
7213	-65.89	kd	CGS001-335	APOA1	Apolipoproteins			
7214	-65.89	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
7215	-65.9	kd	CGS001-5073	PARN	-			
7216	-65.97	oe	ccsbBroad304_04619	GNG8	-			
7217	-65.98	oe	ccsbBroad304_04190	CCDC92	-			
7218	-66.02	kd	CGS001-1718	DHCR24	-			
7219	-66.03	kd	CGS001-9406	ZRANB2	Zinc fingers, RAN-binding domain containing			
7220	-66.08	kd	CGS001-5277	PIGA	Glycosyltransferase group 1 domain containing			
7221	-66.09	cp	BRD-K44442813	pidotimod	Interferon receptor agonist			Interferon receptor agonist, Interleukin receptor agonist
7222	-66.12	oe	ccsbBroad304_07349	MAP7	-			
7223	-66.16	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
7224	-66.16	kd	CGS001-10379	IRF9	-			
7225	-66.22	cp	BRD-A02189320	met-leu-phe	-666			-666
7226	-66.22	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
7227	-66.26	kd	CGS001-3315	HSPB1	Heat shock proteins / HSPB			
7228	-66.26	kd	CGS001-3205	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
7229	-66.27	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
7230	-66.28	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
7231	-66.35	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
7232	-66.36	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
7233	-66.38	oe	ccsbBroad304_06225	FTH1	-			
7234	-66.39	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
7235	-66.39	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
7236	-66.41	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
7237	-66.42	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
7238	-66.46	kd	CGS001-6046	BRD2	Bromodomain kinase (BRDK) family			
7239	-66.5	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
7240	-66.51	kd	CGS001-348	APOE	Apolipoproteins			
7241	-66.54	kd	CGS001-29911	HOOK2	-			
7242	-66.56	kd	CGS001-2017	CTTN	-			
7243	-66.56	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7244	-66.56	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
7245	-66.61	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
7246	-66.64	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
7247	-66.7	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
7248	-66.71	kd	CGS001-8027	STAM	-			
7249	-66.72	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
7250	-66.83	kd	CGS001-256364	EML3	WD repeat domain containing			
7251	-66.85	kd	CGS001-54472	TOLLIP	-			
7252	-66.92	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
7253	-67.02	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
7254	-67.09	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
7255	-67.09	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
7256	-67.15	kd	CGS001-4938	OAS1	-			
7257	-67.18	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
7258	-67.18	kd	CGS001-5636	PRPSAP2	-			
7259	-67.21	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
7260	-67.28	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
7261	-67.28	oe	ccsbBroad304_02292	BCL2L11	-			
7262	-67.31	kd	CGS001-124626	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7263	-67.31	kd	CGS001-192669	EIF2C3	-			
7264	-67.37	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
7265	-67.37	kd	CGS001-1147	CHUK	IKK family			
7266	-67.4	kd	CGS001-9308	CD83	CD molecules			
7267	-67.41	kd	CGS001-55634	ZNF673	-			
7268	-67.42	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
7269	-67.43	oe	ccsbBroad304_00501	EMD	-			
7270	-67.44	cc		Tumor necrosis factor superfamily LOF	-			
7271	-67.48	oe	ccsbBroad304_06639	NFYB	-			
7272	-67.56	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
7273	-67.65	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
7274	-67.74	cc		Bacterial cell wall synthesis inhibitor	-			
7275	-67.74	kd	CGS001-23039	XPO7	Exportins			
7276	-67.76	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
7277	-67.78	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
7278	-67.79	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
7279	-67.8	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
7280	-67.89	kd	CGS001-10342	TFG	-			
7281	-67.94	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
7282	-68	oe	ccsbBroad304_00819	IDH3B	-			
7283	-68.05	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
7284	-68.06	kd	CGS001-5269	SERPINB6	Serine (or cysteine) peptidase inhibitors			
7285	-68.13	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
7286	-68.19	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
7287	-68.22	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7288	-68.26	cc		Bacterial DNA gyrase inhibitor	-			
7289	-68.26	cp	BRD-K92413528	thiazolidinecarboxylic-acid	Reducing agent			Reducing agent
7290	-68.28	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
7291	-68.28	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
7292	-68.32	kd	CGS001-29110	TBK1	IKK family			
7293	-68.39	oe	ccsbBroad304_01485	SC5DL	-			
7294	-68.41	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
7295	-68.42	oe	ccsbBroad304_03625	HIF1AN	-			
7296	-68.47	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
7297	-68.53	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
7298	-68.59	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
7299	-68.61	kd	CGS001-25805	BAMBI	-			
7300	-68.65	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
7301	-68.65	oe	ccsbBroad304_00818	IDH3A	-			
7302	-68.67	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
7303	-68.71	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
7304	-68.75	oe	ccsbBroad304_06683	FURIN	Subtilisin			
7305	-68.77	oe	ccsbBroad304_06870	RNH1	-			
7306	-68.82	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
7307	-68.82	kd	CGS001-345611	IRGM	-			
7308	-68.85	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
7309	-68.85	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
7310	-68.9	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
7311	-68.9	cp	BRD-A56892734	esomeprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
7312	-68.91	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
7313	-68.91	kd	CGS001-55143	CDCA8	-			
7314	-68.93	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
7315	-69.06	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
7316	-69.08	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
7317	-69.09	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
7318	-69.13	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
7319	-69.19	kd	CGS001-3570	IL6R	IL-6 receptor family			
7320	-69.23	kd	CGS001-7032	TFF2	-			
7321	-69.24	kd	CGS001-218	ALDH3A1	Aldehyde dehydrogenases			
7322	-69.27	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
7323	-69.28	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
7324	-69.31	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
7325	-69.33	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
7326	-69.41	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
7327	-69.42	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
7328	-69.49	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
7329	-69.55	oe	ccsbBroad304_06562	MAT1A	-			
7330	-69.58	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
7331	-69.61	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
7332	-69.61	kd	CGS001-5992	RFX4	-			
7333	-69.64	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
7334	-69.79	oe	ccsbBroad304_00816	IDE	Pitrilysin			
7335	-69.8	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
7336	-69.89	kd	CGS001-8317	CDC7	CDC7 family			
7337	-69.91	kd	CGS001-23047	PDS5B	-			
7338	-69.92	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
7339	-69.93	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
7340	-70	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
7341	-70	kd	CGS001-159	ADSS	-			
7342	-70.03	kd	CGS001-23012	STK38L	NDR family			
7343	-70.12	kd	CGS001-9322	TRIP10	-			
7344	-70.12	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
7345	-70.15	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
7346	-70.18	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
7347	-70.21	kd	CGS001-2002	ELK1	ETS Transcription Factors			
7348	-70.28	kd	CGS001-114904	C1QTNF6	-			
7349	-70.3	kd	CGS001-5442	POLRMT	-			
7350	-70.32	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
7351	-70.4	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
7352	-70.45	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
7353	-70.5	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
7354	-70.51	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
7355	-70.53	kd	CGS001-23649	POLA2	DNA polymerases			
7356	-70.53	kd	CGS001-2108	ETFA	-			
7357	-70.56	oe	ccsbBroad304_00529	F3	CD molecules			
7358	-70.56	kd	CGS001-3455	IFNAR2	Interferon receptor family			
7359	-70.58	oe	ccsbBroad304_02138	TRIP10	-			
7360	-70.59	kd	CGS001-6499	SKIV2L	-			
7361	-70.59	kd	CGS001-79902	NUP85	-			
7362	-70.64	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
7363	-70.65	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
7364	-70.66	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
7365	-70.67	kd	CGS001-843	CASP10	Caspases			
7366	-70.69	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
7367	-70.7	oe	ccsbBroad304_14143	NUSAP1	-			
7368	-70.73	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
7369	-70.76	kd	CGS001-5209	PFKFB3	-			
7370	-70.78	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
7371	-70.81	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
7372	-70.84	oe	ccsbBroad304_01855	NCOA4	-			
7373	-70.88	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7374	-70.89	kd	CGS001-286530	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
7375	-70.91	kd	CGS001-174	AFP	-			
7376	-70.97	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
7377	-70.97	kd	CGS001-3985	LIMK2	LIMK subfamily			
7378	-70.98	kd	CGS001-9159	PCSK7	Subtilisin			
7379	-70.99	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
7380	-71.12	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
