Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
2	100	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
3	100	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
4	100	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
5	100	kd	CGS001-7727	ZNF174	Zinc fingers, C2H2-type			
6	100	kd	CGS001-9958	USP15	Ubiquitin-specific peptidases			
7	100	kd	CGS001-9319	TRIP13	ATPases / AAA-type			
8	100	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
9	100	kd	CGS001-6434	TRA2B	RNA binding motif (RRM) containing			
10	100	kd	CGS001-8463	TEAD2	-			
11	100	kd	CGS001-6832	SUPV3L1	-			
12	100	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
13	100	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
14	100	kd	CGS001-10921	RNPS1	RNA binding motif (RRM) containing			
15	100	kd	CGS001-57665	RDH14	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
16	100	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
17	100	kd	CGS001-94103	ORMDL3	-			
18	100	kd	CGS001-55577	NAGK	-			
19	100	kd	CGS001-26292	MYCBP	-			
20	100	kd	CGS001-9961	MVP	-			
21	100	kd	CGS001-10651	MTX2	-			
22	100	kd	CGS001-29079	MED4	-			
23	100	kd	CGS001-221895	JAZF1	Zinc fingers, C2H2-type			
24	100	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
25	100	kd	CGS001-2957	GTF2A1	General transcription factors			
26	100	kd	CGS001-83743	GRWD1	WD repeat domain containing			
27	100	kd	CGS001-2786	GNG4	-			
28	100	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
29	100	kd	CGS001-55500	ETNK1	-			
30	100	kd	CGS001-2109	ETFB	-			
31	100	kd	CGS001-57396	CLK4	CDC-like kinases			
32	100	kd	CGS001-929	CD14	CD molecules			
33	100	kd	CGS001-6046	BRD2	Bromodomain kinase (BRDK) family			
34	100	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
35	100	kd	CGS001-369	ARAF	RAF family			
36	100	kd	CGS001-7915	ALDH5A1	Aldehyde dehydrogenases			
37	100	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
38	99.98	kd	CGS001-171017	ZNF384	Zinc fingers, C2H2-type			
39	99.98	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
40	99.98	kd	CGS001-11073	TOPBP1	-			
41	99.98	kd	CGS001-11198	SUPT16H	-			
42	99.98	kd	CGS001-9709	HERPUD1	-			
43	99.98	kd	CGS001-665	BNIP3L	-			
44	99.96	cc		General transcription factors group 2 LOF	-			
45	99.96	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
46	99.96	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
47	99.96	oe	ccsbBroad304_08322	UFM1	-			
48	99.96	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
49	99.96	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
50	99.96	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
51	99.96	oe	ccsbBroad304_07374	PTPLA	-			
52	99.96	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
53	99.96	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
54	99.96	oe	ccsbBroad304_00880	IRF2	-			
55	99.96	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
56	99.96	oe	ccsbBroad304_00832	IFNB1	Interferons			
57	99.96	oe	ccsbBroad304_00620	GCDH	-			
58	99.96	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
59	99.96	oe	ccsbBroad304_00509	EPHX1	-			
60	99.96	oe	ccsbBroad304_06134	ECH1	-			
61	99.96	oe	ccsbBroad304_03641	ASF1B	-			
62	99.96	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
63	99.96	cp	BRD-K50866992	tropisetron	Serotonin receptor antagonist		HTR3A, GLRA1, GLRA2, GLRB, HTR4	Serotonin receptor antagonist
64	99.96	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
65	99.96	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
66	99.96	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
67	99.96	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
68	99.96	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
69	99.96	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
70	99.96	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
71	99.96	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
72	99.96	kd	CGS001-7090	TLE3	WD repeat domain containing			
73	99.96	kd	CGS001-9014	TAF1B	-			
74	99.96	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
75	99.96	kd	CGS001-2230	FDX1	-			
76	99.96	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
77	99.96	kd	CGS001-2149	F2R	Protease activated receptors			
78	99.96	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
79	99.96	kd	CGS001-10632	ATP5L	ATPases / F-type			
80	99.96	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
81	99.96	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
82	99.94	kd	CGS001-1022	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
83	99.93	oe	ccsbBroad304_02576	MLLT11	-			
84	99.93	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
85	99.93	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
86	99.93	oe	ccsbBroad304_00118	ATIC	-			
87	99.93	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
88	99.93	cp	BRD-K33226500	indinavir	HIV protease inhibitor		CYP3A5	HIV protease inhibitor
89	99.93	cp	BRD-A94543220	bifonazole	Sterol demethylase inhibitor		CYP2B6	Sterol demethylase inhibitor
90	99.93	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
91	99.93	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
92	99.93	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
93	99.93	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
94	99.93	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
95	99.93	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
96	99.93	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
97	99.93	kd	CGS001-80135	RPF1	-			
98	99.93	kd	CGS001-5693	PSMB5	Proteasome subunits			
99	99.93	kd	CGS001-9412	MED21	-			
100	99.93	kd	CGS001-1843	DUSP1	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
101	99.93	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
102	99.93	kd	CGS001-10554	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
103	99.93	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
104	99.91	cc		Proteasome Pathway LOF	-			
105	99.91	cc		Thymidylate synthase inhibitor	-			
106	99.91	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
107	99.91	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
108	99.91	kd	CGS001-9925	ZBTB5	BTB/POZ domain containing			
109	99.91	kd	CGS001-7477	WNT7B	Endogenous ligands			
110	99.91	kd	CGS001-7292	TNFSF4	CD molecules			
111	99.91	kd	CGS001-5915	RARB	Retinoic acid receptors			
112	99.91	kd	CGS001-154197	PNLDC1	-			
113	99.91	kd	CGS001-4947	OAZ2	-			
114	99.91	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
115	99.91	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
116	99.91	kd	CGS001-2168	FABP1	Fatty acid-binding proteins			
117	99.89	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
118	99.89	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
119	99.89	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
120	99.89	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
121	99.89	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
122	99.89	kd	CGS001-8527	DGKD	Pleckstrin homology (PH) domain containing			
123	99.89	kd	CGS001-7263	TST	-			
124	99.89	kd	CGS001-9221	NOLC1	-			
125	99.89	kd	CGS001-4594	MUT	-			
126	99.89	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
127	99.89	kd	CGS001-10014	HDAC5	Histone deacetylases			
128	99.89	kd	CGS001-11151	CORO1A	Coronins			
129	99.89	kd	CGS001-701	BUB1B	Bub family			
130	99.89	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
131	99.87	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
132	99.87	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
133	99.87	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
134	99.87	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
135	99.87	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
136	99.87	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
137	99.87	kd	CGS001-29984	RHOD	-			
138	99.87	kd	CGS001-7025	NR2F1	COUP-TF-like receptors			
139	99.87	kd	CGS001-7181	NR2C1	Testicular receptors			
140	99.87	kd	CGS001-545	ATR	ATR subfamily			
141	99.87	kd	CGS001-50808	AK3	-			
142	99.87	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
143	99.85	cc		Tumor necrosis factor superfamily LOF	-			
144	99.85	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
145	99.85	oe	ccsbBroad304_03182	GLOD4	-			
146	99.85	oe	ccsbBroad304_02501	DCTN6	-			
147	99.85	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
148	99.85	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
149	99.85	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
150	99.85	kd	CGS001-10617	STAMBP	-			
151	99.85	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
152	99.85	kd	CGS001-4700	NDUFA6	LYR motif containing			
153	99.85	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
154	99.85	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
155	99.85	kd	CGS001-2264	FGFR4	Type V RTKs: FGF (fibroblast growth factor) receptor family			
156	99.85	kd	CGS001-1906	EDN1	Endogenous ligands			
157	99.85	kd	CGS001-403	ARL3	ADP-ribosylation factors			
158	99.82	oe	ccsbBroad304_04465	RERG	-			
159	99.82	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
160	99.82	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
161	99.82	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
162	99.82	kd	CGS001-7001	PRDX2	-			
163	99.82	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
164	99.82	kd	CGS001-2872	MKNK2	MKN subfamily			
165	99.82	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
166	99.8	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
167	99.8	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
168	99.8	kd	CGS001-4172	MCM3	-			
169	99.8	kd	CGS001-3909	LAMA3	Laminins			
170	99.8	kd	CGS001-9455	HOMER2	-			
171	99.8	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
172	99.78	oe	ccsbBroad304_00833	IFNG	Interferons			
173	99.78	kd	CGS001-22954	TRIM32	-			
174	99.78	kd	CGS001-8650	NUMB	-			
175	99.78	kd	CGS001-5595	MAPK3	MAPK:ERK subfamily			
176	99.78	kd	CGS001-4299	AFF1	-			
177	99.76	oe	ccsbBroad304_03072	GTPBP8	-			
178	99.76	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
179	99.76	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
180	99.76	kd	CGS001-118738	ZNF488	Zinc fingers, C2H2-type			
181	99.76	kd	CGS001-399664	MEX3D	Mex-3 homologs			
182	99.76	kd	CGS001-2806	GOT2	-			
183	99.76	kd	CGS001-4680	CEACAM6	CD molecules			
184	99.76	kd	CGS001-9451	EIF2AK3	PEK subfamily			
185	99.74	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
186	99.74	oe	ccsbBroad304_01624	SUPV3L1	-			
187	99.74	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
188	99.74	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
189	99.74	kd	CGS001-5682	PSMA1	Proteasome subunits			
190	99.74	kd	CGS001-9943	OXSR1	FRAY subfamily			
191	99.74	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
192	99.73	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
193	99.72	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
194	99.72	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
195	99.72	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
196	99.72	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
197	99.72	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
198	99.72	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
199	99.72	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
200	99.72	kd	CGS001-2023	ENO1	-			
201	99.7	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
202	99.7	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
203	99.69	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
204	99.69	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
205	99.69	kd	CGS001-6678	SPARC	-			
206	99.69	kd	CGS001-5018	OXA1L	-			
207	99.69	kd	CGS001-3596	IL13	Interleukins and interleukin receptors			
208	99.69	kd	CGS001-8780	RIOK3	RIO3 subfamily			
209	99.67	cc		IMPDH inhibitor	-			
210	99.67	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
211	99.67	kd	CGS001-5618	PRLR	Prolactin receptor family			
212	99.67	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
213	99.67	kd	CGS001-629	CFB	Complement system			
214	99.67	kd	CGS001-345	APOC3	Apolipoproteins			
215	99.65	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
216	99.65	kd	CGS001-8681	JMJD7-PLA2G4B	-			
217	99.64	oe	ccsbBroad304_03878	SENP2	-			
218	99.63	oe	ccsbBroad304_10431	HADHB	-			
219	99.63	kd	CGS001-7013	TERF1	-			
220	99.63	kd	CGS001-8467	SMARCA5	-			
221	99.63	kd	CGS001-3155	HMGCL	-			
222	99.63	kd	CGS001-55165	CEP55	-			
223	99.61	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
224	99.61	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
225	99.61	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
226	99.61	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
227	99.61	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
228	99.61	kd	CGS001-51001	MTERFD1	-			
229	99.61	kd	CGS001-23588	KLHDC2	-			
230	99.59	kd	CGS001-2145	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
231	99.58	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
232	99.58	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
233	99.58	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
234	99.56	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
235	99.56	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
236	99.56	oe	ccsbBroad304_03951	NARFL	-			
237	99.54	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
238	99.54	cp	BRD-K62374253	rufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
239	99.54	cp	BRD-K37798499	etoposide	Topoisomerase inhibitor		TOP2A, CYP2E1, CYP3A5, TOP2B	Topoisomerase inhibitor
240	99.54	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
241	99.54	kd	CGS001-79094	CHAC1	-			
242	99.54	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
243	99.53	oe	ccsbBroad304_02838	SDF2L1	-			
244	99.52	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
245	99.52	kd	CGS001-7105	TSPAN6	Tetraspanins			
246	99.52	kd	CGS001-5707	PSMD1	Proteasome subunits			
247	99.52	kd	CGS001-1493	CTLA4	CD molecules			
248	99.51	cc		Kruppel like transcription factors LOF	-			
249	99.5	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
250	99.5	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
251	99.5	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
252	99.5	kd	CGS001-3717	JAK2	Janus kinase (JakA) family			
253	99.5	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
254	99.47	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
255	99.47	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
256	99.47	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
257	99.47	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
258	99.45	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
259	99.45	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
260	99.45	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
261	99.43	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
262	99.43	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
263	99.42	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
264	99.41	kd	CGS001-8649	LAMTOR3	-			
265	99.41	kd	CGS001-2295	FOXF2	Forkhead boxes			
266	99.39	cp	BRD-K66206289	lobeline	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist
267	99.39	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
268	99.39	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
269	99.39	kd	CGS001-4927	NUP88	-			
270	99.37	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
271	99.37	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
272	99.37	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
273	99.37	kd	CGS001-253260	RICTOR	-			
274	99.37	kd	CGS001-822	CAPG	-			
275	99.35	kd	CGS001-22794	CASC3	-			
276	99.34	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
277	99.34	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
278	99.34	kd	CGS001-8895	CPNE3	-			
279	99.33	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
280	99.32	oe	ccsbBroad304_00783	HPRT1	-			
281	99.32	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
282	99.32	kd	CGS001-9415	FADS2	Fatty acid desaturases			
283	99.31	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
284	99.31	kd	CGS001-94234	FOXQ1	Forkhead boxes			
285	99.3	oe	ccsbBroad304_00962	SMAD4	SMADs			
286	99.3	oe	ccsbBroad304_02243	DLGAP5	-			
287	99.3	oe	ccsbBroad304_05931	CAPG	-			
288	99.3	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
289	99.29	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
290	99.28	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
291	99.28	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
292	99.28	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
293	99.28	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
294	99.26	kd	CGS001-4683	NBN	-			
295	99.24	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
296	99.23	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
297	99.23	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
298	99.22	kd	CGS001-3485	IGFBP2	insulin-like growth factor (IGF) binding proteins			
299	99.21	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
300	99.21	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
301	99.21	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
302	99.21	kd	CGS001-538	ATP7A	ATPases / P-type			
303	99.19	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
304	99.18	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
305	99.18	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
306	99.17	oe	ccsbBroad304_02843	FTSJ1	-			
307	99.17	kd	CGS001-114785	MBD6	-			
308	99.15	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
309	99.15	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
310	99.15	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
311	99.15	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
312	99.15	kd	CGS001-5684	PSMA3	Proteasome subunits			
313	99.15	kd	CGS001-3718	JAK3	Janus kinase (JakA) family			
314	99.14	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
315	99.14	kd	CGS001-5997	RGS2	Endogenous ligands			
316	99.13	kd	CGS001-8974	P4HA2	-			
317	99.12	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
318	99.12	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
319	99.11	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
320	99.11	kd	CGS001-93487	MAPK1IP1L	-			
321	99.1	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
322	99.08	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
323	99.08	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
324	99.08	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
325	99.08	kd	CGS001-664	BNIP3	-			
326	99.06	cp	BRD-K70358946	aripiprazole	Serotonin receptor agonist		DRD2, HTR1A, HTR2A, HRH1, HTR1B, HTR1D, HTR2C, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR1E, HTR3A, HTR6, HTR7	Serotonin receptor agonist, Serotonin receptor antagonist
327	99.06	kd	CGS001-54498	SMOX	-			
328	99.06	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
329	99.04	cc		Cyclin dependent kinases LOF	-			
330	99.04	oe	ccsbBroad304_14011	PAPSS1	-			
331	99.04	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
332	99.04	kd	CGS001-23743	BHMT2	-			
333	99.02	oe	ccsbBroad304_06066	CTSL1	-			
334	99	oe	ccsbBroad304_06292	GNAI2	-			
335	98.99	oe	ccsbBroad304_05038	HORMAD2	-			
336	98.97	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
337	98.97	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
338	98.96	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
339	98.95	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
340	98.95	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
341	98.95	kd	CGS001-55872	PBK	TOPK family			
342	98.94	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
343	98.93	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
344	98.93	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
345	98.92	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
346	98.91	kd	CGS001-125919	ZNF543	Zinc fingers, C2H2-type			
347	98.91	kd	CGS001-11015	KDELR3	-			
348	98.91	kd	CGS001-3397	ID1	Basic helix-loop-helix proteins			
349	98.91	kd	CGS001-9917	FAM20B	-			
350	98.9	oe	ccsbBroad304_08292	IP6K2	-			
351	98.88	cp	BRD-K59753975	vindesine	Tubulin inhibitor		TUBB, TUBB1	Tubulin inhibitor
352	98.88	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
353	98.88	kd	CGS001-51160	VPS28	-			
354	98.88	kd	CGS001-8864	PER2	-			
355	98.87	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
356	98.87	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
357	98.86	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
358	98.84	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
359	98.84	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
360	98.84	kd	CGS001-435	ASL	-			
361	98.82	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
362	98.81	cc		Aldehyde dehydrogenases LOF	-			
363	98.81	kd	CGS001-5361	PLXNA1	Plexins			
364	98.8	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
365	98.8	oe	ccsbBroad304_13633	PI4KAP2	-			
366	98.8	oe	ccsbBroad304_06318	GPER	-			
367	98.8	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
368	98.8	kd	CGS001-5695	PSMB7	Proteasome subunits			
369	98.8	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
370	98.78	kd	CGS001-11040	PIM2	PIM family			
371	98.77	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
372	98.77	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
373	98.77	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
374	98.77	kd	CGS001-5985	RFC5	ATPases / AAA-type			
375	98.76	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
376	98.76	kd	CGS001-80274	SCUBE1	-			
377	98.76	kd	CGS001-4174	MCM5	-			
378	98.74	cp	BRD-K47780086	penciclovir	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor
379	98.74	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
380	98.73	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
381	98.73	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
382	98.73	kd	CGS001-84669	USP32	EF-hand domain containing			
383	98.72	kd	CGS001-5887	RAD23B	-			
384	98.7	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
385	98.7	kd	CGS001-388677	NOTCH2NL	-			
386	98.7	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
387	98.68	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
388	98.67	oe	ccsbBroad304_07662	NPRL2	-			
389	98.67	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
390	98.66	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
391	98.65	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
392	98.64	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
393	98.62	cc		Norepinephrine reuptake inhibitor	-			
394	98.6	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
395	98.58	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
396	98.56	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
397	98.54	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
398	98.54	kd	CGS001-6461	SHB	SH2 domain containing			
399	98.54	kd	CGS001-9813	KIAA0494	-			
400	98.53	oe	ccsbBroad304_08645	BCCIP	-			
401	98.53	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
402	98.53	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
403	98.52	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
404	98.51	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
405	98.51	kd	CGS001-10013	HDAC6	Histone deacetylases			
406	98.51	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
407	98.49	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
408	98.48	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
409	98.47	oe	ccsbBroad304_04153	PHF17	-			
410	98.47	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
411	98.47	kd	CGS001-80347	COASY	-			
412	98.47	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
413	98.45	oe	ccsbBroad304_01215	PLAUR	CD molecules			
414	98.45	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
415	98.45	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
416	98.45	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
417	98.44	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
418	98.42	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
419	98.42	kd	CGS001-3053	SERPIND1	Serine (or cysteine) peptidase inhibitors			
420	98.42	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
421	98.4	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
422	98.4	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
423	98.4	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
424	98.39	kd	CGS001-8192	CLPP	ATPases / AAA-type			
425	98.38	kd	CGS001-7020	TFAP2A	-			
426	98.36	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
427	98.36	kd	CGS001-64175	LEPRE1	-			
428	98.34	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
429	98.34	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
430	98.32	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
431	98.32	kd	CGS001-1152	CKB	-			
432	98.32	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
433	98.31	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
434	98.29	oe	ccsbBroad304_01659	TERF1	-			
435	98.29	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
436	98.28	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
437	98.28	kd	CGS001-5053	PAH	Amino acid hydroxylases			
438	98.27	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
439	98.27	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
440	98.26	kd	CGS001-1736	DKC1	-			
441	98.23	kd	CGS001-51128	SAR1B	-			
442	98.23	kd	CGS001-27333	GOLIM4	-			
443	98.21	oe	ccsbBroad304_00995	MECP2	-			
444	98.21	kd	CGS001-8435	SOAT2	-			
445	98.2	kd	CGS001-54681	P4HTM	-			
446	98.2	kd	CGS001-1756	DMD	-			
447	98.18	kd	CGS001-55509	BATF3	basic leucine zipper proteins			
448	98.16	oe	ccsbBroad304_00614	GAMT	-			
449	98.15	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
450	98.15	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
451	98.15	kd	CGS001-116519	APOA5	Apolipoproteins			
452	98.14	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
453	98.14	kd	CGS001-2674	GFRA1	GDNF receptor family			
454	98.13	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
455	98.11	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
456	98.1	kd	CGS001-10308	ZNF267	Zinc fingers, C2H2-type			
457	98.1	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
458	98.09	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
459	98.09	kd	CGS001-3297	HSF1	-			
460	98.05	oe	ccsbBroad304_07800	EXOSC8	-			
461	98.04	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
462	98.03	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
463	98.03	cp	BRD-K59456551	methotrexate	Dihydrofolate reductase inhibitor		DHFR, AOX1, FOLR1, TYMS	Dihydrofolate reductase inhibitor
464	98.02	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
465	98.01	oe	ccsbBroad304_00313	TBCB	-			
466	98.01	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
467	98	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
468	98	kd	CGS001-5829	PXN	-			
469	97.99	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
470	97.99	kd	CGS001-4817	NIT1	-			
471	97.98	kd	CGS001-22930	RAB3GAP1	-			
472	97.97	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
473	97.97	kd	CGS001-9589	WTAP	-			
474	97.95	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
475	97.94	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
476	97.94	kd	CGS001-29102	DROSHA	-			
477	97.92	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
478	97.91	oe	ccsbBroad304_07727	LIAS	-			
479	97.91	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
480	97.9	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
481	97.9	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
482	97.9	kd	CGS001-23464	GCAT	-			
483	97.88	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
484	97.85	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
485	97.85	kd	CGS001-7165	TPD52L2	-			
486	97.84	cc		Bacterial DNA gyrase inhibitor	-			
487	97.8	kd	CGS001-375318	AQP12A	Ion channels / Aquaporins			
488	97.77	oe	ccsbBroad304_04294	ATG10	-			
489	97.76	kd	CGS001-6009	RHEB	-			
490	97.76	kd	CGS001-6387	CXCL12	Endogenous ligands			
491	97.71	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
492	97.7	oe	ccsbBroad304_08386	SMOX	-			
493	97.7	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
494	97.7	kd	CGS001-59286	UBL5	-			
495	97.7	kd	CGS001-57720	GPR107	GPCR / Unclassified : 7TM orphan receptors			
496	97.69	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
497	97.68	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
498	97.68	kd	CGS001-54658	UGT1A1	UDP glucuronosyltransferases			
499	97.66	oe	ccsbBroad304_07834	GGA2	-			
500	97.66	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
501	97.66	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
502	97.64	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
503	97.64	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
504	97.64	kd	CGS001-10652	YKT6	-			
505	97.63	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
506	97.63	kd	CGS001-2260	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
507	97.6	kd	CGS001-657	BMPR1A	Type I receptor serine/threonine kinases			
508	97.58	oe	ccsbBroad304_08684	CXCR7	-			
509	97.57	kd	CGS001-26227	PHGDH	-			
510	97.56	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
511	97.55	kd	CGS001-5062	PAK2	PAKA subfamily			
512	97.54	kd	CGS001-79258	MMEL1	-			
513	97.51	oe	ccsbBroad304_09615	LACC1	-			
514	97.51	oe	ccsbBroad304_03533	CDCA8	-			
515	97.51	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
516	97.51	kd	CGS001-5351	PLOD1	-			
517	97.51	kd	CGS001-54442	KCTD5	-			
518	97.5	kd	CGS001-6934	TCF7L2	-			
519	97.49	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
520	97.49	kd	CGS001-29965	C16ORF5	-			
521	97.48	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
522	97.47	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
523	97.46	kd	CGS001-481	ATP1B1	ATPases / P-type			
524	97.44	kd	CGS001-8892	EIF2B2	-			
525	97.41	kd	CGS001-7295	TXN	-			
526	97.4	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
527	97.4	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
528	97.4	kd	CGS001-7316	UBC	-			
529	97.37	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
530	97.36	kd	CGS001-6199	RPS6KB2	p70 subfamily			
531	97.35	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
532	97.33	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
533	97.33	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
534	97.33	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
535	97.33	kd	CGS001-55837	EAPP	-			
536	97.31	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
537	97.31	kd	CGS001-6652	SORD	-			
538	97.31	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
539	97.29	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
540	97.29	kd	CGS001-4121	MAN1A1	-			
541	97.28	cp	BRD-A42423104	benproperine	Antitussive			Antitussive
542	97.27	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
543	97.25	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
544	97.24	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
545	97.24	kd	CGS001-5586	PKN2	Protein kinase N (PKN) family			
546	97.23	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
547	97.22	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
548	97.2	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
549	97.2	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
550	97.2	kd	CGS001-23378	RRP8	-			
551	97.2	kd	CGS001-5565	PRKAB2	AMPK subfamily			
552	97.17	oe	ccsbBroad304_06278	GK	Glycerol kinases			
553	97.16	kd	CGS001-206358	SLC36A1	SLC36 family of proton-coupled amino acid transporters			
554	97.11	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
555	97.1	cc		PARP inhibitor	-			
556	97.1	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
557	97.09	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
558	97.09	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
559	97.09	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
560	97.09	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
561	97.08	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
562	97.05	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
563	97	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
564	96.99	oe	ccsbBroad304_00626	GDI1	-			
565	96.98	oe	ccsbBroad304_03746	CDC42SE1	-			
566	96.97	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
567	96.97	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
568	96.96	cp	BRD-K22227508	targinine	Nitric oxide synthase inhibitor		NOS2, NOS3	Nitric oxide synthase inhibitor
569	96.96	kd	CGS001-2247	FGF2	Endogenous ligands			
570	96.95	kd	CGS001-7371	UCK2	-			
571	96.94	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
572	96.91	cc		AHSP Pathway LOF	-			
573	96.88	kd	CGS001-160	AP2A1	-			
574	96.87	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
575	96.85	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
576	96.85	kd	CGS001-83737	ITCH	-			
577	96.84	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
578	96.84	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
579	96.83	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
580	96.83	kd	CGS001-2690	GHR	Prolactin receptor family			
581	96.82	cc		NFKB Activation GOF	-			
582	96.79	kd	CGS001-9655	SOCS5	SH2 domain containing			
583	96.76	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
584	96.75	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
585	96.74	kd	CGS001-6519	SLC3A1	SLC3 family			
586	96.74	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
587	96.73	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
588	96.73	kd	CGS001-817	CAMK2D	CAMK2 family			
589	96.69	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
590	96.68	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
591	96.61	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
592	96.6	kd	CGS001-3856	KRT8	Intermediate filaments type II, keratins (basic)			
593	96.6	kd	CGS001-8900	CCNA1	-			
594	96.6	kd	CGS001-6347	CCL2	Chemokine ligands			
595	96.56	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
596	96.56	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
597	96.54	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
598	96.53	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
599	96.52	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
600	96.51	kd	CGS001-9020	MAP3K14	MAPKKK:STE-unique family			
601	96.49	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
602	96.48	kd	CGS001-374291	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
603	96.48	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
604	96.46	kd	CGS001-11168	PSIP1	-			
605	96.44	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
606	96.43	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
607	96.41	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
608	96.39	oe	ccsbBroad304_00221	CASP3	Caspases			
609	96.39	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
610	96.38	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
611	96.37	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
612	96.35	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
613	96.34	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
614	96.33	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
615	96.31	cc		Protein phosphatase catalytic subunits LOF	-			
616	96.3	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
617	96.3	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
618	96.28	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
619	96.28	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
620	96.28	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
621	96.28	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
622	96.27	cc		PI3K Signaling LOF	-			
623	96.27	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
624	96.27	kd	CGS001-9133	CCNB2	-			
625	96.26	kd	CGS001-5445	PON2	Paraoxonases			
626	96.24	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
627	96.22	oe	ccsbBroad304_03640	CEP72	-			
628	96.21	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
629	96.21	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
630	96.2	kd	CGS001-10972	TMED10	-			
631	96.19	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
632	96.19	kd	CGS001-57007	CXCR7	-			
633	96.18	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
634	96.18	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
635	96.15	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
636	96.14	cp	BRD-K55034111	pefloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
637	96.13	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
638	96.13	kd	CGS001-9200	PTPLA	-			
639	96.1	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
640	96.09	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
641	96.06	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
642	96.01	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
643	96.01	kd	CGS001-760	CA2	Carbonic anhydrases			
644	95.98	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
645	95.98	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
646	95.93	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
647	95.93	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
648	95.93	kd	CGS001-23621	BACE1	Pepsin			
649	95.92	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
650	95.9	oe	ccsbBroad304_07761	CORO1A	Coronins			
651	95.9	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
652	95.89	oe	ccsbBroad304_03615	ZNF673	-			
653	95.88	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
654	95.84	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
655	95.83	kd	CGS001-8317	CDC7	CDC7 family			
656	95.82	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
657	95.82	kd	CGS001-5091	PC	Carboxylases			
658	95.76	cc		EIF Proteins LOF	-			
659	95.71	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
660	95.71	oe	ccsbBroad304_09281	TPD52L3	-			
661	95.7	cp	BRD-K96471533	nitazoxanide	Pyruvate ferredoxin oxidoreductase inhibitor			Pyruvate ferredoxin oxidoreductase inhibitor
662	95.69	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
663	95.68	cc		General transcription factors group 1 LOF	-			
664	95.68	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
665	95.68	kd	CGS001-57661	PHRF1	Zinc fingers, PHD-type			
666	95.68	kd	CGS001-4129	MAOB	Catecholamine turnover			
667	95.67	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
668	95.66	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
669	95.65	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
670	95.62	oe	ccsbBroad304_07280	LAMTOR3	-			
671	95.6	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
672	95.6	kd	CGS001-7389	UROD	-			
673	95.59	kd	CGS001-546	ATRX	-			
674	95.58	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
675	95.56	oe	ccsbBroad304_00446	DKC1	-			
676	95.53	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
677	95.52	oe	ccsbBroad304_07326	EIF2B2	-			
678	95.49	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
679	95.47	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
680	95.47	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
681	95.46	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
682	95.43	oe	ccsbBroad304_01985	EIF3H	-			
683	95.43	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
684	95.42	kd	CGS001-23314	SATB2	Homeoboxes / CUT class			
685	95.41	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
686	95.39	oe	ccsbBroad304_01532	SIAH1	-			
687	95.38	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
688	95.38	kd	CGS001-84969	TOX2	-			
689	95.37	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
690	95.33	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
691	95.32	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
692	95.3	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
693	95.29	oe	ccsbBroad304_08325	LIPT1	-			
694	95.29	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
695	95.24	cp	BRD-K85030058	benactyzine	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
696	95.23	kd	CGS001-27102	EIF2AK1	Other PEK family kinases			
697	95.22	cp	BRD-K32311154	nifekalant	Potassium channel blocker			Potassium channel blocker
698	95.19	oe	ccsbBroad304_00423	DAXX	-			
699	95.15	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
700	95.14	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
701	95.14	kd	CGS001-27347	STK39	FRAY subfamily			
702	95.12	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
703	95.1	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
704	95.1	oe	ccsbBroad304_02012	FADD	-			
705	95.07	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
706	95.05	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
707	95.05	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
708	95.04	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
709	94.99	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
710	94.99	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
711	94.91	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
712	94.89	kd	CGS001-677	ZFP36L1	RING-type (C3HC4) zinc fingers			
713	94.86	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
714	94.78	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
715	94.76	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
716	94.75	oe	ccsbBroad304_02292	BCL2L11	-			
717	94.75	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
718	94.73	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
719	94.72	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
720	94.7	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
721	94.7	kd	CGS001-1453	CSNK1D	Casein kinase 1 (CK1) family			
722	94.69	kd	CGS001-10681	GNB5	WD repeat domain containing			
723	94.67	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
724	94.67	kd	CGS001-109	ADCY3	Adenylyl cyclases			
725	94.66	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
726	94.66	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
727	94.65	kd	CGS001-9807	IP6K1	-			
728	94.62	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
729	94.62	kd	CGS001-1457	CSNK2A1	Casein kinase 2 (CK2) family			
730	94.62	kd	CGS001-10180	RBM6	G patch domain containing			
731	94.6	kd	CGS001-6253	RTN2	-			
732	94.59	cc		Progesterone receptor agonist	-			
733	94.57	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
734	94.55	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
735	94.54	cp	BRD-K23369905	oxiconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
736	94.53	kd	CGS001-5566	PRKACA	Protein kinase A			
737	94.52	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
738	94.51	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
739	94.48	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
740	94.47	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
741	94.46	kd	CGS001-472	ATM	Other PIKK family kinases			
742	94.44	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
743	94.43	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
744	94.43	kd	CGS001-5708	PSMD2	Proteasome subunits			
745	94.41	kd	CGS001-1659	DHX8	DEAH-boxes			
746	94.4	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
747	94.35	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
748	94.35	kd	CGS001-821	CANX	-			
749	94.32	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
750	94.32	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
751	94.32	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
752	94.32	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
753	94.27	oe	ccsbBroad304_07197	PDHX	-			
754	94.27	kd	CGS001-8853	ASAP2	Ankyrin repeat domain containing			
755	94.23	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
756	94.21	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
757	94.2	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
758	94.19	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
759	94.19	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
760	94.18	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
761	94.18	kd	CGS001-51290	ERGIC2	-			
762	94.16	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
763	94.16	oe	ccsbBroad304_00179	BTG1	-			
764	94.12	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
765	94.11	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
766	94.09	oe	ccsbBroad304_01186	PHB	-			
767	94.09	oe	ccsbBroad304_05194	LIPH	-			
768	94.07	oe	ccsbBroad304_02862	CCRN4L	-			
769	94.01	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
770	93.99	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
771	93.97	oe	ccsbBroad304_00120	ATOX1	-			
772	93.97	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
773	93.95	oe	ccsbBroad304_02845	PRPF6	-			
774	93.9	kd	CGS001-23536	ADAT1	-			
775	93.88	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
776	93.88	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
777	93.86	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
778	93.86	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
779	93.83	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
780	93.82	kd	CGS001-27336	HTATSF1	RNA binding motif (RRM) containing			
781	93.79	oe	ccsbBroad304_01880	LAGE3	-			
782	93.78	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
783	93.76	oe	ccsbBroad304_06126	TSC22D3	-			
784	93.74	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
785	93.72	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
786	93.72	oe	ccsbBroad304_06174	ERCC1	-			
787	93.72	kd	CGS001-10312	TCIRG1	ATPases / V-type			
788	93.71	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
789	93.7	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
790	93.68	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
791	93.67	oe	ccsbBroad304_02668	PNKP	-			
792	93.66	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
793	93.64	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
794	93.64	kd	CGS001-8536	CAMK1	CAMK1 family			
795	93.6	kd	CGS001-8807	IL18RAP	CD molecules			
796	93.57	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
797	93.54	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
798	93.48	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
799	93.47	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
800	93.45	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
801	93.45	kd	CGS001-1837	DTNA	-			
802	93.44	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
803	93.44	kd	CGS001-9867	PJA2	RING-type (C3HC4) zinc fingers			
804	93.42	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
805	93.41	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
806	93.41	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
807	93.39	kd	CGS001-955	ENTPD6	-			
808	93.37	kd	CGS001-5575	PRKAR1B	Protein kinase A			
809	93.36	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
810	93.36	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
811	93.34	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
812	93.33	kd	CGS001-10153	CEBPZ	-			
813	93.27	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
814	93.24	oe	ccsbBroad304_00941	LIG3	-			
815	93.23	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
816	93.21	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
817	93.19	oe	ccsbBroad304_06420	ICAM3	CD molecules			
818	93.18	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
819	93.17	oe	ccsbBroad304_00515	ERH	-			
820	93.15	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
821	93.12	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
822	93.11	oe	ccsbBroad304_07145	ZFP161	-			
823	93.11	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
824	93.11	kd	CGS001-10434	LYPLA1	-			
825	93.11	kd	CGS001-8022	LHX3	Homeoboxes / LIM class			
826	93.09	kd	CGS001-55765	C1ORF106	-			
827	93.07	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
828	93.06	kd	CGS001-64781	CERK	Ceramide kinase			
829	93.05	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
830	93.04	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
831	93.04	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
832	93.04	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
833	93.02	kd	CGS001-2539	G6PD	-			
834	93.01	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
835	93.01	oe	ccsbBroad304_00632	GGCX	Carboxylases			
836	93	oe	ccsbBroad304_02502	GNA13	-			
837	93	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
838	92.98	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
839	92.97	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
840	92.97	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
841	92.95	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
842	92.92	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
843	92.91	kd	CGS001-539	ATP5O	ATPases / F-type			
844	92.88	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
845	92.87	oe	ccsbBroad304_06975	SMARCC2	-			
846	92.87	cp	BRD-K90733503	cefalexin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
847	92.85	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
848	92.85	oe	ccsbBroad304_03591	ETNK1	-			
849	92.85	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
850	92.83	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
851	92.82	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
852	92.78	oe	ccsbBroad304_06889	RPN2	-			
853	92.75	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
854	92.74	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
855	92.74	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
856	92.73	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
857	92.7	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
858	92.68	kd	CGS001-55229	PANK4	-			
859	92.67	oe	ccsbBroad304_07600	NSA2	-			
860	92.67	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
861	92.64	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
862	92.63	oe	ccsbBroad304_08093	DCPS	-			
863	92.6	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
864	92.59	oe	ccsbBroad304_10758	CTBP2	-			
865	92.59	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
866	92.59	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
867	92.56	kd	CGS001-5590	PRKCZ	Iota subfamily			
868	92.54	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
869	92.54	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
870	92.5	kd	CGS001-1212	CLTB	-			
871	92.49	cc		DNA polymerase inhibitor	-			
872	92.48	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
873	92.48	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
874	92.47	oe	ccsbBroad304_07887	GCAT	-			
875	92.47	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
876	92.47	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
877	92.46	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
878	92.46	kd	CGS001-4976	OPA1	-			
879	92.44	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
880	92.44	kd	CGS001-9833	MELK	MELK subfamily			
881	92.42	kd	CGS001-5621	PRNP	CD molecules			
882	92.38	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
883	92.37	kd	CGS001-389421	LIN28B	-			
884	92.35	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
885	92.31	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
886	92.3	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
887	92.27	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
888	92.21	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
889	92.21	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
890	92.19	oe	ccsbBroad304_06670	OGG1	-			
891	92.14	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
892	92.12	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
893	92.1	kd	CGS001-11140	CDC37	-			
894	92.09	cp	BRD-K34437622	BRD-K34437622	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
895	92.06	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
896	92.05	kd	CGS001-5581	PRKCE	Eta subfamily			
897	92.03	oe	ccsbBroad304_03089	PACSIN3	-			
898	92.02	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
899	92.02	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
900	92	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
901	91.99	kd	CGS001-183	AGT	Endogenous ligands			
902	91.98	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
903	91.96	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
904	91.95	kd	CGS001-10097	ACTR2	-			
905	91.93	oe	ccsbBroad304_07140	XPC	-			
906	91.92	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
907	91.89	kd	CGS001-5579	PRKCB	Alpha subfamily			
908	91.82	kd	CGS001-6364	CCL20	Chemokine ligands			
909	91.81	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
910	91.8	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
911	91.8	kd	CGS001-5498	PPOX	-			
912	91.8	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
913	91.79	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
914	91.79	kd	CGS001-22933	SIRT2	Histone deacetylases			
915	91.78	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
916	91.78	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
917	91.78	kd	CGS001-516	ATP5G1	ATPases / F-type			
918	91.74	kd	CGS001-161725	OTUD7A	OTU domain containing			
919	91.68	kd	CGS001-3693	ITGB5	Integrins			
920	91.67	kd	CGS001-10745	PHTF1	-			
921	91.66	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
922	91.66	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
923	91.64	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
924	91.56	kd	CGS001-115650	TNFRSF13C	Tumour necrosis factor (TNF) receptor family			
925	91.51	oe	ccsbBroad304_02922	TES	-			
926	91.48	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
927	91.47	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
928	91.41	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
929	91.36	cc		Lysine acetyltransferases LOF	-			
930	91.36	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
931	91.33	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
932	91.29	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
933	91.28	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
934	91.24	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
935	91.23	oe	ccsbBroad304_01247	POU2AF1	-			
936	91.23	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
937	91.2	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
938	91.2	kd	CGS001-65263	PYCRL	-			
939	91.19	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
940	91.16	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
941	91.15	kd	CGS001-2710	GK	Glycerol kinases			
942	91.11	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
943	91.07	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
944	91.05	cc		Gamma secretase inhibitor	-			
945	91.03	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
946	90.98	oe	ccsbBroad304_02270	FAM20B	-			
947	90.97	kd	CGS001-5345	SERPINF2	Serine (or cysteine) peptidase inhibitors			
948	90.95	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
949	90.94	kd	CGS001-6929	TCF3	Basic helix-loop-helix proteins			
950	90.92	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
951	90.91	cp	BRD-K10670311	sulfasalazine	Antirheumatic		PTGS1, PTGS2, ACAT1, ALOX5, CHUK, IKBKB, PLA2G1B, PPARG, SLC46A1, SLC7A11, TBXAS1	Antirheumatic, NFkB pathway inhibitor
952	90.91	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
953	90.9	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
954	90.85	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
955	90.85	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