7381	-71.17	cp	BRD-K49404994	levetiracetam	Calcium channel blocker		SV2A, CACNA1B, SCN1A	Calcium channel blocker
7382	-71.19	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
7383	-71.37	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
7384	-71.43	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
7385	-71.43	kd	CGS001-3155	HMGCL	-			
7386	-71.44	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
7387	-71.45	oe	ccsbBroad304_08878	METTL4	-			
7388	-71.45	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
7389	-71.46	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
7390	-71.47	oe	ccsbBroad304_01215	PLAUR	CD molecules			
7391	-71.51	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
7392	-71.59	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
7393	-71.64	oe	ccsbBroad304_00170	BNIP1	-			
7394	-71.68	oe	ccsbBroad304_00960	SMAD1	SMADs			
7395	-71.7	kd	CGS001-79094	CHAC1	-			
7396	-71.71	cp	BRD-A07395371	esmolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
7397	-71.72	oe	ccsbBroad304_00888	ITPK1	-			
7398	-71.77	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
7399	-71.82	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
7400	-71.83	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
7401	-71.88	oe	ccsbBroad304_00389	CTBP1	-			
7402	-71.9	kd	CGS001-6774	STAT3	SH2 domain containing			
7403	-71.91	kd	CGS001-10434	LYPLA1	-			
7404	-71.94	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
7405	-71.95	oe	ccsbBroad304_07024	SYK	Syk family			
7406	-71.96	kd	CGS001-6257	RXRB	Retinoid X receptors			
7407	-71.97	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
7408	-71.99	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
7409	-72.02	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
7410	-72.03	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
7411	-72.03	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
7412	-72.03	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
7413	-72.07	kd	CGS001-130497	OSR1	Zinc fingers, C2H2-type			
7414	-72.09	oe	ccsbBroad304_08426	TEX10	-			
7415	-72.12	kd	CGS001-91433	RCCD1	-			
7416	-72.17	kd	CGS001-5345	SERPINF2	Serine (or cysteine) peptidase inhibitors			
7417	-72.22	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
7418	-72.4	kd	CGS001-11014	KDELR2	-			
7419	-72.59	kd	CGS001-8270	LAGE3	-			
7420	-72.6	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
7421	-72.64	cp	BRD-A11990600	lorazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, TSPO	Benzodiazepine receptor agonist
7422	-72.65	oe	ccsbBroad304_06828	PYCR1	-			
7423	-72.7	kd	CGS001-6520	SLC3A2	SLC3 family			
7424	-72.76	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
7425	-72.77	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
7426	-72.82	cp	BRD-K63343048	orlistat	Lipase inhibitor		PNLIP, DAGLA, FASN, LIPF, CNR1, DAGLB	Lipase inhibitor
7427	-72.82	kd	CGS001-6909	TBX2	T-boxes			
7428	-72.83	kd	CGS001-103	ADAR	-			
7429	-72.86	kd	CGS001-2052	EPHX1	-			
7430	-72.89	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
7431	-72.98	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
7432	-73	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
7433	-73.05	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
7434	-73.05	kd	CGS001-2783	GNB2	WD repeat domain containing			
7435	-73.06	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
7436	-73.09	kd	CGS001-8659	ALDH4A1	Aldehyde dehydrogenases			
7437	-73.1	kd	CGS001-3661	IRF3	-			
7438	-73.18	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
7439	-73.19	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
7440	-73.32	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
7441	-73.33	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
7442	-73.48	kd	CGS001-4706	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
7443	-73.48	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
7444	-73.48	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
7445	-73.51	kd	CGS001-79090	TRAPPC6A	Trafficking protein particle complex			
7446	-73.52	cc		V type ATPases LOF	-			
7447	-73.53	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
7448	-73.54	cc		HIV protease inhibitor	-			
7449	-73.55	kd	CGS001-79711	IPO4	Importins			
7450	-73.57	kd	CGS001-8996	NOL3	-			
7451	-73.58	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
7452	-73.65	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
7453	-73.67	kd	CGS001-5982	RFC2	ATPases / AAA-type			
7454	-73.7	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
7455	-73.74	kd	CGS001-23161	SNX13	Sorting nexins			
7456	-73.78	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
7457	-73.79	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
7458	-73.84	cp	BRD-K22947005	dexbrompheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
7459	-73.84	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
7460	-73.86	kd	CGS001-3339	HSPG2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7461	-73.88	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
7462	-73.89	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
7463	-73.91	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
7464	-73.95	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
7465	-73.98	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
7466	-74.02	oe	ccsbBroad304_02668	PNKP	-			
7467	-74.05	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
7468	-74.08	kd	CGS001-10887	PROKR1	GPCR / Class A : Prokineticin receptors			
7469	-74.11	kd	CGS001-2152	F3	CD molecules			
7470	-74.11	oe	ccsbBroad304_07887	GCAT	-			
7471	-74.16	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
7472	-74.21	kd	CGS001-5167	ENPP1	-			
7473	-74.24	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
7474	-74.29	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
7475	-74.31	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
7476	-74.33	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
7477	-74.34	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
7478	-74.44	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
7479	-74.44	kd	CGS001-10456	HAX1	-			
7480	-74.47	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
7481	-74.61	oe	ccsbBroad304_00490	EIF4EBP1	-			
7482	-74.64	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
7483	-74.66	kd	CGS001-8743	TNFSF10	CD molecules			
7484	-74.69	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
7485	-74.72	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
7486	-74.81	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
7487	-74.82	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
7488	-74.83	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
7489	-74.88	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
7490	-74.88	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
7491	-74.91	oe	ccsbBroad304_02230	HERPUD1	-			
7492	-74.91	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7493	-74.96	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
7494	-74.99	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
7495	-75	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
7496	-75.03	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
7497	-75.03	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
7498	-75.09	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
7499	-75.17	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
7500	-75.21	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
7501	-75.24	oe	ccsbBroad304_06090	DDOST	-			
7502	-75.25	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
7503	-75.27	cc		Tubulin inhibitor	-			
7504	-75.27	cp	BRD-K82109576	vincristine	Tubulin inhibitor		TUBB, TUBA4A	Tubulin inhibitor
7505	-75.3	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
7506	-75.31	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
7507	-75.32	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
7508	-75.33	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
7509	-75.34	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
7510	-75.36	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
7511	-75.36	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
7512	-75.37	kd	CGS001-55229	PANK4	-			
7513	-75.41	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
7514	-75.44	kd	CGS001-471	ATIC	-			
7515	-75.46	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
7516	-75.5	kd	CGS001-5869	RAB5B	RAB, member RAS oncogene			
7517	-75.54	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
7518	-75.54	oe	ccsbBroad304_02249	KIAA0494	-			
7519	-75.57	kd	CGS001-3821	KLRC1	CD molecules			
7520	-75.59	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
7521	-75.59	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
7522	-75.6	kd	CGS001-55379	LRRC59	-			
7523	-75.73	oe	ccsbBroad304_00542	FBP1	-			
7524	-75.74	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
7525	-75.75	kd	CGS001-3705	ITPK1	-			
7526	-75.85	kd	CGS001-6646	SOAT1	-			
7527	-75.87	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
7528	-75.87	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
7529	-75.9	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
7530	-75.95	kd	CGS001-2828	GPR4	GPCR / Class A : Orphans			
7531	-75.98	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
7532	-75.99	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
7533	-76.03	oe	ccsbBroad304_05985	CFL1	-			
7534	-76.06	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
7535	-76.11	kd	CGS001-79170	PRR15L	-			
7536	-76.16	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
7537	-76.17	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
7538	-76.17	kd	CGS001-26959	HBP1	-			
7539	-76.2	kd	CGS001-5887	RAD23B	-			
7540	-76.24	kd	CGS001-3298	HSF2	-			
7541	-76.31	kd	CGS001-645	BLVRB	Short chain dehydrogenase/reductase superfamily / Atypical members			
7542	-76.31	kd	CGS001-122402	TDRD9	Tudor domain containing			
7543	-76.33	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
7544	-76.34	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