956	90.84	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
957	90.83	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
958	90.82	kd	CGS001-8464	SUPT3H	-			
959	90.8	kd	CGS001-3486	IGFBP3	insulin-like growth factor (IGF) binding proteins			
960	90.78	kd	CGS001-57326	PBXIP1	-			
961	90.77	kd	CGS001-10010	TANK	-			
962	90.76	kd	CGS001-8767	RIPK2	Receptor interacting protein kinase (RIPK) family			
963	90.75	oe	ccsbBroad304_00985	MCL1	-			
964	90.74	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
965	90.73	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
966	90.71	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
967	90.7	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
968	90.66	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
969	90.65	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
970	90.64	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
971	90.64	cp	BRD-A68589262	troxipide	Glucosamine synthetase stimulant			Glucosamine synthetase stimulant
972	90.63	kd	CGS001-2963	GTF2F2	General transcription factors			
973	90.62	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
974	90.61	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
975	90.59	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
976	90.51	cp	BRD-K19462402	buflomedil	Adrenergic receptor antagonist		CACNA1C	Adrenergic receptor antagonist, Calcium channel blocker
977	90.51	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
978	90.51	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
979	90.5	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
980	90.48	kd	CGS001-29982	NRBF2	-			
981	90.46	kd	CGS001-9344	TAOK2	TAO subfamily			
982	90.44	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
983	90.44	kd	CGS001-1841	DTYMK	-			
984	90.44	kd	CGS001-54108	CHRAC1	-			
985	90.4	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
986	90.36	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
987	90.35	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
988	90.3	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
989	90.25	cc		MCM family LOF	-			
990	90.25	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
991	90.19	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
992	90.17	kd	CGS001-115	ADCY9	Adenylyl cyclases			
993	90.14	cp	BRD-A16934955	nalbuphine	Opioid receptor agonist		OPRD1, OPRK1, OPRM1	Opioid receptor agonist, Opioid receptor antagonist
994	90.14	kd	CGS001-64219	PJA1	RING-type (C3HC4) zinc fingers			
995	90.11	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
996	90.11	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
997	90.09	oe	ccsbBroad304_07861	COBL	-			
998	90.04	kd	CGS001-79135	APOO	Apolipoproteins			
999	90.03	kd	CGS001-3675	ITGA3	Integrins			
1000	90.03	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
1001	90.01	kd	CGS001-83439	TCF7L1	-			
1002	89.98	kd	CGS001-5710	PSMD4	Proteasome (prosome, macropain) subunits			
1003	89.96	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
1004	89.94	kd	CGS001-5327	PLAT	Chymotrypsin			
1005	89.93	oe	ccsbBroad304_03980	DCLRE1B	-			
1006	89.87	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
1007	89.86	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
1008	89.84	cc		X linked mental retardation group 2 LOF	-			
1009	89.8	kd	CGS001-1528	CYB5A	Cytochrome b genes			
1010	89.77	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
1011	89.77	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
1012	89.77	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
1013	89.77	kd	CGS001-27035	NOX1	-			
1014	89.75	kd	CGS001-2919	CXCL1	Endogenous ligands			
1015	89.71	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
1016	89.7	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
1017	89.69	kd	CGS001-7533	YWHAH	-			
1018	89.67	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
1019	89.67	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
1020	89.67	kd	CGS001-4482	MSRA	-			
1021	89.65	kd	CGS001-2882	GPX7	-			
1022	89.64	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1023	89.62	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
1024	89.59	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
1025	89.58	oe	ccsbBroad304_13813	ARAF	RAF family			
1026	89.54	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
1027	89.53	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
1028	89.53	kd	CGS001-11315	PARK7	Parkinson disease			
1029	89.47	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
1030	89.44	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
1031	89.43	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
1032	89.41	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
1033	89.41	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
1034	89.41	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
1035	89.39	kd	CGS001-2678	GGT1	CD molecules			
1036	89.38	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
1037	89.36	kd	CGS001-399694	SHC4	SH2 domain containing			
1038	89.32	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
1039	89.28	kd	CGS001-3551	IKBKB	IKK family			
1040	89.24	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1041	89.19	kd	CGS001-9687	GREB1	-			
1042	89.16	oe	ccsbBroad304_01105	PNP	-			
1043	89.12	oe	ccsbBroad304_03155	DHH	-			
1044	89.12	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
1045	89.08	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
1046	89.07	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
1047	88.99	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
1048	88.99	kd	CGS001-2877	GPX2	-			
1049	88.98	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
1050	88.98	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
1051	88.97	cp	BRD-K56614220	clofazimine	GK0582 inhibitor			GK0582 inhibitor
1052	88.95	cp	BRD-K89708791	rifaximin	RNA synthesis inhibitor		NR1I2, CYP3A4	RNA synthesis inhibitor
1053	88.91	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
1054	88.89	cp	BRD-K94887716	TFMPP	Serotonin receptor agonist			Serotonin receptor agonist, Serotonin receptor antagonist
1055	88.86	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
1056	88.86	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
1057	88.86	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
1058	88.84	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
1059	88.82	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
1060	88.8	kd	CGS001-6793	STK10	SLK subfamily			
1061	88.79	kd	CGS001-5986	RFNG	Beta 3-glycosyltransferases			
1062	88.76	kd	CGS001-10923	SUB1	-			
1063	88.69	oe	ccsbBroad304_03544	FAIM	-			
1064	88.69	kd	CGS001-6307	MSMO1	Fatty acid hydroxylase domain containing			
1065	88.67	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
1066	88.65	kd	CGS001-50846	DHH	-			
1067	88.64	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1068	88.57	oe	ccsbBroad304_10437	STMN1	-			
1069	88.57	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
1070	88.55	kd	CGS001-11329	STK38	NDR family			
1071	88.53	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
1072	88.53	kd	CGS001-6277	S100A6	EF-hand domain containing			
1073	88.49	oe	ccsbBroad304_11405	UBE3C	-			
1074	88.48	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
1075	88.45	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
1076	88.42	cc		DNA synthesis inhibitor	-			
1077	88.39	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
1078	88.39	kd	CGS001-2115	ETV1	ETS Transcription Factors			
1079	88.37	cc		Adenosine receptor agonist	-			
1080	88.33	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
1081	88.31	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1082	88.3	kd	CGS001-3460	IFNGR2	Interferon receptor family			
1083	88.23	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
1084	88.21	kd	CGS001-9375	TM9SF2	-			
1085	88.16	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
1086	88.1	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
1087	88.1	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
1088	88.08	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
1089	88.03	oe	ccsbBroad304_02596	KDELR3	-			
1090	88.01	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
1091	88	kd	CGS001-23	ABCF1	ATP binding cassette transporters / subfamily F			
1092	87.98	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
1093	87.94	oe	ccsbBroad304_04675	ATG4A	-			
1094	87.9	kd	CGS001-139760	GPR119	GPCR / Class A : Orphans			
1095	87.89	kd	CGS001-4615	MYD88	-			
1096	87.88	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
1097	87.82	kd	CGS001-8553	BHLHE40	Basic helix-loop-helix proteins			
1098	87.81	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
1099	87.74	cc		T-type calcium channel blocker	-			
1100	87.73	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
1101	87.71	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
1102	87.62	kd	CGS001-3456	IFNB1	Interferons			
1103	87.59	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
1104	87.56	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
1105	87.55	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
1106	87.55	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
1107	87.54	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
1108	87.48	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
1109	87.46	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
1110	87.45	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1111	87.45	kd	CGS001-5925	RB1	Endogenous ligands			
1112	87.44	kd	CGS001-5198	PFAS	-			
1113	87.37	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
1114	87.36	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
1115	87.36	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
1116	87.32	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
1117	87.32	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
1118	87.28	cp	BRD-A71009679	KUC103420N	-666			-666
1119	87.28	kd	CGS001-6625	SNRNP70	RNA binding motif (RRM) containing			
1120	87.25	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
1121	87.24	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
1122	87.18	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
1123	87.18	kd	CGS001-8503	PIK3R3	Phosphatidylinositol kinases			
1124	87.15	kd	CGS001-10287	RGS19	Regulators of G-protein signaling			
1125	87.1	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
1126	87.04	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
1127	87.02	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
1128	86.94	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
1129	86.89	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
1130	86.88	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
1131	86.87	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
1132	86.86	cc		Bile acid	-			
1133	86.86	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
1134	86.85	oe	ccsbBroad304_01662	TFDP2	-			
1135	86.85	kd	CGS001-5411	PNN	-			
1136	86.8	oe	ccsbBroad304_00472	EBF1	-			
1137	86.75	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
1138	86.74	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
1139	86.73	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
1140	86.71	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
1141	86.7	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
1142	86.64	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
1143	86.63	cp	BRD-K09471561	levofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
1144	86.62	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
1145	86.6	kd	CGS001-10460	TACC3	-			
1146	86.6	kd	CGS001-661	POLR3D	RNA polymerase subunits			
1147	86.58	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
1148	86.53	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
1149	86.52	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
1150	86.51	oe	ccsbBroad304_02443	HAX1	-			
1151	86.5	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
1152	86.44	oe	ccsbBroad304_01114	NUP88	-			
1153	86.38	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
1154	86.36	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
1155	86.36	kd	CGS001-65975	STK33	CAMK-unique family			
1156	86.34	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
1157	86.33	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
1158	86.32	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
1159	86.31	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
1160	86.3	kd	CGS001-9261	MAPKAPK2	MAPKAPK subfamily			
1161	86.29	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
1162	86.27	kd	CGS001-3980	LIG3	-			
1163	86.26	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
1164	86.26	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
1165	86.23	kd	CGS001-965	CD58	CD molecules			
1166	86.22	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
1167	86.2	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
1168	86.14	cc		LIM class homeoboxes GOF	-			
1169	86.14	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
1170	86.14	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
1171	86.1	cp	BRD-K06388322	pramipexole	Dopamine receptor agonist		DRD3, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
1172	86.09	kd	CGS001-10641	NPRL2	-			
1173	86.04	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
1174	86.02	oe	ccsbBroad304_05936	CASP2	Caspases			
1175	85.99	oe	ccsbBroad304_02446	TADA3	-			
1176	85.99	kd	CGS001-6197	RPS6KA3	RSK subfamily			
1177	85.91	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1178	85.88	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
1179	85.87	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
1180	85.87	kd	CGS001-7010	TEK	Type XII RTKs: TIE family of angiopoietin receptors			
1181	85.85	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
1182	85.84	kd	CGS001-6794	STK11	LKB subfamily			
1183	85.82	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
1184	85.81	kd	CGS001-2194	FASN	Short chain dehydrogenase/reductase superfamily / Atypical members			
1185	85.77	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
1186	85.75	kd	CGS001-11112	HIBADH	-			
1187	85.72	kd	CGS001-80777	CYB5B	-			
1188	85.65	oe	ccsbBroad304_02402	TMEM5	-			
1189	85.64	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
1190	85.54	kd	CGS001-9467	SH3BP5	-			
1191	85.53	oe	ccsbBroad304_06518	LDHA	-			
1192	85.43	kd	CGS001-2512	FTL	-			
1193	85.41	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
1194	85.41	kd	CGS001-6491	STIL	-			
1195	85.38	kd	CGS001-5660	PSAP	Endogenous ligands			
1196	85.36	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
1197	85.33	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
1198	85.32	kd	CGS001-10020	GNE	-			
1199	85.29	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
1200	85.27	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
1201	85.19	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
1202	85.17	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
1203	85.15	kd	CGS001-7444	VRK2	Vaccina related kinase (VRK) family			
1204	85.12	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
1205	85.12	cp	BRD-A35519318	benidipine	Calcium channel blocker		CACNA1C, CACNA1G, CYP3A5	Calcium channel blocker
1206	85.11	oe	ccsbBroad304_00170	BNIP1	-			
1207	85.11	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
1208	85.11	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1209	84.96	kd	CGS001-9180	OSMR	IL-6 receptor family			
1210	84.95	oe	ccsbBroad304_01102	NMT1	-			
1211	84.95	cp	BRD-K44094599	tacrolimus	Calcineurin inhibitor		FKBP1A, CYP3A5, CYP3A7	Calcineurin inhibitor
1212	84.77	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1213	84.73	kd	CGS001-55206	SBNO1	-			
1214	84.72	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
1215	84.7	cc		Tricyclic antidepressant	-			
1216	84.67	kd	CGS001-333929	SNAI3	Snail homologs			
1217	84.63	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
1218	84.63	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
1219	84.62	kd	CGS001-3978	LIG1	-			
1220	84.61	cc		HDAC inhibitor	-			
1221	84.6	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
1222	84.58	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
1223	84.55	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
1224	84.53	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
1225	84.53	kd	CGS001-84878	ZBTB45	BTB/POZ domain containing			
1226	84.5	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
1227	84.45	kd	CGS001-6925	TCF4	Basic helix-loop-helix proteins			
1228	84.43	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
1229	84.43	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
1230	84.42	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
1231	84.4	kd	CGS001-5202	PFDN2	-			
1232	84.38	kd	CGS001-9146	HGS	Zinc fingers, FYVE domain containing			
1233	84.36	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
1234	84.36	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
1235	84.29	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
1236	84.27	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
1237	84.25	kd	CGS001-23223	RRP12	-			
1238	84.2	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
1239	84.2	kd	CGS001-6513	SLC2A1	Solute carriers			
1240	84.18	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
1241	84.17	oe	ccsbBroad304_00226	CAV1	-			
1242	84.09	kd	CGS001-10608	MXD4	Basic helix-loop-helix proteins			
1243	84.03	cp	BRD-K32744045	disulfiram	Aldehyde dehydrogenase inhibitor		ALDH2, ALDH1A2, ALDH5A1, ALDH7A1, CYP2E1, DBH, DNMT1, TRPA1	Aldehyde dehydrogenase inhibitor, TRPV agonist, DNA methyltransferase inhibitor
1244	84.02	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
1245	84.01	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
1246	83.96	oe	ccsbBroad304_06777	PRNP	CD molecules			
1247	83.93	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
1248	83.91	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
1249	83.89	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
1250	83.84	kd	CGS001-2717	GLA	-			
1251	83.81	kd	CGS001-8480	RAE1	WD repeat domain containing			
1252	83.8	kd	CGS001-5373	PMM2	-			
1253	83.74	kd	CGS001-4331	MNAT1	RING-type (C3HC4) zinc fingers			
1254	83.7	kd	CGS001-10769	PLK2	Polo-like kinase (PLK) family			
1255	83.69	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
1256	83.69	kd	CGS001-22850	ADNP2	Zinc fingers, C2H2-type			
1257	83.65	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
1258	83.63	kd	CGS001-8826	IQGAP1	-			
1259	83.61	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
1260	83.6	cc		Aurora kinase inhibitor	-			
1261	83.6	oe	ccsbBroad304_05192	SPRED2	-			
1262	83.55	kd	CGS001-22889	KIAA0907	-			
1263	83.53	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
1264	83.52	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
1265	83.48	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
1266	83.48	kd	CGS001-23786	BCL2L13	-			
1267	83.47	kd	CGS001-5564	PRKAB1	AMPK subfamily			
1268	83.46	kd	CGS001-5328	PLAU	Chymotrypsin			
1269	83.42	kd	CGS001-55536	CDCA7L	-			
1270	83.39	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
1271	83.37	kd	CGS001-55163	PNPO	-			
1272	83.35	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
1273	83.29	kd	CGS001-5901	RAN	-			
1274	83.28	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
1275	83.25	kd	CGS001-23635	SSBP2	-			
1276	83.23	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
1277	83.22	kd	CGS001-6421	SFPQ	RNA binding motif (RRM) containing			
1278	83.16	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
1279	83.14	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
1280	83.05	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
1281	83.02	kd	CGS001-3203	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
1282	83.01	kd	CGS001-51752	ERAP1	Aminopeptidase N			
1283	83	kd	CGS001-55082	ARGLU1	-			
1284	82.98	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
1285	82.95	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
1286	82.94	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1287	82.9	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
1288	82.83	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1289	82.81	kd	CGS001-995	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1290	82.77	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
1291	82.74	oe	ccsbBroad304_03191	NOSIP	-			
1292	82.73	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
1293	82.67	cp	BRD-K18523449	mestanolone	Androgenic steroid			Androgenic steroid
1294	82.65	kd	CGS001-9897	KIAA0196	-			
1295	82.63	kd	CGS001-5063	PAK3	PAKA subfamily			
1296	82.62	kd	CGS001-1827	RCAN1	-			
1297	82.6	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
1298	82.59	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
1299	82.58	kd	CGS001-112812	FDX1L	-			
1300	82.57	kd	CGS001-1196	CLK2	CDC-like kinases			
1301	82.57	kd	CGS001-11257	TP53TG1	-			
1302	82.54	kd	CGS001-634	CEACAM1	CD molecules			
1303	82.51	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
1304	82.49	kd	CGS001-818	CAMK2G	CAMK2 family			
1305	82.48	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
1306	82.48	kd	CGS001-1950	EGF	-			
1307	82.43	kd	CGS001-55011	PIH1D1	-			
1308	82.42	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
1309	82.38	oe	ccsbBroad304_09708	PNLDC1	-			
1310	82.37	oe	ccsbBroad304_00550	FDXR	-			
1311	82.37	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
1312	82.36	cc		Mitogen activated protein kinases LOF	-			
1313	82.34	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
1314	82.31	oe	ccsbBroad304_06367	HK1	-			
1315	82.25	oe	ccsbBroad304_07888	CBX6	-			
1316	82.25	kd	CGS001-3488	IGFBP5	insulin-like growth factor (IGF) binding proteins			
1317	82.23	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
1318	82.22	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
1319	82.2	oe	ccsbBroad304_03311	EVL	-			
1320	82.19	kd	CGS001-1384	CRAT	-			
1321	82.13	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
1322	82.05	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
1323	81.97	kd	CGS001-55662	HIF1AN	-			
1324	81.92	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
1325	81.92	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
1326	81.91	oe	ccsbBroad304_08605	PBK	TOPK family			
1327	81.85	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
1328	81.84	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
1329	81.84	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
1330	81.8	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
1331	81.76	oe	ccsbBroad304_01008	KITLG	-			
1332	81.68	kd	CGS001-10123	ARL4C	ADP-ribosylation factors			
1333	81.63	kd	CGS001-255738	PCSK9	Subtilisin			
1334	81.6	kd	CGS001-5879	RAC1	Endogenous ligands			
1335	81.6	kd	CGS001-11157	LSM6	-			
1336	81.58	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1337	81.57	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
1338	81.53	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
1339	81.51	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
1340	81.5	oe	ccsbBroad304_07768	NISCH	-			
1341	81.46	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
1342	81.46	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
1343	81.45	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
1344	81.41	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
1345	81.36	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
1346	81.34	kd	CGS001-53834	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
1347	81.32	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
1348	81.22	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
1349	81.22	kd	CGS001-7471	WNT1	Endogenous ligands			
1350	81.12	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
1351	81.12	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1352	81.1	oe	ccsbBroad304_07080	TM7SF2	-			
1353	81.03	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
1354	80.98	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
1355	80.95	oe	ccsbBroad304_01699	TPD52L2	-			
1356	80.94	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
1357	80.91	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
1358	80.87	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
1359	80.84	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
1360	80.81	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
1361	80.78	kd	CGS001-7079	TIMP4	-			
1362	80.75	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
1363	80.74	kd	CGS001-2335	FN1	Endogenous ligands			
1364	80.73	kd	CGS001-139135	PASD1	-			
1365	80.7	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
1366	80.67	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
1367	80.66	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
1368	80.63	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
1369	80.59	cc		HIF activator	-			
1370	80.55	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
1371	80.48	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
1372	80.48	kd	CGS001-55781	RIOK2	RIO2 subfamily			
1373	80.38	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
1374	80.33	oe	ccsbBroad304_02115	PTTG1	-			
1375	80.29	oe	ccsbBroad304_02553	BLCAP	-			
1376	80.26	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
1377	80.26	oe	ccsbBroad304_01398	RHEB	-			
1378	80.26	kd	CGS001-213	ALB	-			
1379	80.2	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
1380	80.18	oe	ccsbBroad304_06095	DFFB	-			
1381	80.15	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
1382	80.13	cc		BMP Signaling LOF	-			
1383	80.13	oe	ccsbBroad304_01304	PSEN1	Presenilin			
1384	80.13	kd	CGS001-7103	TSPAN8	Tetraspanins			
1385	80.13	kd	CGS001-4522	MTHFD1	-			
1386	80.11	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
1387	80.1	kd	CGS001-4088	SMAD3	SMADs			
1388	80.04	kd	CGS001-7030	TFE3	Basic helix-loop-helix proteins			
1389	80.02	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
1390	80.02	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
1391	79.99	cc		Cyclins LOF	-			
1392	79.98	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1393	79.96	kd	CGS001-10901	DHRS4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1394	79.92	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
1395	79.91	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
1396	79.91	kd	CGS001-2073	ERCC5	-			
1397	79.9	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
1398	79.89	cp	BRD-K85090592	pilocarpine	Acetylcholine receptor agonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor agonist
1399	79.87	kd	CGS001-2896	GRN	-			
1400	79.85	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
1401	79.84	kd	CGS001-4830	NME1	-			
1402	79.77	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
1403	79.76	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
1404	79.7	kd	CGS001-2961	GTF2E2	General transcription factors			
1405	79.65	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
1406	79.65	kd	CGS001-5546	PRCC	-			
1407	79.61	oe	ccsbBroad304_02875	BRP44	-			
1408	79.61	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
1409	79.59	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
1410	79.58	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
1411	79.52	kd	CGS001-2266	FGG	Endogenous ligands			
1412	79.5	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
1413	79.5	kd	CGS001-1407	CRY1	-			
1414	79.46	oe	ccsbBroad304_01674	TIMP4	-			
1415	79.44	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
1416	79.43	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
1417	79.42	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
1418	79.38	kd	CGS001-1840	DTX1	-			
1419	79.32	kd	CGS001-5744	PTHLH	Endogenous ligands			
1420	79.3	kd	CGS001-4893	NRAS	RAS subfamily			
1421	79.27	kd	CGS001-607	BCL9	-			
1422	79.24	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
1423	79.2	oe	ccsbBroad304_03357	RASD1	-			
1424	79.14	oe	ccsbBroad304_00600	FYN	Src family			
1425	79.14	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
1426	79.13	cp	BRD-A07395371	esmolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
1427	79.12	kd	CGS001-7088	TLE1	WD repeat domain containing			
1428	79.05	kd	CGS001-23386	NUDCD3	-			
1429	78.98	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
1430	78.94	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
1431	78.92	oe	ccsbBroad304_03186	GMNN	-			
1432	78.92	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
1433	78.9	kd	CGS001-324	APC	Armadillo repeat containing			
1434	78.84	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
1435	78.73	kd	CGS001-5092	PCBD1	-			
1436	78.64	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
1437	78.62	cp	BRD-K06878038	deferiprone	Chelating agent		CYP4F2	Chelating agent
1438	78.58	kd	CGS001-22949	PTGR1	-			
1439	78.55	cp	BRD-A64297288	amlodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, ABCG2, CA1, CACNA1B, CACNA1S, CACNA2D3, CACNB1, CACNB2, SMPD1	Calcium channel blocker
1440	78.55	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
1441	78.42	kd	CGS001-3755	KCNG1	Voltage-gated potassium channels			
1442	78.37	kd	CGS001-53340	SPA17	-			
1443	78.37	kd	CGS001-1978	EIF4EBP1	-			
1444	78.35	kd	CGS001-285676	ZNF454	Zinc fingers, C2H2-type			
1445	78.34	oe	ccsbBroad304_08461	CDCA4	-			
1446	78.3	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
1447	78.29	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
1448	78.29	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
1449	78.28	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
1450	78.22	kd	CGS001-25942	SIN3A	-			
1451	78.2	kd	CGS001-3251	HPRT1	-			
1452	78.18	oe	ccsbBroad304_07363	AIFM1	-			
1453	78.17	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
1454	78.15	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
1455	78.14	kd	CGS001-1211	CLTA	-			
1456	78.09	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1457	78.02	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
1458	78.02	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
1459	77.97	oe	ccsbBroad304_06765	PRCC	-			
1460	77.97	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
1461	77.96	cc		Phospholipases GOF	-			
1462	77.94	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
1463	77.94	kd	CGS001-23530	NNT	-			
1464	77.93	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
1465	77.88	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
1466	77.88	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
1467	77.85	cp	BRD-K00532621	midazolam	Benzodiazepine receptor agonist		CYP3A5, CYP3A7, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3	Benzodiazepine receptor agonist
1468	77.82	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
1469	77.81	kd	CGS001-348	APOE	Apolipoproteins			
1470	77.8	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
1471	77.74	oe	ccsbBroad304_00709	GUK1	-			
1472	77.69	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
1473	77.67	cp	BRD-A92630576	trimebutine	Opioid receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Opioid receptor agonist
1474	77.67	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
1475	77.66	kd	CGS001-5950	RBP4	Lipocalins			
1476	77.65	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1477	77.58	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
1478	77.56	cp	BRD-A23637604	oxymetholone	Androgen receptor agonist		AR	Androgen receptor agonist
1479	77.54	oe	ccsbBroad304_02438	FAM3C	-			
1480	77.51	kd	CGS001-4801	NFYB	-			
1481	77.51	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
1482	77.5	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
1483	77.49	kd	CGS001-1488	CTBP2	-			
1484	77.49	kd	CGS001-8738	CRADD	-			
1485	77.48	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
1486	77.47	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
1487	77.44	oe	ccsbBroad304_01401	RIT1	-			
1488	77.43	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
1489	77.4	kd	CGS001-2931	GSK3A	GSK subfamily			
1490	77.39	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
1491	77.38	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
1492	77.37	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
1493	77.36	kd	CGS001-58477	SRPRB	-			
1494	77.34	kd	CGS001-283450	C12ORF51	-			
1495	77.33	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
1496	77.32	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
1497	77.32	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1498	77.13	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
1499	77.12	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
1500	77.1	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
1501	77.06	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
1502	77.02	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
1503	77.01	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
1504	76.88	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
1505	76.86	kd	CGS001-26993	AKAP8L	-			
1506	76.85	kd	CGS001-6723	SRM	-			
1507	76.84	oe	ccsbBroad304_03118	NRBP1	NRBP family			
1508	76.81	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
1509	76.79	kd	CGS001-9929	JOSD1	-			
1510	76.79	kd	CGS001-1616	DAXX	-			
1511	76.76	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
1512	76.74	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
1513	76.71	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
1514	76.7	kd	CGS001-4245	MGAT1	-			
1515	76.69	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
1516	76.67	kd	CGS001-2966	GTF2H2	General transcription factors			
1517	76.65	cc		Androgen receptor modulator	-			
1518	76.62	kd	CGS001-10094	ARPC3	Actin related protein 2/3 complex subunits			
1519	76.56	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
1520	76.48	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
1521	76.46	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
1522	76.39	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
1523	76.35	kd	CGS001-2037	EPB41L2	-			
1524	76.33	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
1525	76.26	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
1526	76.22	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
1527	76.22	kd	CGS001-79733	E2F8	-			
1528	76.22	kd	CGS001-10589	DRAP1	-			
1529	76.17	kd	CGS001-8834	TMEM11	-			
1530	76.15	kd	CGS001-23274	CLEC16A	C-type lectin domain containing			
1531	76.15	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
1532	76.04	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
1533	76.01	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
1534	75.9	kd	CGS001-7485	WRB	-			
1535	75.85	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
1536	75.84	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
1537	75.81	kd	CGS001-3199	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
1538	75.74	kd	CGS001-5033	P4HA1	-			
1539	75.73	kd	CGS001-718	C3	Endogenous ligands			
1540	75.72	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
1541	75.69	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
1542	75.69	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1543	75.68	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
1544	75.66	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
1545	75.55	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
1546	75.55	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
1547	75.54	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
1548	75.5	kd	CGS001-342926	ZNF677	Zinc fingers, C2H2-type			
1549	75.42	kd	CGS001-205	AK4	Adenylate kinases			
1550	75.42	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
1551	75.38	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
1552	75.37	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
1553	75.36	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
1554	75.35	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
1555	75.33	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
1556	75.32	kd	CGS001-5723	PSPH	-			
1557	75.25	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
1558	75.25	kd	CGS001-3476	IGBP1	-			
1559	75.23	oe	ccsbBroad304_06462	ITGAE	Integrins			
1560	75.23	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
1561	75.17	kd	CGS001-1975	EIF4B	RNA binding motif (RRM) containing			
1562	75.17	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
1563	75.15	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
1564	75.12	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
1565	75.07	oe	ccsbBroad304_02884	POT1	-			
1566	75.04	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
1567	75.03	kd	CGS001-5045	FURIN	Subtilisin			
1568	75.01	kd	CGS001-6304	SATB1	Homeoboxes / CUT class			
1569	75	kd	CGS001-23369	PUM2	-			
1570	74.98	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
1571	74.96	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
1572	74.95	kd	CGS001-9531	BAG3	-			
1573	74.93	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
1574	74.93	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
1575	74.92	oe	ccsbBroad304_06290	GNA15	-			
1576	74.92	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
1577	74.85	kd	CGS001-8453	CUL2	-			
1578	74.78	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
1579	74.75	cc		Targets of VEGFR inhibitors GOF	-			
1580	74.75	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
1581	74.6	cp	BRD-K44779798	miglitol	Glucosidase inhibitor		GAA, MGAM, GANAB, GANC, SLC5A4	Glucosidase inhibitor
1582	74.59	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
1583	74.59	kd	CGS001-7024	TFCP2	-			
1584	74.56	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
1585	74.53	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
1586	74.52	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
1587	74.49	kd	CGS001-54899	PXK	Slob family			
1588	74.47	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1589	74.47	kd	CGS001-8193	DPF1	Zinc fingers, PHD-type			
1590	74.45	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
1591	74.42	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
1592	74.4	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1593	74.39	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
1594	74.39	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1595	74.29	kd	CGS001-1605	DAG1	-			
1596	74.23	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1597	74.2	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
1598	74.2	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
1599	74.18	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
1600	74.14	kd	CGS001-57154	SMURF1	-			
1601	74.12	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
1602	74.1	cc		G2 M Checkpoint LOF	-			
1603	74.03	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
1604	74.01	oe	ccsbBroad304_06745	PNN	-			
1605	74	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
1606	73.94	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1607	73.89	oe	ccsbBroad304_02534	UTP14A	-			
1608	73.85	kd	CGS001-7534	YWHAZ	-			
1609	73.81	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
1610	73.81	kd	CGS001-8569	MKNK1	MKN subfamily			
1611	73.78	cc		P38 MAPK inhibitor	-			
1612	73.78	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
1613	73.77	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
1614	73.76	kd	CGS001-5987	TRIM27	-			
1615	73.75	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
1616	73.72	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
1617	73.71	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1618	73.67	oe	ccsbBroad304_02219	MORF4L2	-			
1619	73.67	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
1620	73.67	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1621	73.65	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
1622	73.65	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
1623	73.63	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
1624	73.62	oe	ccsbBroad304_06862	RGS3	-			
1625	73.62	kd	CGS001-55120	FANCL	Fanconi anemia, complementation groups			
1626	73.61	cp	BRD-K94649603	taxifolin	Opioid receptor antagonist		APOB, APP, HMGCR	Opioid receptor antagonist
1627	73.6	kd	CGS001-10456	HAX1	-			
1628	73.59	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
1629	73.56	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
1630	73.5	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
1631	73.48	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
1632	73.48	kd	CGS001-5423	POLB	DNA polymerases			
1633	73.47	kd	CGS001-3560	IL2RB	IL-2 receptor family			
1634	73.45	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
1635	73.45	kd	CGS001-2160	F11	Chymotrypsin			
1636	73.44	kd	CGS001-23509	POFUT1	Fucosyltransferases			
1637	73.43	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
1638	73.41	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
1639	73.41	kd	CGS001-11200	CHEK2	CHK1 subfamily			
1640	73.4	kd	CGS001-11212	PROSC	-			
1641	73.37	kd	CGS001-124583	CANT1	-			
1642	73.32	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
1643	73.32	kd	CGS001-23102	TBC1D2B	-			
1644	73.3	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1645	73.24	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
1646	73.23	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
1647	73.21	oe	ccsbBroad304_07766	RASSF1	-			
1648	73.21	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
1649	73.21	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
1650	73.15	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
1651	73.08	kd	CGS001-55226	NAT10	-			
1652	73.07	kd	CGS001-25797	QPCT	Aminopeptidase Y			
1653	73.07	kd	CGS001-50865	HEBP1	Endogenous ligands			
1654	73.06	kd	CGS001-5230	PGK1	-			
1655	73	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
1656	72.95	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
1657	72.94	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
1658	72.93	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
1659	72.91	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
1660	72.9	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
1661	72.89	cp	BRD-K82109576	vincristine	Tubulin inhibitor		TUBB, TUBA4A	Tubulin inhibitor
1662	72.87	kd	CGS001-5048	PAFAH1B1	WD repeat domain containing			
1663	72.85	cc		Cyclooxygenase inhibitor	-			
1664	72.81	kd	CGS001-8566	PDXK	-			
1665	72.8	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
1666	72.8	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
1667	72.79	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
1668	72.77	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
1669	72.76	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
1670	72.76	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
1671	72.74	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
1672	72.7	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
1673	72.69	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
1674	72.67	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
1675	72.65	oe	ccsbBroad304_00282	CDKN1A	-			
1676	72.65	kd	CGS001-6894	TARBP1	-			
1677	72.65	kd	CGS001-22796	COG2	Components of oligomeric golgi complex			
1678	72.59	oe	ccsbBroad304_02203	MAD2L1BP	-			
1679	72.57	kd	CGS001-5194	PEX13	-			
1680	72.56	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
1681	72.56	kd	CGS001-29888	STRN4	WD repeat domain containing			
1682	72.56	kd	CGS001-831	CAST	-			
1683	72.56	kd	CGS001-111	ADCY5	Adenylate cyclases			
1684	72.54	kd	CGS001-51014	TMED7	-			
1685	72.53	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
1686	72.51	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
1687	72.47	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
1688	72.45	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1689	72.42	kd	CGS001-388	RHOB	-			
1690	72.41	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
1691	72.4	oe	ccsbBroad304_08840	KIF9	Kinesins			
1692	72.4	kd	CGS001-10237	SLC35B1	SLC35 family of nucleotide sugar transporters			
1693	72.39	kd	CGS001-717	C2	Complement system			
1694	72.38	kd	CGS001-56848	SPHK2	Sphingosine kinase			
1695	72.32	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
1696	72.3	kd	CGS001-6927	HNF1A	Homeoboxes / HNF class			
1697	72.28	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
1698	72.23	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
1699	72.18	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
1700	72.17	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
1701	72.1	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1702	72.07	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
1703	72.02	kd	CGS001-51466	EVL	-			
1704	72.01	oe	ccsbBroad304_00394	CTSD	Cathepsins			
1705	72	kd	CGS001-1045	CDX2	Homeoboxes / ANTP class : HOXL subclass			
1706	71.97	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
1707	71.91	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
1708	71.87	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1709	71.83	oe	ccsbBroad304_06845	RARRES3	-			
1710	71.83	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
1711	71.76	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
1712	71.76	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
1713	71.71	oe	ccsbBroad304_06098	DHCR24	-			
1714	71.71	cp	BRD-A43082555	loxoprofen	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
1715	71.66	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
1716	71.65	kd	CGS001-6812	STXBP1	-			
1717	71.65	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
1718	71.62	kd	CGS001-571	BACH1	BTB/POZ domain containing			
1719	71.56	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
1720	71.55	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
1721	71.55	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
1722	71.53	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
1723	71.5	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
1724	71.49	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
1725	71.41	kd	CGS001-54541	DDIT4	-			
1726	71.33	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
1727	71.32	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1728	71.32	kd	CGS001-6603	SMARCD2	-			
1729	71.29	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
1730	71.29	kd	CGS001-4047	LSS	Lanosterol biosynthesis pathway			
1731	71.22	oe	ccsbBroad304_00949	LRPAP1	-			
1732	71.18	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
1733	71.02	oe	ccsbBroad304_07267	PDLIM4	-			
1734	71	cp	BRD-K52080565	rilmenidine	Imidazoline receptor agonist		NISCH	Imidazoline receptor agonist
1735	70.97	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
1736	70.96	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
1737	70.93	kd	CGS001-1879	EBF1	-			
1738	70.88	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
1739	70.87	oe	ccsbBroad304_02231	USP6NL	-			
1740	70.85	kd	CGS001-6259	RYK	Type XV RTKs: RYK			
1741	70.83	kd	CGS001-10857	PGRMC1	-			
1742	70.82	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
1743	70.81	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
1744	70.81	kd	CGS001-5105	PCK1	-			
1745	70.79	kd	CGS001-25966	C2CD2	-			
1746	70.77	oe	ccsbBroad304_07128	VHL	-			
1747	70.77	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
1748	70.74	kd	CGS001-1844	DUSP2	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1749	70.73	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
1750	70.65	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
1751	70.64	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
1752	70.62	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
1753	70.58	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
1754	70.56	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
1755	70.55	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
1756	70.55	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
1757	70.55	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
1758	70.53	kd	CGS001-54881	TEX10	-			
1759	70.53	kd	CGS001-2101	ESRRA	Estrogen-related receptors			
1760	70.52	oe	ccsbBroad304_06574	MDH2	-			
1761	70.46	oe	ccsbBroad304_05135	PARP15	-			
1762	70.46	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
1763	70.45	oe	ccsbBroad304_07124	UROD	-			
1764	70.41	oe	ccsbBroad304_05183	TXLNA	-			
1765	70.33	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
1766	70.32	kd	CGS001-10845	CLPX	ATPases / AAA-type			
1767	70.26	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
1768	70.24	kd	CGS001-170463	SSBP4	-			
1769	70.19	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
1770	70.16	cp	BRD-K73991644	isoquercetin	Aldose reductase inhibitor		AKR1B1, ACE	Aldose reductase inhibitor
1771	70.15	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
1772	70.06	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1773	70.03	cp	BRD-K44353683	nateglinide	Insulin secretagogue		ABCC8, KCNJ11, CYP3A4, INS, KCNJ10, PPARG	Insulin secretagogue
1774	70	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1775	69.97	kd	CGS001-4781	NFIB	-			
1776	69.93	oe	ccsbBroad304_01052	MYB	-			
1777	69.86	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
1778	69.85	oe	ccsbBroad304_00652	GNAS	-			
1779	69.85	kd	CGS001-23030	KDM4B	Histone demethylases			
1780	69.84	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
1781	69.8	kd	CGS001-9854	C2CD2L	-			
1782	69.79	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
1783	69.77	kd	CGS001-23466	CBX6	-			
1784	69.76	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
1785	69.76	kd	CGS001-1119	CHKA	-			
1786	69.75	kd	CGS001-10084	PQBP1	-			
1787	69.75	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
1788	69.72	kd	CGS001-6598	SMARCB1	-			
1789	69.67	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
1790	69.66	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
1791	69.66	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
1792	69.65	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
1793	69.6	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
1794	69.6	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
1795	69.57	oe	ccsbBroad304_07411	LPXN	-			
1796	69.54	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
1797	69.51	oe	ccsbBroad304_02581	ASCC3	-			
1798	69.49	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
1799	69.38	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
1800	69.37	kd	CGS001-54623	PAF1	-			
1801	69.32	oe	ccsbBroad304_00100	RHOA	-			
1802	69.3	oe	ccsbBroad304_02086	PDLIM1	-			
1803	69.28	kd	CGS001-4869	NPM1	-			
1804	69.28	kd	CGS001-133690	CAPSL	EF-hand domain containing			
1805	69.24	kd	CGS001-80025	PANK2	-			
1806	69.21	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
1807	69.19	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
1808	69.19	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
1809	69.18	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
1810	69.12	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
1811	69.11	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
1812	69.1	oe	ccsbBroad304_03910	CCDC90A	-			
1813	69.04	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
1814	69	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
1815	68.99	kd	CGS001-1066	CES1	Carboxylesterases			
1816	68.98	kd	CGS001-55832	CAND1	-			
1817	68.97	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
1818	68.93	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
1819	68.93	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
1820	68.92	kd	CGS001-10314	LANCL1	-			
1821	68.91	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
1822	68.88	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
1823	68.87	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
1824	68.83	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
1825	68.75	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
1826	68.74	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
1827	68.55	oe	ccsbBroad304_01203	PIM1	PIM family			
1828	68.54	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1829	68.53	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
1830	68.53	kd	CGS001-3672	ITGA1	Integrins			
1831	68.5	kd	CGS001-80714	PBX4	Homeoboxes / TALE class			
1832	68.48	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
1833	68.44	kd	CGS001-56916	SMARCAD1	-			
1834	68.43	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
1835	68.42	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
1836	68.41	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
1837	68.4	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
1838	68.37	cp	BRD-K13664374	dichloroacetic-acid	Pyruvate dehydrogenase kinase inhibitor		PDK1	Pyruvate dehydrogenase kinase inhibitor
1839	68.36	kd	CGS001-63892	THADA	-			
1840	68.23	kd	CGS001-6464	SHC1	SH2 domain containing			
1841	68.22	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
1842	68.16	kd	CGS001-1534	CYB561	Cytochrome b genes			
1843	68.14	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
1844	68.12	cc		Glycogen synthase kinase inhibitor	-			
1845	68.12	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
1846	68.07	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
1847	68.07	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
1848	68.06	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
1849	68.02	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
1850	67.93	cc		Calcium channel blocker	-			
1851	67.91	kd	CGS001-2745	GLRX	-			
1852	67.84	kd	CGS001-1719	DHFR	Oxidoreductases			
1853	67.8	kd	CGS001-1869	E2F1	-			
1854	67.77	kd	CGS001-54749	EPDR1	-			
1855	67.76	oe	ccsbBroad304_03420	TOLLIP	-			
1856	67.73	kd	CGS001-8313	AXIN2	-			
1857	67.72	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
1858	67.71	kd	CGS001-178	AGL	-			
1859	67.66	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
1860	67.62	oe	ccsbBroad304_05980	CDKN1B	-			
1861	67.62	kd	CGS001-55718	POLR3E	RNA polymerase subunits			
1862	67.6	kd	CGS001-5688	PSMA7	Proteasome subunits			
1863	67.55	kd	CGS001-9519	TBPL1	-			
1864	67.47	kd	CGS001-10112	KIF20A	Kinesins			
1865	67.4	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
1866	67.4	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
1867	67.37	kd	CGS001-3998	LMAN1	-			
1868	67.36	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1869	67.33	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
1870	67.32	kd	CGS001-25	ABL1	Abl family			
1871	67.31	kd	CGS001-8089	YEATS4	-			
1872	67.27	kd	CGS001-11041	B3GNT1	-			
1873	67.24	kd	CGS001-1314	COPA	Endogenous ligands			
1874	67.23	kd	CGS001-10494	STK25	YSK subfamily			
1875	67.16	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
1876	67.16	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
1877	67.15	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
1878	67.1	oe	ccsbBroad304_12226	NAGK	-			
1879	67.09	oe	ccsbBroad304_02869	ASF1A	-			
1880	67.09	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
1881	67.07	kd	CGS001-9252	RPS6KA5	MSK subfamily			
1882	67.02	kd	CGS001-56139	PCDHA10	Cadherins / Protocadherins : Clustered			
1883	67	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
1884	66.98	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
1885	66.93	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
1886	66.88	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
1887	66.87	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
1888	66.86	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1889	66.86	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
1890	66.83	kd	CGS001-6696	SPP1	Endogenous ligands			
1891	66.82	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
1892	66.81	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
1893	66.79	kd	CGS001-7004	TEAD4	-			
1894	66.77	kd	CGS001-10987	COPS5	-			
1895	66.73	cc		CCK receptor antagonist	-			
1896	66.71	oe	ccsbBroad304_08346	COQ3	-			
1897	66.68	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
1898	66.64	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
1899	66.61	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
1900	66.59	kd	CGS001-25793	FBXO7	F-boxes / other			
1901	66.57	kd	CGS001-11164	NUDT5	Nudix motif containing			
1902	66.52	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
1903	66.49	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
1904	66.46	oe	ccsbBroad304_07511	KIF14	Kinesins			
1905	66.44	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1906	66.43	oe	ccsbBroad304_02756	RRP8	-			
1907	66.42	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
1908	66.42	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
1909	66.39	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
1910	66.31	oe	ccsbBroad304_02094	FIBP	-			
1911	66.27	kd	CGS001-11340	EXOSC8	-			
1912	66.27	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
1913	66.24	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
1914	66.24	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
1915	66.21	cc		Lipocalins GOF	-			
1916	66.2	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
1917	66.16	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
1918	66.16	kd	CGS001-8576	STK16	NAK family			
1919	66.15	oe	ccsbBroad304_07252	DGKZ	-			
1920	66.13	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
1921	66.08	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
1922	66.06	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
1923	66.06	kd	CGS001-5163	PDK1	-			
1924	65.99	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
1925	65.94	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
1926	65.94	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
1927	65.92	kd	CGS001-813	CALU	EF-hand domain containing			
1928	65.9	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
1929	65.87	oe	ccsbBroad304_00964	SMAD7	SMADs			
1930	65.84	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
1931	65.83	oe	ccsbBroad304_02605	PAPD7	-			
1932	65.82	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
1933	65.78	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
1934	65.66	oe	ccsbBroad304_07808	RAB11FIP2	-			
1935	65.64	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
1936	65.63	oe	ccsbBroad304_00549	FDX1	-			
1937	65.62	kd	CGS001-55012	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1938	65.62	kd	CGS001-3029	HAGH	-			
1939	65.61	oe	ccsbBroad304_08104	MED4	-			
1940	65.6	kd	CGS001-64087	MCCC2	-			
1941	65.56	kd	CGS001-79143	MBOAT7	-			
1942	65.52	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
1943	65.5	kd	CGS001-2950	GSTP1	Glutathione S-transferases			
1944	65.47	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
1945	65.44	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
1946	65.36	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
1947	65.33	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
1948	65.28	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
1949	65.21	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
1950	65.16	kd	CGS001-34	ACADM	-			
1951	65.15	kd	CGS001-2348	FOLR1	-			
1952	65.14	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
1953	65.14	kd	CGS001-1676	DFFA	-			
1954	65.12	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
1955	65.09	oe	ccsbBroad304_00033	ADSS	-			
1956	65.03	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
1957	65.03	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
1958	64.98	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
1959	64.98	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
1960	64.97	oe	ccsbBroad304_02566	MORF4L1	-			
1961	64.96	kd	CGS001-286075	ZNF707	Zinc fingers, C2H2-type			
1962	64.9	kd	CGS001-58508	MLL3	-			
1963	64.88	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
1964	64.73	kd	CGS001-8837	CFLAR	Endogenous ligands			
1965	64.7	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
1966	64.67	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
1967	64.67	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
1968	64.66	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
1969	64.65	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
1970	64.59	oe	ccsbBroad304_07515	GFPT2	-			
1971	64.56	oe	ccsbBroad304_07528	DMTF1	-			
1972	64.53	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
1973	64.5	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
1974	64.48	kd	CGS001-9290	GPR55	GPCR / Class A : Orphans			
1975	64.44	kd	CGS001-558	AXL	Fibronectin type III domain containing			
1976	64.43	kd	CGS001-6884	TAF13	-			
1977	64.39	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
1978	64.37	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
1979	64.36	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
1980	64.36	kd	CGS001-149428	BNIPL	-			
1981	64.28	oe	ccsbBroad304_04752	IKBIP	-			
1982	64.27	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
1983	64.22	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
1984	64.22	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
1985	64.17	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1986	64.13	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
1987	64.12	cp	BRD-K96740444	itopride	Dopamine receptor antagonist		DRD2, ACHE, CHRM3	Dopamine receptor antagonist
1988	64.06	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
1989	64.04	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
1990	64.03	cc		Na-K-Cl transporter inhibitor	-			
1991	64.02	cc		C2 domain containing protein kinases LOF	-			
1992	63.98	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
1993	63.97	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
1994	63.92	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
1995	63.91	kd	CGS001-8859	STK19	G11 family			
1996	63.9	kd	CGS001-51005	AMDHD2	-			
1997	63.87	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1998	63.86	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
1999	63.85	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
2000	63.78	oe	ccsbBroad304_02026	NRP1	CD molecules			
2001	63.76	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
2002	63.75	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
2003	63.74	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
2004	63.71	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
2005	63.68	kd	CGS001-9784	SNX17	Sorting nexins			
2006	63.64	kd	CGS001-4012	LNPEP	Aminopeptidase N			
2007	63.63	oe	ccsbBroad304_06301	GOT2	-			
2008	63.5	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
2009	63.46	oe	ccsbBroad304_08775	SQRDL	-			
2010	63.46	kd	CGS001-5538	PPT1	-			
2011	63.45	cc		Ubiquitin-specific peptidases LOF	-			
2012	63.43	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
2013	63.43	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
2014	63.42	oe	ccsbBroad304_03573	BRF2	-			
2015	63.42	kd	CGS001-2634	GBP2	-			
2016	63.38	kd	CGS001-5562	PRKAA1	AMPK subfamily			
2017	63.33	kd	CGS001-328	APEX1	-			
2018	63.28	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
2019	63.24	kd	CGS001-3956	LGALS1	Endogenous ligands			
2020	63.23	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
2021	63.19	kd	CGS001-150280	HORMAD2	-			
2022	63.18	kd	CGS001-81577	GFOD2	-			
2023	63.17	kd	CGS001-51347	TAOK3	TAO subfamily			
2024	63.15	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
2025	63.14	kd	CGS001-8495	PPFIBP2	Sterile alpha motif (SAM) domain containing			
2026	63.1	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
2027	63.07	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
2028	63.07	kd	CGS001-11014	KDELR2	-			
2029	63.06	oe	ccsbBroad304_01184	PGK1	-			
2030	63.02	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
2031	62.99	kd	CGS001-6193	RPS5	S ribosomal proteins			
2032	62.97	cc		HRH1 antagonist	-			
2033	62.97	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
2034	62.96	oe	ccsbBroad304_02677	PDAP1	-			
2035	62.94	kd	CGS001-6788	STK3	MST subfamily			
2036	62.91	kd	CGS001-840	CASP7	Caspases			
2037	62.9	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
2038	62.86	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
2039	62.85	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
2040	62.83	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
2041	62.82	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
2042	62.8	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
2043	62.79	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
2044	62.73	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
2045	62.72	kd	CGS001-9512	PMPCB	-			
2046	62.69	kd	CGS001-3169	FOXA1	Forkhead boxes			
2047	62.68	kd	CGS001-9632	SEC24C	-			
2048	62.58	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
2049	62.57	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
2050	62.48	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
2051	62.42	oe	ccsbBroad304_06458	IRF3	-			
2052	62.42	kd	CGS001-80237	ELL3	-			
2053	62.42	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
2054	62.39	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
2055	62.35	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
2056	62.35	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
2057	62.31	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
2058	62.29	oe	ccsbBroad304_02163	MED7	-			
2059	62.27	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
2060	62.24	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
2061	62.23	kd	CGS001-2793	GNGT2	-			
2062	62.16	kd	CGS001-4602	MYB	-			
2063	62.15	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
2064	62.13	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
2065	62.12	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
2066	62.11	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
2067	62.1	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
2068	62.08	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
2069	62.07	cc		Cell Cycle Inhibition GOF	-			
2070	62.06	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
2071	62.06	kd	CGS001-2098	ESD	-			
2072	62.05	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
2073	62.03	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
2074	62.01	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
2075	61.99	cp	BRD-K96134740	kitasamycin	Protein synthesis inhibitor			Protein synthesis inhibitor
2076	61.98	kd	CGS001-8027	STAM	-			
2077	61.95	oe	ccsbBroad304_12008	NLK	nmo subfamily			
2078	61.92	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
2079	61.9	oe	ccsbBroad304_01769	VEGFB	-			
2080	61.9	kd	CGS001-84333	PCGF5	Polycomb group ring fingers			
2081	61.89	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
2082	61.88	cp	BRD-K07237224	moclobemide	Monoamine oxidase inhibitor		MAOA, CYP2C19, MAOB	Monoamine oxidase inhibitor
2083	61.87	kd	CGS001-3074	HEXB	-			
2084	61.83	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
2085	61.83	kd	CGS001-89766	UMODL1	-			
2086	61.67	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
2087	61.67	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
2088	61.6	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
2089	61.6	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
2090	61.6	kd	CGS001-823	CAPN1	EF-hand domain containing			
2091	61.57	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
2092	61.56	kd	CGS001-9441	MED26	-			
2093	61.53	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
2094	61.48	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
2095	61.42	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
2096	61.4	kd	CGS001-28511	NKIRAS2	-			
2097	61.39	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
2098	61.34	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
2099	61.29	oe	ccsbBroad304_02276	MVP	-			
2100	61.29	kd	CGS001-3032	HADHB	-			
2101	61.25	kd	CGS001-23244	PDS5A	-			
2102	61.23	cc		CDK inhibitor	-			
2103	61.2	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
2104	61.19	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
2105	61.19	kd	CGS001-6648	SOD2	-			
2106	61.13	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
2107	61.11	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
2108	61.06	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2109	61.03	kd	CGS001-604	BCL6	BTB/POZ domain containing			
2110	60.99	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
2111	60.9	cc		Progesterone receptor antagonist	-			
2112	60.86	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
2113	60.85	oe	ccsbBroad304_04038	ELOVL6	-			
2114	60.84	oe	ccsbBroad304_03933	CARD9	-			
2115	60.8	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
2116	60.77	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
2117	60.73	kd	CGS001-221188	GPR114	Adhesion Class GPCRs			
2118	60.7	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
2119	60.53	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
2120	60.47	kd	CGS001-3939	LDHA	-			
2121	60.41	kd	CGS001-80212	CCDC92	-			
2122	60.38	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
2123	60.36	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
2124	60.36	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
2125	60.35	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
2126	60.32	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
2127	60.31	cc		Aromatase inhibitor	-			
2128	60.31	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
2129	60.3	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
2130	60.27	kd	CGS001-1374	CPT1A	-			
2131	60.25	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
2132	60.17	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
2133	60.14	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
2134	60.14	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
2135	60.12	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
2136	60.12	kd	CGS001-23670	TMEM2	-			
2137	60.1	kd	CGS001-2534	FYN	Src family			
2138	60.09	oe	ccsbBroad304_02271	LPGAT1	-			
2139	60.05	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
2140	60.05	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
2141	60	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
2142	60	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
2143	59.96	cc		Interleukins GOF	-			
2144	59.96	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
2145	59.92	oe	ccsbBroad304_03858	SRPRB	-			
2146	59.88	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
2147	59.84	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
2148	59.81	kd	CGS001-55107	ANO1	Calcium activated chloride channel			
2149	59.8	oe	ccsbBroad304_03604	ENOSF1	-			
2150	59.77	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
2151	59.74	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
2152	59.73	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
2153	59.73	kd	CGS001-1026	CDKN1A	-			
2154	59.7	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
2155	59.67	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
2156	59.67	kd	CGS001-23523	CABIN1	-			
2157	59.63	kd	CGS001-6601	SMARCC2	-			
2158	59.63	kd	CGS001-5860	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
2159	59.62	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
2160	59.59	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
2161	59.57	kd	CGS001-4707	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
2162	59.56	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
2163	59.55	kd	CGS001-2280	FKBP1A	Cis-trans-isomerases			
2164	59.5	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
2165	59.5	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
2166	59.5	kd	CGS001-1490	CTGF	-			
2167	59.48	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
2168	59.46	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
2169	59.45	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
2170	59.45	kd	CGS001-25842	ASF1A	-			
2171	59.44	kd	CGS001-7528	YY1	INO80 complex subunits			
2172	59.43	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
2173	59.42	oe	ccsbBroad304_00661	GNGT2	-			
2174	59.4	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
2175	59.39	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
2176	59.38	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
2177	59.35	cp	BRD-K43236057	piceid	ICAM1 inhibitor		GAA, XDH	ICAM1 inhibitor
2178	59.33	kd	CGS001-1386	ATF2	basic leucine zipper proteins			
2179	59.32	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
2180	59.29	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
2181	59.16	cc		Wnt family GOF	-			
2182	59.05	kd	CGS001-2155	F7	Chymotrypsin			
2183	59.01	oe	ccsbBroad304_02837	BHMT2	-			
2184	59	oe	ccsbBroad304_02313	ACTR3	-			
2185	58.97	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
2186	58.94	oe	ccsbBroad304_01394	RFX4	-			
2187	58.94	oe	ccsbBroad304_00237	CCND3	-			
2188	58.94	kd	CGS001-9871	SEC24D	-			
2189	58.93	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
2190	58.92	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
2191	58.9	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
2192	58.9	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
2193	58.89	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
2194	58.87	kd	CGS001-4664	NAB1	-			
2195	58.83	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
2196	58.83	kd	CGS001-25989	ULK3	Unc-51-like kinase (ULK) family			
2197	58.77	kd	CGS001-56731	SLC2A4RG	-			
2198	58.74	kd	CGS001-6257	RXRB	Retinoid X receptors			
2199	58.73	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
2200	58.71	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
2201	58.7	kd	CGS001-10482	NXF1	-			
2202	58.69	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
2203	58.69	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
2204	58.69	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
2205	58.68	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
2206	58.68	kd	CGS001-8635	RNASET2	-			
2207	58.67	kd	CGS001-2990	GUSB	-			
2208	58.66	kd	CGS001-79187	FSD1	Fibronectin type III domain containing			
2209	58.65	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
2210	58.65	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
2211	58.63	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
2212	58.62	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
2213	58.6	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
2214	58.59	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
2215	58.55	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
2216	58.52	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
2217	58.51	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
2218	58.5	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2219	58.5	kd	CGS001-3163	HMOX2	Haem oxygenase			
2220	58.49	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
2221	58.48	kd	CGS001-23636	NUP62	-			
2222	58.47	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
2223	58.42	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2224	58.33	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
2225	58.31	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
2226	58.29	kd	CGS001-10472	ZNF238	-			
2227	58.28	kd	CGS001-7486	WRN	-			
2228	58.23	kd	CGS001-5245	PHB	-			
2229	58.22	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
2230	58.2	kd	CGS001-1431	CS	-			
2231	58.19	kd	CGS001-81544	GDPD5	-			
2232	58.18	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
2233	58.15	kd	CGS001-3708	ITPR1	Ion channels / Inositol triphosphate receptors			
2234	58.14	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
2235	58.13	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
2236	58.11	oe	ccsbBroad304_00795	HSF2	-			
2237	58.05	oe	ccsbBroad304_08879	CASD1	-			
2238	58.05	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
2239	57.99	kd	CGS001-23753	SDF2L1	-			
2240	57.98	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
2241	57.94	oe	ccsbBroad304_02834	GABARAPL1	-			
2242	57.87	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
2243	57.87	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
2244	57.85	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
2245	57.84	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
2246	57.83	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
2247	57.82	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
2248	57.78	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
2249	57.72	kd	CGS001-857	CAV1	-			
2250	57.71	oe	ccsbBroad304_01379	RBBP6	-			
2251	57.7	kd	CGS001-57504	MTA3	GATA zinc finger domain containing			
2252	57.68	cp	BRD-K53220666	trimetozine	Sedative			Sedative
2253	57.65	oe	ccsbBroad304_00738	HINT1	-			
2254	57.65	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
2255	57.64	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
2256	57.63	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
2257	57.61	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2258	57.59	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
2259	57.55	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
2260	57.51	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
2261	57.5	oe	ccsbBroad304_05439	O3FAR1	-			
2262	57.48	oe	ccsbBroad304_07491	IP6K1	-			
2263	57.44	kd	CGS001-3897	L1CAM	CD molecules			
2264	57.44	kd	CGS001-10142	AKAP9	A-kinase anchor proteins			
2265	57.41	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
2266	57.38	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
2267	57.37	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
2268	57.32	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
2269	57.28	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
2270	57.27	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
2271	57.27	kd	CGS001-8505	PARG	-			
2272	57.26	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
2273	57.22	oe	ccsbBroad304_02052	KYNU	-			
2274	57.18	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
2275	57.1	kd	CGS001-375133	PI4KAP2	-			
2276	57.08	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
2277	57.08	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
2278	57.06	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
2279	57.03	cc		Dihydrofolate reductase inhibitor	-			
2280	57.03	kd	CGS001-7965	AIMP2	-			
2281	56.98	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
2282	56.96	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
2283	56.95	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
2284	56.95	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
2285	56.86	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
2286	56.79	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
2287	56.78	oe	ccsbBroad304_02345	TXNDC9	-			
2288	56.73	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
2289	56.73	kd	CGS001-2184	FAH	-			
2290	56.72	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
2291	56.72	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
2292	56.7	kd	CGS001-57167	SALL4	Zinc fingers, C2H2-type			
2293	56.65	kd	CGS001-3589	IL11	Endogenous ligands			
2294	56.62	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
2295	56.56	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
2296	56.55	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
2297	56.55	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
2298	56.51	kd	CGS001-81533	ITFG1	-			
2299	56.4	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
2300	56.38	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
2301	56.35	oe	ccsbBroad304_02804	KLHDC2	-			
2302	56.32	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
2303	56.27	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
2304	56.27	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
2305	56.25	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2306	56.24	kd	CGS001-4194	MDM4	-			
2307	56.16	oe	ccsbBroad304_02801	CASP14	Caspases			
2308	56.13	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
2309	56.13	cp	BRD-A52282606	lacidipine	Calcium channel blocker		CACNA1C	Calcium channel blocker
2310	56.08	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
2311	56.06	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
2312	56.04	oe	ccsbBroad304_03047	BZW2	-			
2313	56.02	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
2314	56.01	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
2315	55.99	kd	CGS001-2203	FBP1	-			
2316	55.95	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
2317	55.89	kd	CGS001-55869	HDAC8	Histone deacetylases			
2318	55.87	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
2319	55.87	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
2320	55.86	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
2321	55.84	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
2322	55.83	oe	ccsbBroad304_04406	PLA2G12B	-			
2323	55.83	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
2324	55.78	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
2325	55.77	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
2326	55.77	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
2327	55.76	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
2328	55.72	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
2329	55.71	kd	CGS001-5567	PRKACB	Protein kinase A			
2330	55.71	kd	CGS001-7919	DDX39B	DEAD-boxes			
2331	55.67	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
2332	55.67	kd	CGS001-5591	PRKDC	Other PIKK family kinases			
2333	55.67	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
2334	55.66	kd	CGS001-54788	DNAJB12	Heat shock proteins / DNAJ (HSP40)			
2335	55.61	oe	ccsbBroad304_02058	PLOD3	-			
2336	55.57	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
2337	55.57	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
2338	55.57	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
2339	55.57	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
2340	55.53	kd	CGS001-9868	TOMM70A	Tetratricopeptide (TTC) repeat domain containing			
2341	55.51	kd	CGS001-51172	NAGPA	-			
2342	55.5	oe	ccsbBroad304_02484	PAICS	-			
2343	55.45	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
2344	55.44	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
2345	55.44	kd	CGS001-79947	DHDDS	-			
2346	55.4	kd	CGS001-2243	FGA	Endogenous ligands			
2347	55.37	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
2348	55.34	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
2349	55.32	kd	CGS001-6932	TCF7	-			
2350	55.27	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
2351	55.2	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
2352	55.17	kd	CGS001-8833	GMPS	-			
2353	55.09	kd	CGS001-32	ACACB	Carboxylases			
2354	55.08	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
2355	55.07	kd	CGS001-7247	TSN	-			
2356	55.07	kd	CGS001-60	ACTB	-			
2357	55.05	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
2358	55.04	kd	CGS001-3601	IL15RA	IL-2 receptor family			
2359	55.01	kd	CGS001-5338	PLD2	Hydrolases			
2360	55	oe	ccsbBroad304_09195	MCM8	-			
2361	54.9	kd	CGS001-84775	ZNF607	Zinc fingers, C2H2-type			
2362	54.89	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
2363	54.88	kd	CGS001-2821	GPI	-			
2364	54.87	kd	CGS001-126208	ZNF787	Zinc fingers, C2H2-type			
2365	54.87	kd	CGS001-2021	ENDOG	-			
2366	54.86	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
2367	54.86	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
2368	54.84	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
2369	54.74	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
2370	54.74	kd	CGS001-7054	TH	Amino acid hydroxylases			
2371	54.74	kd	CGS001-5004	ORM1	Lipocalins			
2372	54.72	kd	CGS001-1376	CPT2	-			
2373	54.67	oe	ccsbBroad304_01519	SET	-			
2374	54.66	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
2375	54.64	cc		Calmodulin antagonist	-			
2376	54.63	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
2377	54.63	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
2378	54.62	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
2379	54.58	cp	BRD-K82795137	loratadine	Histamine receptor antagonist		HRH1, CYP2C19, CYP3A5	Histamine receptor antagonist
2380	54.51	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
2381	54.5	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
2382	54.47	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
2383	54.46	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
2384	54.43	oe	ccsbBroad304_03850	TRIB3	Trbl family			
2385	54.42	oe	ccsbBroad304_00020	ACY1	-			
2386	54.38	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
2387	54.33	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
2388	54.3	kd	CGS001-54861	SNRK	SNRK subfamily			
2389	54.24	kd	CGS001-9817	KEAP1	Kelch-like proteins			
2390	54.18	oe	ccsbBroad304_01166	PDK2	PDHK family			
2391	54.18	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
2392	54.15	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
2393	54.09	cc		Dopamine receptor antagonist	-			
2394	54.09	oe	ccsbBroad304_00231	CBFB	-			
2395	54.07	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
2396	54.02	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
2397	54	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
2398	53.99	kd	CGS001-9797	TATDN2	-			
2399	53.97	kd	CGS001-23710	GABARAPL1	-			
2400	53.94	oe	ccsbBroad304_07531	TANK	-			
2401	53.88	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
2402	53.85	kd	CGS001-140612	ZFP28	Zinc fingers, C2H2-type			
2403	53.82	kd	CGS001-29899	GPSM2	Tetratricopeptide (TTC) repeat domain containing			
2404	53.81	kd	CGS001-6050	RNH1	-			
2405	53.74	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
2406	53.74	kd	CGS001-9788	MTSS1	-			
2407	53.73	oe	ccsbBroad304_05907	BUB1B	Bub family			
2408	53.71	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
2409	53.68	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
2410	53.67	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
2411	53.55	oe	ccsbBroad304_00551	FECH	-			
2412	53.53	kd	CGS001-53343	NUDT9	Nudix motif containing			
2413	53.52	oe	ccsbBroad304_01672	TIMP2	-			
2414	53.51	kd	CGS001-3066	HDAC2	Histone deacetylases			
2415	53.5	oe	ccsbBroad304_00650	GNA11	-			
2416	53.49	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
2417	53.47	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
2418	53.46	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
2419	53.45	oe	ccsbBroad304_02485	STAMBP	-			
2420	53.45	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
2421	53.39	kd	CGS001-10452	TOMM40	-			
2422	53.37	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
2423	53.34	kd	CGS001-7421	VDR	Vitamin D receptors			
2424	53.34	kd	CGS001-51447	IP6K2	-			
2425	53.3	oe	ccsbBroad304_06538	LSP1	-			
2426	53.3	oe	ccsbBroad304_02671	ECD	-			
2427	53.24	kd	CGS001-6778	STAT6	SH2 domain containing			
2428	53.22	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
2429	53.22	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
2430	53.22	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
2431	53.18	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2432	53.15	kd	CGS001-147686	ZNF418	Zinc fingers, C2H2-type			
2433	53.11	kd	CGS001-151126	ZNF385B	-			
2434	53.09	cc		Apolipoproteins LOF	-			
2435	53.09	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
2436	53.07	kd	CGS001-7039	TGFA	-			
2437	53.07	kd	CGS001-347736	NME9	-			
2438	53.02	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
2439	52.99	cp	BRD-K57930253	nitrazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, SCN1A	Benzodiazepine receptor agonist
2440	52.95	kd	CGS001-5460	POU5F1	Homeoboxes / POU class			
2441	52.93	kd	CGS001-23013	SPEN	RNA binding motif (RRM) containing			
2442	52.93	kd	CGS001-6990	DYNLT3	Cytoplasmic dyneins			
2443	52.9	kd	CGS001-5894	RAF1	RAF family			
2444	52.87	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2445	52.87	kd	CGS001-81539	SLC38A1	System A-like transporters			
2446	52.86	kd	CGS001-1856	DVL2	Dishevelled homologs			
2447	52.85	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
2448	52.85	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
2449	52.82	kd	CGS001-57121	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2450	52.77	oe	ccsbBroad304_03097	CNOT7	-			
2451	52.76	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
2452	52.73	cc		MEK inhibitor	-			
2453	52.73	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
2454	52.69	kd	CGS001-29998	GLTSCR1	-			
2455	52.67	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
2456	52.64	oe	ccsbBroad304_01723	TTK	TTK family			
2457	52.64	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
2458	52.62	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
2459	52.6	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
2460	52.59	oe	ccsbBroad304_00489	EHHADH	-			
2461	52.59	kd	CGS001-84811	BUD13	-			
2462	52.57	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
2463	52.51	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
2464	52.5	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
2465	52.48	oe	ccsbBroad304_01560	SNAPC1	-			
2466	52.48	kd	CGS001-23566	LPAR3	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2467	52.46	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
2468	52.46	kd	CGS001-350	APOH	Apolipoproteins			
2469	52.45	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
2470	52.4	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
2471	52.39	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
2472	52.33	cp	BRD-K84566043	fenpiverinium	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
2473	52.27	cc		Integrin subunits alpha LOF	-			
2474	52.22	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
2475	52.2	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
2476	52.17	kd	CGS001-133522	PPARGC1B	RNA binding motif (RRM) containing			
2477	52.15	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
2478	52.14	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
2479	52.14	kd	CGS001-56889	TM9SF3	-			
2480	52.08	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2481	52.03	oe	ccsbBroad304_06739	PLOD1	-			
2482	52.03	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
2483	52.03	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2484	51.96	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
2485	51.91	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
2486	51.86	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
2487	51.86	cp	BRD-A96107863	nisoldipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNB2, CYP3A5	Calcium channel blocker
2488	51.84	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
2489	51.81	kd	CGS001-5898	RALA	-			
2490	51.8	cp	BRD-K86003836	flubendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
2491	51.77	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
2492	51.75	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
2493	51.74	kd	CGS001-10392	NOD1	Nucleotide-binding domain and leucine rich repeat containing			
2494	51.73	oe	ccsbBroad304_00854	IL8	-			
2495	51.72	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
2496	51.7	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
2497	51.68	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
2498	51.59	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2499	51.57	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
2500	51.56	kd	CGS001-5253	PHF2	Histone demethylases			
2501	51.56	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
2502	51.52	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
2503	51.52	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
2504	51.51	cp	BRD-K39983086	loteprednol	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Phospholipase inhibitor
2505	51.45	oe	ccsbBroad304_02287	GNPDA1	-			
2506	51.43	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
2507	51.4	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
2508	51.39	oe	ccsbBroad304_07561	YAF2	-			
2509	51.36	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
2510	51.36	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
2511	51.35	oe	ccsbBroad304_00747	HLF	-			
2512	51.33	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
2513	51.33	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
2514	51.28	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
2515	51.27	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
2516	51.26	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
2517	51.23	kd	CGS001-9453	GGPS1	Lanosterol biosynthesis pathway			
2518	51.21	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
2519	51.18	cp	BRD-K93618743	ipriflavone	Bone resorption inhibitor			Bone resorption inhibitor
2520	51.17	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
2521	51.16	kd	CGS001-3119	HLA-DQB1	Immunoglobulin superfamily / C1-set domain containing			
2522	51.15	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
2523	51.15	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
2524	51.15	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
2525	51.14	oe	ccsbBroad304_08152	PSAT1	-			
2526	51.13	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
2527	51.13	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
2528	51.13	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
2529	51.06	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
2530	51.06	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
2531	51.06	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
2532	51.04	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
2533	51.04	kd	CGS001-3608	ILF2	-			
2534	50.95	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
2535	50.95	kd	CGS001-8764	TNFRSF14	Tumour necrosis factor (TNF) receptor family			
2536	50.91	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
2537	50.9	kd	CGS001-29110	TBK1	IKK family			
2538	50.88	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
2539	50.8	kd	CGS001-5217	PFN2	-			
2540	50.79	oe	ccsbBroad304_07053	TFPI	-			
2541	50.79	oe	ccsbBroad304_01002	METTL1	-			
2542	50.78	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
2543	50.74	kd	CGS001-84515	MCM8	-			
2544	50.66	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
2545	50.64	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2546	50.63	oe	ccsbBroad304_04544	RCCD1	-			
2547	50.57	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2548	50.55	cp	BRD-K46435977	valaciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
2549	50.54	kd	CGS001-801	CALM1	EF-hand domain containing			
2550	50.49	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2551	50.48	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
2552	50.45	kd	CGS001-2673	GFPT1	-			
2553	50.38	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
2554	50.38	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
2555	50.38	kd	CGS001-637	BID	Endogenous ligands			
2556	50.37	cc		Purinergic receptors P2Y GOF	-			
2557	50.37	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
2558	50.35	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
2559	50.32	cc		FXR antagonist	-			
2560	50.28	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
2561	50.23	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
2562	50.22	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
2563	50.19	oe	ccsbBroad304_03696	C19ORF10	-			
2564	50.15	oe	ccsbBroad304_00183	C1S	Complement system			
2565	50.15	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
2566	50.13	oe	ccsbBroad304_01146	PARN	-			
2567	50.12	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
2568	50.1	kd	CGS001-9475	ROCK2	Pleckstrin homology (PH) domain containing			
2569	50.09	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
2570	50.07	kd	CGS001-30836	DNTTIP2	-			
2571	50.05	oe	ccsbBroad304_00239	CCNG1	-			
2572	50.05	kd	CGS001-51135	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
2573	50.04	kd	CGS001-7431	VIM	Intermediate filaments type III			
2574	50.02	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
2575	50	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
2576	49.95	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
2577	49.94	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
2578	49.94	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
2579	49.88	kd	CGS001-5594	MAPK1	MAPK:ERK subfamily			
2580	49.85	kd	CGS001-79960	PHF17	-			
2581	49.85	kd	CGS001-11154	AP4S1	-			
2582	49.84	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
2583	49.83	kd	CGS001-5654	HTRA1	Serine peptidases / Serine peptidases			
2584	49.8	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
2585	49.79	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
2586	49.78	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
2587	49.73	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
2588	49.73	kd	CGS001-54566	EPB41L4B	-			
2589	49.7	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
2590	49.69	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
2591	49.59	cc		GATA Zinc finger domain containing LOF	-			
2592	49.58	oe	ccsbBroad304_03164	MTERFD1	-			
2593	49.57	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
2594	49.57	kd	CGS001-4791	NFKB2	NFkappaB transcription factor family			
2595	49.47	kd	CGS001-10138	YAF2	-			
2596	49.46	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
2597	49.44	kd	CGS001-3376	IARS	Aminoacyl tRNA synthetases / Class I			
2598	49.44	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
2599	49.42	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2600	49.4	oe	ccsbBroad304_03056	MCTS1	-			
2601	49.36	oe	ccsbBroad304_00222	CASP6	Caspases			
2602	49.36	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
2603	49.27	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
2604	49.27	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2605	49.24	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
2606	49.22	oe	ccsbBroad304_07217	AXIN2	-			
2607	49.21	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
2608	49.18	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
2609	49.15	kd	CGS001-51684	SUFU	-			
2610	49.14	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
2611	49.14	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
2612	49.1	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
2613	49.09	kd	CGS001-54815	GATAD2A	GATA zinc finger domain containing			
2614	49.05	kd	CGS001-6829	SUPT5H	-			
2615	49.04	kd	CGS001-50604	IL20	Interleukins and interleukin receptors			
2616	49.03	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
2617	48.98	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
2618	48.86	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
2619	48.85	oe	ccsbBroad304_08802	ELAC2	-			
2620	48.82	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
2621	48.8	kd	CGS001-2618	GART	Ribosyl transferases			
2622	48.79	cc		Estrogen receptor antagonist	-			
2623	48.79	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
2624	48.75	oe	ccsbBroad304_00101	RHOC	-			
2625	48.75	kd	CGS001-3638	INSIG1	-			
2626	48.73	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
2627	48.71	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
2628	48.67	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
2629	48.65	kd	CGS001-597	BCL2A1	-			
2630	48.65	kd	CGS001-9131	AIFM1	-			
2631	48.64	kd	CGS001-51026	GOLT1B	-			
2632	48.63	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
2633	48.62	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
2634	48.56	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
2635	48.55	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
2636	48.51	oe	ccsbBroad304_07238	STK24	YSK subfamily			
2637	48.51	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
2638	48.47	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2639	48.44	oe	ccsbBroad304_06976	SMARCE1	-			
2640	48.43	kd	CGS001-29940	DSE	-			
2641	48.42	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
2642	48.41	kd	CGS001-7052	TGM2	Transglutaminases			
2643	48.39	kd	CGS001-7374	UNG	-			
2644	48.38	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
2645	48.34	kd	CGS001-5052	PRDX1	-			
2646	48.34	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
2647	48.33	oe	ccsbBroad304_03129	ERO1L	-			
2648	48.33	cp	BRD-K82147103	lofepramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
2649	48.3	kd	CGS001-4023	LPL	-			
2650	48.29	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
2651	48.21	cp	BRD-K60160658	tiagabine	GABA uptake inhibitor		SLC6A1, CYP2C19	GABA uptake inhibitor
2652	48.2	kd	CGS001-3664	IRF6	-			
2653	48.19	oe	ccsbBroad304_03961	SMURF2	-			
2654	48.18	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
2655	48.12	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
2656	48.11	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
2657	48.07	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
2658	48.06	oe	ccsbBroad304_07605	LYPLA1	-			
2659	48.03	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
2660	48.03	kd	CGS001-30	ACAA1	-			
2661	48.01	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2662	47.99	cc		Serotonin receptor agonist	-			
2663	47.97	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
2664	47.97	kd	CGS001-776	CACNA1D	Calcium channel subunits			
2665	47.92	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2666	47.91	kd	CGS001-1499	CTNNB1	Catenins			
2667	47.9	cc		Angiotensin receptor antagonist	-			
2668	47.89	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
2669	47.84	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
2670	47.83	kd	CGS001-5134	PDCD2	Zinc fingers, MYND-type			
2671	47.82	kd	CGS001-25925	ZNF521	Zinc fingers, C2H2-type			
2672	47.8	kd	CGS001-91949	COG7	Components of oligomeric golgi complex			
2673	47.78	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
2674	47.71	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
2675	47.7	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
2676	47.68	oe	ccsbBroad304_06287	GM2A	-			
2677	47.65	oe	ccsbBroad304_05756	ACAA1	-			
2678	47.65	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
2679	47.65	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
2680	47.65	kd	CGS001-51520	LARS	Aminoacyl tRNA synthetases / Class I			
2681	47.61	kd	CGS001-23242	COBL	-			
2682	47.6	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
2683	47.55	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
2684	47.53	kd	CGS001-9710	KIAA0355	-			
2685	47.53	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
2686	47.48	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
2687	47.47	cc		Vitamin D receptor agonist	-			
2688	47.47	cc		Benzodiazepine receptor agonist	-			
2689	47.41	kd	CGS001-51750	RTEL1	-			
2690	47.4	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
2691	47.33	kd	CGS001-7097	TLR2	Toll-like receptor family			
2692	47.32	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
2693	47.31	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
2694	47.29	kd	CGS001-1977	EIF4E	Translation Initiation Factor 4E			
2695	47.26	kd	CGS001-1611	DAP	-			
2696	47.26	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
2697	47.24	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
2698	47.23	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
2699	47.13	kd	CGS001-7018	TF	-			
2700	47.1	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
2701	47.08	kd	CGS001-808	CALM3	EF-hand domain containing			
2702	47.05	kd	CGS001-9134	CCNE2	-			
2703	47.04	oe	ccsbBroad304_02414	IRF9	-			
2704	47.03	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
2705	46.98	cp	BRD-K28849549	mesalazine	Cyclooxygenase inhibitor		PTGS1, PPARG, PTGS2, ALOX5, CHUK, CTNNB1, IKBKB, MPO, NAT1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor, Prostanoid receptor antagonist
2706	46.96	oe	ccsbBroad304_06136	ECHS1	-			
2707	46.92	oe	ccsbBroad304_02452	NXF1	-			
2708	46.91	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
2709	46.9	kd	CGS001-1763	DNA2	-			
2710	46.9	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
2711	46.87	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
2712	46.87	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2713	46.87	kd	CGS001-7187	TRAF3	-			
2714	46.84	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
2715	46.83	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
2716	46.83	kd	CGS001-27109	ATP5S	-			
2717	46.82	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
2718	46.81	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
2719	46.8	oe	ccsbBroad304_00212	CAMLG	-			
2720	46.77	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
2721	46.75	oe	ccsbBroad304_10487	BPHL	-			
2722	46.75	cp	BRD-K50938287	sumatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1A, HTR1F, HTR1E, HTR5A, HTR6, HTR7	Serotonin receptor agonist
2723	46.71	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
2724	46.64	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
2725	46.63	kd	CGS001-6790	AURKA	Aurora kinase			
2726	46.59	oe	ccsbBroad304_02017	PEX11A	-			
2727	46.59	kd	CGS001-944	TNFSF8	CD molecules			
2728	46.57	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
2729	46.53	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2730	46.51	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
2731	46.51	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
2732	46.5	oe	ccsbBroad304_08553	STAP2	-			
2733	46.5	kd	CGS001-5743	PTGS2	Cyclooxygenase			
2734	46.48	cp	BRD-A37052580	physostigmine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Cholinesterase inhibitor
2735	46.46	oe	ccsbBroad304_00552	FEN1	-			
2736	46.46	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
2737	46.44	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
2738	46.42	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
2739	46.41	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
2740	46.41	kd	CGS001-6713	SQLE	Lanosterol biosynthesis pathway			
2741	46.41	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
2742	46.39	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
2743	46.38	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
2744	46.34	cc		HIV protease inhibitor	-			
2745	46.32	oe	ccsbBroad304_01371	RALA	-			
2746	46.32	oe	ccsbBroad304_09354	IGSF8	CD molecules			
2747	46.31	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
2748	46.29	kd	CGS001-338557	O3FAR1	-			
2749	46.28	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
2750	46.28	kd	CGS001-1728	NQO1	-			
2751	46.25	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
2752	46.25	kd	CGS001-4709	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
2753	46.25	kd	CGS001-10523	CHERP	G patch domain containing			
2754	46.21	kd	CGS001-7345	UCHL1	Ubiquitin C-terminal hydrolase			
2755	46.19	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
2756	46.19	kd	CGS001-10401	PIAS3	Zinc fingers, MIZ-type			
2757	46.19	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
2758	46.18	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
2759	46.13	kd	CGS001-10253	SPRY2	-			
2760	46.12	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
2761	46.11	kd	CGS001-1105	CHD1	-			
2762	46.08	kd	CGS001-9275	BCL7B	-			
2763	46.08	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
2764	46.06	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
2765	46.06	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
2766	46.04	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
2767	46.04	kd	CGS001-79581	GPR172A	-			
2768	46.01	kd	CGS001-2167	FABP4	Fatty acid binding protein family			
2769	45.99	kd	CGS001-8804	CREG1	-			
2770	45.97	kd	CGS001-3565	IL4	Interleukins and interleukin receptors			
2771	45.96	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
2772	45.95	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
2773	45.94	oe	ccsbBroad304_07827	STK38L	NDR family			
2774	45.93	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
2775	45.93	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
2776	45.92	kd	CGS001-222894	FERD3L	Basic helix-loop-helix proteins			
2777	45.92	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
2778	45.91	cc		MDM inhibitor	-			
2779	45.89	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
2780	45.86	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
2781	45.86	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
2782	45.85	cc		Protein synthesis inhibitor	-			
2783	45.85	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
2784	45.83	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
2785	45.82	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
2786	45.82	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
2787	45.79	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
2788	45.71	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2789	45.58	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
2790	45.57	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
2791	45.57	kd	CGS001-83637	ZMIZ2	Zinc fingers, MIZ-type			
2792	45.56	oe	ccsbBroad304_06789	PSEN2	Presenilin			
2793	45.54	kd	CGS001-10051	SMC4	Structural maintenance of chromosomes proteins			
2794	45.53	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
2795	45.48	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
2796	45.44	kd	CGS001-7428	VHL	-			
2797	45.43	oe	ccsbBroad304_01576	SOAT1	-			
2798	45.36	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
2799	45.36	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
2800	45.36	kd	CGS001-4734	NEDD4	-			
2801	45.35	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
2802	45.34	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
2803	45.32	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
2804	45.3	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
2805	45.27	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
2806	45.27	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
2807	45.24	oe	ccsbBroad304_02002	RNMT	-			
2808	45.19	cp	BRD-K86887724	dofetilide	Potassium channel blocker		KCNH2, KCNH1, KCNJ12, KCNK2	Potassium channel blocker
2809	45.17	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
2810	45.17	kd	CGS001-2277	FIGF	-			
2811	45.16	cp	BRD-K70883034	nimetazepam	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA receptor agonist
2812	45.16	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
2813	45.15	kd	CGS001-6722	SRF	-			
2814	45.14	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
2815	45.14	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
2816	45.13	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
2817	45.11	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
2818	45.08	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2819	45.03	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
2820	45.01	oe	ccsbBroad304_03372	CAB39	-			