7545	-76.4	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
7546	-76.4	kd	CGS001-79796	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
7547	-76.47	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
7548	-76.5	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
7549	-76.5	oe	ccsbBroad304_05098	MAGEB6	-			
7550	-76.53	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
7551	-76.55	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
7552	-76.57	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
7553	-76.59	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
7554	-76.6	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
7555	-76.61	kd	CGS001-9128	PRPF4	WD repeat domain containing			
7556	-76.64	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
7557	-76.66	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
7558	-76.75	oe	ccsbBroad304_02229	TRAM2	-			
7559	-76.79	kd	CGS001-9377	COX5A	Mitochondrial respiratory chain complex			
7560	-76.81	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
7561	-76.82	kd	CGS001-2004	ELK3	ETS Transcription Factors			
7562	-76.83	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
7563	-76.83	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
7564	-76.96	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
7565	-76.97	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
7566	-77.02	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
7567	-77.1	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
7568	-77.17	kd	CGS001-5498	PPOX	-			
7569	-77.19	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
7570	-77.27	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7571	-77.29	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
7572	-77.34	kd	CGS001-5595	MAPK3	MAPK:ERK subfamily			
7573	-77.35	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
7574	-77.37	kd	CGS001-9655	SOCS5	SH2 domain containing			
7575	-77.4	cp	BRD-K70883034	nimetazepam	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA receptor agonist
7576	-77.42	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
7577	-77.42	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
7578	-77.49	kd	CGS001-4303	FOXO4	Forkhead boxes			
7579	-77.5	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
7580	-77.5	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
7581	-77.51	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
7582	-77.61	kd	CGS001-8859	STK19	G11 family			
7583	-77.64	kd	CGS001-8438	RAD54L	-			
7584	-77.65	kd	CGS001-80762	NDFIP1	-			
7585	-77.7	oe	ccsbBroad304_00116	ASS1	-			
7586	-77.7	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
7587	-77.7	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
7588	-77.74	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
7589	-77.74	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
7590	-77.75	kd	CGS001-9053	MAP7	-			
7591	-77.76	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
7592	-77.77	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
7593	-77.79	kd	CGS001-80347	COASY	-			
7594	-77.91	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
7595	-77.96	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
7596	-77.98	kd	CGS001-166	AES	-			
7597	-78.04	kd	CGS001-8914	TIMELESS	-			
7598	-78.07	oe	ccsbBroad304_06126	TSC22D3	-			
7599	-78.11	kd	CGS001-4171	MCM2	-			
7600	-78.11	oe	ccsbBroad304_02838	SDF2L1	-			
7601	-78.13	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
7602	-78.18	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
7603	-78.2	oe	ccsbBroad304_02173	ATG5	-			
7604	-78.24	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
7605	-78.31	kd	CGS001-2745	GLRX	-			
7606	-78.35	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
7607	-78.38	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
7608	-78.45	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
7609	-78.53	kd	CGS001-23075	SWAP70	EF-hand domain containing			
7610	-78.54	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
7611	-78.55	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
7612	-78.56	kd	CGS001-81544	GDPD5	-			
7613	-78.59	kd	CGS001-64087	MCCC2	-			
7614	-78.65	kd	CGS001-4904	YBX1	-			
7615	-78.67	kd	CGS001-663	BNIP2	-			
7616	-78.76	kd	CGS001-1198	CLK3	CDC-like kinases			
7617	-78.85	kd	CGS001-10898	CPSF4	-			
7618	-78.88	oe	ccsbBroad304_08023	EIF2C1	-			
7619	-78.9	cp	BRD-K31491153	1-phenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
7620	-78.92	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
7621	-78.96	kd	CGS001-3479	IGF1	Endogenous ligands			
7622	-78.97	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
7623	-79	cp	BRD-K49668410	clarithromycin	Bacterial 50S ribosomal subunit inhibitor		CYP2C19, CYP3A4, CYP3A5, CYP3A7	Bacterial 50S ribosomal subunit inhibitor
7624	-79.05	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
7625	-79.05	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
7626	-79.07	kd	CGS001-390	RND3	-			
7627	-79.14	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
7628	-79.15	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
7629	-79.18	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
7630	-79.3	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
7631	-79.36	kd	CGS001-10298	PAK4	PAKB subfamily			
7632	-79.4	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
7633	-79.43	kd	CGS001-51655	RASD1	-			
7634	-79.48	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
7635	-79.5	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
7636	-79.51	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
7637	-79.54	kd	CGS001-22841	RAB11FIP2	-			
7638	-79.55	kd	CGS001-9955	HS3ST3A1	Sulfotransferases, membrane-bound			
7639	-79.57	kd	CGS001-168374	ZNF92	Zinc fingers, C2H2-type			
7640	-79.57	kd	CGS001-64754	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
7641	-79.62	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
7642	-79.64	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
7643	-79.69	kd	CGS001-4790	NFKB1	NFkappaB transcription factor family			
7644	-79.73	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
7645	-79.76	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
7646	-79.79	oe	ccsbBroad304_00150	BAX	-			
7647	-79.81	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
7648	-79.82	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
7649	-79.85	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
7650	-79.98	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
7651	-80	oe	ccsbBroad304_07548	TSSC4	-			
7652	-80.01	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
7653	-80.04	kd	CGS001-4916	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
7654	-80.1	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
7655	-80.14	oe	ccsbBroad304_01640	TAF12	-			
7656	-80.17	kd	CGS001-54807	ZNF586	Zinc fingers, C2H2-type			
7657	-80.17	kd	CGS001-55893	ZNF395	Zinc fingers, C2H2-type			
7658	-80.18	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
7659	-80.27	kd	CGS001-162	AP1B1	-			
7660	-80.28	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
7661	-80.29	kd	CGS001-24140	FTSJ1	-			
7662	-80.41	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
7663	-80.41	kd	CGS001-3459	IFNGR1	Interferon receptor family			
7664	-80.42	kd	CGS001-143187	VTI1A	-			
7665	-80.43	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
7666	-80.45	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
7667	-80.49	kd	CGS001-2592	GALT	-			
7668	-80.51	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
7669	-80.53	cp	BRD-K33226500	indinavir	HIV protease inhibitor		CYP3A5	HIV protease inhibitor
7670	-80.57	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
7671	-80.67	kd	CGS001-1892	ECHS1	-			
7672	-80.69	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
7673	-80.74	cc		Mitochondrial complex IV LOF	-			
7674	-80.87	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
7675	-80.87	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
7676	-80.93	kd	CGS001-2274	FHL2	-			
7677	-80.93	kd	CGS001-1509	CTSD	Cathepsins			
7678	-80.94	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
7679	-80.99	kd	CGS001-2697	GJA1	Ion channels / Gap junction proteins (connexins)			
7680	-81.05	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
7681	-81.06	kd	CGS001-219333	USP12	Ubiquitin-specific peptidases			
7682	-81.11	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
7683	-81.12	oe	ccsbBroad304_04465	RERG	-			
7684	-81.17	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
7685	-81.18	kd	CGS001-2078	ERG	ETS Transcription Factors			
7686	-81.23	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
7687	-81.25	kd	CGS001-9474	ATG5	-			
7688	-81.32	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
7689	-81.33	kd	CGS001-10657	KHDRBS1	-			
7690	-81.37	kd	CGS001-10269	ZMPSTE24	-			
7691	-81.42	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
7692	-81.45	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
7693	-81.52	kd	CGS001-9854	C2CD2L	-			
7694	-81.54	oe	ccsbBroad304_03573	BRF2	-			
7695	-81.57	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
7696	-81.63	kd	CGS001-7625	ZNF74	Zinc fingers, C2H2-type			
7697	-81.68	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
7698	-81.72	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
7699	-81.74	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
7700	-81.78	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
7701	-81.78	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
7702	-81.79	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
7703	-81.79	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
7704	-81.82	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
7705	-81.87	oe	ccsbBroad304_08879	CASD1	-			
7706	-81.9	oe	ccsbBroad304_02822	ARFIP2	-			
7707	-81.91	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