2821	45	kd	CGS001-8233	ZRSR2	RNA binding motif (RRM) containing			
2822	44.99	kd	CGS001-6714	SRC	Src family			
2823	44.99	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
2824	44.97	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
2825	44.95	oe	ccsbBroad304_00665	GOT1	-			
2826	44.94	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
2827	44.94	kd	CGS001-439	ASNA1	-			
2828	44.93	cc		Non Homologous End Joining LOF	-			
2829	44.93	kd	CGS001-147179	WIPF2	-			
2830	44.91	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
2831	44.91	kd	CGS001-6709	SPTAN1	EF-hand domain containing			
2832	44.87	oe	ccsbBroad304_00624	GCK	Hexokinases			
2833	44.86	oe	ccsbBroad304_06435	RBPJ	-			
2834	44.86	kd	CGS001-10587	TXNRD2	-			
2835	44.83	oe	ccsbBroad304_03798	PHTF2	-			
2836	44.81	cc		Tubulin inhibitor	-			
2837	44.8	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
2838	44.79	cc		Potassium channel activator	-			
2839	44.79	kd	CGS001-4773	NFATC2	Nuclear factor of activated T-cells			
2840	44.75	cp	BRD-K15916496	clotrimazole	Cytochrome P450 inhibitor		KCNN4, CYP3A4, CYP51A1, NR1I2, NR1I3, TRPM2, TRPM4, TRPM8	Cytochrome P450 inhibitor, Imidazoline receptor ligand
2841	44.74	kd	CGS001-5335	PLCG1	Phosphoinositide-specific phospholipase C			
2842	44.73	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
2843	44.73	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
2844	44.72	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
2845	44.72	kd	CGS001-8836	GGH	Gamma-glutamyl hydrolase			
2846	44.69	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
2847	44.68	oe	ccsbBroad304_13939	MOK	RCK family			
2848	44.68	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
2849	44.64	oe	ccsbBroad304_06255	LRRC32	-			
2850	44.63	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
2851	44.6	kd	CGS001-115201	ATG4A	-			
2852	44.57	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
2853	44.5	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
2854	44.49	kd	CGS001-27148	STK36	Unc-51-like kinase (ULK) family			
2855	44.48	oe	ccsbBroad304_02589	COPS5	-			
2856	44.48	kd	CGS001-4552	MTRR	-			
2857	44.47	oe	ccsbBroad304_02373	SPRY2	-			
2858	44.45	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
2859	44.44	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
2860	44.43	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
2861	44.42	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
2862	44.41	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
2863	44.39	oe	ccsbBroad304_06090	DDOST	-			
2864	44.39	kd	CGS001-7311	UBA52	L ribosomal proteins			
2865	44.35	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
2866	44.35	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
2867	44.32	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
2868	44.3	kd	CGS001-8575	PRKRA	-			
2869	44.29	kd	CGS001-26149	ZNF658	Zinc fingers, C2H2-type			
2870	44.28	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
2871	44.24	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
2872	44.24	kd	CGS001-4190	MDH1	-			
2873	44.24	kd	CGS001-3033	HADH	-			
2874	44.23	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
2875	44.22	kd	CGS001-1633	DCK	-			
2876	44.21	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
2877	44.2	kd	CGS001-29937	NENF	-			
2878	44.15	kd	CGS001-90655	TGIF2LY	Homeoboxes / TALE class			
2879	44.15	kd	CGS001-9767	PHF16	-			
2880	44.15	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2881	44.14	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
2882	44.12	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
2883	44.12	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
2884	44.11	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
2885	44.09	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
2886	44.06	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
2887	44.02	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
2888	44	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
2889	43.99	kd	CGS001-4953	ODC1	Decarboxylases			
2890	43.96	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
2891	43.95	kd	CGS001-55699	IARS2	Aminoacyl tRNA synthetases / Class I			
2892	43.94	cc		Structural maintenance of chromosomes proteins LOF	-			
2893	43.94	cp	BRD-K48932581	cetraxate	Mucus protecting agent		GAST	Mucus protecting agent
2894	43.93	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
2895	43.93	kd	CGS001-51569	UFM1	-			
2896	43.92	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
2897	43.86	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
2898	43.85	kd	CGS001-191	AHCY	Adenosine turnover			
2899	43.81	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
2900	43.8	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
2901	43.8	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
2902	43.79	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
2903	43.79	kd	CGS001-1030	CDKN2B	-			
2904	43.75	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2905	43.69	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
2906	43.66	oe	ccsbBroad304_03950	ATG3	-			
2907	43.66	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
2908	43.65	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
2909	43.63	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
2910	43.62	kd	CGS001-8050	PDHX	-			
2911	43.59	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
2912	43.57	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
2913	43.57	oe	ccsbBroad304_04399	PGBD1	-			
2914	43.54	oe	ccsbBroad304_00112	ASNA1	-			
2915	43.52	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
2916	43.52	kd	CGS001-537	ATP6AP1	-			
2917	43.44	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
2918	43.4	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
2919	43.37	kd	CGS001-5763	PTMS	-			
2920	43.36	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
2921	43.35	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
2922	43.34	cp	BRD-K94144010	cotinine	Nicotine metabolite			Nicotine metabolite
2923	43.33	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
2924	43.32	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
2925	43.29	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
2926	43.27	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
2927	43.27	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
2928	43.21	kd	CGS001-8659	ALDH4A1	Aldehyde dehydrogenases			
2929	43.18	kd	CGS001-8874	ARHGEF7	Rho guanine nucleotide exchange factors			
2930	43.16	oe	ccsbBroad304_05098	MAGEB6	-			
2931	43.16	oe	ccsbBroad304_02415	TUBB3	Tubulins			
2932	43.12	kd	CGS001-56647	BCCIP	-			
2933	43.09	cp	BRD-K33312228	halometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2934	43.08	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2935	43.06	oe	ccsbBroad304_01632	SYPL1	-			
2936	43.06	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
2937	43.04	kd	CGS001-5479	PPIB	-			
2938	43.04	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2939	43.03	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
2940	43	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
2941	42.97	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
2942	42.97	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
2943	42.96	oe	ccsbBroad304_02964	TIMM9	-			
2944	42.96	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
2945	42.95	cp	BRD-A23359898	sibutramine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, CYP2B6, CYP2C19, CYP3A5	Serotonin reuptake inhibitor
2946	42.95	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2947	42.88	kd	CGS001-2053	EPHX2	-			
2948	42.87	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
2949	42.86	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
2950	42.84	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
2951	42.8	kd	CGS001-9061	PAPSS1	-			
2952	42.77	kd	CGS001-9870	KIAA0317	-			
2953	42.75	kd	CGS001-55311	ZNF444	Zinc fingers, C2H2-type			
2954	42.73	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
2955	42.71	oe	ccsbBroad304_00268	CD81	CD molecules			
2956	42.71	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
2957	42.66	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2958	42.65	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
2959	42.6	kd	CGS001-81620	CDT1	-			
2960	42.57	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
2961	42.55	oe	ccsbBroad304_01948	GAS7	-			
2962	42.53	oe	ccsbBroad304_00963	SMAD5	SMADs			
2963	42.53	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2964	42.52	cp	BRD-K16336526	capsaicin	TRPV agonist		TRPV1, CFTR, ENOX2	TRPV agonist
2965	42.47	kd	CGS001-1718	DHCR24	-			
2966	42.45	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
2967	42.4	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
2968	42.4	kd	CGS001-4176	MCM7	-			
2969	42.39	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
2970	42.33	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
2971	42.27	kd	CGS001-2118	ETV4	ETS Transcription Factors			
2972	42.22	kd	CGS001-10474	TADA3	-			
2973	42.2	oe	ccsbBroad304_01640	TAF12	-			
2974	42.2	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
2975	42.16	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
2976	42.15	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
2977	42.14	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
2978	42.14	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
2979	42.09	oe	ccsbBroad304_01960	CASK	CASK family			
2980	42.07	kd	CGS001-7353	UFD1L	-			
2981	42.06	oe	ccsbBroad304_02249	KIAA0494	-			
2982	42.06	kd	CGS001-79885	HDAC11	Histone deacetylases			
2983	42.03	kd	CGS001-5993	RFX5	-			
2984	42.03	kd	CGS001-4548	MTR	-			
2985	42.02	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
2986	42.01	oe	ccsbBroad304_01205	PIN1	-			
2987	41.97	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
2988	41.96	oe	ccsbBroad304_01054	GADD45B	-			
2989	41.93	cc		Kinase anchoring proteins LOF	-			
2990	41.86	kd	CGS001-2356	FPGS	-			
2991	41.85	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
2992	41.84	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
2993	41.82	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
2994	41.82	kd	CGS001-83593	RASSF5	-			
2995	41.81	oe	ccsbBroad304_01527	SGK1	SGK family			
2996	41.79	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
2997	41.75	kd	CGS001-5580	PRKCD	Delta subfamily			
2998	41.75	kd	CGS001-10725	NFAT5	Nuclear factor of activated T-cells			
2999	41.73	oe	ccsbBroad304_09006	RPF1	-			
3000	41.71	kd	CGS001-26086	GPSM1	Tetratricopeptide (TTC) repeat domain containing			
3001	41.68	oe	ccsbBroad304_03859	ENOPH1	-			
3002	41.67	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
3003	41.66	kd	CGS001-5588	PRKCQ	Delta subfamily			
3004	41.65	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
3005	41.65	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
3006	41.63	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
3007	41.63	kd	CGS001-4173	MCM4	-			
3008	41.62	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
3009	41.61	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
3010	41.61	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
3011	41.61	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3012	41.61	kd	CGS001-23266	LPHN2	Adhesion Class GPCRs			
3013	41.56	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
3014	41.54	kd	CGS001-22934	RPIA	-			
3015	41.53	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
3016	41.53	kd	CGS001-10969	EBNA1BP2	-			
3017	41.52	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
3018	41.52	kd	CGS001-670	BPHL	-			
3019	41.52	kd	CGS001-367	AR	Nuclear hormone receptors			
3020	41.5	cp	BRD-K10961822	latanoprost	Prostanoid receptor agonist		PTGFR	Prostanoid receptor agonist
3021	41.49	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
3022	41.47	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
3023	41.46	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
3024	41.45	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
3025	41.37	cp	BRD-K69650333	idarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
3026	41.36	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
3027	41.36	kd	CGS001-51586	MED15	-			
3028	41.36	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
3029	41.33	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
3030	41.29	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
3031	41.28	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
3032	41.28	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
3033	41.26	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
3034	41.24	kd	CGS001-10252	SPRY1	-			
3035	41.22	oe	ccsbBroad304_02579	YWHAQ	-			
3036	41.2	kd	CGS001-121549	ASCL4	Basic helix-loop-helix proteins			
3037	41.18	kd	CGS001-4926	NUMA1	-			
3038	41.16	oe	ccsbBroad304_00164	BLMH	-			
3039	41.15	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
3040	41.12	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
3041	41.11	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
3042	41.08	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
3043	41.07	oe	ccsbBroad304_01832	PAX8	Paired boxes			
3044	41.05	oe	ccsbBroad304_02526	POP4	-			
3045	41.05	oe	ccsbBroad304_07208	NRIP1	-			
3046	41.05	kd	CGS001-2114	ETS2	ETS Transcription Factors			
3047	41.04	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3048	40.99	kd	CGS001-51027	BOLA1	-			
3049	40.97	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
3050	40.96	kd	CGS001-10451	VAV3	Rho guanine nucleotide exchange factors			
3051	40.95	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
3052	40.92	oe	ccsbBroad304_06836	RAD23B	-			
3053	40.92	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
3054	40.89	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
3055	40.84	oe	ccsbBroad304_08266	PIPOX	-			
3056	40.84	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
3057	40.84	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
3058	40.78	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
3059	40.76	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
3060	40.73	kd	CGS001-84647	PLA2G12B	-			
3061	40.69	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
3062	40.68	kd	CGS001-8896	BUD31	-			
3063	40.66	oe	ccsbBroad304_00392	CTLA4	CD molecules			
3064	40.6	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3065	40.59	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
3066	40.59	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
3067	40.51	kd	CGS001-1644	DDC	Catecholamine turnover			
3068	40.5	kd	CGS001-56654	NPDC1	-			
3069	40.49	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
3070	40.48	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
3071	40.47	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
3072	40.46	oe	ccsbBroad304_00184	C2	Complement system			
3073	40.45	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
3074	40.45	oe	ccsbBroad304_03121	NRBF2	-			
3075	40.4	kd	CGS001-64750	SMURF2	-			
3076	40.4	kd	CGS001-81611	ANP32E	ANP32 acidic nuclear phosphoproteins			
3077	40.38	kd	CGS001-9380	GRHPR	-			
3078	40.38	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
3079	40.37	kd	CGS001-7159	TP53BP2	Ankyrin repeat domain containing			
3080	40.36	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
3081	40.32	kd	CGS001-5442	POLRMT	-			
3082	40.29	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
3083	40.25	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
3084	40.23	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
3085	40.22	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
3086	40.22	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
3087	40.22	kd	CGS001-2869	GRK5	GRK1/3 subfamily			
3088	40.19	kd	CGS001-6286	S100P	EF-hand domain containing			
3089	40.18	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
3090	40.17	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
3091	40.16	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
3092	40.14	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
3093	40.14	kd	CGS001-2837	UTS2R	Urotensin receptor			
3094	40.12	oe	ccsbBroad304_04655	TRIM9	-			
3095	40.11	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
3096	40.11	cp	BRD-K39621635	artemether	Antimalarial		ATP1A1, CYP2B6, CYP2C19, CYP3A5	Antimalarial
3097	40.09	kd	CGS001-5355	PLP2	-			
3098	40.06	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
3099	40.06	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
3100	40.05	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
3101	40.05	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
3102	40.04	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
3103	40.01	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
3104	40.01	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
3105	39.99	kd	CGS001-54821	ERCC6L	-			
3106	39.97	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
3107	39.97	kd	CGS001-1514	CTSL1	-			
3108	39.95	oe	ccsbBroad304_08596	EAPP	-			
3109	39.94	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
3110	39.94	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
3111	39.9	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
3112	39.88	oe	ccsbBroad304_04649	ADC	-			
3113	39.83	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3114	39.8	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
3115	39.79	kd	CGS001-8204	NRIP1	-			
3116	39.79	kd	CGS001-344	APOC2	Apolipoproteins			
3117	39.77	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
3118	39.76	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
3119	39.72	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
3120	39.68	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
3121	39.64	oe	ccsbBroad304_02653	PRAF2	-			
3122	39.64	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
3123	39.64	kd	CGS001-4779	NFE2L1	basic leucine zipper proteins			
3124	39.64	kd	CGS001-2181	ACSL3	Acyl-CoA synthetase family			
3125	39.63	kd	CGS001-10943	MSL3	-			
3126	39.62	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
3127	39.51	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
3128	39.51	kd	CGS001-57787	MARK4	MARK subfamily			
3129	39.5	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3130	39.5	kd	CGS001-57657	HCN3	Cyclic nucleotide-regulated channels			
3131	39.48	kd	CGS001-8935	SKAP2	Pleckstrin homology (PH) domain containing			
3132	39.47	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
3133	39.45	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
3134	39.44	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
3135	39.43	kd	CGS001-5891	MOK	RCK family			
3136	39.42	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
3137	39.42	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
3138	39.42	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
3139	39.39	oe	ccsbBroad304_00519	ETFB	-			
3140	39.39	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
3141	39.39	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
3142	39.38	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
3143	39.37	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
3144	39.35	oe	ccsbBroad304_03497	TXNL4B	-			
3145	39.34	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
3146	39.33	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
3147	39.29	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
3148	39.29	kd	CGS001-117154	DACH2	-			
3149	39.24	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
3150	39.24	kd	CGS001-301	ANXA1	Annexins			
3151	39.23	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
3152	39.22	kd	CGS001-1209	CLPTM1	-			
3153	39.19	kd	CGS001-84109	QRFPR	GPCR / Class A : RF amide peptide receptors			
3154	39.13	kd	CGS001-7276	TTR	-			
3155	39.08	oe	ccsbBroad304_00249	CD14	CD molecules			
3156	39.08	kd	CGS001-6622	SNCA	Parkinson disease			
3157	39.01	oe	ccsbBroad304_03415	GFOD1	-			
3158	39.01	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3159	39	kd	CGS001-6337	SCNN1A	Epithelial sodium channels (ENaC)			
3160	38.96	kd	CGS001-25861	DFNB31	-			
3161	38.93	kd	CGS001-10468	FST	-			
3162	38.91	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
3163	38.91	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
3164	38.91	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
3165	38.86	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
3166	38.84	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
3167	38.82	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
3168	38.81	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
3169	38.79	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
3170	38.76	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
3171	38.75	kd	CGS001-805	CALM2	EF-hand domain containing			
3172	38.74	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
3173	38.73	kd	CGS001-7272	TTK	TTK family			
3174	38.72	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
3175	38.69	kd	CGS001-3614	IMPDH1	Oxidoreductases			
3176	38.67	cc		Retinoid receptor agonist	-			
3177	38.67	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
3178	38.66	oe	ccsbBroad304_02398	LANCL1	-			
3179	38.66	kd	CGS001-8634	RTCD1	-			
3180	38.65	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
3181	38.6	kd	CGS001-4089	SMAD4	SMADs			
3182	38.59	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3183	38.58	kd	CGS001-9232	PTTG1	-			
3184	38.57	kd	CGS001-23224	SYNE2	-			
3185	38.55	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
3186	38.55	kd	CGS001-775	CACNA1C	Calcium channel subunits			
3187	38.54	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
3188	38.48	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
3189	38.47	kd	CGS001-836	CASP3	Caspases			
3190	38.42	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
3191	38.42	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
3192	38.42	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
3193	38.41	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
3194	38.41	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
3195	38.35	kd	CGS001-28985	MCTS1	-			
3196	38.33	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
3197	38.31	kd	CGS001-55278	QRSL1	-			
3198	38.31	kd	CGS001-8477	GPR65	GPCR / Class A : Orphans			
3199	38.29	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
3200	38.29	kd	CGS001-90861	HN1L	-			
3201	38.28	kd	CGS001-10400	PEMT	-			
3202	38.27	kd	CGS001-6757	SSX2	-			
3203	38.23	oe	ccsbBroad304_06085	DCK	-			
3204	38.21	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
3205	38.21	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
3206	38.21	kd	CGS001-29978	UBQLN2	Ubiquilin family			
3207	38.21	kd	CGS001-182	JAG1	CD molecules			
3208	38.2	oe	ccsbBroad304_01164	PDHB	-			
3209	38.2	kd	CGS001-64121	RRAGC	-			
3210	38.19	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
3211	38.19	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3212	38.17	kd	CGS001-4547	MTTP	-			
3213	38.14	kd	CGS001-3572	IL6ST	IL-6 receptor family			
3214	38.09	kd	CGS001-9898	UBAP2L	-			
3215	38.08	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
3216	38.07	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
3217	38.04	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
3218	38.03	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
3219	38.02	cc		MTOR inhibitor	-			
3220	37.98	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
3221	37.95	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
3222	37.94	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
3223	37.89	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
3224	37.87	kd	CGS001-340371	NRBP2	NRBP family			
3225	37.86	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
3226	37.83	oe	ccsbBroad304_02278	THRAP3	-			
3227	37.83	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
3228	37.83	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
3229	37.81	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
3230	37.81	kd	CGS001-51375	SNX7	Sorting nexins			
3231	37.8	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
3232	37.77	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
3233	37.74	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
3234	37.71	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
3235	37.69	kd	CGS001-84328	LZIC	-			
3236	37.67	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
3237	37.65	oe	ccsbBroad304_03264	UBAP1	-			
3238	37.65	oe	ccsbBroad304_00072	ANXA7	Annexins			
3239	37.64	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
3240	37.62	cp	BRD-A87387433	cefpodoxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3241	37.56	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3242	37.56	kd	CGS001-58492	ZNF77	Zinc fingers, C2H2-type			
3243	37.55	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
3244	37.54	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
3245	37.5	kd	CGS001-3665	IRF7	-			
3246	37.49	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
3247	37.49	kd	CGS001-2274	FHL2	-			
3248	37.47	kd	CGS001-345611	IRGM	-			
3249	37.46	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
3250	37.45	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
3251	37.44	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
3252	37.43	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
3253	37.42	kd	CGS001-79071	ELOVL6	-			
3254	37.4	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
3255	37.38	oe	ccsbBroad304_00651	GNAI3	-			
3256	37.37	kd	CGS001-2004	ELK3	ETS Transcription Factors			
3257	37.36	oe	ccsbBroad304_06282	GLDC	-			
3258	37.34	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
3259	37.33	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
3260	37.33	kd	CGS001-5727	PTCH1	-			
3261	37.31	oe	ccsbBroad304_09954	PTRF	-			
3262	37.31	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
3263	37.3	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
3264	37.3	kd	CGS001-10891	PPARGC1A	RNA binding motif (RRM) containing			
3265	37.28	oe	ccsbBroad304_00459	DPYD	-			
3266	37.28	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
3267	37.24	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
3268	37.16	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
3269	37.12	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
3270	37.11	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
3271	37.1	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
3272	37.08	cc		Topoisomerase inhibitor	-			
3273	37.08	kd	CGS001-113878	DTX2	RING-type (C3HC4) zinc fingers			
3274	37.07	kd	CGS001-5432	POLR2C	RNA polymerase subunits			
3275	37.04	oe	ccsbBroad304_04379	LZIC	-			
3276	37.02	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
3277	37.01	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
3278	36.97	kd	CGS001-284119	PTRF	-			
3279	36.94	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
3280	36.94	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
3281	36.93	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
3282	36.9	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
3283	36.89	oe	ccsbBroad304_01593	SRP14	-			
3284	36.89	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
3285	36.86	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
3286	36.85	kd	CGS001-23650	TRIM29	-			
3287	36.85	kd	CGS001-3685	ITGAV	Integrins			
3288	36.83	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
3289	36.81	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
3290	36.78	kd	CGS001-11284	PNKP	-			
3291	36.77	oe	ccsbBroad304_00054	ALDOC	-			
3292	36.76	kd	CGS001-7076	TIMP1	-			
3293	36.74	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3294	36.74	kd	CGS001-54505	DHX29	DEAH-boxes			
3295	36.72	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
3296	36.69	kd	CGS001-83448	PUS7L	-			
3297	36.69	kd	CGS001-4069	LYZ	-			
3298	36.67	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
3299	36.66	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
3300	36.65	kd	CGS001-3992	FADS1	Fatty acid desaturases			
3301	36.64	oe	ccsbBroad304_02738	RRS1	-			
3302	36.62	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
3303	36.62	kd	CGS001-10111	RAD50	-			
3304	36.6	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
3305	36.58	oe	ccsbBroad304_03037	TMEM97	-			
3306	36.57	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
3307	36.52	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3308	36.52	kd	CGS001-5019	OXCT1	-			
3309	36.5	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
3310	36.49	oe	ccsbBroad304_01034	MSH2	-			
3311	36.49	kd	CGS001-5932	RBBP8	-			
3312	36.47	kd	CGS001-1399	CRKL	SH2 domain containing			
3313	36.44	oe	ccsbBroad304_08878	METTL4	-			
3314	36.44	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
3315	36.41	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
3316	36.39	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
3317	36.39	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
3318	36.36	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
3319	36.34	kd	CGS001-9869	SETDB1	Histone methyltransferases (HMTs)			
3320	36.32	kd	CGS001-1468	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
3321	36.29	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3322	36.29	kd	CGS001-5292	PIM1	PIM family			
3323	36.29	kd	CGS001-79109	MAPKAP1	-			
3324	36.28	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
3325	36.23	kd	CGS001-8431	NR0B2	DAX-like receptors			
3326	36.22	oe	ccsbBroad304_09503	KLHDC9	-			
3327	36.22	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
3328	36.22	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
3329	36.21	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
3330	36.19	oe	ccsbBroad304_03444	PAF1	-			
3331	36.19	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
3332	36.15	kd	CGS001-5255	PHKA1	-			
3333	36.11	kd	CGS001-27097	TAF5L	WD repeat domain containing			
3334	36.07	kd	CGS001-6119	RPA3	-			
3335	36.06	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
3336	36.06	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3337	36.05	oe	ccsbBroad304_04775	NTAN1	-			
3338	36.03	oe	ccsbBroad304_00032	ADSL	-			
3339	36.03	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
3340	36	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
3341	35.96	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
3342	35.96	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
3343	35.95	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
3344	35.95	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
3345	35.94	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
3346	35.83	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
3347	35.83	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
3348	35.79	cc		GPCR Subset GOF	-			
3349	35.74	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
3350	35.73	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
3351	35.73	kd	CGS001-8850	KAT2B	Histone acetyltransferases (HATs)			
3352	35.72	oe	ccsbBroad304_02496	MTX2	-			
3353	35.7	kd	CGS001-4292	MLH1	-			
3354	35.66	oe	ccsbBroad304_06562	MAT1A	-			
3355	35.64	kd	CGS001-6611	SMS	-			
3356	35.62	kd	CGS001-129685	TAF8	-			
3357	35.6	kd	CGS001-5583	PRKCH	Eta subfamily			
3358	35.6	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3359	35.6	kd	CGS001-79145	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
3360	35.6	oe	ccsbBroad304_06383	HMMR	CD molecules			
3361	35.58	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
3362	35.57	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
3363	35.56	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
3364	35.53	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
3365	35.51	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
3366	35.5	kd	CGS001-10939	AFG3L2	ATPases / AAA-type			
3367	35.49	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
3368	35.49	kd	CGS001-1647	GADD45A	-			
3369	35.47	oe	ccsbBroad304_07277	RTCD1	-			
3370	35.46	kd	CGS001-51547	SIRT7	Histone deacetylases (HDACs)			
3371	35.43	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
3372	35.37	cp	BRD-K63265447	docetaxel	Tubulin inhibitor		TUBB, BCL2, MAP2, MAP4, MAPT, NR1I2, TUBB1	Tubulin inhibitor
3373	35.36	oe	ccsbBroad304_02340	SORBS3	-			
3374	35.33	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
3375	35.32	oe	ccsbBroad304_00113	ASNS	-			
3376	35.32	kd	CGS001-5920	RARRES3	-			
3377	35.31	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
3378	35.29	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
3379	35.28	cc		X linked mental retardation group 1 LOF	-			
3380	35.28	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
3381	35.27	kd	CGS001-9670	IPO13	Importins			
3382	35.25	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
3383	35.23	oe	ccsbBroad304_07890	CBX7	-			
3384	35.23	kd	CGS001-7003	TEAD1	-			
3385	35.23	kd	CGS001-9700	ESPL1	-			
3386	35.22	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
3387	35.14	kd	CGS001-11333	PDAP1	-			
3388	35.13	oe	ccsbBroad304_06382	HMGCL	-			
3389	35.13	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
3390	35.12	oe	ccsbBroad304_06870	RNH1	-			
3391	35.11	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
3392	35.09	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
3393	35.03	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
3394	35.03	kd	CGS001-51548	SIRT6	Histone deacetylases (HDACs)			
3395	35.02	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
3396	35.02	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
3397	35.01	kd	CGS001-1512	CTSH	Cathepsins			
3398	34.96	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
3399	34.96	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
3400	34.96	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
3401	34.96	kd	CGS001-652	BMP4	Bone morphogenetic proteins			
3402	34.95	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
3403	34.95	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
3404	34.94	oe	ccsbBroad304_01066	NDUFA4	-			
3405	34.92	kd	CGS001-8148	TAF15	RNA binding motif (RRM) containing			
3406	34.88	kd	CGS001-8743	TNFSF10	CD molecules			
3407	34.88	kd	CGS001-10397	NDRG1	-			
3408	34.87	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
3409	34.86	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
3410	34.86	oe	ccsbBroad304_01139	PA2G4	-			
3411	34.85	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
3412	34.84	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
3413	34.83	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3414	34.83	kd	CGS001-2639	GCDH	-			
3415	34.82	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
3416	34.81	oe	ccsbBroad304_03112	NENF	-			
3417	34.81	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
3418	34.8	oe	ccsbBroad304_06720	PHYH	-			
3419	34.8	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
3420	34.76	oe	ccsbBroad304_06008	AP2M1	-			
3421	34.75	cc		FOS transcription factor family GOF	-			
3422	34.75	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
3423	34.73	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
3424	34.72	oe	ccsbBroad304_03506	AURKAIP1	-			
3425	34.71	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
3426	34.68	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
3427	34.67	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
3428	34.67	oe	ccsbBroad304_08993	DHDDS	-			
3429	34.63	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
3430	34.62	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
3431	34.61	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
3432	34.61	kd	CGS001-51465	UBE2J1	Ubiquitin-conjugating enzymes E2			
3433	34.6	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
3434	34.6	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
3435	34.57	kd	CGS001-6924	TCEB3	-			
3436	34.57	kd	CGS001-2782	GNB1	WD repeat domain containing			
3437	34.54	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
3438	34.53	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
3439	34.52	kd	CGS001-57026	PDXP	-			
3440	34.51	kd	CGS001-8797	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
3441	34.5	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
3442	34.49	oe	ccsbBroad304_07506	UBAP2L	-			
3443	34.49	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
3444	34.44	oe	ccsbBroad304_01872	DGCR14	-			
3445	34.4	kd	CGS001-5966	REL	NFkappaB transcription factor family			
3446	34.4	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
3447	34.39	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
3448	34.39	kd	CGS001-3455	IFNAR2	Interferon receptor family			
3449	34.35	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
3450	34.35	kd	CGS001-55556	ENOSF1	-			
3451	34.34	oe	ccsbBroad304_07018	SUPT5H	-			
3452	34.33	oe	ccsbBroad304_00510	EPHX2	-			
3453	34.33	kd	CGS001-883	CCBL1	Hydrogen sulphide synthesis			
3454	34.32	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
3455	34.32	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
3456	34.32	kd	CGS001-275	AMT	-			
3457	34.31	kd	CGS001-162	AP1B1	-			
3458	34.3	kd	CGS001-1497	CTNS	-			
3459	34.28	oe	ccsbBroad304_02298	DNM1L	-			
3460	34.24	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
3461	34.21	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
3462	34.18	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
3463	34.18	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
3464	34.16	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
3465	34.16	oe	ccsbBroad304_06324	GPX7	-			
3466	34.15	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
3467	34.13	cc		Estrogen receptor agonist	-			
3468	34.13	oe	ccsbBroad304_01257	PPOX	-			
3469	34.11	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
3470	34.1	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
3471	34.08	kd	CGS001-140465	MYL6B	EF-hand domain containing			
3472	34.05	kd	CGS001-2768	GNA12	-			
3473	34.02	kd	CGS001-3995	FADS3	Fatty acid desaturases			
3474	34.01	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
3475	34	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
3476	34	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
3477	34	kd	CGS001-10810	WASF3	-			
3478	33.98	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
3479	33.95	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
3480	33.94	kd	CGS001-6895	TARBP2	-			
3481	33.92	kd	CGS001-4671	NAIP	Inhibitors of apoptosis (IAP) protein family			
3482	33.9	kd	CGS001-2878	GPX3	-			
3483	33.89	kd	CGS001-392	ARHGAP1	Rho GTPase activating proteins			
3484	33.88	kd	CGS001-54732	TMED9	-			
3485	33.88	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
3486	33.86	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
3487	33.84	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
3488	33.83	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
3489	33.79	kd	CGS001-5315	PKM2	-			
3490	33.78	kd	CGS001-124535	HSF5	-			
3491	33.75	kd	CGS001-4090	SMAD5	SMADs			
3492	33.74	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
3493	33.74	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
3494	33.72	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
3495	33.72	kd	CGS001-10214	SSX3	-			
3496	33.71	kd	CGS001-9748	SLK	SLK subfamily			
3497	33.68	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
3498	33.67	kd	CGS001-64710	NUCKS1	-			
3499	33.65	oe	ccsbBroad304_01174	PEX13	-			
3500	33.64	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
3501	33.63	kd	CGS001-7175	TPR	-			
3502	33.62	cp	BRD-M47937986	cefatrizine	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3503	33.62	kd	CGS001-4507	MTAP	-			
3504	33.59	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
3505	33.56	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
3506	33.56	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
3507	33.54	kd	CGS001-7424	VEGFC	-			
3508	33.54	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
3509	33.49	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
3510	33.48	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
3511	33.47	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
3512	33.47	kd	CGS001-5624	PROC	Endogenous ligands			
3513	33.47	kd	CGS001-2	A2M	-			
3514	33.45	kd	CGS001-2002	ELK1	ETS Transcription Factors			
3515	33.45	kd	CGS001-174	AFP	-			
3516	33.44	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
3517	33.39	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
3518	33.38	oe	ccsbBroad304_00486	EFNB2	Ephrins			
3519	33.38	kd	CGS001-2015	EMR1	Adhesion Class GPCRs			
3520	33.35	kd	CGS001-391013	PLA2G2C	-			
3521	33.3	oe	ccsbBroad304_06178	ERCC5	-			
3522	33.3	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3523	33.24	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
3524	33.23	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
3525	33.22	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
3526	33.22	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
3527	33.2	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
3528	33.2	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
3529	33.19	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
3530	33.18	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
3531	33.17	oe	ccsbBroad304_06852	RBP4	Lipocalins			
3532	33.16	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
3533	33.16	oe	ccsbBroad304_06089	DDIT3	-			
3534	33.13	kd	CGS001-5550	PREP	Prolyl oligopeptidase			
3535	33.1	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
3536	33.09	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3537	33.08	kd	CGS001-79902	NUP85	-			
3538	33.08	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
3539	33.08	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
3540	33.08	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
3541	33.04	kd	CGS001-5223	PGAM1	-			
3542	33.02	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
3543	33.01	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
3544	33.01	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
3545	32.95	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
3546	32.94	kd	CGS001-2876	GPX1	-			
3547	32.92	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
3548	32.92	kd	CGS001-10975	UQCR11	Mitochondrial respiratory chain complex / Complex III			
3549	32.89	oe	ccsbBroad304_00818	IDH3A	-			
3550	32.88	kd	CGS001-3225	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
3551	32.86	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
3552	32.84	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
3553	32.83	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
3554	32.83	kd	CGS001-56993	TOMM22	-			
3555	32.82	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
3556	32.81	kd	CGS001-5573	PRKAR1A	Protein kinase A			
3557	32.81	kd	CGS001-10046	MAMLD1	-			
3558	32.8	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
3559	32.77	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
3560	32.75	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
3561	32.75	kd	CGS001-1072	CFL1	-			
3562	32.73	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
3563	32.72	kd	CGS001-57018	CCNL1	-			
3564	32.71	oe	ccsbBroad304_02554	TRAFD1	-			
3565	32.71	kd	CGS001-51022	GLRX2	-			
3566	32.7	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
3567	32.7	kd	CGS001-23043	TNIK	MSN subfamily			
3568	32.68	oe	ccsbBroad304_05528	TICAM2	-			
3569	32.67	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
3570	32.66	kd	CGS001-338	APOB	Apolipoproteins			
3571	32.65	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
3572	32.65	kd	CGS001-5471	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
3573	32.65	kd	CGS001-57721	METTL14	-			
3574	32.63	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
3575	32.63	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
3576	32.63	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
3577	32.56	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
3578	32.56	kd	CGS001-506	ATP5B	ATPases / F-type			
3579	32.55	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
3580	32.54	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
3581	32.53	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
3582	32.53	kd	CGS001-51564	HDAC7	Histone deacetylases			
3583	32.51	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
3584	32.48	kd	CGS001-169436	C9ORF96	-			
3585	32.46	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
3586	32.44	oe	ccsbBroad304_00572	FKBP3	-			
3587	32.42	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
3588	32.42	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
3589	32.4	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
3590	32.4	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
3591	32.39	kd	CGS001-1440	CSF3	Endogenous ligands			
3592	32.38	kd	CGS001-51097	SCCPDH	-			
3593	32.37	oe	ccsbBroad304_01327	PSPH	-			
3594	32.36	cc		Homeobox Gene GOF	-			
3595	32.36	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
3596	32.36	kd	CGS001-83694	RPS6KL1	RSKL family			
3597	32.35	oe	ccsbBroad304_00501	EMD	-			
3598	32.33	kd	CGS001-716	C1S	Complement system			
3599	32.32	kd	CGS001-5535	PPP3R2	EF-hand domain containing			
3600	32.32	kd	CGS001-10775	POP4	-			
3601	32.31	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
3602	32.3	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
3603	32.3	kd	CGS001-29116	MYLIP	-			
3604	32.3	kd	CGS001-3054	HCFC1	-			
3605	32.26	oe	ccsbBroad304_04457	TOX2	-			
3606	32.23	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
3607	32.23	kd	CGS001-4191	MDH2	-			
3608	32.21	oe	ccsbBroad304_01658	PRDX2	-			
3609	32.21	kd	CGS001-7078	TIMP3	-			
3610	32.21	kd	CGS001-23046	KIF21B	Kinesins			
3611	32.15	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
3612	32.14	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
3613	32.12	kd	CGS001-3920	LAMP2	CD molecules			
3614	32.06	kd	CGS001-148327	CREB3L4	basic leucine zipper proteins			
3615	32.05	cc		HSP inhibitor	-			
3616	32.02	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
3617	32	kd	CGS001-9616	RNF7	RING-type (C3HC4) zinc fingers			
3618	31.96	oe	ccsbBroad304_08452	PIH1D1	-			
3619	31.96	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
3620	31.94	kd	CGS001-7083	TK1	-			
3621	31.94	kd	CGS001-578	BAK1	-			
3622	31.92	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
3623	31.88	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
3624	31.85	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
3625	31.82	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
3626	31.8	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
3627	31.78	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
3628	31.77	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
3629	31.77	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
3630	31.77	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
3631	31.77	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
3632	31.76	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
3633	31.75	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
3634	31.73	kd	CGS001-94235	GNG8	-			
3635	31.72	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
3636	31.7	oe	ccsbBroad304_02136	COPS2	-			
3637	31.68	kd	CGS001-4967	OGDH	-			
3638	31.67	kd	CGS001-390980	ZNF805	Zinc fingers, C2H2-type			
3639	31.66	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
3640	31.65	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
3641	31.63	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
3642	31.6	kd	CGS001-1001	CDH3	Cadherins / Major cadherins			
3643	31.59	kd	CGS001-8531	CSDA	-			
3644	31.58	kd	CGS001-2048	EPHB2	Type XIII RTKs: Ephrin receptor family			
3645	31.58	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
3646	31.57	oe	ccsbBroad304_08839	IFIH1	-			
3647	31.56	cc		Vesicular Transport LOF	-			
3648	31.56	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
3649	31.56	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
3650	31.53	oe	ccsbBroad304_01208	PITPNA	-			
3651	31.48	oe	ccsbBroad304_05745	CD24	CD molecules			
3652	31.48	kd	CGS001-6595	SMARCA2	Non-enzymatic BRD containing proteins			
3653	31.46	kd	CGS001-4175	MCM6	-			
3654	31.42	kd	CGS001-400	ARL1	ADP-ribosylation factors			
3655	31.39	kd	CGS001-7423	VEGFB	-			
3656	31.35	kd	CGS001-2197	FAU	S ribosomal proteins			
3657	31.31	kd	CGS001-1662	DDX10	DEAD-boxes			
3658	31.28	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
3659	31.28	kd	CGS001-10018	BCL2L11	-			
3660	31.24	kd	CGS001-4836	NMT1	-			
3661	31.22	kd	CGS001-4072	EPCAM	CD molecules			
3662	31.21	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
3663	31.2	oe	ccsbBroad304_07889	QPRT	-			
3664	31.18	kd	CGS001-25937	WWTR1	Hippo Signaling			
3665	31.14	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
3666	31.13	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
3667	31.13	kd	CGS001-5914	RARA	Retinoic acid receptors			
3668	31.13	kd	CGS001-390212	GPR152	GPCR / Class A : Orphans			
3669	31.1	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
3670	31.09	kd	CGS001-9322	TRIP10	-			
3671	31.04	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
3672	31.03	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
3673	31.01	kd	CGS001-23355	VPS8	-			
3674	31.01	kd	CGS001-51593	SRRT	-			
3675	31.01	kd	CGS001-662	BNIP1	-			
3676	30.98	kd	CGS001-221391	OPN5	GPCR / Class A : Opsin receptors			
3677	30.97	kd	CGS001-2287	FKBP3	-			
3678	30.96	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
3679	30.96	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
3680	30.94	oe	ccsbBroad304_08339	CMPK1	-			
3681	30.93	kd	CGS001-10078	TSSC4	-			
3682	30.92	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
3683	30.88	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
3684	30.87	kd	CGS001-5184	PEPD	Methionyl aminopeptidase			
3685	30.86	kd	CGS001-10991	SLC38A3	System N-like transporters			
3686	30.86	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
3687	30.86	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
3688	30.85	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3689	30.85	kd	CGS001-9447	AIM2	-			
3690	30.84	kd	CGS001-11044	PAPD7	-			
3691	30.84	kd	CGS001-3482	IGF2R	CD molecules			
3692	30.83	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
3693	30.79	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
3694	30.74	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
3695	30.74	kd	CGS001-124641	OVCA2	-			
3696	30.74	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
3697	30.73	cc		Interleukin receptors LOF	-			
3698	30.7	kd	CGS001-9122	SLC16A4	SLC16 family of monocarboxylate transporters			
3699	30.66	oe	ccsbBroad304_00817	IDH2	-			
3700	30.66	kd	CGS001-10329	TMEM5	-			
3701	30.64	kd	CGS001-8878	SQSTM1	-			
3702	30.62	kd	CGS001-7099	TLR4	Toll-like receptor family			
3703	30.62	kd	CGS001-5584	PRKCI	Iota subfamily			
3704	30.61	kd	CGS001-4436	MSH2	-			
3705	30.58	kd	CGS001-2731	GLDC	-			
3706	30.57	kd	CGS001-1173	AP2M1	-			
3707	30.56	kd	CGS001-6608	SMO	GPCR / Class F : Frizzled receptors			
3708	30.55	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
3709	30.48	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
3710	30.48	kd	CGS001-4300	MLLT3	-			
3711	30.47	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
3712	30.46	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
3713	30.46	kd	CGS001-523	ATP6V1A	ATPases / V-type			
3714	30.45	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
3715	30.45	kd	CGS001-149233	IL23R	IL-12 receptor family			
3716	30.44	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
3717	30.43	oe	ccsbBroad304_09095	PUS7L	-			
3718	30.43	kd	CGS001-283	ANG	Ribonucleases, RNase A			
3719	30.38	kd	CGS001-55234	SMU1	WD repeat domain containing			
3720	30.37	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
3721	30.35	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
3722	30.35	kd	CGS001-4200	ME2	-			
3723	30.34	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
3724	30.33	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
3725	30.31	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
3726	30.3	kd	CGS001-3416	IDE	Pitrilysin			
3727	30.29	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
3728	30.28	cc		BCL inhibitor	-			
3729	30.28	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
3730	30.26	oe	ccsbBroad304_00883	ISG20	-			
3731	30.24	kd	CGS001-6391	SDHC	Mitochondrial respiratory chain complex / Complex II			
3732	30.24	kd	CGS001-57521	RPTOR	WD repeat domain containing			
3733	30.19	kd	CGS001-8508	NIPSNAP1	-			
3734	30.18	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
3735	30.17	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
3736	30.16	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
3737	30.16	kd	CGS001-2254	FGF9	Endogenous ligands			
3738	30.13	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3739	30.08	kd	CGS001-6827	SUPT4H1	-			
3740	30.08	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
3741	30.07	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
3742	30.05	cp	BRD-K82143716	flucytosine	Antifungal		DNMT1	Antifungal
3743	30.05	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3744	30.04	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
3745	30.03	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
3746	30.03	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
3747	30.02	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
3748	30	kd	CGS001-2550	GABBR1	GABA receptors			
3749	29.98	cc		Toll like receptors LOF	-			
3750	29.97	kd	CGS001-10645	CAMKK2	Meta subfamily			
3751	29.97	kd	CGS001-8573	CASK	CASK family			
3752	29.95	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
3753	29.95	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
3754	29.91	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
3755	29.91	kd	CGS001-84875	PARP10	Poly (ADP-ribose) polymerases			
3756	29.89	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
3757	29.88	oe	ccsbBroad304_00370	CS	-			
3758	29.87	kd	CGS001-9263	STK17A	Death-associated kinase (DAPK) family			
3759	29.86	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
3760	29.86	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
3761	29.86	kd	CGS001-1184	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
3762	29.83	kd	CGS001-5378	PMS1	-			
3763	29.77	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
3764	29.74	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
3765	29.73	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
3766	29.73	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
3767	29.7	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
3768	29.69	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3769	29.67	oe	ccsbBroad304_07478	CCP110	-			
3770	29.61	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
3771	29.61	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
3772	29.57	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
3773	29.55	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
3774	29.55	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
3775	29.54	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3776	29.52	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
3777	29.52	kd	CGS001-811	CALR	-			
3778	29.48	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