7708	-81.99	cp	BRD-A24191444	ifenprodil	Adrenergic receptor antagonist		GRIN1, GRIN2B	Adrenergic receptor antagonist, Glutamate receptor antagonist
7709	-81.99	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
7710	-82.01	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7711	-82.03	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
7712	-82.03	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
7713	-82.12	kd	CGS001-523	ATP6V1A	ATPases / V-type			
7714	-82.13	kd	CGS001-5608	MAP2K6	MAPKK:STE7 family			
7715	-82.18	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
7716	-82.25	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7717	-82.28	kd	CGS001-5825	ABCD3	ATP binding cassette transporters / subfamily D			
7718	-82.28	cp	BRD-A39390670	rabeprazole	ATPase inhibitor		ATP4A, CYP2C19	ATPase inhibitor, Gastrin inhibitor
7719	-82.31	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
7720	-82.37	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
7721	-82.43	kd	CGS001-39	ACAT2	Lanosterol biosynthesis pathway			
7722	-82.49	kd	CGS001-8892	EIF2B2	-			
7723	-82.5	kd	CGS001-3995	FADS3	Fatty acid desaturases			
7724	-82.58	cp	BRD-K86003836	flubendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
7725	-82.59	kd	CGS001-9961	MVP	-			
7726	-82.62	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
7727	-82.63	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
7728	-82.64	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
7729	-82.72	kd	CGS001-2857	GPR34	GPCR / Class A : Orphans			
7730	-82.79	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
7731	-82.83	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
7732	-82.88	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
7733	-82.92	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
7734	-82.94	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
7735	-82.99	kd	CGS001-5898	RALA	-			
7736	-83.01	oe	ccsbBroad304_02831	SGK3	SGK family			
7737	-83.03	kd	CGS001-150962	PUS10	-			
7738	-83.03	oe	ccsbBroad304_01183	PGD	-			
7739	-83.06	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
7740	-83.14	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
7741	-83.15	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
7742	-83.17	kd	CGS001-440	ASNS	-			
7743	-83.24	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
7744	-83.25	kd	CGS001-23139	MAST2	MAST family			
7745	-83.3	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
7746	-83.33	kd	CGS001-2771	GNAI2	-			
7747	-83.35	kd	CGS001-3672	ITGA1	Integrins			
7748	-83.39	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
7749	-83.41	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
7750	-83.44	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
7751	-83.45	kd	CGS001-11182	SLC2A6	Solute carriers			
7752	-83.46	kd	CGS001-8893	EIF2B5	-			
7753	-83.57	kd	CGS001-8660	IRS2	Pleckstrin homology (PH) domain containing			
7754	-83.59	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
7755	-83.63	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
7756	-83.66	kd	CGS001-6605	SMARCE1	-			
7757	-83.68	kd	CGS001-5460	POU5F1	Homeoboxes / POU class			
7758	-83.69	kd	CGS001-100133941	CD24	CD molecules			
7759	-83.69	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
7760	-83.7	oe	ccsbBroad304_00155	CCND1	-			
7761	-83.75	kd	CGS001-94239	H2AFV	Histones / Replication-independent			
7762	-83.76	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
7763	-83.77	kd	CGS001-56005	C19ORF10	-			
7764	-83.79	oe	ccsbBroad304_00184	C2	Complement system			
7765	-83.84	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
7766	-83.84	kd	CGS001-23211	ZC3H4	Zinc fingers, CCCH-type domain containing			
7767	-83.85	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
7768	-83.88	kd	CGS001-2643	GCH1	-			
7769	-83.92	kd	CGS001-51466	EVL	-			
7770	-83.94	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
7771	-83.99	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
7772	-83.99	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
7773	-84	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
7774	-84.05	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
7775	-84.07	kd	CGS001-80025	PANK2	-			
7776	-84.09	kd	CGS001-3659	IRF1	-			
7777	-84.09	kd	CGS001-1594	CYP27B1	Cytochrome P450s			
7778	-84.16	kd	CGS001-3575	IL7R	IL-2 receptor family			
7779	-84.17	kd	CGS001-9213	XPR1	-			
7780	-84.17	kd	CGS001-10857	PGRMC1	-			
7781	-84.18	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
7782	-84.22	kd	CGS001-116443	GRIN3A	Glutamate receptors			
7783	-84.28	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
7784	-84.4	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
7785	-84.4	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
7786	-84.47	kd	CGS001-51530	ZC3HC1	Zinc fingers, C3HC-type			
7787	-84.48	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
7788	-84.54	oe	ccsbBroad304_07145	ZFP161	-			
7789	-84.55	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
7790	-84.55	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
7791	-84.58	kd	CGS001-6342	SCP2	-			
7792	-84.71	oe	ccsbBroad304_02578	EBNA1BP2	-			
7793	-84.73	oe	ccsbBroad304_00991	MDH1	-			
7794	-84.74	kd	CGS001-5335	PLCG1	Phosphoinositide-specific phospholipase C			
7795	-84.89	cc		Aminoacyl tRNA synthetases class II LOF	-			
7796	-84.96	oe	ccsbBroad304_02741	PDS5A	-			
7797	-84.97	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
7798	-85.01	kd	CGS001-10606	PAICS	-			
7799	-85.03	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
7800	-85.11	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
7801	-85.14	cp	BRD-K29113274	ketoconazole	Sterol demethylase inhibitor		AR, CYP19A1, CYP21A2, CYP2C19, CYP3A5, CYP3A7, KCNA10	Sterol demethylase inhibitor
7802	-85.15	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7803	-85.16	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
7804	-85.17	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
7805	-85.17	kd	CGS001-1642	DDB1	-			
7806	-85.2	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
7807	-85.2	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7808	-85.22	oe	ccsbBroad304_06066	CTSL1	-			
7809	-85.27	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
7810	-85.31	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
7811	-85.43	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
7812	-85.46	kd	CGS001-2056	EPO	Endogenous ligands			
7813	-85.6	oe	ccsbBroad304_06888	RPN1	-			
7814	-85.6	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
7815	-85.61	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
7816	-85.63	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
7817	-85.64	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
7818	-85.67	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
7819	-85.71	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
7820	-85.71	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
7821	-85.77	kd	CGS001-2752	GLUL	-			
7822	-85.78	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
7823	-85.79	oe	ccsbBroad304_03980	DCLRE1B	-			
7824	-85.79	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
7825	-85.81	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
7826	-85.85	kd	CGS001-55907	CMAS	-			
7827	-85.88	kd	CGS001-6732	SRPK1	SRPK family			
7828	-85.92	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
7829	-85.93	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
7830	-85.95	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
7831	-86.01	cc		General transcription factors group 1 LOF	-			
7832	-86.01	kd	CGS001-3376	IARS	Aminoacyl tRNA synthetases / Class I			
7833	-86.03	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
7834	-86.04	oe	ccsbBroad304_01754	UCK2	-			
7835	-86.1	kd	CGS001-10472	ZNF238	-			
7836	-86.19	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
7837	-86.2	kd	CGS001-10198	MPHOSPH9	-			
7838	-86.21	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
7839	-86.25	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
7840	-86.26	kd	CGS001-167826	OLIG3	Basic helix-loop-helix proteins			
7841	-86.26	oe	ccsbBroad304_06574	MDH2	-			
7842	-86.3	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
7843	-86.34	oe	ccsbBroad304_00986	MCM2	-			
7844	-86.45	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
7845	-86.51	kd	CGS001-3569	IL6	Interferons			
7846	-86.53	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
7847	-86.54	kd	CGS001-4092	SMAD7	SMADs			
7848	-86.54	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
7849	-86.56	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
7850	-86.59	oe	ccsbBroad304_02576	MLLT11	-			
7851	-86.59	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
7852	-86.6	oe	ccsbBroad304_01413	RPA2	-			
7853	-86.66	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
7854	-86.66	kd	CGS001-9988	DMTF1	-			
7855	-86.67	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
7856	-86.68	oe	ccsbBroad304_04490	RSPH1	-			
7857	-86.73	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
7858	-86.75	cc		Phospholipases LOF	-			
7859	-86.75	kd	CGS001-9975	NR1D2	Rev-Erb receptors			
7860	-86.84	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
7861	-86.88	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
7862	-86.9	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
7863	-86.92	kd	CGS001-602	BCL3	Ankyrin repeat domain containing			
7864	-86.99	oe	ccsbBroad304_06648	CNOT3	-			
7865	-87.04	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
7866	-87.13	kd	CGS001-9774	BCLAF1	-			
7867	-87.15	kd	CGS001-5831	PYCR1	-			
7868	-87.18	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
7869	-87.19	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
7870	-87.2	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
7871	-87.2	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
7872	-87.21	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
7873	-87.22	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
7874	-87.25	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