3779	29.43	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
3780	29.42	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
3781	29.39	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3782	29.38	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
3783	29.38	kd	CGS001-283455	KSR2	RAF family			
3784	29.37	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3785	29.35	kd	CGS001-4329	ALDH6A1	Aldehyde dehydrogenases			
3786	29.34	kd	CGS001-22921	MSRB2	-			
3787	29.31	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
3788	29.3	kd	CGS001-9318	COPS2	-			
3789	29.29	kd	CGS001-57215	THAP11	THAP (C2CH-type zinc finger) domain containing			
3790	29.25	kd	CGS001-23475	QPRT	-			
3791	29.23	oe	ccsbBroad304_00975	MAT2A	-			
3792	29.23	kd	CGS001-10525	HYOU1	Heat shock proteins / HSP70			
3793	29.22	kd	CGS001-114609	TIRAP	-			
3794	29.21	kd	CGS001-4856	NOV	-			
3795	29.16	cp	BRD-A70083328	secnidazole	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Microtubule inhibitor, Antiprotozoal
3796	29.16	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
3797	29.12	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
3798	29.1	oe	ccsbBroad304_02840	PISD	Decarboxylases			
3799	29.1	kd	CGS001-6871	TADA2A	-			
3800	29.04	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
3801	29.04	kd	CGS001-3566	IL4R	IL-2 receptor family			
3802	29.03	oe	ccsbBroad304_00036	AFP	-			
3803	29.01	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
3804	29.01	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
3805	29.01	kd	CGS001-24140	FTSJ1	-			
3806	28.98	cc		SMAD family LOF	-			
3807	28.98	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
3808	28.96	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
3809	28.93	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
3810	28.93	kd	CGS001-51451	LCMT1	-			
3811	28.92	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
3812	28.91	kd	CGS001-29946	SERTAD3	-			
3813	28.9	oe	ccsbBroad304_00099	ARG2	Arginase			
3814	28.9	kd	CGS001-51655	RASD1	-			
3815	28.88	oe	ccsbBroad304_07592	CEPT1	-			
3816	28.88	oe	ccsbBroad304_03269	CD320	CD molecules			
3817	28.88	kd	CGS001-22938	SNW1	-			
3818	28.85	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
3819	28.81	kd	CGS001-11182	SLC2A6	Solute carriers			
3820	28.81	kd	CGS001-5193	PEX12	-			
3821	28.79	kd	CGS001-7862	BRPF1	Non-enzymatic BRD containing proteins			
3822	28.78	oe	ccsbBroad304_06711	PFAS	-			
3823	28.78	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
3824	28.76	kd	CGS001-8829	NRP1	CD molecules			
3825	28.74	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
3826	28.72	kd	CGS001-1650	DDOST	-			
3827	28.65	kd	CGS001-7852	CXCR4	Chemokine receptors			
3828	28.62	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
3829	28.6	kd	CGS001-10755	GIPC1	-			
3830	28.59	oe	ccsbBroad304_10207	ERLIN1	-			
3831	28.59	kd	CGS001-873	CBR1	Prostaglandin synthases			
3832	28.58	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
3833	28.57	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
3834	28.57	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3835	28.56	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
3836	28.55	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
3837	28.53	cp	BRD-A12560204	nitrendipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1H, CACNA1S, CACNA2D2, CACNB2, CACNG1, KCNN4	Calcium channel blocker
3838	28.53	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
3839	28.52	kd	CGS001-3176	HNMT	-			
3840	28.51	kd	CGS001-5073	PARN	-			
3841	28.5	kd	CGS001-23429	RYBP	-			
3842	28.5	kd	CGS001-2787	GNG5	-			
3843	28.49	kd	CGS001-8870	IER3	-			
3844	28.48	kd	CGS001-58478	ENOPH1	-			
3845	28.47	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
3846	28.46	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
3847	28.46	kd	CGS001-53836	GPR87	GPCR / Class A : Orphans			
3848	28.42	kd	CGS001-2621	GAS6	-			
3849	28.39	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
3850	28.33	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
3851	28.33	oe	ccsbBroad304_08480	PNPO	-			
3852	28.33	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
3853	28.33	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3854	28.32	kd	CGS001-26520	TIMM9	-			
3855	28.3	kd	CGS001-54386	TERF2IP	-			
3856	28.3	kd	CGS001-9759	HDAC4	Histone deacetylases			
3857	28.29	kd	CGS001-7879	RAB7A	RAB, member RAS oncogene			
3858	28.28	kd	CGS001-6098	ROS1	Type XVII RTKs: ROS receptors			
3859	28.27	kd	CGS001-9805	SCRN1	-			
3860	28.25	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
3861	28.19	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
3862	28.18	cc		ATP synthase inhibitor	-			
3863	28.18	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
3864	28.18	kd	CGS001-7056	THBD	CD molecules			
3865	28.16	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
3866	28.16	kd	CGS001-595	CCND1	-			
3867	28.15	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
3868	28.15	kd	CGS001-6727	SRP14	-			
3869	28.11	kd	CGS001-1649	DDIT3	-			
3870	28.1	kd	CGS001-23647	ARFIP2	-			
3871	28.08	kd	CGS001-57222	ERGIC1	-			
3872	28.05	kd	CGS001-64223	MLST8	WD repeat domain containing			
3873	28.05	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
3874	28.04	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
3875	28.01	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
3876	27.96	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
3877	27.96	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3878	27.94	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
3879	27.93	kd	CGS001-2776	GNAQ	-			
3880	27.91	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
3881	27.86	kd	CGS001-3242	HPD	Oxidoreductases			
3882	27.85	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
3883	27.85	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
3884	27.82	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
3885	27.8	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
3886	27.79	kd	CGS001-3419	IDH3A	-			
3887	27.79	kd	CGS001-10421	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3888	27.73	kd	CGS001-3669	ISG20	-			
3889	27.72	kd	CGS001-6919	TCEA2	-			
3890	27.72	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3891	27.71	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
3892	27.69	kd	CGS001-1737	DLAT	-			
3893	27.65	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
3894	27.65	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
3895	27.63	cc		PPAR receptor agonist	-			
3896	27.63	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
3897	27.63	kd	CGS001-5050	PAFAH1B3	-			
3898	27.62	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
3899	27.62	kd	CGS001-199704	ZNF585A	Zinc fingers, C2H2-type			
3900	27.62	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
3901	27.54	oe	ccsbBroad304_06671	OPA1	-			
3902	27.54	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
3903	27.52	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
3904	27.51	cc		Wnt family LOF	-			
3905	27.5	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
3906	27.49	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
3907	27.48	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
3908	27.45	kd	CGS001-55612	FERMT1	Fermitins			
3909	27.44	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
3910	27.43	kd	CGS001-4860	PNP	-			
3911	27.42	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
3912	27.39	kd	CGS001-2565	GABRG1	GABA receptors			
3913	27.38	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
3914	27.37	kd	CGS001-5571	PRKAG1	AMPK subfamily			
3915	27.36	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
3916	27.36	kd	CGS001-6591	SNAI2	Snail homologs			
3917	27.35	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
3918	27.34	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
3919	27.27	kd	CGS001-4199	ME1	-			
3920	27.26	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
3921	27.24	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
3922	27.22	kd	CGS001-891	CCNB1	-			
3923	27.19	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
3924	27.19	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
3925	27.18	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
3926	27.16	oe	ccsbBroad304_06888	RPN1	-			
3927	27.15	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
3928	27.14	kd	CGS001-9354	UBE4A	U-box domain containing			
3929	27.13	kd	CGS001-1606	DGKA	EF-hand domain containing			
3930	27.11	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
3931	27.08	kd	CGS001-1545	CYP1B1	Cytochrome P450s			
3932	27.07	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
3933	27.06	kd	CGS001-1642	DDB1	-			
3934	27.05	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
3935	27.05	kd	CGS001-29775	CARD10	-			
3936	27.04	oe	ccsbBroad304_07101	TSC2	-			
3937	27.01	cc		Glucocorticoid receptor agonist	-			
3938	27	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
3939	27	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
3940	26.98	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
3941	26.97	cp	BRD-K37516142	idebenone	Calcium channel modulator			Calcium channel modulator
3942	26.96	kd	CGS001-10614	HEXIM1	-			
3943	26.95	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
3944	26.94	kd	CGS001-843	CASP10	Caspases			
3945	26.94	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3946	26.93	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
3947	26.93	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
3948	26.92	kd	CGS001-7849	PAX8	Paired boxes			
3949	26.91	oe	ccsbBroad304_02092	SYNGR3	-			
3950	26.89	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
3951	26.87	kd	CGS001-2770	GNAI1	-			
3952	26.86	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3953	26.84	kd	CGS001-63948	DMRTB1	-			
3954	26.84	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
3955	26.83	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
3956	26.82	kd	CGS001-4904	YBX1	-			
3957	26.79	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
3958	26.76	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
3959	26.75	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
3960	26.74	kd	CGS001-7511	XPNPEP1	Methionyl aminopeptidase			
3961	26.73	kd	CGS001-5982	RFC2	ATPases / AAA-type			
3962	26.72	kd	CGS001-5962	RDX	-			
3963	26.71	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3964	26.7	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
3965	26.69	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
3966	26.68	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
3967	26.67	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
3968	26.66	kd	CGS001-54512	EXOSC4	-			
3969	26.65	kd	CGS001-5696	PSMB8	Proteasome (prosome, macropain) subunits			
3970	26.62	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
3971	26.56	kd	CGS001-415116	PIM3	PIM family			
3972	26.53	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
3973	26.51	kd	CGS001-11320	MGAT4A	-			
3974	26.51	kd	CGS001-57822	GRHL3	-			
3975	26.5	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
3976	26.49	cp	BRD-A49172652	lansoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4, CYP3A5	ATPase inhibitor
3977	26.44	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
3978	26.42	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3979	26.42	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
3980	26.4	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
3981	26.39	kd	CGS001-2138	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
3982	26.38	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
3983	26.36	kd	CGS001-84108	PCGF6	Polycomb group ring fingers			
3984	26.32	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
3985	26.32	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
3986	26.3	kd	CGS001-2959	GTF2B	General transcription factors			
3987	26.29	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
3988	26.27	kd	CGS001-1356	CP	-			
3989	26.25	kd	CGS001-10795	ZNF268	Zinc fingers, C2H2-type			
3990	26.19	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
3991	26.19	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
3992	26.12	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
3993	26.1	kd	CGS001-2523	FUT1	Fucosyltransferases			
3994	26.06	kd	CGS001-1128	CHRM1	Cholinergic receptors			
3995	26.05	kd	CGS001-58472	SQRDL	-			
3996	26	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
3997	25.99	kd	CGS001-204851	HIPK1	HIPK subfamily			
3998	25.97	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
3999	25.97	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
4000	25.93	kd	CGS001-2235	FECH	-			
4001	25.9	kd	CGS001-9712	USP6NL	-			
4002	25.88	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
4003	25.88	kd	CGS001-257397	TAB3	-			
4004	25.88	kd	CGS001-1962	EHHADH	-			
4005	25.84	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
4006	25.83	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4007	25.82	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4008	25.82	kd	CGS001-8741	TNFSF13	CD molecules			
4009	25.82	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
4010	25.81	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
4011	25.81	cp	BRD-K54316499	tolterodine	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRM1, CHRM4, CHRM5	Acetylcholine receptor antagonist
4012	25.8	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
4013	25.8	kd	CGS001-2664	GDI1	-			
4014	25.78	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
4015	25.77	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
4016	25.75	kd	CGS001-10221	TRIB1	Trbl family			
4017	25.74	cp	BRD-K40758068	efavirenz	HIV protease inhibitor		CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5	HIV protease inhibitor
4018	25.71	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
4019	25.71	cp	BRD-A39390670	rabeprazole	ATPase inhibitor		ATP4A, CYP2C19	ATPase inhibitor, Gastrin inhibitor
4020	25.69	kd	CGS001-6617	SNAPC1	-			
4021	25.65	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
4022	25.65	kd	CGS001-306	ANXA3	Annexins			
4023	25.64	kd	CGS001-949	SCARB1	-			
4024	25.61	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
4025	25.57	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
4026	25.55	oe	ccsbBroad304_08888	ACD	-			
4027	25.51	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
4028	25.51	kd	CGS001-4316	MMP7	Matrix metallopeptidase			
4029	25.48	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
4030	25.47	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
4031	25.46	cc		IGF-1 inhibitor	-			
4032	25.46	kd	CGS001-204	AK2	Adenylate kinases			
4033	25.44	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
4034	25.43	kd	CGS001-112858	TP53RK	Bud32 family			
4035	25.38	kd	CGS001-190	NR0B1	DAX-like receptors			
4036	25.31	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
4037	25.29	kd	CGS001-7360	UGP2	-			
4038	25.27	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
4039	25.25	kd	CGS001-164091	PAQR7	-			
4040	25.21	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
4041	25.2	kd	CGS001-3586	IL10	Interleukins and interleukin receptors			
4042	25.14	kd	CGS001-51588	PIAS4	Zinc fingers, MIZ-type			
4043	25.09	cc		TGF beta receptor inhibitor	-			
4044	25.04	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
4045	25.02	kd	CGS001-9474	ATG5	-			
4046	25.01	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
4047	24.99	kd	CGS001-6210	RPS15A	S ribosomal proteins			
4048	24.98	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
4049	24.98	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
4050	24.98	kd	CGS001-162655	ZNF519	Zinc fingers, C2H2-type			
4051	24.98	kd	CGS001-5576	PRKAR2A	Protein kinase A			
4052	24.95	kd	CGS001-50943	FOXP3	Forkhead boxes			
4053	24.92	kd	CGS001-57147	SCYL3	-			
4054	24.87	kd	CGS001-54556	ING3	Zinc fingers, PHD-type			
4055	24.85	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
4056	24.8	kd	CGS001-9641	IKBKE	IKK family			
4057	24.8	kd	CGS001-9034	CCRL2	Chemokine receptors			
4058	24.78	kd	CGS001-4849	CNOT3	-			
4059	24.77	kd	CGS001-6775	STAT4	SH2 domain containing			
4060	24.76	kd	CGS001-861	RUNX1	-			
4061	24.76	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
4062	24.75	kd	CGS001-3459	IFNGR1	Interferon receptor family			
4063	24.73	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
4064	24.7	kd	CGS001-10613	ERLIN1	-			
4065	24.7	kd	CGS001-11214	AKAP13	A-kinase anchor proteins			
4066	24.68	kd	CGS001-11129	CLASRP	-			
4067	24.64	cp	BRD-K32398298	alprazolam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, CYP3A5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
4068	24.63	kd	CGS001-58528	RRAGD	-			
4069	24.62	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
4070	24.61	oe	ccsbBroad304_08709	SCYL3	-			
4071	24.61	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
4072	24.6	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
4073	24.58	kd	CGS001-8449	DHX16	DEAH-boxes			
4074	24.57	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
4075	24.55	kd	CGS001-256364	EML3	WD repeat domain containing			
4076	24.54	kd	CGS001-27161	EIF2C2	-			
4077	24.53	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
4078	24.53	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
4079	24.52	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
4080	24.5	oe	ccsbBroad304_07798	EXOC3	-			
4081	24.48	kd	CGS001-2242	FES	Fer family			
4082	24.46	kd	CGS001-7100	TLR5	Toll-like receptor family			
4083	24.33	kd	CGS001-9903	KLHL21	BTB/POZ domain containing			
4084	24.32	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
4085	24.29	kd	CGS001-51174	TUBD1	Tubulins			
4086	24.26	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
4087	24.25	cc		Rho associated kinase inhibitor	-			
4088	24.22	oe	ccsbBroad304_06188	F10	Chymotrypsin			
4089	24.2	kd	CGS001-23408	SIRT5	Histone deacetylases			
4090	24.17	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
4091	24.16	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
4092	24.15	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
4093	24.09	kd	CGS001-6647	SOD1	-			
4094	24.04	kd	CGS001-58497	PRUNE	-			
4095	24.04	kd	CGS001-10390	CEPT1	-			
4096	24.02	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
4097	24.02	kd	CGS001-51601	LIPT1	-			
4098	24.02	kd	CGS001-515	ATP5F1	ATPases / F-type			
4099	24.01	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
4100	24.01	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
4101	24	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
4102	24	kd	CGS001-7342	UBP1	-			
4103	23.99	oe	ccsbBroad304_00262	CD59	CD molecules			
4104	23.98	cc		IL4 Pathway LOF	-			
4105	23.96	kd	CGS001-79139	DERL1	-			
4106	23.93	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
4107	23.93	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
4108	23.91	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
4109	23.9	kd	CGS001-2172	FABP6	Fatty acid binding protein family			
4110	23.86	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
4111	23.81	kd	CGS001-26523	EIF2C1	-			
4112	23.78	kd	CGS001-10873	ME3	-			
4113	23.76	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
4114	23.76	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
4115	23.73	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4116	23.71	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
4117	23.65	kd	CGS001-1810	DR1	-			
4118	23.61	kd	CGS001-4811	NID1	-			
4119	23.61	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
4120	23.59	kd	CGS001-3098	HK1	-			
4121	23.56	cc		Serpin peptidase inhibitors LOF	-			
4122	23.56	kd	CGS001-4094	MAF	-			
4123	23.55	kd	CGS001-66008	TRAK2	-			
4124	23.52	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
4125	23.52	kd	CGS001-64080	RBKS	-			
4126	23.48	kd	CGS001-85442	KNDC1	-			
4127	23.48	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
4128	23.46	oe	ccsbBroad304_06264	GBP2	-			
4129	23.45	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
4130	23.44	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
4131	23.43	oe	ccsbBroad304_00789	HSBP1	-			
4132	23.43	kd	CGS001-7077	TIMP2	-			
4133	23.43	kd	CGS001-8535	CBX4	-			
4134	23.42	kd	CGS001-9337	CNOT8	-			
4135	23.34	cc		GABA receptor antagonist	-			
4136	23.34	kd	CGS001-3927	LASP1	-			
4137	23.32	cc		PKC activator	-			
4138	23.32	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
4139	23.32	kd	CGS001-290	ANPEP	Aminopeptidase N			
4140	23.32	kd	CGS001-185	AGTR1	Angiotensin receptors			
4141	23.3	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
4142	23.28	kd	CGS001-9184	BUB3	WD repeat domain containing			
4143	23.25	cc		RAF inhibitor	-			
4144	23.23	kd	CGS001-2224	FDPS	Lanosterol biosynthesis pathway			
4145	23.21	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
4146	23.19	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
4147	23.15	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
4148	23.13	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
4149	23.1	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
4150	23.08	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
4151	23.08	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
4152	23.05	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4153	23.03	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
4154	23.01	kd	CGS001-286380	FOXD4L3	-			
4155	22.99	kd	CGS001-488	ATP2A2	Calcium-ATPases			
4156	22.98	kd	CGS001-10318	TNIP1	-			
4157	22.98	kd	CGS001-30001	ERO1L	-			
4158	22.95	cc		Serotonin receptor antagonist	-			
4159	22.94	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
4160	22.93	kd	CGS001-3660	IRF2	-			
4161	22.88	kd	CGS001-572	BAD	-			
4162	22.8	oe	ccsbBroad304_07832	XPO7	Exportins			
4163	22.79	kd	CGS001-8678	BECN1	-			
4164	22.76	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
4165	22.75	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
4166	22.75	kd	CGS001-10765	KDM5B	Histone demethylases			
4167	22.74	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
4168	22.73	oe	ccsbBroad304_07220	CDC45	-			
4169	22.71	kd	CGS001-375	ARF1	ADP-ribosylation factors			
4170	22.7	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
4171	22.7	kd	CGS001-6883	TAF12	-			
4172	22.69	kd	CGS001-3298	HSF2	-			
4173	22.66	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
4174	22.66	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
4175	22.65	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
4176	22.65	kd	CGS001-9276	COPB2	WD repeat domain containing			
4177	22.64	kd	CGS001-2852	GPER	-			
4178	22.6	kd	CGS001-3516	RBPJ	-			
4179	22.58	oe	ccsbBroad304_07178	ZFP112	-			
4180	22.57	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
4181	22.56	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
4182	22.51	kd	CGS001-103	ADAR	-			
4183	22.46	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
4184	22.44	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
4185	22.43	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
4186	22.42	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
4187	22.42	kd	CGS001-9568	GABBR2	GABA receptors			
4188	22.41	kd	CGS001-4122	MAN2A2	-			
4189	22.4	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
4190	22.39	oe	ccsbBroad304_03310	LCMT1	-			
4191	22.39	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
4192	22.38	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
4193	22.38	kd	CGS001-10797	MTHFD2	-			
4194	22.36	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
4195	22.35	kd	CGS001-673	BRAF	RAF family			
4196	22.34	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
4197	22.32	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
4198	22.3	kd	CGS001-6217	RPS16	S ribosomal proteins			
4199	22.29	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
4200	22.28	kd	CGS001-3123	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
4201	22.27	oe	ccsbBroad304_00376	CSK	Csk family			
4202	22.27	kd	CGS001-10628	TXNIP	-			
4203	22.25	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
4204	22.21	kd	CGS001-7150	TOP1	DNA Topoisomerases			
4205	22.2	cc		PI3K inhibitor	-			
4206	22.19	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
4207	22.16	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
4208	22.16	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
4209	22.12	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
4210	22.12	kd	CGS001-3845	KRAS	RAS subfamily			
4211	22.11	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
4212	22.08	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
4213	22.04	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
4214	22.02	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
4215	21.99	kd	CGS001-1635	DCTD	-			
4216	21.94	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
4217	21.92	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
4218	21.91	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
4219	21.9	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
4220	21.86	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
4221	21.84	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
4222	21.83	oe	ccsbBroad304_06952	SKP1	-			
4223	21.83	kd	CGS001-6643	SNX2	Sorting nexins			
4224	21.77	cp	BRD-K29653726	topiramate	Carbonic anhydrase inhibitor		CA2, CA4, GRIK1, CA1, CA12, CA7, CYP2C19, CYP3A4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA1, SCN1A, SCN5A	Carbonic anhydrase inhibitor, Glutamate receptor antagonist, Kainate receptor antagonist
4225	21.73	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
4226	21.56	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
4227	21.52	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
4228	21.5	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
4229	21.5	kd	CGS001-5883	RAD9A	-			
4230	21.49	kd	CGS001-25949	SYF2	-			
4231	21.48	kd	CGS001-8334	HIST1H2AC	Histones / Replication-dependent			
4232	21.44	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
4233	21.43	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
4234	21.43	kd	CGS001-25948	KBTBD2	BTB/POZ domain containing			
4235	21.41	kd	CGS001-84890	ADO	-			
4236	21.38	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
4237	21.24	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4238	21.19	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
4239	21.17	kd	CGS001-1445	CSK	Csk family			
4240	21.15	cp	BRD-K73196317	urapidil	Adrenergic receptor antagonist		HTR1A	Adrenergic receptor antagonist
4241	21.13	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
4242	21.13	kd	CGS001-51079	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
4243	21.02	kd	CGS001-3725	JUN	basic leucine zipper proteins			
4244	21.02	kd	CGS001-116535	MRGPRF	GPCR / Class A : Orphans			
4245	20.96	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
4246	20.95	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
4247	20.94	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
4248	20.9	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
4249	20.86	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
4250	20.79	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
4251	20.78	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
4252	20.74	kd	CGS001-65123	INTS3	-			
4253	20.7	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
4254	20.7	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
4255	20.61	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
4256	20.56	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
4257	20.51	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
4258	20.43	cp	BRD-A79903587	tegafur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
4259	20.36	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
4260	20.34	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
4261	20.3	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
4262	20.26	kd	CGS001-4221	MEN1	-			
4263	20.23	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4264	20.2	kd	CGS001-310	ANXA7	Annexins			
4265	20.16	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
4266	20.16	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
4267	20.11	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
4268	20.05	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
4269	20.01	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
4270	19.95	cc		Sigma receptor antagonist	-			
4271	19.91	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
4272	19.87	kd	CGS001-8525	DGKZ	-			
4273	19.86	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
4274	19.84	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
4275	19.79	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
4276	19.71	kd	CGS001-5686	PSMA5	Proteasome subunits			
4277	19.67	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
4278	19.55	cp	BRD-K22009844	phenprobamate	Muscle relaxant			Muscle relaxant
4279	19.53	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
4280	19.53	kd	CGS001-1111	CHEK1	CHK1 subfamily			
4281	19.34	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
4282	19.26	kd	CGS001-84923	FAM104A	-			
4283	19.24	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
4284	19.2	kd	CGS001-9643	MORF4L2	-			
4285	19.15	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
4286	19.14	kd	CGS001-5900	RALGDS	-			
4287	19.12	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
4288	19.1	cp	BRD-K82357231	desloratadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4289	19.01	kd	CGS001-58533	SNX6	Sorting nexins			
4290	18.96	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
4291	18.87	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
4292	18.78	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
4293	18.7	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
4294	18.69	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
4295	18.63	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4296	18.61	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
4297	18.55	oe	ccsbBroad304_00420	DAP	-			
4298	18.52	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
4299	18.49	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
4300	18.38	kd	CGS001-10285	SMNDC1	Tudor domain containing			
4301	18.33	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
4302	18.33	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
4303	18.26	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
4304	18.22	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
4305	18.13	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
4306	18.12	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
4307	18.09	cc		DNA dependent protein kinase inhibitor	-			
4308	17.98	kd	CGS001-6897	TARS	Aminoacyl tRNA synthetases / Class II			
4309	17.95	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
4310	17.95	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4311	17.9	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
4312	17.81	cc		ATPase inhibitor	-			
4313	17.76	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
4314	17.73	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
4315	17.7	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4316	17.7	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
4317	17.67	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
4318	17.67	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
4319	17.58	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4320	17.48	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
4321	17.44	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
4322	17.38	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
4323	17.3	cc		PKC inhibitor	-			
4324	17.24	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
4325	17.22	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
4326	17.22	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
4327	17.17	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
4328	17.17	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
4329	17.14	kd	CGS001-10105	PPIF	-			
4330	16.8	kd	CGS001-1305	COL13A1	Collagens			
4331	16.66	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
4332	16.63	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
4333	16.58	kd	CGS001-3421	IDH3G	-			
4334	16.55	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
4335	16.54	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
4336	16.47	kd	CGS001-2769	GNA15	-			
4337	16.21	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
4338	16.21	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
4339	16.17	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4340	16.17	kd	CGS001-1362	CPD	Carboxypeptidase A			
4341	16.11	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
4342	16.07	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
4343	15.95	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
4344	15.79	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
4345	15.55	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
4346	15.5	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
4347	15.44	kd	CGS001-2475	MTOR	FRAP subfamily			
4348	15.42	cp	BRD-K88679075	methandriol	Androgenic steroid			Androgenic steroid
4349	15.11	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
4350	15.1	cc		Nucleoside reverse transcriptase inhibitor	-			
4351	15	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
4352	14.93	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
4353	14.81	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4354	14.74	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
4355	14.69	cp	BRD-K13800121	parecoxib	Cyclooxygenase inhibitor		LTF, PTGS2	Cyclooxygenase inhibitor
4356	14.54	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
4357	14.5	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
4358	14.4	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
4359	14.39	cc		FGFR inhibitor	-			
4360	14.32	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
4361	14.2	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
4362	14.08	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
4363	14.07	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
4364	14.06	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
4365	14.01	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
4366	13.96	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
4367	13.86	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
4368	13.65	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
4369	13.34	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
4370	13.23	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
4371	13.23	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
4372	13.2	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
4373	13.12	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
4374	13.07	cp	BRD-K99063460	didanosine	Nucleoside reverse transcriptase inhibitor		PNP	Nucleoside reverse transcriptase inhibitor
4375	13.07	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
4376	13.06	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
4377	13.04	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
4378	13.03	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
4379	12.98	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
4380	12.9	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
4381	12.88	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
4382	12.78	kd	CGS001-5608	MAP2K6	MAPKK:STE7 family			
4383	12.66	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
4384	12.64	cp	BRD-A11990600	lorazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, TSPO	Benzodiazepine receptor agonist
4385	12.64	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
4386	12.53	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
4387	12.5	kd	CGS001-51268	PIPOX	-			
4388	12.46	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
4389	12.27	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
4390	12.11	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4391	12	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
4392	11.77	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
4393	11.59	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
4394	11.56	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
4395	11.55	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
4396	11.4	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
4397	11.18	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
4398	11.07	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
4399	10.92	cp	BRD-K00673382	famotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
4400	10.85	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
4401	10.77	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
4402	10.65	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
4403	10.61	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
4404	10.59	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
4405	10.48	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
4406	10.42	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4407	10.41	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
4408	10.39	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
4409	10.33	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
4410	10.29	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
4411	10.25	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
4412	10.2	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
4413	10.19	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
4414	10.09	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
4415	9.98	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
4416	9.85	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
4417	9.82	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
4418	9.82	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
4419	9.61	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
4420	9.53	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
4421	9.46	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
4422	9.46	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
4423	9.4	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
4424	9.25	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
4425	9.15	cp	BRD-K29530284	amlexanox	Histamine receptor modulator		FGF1, IL3, S100A12, S100A13	Histamine receptor modulator
4426	8.9	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
4427	8.88	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
4428	8.88	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
4429	8.73	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
4430	8.58	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
4431	8.54	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
4432	8.46	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
4433	8.32	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
4434	8.32	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
4435	8.31	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
4436	8.28	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
4437	7.7	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
4438	7.64	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
4439	7.26	cc		Akt Signaling LOF	-			
4440	7.26	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4441	6.33	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
4442	6.2	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
4443	5.91	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
4444	5.86	cc		Reverse transcriptase inhibitor	-			
4445	5.78	cc		VEGFR inhibitor	-			
4446	5.77	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
4447	5.76	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4448	5.25	cc		PRD class homeoboxes and psudogenes LOF	-			
4449	4.9	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
4450	4.75	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
4451	-4.29	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
4452	-6.1	cp	BRD-K04196797	oxcarbazepine	Sodium channel blocker		CYP2C19, CYP3A4, CYP3A5, SCN1A, SCN3A, SCN5A	Sodium channel blocker
4453	-6.17	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
4454	-6.2	cc		DNA Replication LOF	-			
4455	-6.4	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
4456	-6.7	cp	BRD-K47278471	diphenhydramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4457	-6.76	cp	BRD-K34508425	KUC103898N	-666			-666
4458	-6.76	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
4459	-7	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
4460	-7.11	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
4461	-7.11	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
4462	-7.19	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
4463	-7.24	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
4464	-7.33	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
4465	-7.44	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
4466	-7.61	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
4467	-8.88	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
4468	-8.89	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
4469	-9.1	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
4470	-9.17	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4471	-9.19	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
4472	-9.35	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
4473	-9.47	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
4474	-9.52	cc		Minor histocompatibility antigens LOF	-			
4475	-9.52	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
4476	-9.6	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
4477	-9.87	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
4478	-9.89	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4479	-9.89	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
4480	-9.9	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4481	-9.9	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4482	-10.03	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
4483	-10.07	cp	BRD-K62858456	lomerizine	Calcium channel blocker		ABCB1, CACNA1B, SCN5A	Calcium channel blocker
4484	-10.21	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
4485	-10.32	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
4486	-10.43	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
4487	-10.54	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
4488	-10.55	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
4489	-10.59	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
4490	-10.79	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
4491	-10.9	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
4492	-11.07	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
4493	-11.09	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
4494	-11.1	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
4495	-11.14	cp	BRD-K98493452	honokiol	AKT inhibitor		ALOX5, PTGS1, PTGS2	AKT inhibitor
4496	-11.16	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
4497	-11.21	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
4498	-11.24	kd	CGS001-29968	PSAT1	-			
4499	-11.44	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4500	-11.51	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
4501	-11.56	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
4502	-11.69	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
4503	-12.03	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
4504	-12.04	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
4505	-12.05	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
4506	-12.14	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
4507	-12.15	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
4508	-12.18	cc		Sterol demethylase inhibitor	-			
4509	-12.23	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
4510	-12.41	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
4511	-12.5	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
4512	-12.54	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
4513	-12.56	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
4514	-12.61	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
4515	-12.75	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
4516	-12.75	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
4517	-12.79	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
4518	-13.21	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
4519	-13.25	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4520	-13.34	cp	BRD-A24381660	zeranol	Estrogen receptor agonist			Estrogen receptor agonist
4521	-13.42	kd	CGS001-203	AK1	Adenylate kinases			
4522	-13.6	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
4523	-13.61	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
4524	-13.65	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
4525	-13.8	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
4526	-13.82	cp	BRD-K81916719	triclabendazole	Microtubule inhibitor		DNMT1	Microtubule inhibitor
4527	-14.01	cc		PDGFR/KIT inhibitor	-			
4528	-14.05	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
4529	-14.2	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
4530	-14.26	cp	BRD-K02227374	milnacipran	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Serotonin reuptake inhibitor
4531	-14.29	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
4532	-14.45	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
4533	-14.46	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
4534	-14.94	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
4535	-15.13	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
4536	-15.22	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
4537	-15.3	cc		HMGCR inhibitor	-			
4538	-15.41	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
4539	-15.42	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
4540	-15.52	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
4541	-15.7	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
4542	-15.85	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
4543	-15.96	oe	ccsbBroad304_02197	VPS26A	-			
4544	-15.99	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
4545	-16.05	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
4546	-16.23	kd	CGS001-55239	OGFOD1	-			
4547	-16.27	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
4548	-16.29	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
4549	-16.35	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
4550	-16.44	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
4551	-16.52	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
4552	-16.61	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4553	-16.67	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
4554	-16.8	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
4555	-16.88	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
4556	-16.95	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
4557	-17.03	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
4558	-17.07	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
4559	-17.12	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
4560	-17.34	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
4561	-17.57	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
4562	-17.62	kd	CGS001-7525	YES1	Src family			
4563	-17.7	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
4564	-17.7	kd	CGS001-8772	FADD	-			
4565	-17.76	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
4566	-17.81	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
4567	-17.86	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
4568	-17.9	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
4569	-18.05	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
4570	-18.05	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
4571	-18.17	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
4572	-18.23	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
4573	-18.33	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
4574	-18.36	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
4575	-18.36	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
4576	-18.45	kd	CGS001-9212	AURKB	Aurora kinase			
4577	-18.58	kd	CGS001-5578	PRKCA	Delta subfamily			
4578	-18.63	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
4579	-18.69	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
4580	-18.75	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
4581	-18.84	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
4582	-18.88	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
4583	-18.88	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
4584	-18.95	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4585	-18.96	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
4586	-18.97	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4587	-19.06	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4588	-19.1	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
4589	-19.27	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
4590	-19.3	kd	CGS001-35	ACADS	-			
4591	-19.32	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
4592	-19.47	kd	CGS001-6275	S100A4	EF-hand domain containing			
4593	-19.5	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
4594	-19.72	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4595	-19.74	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
4596	-19.74	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
4597	-19.75	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
4598	-19.78	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
4599	-19.88	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
4600	-20.01	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
4601	-20.07	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
4602	-20.07	kd	CGS001-132	ADK	Adenosine turnover			
4603	-20.08	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
4604	-20.08	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
4605	-20.12	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4606	-20.24	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
4607	-20.31	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
4608	-20.41	kd	CGS001-79006	METRN	-			
4609	-20.48	kd	CGS001-5110	PCMT1	-			
4610	-20.48	kd	CGS001-1675	CFD	Complement system			
4611	-20.51	kd	CGS001-5362	PLXNA2	Plexins			
4612	-20.53	kd	CGS001-998	CDC42	-			
4613	-20.6	kd	CGS001-165082	GPR113	Adhesion Class GPCRs			
4614	-20.61	kd	CGS001-1861	TOR1A	-			
4615	-20.7	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
4616	-20.75	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
4617	-20.8	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
4618	-20.95	cc		Zinc fingers RanBP2 type LOF	-			
4619	-21.05	kd	CGS001-18	ABAT	GABA turnover			
4620	-21.09	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
4621	-21.09	kd	CGS001-10058	ABCB6	ATP binding cassette transporters / subfamily B			
4622	-21.13	kd	CGS001-23499	MACF1	EF-hand domain containing			
4623	-21.19	kd	CGS001-54884	RETSAT	-			
4624	-21.35	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
4625	-21.37	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
4626	-21.42	kd	CGS001-5613	PRKX	Protein kinase A			
4627	-21.43	kd	CGS001-900	CCNG1	-			
4628	-21.46	cp	BRD-K85503079	perospirone	Dopamine receptor antagonist		DRD2, HTR2A, DRD3, DRD4, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
4629	-21.58	cp	BRD-K99447003	enalaprilat	ACE inhibitor		ACE	ACE inhibitor
4630	-21.58	kd	CGS001-4171	MCM2	-			
4631	-21.63	kd	CGS001-5664	PSEN2	Presenilin			
4632	-21.64	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
4633	-21.65	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
4634	-21.72	kd	CGS001-29880	ALG5	Glycosyltransferase family 2 domain containing			
4635	-21.73	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
4636	-21.79	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
4637	-21.83	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
4638	-21.88	kd	CGS001-397	ARHGDIB	Endogenous ligands			
4639	-21.9	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
4640	-21.9	kd	CGS001-4144	MAT2A	-			
4641	-22.01	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
4642	-22.09	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
4643	-22.13	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
4644	-22.15	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
4645	-22.15	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
4646	-22.2	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
4647	-22.23	kd	CGS001-9900	SV2A	Major facilitator superfamily (MFS) of transporters			
4648	-22.25	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
4649	-22.25	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
4650	-22.25	kd	CGS001-84759	PCGF1	Polycomb group ring fingers			
4651	-22.28	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
4652	-22.31	kd	CGS001-10381	TUBB3	Tubulins			
4653	-22.35	kd	CGS001-8720	MBTPS1	Subtilisin			
4654	-22.37	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
4655	-22.37	kd	CGS001-1465	CSRP1	-			
4656	-22.37	kd	CGS001-501	ALDH7A1	Aldehyde dehydrogenases			
4657	-22.38	oe	ccsbBroad304_14242	MCCC2	-			
4658	-22.39	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
4659	-22.4	kd	CGS001-6856	SYPL1	-			
4660	-22.4	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
4661	-22.44	kd	CGS001-6885	MAP3K7	MAPKKK:TAK1 subfamily			
4662	-22.51	kd	CGS001-4439	MSH5	-			
4663	-22.53	kd	CGS001-6721	SREBF2	Basic helix-loop-helix proteins			
4664	-22.56	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
4665	-22.57	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
4666	-22.57	kd	CGS001-4067	LYN	Src family			
4667	-22.64	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
4668	-22.71	kd	CGS001-5257	PHKB	-			
4669	-22.71	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
4670	-22.81	kd	CGS001-26277	TINF2	-			
4671	-22.82	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
4672	-22.82	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
4673	-22.83	kd	CGS001-10673	TNFSF13B	CD molecules			
4674	-22.85	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
4675	-22.95	kd	CGS001-2057	EPOR	Prolactin receptor family			
4676	-22.98	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
4677	-23.01	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
4678	-23.05	kd	CGS001-11343	MGLL	Endocannabinoid turnover			
4679	-23.09	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
4680	-23.18	kd	CGS001-55770	EXOC2	-			
4681	-23.21	oe	ccsbBroad304_02175	MAGED1	-			
4682	-23.22	kd	CGS001-89910	UBE3B	-			
4683	-23.23	kd	CGS001-4946	OAZ1	-			
4684	-23.24	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
4685	-23.37	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
4686	-23.4	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
4687	-23.43	kd	CGS001-4254	KITLG	-			
4688	-23.46	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
4689	-23.46	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
4690	-23.49	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
4691	-23.49	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