7875	-87.25	kd	CGS001-79001	VKORC1	Oxidoreductases			
7876	-87.34	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
7877	-87.35	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
7878	-87.37	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
7879	-87.38	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
7880	-87.39	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
7881	-87.4	cp	BRD-A87387433	cefpodoxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7882	-87.44	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
7883	-87.47	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
7884	-87.53	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
7885	-87.53	kd	CGS001-10123	ARL4C	ADP-ribosylation factors			
7886	-87.57	oe	ccsbBroad304_02716	NMNAT2	-			
7887	-87.74	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
7888	-87.82	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
7889	-87.83	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
7890	-87.85	kd	CGS001-9061	PAPSS1	-			
7891	-87.86	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
7892	-87.87	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
7893	-87.88	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
7894	-87.88	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
7895	-87.88	kd	CGS001-3046	HBE1	-			
7896	-87.91	oe	ccsbBroad304_01374	RAP1A	-			
7897	-87.93	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
7898	-87.94	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
7899	-87.94	kd	CGS001-4709	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
7900	-88.03	kd	CGS001-27161	EIF2C2	-			
7901	-88.06	kd	CGS001-340371	NRBP2	NRBP family			
7902	-88.07	kd	CGS001-136	ADORA2B	GPCR / Class A : Adenosine receptors			
7903	-88.12	cp	BRD-A41450521	tosufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
7904	-88.14	kd	CGS001-5918	RARRES1	-			
7905	-88.29	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
7906	-88.3	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
7907	-88.31	oe	ccsbBroad304_09954	PTRF	-			
7908	-88.33	kd	CGS001-6647	SOD1	-			
7909	-88.34	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
7910	-88.41	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
7911	-88.43	kd	CGS001-5981	RFC1	ATPases / AAA-type			
7912	-88.52	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
7913	-88.53	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
7914	-88.55	kd	CGS001-26511	CHIC2	-			
7915	-88.56	oe	ccsbBroad304_00034	AES	-			
7916	-88.56	kd	CGS001-162655	ZNF519	Zinc fingers, C2H2-type			
7917	-88.59	oe	ccsbBroad304_02357	SSX3	-			
7918	-88.63	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
7919	-88.68	kd	CGS001-5563	PRKAA2	AMPK subfamily			
7920	-88.72	kd	CGS001-25825	BACE2	Pepsin			
7921	-88.74	oe	ccsbBroad304_00651	GNAI3	-			
7922	-88.75	oe	ccsbBroad304_06253	GALT	-			
7923	-88.75	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
7924	-88.76	kd	CGS001-55033	FKBP14	EF-hand domain containing			
7925	-88.77	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
7926	-88.79	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
7927	-88.8	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
7928	-88.82	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7929	-88.86	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
7930	-88.87	kd	CGS001-22883	CLSTN1	Cadherins / Cadherin-related			
7931	-88.9	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
7932	-88.91	kd	CGS001-8905	AP1S2	-			
7933	-88.96	kd	CGS001-4967	OGDH	-			
7934	-88.98	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
7935	-88.98	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
7936	-89	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
7937	-89.01	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7938	-89.02	kd	CGS001-3420	IDH3B	-			
7939	-89.17	kd	CGS001-60	ACTB	-			
7940	-89.19	oe	ccsbBroad304_01351	PEX19	-			
7941	-89.21	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
7942	-89.24	kd	CGS001-10557	RPP38	-			
7943	-89.26	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
7944	-89.27	kd	CGS001-375346	TMEM110	-			
7945	-89.29	kd	CGS001-84619	ZGPAT	G patch domain containing			
7946	-89.3	kd	CGS001-6251	RSU1	-			
7947	-89.3	oe	ccsbBroad304_02405	TFG	-			
7948	-89.3	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
7949	-89.35	oe	ccsbBroad304_05981	CDO1	-			
7950	-89.39	oe	ccsbBroad304_00725	HADHA	-			
7951	-89.4	kd	CGS001-6793	STK10	SLK subfamily			
7952	-89.43	oe	ccsbBroad304_00249	CD14	CD molecules			
7953	-89.45	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
7954	-89.45	kd	CGS001-64921	CASD1	-			
7955	-89.48	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
7956	-89.51	kd	CGS001-9200	PTPLA	-			
7957	-89.51	kd	CGS001-87	ACTN1	EF-hand domain containing			
7958	-89.58	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
7959	-89.64	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
7960	-89.65	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
7961	-89.67	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
7962	-89.72	kd	CGS001-8777	MPDZ	-			
7963	-89.79	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7964	-89.81	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
7965	-89.81	oe	ccsbBroad304_00810	HYAL1	-			
7966	-89.84	kd	CGS001-23549	DNPEP	Aminopeptidase I			
7967	-89.85	kd	CGS001-10962	MLLT11	-			
7968	-89.86	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
7969	-89.87	kd	CGS001-533	ATP6V0B	ATPases / V-type			
7970	-89.87	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
7971	-89.88	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
7972	-89.89	kd	CGS001-4782	NFIC	-			
7973	-89.89	oe	ccsbBroad304_07851	FAM120A	-			
7974	-89.96	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
7975	-90.01	kd	CGS001-330	BIRC3	Inhibitors of apoptosis (IAP) protein family			
7976	-90.02	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
7977	-90.04	kd	CGS001-10523	CHERP	G patch domain containing			
7978	-90.09	kd	CGS001-6203	RPS9	S ribosomal proteins			
7979	-90.16	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
7980	-90.18	oe	ccsbBroad304_01862	YEATS4	-			
7981	-90.2	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
7982	-90.22	kd	CGS001-55722	CEP72	-			
7983	-90.23	kd	CGS001-1843	DUSP1	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
7984	-90.23	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
7985	-90.25	oe	ccsbBroad304_00657	GNG4	-			
7986	-90.3	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
7987	-90.31	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
7988	-90.35	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
7989	-90.36	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
7990	-90.37	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
7991	-90.44	oe	ccsbBroad304_02092	SYNGR3	-			
7992	-90.5	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
7993	-90.51	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
7994	-90.55	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
7995	-90.56	cp	BRD-K51485625	ritonavir	HIV protease inhibitor		CYP3A4, CYP1A2, CYP2B6, CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
7996	-90.59	cp	BRD-K50938287	sumatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1A, HTR1F, HTR1E, HTR5A, HTR6, HTR7	Serotonin receptor agonist
7997	-90.6	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
7998	-90.62	kd	CGS001-5300	PIN1	-			
7999	-90.65	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
8000	-90.65	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
8001	-90.7	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
8002	-90.7	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
8003	-90.73	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
8004	-90.76	kd	CGS001-56922	MCCC1	-			
8005	-90.79	kd	CGS001-5450	POU2AF1	-			
8006	-90.85	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
8007	-90.91	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
8008	-90.98	kd	CGS001-6208	RPS14	S ribosomal proteins			
8009	-91.04	oe	ccsbBroad304_00060	AMBP	Lipocalins			
8010	-91.05	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
8011	-91.06	oe	ccsbBroad304_07889	QPRT	-			
8012	-91.06	oe	ccsbBroad304_00811	ICAM1	CD molecules			
8013	-91.07	kd	CGS001-4688	NCF2	Tetratricopeptide (TTC) repeat domain containing			
8014	-91.07	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
8015	-91.09	oe	ccsbBroad304_14020	SH3BP5	-			
8016	-91.09	kd	CGS001-9352	TXNL1	-			
8017	-91.09	kd	CGS001-1201	CLN3	-			
8018	-91.26	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
8019	-91.27	cp	BRD-A43082555	loxoprofen	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
8020	-91.27	oe	ccsbBroad304_07832	XPO7	Exportins			
8021	-91.27	oe	ccsbBroad304_07605	LYPLA1	-			
8022	-91.3	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
8023	-91.33	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
8024	-91.41	kd	CGS001-6309	SC5DL	-			
8025	-91.42	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
8026	-91.47	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
8027	-91.51	kd	CGS001-1390	CREM	basic leucine zipper proteins			
8028	-91.58	kd	CGS001-10398	MYL9	EF-hand domain containing			
8029	-91.6	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
8030	-91.64	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
8031	-91.67	kd	CGS001-6919	TCEA2	-			
8032	-91.69	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
8033	-91.84	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
8034	-91.86	kd	CGS001-5649	RELN	-			
8035	-91.87	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
8036	-91.9	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
8037	-91.9	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
8038	-91.91	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
8039	-91.94	kd	CGS001-9632	SEC24C	-			
8040	-91.95	cp	BRD-A09495397	bicuculline	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, KCNN1	GABA receptor antagonist