4692	-23.52	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
4693	-23.55	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
4694	-23.63	kd	CGS001-3821	KLRC1	CD molecules			
4695	-23.65	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
4696	-23.65	kd	CGS001-10489	LRRC41	-			
4697	-23.81	oe	ccsbBroad304_03658	DCP1A	-			
4698	-23.82	kd	CGS001-8522	GAS7	-			
4699	-23.85	kd	CGS001-6118	RPA2	-			
4700	-23.9	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
4701	-23.92	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
4702	-23.96	cp	BRD-K52020312	metronidazole	DNA inhibitor		CYP2C8, CYP2E1, CYP3A5, CYP3A7	DNA inhibitor, Antiprotozoal
4703	-23.98	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
4704	-24	kd	CGS001-6773	STAT2	SH2 domain containing			
4705	-24.04	oe	ccsbBroad304_03405	CHRAC1	-			
4706	-24.05	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
4707	-24.05	kd	CGS001-23161	SNX13	Sorting nexins			
4708	-24.06	oe	ccsbBroad304_00648	GLRX	-			
4709	-24.06	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
4710	-24.09	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
4711	-24.09	kd	CGS001-2864	FFAR1	Fatty acid receptors			
4712	-24.1	oe	ccsbBroad304_03080	C16ORF80	-			
4713	-24.15	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
4714	-24.15	kd	CGS001-167826	OLIG3	Basic helix-loop-helix proteins			
4715	-24.17	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
4716	-24.2	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
4717	-24.2	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
4718	-24.24	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
4719	-24.25	kd	CGS001-29763	PACSIN3	-			
4720	-24.26	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
4721	-24.28	kd	CGS001-26128	KIAA1279	-			
4722	-24.3	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
4723	-24.31	kd	CGS001-10254	STAM2	-			
4724	-24.32	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
4725	-24.36	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
4726	-24.36	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
4727	-24.36	oe	ccsbBroad304_01613	STK11	LKB subfamily			
4728	-24.39	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
4729	-24.4	cc		IKK inhibitor	-			
4730	-24.44	kd	CGS001-1632	ECI1	-			
4731	-24.46	oe	ccsbBroad304_00957	M6PR	-			
4732	-24.54	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
4733	-24.55	kd	CGS001-8669	EIF3J	-			
4734	-24.57	cp	BRD-K11630072	carmofur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
4735	-24.63	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
4736	-24.64	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
4737	-24.65	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
4738	-24.74	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
4739	-24.76	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
4740	-24.78	kd	CGS001-4351	MPI	-			
4741	-24.81	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
4742	-24.82	kd	CGS001-6821	SUOX	-			
4743	-24.84	kd	CGS001-5427	POLE2	DNA polymerases			
4744	-24.86	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
4745	-24.87	kd	CGS001-55810	FOXJ2	Forkhead boxes			
4746	-24.88	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
4747	-24.89	kd	CGS001-5577	PRKAR2B	Protein kinase A			
4748	-24.94	cp	BRD-K29113274	ketoconazole	Sterol demethylase inhibitor		AR, CYP19A1, CYP21A2, CYP2C19, CYP3A5, CYP3A7, KCNA10	Sterol demethylase inhibitor
4749	-24.99	cp	BRD-K46742498	alosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
4750	-25.03	kd	CGS001-2182	ACSL4	Acyl-CoA synthetase family			
4751	-25.07	oe	ccsbBroad304_03450	TMED9	-			
4752	-25.09	kd	CGS001-25888	ZNF473	Zinc fingers, C2H2-type			
4753	-25.12	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
4754	-25.14	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
4755	-25.22	kd	CGS001-5777	PTPN6	Protein tyrosine phosphatases			
4756	-25.28	kd	CGS001-57804	POLD4	DNA polymerases			
4757	-25.29	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
4758	-25.31	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
4759	-25.34	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
4760	-25.36	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
4761	-25.44	kd	CGS001-51292	GMPR2	-			
4762	-25.46	kd	CGS001-10476	ATP5H	ATPases / F-type			
4763	-25.48	cp	BRD-A24543851	nornicotine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
4764	-25.49	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
4765	-25.5	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
4766	-25.59	kd	CGS001-899	CCNF	F-boxes / other			
4767	-25.6	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
4768	-25.61	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
4769	-25.68	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
4770	-25.71	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
4771	-25.75	kd	CGS001-5108	PCM1	-			
4772	-25.75	kd	CGS001-84539	MCHR2	GPCR / Class A : MCH receptors			
4773	-25.79	cc		Histone deacetylases LOF	-			
4774	-25.8	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
4775	-25.83	kd	CGS001-573	BAG1	-			
4776	-25.86	kd	CGS001-7089	TLE2	WD repeat domain containing			
4777	-25.86	kd	CGS001-57057	TBX20	T-boxes			
4778	-25.89	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
4779	-25.92	oe	ccsbBroad304_00238	CCNE1	-			
4780	-25.95	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
4781	-25.97	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
4782	-26.04	kd	CGS001-81848	SPRY4	-			
4783	-26.06	oe	ccsbBroad304_00529	F3	CD molecules			
4784	-26.06	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
4785	-26.06	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
4786	-26.11	kd	CGS001-116113	FOXP4	Forkhead boxes			
4787	-26.12	kd	CGS001-3912	LAMB1	Laminins			
4788	-26.16	cc		Ribonucleotide reductase inhibitor	-			
4789	-26.2	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
4790	-26.27	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
4791	-26.27	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4792	-26.27	kd	CGS001-4282	MIF	-			
4793	-26.28	kd	CGS001-23118	TAB2	-			
4794	-26.28	kd	CGS001-80762	NDFIP1	-			
4795	-26.29	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
4796	-26.3	kd	CGS001-65243	ZNF643	-			
4797	-26.31	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
4798	-26.33	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
4799	-26.35	kd	CGS001-624	BDKRB2	Bradykinin receptors			
4800	-26.38	kd	CGS001-10544	PROCR	CD molecules			
4801	-26.43	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4802	-26.49	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
4803	-26.52	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
4804	-26.52	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
4805	-26.54	kd	CGS001-4665	NAB2	-			
4806	-26.59	kd	CGS001-5037	PEBP1	-			
4807	-26.66	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
4808	-26.69	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
4809	-26.72	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
4810	-26.74	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
4811	-26.74	kd	CGS001-7280	TUBB2A	Tubulins			
4812	-26.76	kd	CGS001-23239	PHLPP1	Pleckstrin homology (PH) domain containing			
4813	-26.83	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
4814	-26.89	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
4815	-26.94	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
4816	-27.04	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
4817	-27.06	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
4818	-27.07	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
4819	-27.08	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
4820	-27.11	kd	CGS001-2079	ERH	-			
4821	-27.15	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
4822	-27.17	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
4823	-27.17	kd	CGS001-644	BLVRA	-			
4824	-27.23	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
4825	-27.25	kd	CGS001-10962	MLLT11	-			
4826	-27.27	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
4827	-27.28	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
4828	-27.29	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
4829	-27.34	kd	CGS001-5612	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
4830	-27.36	kd	CGS001-64863	METTL4	-			
4831	-27.39	kd	CGS001-2967	GTF2H3	General transcription factors			
4832	-27.42	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
4833	-27.42	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
4834	-27.43	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
4835	-27.45	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
4836	-27.46	oe	ccsbBroad304_10230	STK19	G11 family			
4837	-27.46	oe	ccsbBroad304_00152	BCAT2	-			
4838	-27.46	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
4839	-27.48	kd	CGS001-10493	VAT1	-			
4840	-27.48	kd	CGS001-1643	DDB2	WD repeat domain containing			
4841	-27.48	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
4842	-27.49	kd	CGS001-91304	C19ORF6	-			
4843	-27.51	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
4844	-27.54	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
4845	-27.54	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
4846	-27.54	kd	CGS001-2937	GSS	-			
4847	-27.55	kd	CGS001-4208	MEF2C	Myocyte enhancer factors			
4848	-27.56	kd	CGS001-3985	LIMK2	LIMK subfamily			
4849	-27.56	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
4850	-27.61	kd	CGS001-163688	CALML6	EF-hand domain containing			
4851	-27.61	kd	CGS001-383	ARG1	Arginase			
4852	-27.62	kd	CGS001-222546	RFX6	-			
4853	-27.64	kd	CGS001-51422	PRKAG2	AMPK subfamily			
4854	-27.67	kd	CGS001-9156	EXO1	-			
4855	-27.69	oe	ccsbBroad304_07337	TAF1B	-			
4856	-27.77	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
4857	-27.77	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
4858	-27.79	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
4859	-27.8	kd	CGS001-7917	BAG6	-			
4860	-27.83	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
4861	-27.83	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
4862	-27.87	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
4863	-27.87	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4864	-27.92	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
4865	-27.94	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
4866	-27.94	kd	CGS001-10165	SLC25A13	Mitochondrial amino acid transporter subfamily			
4867	-27.94	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
4868	-27.95	kd	CGS001-6804	STX1A	-			
4869	-27.98	kd	CGS001-5881	RAC3	Endogenous ligands			
4870	-28.03	kd	CGS001-378	ARF4	ADP-ribosylation factors			
4871	-28.04	kd	CGS001-85480	TSLP	-			
4872	-28.05	kd	CGS001-2735	GLI1	Zinc fingers, C2H2-type			
4873	-28.07	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
4874	-28.07	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
4875	-28.16	kd	CGS001-8702	B4GALT4	Beta 4-glycosyltransferases			
4876	-28.17	oe	ccsbBroad304_08694	TBX20	T-boxes			
4877	-28.18	kd	CGS001-7982	ST7	-			
4878	-28.18	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
4879	-28.21	kd	CGS001-10513	APPBP2	-			
4880	-28.28	kd	CGS001-100	ADA	Adenosine turnover			
4881	-28.34	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
4882	-28.34	kd	CGS001-150094	SIK1	QIK subfamily			
4883	-28.37	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
4884	-28.38	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
4885	-28.38	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
4886	-28.39	kd	CGS001-158	ADSL	-			
4887	-28.43	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4888	-28.44	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
4889	-28.45	cc		Leucine rich repeat kinase inhibitor	-			
4890	-28.45	oe	ccsbBroad304_01651	TCF7L2	-			
4891	-28.47	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
4892	-28.48	oe	ccsbBroad304_01061	NAB2	-			
4893	-28.51	kd	CGS001-27	ABL2	Abl family			
4894	-28.53	kd	CGS001-8428	STK24	YSK subfamily			
4895	-28.55	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
4896	-28.57	cp	BRD-K41903098	diphenoxylate	Opioid receptor agonist		OPRM1, OPRD1	Opioid receptor agonist
4897	-28.61	kd	CGS001-10398	MYL9	EF-hand domain containing			
4898	-28.61	kd	CGS001-4170	MCL1	-			
4899	-28.62	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
4900	-28.62	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
4901	-28.66	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
4902	-28.66	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
4903	-28.67	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
4904	-28.68	kd	CGS001-3420	IDH3B	-			
4905	-28.68	kd	CGS001-238	ALK	Leukocyte tyrosine kinase (LTK) receptor family			
4906	-28.69	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
4907	-28.7	kd	CGS001-5211	PFKL	-			
4908	-28.71	oe	ccsbBroad304_05985	CFL1	-			
4909	-28.72	kd	CGS001-22978	NT5C2	Adenosine turnover			
4910	-28.73	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
4911	-28.78	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
4912	-28.78	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
4913	-28.82	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
4914	-28.82	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
4915	-28.83	oe	ccsbBroad304_00161	BID	Endogenous ligands			
4916	-28.84	kd	CGS001-10437	IFI30	-			
4917	-28.85	kd	CGS001-7296	TXNRD1	-			
4918	-28.92	cp	BRD-K27184429	levocetirizine	Histamine receptor antagonist		HRH1, CXCL8	Histamine receptor antagonist
4919	-29.01	kd	CGS001-3431	SP110	Non-enzymatic BRD containing proteins			
4920	-29.06	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
4921	-29.09	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
4922	-29.11	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
4923	-29.14	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4924	-29.14	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
4925	-29.18	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
4926	-29.18	kd	CGS001-39	ACAT2	Lanosterol biosynthesis pathway			
4927	-29.19	oe	ccsbBroad304_06855	RDX	-			
4928	-29.19	kd	CGS001-83933	HDAC10	Histone deacetylases			
4929	-29.22	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
4930	-29.23	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4931	-29.23	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
4932	-29.23	kd	CGS001-2909	ARHGAP35	Rho GTPase activating proteins			
4933	-29.25	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
4934	-29.26	kd	CGS001-3161	HMMR	CD molecules			
4935	-29.29	kd	CGS001-55907	CMAS	-			
4936	-29.31	cp	BRD-K65910366	KUC103904N	-666			-666
4937	-29.34	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
4938	-29.39	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
4939	-29.41	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
4940	-29.44	kd	CGS001-7468	WHSC1	Zinc fingers, PHD-type			
4941	-29.44	kd	CGS001-8805	TRIM24	TIF1 family			
4942	-29.45	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
4943	-29.47	cc		NFkB pathway inhibitor	-			
4944	-29.47	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
4945	-29.48	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
4946	-29.49	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
4947	-29.5	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
4948	-29.54	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
4949	-29.62	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
4950	-29.62	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
4951	-29.67	cp	BRD-K33106058	cytarabine	Ribonucleotide reductase inhibitor		POLB, POLA1	Ribonucleotide reductase inhibitor
4952	-29.68	oe	ccsbBroad304_09284	UBE3B	-			
4953	-29.7	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
4954	-29.71	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
4955	-29.72	kd	CGS001-1147	CHUK	IKK family			
4956	-29.73	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
4957	-29.75	kd	CGS001-898	CCNE1	-			
4958	-29.79	kd	CGS001-5209	PFKFB3	-			
4959	-29.8	kd	CGS001-444	ASPH	-			
4960	-29.81	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
4961	-29.82	oe	ccsbBroad304_04616	ORMDL3	-			
4962	-29.83	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
4963	-29.83	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
4964	-29.86	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
4965	-29.88	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
4966	-29.88	kd	CGS001-5269	SERPINB6	Serine (or cysteine) peptidase inhibitors			
4967	-29.99	kd	CGS001-126823	KLHDC9	-			
4968	-29.99	kd	CGS001-699	BUB1	Bub family			
4969	-30.07	kd	CGS001-7465	WEE1	WEE family			
4970	-30.12	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
4971	-30.13	cp	BRD-K18895904	olanzapine	Dopamine receptor antagonist		DRD2, HTR2A, HTR2C, DRD1, DRD3, DRD4, HRH1, HTR1A, HTR1B, HTR1D, HTR1E, HTR6, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C8, DRD5, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH2, HRH4, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
4972	-30.13	kd	CGS001-51380	CSAD	-			
4973	-30.14	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
4974	-30.16	kd	CGS001-10477	UBE2E3	Ubiquitin-conjugating enzymes E2			
4975	-30.16	kd	CGS001-3339	HSPG2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4976	-30.19	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
4977	-30.19	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
4978	-30.2	kd	CGS001-2119	ETV5	ETS Transcription Factors			
4979	-30.24	kd	CGS001-4837	NNMT	-			
4980	-30.25	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
4981	-30.43	kd	CGS001-55958	KLHL9	BTB/POZ domain containing			
4982	-30.44	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
4983	-30.45	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
4984	-30.45	kd	CGS001-10626	TRIM16	Tripartite motif containing			
4985	-30.47	kd	CGS001-8639	AOC3	Oxidoreductases			
4986	-30.5	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
4987	-30.5	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
4988	-30.55	kd	CGS001-1312	COMT	Catecholamine turnover			
4989	-30.56	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
4990	-30.57	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4991	-30.57	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
4992	-30.58	kd	CGS001-79711	IPO4	Importins			
4993	-30.6	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
4994	-30.67	oe	ccsbBroad304_02500	RRAGA	-			
4995	-30.68	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
4996	-30.69	oe	ccsbBroad304_00174	BRAF	RAF family			
4997	-30.69	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
4998	-30.7	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
4999	-30.7	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
5000	-30.72	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
5001	-30.73	kd	CGS001-113451	ADC	-			
5002	-30.74	kd	CGS001-9443	MED7	-			
5003	-30.76	oe	ccsbBroad304_06665	OAT	-			
5004	-30.82	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
5005	-30.84	oe	ccsbBroad304_02674	STK38	NDR family			
5006	-30.84	oe	ccsbBroad304_07362	NMI	-			
5007	-30.84	kd	CGS001-24148	PRPF6	-			
5008	-30.89	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
5009	-30.9	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
5010	-30.91	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
5011	-30.97	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
5012	-31	kd	CGS001-5817	PVR	Immunoglobulin superfamily / C2-set domain containing			
5013	-31.02	kd	CGS001-4668	NAGA	-			
5014	-31.04	oe	ccsbBroad304_09358	MAPK1IP1L	-			
5015	-31.04	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
5016	-31.04	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
5017	-31.08	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
5018	-31.09	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
5019	-31.14	kd	CGS001-51734	SEPX1	-			
5020	-31.18	kd	CGS001-23549	DNPEP	Aminopeptidase I			
5021	-31.2	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
5022	-31.23	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
5023	-31.25	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
5024	-31.31	kd	CGS001-10670	RRAGA	-			
5025	-31.31	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
5026	-31.34	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
5027	-31.36	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
5028	-31.42	kd	CGS001-6469	SHH	-			
5029	-31.44	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
5030	-31.48	kd	CGS001-51727	CMPK1	-			
5031	-31.5	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
5032	-31.52	kd	CGS001-2159	F10	Chymotrypsin			
5033	-31.53	oe	ccsbBroad304_14047	TACC3	-			
5034	-31.53	oe	ccsbBroad304_04064	PRR15L	-			
5035	-31.53	kd	CGS001-2828	GPR4	GPCR / Class A : Orphans			
5036	-31.57	kd	CGS001-286530	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
5037	-31.67	kd	CGS001-6887	TAL2	Basic helix-loop-helix proteins			
5038	-31.7	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
5039	-31.71	kd	CGS001-2747	GLUD2	-			
5040	-31.73	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
5041	-31.73	kd	CGS001-7032	TFF2	-			
5042	-31.74	kd	CGS001-1677	DFFB	-			
5043	-31.77	oe	ccsbBroad304_02578	EBNA1BP2	-			
5044	-31.8	oe	ccsbBroad304_06449	ILF3	-			
5045	-31.8	kd	CGS001-478	ATP1A3	ATPases / P-type			
5046	-31.83	oe	ccsbBroad304_01147	PC	Carboxylases			
5047	-31.98	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
5048	-31.99	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
5049	-32	kd	CGS001-6715	SRD5A1	-			
5050	-32.08	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
5051	-32.08	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5052	-32.09	kd	CGS001-7251	TSG101	-			
5053	-32.1	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
5054	-32.1	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
5055	-32.12	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
5056	-32.13	kd	CGS001-336	APOA2	Apolipoproteins			
5057	-32.14	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
5058	-32.14	kd	CGS001-11319	ECD	-			
5059	-32.23	kd	CGS001-847	CAT	-			
5060	-32.26	kd	CGS001-4323	MMP14	Matrix metallopeptidase			
5061	-32.27	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
5062	-32.28	kd	CGS001-1727	CYB5R3	-			
5063	-32.29	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
5064	-32.29	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
5065	-32.31	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
5066	-32.32	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
5067	-32.32	kd	CGS001-2309	FOXO3	Forkhead boxes			
5068	-32.33	kd	CGS001-10553	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
5069	-32.34	cc		Potassium channel blocker	-			
5070	-32.35	oe	ccsbBroad304_02633	LSM6	-			
5071	-32.36	kd	CGS001-9815	GIT2	Ankyrin repeat domain containing			
5072	-32.37	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
5073	-32.39	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
5074	-32.41	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
5075	-32.5	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
5076	-32.51	kd	CGS001-1788	DNMT3A	Methyltransferases			
5077	-32.52	kd	CGS001-4758	NEU1	-			
5078	-32.53	oe	ccsbBroad304_02759	DICER1	-			
5079	-32.53	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5080	-32.57	kd	CGS001-826	CAPNS1	EF-hand domain containing			
5081	-32.58	kd	CGS001-6774	STAT3	SH2 domain containing			
5082	-32.59	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
5083	-32.6	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
5084	-32.61	kd	CGS001-7157	TP53	-			
5085	-32.61	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
5086	-32.65	kd	CGS001-29915	HCFC2	-			
5087	-32.66	kd	CGS001-2100	ESR2	Estrogen receptors			
5088	-32.7	kd	CGS001-5734	PTGER4	GPCR / Class A : Prostanoid receptors			
5089	-32.71	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
5090	-32.73	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
5091	-32.73	kd	CGS001-10606	PAICS	-			
5092	-32.75	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
5093	-32.79	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
5094	-32.8	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
5095	-32.91	oe	ccsbBroad304_02708	TRIM32	-			
5096	-32.92	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
5097	-32.96	kd	CGS001-1028	CDKN1C	-			
5098	-32.99	kd	CGS001-2645	GCK	Hexokinases			
5099	-33	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
5100	-33.01	kd	CGS001-256281	NUDT14	Nudix motif containing			
5101	-33.02	kd	CGS001-2810	SFN	-			
5102	-33.05	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
5103	-33.05	kd	CGS001-79722	ANKRD55	Ankyrin repeat domain containing			
5104	-33.07	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
5105	-33.11	kd	CGS001-7504	XK	Blood group antigens			
5106	-33.13	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
5107	-33.14	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
5108	-33.15	kd	CGS001-11019	LIAS	-			
5109	-33.17	kd	CGS001-2289	FKBP5	Tetratricopeptide (TTC) repeat domain containing			
5110	-33.18	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5111	-33.22	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5112	-33.26	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
5113	-33.27	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
5114	-33.28	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
5115	-33.28	kd	CGS001-55191	NADSYN1	-			
5116	-33.29	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
5117	-33.36	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
5118	-33.36	kd	CGS001-123803	NTAN1	-			
5119	-33.38	kd	CGS001-4763	NF1	-			
5120	-33.39	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
5121	-33.39	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
5122	-33.4	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5123	-33.45	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
5124	-33.46	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5125	-33.47	cc		EGFR inhibitor	-			
5126	-33.52	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
5127	-33.53	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
5128	-33.54	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
5129	-33.56	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
5130	-33.56	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
5131	-33.6	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
5132	-33.7	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
5133	-33.71	kd	CGS001-3659	IRF1	-			
5134	-33.75	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
5135	-33.76	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
5136	-33.78	kd	CGS001-271	AMPD2	-			
5137	-33.84	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
5138	-33.87	cp	BRD-A24191444	ifenprodil	Adrenergic receptor antagonist		GRIN1, GRIN2B	Adrenergic receptor antagonist, Glutamate receptor antagonist
5139	-33.88	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
5140	-33.89	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
5141	-33.89	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
5142	-33.91	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
5143	-33.93	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
5144	-33.95	kd	CGS001-5306	PITPNA	-			
5145	-33.96	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
5146	-33.97	cp	BRD-K97752965	nicorandil	Nitric oxide donor		ABCC9, KCNJ11, KCNJ8	Nitric oxide donor, Potassium channel activator
5147	-33.99	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
5148	-34.01	kd	CGS001-5810	RAD1	-			
5149	-34.02	oe	ccsbBroad304_00956	LYZ	-			
5150	-34.09	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
5151	-34.15	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
5152	-34.16	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
5153	-34.16	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
5154	-34.17	kd	CGS001-5446	PON3	Paraoxonases			
5155	-34.17	kd	CGS001-4704	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5156	-34.22	kd	CGS001-1604	CD55	CD molecules			
5157	-34.25	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
5158	-34.25	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
5159	-34.26	kd	CGS001-83729	INHBE	-			
5160	-34.27	kd	CGS001-6271	S100A1	EF-hand domain containing			
5161	-34.35	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
5162	-34.35	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
5163	-34.36	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
5164	-34.41	cp	BRD-K21806131	tegaserod	Serotonin receptor partial agonist		HTR4, HTR2B, HTR2A, HTR2C	Serotonin receptor partial agonist
5165	-34.45	kd	CGS001-55033	FKBP14	EF-hand domain containing			
5166	-34.51	kd	CGS001-7484	WNT9B	Wingless-type MMTV integration sites			
5167	-34.52	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
5168	-34.54	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
5169	-34.58	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
5170	-34.63	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
5171	-34.64	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
5172	-34.65	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
5173	-34.65	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
5174	-34.66	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
5175	-34.66	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
5176	-34.66	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5177	-34.67	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
5178	-34.68	cc		S100 calcium binding proteins LOF	-			
5179	-34.71	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
5180	-34.74	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
5181	-34.74	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
5182	-34.78	oe	ccsbBroad304_08365	CYCS	-			
5183	-34.79	kd	CGS001-9697	TRAM2	-			
5184	-34.8	kd	CGS001-6813	STXBP2	-			
5185	-34.8	kd	CGS001-2629	GBA	-			
5186	-34.82	kd	CGS001-7693	ZNF134	Zinc fingers, C2H2-type			
5187	-34.83	kd	CGS001-4708	NDUFB2	Mitochondrial respiratory chain complex / Complex I			
5188	-34.86	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
5189	-34.99	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
5190	-35	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
5191	-35.04	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
5192	-35.05	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
5193	-35.09	oe	ccsbBroad304_07843	FCHO1	-			
5194	-35.09	kd	CGS001-3109	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
5195	-35.11	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
5196	-35.11	kd	CGS001-7541	ZFP161	-			
5197	-35.14	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
5198	-35.14	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
5199	-35.17	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
5200	-35.18	kd	CGS001-117581	TWIST2	Basic helix-loop-helix proteins			
5201	-35.2	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
5202	-35.24	oe	ccsbBroad304_01165	PDK1	-			
5203	-35.24	kd	CGS001-54490	UGT2B28	UDP glucuronosyltransferases			
5204	-35.3	kd	CGS001-5689	PSMB1	Proteasome subunits			
5205	-35.4	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5206	-35.45	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
5207	-35.47	kd	CGS001-50814	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5208	-35.48	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
5209	-35.5	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
5210	-35.53	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
5211	-35.54	kd	CGS001-2760	GM2A	-			
5212	-35.55	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
5213	-35.55	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
5214	-35.57	oe	ccsbBroad304_01577	SOD1	-			
5215	-35.57	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
5216	-35.57	kd	CGS001-3170	FOXA2	Forkhead boxes			
5217	-35.58	oe	ccsbBroad304_00469	DUT	-			
5218	-35.59	kd	CGS001-3690	ITGB3	Integrins			
5219	-35.62	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
5220	-35.62	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
5221	-35.65	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
5222	-35.67	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
5223	-35.7	kd	CGS001-5933	RBL1	-			
5224	-35.71	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
5225	-35.72	kd	CGS001-27113	BBC3	-			
5226	-35.76	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
5227	-35.78	kd	CGS001-4255	MGMT	-			
5228	-35.79	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
5229	-35.79	kd	CGS001-10048	RANBP9	-			
5230	-35.81	cp	BRD-K81855038	roxatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
5231	-35.83	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
5232	-35.83	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
5233	-35.86	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
5234	-35.86	kd	CGS001-3265	HRAS	RAS subfamily			
5235	-35.87	oe	ccsbBroad304_03177	FIS1	-			
5236	-35.91	cc		Sodium channel blocker	-			
5237	-35.91	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5238	-35.93	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
5239	-35.94	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
5240	-35.97	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5241	-35.98	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
5242	-35.99	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
5243	-35.99	kd	CGS001-162699	TCEB3C	-			
5244	-36.02	kd	CGS001-1859	DYRK1A	Dyrk1 subfamily			
5245	-36.03	oe	ccsbBroad304_00991	MDH1	-			
5246	-36.05	kd	CGS001-3034	HAL	-			
5247	-36.07	kd	CGS001-5300	PIN1	-			
5248	-36.12	kd	CGS001-55746	NUP133	-			
5249	-36.17	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
5250	-36.17	kd	CGS001-8226	HDHD1	-			
5251	-36.18	kd	CGS001-9690	UBE3C	-			
5252	-36.2	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
5253	-36.2	kd	CGS001-9459	ARHGEF6	Rho guanine nucleotide exchange factors			
5254	-36.23	oe	ccsbBroad304_09035	COASY	-			
5255	-36.25	oe	ccsbBroad304_06783	LGMN	Legumain			
5256	-36.25	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
5257	-36.28	cp	BRD-K41051431	mecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5258	-36.3	kd	CGS001-7771	ZFP112	-			
5259	-36.36	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
5260	-36.4	oe	ccsbBroad304_00146	BAD	-			
5261	-36.4	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
5262	-36.41	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
5263	-36.48	kd	CGS001-527	ATP6V0C	ATPases / V-type			
5264	-36.49	cc		PKA inhibitor	-			
5265	-36.52	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
5266	-36.56	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
5267	-36.58	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
5268	-36.59	kd	CGS001-51176	LEF1	-			
5269	-36.61	kd	CGS001-10538	BATF	basic leucine zipper proteins			
5270	-36.66	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
5271	-36.67	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
5272	-36.69	kd	CGS001-1955	MEGF9	-			
5273	-36.7	oe	ccsbBroad304_02569	BTG3	-			
5274	-36.72	kd	CGS001-148103	ZNF599	Zinc fingers, C2H2-type			
5275	-36.73	oe	ccsbBroad304_02143	CNOT8	-			
5276	-36.74	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
5277	-36.75	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5278	-36.77	kd	CGS001-7029	TFDP2	-			
5279	-36.81	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
5280	-36.82	oe	ccsbBroad304_00961	SMAD2	SMADs			
5281	-36.82	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
5282	-36.83	oe	ccsbBroad304_07724	KDELR2	-			
5283	-36.84	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
5284	-36.87	kd	CGS001-55214	LEPREL1	-			
5285	-36.87	oe	ccsbBroad304_02506	EBP	-			
5286	-36.9	kd	CGS001-10135	NAMPT	-			
5287	-36.91	cc		SRC inhibitor	-			
5288	-36.91	oe	ccsbBroad304_02890	SYF2	-			
5289	-36.92	kd	CGS001-55193	PBRM1	Non-enzymatic BRD containing proteins			
5290	-36.94	oe	ccsbBroad304_08511	RFK	-			
5291	-36.97	kd	CGS001-91433	RCCD1	-			
5292	-37.03	kd	CGS001-284	ANGPT1	Fibrinogen C domain containing			
5293	-37.06	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
5294	-37.09	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
5295	-37.1	kd	CGS001-170591	S100Z	EF-hand domain containing			
5296	-37.14	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
5297	-37.16	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
5298	-37.17	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
5299	-37.22	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
5300	-37.23	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
5301	-37.23	kd	CGS001-11113	CIT	Other DMPK family kinases			
5302	-37.24	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
5303	-37.29	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
5304	-37.31	cp	BRD-A16444946	acarbose	Glucosidase inhibitor		GAA, MGAM, AMY2A, SI	Glucosidase inhibitor
5305	-37.39	kd	CGS001-55723	ASF1B	-			
5306	-37.4	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
5307	-37.41	oe	ccsbBroad304_02372	SPRY1	-			
5308	-37.46	kd	CGS001-54851	ANKRD49	Ankyrin repeat domain containing			
5309	-37.52	kd	CGS001-2010	EMD	-			
5310	-37.54	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
5311	-37.54	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
5312	-37.57	oe	ccsbBroad304_07557	NAMPT	-			
5313	-37.58	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5314	-37.58	kd	CGS001-57761	TRIB3	Trbl family			
5315	-37.62	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
5316	-37.63	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
5317	-37.64	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
5318	-37.64	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
5319	-37.67	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
5320	-37.73	kd	CGS001-6908	TBP	General transcription factors			
5321	-37.74	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
5322	-37.84	kd	CGS001-2568	GABRP	GABA receptors			
5323	-37.84	kd	CGS001-1112	FOXN3	Forkhead boxes			
5324	-37.85	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
5325	-37.86	kd	CGS001-11188	NISCH	-			
5326	-37.88	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5327	-37.9	kd	CGS001-11007	CCDC85B	-			
5328	-37.97	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
5329	-37.97	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
5330	-37.98	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
5331	-37.98	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
5332	-38.05	oe	ccsbBroad304_00841	IKBKB	IKK family			
5333	-38.07	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
5334	-38.09	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
5335	-38.09	kd	CGS001-2237	FEN1	-			
5336	-38.11	kd	CGS001-5294	PIK3CG	Phosphatidylinositol kinases			
5337	-38.14	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
5338	-38.14	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
5339	-38.14	kd	CGS001-5025	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
5340	-38.15	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
5341	-38.16	oe	ccsbBroad304_00116	ASS1	-			
5342	-38.16	kd	CGS001-8408	ULK1	Unc-51-like kinase (ULK) family			
5343	-38.19	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
5344	-38.2	kd	CGS001-10250	SRRM1	-			
5345	-38.22	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
5346	-38.23	oe	ccsbBroad304_02205	WTAP	-			
5347	-38.25	oe	ccsbBroad304_00645	GCLM	-			
5348	-38.25	kd	CGS001-563	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
5349	-38.26	cp	BRD-K51485625	ritonavir	HIV protease inhibitor		CYP3A4, CYP1A2, CYP2B6, CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
5350	-38.27	kd	CGS001-375449	MAST4	MAST family			
5351	-38.27	kd	CGS001-8872	CDC123	-			
5352	-38.27	kd	CGS001-29105	C16ORF80	-			
5353	-38.3	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
5354	-38.35	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5355	-38.36	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
5356	-38.38	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
5357	-38.39	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
5358	-38.41	kd	CGS001-5928	RBBP4	WD repeat domain containing			
5359	-38.44	kd	CGS001-10298	PAK4	PAKB subfamily			
5360	-38.45	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
5361	-38.46	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
5362	-38.48	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
5363	-38.49	kd	CGS001-218	ALDH3A1	Aldehyde dehydrogenases			
5364	-38.52	kd	CGS001-9218	VAPA	-			
5365	-38.54	oe	ccsbBroad304_00250	CD19	CD molecules			
5366	-38.56	kd	CGS001-6810	STX4	-			
5367	-38.58	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
5368	-38.63	kd	CGS001-87	ACTN1	EF-hand domain containing			
5369	-38.66	kd	CGS001-8548	BLZF1	-			
5370	-38.67	kd	CGS001-11336	EXOC3	-			
5371	-38.7	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
5372	-38.71	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
5373	-38.76	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
5374	-38.77	kd	CGS001-4835	NQO2	-			
5375	-38.78	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
5376	-38.81	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
5377	-38.81	kd	CGS001-2147	F2	Endogenous ligands			
5378	-38.83	kd	CGS001-84971	ATG4D	-			
5379	-38.92	kd	CGS001-84547	PGBD1	-			
5380	-38.99	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
5381	-38.99	kd	CGS001-7572	ZNF24	Zinc fingers, C2H2-type			
5382	-39.01	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
5383	-39.01	kd	CGS001-63874	ABHD4	Abhydrolase domain containing			
5384	-39.02	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
5385	-39.04	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
5386	-39.07	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
5387	-39.07	kd	CGS001-23077	MYCBP2	-			
5388	-39.08	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
5389	-39.09	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
5390	-39.12	oe	ccsbBroad304_09881	RFX6	-			
5391	-39.12	kd	CGS001-10174	SORBS3	-			
5392	-39.14	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
5393	-39.16	kd	CGS001-23057	NMNAT2	-			
5394	-39.18	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
5395	-39.19	oe	ccsbBroad304_06226	FTL	-			
5396	-39.22	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
5397	-39.33	kd	CGS001-7057	THBS1	-			
5398	-39.35	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
5399	-39.36	kd	CGS001-6502	SKP2	F-boxes / Leucine-rich repeats			
5400	-39.38	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
5401	-39.39	kd	CGS001-54555	DDX49	DEAD-boxes			
5402	-39.41	kd	CGS001-84288	EFCAB2	EF-hand domain containing			
5403	-39.45	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
5404	-39.47	kd	CGS001-3481	IGF2	-			
5405	-39.49	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5406	-39.51	kd	CGS001-27125	AFF4	-			
5407	-39.52	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
5408	-39.53	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
5409	-39.54	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
5410	-39.56	kd	CGS001-253430	IPMK	-			
5411	-39.59	kd	CGS001-152	ADRA2C	GPCR / Class A : Adrenoceptors : alpha			
5412	-39.61	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
5413	-39.61	kd	CGS001-8945	BTRC	F-boxes / WD-40 domains			
5414	-39.63	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
5415	-39.64	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
5416	-39.65	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
5417	-39.72	cc		Akt Signaling GOF	-			
5418	-39.72	oe	ccsbBroad304_03652	EXOC2	-			
5419	-39.73	oe	ccsbBroad304_01234	POLB	DNA polymerases			
5420	-39.73	kd	CGS001-23463	ICMT	-			
5421	-39.74	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
5422	-39.76	oe	ccsbBroad304_07920	NUP62	-			
5423	-39.81	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5424	-39.82	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
5425	-39.85	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
5426	-39.85	kd	CGS001-51070	NOSIP	-			
5427	-39.91	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
5428	-39.92	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
5429	-39.92	cp	BRD-K17705806	JTC-801	Opioid receptor antagonist		OPRL1	Opioid receptor antagonist
5430	-39.92	kd	CGS001-1120	CHKB	-			
5431	-39.94	kd	CGS001-210	ALAD	-			
5432	-39.99	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
5433	-40.07	kd	CGS001-9213	XPR1	-			
5434	-40.08	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
5435	-40.11	kd	CGS001-5170	PDPK1	PDK1 family			
5436	-40.18	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
5437	-40.21	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
5438	-40.26	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
5439	-40.41	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
5440	-40.44	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
5441	-40.45	oe	ccsbBroad304_10846	GGT1	CD molecules			
5442	-40.51	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
5443	-40.53	kd	CGS001-7357	UGCG	Glycosyltransferase family 2 domain containing			
5444	-40.54	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
5445	-40.58	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
5446	-40.58	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5447	-40.64	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
5448	-40.64	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
5449	-40.66	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
5450	-40.78	kd	CGS001-6198	RPS6KB1	p70 subfamily			
5451	-40.84	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
5452	-40.84	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5453	-40.92	kd	CGS001-10131	TRAP1	Heat shock proteins / HSPC			
5454	-40.94	oe	ccsbBroad304_00564	FGR	Src family			
5455	-40.94	kd	CGS001-708	C1QBP	-			
5456	-40.96	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
5457	-41.01	oe	ccsbBroad304_01962	STK16	NAK family			
5458	-41.05	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
5459	-41.05	kd	CGS001-4193	MDM2	-			
5460	-41.09	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
5461	-41.1	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
5462	-41.12	oe	ccsbBroad304_07704	SUB1	-			
5463	-41.12	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
5464	-41.13	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
5465	-41.15	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
5466	-41.18	kd	CGS001-55631	LRRC40	-			
5467	-41.19	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
5468	-41.2	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
5469	-41.21	oe	ccsbBroad304_04626	EGLN3	-			
5470	-41.21	kd	CGS001-26959	HBP1	-			
5471	-41.22	kd	CGS001-6223	RPS19	S ribosomal proteins			
5472	-41.24	kd	CGS001-55256	ADI1	-			
5473	-41.28	kd	CGS001-57616	TSHZ3	Teashirt zinc fingers			
5474	-41.29	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
5475	-41.38	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
5476	-41.4	oe	ccsbBroad304_00115	ASPH	-			
5477	-41.41	cc		V type ATPases LOF	-			
5478	-41.42	cc		Nucleoporin LOF	-			
5479	-41.42	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
5480	-41.44	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
5481	-41.48	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
5482	-41.49	kd	CGS001-79618	HMBOX1	Homeoboxes / HNF class			
5483	-41.5	oe	ccsbBroad304_13998	PDXK	-			
5484	-41.5	kd	CGS001-641	BLM	-			
5485	-41.54	cp	BRD-K92870997	pterostilbene	Cyclooxygenase inhibitor		FAAH, PPARA, PTGS1, PTGS2	Cyclooxygenase inhibitor, PPAR receptor agonist
5486	-41.54	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
5487	-41.55	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
5488	-41.56	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
5489	-41.56	kd	CGS001-3579	CXCR2	Chemokine receptors			
5490	-41.58	oe	ccsbBroad304_05152	SSBP4	-			
5491	-41.59	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
5492	-41.62	oe	ccsbBroad304_02361	MFSD10	-			
5493	-41.66	kd	CGS001-5906	RAP1A	-			
5494	-41.69	kd	CGS001-1062	CENPE	Kinesins			
5495	-41.7	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
5496	-41.72	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
5497	-41.74	kd	CGS001-3017	HIST1H2BD	Histones / Replication-dependent			
5498	-41.78	kd	CGS001-3799	KIF5B	Kinesins			
5499	-41.79	cp	BRD-A75935363	atracurium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
5500	-41.83	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
5501	-41.87	kd	CGS001-6772	STAT1	SH2 domain containing			
5502	-41.92	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
5503	-41.95	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
5504	-41.96	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
5505	-41.98	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
5506	-42.01	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
5507	-42.06	kd	CGS001-51181	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5508	-42.09	kd	CGS001-7016	TESK1	TESK subfamily			
5509	-42.21	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
5510	-42.25	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
5511	-42.27	kd	CGS001-6446	SGK1	SGK family			
5512	-42.28	oe	ccsbBroad304_02239	RASSF2	-			
5513	-42.28	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
5514	-42.3	oe	ccsbBroad304_06349	HAGH	-			
5515	-42.31	kd	CGS001-211	ALAS1	-			
5516	-42.36	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
5517	-42.38	oe	ccsbBroad304_10240	CROT	-			
5518	-42.43	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
5519	-42.47	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
5520	-42.47	kd	CGS001-1892	ECHS1	-			
5521	-42.5	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
5522	-42.55	kd	CGS001-57819	LSM2	-			
5523	-42.61	kd	CGS001-122809	SOCS4	SH2 domain containing			
5524	-42.66	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
5525	-42.7	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
5526	-42.71	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
5527	-42.78	kd	CGS001-7466	WFS1	-			
5528	-42.8	oe	ccsbBroad304_07097	TRAF1	-			
5529	-42.81	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
5530	-42.81	kd	CGS001-9887	SMG7	-			
5531	-42.85	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
5532	-42.89	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
5533	-42.89	kd	CGS001-9360	PPIG	-			
5534	-42.89	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
5535	-42.93	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
5536	-42.94	oe	ccsbBroad304_03853	LSM2	-			
5537	-42.94	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
5538	-42.94	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
5539	-42.98	oe	ccsbBroad304_04471	C5ORF62	-			
5540	-42.98	kd	CGS001-55632	G2E3	Zinc fingers, PHD-type			
5541	-43	kd	CGS001-79712	GTDC1	Glycosyltransferase group 1 domain containing			
5542	-43.08	kd	CGS001-51495	PTPLAD1	-			
5543	-43.09	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
5544	-43.11	oe	ccsbBroad304_03554	NAT10	-			
5545	-43.12	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
5546	-43.13	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
5547	-43.15	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
5548	-43.17	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
5549	-43.19	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
5550	-43.25	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
5551	-43.25	kd	CGS001-54901	CDKAL1	-			
5552	-43.3	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
5553	-43.33	kd	CGS001-892	CCNC	-			
5554	-43.36	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
5555	-43.37	kd	CGS001-2212	FCGR2A	CD molecules			
5556	-43.43	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
5557	-43.44	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5558	-43.5	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
5559	-43.58	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
5560	-43.66	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
5561	-43.68	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5562	-43.68	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
5563	-43.68	kd	CGS001-3957	LGALS2	Lectins, galactoside-binding			
5564	-43.7	kd	CGS001-638	BIK	-			
5565	-43.71	kd	CGS001-56675	NRIP3	-			
5566	-43.72	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
5567	-43.72	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
5568	-43.77	kd	CGS001-7846	TUBA1A	Tubulins			
5569	-43.78	kd	CGS001-55379	LRRC59	-			
5570	-43.8	oe	ccsbBroad304_01701	TPI1	-			
5571	-43.81	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
5572	-43.82	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
5573	-43.82	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5574	-43.83	kd	CGS001-10128	LRPPRC	-			
5575	-43.84	kd	CGS001-64077	LHPP	-			
5576	-43.86	cp	BRD-K84955386	hyperoside	Glucosidase inhibitor		ACE, AKR1B1, GAA	Glucosidase inhibitor
5577	-43.95	oe	ccsbBroad304_03040	NKIRAS2	-			
5578	-43.95	kd	CGS001-9761	MLEC	-			
5579	-43.98	kd	CGS001-8543	LMO4	-			
5580	-44	oe	ccsbBroad304_02018	SUCLA2	-			
5581	-44.03	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
5582	-44.03	kd	CGS001-5451	POU2F1	Homeoboxes / POU class			
5583	-44.05	oe	ccsbBroad304_06837	RAF1	RAF family			
5584	-44.11	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
5585	-44.14	oe	ccsbBroad304_05749	A2M	-			
5586	-44.17	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
5587	-44.19	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
5588	-44.19	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5589	-44.23	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
5590	-44.25	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
5591	-44.26	kd	CGS001-2778	GNAS	-			
5592	-44.27	kd	CGS001-467	ATF3	basic leucine zipper proteins			
5593	-44.28	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
5594	-44.33	kd	CGS001-8985	PLOD3	-			
5595	-44.41	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
5596	-44.41	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5597	-44.45	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
5598	-44.51	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
5599	-44.61	kd	CGS001-5371	PML	RING-type (C3HC4) zinc fingers			
5600	-44.63	kd	CGS001-118442	GPR62	GPCR / Class A : Orphans			
5601	-44.64	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
5602	-44.66	kd	CGS001-6822	SULT2A1	Sulfotransferases, cytosolic			
5603	-44.67	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5604	-44.68	oe	ccsbBroad304_06993	SRD5A1	-			
5605	-44.69	kd	CGS001-9988	DMTF1	-			
5606	-44.71	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
5607	-44.72	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
5608	-44.8	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
5609	-44.81	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
5610	-44.83	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
5611	-44.83	kd	CGS001-4638	MYLK	Myosin Light Chain Kinase (MLCK) family			
5612	-44.85	oe	ccsbBroad304_01372	RALB	-			
5613	-44.86	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5614	-44.87	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