8041	-91.97	kd	CGS001-1453	CSNK1D	Casein kinase 1 (CK1) family			
8042	-92	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
8043	-92.04	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
8044	-92.05	kd	CGS001-4953	ODC1	Decarboxylases			
8045	-92.09	kd	CGS001-1949	EFNB3	Ephrins			
8046	-92.11	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
8047	-92.13	kd	CGS001-4811	NID1	-			
8048	-92.14	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
8049	-92.21	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
8050	-92.21	kd	CGS001-4616	GADD45B	-			
8051	-92.24	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
8052	-92.24	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
8053	-92.28	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
8054	-92.3	kd	CGS001-1312	COMT	Catecholamine turnover			
8055	-92.34	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
8056	-92.38	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
8057	-92.41	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
8058	-92.42	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
8059	-92.43	kd	CGS001-191	AHCY	Adenosine turnover			
8060	-92.46	kd	CGS001-23196	FAM120A	-			
8061	-92.49	cp	BRD-A01787639	naftopidil	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
8062	-92.51	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
8063	-92.56	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
8064	-92.57	kd	CGS001-23325	KIAA1033	-			
8065	-92.59	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
8066	-92.59	kd	CGS001-6272	SORT1	-			
8067	-92.64	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
8068	-92.7	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
8069	-92.76	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
8070	-92.78	oe	ccsbBroad304_03555	PANK4	-			
8071	-92.82	kd	CGS001-163486	DENND1B	DENN/MADD domain containing			
8072	-92.83	kd	CGS001-51014	TMED7	-			
8073	-92.85	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
8074	-92.85	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
8075	-92.85	oe	ccsbBroad304_05763	ACTB	-			
8076	-92.86	kd	CGS001-821	CANX	-			
8077	-92.88	oe	ccsbBroad304_01203	PIM1	PIM family			
8078	-92.9	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
8079	-92.9	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
8080	-92.93	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
8081	-92.99	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
8082	-93.02	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
8083	-93.03	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
8084	-93.03	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
8085	-93.1	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
8086	-93.11	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
8087	-93.14	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
8088	-93.19	oe	ccsbBroad304_03023	CRCP	-			
8089	-93.19	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
8090	-93.2	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
8091	-93.21	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
8092	-93.25	kd	CGS001-7750	ZMYM2	Zinc fingers, MYM type			
8093	-93.25	kd	CGS001-26574	AATF	-			
8094	-93.26	kd	CGS001-29946	SERTAD3	-			
8095	-93.31	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
8096	-93.36	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
8097	-93.38	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
8098	-93.38	oe	ccsbBroad304_01617	STX4	-			
8099	-93.44	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
8100	-93.49	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
8101	-93.52	oe	ccsbBroad304_09358	MAPK1IP1L	-			
8102	-93.54	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
8103	-93.57	kd	CGS001-55608	ANKRD10	Ankyrin repeat domain containing			
8104	-93.58	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
8105	-93.59	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
8106	-93.59	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
8107	-93.65	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
8108	-93.67	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
8109	-93.71	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
8110	-93.74	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
8111	-93.75	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
8112	-93.79	kd	CGS001-6199	RPS6KB2	p70 subfamily			
8113	-93.81	oe	ccsbBroad304_04752	IKBIP	-			
8114	-93.84	kd	CGS001-999	CDH1	CD molecules			
8115	-93.85	kd	CGS001-7314	UBB	-			
8116	-93.86	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
8117	-93.91	oe	ccsbBroad304_07888	CBX6	-			
8118	-93.93	oe	ccsbBroad304_00568	FHL2	-			
8119	-93.97	oe	ccsbBroad304_00518	ETFA	-			
8120	-93.99	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
8121	-94.05	kd	CGS001-51742	ARID4B	-			
8122	-94.1	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
8123	-94.1	oe	ccsbBroad304_00313	TBCB	-			
8124	-94.11	kd	CGS001-2621	GAS6	-			
8125	-94.11	kd	CGS001-8667	EIF3H	-			
8126	-94.12	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
8127	-94.12	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
8128	-94.14	kd	CGS001-2534	FYN	Src family			
8129	-94.15	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
8130	-94.16	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
8131	-94.2	kd	CGS001-9712	USP6NL	-			
8132	-94.21	kd	CGS001-51460	SFMBT1	Sterile alpha motif (SAM) domain containing			
8133	-94.23	kd	CGS001-2896	GRN	-			
8134	-94.25	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
8135	-94.25	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
8136	-94.25	kd	CGS001-6307	MSMO1	Fatty acid hydroxylase domain containing			
8137	-94.27	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
8138	-94.34	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
8139	-94.43	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
8140	-94.44	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
8141	-94.46	kd	CGS001-90655	TGIF2LY	Homeoboxes / TALE class			
8142	-94.48	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
8143	-94.5	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
8144	-94.52	kd	CGS001-11179	ZNF277	-			
8145	-94.54	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
8146	-94.58	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
8147	-94.61	kd	CGS001-11344	TWF2	Twinfilin subfamily			
8148	-94.62	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
8149	-94.62	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
8150	-94.64	kd	CGS001-3897	L1CAM	CD molecules			
8151	-94.7	kd	CGS001-11325	DDX42	DEAD-boxes			
8152	-94.72	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
8153	-94.77	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
8154	-94.79	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
8155	-94.8	kd	CGS001-23384	SPECC1L	-			
8156	-94.81	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
8157	-94.82	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
8158	-94.84	kd	CGS001-5188	PET112	-			
8159	-94.84	kd	CGS001-4297	MLL	-			
8160	-94.89	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
8161	-94.89	kd	CGS001-2944	GSTM1	Glutathione S-transferases / Soluble			
8162	-94.89	kd	CGS001-10672	GNA13	-			
8163	-94.92	kd	CGS001-113878	DTX2	RING-type (C3HC4) zinc fingers			
8164	-94.92	oe	ccsbBroad304_01716	TSN	-			
8165	-94.96	kd	CGS001-1497	CTNS	-			
8166	-94.98	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
8167	-95	kd	CGS001-55781	RIOK2	RIO2 subfamily			
8168	-95	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
8169	-95.03	kd	CGS001-10745	PHTF1	-			
8170	-95.04	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
8171	-95.05	oe	ccsbBroad304_02533	NOXA1	-			
8172	-95.07	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
8173	-95.07	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
8174	-95.08	kd	CGS001-3428	IFI16	-			
8175	-95.1	kd	CGS001-93349	SP140L	Zinc fingers, PHD-type			
8176	-95.16	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
8177	-95.17	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
8178	-95.17	kd	CGS001-29775	CARD10	-			
8179	-95.19	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
8180	-95.22	kd	CGS001-5096	PCCB	Carboxylases			
8181	-95.22	kd	CGS001-2130	EWSR1	RNA binding motif (RRM) containing			
8182	-95.26	kd	CGS001-2524	FUT2	Fucosyltransferases			
8183	-95.28	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
8184	-95.29	kd	CGS001-57018	CCNL1	-			
8185	-95.32	kd	CGS001-2617	GARS	Aminoacyl tRNA synthetases / Class II			
8186	-95.38	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
8187	-95.39	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
8188	-95.41	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
8189	-95.43	kd	CGS001-4795	NFKBIL1	-			
8190	-95.43	kd	CGS001-85027	C5ORF62	-			
8191	-95.44	kd	CGS001-10776	ARPP19	-			
8192	-95.49	kd	CGS001-5810	RAD1	-			
8193	-95.54	cc		Baculoviral IAP repeat domain containing LOF	-			
8194	-95.56	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
8195	-95.62	kd	CGS001-1611	DAP	-			
8196	-95.63	kd	CGS001-538	ATP7A	ATPases / P-type			
8197	-95.66	oe	ccsbBroad304_01974	RNASET2	-			
8198	-95.69	kd	CGS001-2197	FAU	S ribosomal proteins			
8199	-95.7	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
8200	-95.7	kd	CGS001-55008	HERC6	-			
8201	-95.71	kd	CGS001-66008	TRAK2	-			
8202	-95.74	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
8203	-95.74	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
8204	-95.79	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
8205	-95.81	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
8206	-95.81	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
8207	-95.82	oe	ccsbBroad304_02368	TIMM17B	-			
8208	-95.83	kd	CGS001-51805	COQ3	-			
8209	-95.87	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
8210	-95.88	kd	CGS001-8140	SLC7A5	SLC7 family			
8211	-95.88	oe	ccsbBroad304_06464	ITGB2	Integrins			
8212	-95.89	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
8213	-95.93	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
8214	-95.95	kd	CGS001-23242	COBL	-			
8215	-96	kd	CGS001-51375	SNX7	Sorting nexins			
8216	-96.01	cp	BRD-K59753975	vindesine	Tubulin inhibitor		TUBB, TUBB1	Tubulin inhibitor
8217	-96.06	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
8218	-96.06	kd	CGS001-151306	GPBAR1	Bile acid receptor			
8219	-96.07	oe	ccsbBroad304_09881	RFX6	-			
8220	-96.11	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
8221	-96.16	cc		Kruppel like transcription factors LOF	-			
8222	-96.18	oe	ccsbBroad304_02864	PRDX5	-			
8223	-96.19	kd	CGS001-6275	S100A4	EF-hand domain containing			
8224	-96.19	kd	CGS001-143	PARP4	Poly (ADP-ribose) polymerases			
8225	-96.19	kd	CGS001-1977	EIF4E	Translation Initiation Factor 4E			
8226	-96.21	kd	CGS001-9870	KIAA0317	-			
8227	-96.21	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
8228	-96.23	kd	CGS001-55422	ZNF331	Zinc fingers, C2H2-type			
8229	-96.24	kd	CGS001-51335	NGRN	-			
8230	-96.27	kd	CGS001-1727	CYB5R3	-			
8231	-96.28	oe	ccsbBroad304_00817	IDH2	-			
8232	-96.28	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
8233	-96.35	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
8234	-96.35	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
8235	-96.36	kd	CGS001-5371	PML	RING-type (C3HC4) zinc fingers			
8236	-96.39	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
8237	-96.39	kd	CGS001-5433	POLR2D	RNA polymerase subunits			
8238	-96.39	kd	CGS001-55038	CDCA4	-			
8239	-96.44	oe	ccsbBroad304_01483	SAT1	-			
8240	-96.46	kd	CGS001-10933	MORF4L1	-			
8241	-96.5	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
8242	-96.51	kd	CGS001-55765	C1ORF106	-			
8243	-96.52	kd	CGS001-1728	NQO1	-			
8244	-96.53	kd	CGS001-24148	PRPF6	-			
8245	-96.54	kd	CGS001-3017	HIST1H2BD	Histones / Replication-dependent			
8246	-96.55	kd	CGS001-7270	TTF1	-			
8247	-96.56	oe	ccsbBroad304_00100	RHOA	-			
8248	-96.56	kd	CGS001-6813	STXBP2	-			
8249	-96.57	kd	CGS001-23581	CASP14	Caspases			
8250	-96.57	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
8251	-96.65	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
8252	-96.68	cc		EIF Proteins LOF	-			
8253	-96.69	kd	CGS001-79862	ZNF669	Zinc fingers, C2H2-type			
8254	-96.73	kd	CGS001-6643	SNX2	Sorting nexins			
8255	-96.74	oe	ccsbBroad304_03917	RBKS	-			
8256	-96.74	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
8257	-96.76	kd	CGS001-5699	PSMB10	Proteasome (prosome, macropain) subunits			
8258	-96.77	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
8259	-96.77	kd	CGS001-4046	LSP1	-			
8260	-96.79	kd	CGS001-1975	EIF4B	RNA binding motif (RRM) containing			
8261	-96.8	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
8262	-96.81	oe	ccsbBroad304_00418	CD55	CD molecules			
8263	-96.86	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
8264	-96.88	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
8265	-96.9	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
8266	-96.91	kd	CGS001-391013	PLA2G2C	-			
8267	-96.92	cc		RNA Polymerase Enzymes LOF	-			
8268	-96.92	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
8269	-96.93	kd	CGS001-7031	TFF1	-			
8270	-96.94	kd	CGS001-6676	SPAG4	-			
8271	-96.96	kd	CGS001-84547	PGBD1	-			
8272	-96.97	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
8273	-96.97	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
8274	-97.01	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
8275	-97.02	cp	BRD-K56614220	clofazimine	GK0582 inhibitor			GK0582 inhibitor
8276	-97.04	oe	ccsbBroad304_06136	ECHS1	-			
8277	-97.09	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
8278	-97.09	kd	CGS001-6812	STXBP1	-			
8279	-97.09	kd	CGS001-10447	FAM3C	-			
8280	-97.11	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
8281	-97.14	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
8282	-97.15	kd	CGS001-3988	LIPA	-			
8283	-97.16	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
8284	-97.18	oe	ccsbBroad304_01951	BLZF1	-			
8285	-97.18	kd	CGS001-51282	SCAND1	-			
8286	-97.18	kd	CGS001-10755	GIPC1	-			
8287	-97.2	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
8288	-97.23	kd	CGS001-1452	CSNK1A1	Casein kinase 1 (CK1) family			
8289	-97.28	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
8290	-97.29	kd	CGS001-5080	PAX6	Paired boxes			
8291	-97.32	kd	CGS001-5932	RBBP8	-			
8292	-97.33	oe	ccsbBroad304_06159	CTTN	-			
8293	-97.34	kd	CGS001-1831	TSC22D3	-			
8294	-97.35	kd	CGS001-6188	RPS3	S ribosomal proteins			
8295	-97.36	oe	ccsbBroad304_02604	B3GNT1	-			
8296	-97.37	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
8297	-97.42	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
8298	-97.44	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
8299	-97.44	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
8300	-97.45	kd	CGS001-955	ENTPD6	-			
8301	-97.46	kd	CGS001-6944	VPS72	-			
8302	-97.5	kd	CGS001-122618	PLD4	-			
8303	-97.5	kd	CGS001-5771	PTPN2	Protein tyrosine phosphatases			
8304	-97.53	kd	CGS001-5511	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
8305	-97.61	kd	CGS001-5578	PRKCA	Delta subfamily			
8306	-97.68	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
8307	-97.71	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
8308	-97.71	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
8309	-97.72	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
8310	-97.72	kd	CGS001-50865	HEBP1	Endogenous ligands			
8311	-97.73	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
8312	-97.78	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
8313	-97.79	kd	CGS001-55793	FAM63A	-			
8314	-97.83	kd	CGS001-80150	ASRGL1	-			
8315	-97.84	kd	CGS001-8295	TRRAP	TRRAP subfamily			
8316	-97.84	kd	CGS001-60528	ELAC2	-			
8317	-97.85	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
8318	-97.85	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
8319	-97.87	oe	ccsbBroad304_14047	TACC3	-			
8320	-97.88	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
8321	-97.88	oe	ccsbBroad304_01394	RFX4	-			
8322	-97.89	kd	CGS001-6455	SH3GL1	-			
8323	-97.92	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
8324	-97.93	kd	CGS001-944	TNFSF8	CD molecules			
8325	-97.96	kd	CGS001-118442	GPR62	GPCR / Class A : Orphans			
8326	-98	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
8327	-98.01	oe	ccsbBroad304_07101	TSC2	-			
8328	-98.01	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
8329	-98.01	cp	BRD-K66206289	lobeline	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist
8330	-98.01	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
8331	-98.02	kd	CGS001-7728	ZNF175	Zinc fingers, C2H2-type			
8332	-98.03	kd	CGS001-5781	PTPN11	Protein tyrosine phosphatases			
8333	-98.06	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
8334	-98.06	kd	CGS001-648	BMI1	Polycomb group ring fingers			
8335	-98.07	kd	CGS001-3934	LCN2	Lipocalins			
8336	-98.09	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
8337	-98.11	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
8338	-98.13	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
8339	-98.13	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
8340	-98.13	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
8341	-98.14	oe	ccsbBroad304_02955	MYCBP	-			
8342	-98.14	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
8343	-98.15	kd	CGS001-9467	SH3BP5	-			
8344	-98.17	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
8345	-98.18	kd	CGS001-3421	IDH3G	-			
8346	-98.2	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
8347	-98.21	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
8348	-98.21	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
8349	-98.24	kd	CGS001-2542	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
8350	-98.24	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
8351	-98.26	kd	CGS001-4016	LOXL1	-			
8352	-98.28	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
8353	-98.29	kd	CGS001-1595	CYP51A1	Cytochrome P450s			
8354	-98.31	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
8355	-98.31	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
8356	-98.33	kd	CGS001-11333	PDAP1	-			
8357	-98.38	oe	ccsbBroad304_02419	NDRG1	-			
8358	-98.39	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
8359	-98.41	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
8360	-98.42	kd	CGS001-23077	MYCBP2	-			
8361	-98.42	oe	ccsbBroad304_00053	ALDOA	-			
8362	-98.45	kd	CGS001-5813	PURA	-			
8363	-98.45	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
8364	-98.46	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
8365	-98.47	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
8366	-98.47	kd	CGS001-9344	TAOK2	TAO subfamily			
8367	-98.5	oe	ccsbBroad304_02592	KIF2C	Kinesins			
8368	-98.52	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
8369	-98.52	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
8370	-98.53	kd	CGS001-2194	FASN	Short chain dehydrogenase/reductase superfamily / Atypical members			
8371	-98.55	kd	CGS001-27097	TAF5L	WD repeat domain containing			
8372	-98.56	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
8373	-98.56	oe	ccsbBroad304_07651	HEXIM1	-			
8374	-98.61	kd	CGS001-8508	NIPSNAP1	-			
8375	-98.61	kd	CGS001-51293	CD320	CD molecules			
8376	-98.61	oe	ccsbBroad304_05948	CCND2	-			
8377	-98.63	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
8378	-98.63	kd	CGS001-6767	ST13	Tetratricopeptide (TTC) repeat domain containing			
8379	-98.64	kd	CGS001-7466	WFS1	-			
8380	-98.65	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
8381	-98.7	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
8382	-98.71	kd	CGS001-10325	RRAGB	-			
8383	-98.71	kd	CGS001-4717	NDUFC1	Mitochondrial respiratory chain complex / Complex I			
8384	-98.71	kd	CGS001-93185	IGSF8	CD molecules			
8385	-98.72	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