5615	-44.9	kd	CGS001-4724	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
5616	-44.91	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
5617	-44.93	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
5618	-44.97	cp	BRD-K25310650	ormetoprim	Bacterial antifolate			Bacterial antifolate
5619	-45.01	kd	CGS001-11004	KIF2C	Kinesins			
5620	-45.05	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
5621	-45.06	oe	ccsbBroad304_02990	LYPD3	-			
5622	-45.13	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
5623	-45.14	kd	CGS001-1509	CTSD	Cathepsins			
5624	-45.16	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
5625	-45.17	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
5626	-45.22	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
5627	-45.32	kd	CGS001-4092	SMAD7	SMADs			
5628	-45.37	oe	ccsbBroad304_02702	MSRB2	-			
5629	-45.55	cc		Bacterial cell wall synthesis inhibitor	-			
5630	-45.55	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
5631	-45.56	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
5632	-45.56	oe	ccsbBroad304_00077	APEX1	-			
5633	-45.58	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
5634	-45.61	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
5635	-45.67	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
5636	-45.68	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5637	-45.74	kd	CGS001-5167	ENPP1	-			
5638	-45.76	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
5639	-45.79	kd	CGS001-27297	CRCP	-			
5640	-45.94	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
5641	-46	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
5642	-46.1	kd	CGS001-9231	DLG5	-			
5643	-46.12	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
5644	-46.16	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
5645	-46.2	kd	CGS001-1029	CDKN2A	-			
5646	-46.22	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
5647	-46.36	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
5648	-46.37	kd	CGS001-29883	CNOT7	-			
5649	-46.46	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
5650	-46.47	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
5651	-46.48	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
5652	-46.52	cc		Cannabinoid receptor agonist	-			
5653	-46.52	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
5654	-46.63	oe	ccsbBroad304_08023	EIF2C1	-			
5655	-46.63	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
5656	-46.64	kd	CGS001-262	AMD1	Decarboxylases			
5657	-46.68	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
5658	-46.71	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
5659	-46.72	kd	CGS001-23012	STK38L	NDR family			
5660	-46.73	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
5661	-46.74	kd	CGS001-9891	NUAK1	NuaK subfamily			
5662	-46.76	oe	ccsbBroad304_08825	LHPP	-			
5663	-46.79	kd	CGS001-23365	ARHGEF12	Rho guanine nucleotide exchange factors			
5664	-46.8	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
5665	-46.81	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
5666	-46.83	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
5667	-46.86	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
5668	-46.87	kd	CGS001-51720	UIMC1	-			
5669	-46.88	kd	CGS001-2773	GNAI3	-			
5670	-46.89	kd	CGS001-4143	MAT1A	-			
5671	-46.96	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
5672	-46.99	kd	CGS001-3569	IL6	Interferons			
5673	-47.01	kd	CGS001-837	CASP4	Caspases			
5674	-47.01	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
5675	-47.05	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
5676	-47.09	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
5677	-47.11	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
5678	-47.11	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
5679	-47.13	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
5680	-47.14	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
5681	-47.2	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
5682	-47.2	kd	CGS001-9258	MFHAS1	-			
5683	-47.24	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
5684	-47.26	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
5685	-47.28	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
5686	-47.3	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
5687	-47.31	kd	CGS001-9738	CCP110	-			
5688	-47.38	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
5689	-47.41	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
5690	-47.45	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
5691	-47.49	oe	ccsbBroad304_09821	TMEM154	-			
5692	-47.6	kd	CGS001-230	ALDOC	-			
5693	-47.65	kd	CGS001-9791	PTDSS1	-			
5694	-47.7	oe	ccsbBroad304_01748	UFD1L	-			
5695	-47.71	kd	CGS001-509	ATP5C1	ATPases / F-type			
5696	-47.77	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
5697	-47.81	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
5698	-47.82	kd	CGS001-5979	RET	Type XIV RTKs: RET			
5699	-47.84	cp	BRD-K81169441	cerivastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A5	HMGCR inhibitor
5700	-47.87	kd	CGS001-10914	PAPOLA	-			
5701	-47.9	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
5702	-47.92	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
5703	-47.93	kd	CGS001-645	BLVRB	Short chain dehydrogenase/reductase superfamily / Atypical members			
5704	-47.95	cc		FLT3 inhibitor	-			
5705	-47.96	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
5706	-47.96	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
5707	-47.97	kd	CGS001-9	NAT1	-			
5708	-47.97	kd	CGS001-135	ADORA2A	GPCR / Class A : Adenosine receptors			
5709	-47.98	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
5710	-48	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
5711	-48.02	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
5712	-48.02	oe	ccsbBroad304_08167	DNTTIP2	-			
5713	-48.02	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
5714	-48.08	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
5715	-48.13	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
5716	-48.23	kd	CGS001-3269	HRH1	Histamine receptors			
5717	-48.28	kd	CGS001-51002	TPRKB	-			
5718	-48.33	cc		Sirtuins GOF	-			
5719	-48.34	kd	CGS001-79073	TMEM109	-			
5720	-48.35	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
5721	-48.39	kd	CGS001-3880	KRT19	Intermediate filaments type I, keratins (acidic)			
5722	-48.42	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
5723	-48.44	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
5724	-48.47	oe	ccsbBroad304_03173	TMED7	-			
5725	-48.47	oe	ccsbBroad304_10212	GRHL3	-			
5726	-48.49	oe	ccsbBroad304_00471	E2F6	-			
5727	-48.49	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
5728	-48.54	kd	CGS001-5910	RAP1GDS1	Armadillo repeat containing			
5729	-48.57	oe	ccsbBroad304_00006	ACADM	-			
5730	-48.57	kd	CGS001-81550	TDRD3	Tudor domain containing			
5731	-48.58	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
5732	-48.59	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
5733	-48.59	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
5734	-48.61	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
5735	-48.64	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
5736	-48.66	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
5737	-48.68	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
5738	-48.71	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
5739	-48.73	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
5740	-48.8	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
5741	-48.84	oe	ccsbBroad304_00491	EIF4EBP2	-			
5742	-48.93	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
5743	-49	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
5744	-49.01	kd	CGS001-581	BAX	-			
5745	-49.07	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
5746	-49.12	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
5747	-49.14	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
5748	-49.15	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
5749	-49.18	kd	CGS001-10657	KHDRBS1	-			
5750	-49.19	kd	CGS001-8655	DYNLL1	Cytoplasmic dyneins			
5751	-49.21	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
5752	-49.23	cp	BRD-A88254928	salbutamol	Adrenergic receptor agonist		ADRB2, ADRB1	Adrenergic receptor agonist
5753	-49.24	kd	CGS001-384	ARG2	Arginase			
5754	-49.24	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
5755	-49.32	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
5756	-49.34	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
5757	-49.34	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
5758	-49.4	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
5759	-49.41	oe	ccsbBroad304_03266	ERGIC2	-			
5760	-49.44	kd	CGS001-50	ACO2	-			
5761	-49.52	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
5762	-49.53	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
5763	-49.56	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
5764	-49.56	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
5765	-49.71	oe	ccsbBroad304_08217	SCCPDH	-			
5766	-49.71	oe	ccsbBroad304_02788	PRAME	-			
5767	-49.71	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5768	-49.81	oe	ccsbBroad304_03874	UBL5	-			
5769	-49.81	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
5770	-49.82	oe	ccsbBroad304_01038	MSRA	-			
5771	-49.88	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
5772	-49.9	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
5773	-49.9	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
5774	-49.9	kd	CGS001-4711	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
5775	-49.92	oe	ccsbBroad304_02864	PRDX5	-			
5776	-49.96	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
5777	-50.03	oe	ccsbBroad304_01664	TGFA	-			
5778	-50.03	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
5779	-50.08	oe	ccsbBroad304_00993	MDM4	-			
5780	-50.08	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
5781	-50.08	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
5782	-50.09	oe	ccsbBroad304_01373	RAN	-			
5783	-50.09	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
5784	-50.11	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
5785	-50.14	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
5786	-50.19	kd	CGS001-3428	IFI16	-			
5787	-50.2	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
5788	-50.22	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
5789	-50.23	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
5790	-50.23	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
5791	-50.24	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
5792	-50.27	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
5793	-50.32	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
5794	-50.36	kd	CGS001-1345	COX6C	Mitochondrial respiratory chain complex			
5795	-50.44	kd	CGS001-991	CDC20	WD repeat domain containing			
5796	-50.46	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
5797	-50.46	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
5798	-50.46	kd	CGS001-1738	DLD	-			
5799	-50.47	kd	CGS001-4795	NFKBIL1	-			
5800	-50.48	kd	CGS001-6493	SIM2	Basic helix-loop-helix proteins			
5801	-50.48	kd	CGS001-83999	KREMEN1	-			
5802	-50.52	kd	CGS001-4790	NFKB1	NFkappaB transcription factor family			
5803	-50.55	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
5804	-50.6	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
5805	-50.65	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
5806	-50.66	kd	CGS001-4048	LTA4H	Hydrolases			
5807	-50.72	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
5808	-50.75	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
5809	-50.79	kd	CGS001-3590	IL11RA	IL-6 receptor family			
5810	-50.82	oe	ccsbBroad304_03479	YTHDF1	-			
5811	-50.91	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
5812	-50.95	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
5813	-50.96	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
5814	-50.96	kd	CGS001-6670	SP3	Specificity protein transcription factors			
5815	-50.97	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
5816	-50.97	kd	CGS001-771	CA12	Carbonic anhydrases			
5817	-51.04	oe	ccsbBroad304_06642	NIT1	-			
5818	-51.05	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
5819	-51.05	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
5820	-51.05	kd	CGS001-4234	METTL1	-			
5821	-51.12	oe	ccsbBroad304_07923	LSM5	-			
5822	-51.12	oe	ccsbBroad304_00155	CCND1	-			
5823	-51.13	kd	CGS001-200879	LIPH	-			
5824	-51.19	oe	ccsbBroad304_00001	NAT1	-			
5825	-51.29	oe	ccsbBroad304_05947	CCNC	-			
5826	-51.29	kd	CGS001-25898	RCHY1	RING-type (C3HC4) zinc fingers			
5827	-51.32	kd	CGS001-5036	PA2G4	-			
5828	-51.45	kd	CGS001-5106	PCK2	-			
5829	-51.5	oe	ccsbBroad304_13598	NRBP2	NRBP family			
5830	-51.5	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
5831	-51.55	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
5832	-51.58	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
5833	-51.63	oe	ccsbBroad304_07875	SPECC1L	-			
5834	-51.69	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
5835	-51.69	kd	CGS001-2936	GSR	Oxidoreductases			
5836	-51.71	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
5837	-51.75	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
5838	-51.78	kd	CGS001-55876	GSDMB	-			
5839	-51.81	oe	ccsbBroad304_06695	PCK2	-			
5840	-51.81	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
5841	-51.86	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
5842	-51.88	cp	BRD-A02189320	met-leu-phe	-666			-666
5843	-51.9	oe	ccsbBroad304_04786	CANT1	-			
5844	-51.9	kd	CGS001-3776	KCNK2	Two-P potassium channels			
5845	-51.92	kd	CGS001-6443	SGCB	-			
5846	-51.93	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
5847	-51.93	kd	CGS001-53347	UBASH3A	-			
5848	-51.99	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
5849	-52	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
5850	-52.07	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5851	-52.13	kd	CGS001-3692	EIF6	-			
5852	-52.14	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
5853	-52.17	oe	ccsbBroad304_03570	QRSL1	-			
5854	-52.19	kd	CGS001-54811	ZNF562	Zinc fingers, C2H2-type			
5855	-52.23	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
5856	-52.25	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5857	-52.28	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
5858	-52.28	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
5859	-52.3	kd	CGS001-1903	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
5860	-52.32	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
5861	-52.36	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
5862	-52.46	kd	CGS001-382	ARF6	ADP-ribosylation factors			
5863	-52.47	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5864	-52.53	oe	ccsbBroad304_00819	IDH3B	-			
5865	-52.55	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
5866	-52.57	kd	CGS001-10898	CPSF4	-			
5867	-52.59	kd	CGS001-47	ACLY	-			
5868	-52.61	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
5869	-52.65	oe	ccsbBroad304_01101	NME1	-			
5870	-52.65	kd	CGS001-122402	TDRD9	Tudor domain containing			
5871	-52.85	oe	ccsbBroad304_05758	ACADSB	-			
5872	-52.86	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
5873	-52.94	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
5874	-52.94	kd	CGS001-10906	TRAFD1	-			
5875	-53	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
5876	-53	kd	CGS001-6285	S100B	EF-hand domain containing			
5877	-53.01	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
5878	-53.15	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
5879	-53.19	oe	ccsbBroad304_01841	BAG6	-			
5880	-53.26	kd	CGS001-23335	WDR7	WD repeat domain containing			
5881	-53.28	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
5882	-53.35	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
5883	-53.35	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
5884	-53.36	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
5885	-53.55	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5886	-53.59	cc		JAK inhibitor	-			
5887	-53.62	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
5888	-53.65	oe	ccsbBroad304_02057	P4HA2	-			
5889	-53.65	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
5890	-53.65	kd	CGS001-54106	TLR9	Toll-like receptor family			
5891	-53.73	kd	CGS001-6621	SNAPC4	-			
5892	-53.74	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
5893	-53.81	kd	CGS001-51203	NUSAP1	-			
5894	-53.82	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
5895	-53.83	cp	BRD-K30563334	rifabutin	Protein synthesis inhibitor		CYP3A4, HSP90AA1, HSP90B1	Protein synthesis inhibitor
5896	-53.87	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
5897	-53.89	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
5898	-53.9	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
5899	-53.92	kd	CGS001-4929	NR4A2	Nerve growth factor IB-like receptors			
5900	-53.93	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
5901	-53.94	oe	ccsbBroad304_00954	LYN	Src family			
5902	-54	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
5903	-54	kd	CGS001-10023	FRAT1	-			
5904	-54.05	kd	CGS001-440	ASNS	-			
5905	-54.07	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
5906	-54.08	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
5907	-54.08	kd	CGS001-10955	SERINC3	-			
5908	-54.16	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
5909	-54.16	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
5910	-54.18	oe	ccsbBroad304_01084	NEU1	-			
5911	-54.18	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
5912	-54.21	kd	CGS001-6196	RPS6KA2	RSK subfamily			
5913	-54.28	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
5914	-54.29	kd	CGS001-23196	FAM120A	-			
5915	-54.36	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
5916	-54.46	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
5917	-54.46	kd	CGS001-308	ANXA5	Annexins			
5918	-54.52	oe	ccsbBroad304_02425	CDIPT	-			
5919	-54.52	kd	CGS001-55937	APOM	Apolipoproteins			
5920	-54.53	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
5921	-54.54	cp	BRD-K01649396	indatraline	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine transporter inhibitor
5922	-54.54	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
5923	-54.61	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
5924	-54.64	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
5925	-54.65	oe	ccsbBroad304_02509	GMEB1	-			
5926	-54.69	oe	ccsbBroad304_01951	BLZF1	-			
5927	-54.7	kd	CGS001-5422	POLA1	DNA polymerases			
5928	-54.7	kd	CGS001-11325	DDX42	DEAD-boxes			
5929	-54.73	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
5930	-54.76	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
5931	-54.78	kd	CGS001-31	ACACA	Carboxylases			
5932	-54.79	kd	CGS001-3458	IFNG	Interferons			
5933	-54.8	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
5934	-54.83	oe	ccsbBroad304_06048	CRYZ	-			
5935	-54.85	cc		RNA Polymerase Enzymes LOF	-			
5936	-54.96	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
5937	-54.98	kd	CGS001-23212	RRS1	-			
5938	-55.1	oe	ccsbBroad304_14291	GDPD5	-			
5939	-55.12	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
5940	-55.13	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5941	-55.13	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
5942	-55.15	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
5943	-55.16	kd	CGS001-26271	FBXO5	F-boxes / other			
5944	-55.21	kd	CGS001-26298	EHF	-			
5945	-55.22	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
5946	-55.23	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
5947	-55.24	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
5948	-55.24	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
5949	-55.28	kd	CGS001-84290	CAPNS2	EF-hand domain containing			
5950	-55.31	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
5951	-55.33	kd	CGS001-10198	MPHOSPH9	-			
5952	-55.36	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
5953	-55.36	kd	CGS001-3226	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
5954	-55.37	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
5955	-55.43	kd	CGS001-57157	PHTF2	-			
5956	-55.47	kd	CGS001-23678	SGK3	SGK family			
5957	-55.54	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
5958	-55.57	cp	BRD-K85925969	zalcitabine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
5959	-55.57	kd	CGS001-5359	PLSCR1	-			
5960	-55.6	cc		Proteasome inhibitor	-			
5961	-55.65	oe	ccsbBroad304_01001	MEST	-			
5962	-55.71	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
5963	-55.71	kd	CGS001-54957	TXNL4B	-			
5964	-55.72	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
5965	-55.74	oe	ccsbBroad304_03934	LEPRE1	-			
5966	-55.74	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
5967	-55.87	oe	ccsbBroad304_02416	TUBB4B	-			
5968	-55.9	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
5969	-55.91	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
5970	-55.91	kd	CGS001-9978	RBX1	RING-type (C3HC4) zinc fingers			
5971	-56.01	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
5972	-56.06	kd	CGS001-89765	RSPH1	-			
5973	-56.08	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
5974	-56.08	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5975	-56.09	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
5976	-56.18	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
5977	-56.19	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
5978	-56.22	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5979	-56.25	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
5980	-56.26	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
5981	-56.26	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
5982	-56.27	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
5983	-56.29	kd	CGS001-4968	OGG1	-			
5984	-56.33	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
5985	-56.38	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
5986	-56.38	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
5987	-56.41	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
5988	-56.45	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
5989	-56.55	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
5990	-56.55	kd	CGS001-11186	RASSF1	-			
5991	-56.6	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
5992	-56.65	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
5993	-56.65	kd	CGS001-2729	GCLC	-			
5994	-56.68	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
5995	-56.83	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
5996	-56.85	cc		Canonical high mobility group proteins LOF	-			
5997	-56.94	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
5998	-56.95	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
5999	-56.96	oe	ccsbBroad304_02386	EIF1B	-			
6000	-56.96	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
6001	-56.97	oe	ccsbBroad304_07569	TRIB1	Trbl family			
6002	-56.97	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
6003	-56.99	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
6004	-57.01	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
6005	-57.02	oe	ccsbBroad304_00836	IGF2	-			
6006	-57.03	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
6007	-57.03	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
6008	-57.13	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6009	-57.18	kd	CGS001-23387	SIK3	QIK subfamily			
6010	-57.2	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
6011	-57.26	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
6012	-57.26	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
6013	-57.28	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
6014	-57.37	kd	CGS001-10007	GNPDA1	-			
6015	-57.38	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
6016	-57.4	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
6017	-57.4	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
6018	-57.45	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
6019	-57.51	kd	CGS001-2853	GPR31	GPCR / Class A : Orphans			
6020	-57.52	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
6021	-57.6	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
6022	-57.7	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
6023	-57.72	kd	CGS001-1997	ELF1	ETS Transcription Factors			
6024	-57.76	kd	CGS001-3149	HMGB3	High-mobility group / Canonical			
6025	-57.79	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
6026	-57.8	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6027	-57.81	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
6028	-57.82	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
6029	-57.82	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
6030	-57.84	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
6031	-57.9	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
6032	-57.9	cp	BRD-K04710043	hexamethylenebisacetamide	AKT inhibitor			AKT inhibitor, Differentiation inducer, NFkB pathway inhibitor
6033	-58.03	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
6034	-58.05	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
6035	-58.06	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
6036	-58.18	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
6037	-58.19	oe	ccsbBroad304_08426	TEX10	-			
6038	-58.3	kd	CGS001-9377	COX5A	Mitochondrial respiratory chain complex			
6039	-58.36	kd	CGS001-1460	CSNK2B	Casein kinase 2 (CK2) family			
6040	-58.37	oe	ccsbBroad304_00223	CASP9	Caspases			
6041	-58.37	kd	CGS001-64858	DCLRE1B	-			
6042	-58.37	kd	CGS001-2017	CTTN	-			
6043	-58.38	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
6044	-58.44	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
6045	-58.44	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6046	-58.44	kd	CGS001-2495	FTH1	-			
6047	-58.47	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
6048	-58.48	oe	ccsbBroad304_07017	SUOX	-			
6049	-58.51	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6050	-58.58	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
6051	-58.6	oe	ccsbBroad304_00728	HBE1	-			
6052	-58.6	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
6053	-58.61	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
6054	-58.7	kd	CGS001-6663	SOX10	SRY (sex determining region Y)-boxes			
6055	-58.78	oe	ccsbBroad304_02306	PQBP1	-			
6056	-58.84	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
6057	-58.85	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
6058	-58.88	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
6059	-58.9	kd	CGS001-51545	ZNF581	Zinc fingers, C2H2-type			
6060	-58.92	oe	ccsbBroad304_02218	IKBKE	IKK family			
6061	-58.95	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
6062	-59.01	oe	ccsbBroad304_01148	PCBD1	-			
6063	-59.05	kd	CGS001-94239	H2AFV	Histones / Replication-independent			
6064	-59.19	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
6065	-59.19	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
6066	-59.27	cc		Trace amine receptors LOF	-			
6067	-59.32	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
6068	-59.33	oe	ccsbBroad304_00933	LDHB	-			
6069	-59.4	oe	ccsbBroad304_06651	NOV	-			
6070	-59.5	kd	CGS001-3832	KIF11	Kinesins			
6071	-59.5	oe	ccsbBroad304_00225	CAT	-			
6072	-59.59	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
6073	-59.62	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
6074	-59.71	cc		SRY LOF	-			
6075	-59.77	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
6076	-59.79	kd	CGS001-9308	CD83	CD molecules			
6077	-59.84	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
6078	-59.93	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6079	-59.94	kd	CGS001-23658	LSM5	-			
6080	-59.96	kd	CGS001-1503	CTPS	-			
6081	-59.97	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
6082	-60.01	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
6083	-60.03	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
6084	-60.24	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
6085	-60.24	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
6086	-60.29	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
6087	-60.33	kd	CGS001-678	ZFP36L2	RING-type (C3HC4) zinc fingers			
6088	-60.33	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
6089	-60.37	kd	CGS001-406	ARNTL	Basic helix-loop-helix proteins			
6090	-60.38	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
6091	-60.39	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6092	-60.4	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
6093	-60.4	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
6094	-60.45	kd	CGS001-533	ATP6V0B	ATPases / V-type			
6095	-60.55	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
6096	-60.56	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
6097	-60.57	oe	ccsbBroad304_09225	BUD13	-			
6098	-60.62	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
6099	-60.63	cc		Imidazoline ligand	-			
6100	-60.71	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
6101	-60.76	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
6102	-60.8	cp	BRD-K66896231	BRD-K66896231	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
6103	-60.85	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
6104	-60.93	oe	ccsbBroad304_06639	NFYB	-			
6105	-61.02	oe	ccsbBroad304_03773	CIAPIN1	-			
6106	-61.02	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
6107	-61.14	kd	CGS001-5277	PIGA	Glycosyltransferase group 1 domain containing			
6108	-61.15	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
6109	-61.17	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
6110	-61.2	kd	CGS001-3127	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
6111	-61.27	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
6112	-61.29	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
6113	-61.39	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
6114	-61.43	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
6115	-61.48	cc		NADH ubiquinone oxidoreductase supernumerary subunits LOF	-			
6116	-61.53	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
6117	-61.54	kd	CGS001-95	ACY1	-			
6118	-61.55	kd	CGS001-6605	SMARCE1	-			
6119	-61.58	kd	CGS001-9787	DLGAP5	-			
6120	-61.59	oe	ccsbBroad304_00060	AMBP	Lipocalins			
6121	-61.61	kd	CGS001-51053	GMNN	-			
6122	-61.75	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
6123	-61.83	kd	CGS001-25819	CCRN4L	-			
6124	-61.89	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
6125	-61.95	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
6126	-61.97	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
6127	-61.97	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
6128	-61.97	kd	CGS001-23325	KIAA1033	-			
6129	-61.99	kd	CGS001-11344	TWF2	Twinfilin subfamily			
6130	-62	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
6131	-62.06	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
6132	-62.15	kd	CGS001-8996	NOL3	-			
6133	-62.16	oe	ccsbBroad304_07820	SNW1	-			
6134	-62.16	kd	CGS001-285267	ZNF619	Zinc fingers, C2H2-type			
6135	-62.18	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
6136	-62.2	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
6137	-62.23	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
6138	-62.3	oe	ccsbBroad304_01091	NFIB	-			
6139	-62.44	kd	CGS001-54472	TOLLIP	-			
6140	-62.53	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6141	-62.78	kd	CGS001-3030	HADHA	-			
6142	-62.82	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
6143	-62.9	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
6144	-62.95	oe	ccsbBroad304_02367	CALCOCO2	-			
6145	-62.95	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
6146	-63.04	kd	CGS001-4087	SMAD2	SMADs			
6147	-63.05	kd	CGS001-4905	NSF	ATPases / AAA-type			
6148	-63.07	oe	ccsbBroad304_06004	CKB	-			
6149	-63.08	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
6150	-63.11	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
6151	-63.16	kd	CGS001-84936	ZFYVE19	Zinc fingers, FYVE domain containing			
6152	-63.28	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
6153	-63.31	oe	ccsbBroad304_14143	NUSAP1	-			
6154	-63.33	oe	ccsbBroad304_03268	GMPR2	-			
6155	-63.58	kd	CGS001-10887	PROKR1	GPCR / Class A : Prokineticin receptors			
6156	-63.68	kd	CGS001-84634	KISS1R	GPCR / Class A : RF amide peptide receptors			
6157	-63.68	kd	CGS001-3593	IL12B	Interleukins and interleukin receptors			
6158	-63.77	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
6159	-63.8	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
6160	-63.84	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
6161	-63.86	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
6162	-63.89	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6163	-63.94	kd	CGS001-10682	EBP	-			
6164	-64.02	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
6165	-64.08	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6166	-64.1	kd	CGS001-6195	RPS6KA1	RSK subfamily			
6167	-64.17	cp	BRD-K33483813	actarit	Interleukin receptor agonist			Interleukin receptor agonist
6168	-64.21	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
6169	-64.22	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
6170	-64.28	kd	CGS001-9637	FEZ2	-			
6171	-64.53	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
6172	-64.62	kd	CGS001-259	AMBP	Lipocalins			
6173	-64.63	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
6174	-64.63	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
6175	-64.63	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6176	-64.63	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6177	-64.63	kd	CGS001-5159	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6178	-64.67	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
6179	-64.68	kd	CGS001-3248	HPGD	Prostaglandin synthases			
6180	-64.7	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
6181	-64.73	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
6182	-64.83	kd	CGS001-5515	PPP2CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6183	-64.84	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
6184	-64.84	kd	CGS001-5645	PRSS2	Serine peptidases			
6185	-64.88	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
6186	-64.91	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
6187	-64.91	kd	CGS001-2099	ESR1	Estrogen receptors			
6188	-64.94	oe	ccsbBroad304_00106	ARRB1	-			
6189	-64.97	oe	ccsbBroad304_06094	DFFA	-			
6190	-64.97	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
6191	-64.99	kd	CGS001-121599	SPIC	ETS Transcription Factors			
6192	-65.01	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6193	-65.02	kd	CGS001-4846	NOS3	Nitric oxide synthases			
6194	-65.06	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
6195	-65.11	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
6196	-65.13	oe	ccsbBroad304_00038	AGL	-			
6197	-65.13	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
6198	-65.14	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
6199	-65.19	cc		HOXL subclass homeoboxes LOF	-			
6200	-65.21	kd	CGS001-433	ASGR2	C-type lectin domain containing			
6201	-65.3	kd	CGS001-8220	DGCR14	-			
6202	-65.36	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
6203	-65.4	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
6204	-65.44	oe	ccsbBroad304_04619	GNG8	-			
6205	-65.48	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
6206	-65.53	kd	CGS001-10915	TCERG1	-			
6207	-65.57	kd	CGS001-53632	PRKAG3	AMPK subfamily			
6208	-65.57	kd	CGS001-54438	GFOD1	-			
6209	-65.58	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
6210	-65.58	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
6211	-65.59	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
6212	-65.61	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
6213	-65.64	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
6214	-65.66	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
6215	-65.67	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
6216	-65.71	kd	CGS001-2153	F5	Blood coagulation components			
6217	-65.72	oe	ccsbBroad304_00644	GCLC	-			
6218	-65.72	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
6219	-65.74	oe	ccsbBroad304_03848	METTL14	-			
6220	-65.78	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
6221	-65.9	kd	CGS001-11267	SNF8	-			
6222	-65.97	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
6223	-66.03	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
6224	-66.07	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
6225	-66.14	kd	CGS001-6500	SKP1	-			
6226	-66.15	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
6227	-66.21	kd	CGS001-3676	ITGA4	Integrins			
6228	-66.29	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
6229	-66.31	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
6230	-66.31	kd	CGS001-10427	SEC24B	-			
6231	-66.36	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
6232	-66.4	kd	CGS001-51284	TLR7	Toll-like receptor family			
6233	-66.44	kd	CGS001-57459	GATAD2B	GATA zinc finger domain containing			
6234	-66.47	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6235	-66.48	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
6236	-66.48	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
6237	-66.53	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
6238	-66.54	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
6239	-66.56	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
6240	-66.57	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
6241	-66.64	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
6242	-66.66	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
6243	-66.69	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
6244	-66.71	kd	CGS001-10607	TBL3	WD repeat domain containing			
6245	-66.71	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
6246	-66.75	oe	ccsbBroad304_06535	LPL	-			
6247	-66.77	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
6248	-66.87	oe	ccsbBroad304_06159	CTTN	-			
6249	-66.97	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
6250	-67	oe	ccsbBroad304_04194	ELL3	-			
6251	-67	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
6252	-67.13	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
6253	-67.15	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
6254	-67.2	oe	ccsbBroad304_00888	ITPK1	-			
6255	-67.2	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
6256	-67.29	kd	CGS001-4077	NBR1	-			
6257	-67.32	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
6258	-67.33	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6259	-67.34	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
6260	-67.38	kd	CGS001-2000	ELF4	ETS Transcription Factors			
6261	-67.47	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
6262	-67.49	oe	ccsbBroad304_00390	CTGF	-			
6263	-67.49	kd	CGS001-116443	GRIN3A	Glutamate receptors			
6264	-67.52	kd	CGS001-3783	KCNN4	Calcium-activated potassium channels			
6265	-67.55	kd	CGS001-23492	CBX7	-			
6266	-67.61	kd	CGS001-9703	KIAA0100	-			
6267	-67.68	kd	CGS001-8446	DUSP11	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6268	-67.69	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6269	-67.72	kd	CGS001-23066	CAND2	-			
6270	-67.75	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
6271	-67.87	kd	CGS001-1195	CLK1	CDC-like kinases			
6272	-67.89	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
6273	-67.98	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
6274	-68.06	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
6275	-68.16	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6276	-68.17	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
6277	-68.2	kd	CGS001-2879	GPX4	-			
6278	-68.32	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6279	-68.32	kd	CGS001-79862	ZNF669	Zinc fingers, C2H2-type			
6280	-68.34	oe	ccsbBroad304_02109	XPR1	-			
6281	-68.34	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
6282	-68.38	kd	CGS001-56616	DIABLO	-			
6283	-68.4	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
6284	-68.4	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
6285	-68.41	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
6286	-68.45	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
6287	-68.46	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6288	-68.54	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
6289	-68.59	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
6290	-68.61	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
6291	-68.65	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
6292	-68.69	kd	CGS001-36	ACADSB	-			
6293	-68.73	kd	CGS001-2263	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
6294	-68.81	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
6295	-68.84	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
6296	-68.85	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
6297	-68.89	oe	ccsbBroad304_07814	SACM1L	-			
6298	-68.93	kd	CGS001-5164	PDK2	PDHK family			
6299	-68.96	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
6300	-68.96	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6301	-69.02	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
6302	-69.03	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
6303	-69.08	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
6304	-69.15	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
6305	-69.17	oe	ccsbBroad304_00874	INS	-			
6306	-69.3	cp	BRD-K51671335	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
6307	-69.33	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
6308	-69.38	oe	ccsbBroad304_02195	SPAG7	-			
6309	-69.43	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
6310	-69.47	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
6311	-69.55	kd	CGS001-486	FXYD2	Ion transport regulator			
6312	-69.59	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
6313	-69.6	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
6314	-69.62	oe	ccsbBroad304_01180	PFKFB3	-			
6315	-69.68	oe	ccsbBroad304_06144	EFNB3	Ephrins			
6316	-69.68	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
6317	-69.69	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
6318	-69.7	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
6319	-69.72	kd	CGS001-10841	FTCD	-			
6320	-69.73	oe	ccsbBroad304_02956	EHF	-			
6321	-69.81	kd	CGS001-10957	PNRC1	-			
6322	-69.82	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
6323	-69.99	kd	CGS001-3383	ICAM1	CD molecules			
6324	-70.08	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
6325	-70.13	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
6326	-70.2	oe	ccsbBroad304_01673	TIMP3	-			
6327	-70.22	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
6328	-70.23	kd	CGS001-1287	COL4A5	Collagens			
6329	-70.26	kd	CGS001-56882	CDC42SE1	-			
6330	-70.33	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
6331	-70.36	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6332	-70.39	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
6333	-70.41	kd	CGS001-3171	FOXA3	Forkhead boxes			
6334	-70.43	oe	ccsbBroad304_06828	PYCR1	-			
6335	-70.44	cc		Bromodomain Inhibitor	-			
6336	-70.44	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
6337	-70.44	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
6338	-70.47	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
6339	-70.5	oe	ccsbBroad304_06992	SRC	Src family			
6340	-70.52	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
6341	-70.56	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
6342	-70.56	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6343	-70.57	oe	ccsbBroad304_08055	ATP5S	-			
6344	-70.58	oe	ccsbBroad304_00034	AES	-			
6345	-70.58	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
6346	-70.61	kd	CGS001-3559	IL2RA	IL-2 receptor family			
6347	-70.63	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
6348	-70.67	kd	CGS001-6857	SYT1	Synaptotagmins			
6349	-70.72	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
6350	-70.76	kd	CGS001-64376	IKZF5	IKAROS zinc fingers			
6351	-70.77	kd	CGS001-1036	CDO1	-			
6352	-70.78	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
6353	-70.79	kd	CGS001-9406	ZRANB2	Zinc fingers, RAN-binding domain containing			
6354	-70.88	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
6355	-70.89	oe	ccsbBroad304_00532	F11	Chymotrypsin			
6356	-70.9	kd	CGS001-28964	GIT1	Ankyrin repeat domain containing			
6357	-70.92	kd	CGS001-25913	POT1	-			
6358	-71	kd	CGS001-23451	SF3B1	-			
6359	-71.05	oe	ccsbBroad304_00397	CTSK	Cathepsins			
6360	-71.09	kd	CGS001-3689	ITGB2	Integrins			
6361	-71.17	oe	ccsbBroad304_00617	GBA	-			
6362	-71.2	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
6363	-71.25	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
6364	-71.27	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6365	-71.28	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
6366	-71.29	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6367	-71.3	kd	CGS001-2355	FOSL2	basic leucine zipper proteins			
6368	-71.33	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6369	-71.39	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
6370	-71.41	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
6371	-71.41	oe	ccsbBroad304_05981	CDO1	-			
6372	-71.45	oe	ccsbBroad304_00009	ACLY	-			
6373	-71.47	kd	CGS001-7172	TPMT	-			
6374	-71.48	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
6375	-71.51	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
6376	-71.51	kd	CGS001-23597	ACOT9	Acyl CoA thioesterases			
6377	-71.53	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
6378	-71.54	kd	CGS001-2538	G6PC	-			
6379	-71.57	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6380	-71.59	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
6381	-71.68	kd	CGS001-22818	COPZ1	-			
6382	-71.72	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
6383	-71.77	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
6384	-71.79	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
6385	-71.82	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6386	-71.82	kd	CGS001-64422	ATG3	-			
6387	-71.84	kd	CGS001-835	CASP2	Caspases			
6388	-71.85	kd	CGS001-9374	PPT2	-			
6389	-71.89	kd	CGS001-26574	AATF	-			
6390	-71.93	kd	CGS001-84365	MKI67IP	-			
6391	-71.96	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
6392	-72.09	kd	CGS001-84722	PSRC1	-			
6393	-72.11	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
6394	-72.11	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
6395	-72.12	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
6396	-72.13	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
6397	-72.13	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
6398	-72.15	kd	CGS001-7625	ZNF74	Zinc fingers, C2H2-type			
6399	-72.21	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
6400	-72.24	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
6401	-72.29	kd	CGS001-55437	STRADB	STLK subfamily			
6402	-72.35	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
6403	-72.38	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6404	-72.38	kd	CGS001-2783	GNB2	WD repeat domain containing			
6405	-72.39	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
6406	-72.56	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
6407	-72.57	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
6408	-72.6	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
6409	-72.63	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
6410	-72.63	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
6411	-72.65	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
6412	-72.66	kd	CGS001-2987	GUK1	-			
6413	-72.72	kd	CGS001-23211	ZC3H4	Zinc fingers, CCCH-type domain containing			
6414	-72.74	oe	ccsbBroad304_02822	ARFIP2	-			
6415	-72.74	kd	CGS001-9638	FEZ1	-			
6416	-72.77	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
6417	-72.78	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
6418	-72.8	kd	CGS001-833	CARS	Aminoacyl tRNA synthetases / Class I			
6419	-72.82	kd	CGS001-19	ABCA1	ATP binding cassette transporters / subfamily A			
6420	-72.94	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
6421	-72.95	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
6422	-73.03	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
6423	-73.03	kd	CGS001-901	CCNG2	-			
6424	-73.04	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
6425	-73.08	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
6426	-73.1	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
6427	-73.16	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
6428	-73.24	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
6429	-73.26	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
6430	-73.32	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
6431	-73.47	kd	CGS001-7155	TOP2B	DNA Topoisomerases			
6432	-73.48	kd	CGS001-8295	TRRAP	TRRAP subfamily			
6433	-73.5	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
6434	-73.53	kd	CGS001-3046	HBE1	-			
6435	-73.58	kd	CGS001-64147	KIF9	Kinesins			
6436	-73.62	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6437	-73.64	oe	ccsbBroad304_07548	TSSC4	-			
6438	-73.64	kd	CGS001-6514	SLC2A2	Solute carriers			
6439	-73.67	kd	CGS001-23062	GGA2	-			
6440	-73.72	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
6441	-73.75	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
6442	-73.77	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
6443	-73.77	kd	CGS001-6909	TBX2	T-boxes			
6444	-73.84	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
6445	-73.95	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
6446	-73.97	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6447	-73.97	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
6448	-74.16	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
6449	-74.3	oe	ccsbBroad304_02772	ICMT	-			
6450	-74.34	kd	CGS001-3988	LIPA	-			
6451	-74.35	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
6452	-74.45	kd	CGS001-1198	CLK3	CDC-like kinases			
6453	-74.46	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
6454	-74.5	oe	ccsbBroad304_02458	STK25	YSK subfamily			
6455	-74.5	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
6456	-74.54	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
6457	-74.58	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
6458	-74.6	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
6459	-74.63	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
6460	-74.65	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
6461	-74.69	oe	ccsbBroad304_09054	EGFL8	-			
6462	-74.69	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
6463	-74.84	oe	ccsbBroad304_00150	BAX	-			
6464	-74.84	kd	CGS001-5162	PDHB	-			
6465	-74.84	kd	CGS001-593	BCKDHA	-			
6466	-74.85	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
6467	-74.86	oe	ccsbBroad304_01754	UCK2	-			
6468	-74.86	kd	CGS001-1284	COL4A2	Collagens			
6469	-75	kd	CGS001-1999	ELF3	ETS Transcription Factors			
6470	-75.01	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
6471	-75.07	oe	ccsbBroad304_00098	ARG1	Arginase			
6472	-75.11	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6473	-75.13	kd	CGS001-64094	SMOC2	EF-hand domain containing			
6474	-75.13	kd	CGS001-2834	PRLHR	GPCR / Class A : RF amide peptide receptors			
6475	-75.16	kd	CGS001-1070	CETN3	EF-hand domain containing			
6476	-75.16	kd	CGS001-930	CD19	CD molecules			
6477	-75.17	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
6478	-75.26	kd	CGS001-10295	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
6479	-75.32	oe	ccsbBroad304_00960	SMAD1	SMADs			
6480	-75.32	kd	CGS001-1622	DBI	-			
6481	-75.35	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
6482	-75.39	oe	ccsbBroad304_03917	RBKS	-			
6483	-75.41	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
6484	-75.42	kd	CGS001-337867	UBAC2	-			
6485	-75.44	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
6486	-75.46	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
6487	-75.47	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
6488	-75.51	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
6489	-75.57	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
6490	-75.59	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
6491	-75.64	kd	CGS001-3827	KNG1	Endogenous ligands			
6492	-75.64	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
6493	-75.68	oe	ccsbBroad304_06350	HAL	-			
6494	-75.68	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
6495	-75.71	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
6496	-75.76	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
6497	-75.81	kd	CGS001-5336	PLCG2	Phosphoinositide-specific phospholipase C			
6498	-75.87	oe	ccsbBroad304_00492	EIF5A	-			
6499	-75.88	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
6500	-75.91	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6501	-75.99	kd	CGS001-9181	ARHGEF2	Rho guanine nucleotide exchange factors			
6502	-76	oe	ccsbBroad304_00568	FHL2	-			
6503	-76.07	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
6504	-76.09	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
6505	-76.12	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
6506	-76.26	kd	CGS001-650	BMP2	Bone morphogenetic proteins			
6507	-76.27	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
6508	-76.28	kd	CGS001-2976	GTF3C2	General transcription factors			
6509	-76.29	kd	CGS001-84930	MASTL	MAST family			
6510	-76.34	cp	BRD-K49404994	levetiracetam	Calcium channel blocker		SV2A, CACNA1B, SCN1A	Calcium channel blocker
6511	-76.37	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
6512	-76.47	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
6513	-76.53	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
6514	-76.57	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
6515	-76.6	cc		Thromboxane receptor antagonist	-			
6516	-76.68	kd	CGS001-7337	UBE3A	-			
6517	-76.68	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
6518	-76.77	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
6519	-76.84	kd	CGS001-353	APRT	-			
6520	-76.88	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
6521	-76.88	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
6522	-76.91	oe	ccsbBroad304_06286	GLUL	-			
6523	-76.92	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
6524	-76.95	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
6525	-76.96	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
6526	-76.97	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
6527	-77.08	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
6528	-77.08	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
6529	-77.08	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
6530	-77.17	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
6531	-77.22	kd	CGS001-2152	F3	CD molecules			
6532	-77.24	kd	CGS001-2108	ETFA	-			
6533	-77.26	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
6534	-77.27	kd	CGS001-85027	C5ORF62	-			
6535	-77.35	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