8386	-98.74	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
8387	-98.76	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
8388	-98.76	kd	CGS001-134288	TMEM174	-			
8389	-98.78	kd	CGS001-22944	KIN	-			
8390	-98.79	kd	CGS001-466	ATF1	basic leucine zipper proteins			
8391	-98.84	kd	CGS001-51447	IP6K2	-			
8392	-98.85	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
8393	-98.86	kd	CGS001-23142	DCUN1D4	-			
8394	-98.87	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
8395	-98.87	kd	CGS001-89910	UBE3B	-			
8396	-98.89	oe	ccsbBroad304_01174	PEX13	-			
8397	-98.89	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
8398	-98.91	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
8399	-98.94	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
8400	-98.95	kd	CGS001-25987	TSKU	-			
8401	-98.95	kd	CGS001-8986	RPS6KA4	MSK subfamily			
8402	-98.96	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
8403	-98.98	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
8404	-98.98	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
8405	-99.03	kd	CGS001-2859	GPR35	GPCR / Class A : Orphans			
8406	-99.03	kd	CGS001-8891	EIF2B3	-			
8407	-99.03	kd	CGS001-1738	DLD	-			
8408	-99.03	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
8409	-99.04	kd	CGS001-54925	ZNF434	-			
8410	-99.05	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
8411	-99.05	kd	CGS001-5063	PAK3	PAKA subfamily			
8412	-99.05	kd	CGS001-2849	GPR26	GPCR / Class A : Orphans			
8413	-99.06	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
8414	-99.08	oe	ccsbBroad304_06862	RGS3	-			
8415	-99.08	kd	CGS001-5546	PRCC	-			
8416	-99.09	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
8417	-99.11	kd	CGS001-27076	LYPD3	-			
8418	-99.13	kd	CGS001-23338	PHF15	-			
8419	-99.15	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
8420	-99.15	kd	CGS001-6799	SULT1A2	Sulfotransferases, cytosolic			
8421	-99.17	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
8422	-99.17	oe	ccsbBroad304_02674	STK38	NDR family			
8423	-99.18	kd	CGS001-7297	TYK2	Janus kinase (JakA) family			
8424	-99.18	kd	CGS001-3033	HADH	-			
8425	-99.18	kd	CGS001-2969	GTF2I	General transcription factors			
8426	-99.19	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
8427	-99.21	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
8428	-99.21	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
8429	-99.26	kd	CGS001-6146	RPL22	L ribosomal proteins			
8430	-99.3	cp	BRD-M41783010	acamprosate	Glutamate receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B, GRM5	Glutamate receptor antagonist
8431	-99.3	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
8432	-99.3	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
8433	-99.31	oe	ccsbBroad304_00600	FYN	Src family			
8434	-99.32	kd	CGS001-4125	MAN2B1	-			
8435	-99.33	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
8436	-99.34	kd	CGS001-5351	PLOD1	-			
8437	-99.34	kd	CGS001-2114	ETS2	ETS Transcription Factors			
8438	-99.35	oe	ccsbBroad304_00020	ACY1	-			
8439	-99.37	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
8440	-99.37	kd	CGS001-23223	RRP12	-			
8441	-99.39	kd	CGS001-10190	TXNDC9	-			
8442	-99.4	oe	ccsbBroad304_05183	TXLNA	-			
8443	-99.4	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
8444	-99.4	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
8445	-99.45	kd	CGS001-1487	CTBP1	-			
8446	-99.45	kd	CGS001-5049	PAFAH1B2	-			
8447	-99.45	kd	CGS001-4234	METTL1	-			
8448	-99.47	kd	CGS001-5970	RELA	NFkappaB transcription factor family			
8449	-99.47	kd	CGS001-2580	GAK	Heat shock proteins / DNAJ (HSP40)			
8450	-99.47	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
8451	-99.48	kd	CGS001-23585	TMEM50A	-			
8452	-99.49	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
8453	-99.5	kd	CGS001-1650	DDOST	-			
8454	-99.51	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
8455	-99.53	kd	CGS001-10245	TIMM17B	-			
8456	-99.53	kd	CGS001-4204	MECP2	-			
8457	-99.54	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
8458	-99.54	oe	ccsbBroad304_08888	ACD	-			
8459	-99.55	kd	CGS001-4547	MTTP	-			
8460	-99.56	kd	CGS001-3663	IRF5	-			
8461	-99.58	kd	CGS001-51311	TLR8	Toll-like receptor family			
8462	-99.58	kd	CGS001-2597	GAPDH	-			
8463	-99.59	kd	CGS001-51701	NLK	nmo subfamily			
8464	-99.6	kd	CGS001-2958	GTF2A2	General transcription factors			
8465	-99.61	kd	CGS001-6632	SNRPD1	-			
8466	-99.61	kd	CGS001-9140	ATG12	-			
8467	-99.63	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
8468	-99.66	kd	CGS001-6886	TAL1	Basic helix-loop-helix proteins			
8469	-99.66	kd	CGS001-6741	SSB	La ribonucleoprotein domain containing			
8470	-99.66	kd	CGS001-2677	GGCX	Carboxylases			
8471	-99.68	oe	ccsbBroad304_01663	TFF2	-			
8472	-99.68	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
8473	-99.68	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
8474	-99.72	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
8475	-99.72	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
8476	-99.72	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
8477	-99.72	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
8478	-99.74	kd	CGS001-6391	SDHC	Mitochondrial respiratory chain complex / Complex II			
8479	-99.76	kd	CGS001-10652	YKT6	-			
8480	-99.76	kd	CGS001-51002	TPRKB	-			
8481	-99.76	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
8482	-99.77	oe	ccsbBroad304_09821	TMEM154	-			
8483	-99.77	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
8484	-99.79	kd	CGS001-57822	GRHL3	-			
8485	-99.79	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
8486	-99.79	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
8487	-99.79	kd	CGS001-5422	POLA1	DNA polymerases			
8488	-99.81	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
8489	-99.82	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
8490	-99.82	kd	CGS001-6599	SMARCC1	-			
8491	-99.82	kd	CGS001-9805	SCRN1	-			
8492	-99.82	kd	CGS001-6129	RPL7	L ribosomal proteins			
8493	-99.82	kd	CGS001-5480	PPIC	-			
8494	-99.82	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
8495	-99.82	kd	CGS001-5315	PKM2	-			
8496	-99.82	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
8497	-99.82	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
8498	-99.84	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
8499	-99.84	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
8500	-99.86	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
8501	-99.86	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
8502	-99.87	kd	CGS001-7128	TNFAIP3	OTU domain containing			
8503	-99.87	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
8504	-99.87	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
8505	-99.87	kd	CGS001-2067	ERCC1	-			
8506	-99.87	kd	CGS001-56998	CTNNBIP1	Catenins			
8507	-99.87	kd	CGS001-23365	ARHGEF12	Rho guanine nucleotide exchange factors			
8508	-99.89	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
8509	-99.89	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
8510	-99.89	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
8511	-99.89	kd	CGS001-55111	PLEKHJ1	Pleckstrin homology (PH) domain containing			
8512	-99.89	kd	CGS001-3909	LAMA3	Laminins			
8513	-99.89	kd	CGS001-221393	GPR115	Adhesion Class GPCRs			
8514	-99.89	kd	CGS001-960	CD44	CD molecules			
8515	-99.89	kd	CGS001-883	CCBL1	Hydrogen sulphide synthesis			
8516	-99.89	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
8517	-99.91	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
8518	-99.91	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
8519	-99.91	oe	ccsbBroad304_00237	CCND3	-			
8520	-99.92	kd	CGS001-26520	TIMM9	-			
8521	-99.92	kd	CGS001-6883	TAF12	-			
8522	-99.92	kd	CGS001-51128	SAR1B	-			
8523	-99.92	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
8524	-99.92	kd	CGS001-10113	PREB	WD repeat domain containing			
8525	-99.92	kd	CGS001-50814	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
8526	-99.92	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
8527	-99.92	kd	CGS001-2059	EPS8	-			
8528	-99.92	kd	CGS001-8824	CES2	Carboxylesterases			
8529	-99.92	kd	CGS001-10904	BLCAP	-			
8530	-99.92	kd	CGS001-23461	ABCA5	ATP binding cassette transporters / subfamily A			
8531	-99.93	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
8532	-99.93	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
8533	-99.95	kd	CGS001-147948	ZNF582	Zinc fingers, C2H2-type			
8534	-99.95	kd	CGS001-11180	WDR6	WD repeat domain containing			
8535	-99.95	kd	CGS001-8717	TRADD	-			
8536	-99.95	kd	CGS001-7157	TP53	-			
8537	-99.95	kd	CGS001-6894	TARBP1	-			
8538	-99.95	kd	CGS001-6777	STAT5B	SH2 domain containing			
8539	-99.95	kd	CGS001-6429	SRSF4	RNA binding motif (RRM) containing			
8540	-99.95	kd	CGS001-6670	SP3	Specificity protein transcription factors			
8541	-99.95	kd	CGS001-6478	SIAH2	-			
8542	-99.95	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
8543	-99.95	kd	CGS001-5930	RBBP6	-			
8544	-99.95	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
8545	-99.95	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
8546	-99.95	kd	CGS001-55872	PBK	TOPK family			
8547	-99.95	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
8548	-99.95	kd	CGS001-4771	NF2	A-kinase anchor proteins			
8549	-99.95	kd	CGS001-3312	HSPA8	Heat shock proteins / HSP70			
8550	-99.95	kd	CGS001-2952	GSTT1	Glutathione S-transferases / Soluble			
8551	-99.95	kd	CGS001-50943	FOXP3	Forkhead boxes			
8552	-99.95	kd	CGS001-2264	FGFR4	Type V RTKs: FGF (fibroblast growth factor) receptor family			
8553	-99.95	kd	CGS001-9637	FEZ2	-			
8554	-99.95	kd	CGS001-125965	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
8555	-99.95	kd	CGS001-894	CCND2	-			
8556	-99.95	kd	CGS001-154	ADRB2	GPCR / Class A : Adrenoceptors : beta			
8557	-99.95	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
8558	-99.98	cc		X linked mental retardation group 1 LOF	-			
8559	-100	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