6536	-77.36	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
6537	-77.38	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
6538	-77.4	kd	CGS001-80314	EPC1	-			
6539	-77.44	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
6540	-77.45	cp	BRD-K92413528	thiazolidinecarboxylic-acid	Reducing agent			Reducing agent
6541	-77.47	oe	ccsbBroad304_00053	ALDOA	-			
6542	-77.51	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
6543	-77.52	cp	BRD-K39391626	ethylestrenol	Progesterone receptor agonist		AR	Progesterone receptor agonist
6544	-77.54	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
6545	-77.55	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
6546	-77.56	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
6547	-77.63	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
6548	-77.65	kd	CGS001-2767	GNA11	-			
6549	-77.66	kd	CGS001-3925	STMN1	-			
6550	-77.68	kd	CGS001-663	BNIP2	-			
6551	-77.71	kd	CGS001-5663	PSEN1	Presenilin			
6552	-77.72	kd	CGS001-11254	SLC6A14	Glycine transporter subfamily			
6553	-77.8	kd	CGS001-3682	ITGAE	Integrins			
6554	-77.92	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
6555	-78.18	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
6556	-78.18	kd	CGS001-6776	STAT5A	SH2 domain containing			
6557	-78.27	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
6558	-78.28	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
6559	-78.32	oe	ccsbBroad304_00070	ANXA5	Annexins			
6560	-78.33	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
6561	-78.36	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
6562	-78.52	cp	BRD-K10065684	dantron	Laxative			Laxative
6563	-78.57	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
6564	-78.63	kd	CGS001-3575	IL7R	IL-2 receptor family			
6565	-78.64	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6566	-78.67	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
6567	-78.68	oe	ccsbBroad304_04190	CCDC92	-			
6568	-78.69	cc		KCNJ11 modulator	-			
6569	-78.7	kd	CGS001-839	CASP6	Caspases			
6570	-78.75	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
6571	-78.76	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
6572	-78.86	kd	CGS001-4016	LOXL1	-			
6573	-78.87	kd	CGS001-166793	ZBTB49	BTB/POZ domain containing			
6574	-78.92	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6575	-78.93	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
6576	-78.97	kd	CGS001-10481	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
6577	-79.05	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
6578	-79.06	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
6579	-79.1	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
6580	-79.23	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
6581	-79.24	cc		Serine proteases GOF	-			
6582	-79.33	cp	BRD-A39172021	ampiroxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6583	-79.33	kd	CGS001-10671	DCTN6	-			
6584	-79.39	kd	CGS001-1948	EFNB2	Ephrins			
6585	-79.39	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
6586	-79.49	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6587	-79.51	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
6588	-79.53	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6589	-79.54	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
6590	-79.58	kd	CGS001-8777	MPDZ	-			
6591	-79.6	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
6592	-79.62	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
6593	-79.66	oe	ccsbBroad304_01222	PLP2	-			
6594	-79.66	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
6595	-79.71	oe	ccsbBroad304_06820	PTS	-			
6596	-79.71	kd	CGS001-10695	CNPY3	Trinucleotide (CAG) repeat containing			
6597	-79.78	kd	CGS001-64241	ABCG8	ATP binding cassette transporters / subfamily G			
6598	-79.81	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
6599	-79.91	oe	ccsbBroad304_02318	KIF20A	Kinesins			
6600	-79.94	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
6601	-79.98	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
6602	-80.01	kd	CGS001-54659	UGT1A3	UDP glucuronosyltransferases			
6603	-80.04	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
6604	-80.04	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
6605	-80.22	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
6606	-80.33	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
6607	-80.35	oe	ccsbBroad304_06523	LIG1	-			
6608	-80.38	kd	CGS001-283150	FOXR1	Forkhead boxes			
6609	-80.44	oe	ccsbBroad304_00518	ETFA	-			
6610	-80.47	kd	CGS001-4637	MYL6	EF-hand domain containing			
6611	-80.53	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
6612	-80.55	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
6613	-80.64	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
6614	-80.67	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
6615	-80.67	kd	CGS001-6720	SREBF1	Basic helix-loop-helix proteins			
6616	-80.69	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
6617	-80.77	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
6618	-80.78	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
6619	-80.81	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
6620	-80.81	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
6621	-80.83	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
6622	-80.86	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
6623	-80.86	kd	CGS001-114112	TXNRD3	-			
6624	-80.88	kd	CGS001-9341	VAMP3	Vesicle-associated membrane proteins			
6625	-80.92	kd	CGS001-7358	UGDH	-			
6626	-80.93	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
6627	-80.96	kd	CGS001-351	APP	Endogenous ligands			
6628	-81	oe	ccsbBroad304_00464	DTNA	-			
6629	-81.12	oe	ccsbBroad304_00542	FBP1	-			
6630	-81.23	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
6631	-81.24	kd	CGS001-2805	GOT1	-			
6632	-81.25	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
6633	-81.27	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
6634	-81.34	kd	CGS001-8692	HYAL2	-			
6635	-81.37	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
6636	-81.57	kd	CGS001-3281	HSBP1	-			
6637	-81.58	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
6638	-81.61	oe	ccsbBroad304_01556	SMARCB1	-			
6639	-81.71	oe	ccsbBroad304_08481	CEP55	-			
6640	-81.71	kd	CGS001-6309	SC5DL	-			
6641	-81.71	kd	CGS001-2958	GTF2A2	General transcription factors			
6642	-81.78	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
6643	-81.9	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
6644	-81.91	kd	CGS001-335	APOA1	Apolipoproteins			
6645	-81.97	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
6646	-81.97	kd	CGS001-3177	SLC29A2	SLC29 family			
6647	-81.98	oe	ccsbBroad304_06253	GALT	-			
6648	-82.04	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
6649	-82.14	kd	CGS001-4798	NFRKB	INO80 complex subunits			
6650	-82.2	oe	ccsbBroad304_00389	CTBP1	-			
6651	-82.2	kd	CGS001-6541	SLC7A1	SLC7 family			
6652	-82.26	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
6653	-82.28	oe	ccsbBroad304_00657	GNG4	-			
6654	-82.41	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
6655	-82.42	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
6656	-82.43	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
6657	-82.54	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
6658	-82.6	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
6659	-82.62	oe	ccsbBroad304_02349	MPHOSPH9	-			
6660	-82.64	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
6661	-82.65	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
6662	-82.73	oe	ccsbBroad304_07851	FAM120A	-			
6663	-82.74	kd	CGS001-5699	PSMB10	Proteasome (prosome, macropain) subunits			
6664	-82.84	oe	ccsbBroad304_05948	CCND2	-			
6665	-82.88	oe	ccsbBroad304_06683	FURIN	Subtilisin			
6666	-82.89	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
6667	-82.93	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
6668	-82.96	cc		Bacterial 30S ribosomal subunit inhibitor	-			
6669	-82.99	kd	CGS001-130497	OSR1	Zinc fingers, C2H2-type			
6670	-83.01	oe	ccsbBroad304_02572	SERINC3	-			
6671	-83.03	oe	ccsbBroad304_06235	G6PD	-			
6672	-83.06	kd	CGS001-339403	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
6673	-83.07	kd	CGS001-7474	WNT5A	Endogenous ligands			
6674	-83.09	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
6675	-83.1	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
6676	-83.17	kd	CGS001-23075	SWAP70	EF-hand domain containing			
6677	-83.18	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
6678	-83.2	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
6679	-83.2	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
6680	-83.22	cp	BRD-A68888262	azelastine	Histamine receptor antagonist		HRH1, CYP2C19	Histamine receptor antagonist
6681	-83.22	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
6682	-83.31	kd	CGS001-4833	NME4	-			
6683	-83.32	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
6684	-83.41	oe	ccsbBroad304_00490	EIF4EBP1	-			
6685	-83.48	kd	CGS001-2771	GNAI2	-			
6686	-83.49	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
6687	-83.52	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
6688	-83.53	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
6689	-83.54	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
6690	-83.59	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
6691	-83.64	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
6692	-83.68	cc		Supressors of cytokine signaling GOF	-			
6693	-83.73	oe	ccsbBroad304_14174	CDKAL1	-			
6694	-83.75	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
6695	-83.79	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
6696	-83.81	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
6697	-83.94	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
6698	-83.99	kd	CGS001-9140	ATG12	-			
6699	-84.01	kd	CGS001-6675	UAP1	-			
6700	-84.05	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
6701	-84.06	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
6702	-84.07	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
6703	-84.1	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
6704	-84.14	oe	ccsbBroad304_01654	TCTA	-			
6705	-84.14	kd	CGS001-975	CD81	CD molecules			
6706	-84.14	kd	CGS001-586	BCAT1	-			
6707	-84.16	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
6708	-84.23	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
6709	-84.29	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
6710	-84.33	kd	CGS001-7248	TSC1	-			
6711	-84.41	kd	CGS001-3065	HDAC1	Histone deacetylases			
6712	-84.46	oe	ccsbBroad304_00085	APRT	-			
6713	-84.56	oe	ccsbBroad304_00418	CD55	CD molecules			
6714	-84.58	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
6715	-84.66	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
6716	-84.66	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
6717	-84.68	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
6718	-84.69	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
6719	-84.72	kd	CGS001-2956	MSH6	-			
6720	-84.77	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
6721	-84.79	kd	CGS001-89882	TPD52L3	-			
6722	-84.82	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6723	-84.84	kd	CGS001-23192	ATG4B	Aut2 peptidase			
6724	-84.86	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
6725	-84.95	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
6726	-84.95	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
6727	-85	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6728	-85	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
6729	-85.15	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
6730	-85.2	oe	ccsbBroad304_00316	CKS1B	-			
6731	-85.21	kd	CGS001-23576	DDAH1	Dimethylarginine dimethylaminohydrolases			
6732	-85.26	kd	CGS001-1515	CTSL2	-			
6733	-85.27	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
6734	-85.37	oe	ccsbBroad304_02032	TSC22D1	-			
6735	-85.37	kd	CGS001-5264	PHYH	-			
6736	-85.44	kd	CGS001-11136	SLC7A9	SLC7 family			
6737	-85.51	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
6738	-85.51	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
6739	-85.53	kd	CGS001-890	CCNA2	-			
6740	-85.54	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
6741	-85.61	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
6742	-85.63	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
6743	-85.65	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
6744	-85.81	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
6745	-85.86	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6746	-85.92	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
6747	-85.92	kd	CGS001-6799	SULT1A2	Sulfotransferases, cytosolic			
6748	-85.95	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
6749	-85.98	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
6750	-86.03	kd	CGS001-475	ATOX1	-			
6751	-86.04	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6752	-86.1	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
6753	-86.12	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
6754	-86.19	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6755	-86.2	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
6756	-86.21	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
6757	-86.22	kd	CGS001-10059	DNM1L	-			
6758	-86.28	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
6759	-86.32	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
6760	-86.32	kd	CGS001-147948	ZNF582	Zinc fingers, C2H2-type			
6761	-86.33	kd	CGS001-6520	SLC3A2	SLC3 family			
6762	-86.35	kd	CGS001-7832	BTG2	-			
6763	-86.39	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
6764	-86.44	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
6765	-86.46	oe	ccsbBroad304_00462	DR1	-			
6766	-86.49	kd	CGS001-11243	PMF1	-			
6767	-86.52	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6768	-86.53	cc		Tachykinin antagonist	-			
6769	-86.53	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
6770	-86.54	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
6771	-86.54	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
6772	-86.57	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
6773	-86.59	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
6774	-86.6	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
6775	-86.62	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
6776	-86.67	kd	CGS001-9326	ZNHIT3	Zinc fingers, HIT-type			
6777	-86.71	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
6778	-86.72	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
6779	-86.73	oe	ccsbBroad304_07219	CDC7	CDC7 family			
6780	-86.73	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
6781	-86.82	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
6782	-86.85	kd	CGS001-1513	CTSK	Cathepsins			
6783	-86.9	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
6784	-86.97	kd	CGS001-960	CD44	CD molecules			
6785	-87.05	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
6786	-87.1	kd	CGS001-91392	ZNF502	Zinc fingers, C2H2-type			
6787	-87.17	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
6788	-87.18	kd	CGS001-408	ARRB1	-			
6789	-87.22	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
6790	-87.24	oe	ccsbBroad304_02741	PDS5A	-			
6791	-87.32	cp	BRD-K05350981	oligomycin-c	ATPase inhibitor		ATP5A1	ATPase inhibitor, ATP synthase inhibitor
6792	-87.39	cp	BRD-K66412701	pazufloxacin	Topoisomerase inhibitor			Topoisomerase inhibitor
6793	-87.45	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
6794	-87.48	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
6795	-87.58	kd	CGS001-29959	NRBP1	NRBP family			
6796	-87.59	kd	CGS001-440387	CTRB2	-			
6797	-87.7	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
6798	-87.72	kd	CGS001-5293	PIK3CD	Phosphatidylinositol kinases			
6799	-87.77	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
6800	-87.79	oe	ccsbBroad304_03732	NPDC1	-			
6801	-87.81	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
6802	-87.85	oe	ccsbBroad304_07275	PSMG1	-			
6803	-87.85	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
6804	-87.85	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6805	-87.9	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
6806	-87.92	kd	CGS001-5058	PAK1	PAKA subfamily			
6807	-87.95	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
6808	-87.97	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
6809	-88.03	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
6810	-88.05	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
6811	-88.05	kd	CGS001-136	ADORA2B	GPCR / Class A : Adenosine receptors			
6812	-88.13	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
6813	-88.16	oe	ccsbBroad304_12106	PXK	Slob family			
6814	-88.18	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
6815	-88.27	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
6816	-88.27	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
6817	-88.29	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
6818	-88.3	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
6819	-88.41	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
6820	-88.41	kd	CGS001-54536	EXOC6	-			
6821	-88.43	oe	ccsbBroad304_03555	PANK4	-			
6822	-88.56	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
6823	-88.58	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
6824	-88.64	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
6825	-88.65	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
6826	-88.69	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
6827	-88.7	kd	CGS001-8848	TSC22D1	-			
6828	-88.75	oe	ccsbBroad304_02626	PKIG	-			
6829	-88.79	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
6830	-88.8	oe	ccsbBroad304_00447	DLD	-			
6831	-88.8	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
6832	-88.82	kd	CGS001-5228	PGF	-			
6833	-88.82	kd	CGS001-976	CD97	Adhesion Class GPCRs			
6834	-88.84	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
6835	-88.85	cc		EMSY complex LOF	-			
6836	-88.87	oe	ccsbBroad304_02217	FEZ1	-			
6837	-88.9	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
6838	-88.94	oe	ccsbBroad304_08536	PARL	-			
6839	-89	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
6840	-89.01	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
6841	-89.03	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
6842	-89.12	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
6843	-89.15	kd	CGS001-2542	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
6844	-89.16	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
6845	-89.21	kd	CGS001-2353	FOS	basic leucine zipper proteins			
6846	-89.28	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
6847	-89.3	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
6848	-89.39	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
6849	-89.4	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
6850	-89.46	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
6851	-89.53	kd	CGS001-54205	CYCS	-			
6852	-89.55	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
6853	-89.57	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
6854	-89.57	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6855	-89.62	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
6856	-89.64	kd	CGS001-50813	COPS7A	-			
6857	-89.65	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
6858	-89.65	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
6859	-89.68	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
6860	-89.69	kd	CGS001-10928	RALBP1	-			
6861	-89.7	kd	CGS001-27034	ACAD8	-			
6862	-89.72	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6863	-89.78	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
6864	-89.8	kd	CGS001-6207	RPS13	S ribosomal proteins			
6865	-89.81	oe	ccsbBroad304_05590	NOTCH2NL	-			
6866	-89.82	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
6867	-89.82	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
6868	-89.83	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
6869	-89.83	kd	CGS001-3479	IGF1	Endogenous ligands			
6870	-89.89	kd	CGS001-26036	ZNF451	Zinc fingers, C2H2-type			
6871	-89.91	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
6872	-89.99	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
6873	-90	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
6874	-90.08	kd	CGS001-2752	GLUL	-			
6875	-90.12	kd	CGS001-3663	IRF5	-			
6876	-90.13	oe	ccsbBroad304_03122	RHOD	-			
6877	-90.15	kd	CGS001-319100	TAAR6	GPCR / Class A : Trace amine associated receptors			
6878	-90.16	oe	ccsbBroad304_07466	VGLL4	-			
6879	-90.16	kd	CGS001-3705	ITPK1	-			
6880	-90.17	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
6881	-90.22	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6882	-90.31	oe	ccsbBroad304_04257	SPRY4	-			
6883	-90.33	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
6884	-90.35	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
6885	-90.36	oe	ccsbBroad304_03433	DDIT4	-			
6886	-90.36	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
6887	-90.37	oe	ccsbBroad304_00329	CLTA	-			
6888	-90.45	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
6889	-90.46	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
6890	-90.48	kd	CGS001-4718	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
6891	-90.49	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
6892	-90.52	kd	CGS001-1429	CRYZ	-			
6893	-90.56	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
6894	-90.58	cp	BRD-K49668410	clarithromycin	Bacterial 50S ribosomal subunit inhibitor		CYP2C19, CYP3A4, CYP3A5, CYP3A7	Bacterial 50S ribosomal subunit inhibitor
6895	-90.63	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
6896	-90.66	oe	ccsbBroad304_04170	PANK2	-			
6897	-90.72	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
6898	-90.72	kd	CGS001-4179	CD46	CD molecules			
6899	-90.75	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
6900	-90.77	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
6901	-90.82	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
6902	-90.86	kd	CGS001-466	ATF1	basic leucine zipper proteins			
6903	-90.93	kd	CGS001-55818	KDM3A	Histone demethylases			
6904	-90.95	kd	CGS001-327	APEH	Prolyl oligopeptidase			
6905	-90.98	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
6906	-91.03	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
6907	-91.11	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
6908	-91.14	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
6909	-91.16	kd	CGS001-2593	GAMT	-			
6910	-91.17	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
6911	-91.17	kd	CGS001-4697	NDUFA4	-			
6912	-91.2	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
6913	-91.25	kd	CGS001-6203	RPS9	S ribosomal proteins			
6914	-91.25	kd	CGS001-8986	RPS6KA4	MSK subfamily			
6915	-91.32	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
6916	-91.38	oe	ccsbBroad304_02133	CD83	CD molecules			
6917	-91.42	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
6918	-91.43	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
6919	-91.43	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
6920	-91.43	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
6921	-91.44	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
6922	-91.44	kd	CGS001-1163	CKS1B	-			
6923	-91.46	kd	CGS001-9352	TXNL1	-			
6924	-91.49	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6925	-91.51	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
6926	-91.53	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6927	-91.68	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
6928	-91.72	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
6929	-91.75	kd	CGS001-8800	PEX11A	-			
6930	-91.76	oe	ccsbBroad304_01183	PGD	-			
6931	-91.76	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
6932	-91.77	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
6933	-91.77	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
6934	-91.78	kd	CGS001-6272	SORT1	-			
6935	-91.8	oe	ccsbBroad304_00810	HYAL1	-			
6936	-91.8	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
6937	-91.83	kd	CGS001-2077	ERF	ETS Transcription Factors			
6938	-91.9	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
6939	-91.9	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
6940	-91.92	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
6941	-91.96	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
6942	-91.97	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
6943	-91.99	oe	ccsbBroad304_07029	TADA2A	-			
6944	-92.01	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6945	-92.03	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
6946	-92.04	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
6947	-92.04	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
6948	-92.06	cp	BRD-A84134924	pancuronium	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRNA1, CHRNA2	Acetylcholine receptor antagonist
6949	-92.1	oe	ccsbBroad304_07088	TP53	-			
6950	-92.18	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
6951	-92.18	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
6952	-92.29	kd	CGS001-3934	LCN2	Lipocalins			
6953	-92.3	kd	CGS001-51271	UBAP1	-			
6954	-92.32	kd	CGS001-1020	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
6955	-92.34	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
6956	-92.42	oe	ccsbBroad304_02497	YKT6	-			
6957	-92.46	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
6958	-92.51	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
6959	-92.51	kd	CGS001-498	ATP5A1	ATPases / F-type			
6960	-92.52	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
6961	-92.53	oe	ccsbBroad304_00966	MAFG	-			
6962	-92.56	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6963	-92.56	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6964	-92.59	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
6965	-92.6	kd	CGS001-4907	NT5E	Adenosine turnover			
6966	-92.62	oe	ccsbBroad304_08952	E2F8	-			
6967	-92.64	oe	ccsbBroad304_06494	KLRC1	CD molecules			
6968	-92.64	kd	CGS001-3670	ISL1	Homeoboxes / LIM class			
6969	-92.64	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
6970	-92.71	kd	CGS001-6429	SRSF4	RNA binding motif (RRM) containing			
6971	-92.71	kd	CGS001-3654	IRAK1	Interleukin-1 receptor-associated kinase (IRAK) family			
6972	-92.8	cp	BRD-K49481516	galantamine	Acetylcholinesterase inhibitor		ACHE, BCHE, CHRNA1, CHRNA10, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNA9, CHRNB1, CHRNB2, CHRNB3, CHRNB4, CHRND, CHRNE, CHRNG	Acetylcholinesterase inhibitor
6973	-92.89	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
6974	-92.89	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
6975	-92.92	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
6976	-92.93	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
6977	-92.98	oe	ccsbBroad304_04490	RSPH1	-			
6978	-92.98	kd	CGS001-23047	PDS5B	-			
6979	-92.99	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
6980	-93.02	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
6981	-93.03	kd	CGS001-8438	RAD54L	-			
6982	-93.11	oe	ccsbBroad304_00658	GNG5	-			
6983	-93.14	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
6984	-93.15	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
6985	-93.15	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
6986	-93.16	kd	CGS001-2232	FDXR	-			
6987	-93.21	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
6988	-93.24	oe	ccsbBroad304_03308	YTHDF2	-			
6989	-93.35	oe	ccsbBroad304_03113	DSE	-			
6990	-93.35	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
6991	-93.37	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
6992	-93.37	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
6993	-93.39	kd	CGS001-5934	RBL2	-			
6994	-93.4	kd	CGS001-23384	SPECC1L	-			
6995	-93.46	oe	ccsbBroad304_07320	SQSTM1	-			
6996	-93.46	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
6997	-93.47	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
6998	-93.48	oe	ccsbBroad304_00615	GAPDH	-			
6999	-93.5	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
7000	-93.53	kd	CGS001-1949	EFNB3	Ephrins			
7001	-93.59	oe	ccsbBroad304_02686	COPZ1	-			
7002	-93.61	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
7003	-93.64	kd	CGS001-4717	NDUFC1	Mitochondrial respiratory chain complex / Complex I			
7004	-93.69	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
7005	-93.69	kd	CGS001-84619	ZGPAT	G patch domain containing			
7006	-93.71	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
7007	-93.73	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
7008	-93.76	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
7009	-93.8	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
7010	-93.84	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
7011	-93.84	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
7012	-93.9	oe	ccsbBroad304_01617	STX4	-			
7013	-93.92	oe	ccsbBroad304_03565	ADI1	-			
7014	-93.92	kd	CGS001-6016	RIT1	-			
7015	-93.94	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
7016	-93.96	cp	BRD-A00520476	otenzepad	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
7017	-94.01	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
7018	-94.02	oe	ccsbBroad304_02815	SSBP2	-			
7019	-94.03	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
7020	-94.04	kd	CGS001-1495	CTNNA1	Catenins			
7021	-94.06	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
7022	-94.06	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
7023	-94.08	kd	CGS001-147837	ZNF563	Zinc fingers, C2H2-type			
7024	-94.09	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
7025	-94.1	kd	CGS001-60493	FASTKD5	-			
7026	-94.12	oe	ccsbBroad304_00147	BAG1	-			
7027	-94.12	kd	CGS001-23657	SLC7A11	Solute carriers			
7028	-94.13	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
7029	-94.15	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
7030	-94.15	kd	CGS001-4287	ATXN3	Ataxins			
7031	-94.16	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
7032	-94.17	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7033	-94.27	kd	CGS001-83440	ADPGK	-			
7034	-94.28	kd	CGS001-5160	PDHA1	-			
7035	-94.32	cp	BRD-A41450521	tosufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
7036	-94.36	kd	CGS001-54807	ZNF586	Zinc fingers, C2H2-type			
7037	-94.37	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
7038	-94.38	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
7039	-94.43	kd	CGS001-2161	F12	Chymotrypsin			
7040	-94.45	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
7041	-94.49	oe	ccsbBroad304_02487	TXNIP	-			
7042	-94.51	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
7043	-94.51	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
7044	-94.54	oe	ccsbBroad304_03772	CCNL1	-			
7045	-94.55	kd	CGS001-10933	MORF4L1	-			
7046	-94.55	kd	CGS001-23210	JMJD6	-			
7047	-94.62	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
7048	-94.7	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
7049	-94.74	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
7050	-94.74	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
7051	-94.74	kd	CGS001-9541	CIR1	-			
7052	-94.76	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
7053	-94.77	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
7054	-94.79	kd	CGS001-57048	PLSCR3	-			
7055	-94.89	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
7056	-94.89	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
7057	-94.97	cp	BRD-K83144676	olmesartan	Angiotensin antagonist		AGTR1	Angiotensin antagonist
7058	-95.03	oe	ccsbBroad304_01623	SUPT4H1	-			
7059	-95.08	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
7060	-95.12	oe	ccsbBroad304_00816	IDE	Pitrilysin			
7061	-95.13	cc		Baculoviral IAP repeat domain containing LOF	-			
7062	-95.15	kd	CGS001-55634	ZNF673	-			
7063	-95.17	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
7064	-95.17	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
7065	-95.2	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
7066	-95.22	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
7067	-95.25	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
7068	-95.25	kd	CGS001-7297	TYK2	Janus kinase (JakA) family			
7069	-95.25	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
7070	-95.29	kd	CGS001-64343	AZI2	-			
7071	-95.3	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
7072	-95.31	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
7073	-95.32	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
7074	-95.34	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
7075	-95.35	kd	CGS001-51776	ZAK	MLK subfamily			
7076	-95.4	cp	BRD-A48261811	argatroban	Thrombin inhibitor		F2, CYP3A5	Thrombin inhibitor
7077	-95.43	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
7078	-95.55	kd	CGS001-6184	RPN1	-			
7079	-95.65	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
7080	-95.67	kd	CGS001-405	ARNT	Basic helix-loop-helix proteins			
7081	-95.71	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
7082	-95.75	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7083	-95.8	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
7084	-95.82	oe	ccsbBroad304_01974	RNASET2	-			
7085	-95.86	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
7086	-95.87	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
7087	-95.95	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
7088	-95.96	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
7089	-95.96	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
7090	-96	kd	CGS001-1831	TSC22D3	-			
7091	-96.02	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
7092	-96.03	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
7093	-96.06	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
7094	-96.11	kd	CGS001-7298	TYMS	Methyltransferases			
7095	-96.13	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
7096	-96.14	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
7097	-96.14	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
7098	-96.17	oe	ccsbBroad304_05757	ACADS	-			
7099	-96.21	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
7100	-96.23	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
7101	-96.23	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
7102	-96.25	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7103	-96.26	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
7104	-96.27	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
7105	-96.3	oe	ccsbBroad304_02432	IFI30	-			
7106	-96.31	cp	BRD-K88304388	dextrorphan	Glutamate receptor antagonist		OPRM1, OPRK1, OPRD1, GRIN1, HTR1A, SLC6A2	Glutamate receptor antagonist
7107	-96.33	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
7108	-96.34	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
7109	-96.35	kd	CGS001-64425	POLR1E	RNA polymerase subunits			
7110	-96.36	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
7111	-96.39	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
7112	-96.41	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
7113	-96.44	cc		Aminoacyl tRNA synthetases class II LOF	-			
7114	-96.44	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
7115	-96.45	oe	ccsbBroad304_09578	PASD1	-			
7116	-96.46	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
7117	-96.48	kd	CGS001-93349	SP140L	Zinc fingers, PHD-type			
7118	-96.53	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
7119	-96.54	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
7120	-96.58	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
7121	-96.59	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7122	-96.6	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
7123	-96.61	kd	CGS001-25824	PRDX5	-			
7124	-96.62	kd	CGS001-6944	VPS72	-			
7125	-96.62	kd	CGS001-1201	CLN3	-			
7126	-96.63	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
7127	-96.64	kd	CGS001-6599	SMARCC1	-			
7128	-96.65	kd	CGS001-2592	GALT	-			
7129	-96.69	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
7130	-96.7	cp	BRD-K63343048	orlistat	Lipase inhibitor		PNLIP, DAGLA, FASN, LIPF, CNR1, DAGLB	Lipase inhibitor
7131	-96.74	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
7132	-96.76	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
7133	-96.81	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
7134	-96.81	kd	CGS001-6282	S100A11	EF-hand domain containing			
7135	-96.83	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
7136	-96.85	oe	ccsbBroad304_05823	ANXA2	Annexins			
7137	-96.89	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
7138	-96.89	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
7139	-96.93	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
7140	-96.94	kd	CGS001-79174	CRELD2	-			
7141	-96.98	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
7142	-96.99	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
7143	-96.99	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
7144	-97.05	kd	CGS001-5916	RARG	Retinoic acid receptors			
7145	-97.07	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
7146	-97.09	oe	ccsbBroad304_01716	TSN	-			
7147	-97.09	kd	CGS001-302	ANXA2	Annexins			
7148	-97.12	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
7149	-97.15	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
7150	-97.16	oe	ccsbBroad304_02565	RALBP1	-			
7151	-97.16	kd	CGS001-4916	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
7152	-97.16	kd	CGS001-2859	GPR35	GPCR / Class A : Orphans			
7153	-97.16	kd	CGS001-9695	EDEM1	-			
7154	-97.17	kd	CGS001-2730	GCLM	-			
7155	-97.18	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
7156	-97.21	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
7157	-97.22	kd	CGS001-7086	TKT	-			
7158	-97.23	oe	ccsbBroad304_00210	CALR	-			
7159	-97.24	oe	ccsbBroad304_02230	HERPUD1	-			
7160	-97.24	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
7161	-97.27	oe	ccsbBroad304_06663	OAS1	-			
7162	-97.29	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
7163	-97.3	kd	CGS001-93185	IGSF8	CD molecules			
7164	-97.32	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
7165	-97.37	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
7166	-97.39	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
7167	-97.41	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
7168	-97.41	kd	CGS001-11142	PKIG	-			
7169	-97.43	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
7170	-97.47	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
7171	-97.51	oe	ccsbBroad304_13499	KSR2	RAF family			
7172	-97.53	kd	CGS001-6632	SNRPD1	-			
7173	-97.55	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7174	-97.55	oe	ccsbBroad304_06386	HNMT	-			
7175	-97.57	kd	CGS001-85315	PAQR8	-			
7176	-97.58	kd	CGS001-5563	PRKAA2	AMPK subfamily			
7177	-97.59	kd	CGS001-6233	RPS27A	S ribosomal proteins			
7178	-97.59	kd	CGS001-23761	PISD	Decarboxylases			
7179	-97.62	oe	ccsbBroad304_07490	SCRN1	-			
7180	-97.64	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
7181	-97.66	kd	CGS001-25801	GCA	EF-hand domain containing			
7182	-97.67	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
7183	-97.68	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7184	-97.69	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
7185	-97.7	kd	CGS001-4938	OAS1	-			
7186	-97.72	kd	CGS001-1594	CYP27B1	Cytochrome P450s			
7187	-97.74	kd	CGS001-54805	CNNM2	-			
7188	-97.75	kd	CGS001-23142	DCUN1D4	-			
7189	-97.75	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
7190	-97.77	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
7191	-97.79	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
7192	-97.81	cp	BRD-K44442813	pidotimod	Interferon receptor agonist			Interferon receptor agonist, Interleukin receptor agonist
7193	-97.84	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
7194	-97.85	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
7195	-97.85	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
7196	-97.9	oe	ccsbBroad304_02045	BUD31	-			
7197	-97.9	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7198	-97.92	oe	ccsbBroad304_05902	BNIP3	-			
7199	-97.93	oe	ccsbBroad304_01933	TEAD2	-			
7200	-97.94	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
7201	-97.94	kd	CGS001-115727	RASGRP4	EF-hand domain containing			
7202	-97.95	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
7203	-97.95	kd	CGS001-54584	GNB1L	WD repeat domain containing			
7204	-97.98	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
7205	-97.98	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
7206	-98	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
7207	-98.03	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
7208	-98.03	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
7209	-98.04	kd	CGS001-6303	SAT1	-			
7210	-98.06	kd	CGS001-4097	MAFG	-			
7211	-98.07	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
7212	-98.1	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
7213	-98.12	kd	CGS001-8667	EIF3H	-			
7214	-98.14	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
7215	-98.14	kd	CGS001-4706	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
7216	-98.15	kd	CGS001-51335	NGRN	-			
7217	-98.18	kd	CGS001-2580	GAK	Heat shock proteins / DNAJ (HSP40)			
7218	-98.19	kd	CGS001-6850	SYK	Syk family			
7219	-98.2	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
7220	-98.21	kd	CGS001-2261	FGFR3	Type V RTKs: FGF (fibroblast growth factor) receptor family			
7221	-98.21	kd	CGS001-4204	MECP2	-			
7222	-98.25	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
7223	-98.25	kd	CGS001-5428	POLG	DNA polymerases			
7224	-98.26	kd	CGS001-1984	EIF5A	-			
7225	-98.27	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
7226	-98.34	oe	ccsbBroad304_00931	LCN2	Lipocalins			
7227	-98.34	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
7228	-98.36	kd	CGS001-9967	THRAP3	-			
7229	-98.38	oe	ccsbBroad304_02419	NDRG1	-			
7230	-98.4	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
7231	-98.4	kd	CGS001-7314	UBB	-			
7232	-98.44	kd	CGS001-221393	GPR115	Adhesion Class GPCRs			
7233	-98.45	oe	ccsbBroad304_02048	BCL10	-			
7234	-98.45	oe	ccsbBroad304_06294	GNAZ	-			
7235	-98.47	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
7236	-98.52	kd	CGS001-64921	CASD1	-			
7237	-98.53	kd	CGS001-966	CD59	CD molecules			
7238	-98.56	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
7239	-98.56	kd	CGS001-2588	GALNS	Arylsulfatase family			
7240	-98.57	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
7241	-98.6	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
7242	-98.61	oe	ccsbBroad304_01787	YES1	Src family			
7243	-98.62	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
7244	-98.64	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
7245	-98.64	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
7246	-98.64	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
7247	-98.64	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
7248	-98.67	kd	CGS001-6658	SOX3	SRY (sex determining region Y)-boxes			
7249	-98.67	kd	CGS001-55312	RFK	-			
7250	-98.68	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
7251	-98.69	kd	CGS001-5450	POU2AF1	-			
7252	-98.69	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
7253	-98.71	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
7254	-98.73	cp	BRD-K51730347	diphencyprone	Immunostimulant			Immunostimulant
7255	-98.73	kd	CGS001-1154	CISH	SH2 domain containing			
7256	-98.74	kd	CGS001-10325	RRAGB	-			
7257	-98.75	kd	CGS001-6732	SRPK1	SRPK family			
7258	-98.75	kd	CGS001-10465	PPIH	-			
7259	-98.75	kd	CGS001-10001	MED6	-			
7260	-98.77	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
7261	-98.77	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
7262	-98.77	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
7263	-98.78	cc		Beta-adrenergic receptor agonist	-			
7264	-98.78	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
7265	-98.79	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
7266	-98.8	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
7267	-98.81	kd	CGS001-6194	RPS6	S ribosomal proteins			
7268	-98.82	kd	CGS001-2597	GAPDH	-			
7269	-98.84	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
7270	-98.85	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
7271	-98.88	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
7272	-98.88	kd	CGS001-11179	ZNF277	-			
7273	-98.88	kd	CGS001-978	CDA	-			
7274	-98.9	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
7275	-98.9	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
7276	-98.94	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
7277	-98.94	kd	CGS001-2078	ERG	ETS Transcription Factors			
7278	-98.95	kd	CGS001-2932	GSK3B	GSK subfamily			
7279	-98.99	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
7280	-99.02	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
7281	-99.02	kd	CGS001-9404	LPXN	-			
7282	-99.03	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
7283	-99.03	kd	CGS001-55038	CDCA4	-			
7284	-99.04	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
7285	-99.04	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7286	-99.04	kd	CGS001-6258	RXRG	Retinoid X receptors			
7287	-99.06	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7288	-99.06	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
7289	-99.06	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
7290	-99.07	kd	CGS001-7128	TNFAIP3	OTU domain containing			
7291	-99.1	oe	ccsbBroad304_07287	HYAL2	-			
7292	-99.12	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
7293	-99.15	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
7294	-99.15	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
7295	-99.15	kd	CGS001-10672	GNA13	-			
7296	-99.2	cc		Mediator complex LOF	-			
7297	-99.23	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
7298	-99.23	oe	ccsbBroad304_00003	ABAT	GABA turnover			
7299	-99.23	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
7300	-99.24	oe	ccsbBroad304_03119	C16ORF5	-			
7301	-99.24	kd	CGS001-23534	TNPO3	Importins			
7302	-99.25	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
7303	-99.26	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
7304	-99.28	oe	ccsbBroad304_09756	PAQR7	-			
7305	-99.28	oe	ccsbBroad304_02173	ATG5	-			
7306	-99.28	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
7307	-99.28	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
7308	-99.29	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
7309	-99.3	kd	CGS001-727	C5	Endogenous ligands			
7310	-99.32	kd	CGS001-462	SERPINC1	Serine (or cysteine) peptidase inhibitors			
7311	-99.32	kd	CGS001-5641	LGMN	Legumain			
7312	-99.34	cp	BRD-A01787639	naftopidil	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
7313	-99.34	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
7314	-99.35	kd	CGS001-5992	RFX4	-			
7315	-99.37	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7316	-99.37	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
7317	-99.37	kd	CGS001-6189	RPS3A	S ribosomal proteins			
7318	-99.37	kd	CGS001-894	CCND2	-			
7319	-99.39	kd	CGS001-26191	PTPN22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
7320	-99.39	kd	CGS001-9774	BCLAF1	-			
7321	-99.41	kd	CGS001-51222	ZNF219	Zinc fingers, C2H2-type			
7322	-99.41	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
7323	-99.41	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
7324	-99.43	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
7325	-99.43	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
7326	-99.43	kd	CGS001-1910	EDNRB	Endothelin receptors			
7327	-99.44	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
7328	-99.45	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
7329	-99.45	kd	CGS001-7343	UBTF	-			
7330	-99.45	kd	CGS001-9945	GFPT2	-			
7331	-99.47	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
7332	-99.5	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
7333	-99.5	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
7334	-99.52	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
7335	-99.52	kd	CGS001-23585	TMEM50A	-			
7336	-99.52	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
7337	-99.52	kd	CGS001-5927	KDM5A	Histone demethylases			
7338	-99.52	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
7339	-99.54	oe	ccsbBroad304_03928	RRAGC	-			
7340	-99.54	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
7341	-99.54	kd	CGS001-5433	POLR2D	RNA polymerase subunits			
7342	-99.54	kd	CGS001-5387	PMS2P3	-			
7343	-99.54	kd	CGS001-140690	CTCFL	Zinc fingers, C2H2-type			
7344	-99.55	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
7345	-99.56	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
7346	-99.56	kd	CGS001-3651	PDX1	Homeoboxes / ANTP class : HOXL subclass			
7347	-99.58	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
7348	-99.61	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
7349	-99.61	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
7350	-99.61	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
7351	-99.61	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
7352	-99.61	kd	CGS001-51701	NLK	nmo subfamily			
7353	-99.63	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
7354	-99.63	oe	ccsbBroad304_03386	SPA17	-			
7355	-99.63	oe	ccsbBroad304_14020	SH3BP5	-			
7356	-99.63	kd	CGS001-5981	RFC1	ATPases / AAA-type			
7357	-99.63	kd	CGS001-226	ALDOA	-			
7358	-99.65	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
7359	-99.65	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
7360	-99.65	kd	CGS001-203523	ZNF449	Zinc fingers, C2H2-type			
7361	-99.65	kd	CGS001-8802	SUCLG1	-			
7362	-99.65	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
7363	-99.66	kd	CGS001-5320	PLA2G2A	Hydrolases			
7364	-99.67	oe	ccsbBroad304_03618	OSGEP	-			
7365	-99.67	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
7366	-99.67	kd	CGS001-6741	SSB	La ribonucleoprotein domain containing			
7367	-99.67	kd	CGS001-23581	CASP14	Caspases			
7368	-99.69	oe	ccsbBroad304_08045	NOX1	-			
7369	-99.69	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
7370	-99.69	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
7371	-99.71	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
7372	-99.72	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
7373	-99.72	kd	CGS001-7535	ZAP70	Syk family			
7374	-99.72	kd	CGS001-7167	TPI1	-			
7375	-99.72	kd	CGS001-9928	KIF14	Kinesins			
7376	-99.72	kd	CGS001-2849	GPR26	GPCR / Class A : Orphans			
7377	-99.73	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7378	-99.74	oe	ccsbBroad304_07632	PROCR	CD molecules			
7379	-99.74	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
7380	-99.76	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
7381	-99.76	oe	ccsbBroad304_02737	JMJD6	-			
7382	-99.76	kd	CGS001-3373	HYAL1	-			
7383	-99.76	kd	CGS001-8841	HDAC3	Histone deacetylases			
7384	-99.78	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
7385	-99.78	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
7386	-99.78	kd	CGS001-5352	PLOD2	-			
7387	-99.8	oe	ccsbBroad304_06234	G6PC	-			
7388	-99.8	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
7389	-99.8	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
7390	-99.8	kd	CGS001-6188	RPS3	S ribosomal proteins			
7391	-99.8	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
7392	-99.8	kd	CGS001-4942	OAT	-			
7393	-99.8	kd	CGS001-3673	ITGA2	Integrins			
7394	-99.8	kd	CGS001-84433	CARD11	-			
7395	-99.82	oe	ccsbBroad304_00398	CTSL2	-			
7396	-99.82	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
7397	-99.82	kd	CGS001-54925	ZNF434	-			
7398	-99.82	kd	CGS001-390	RND3	-			
7399	-99.82	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
7400	-99.85	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
7401	-99.85	oe	ccsbBroad304_03808	ERGIC1	-			
7402	-99.85	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
7403	-99.87	oe	ccsbBroad304_02533	NOXA1	-			
7404	-99.87	oe	ccsbBroad304_05821	ANXA1	Annexins			
7405	-99.87	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7406	-99.87	kd	CGS001-85004	RERG	-			
7407	-99.87	kd	CGS001-116931	MED12L	-			
7408	-99.87	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
7409	-99.87	kd	CGS001-2056	EPO	Endogenous ligands			
7410	-99.87	kd	CGS001-1452	CSNK1A1	Casein kinase 1 (CK1) family			
7411	-99.87	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
7412	-99.89	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
7413	-99.89	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7414	-99.89	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
7415	-99.89	cp	BRD-A56892734	esomeprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
7416	-99.89	kd	CGS001-143187	VTI1A	-			
7417	-99.89	kd	CGS001-55176	SEC61A2	-			
7418	-99.89	kd	CGS001-23139	MAST2	MAST family			
7419	-99.91	oe	ccsbBroad304_06237	GAA	Glycosidases			
7420	-99.91	oe	ccsbBroad304_00986	MCM2	-			
7421	-99.91	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
7422	-99.91	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
7423	-99.91	kd	CGS001-3958	LGALS3	Endogenous ligands			
7424	-99.93	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
7425	-99.93	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
7426	-99.93	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
7427	-99.93	oe	ccsbBroad304_01347	RAD1	-			
7428	-99.93	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
7429	-99.93	oe	ccsbBroad304_02285	MED6	-			
7430	-99.93	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
7431	-99.93	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
7432	-99.93	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
7433	-99.93	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
7434	-99.93	kd	CGS001-4605	MYBL2	-			
7435	-99.93	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
7436	-99.93	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
7437	-99.93	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
7438	-99.95	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
7439	-99.96	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
7440	-99.96	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
7441	-99.96	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
7442	-99.96	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
7443	-99.96	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
7444	-99.96	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
7445	-99.96	oe	ccsbBroad304_02604	B3GNT1	-			
7446	-99.96	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
7447	-99.96	cp	BRD-K22947005	dexbrompheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
7448	-99.96	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
7449	-99.96	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
7450	-99.96	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
7451	-99.96	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
7452	-99.96	cp	BRD-K15842202	eudesmic-acid	-666			-666
7453	-99.96	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
7454	-99.96	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
7455	-99.96	kd	CGS001-10284	SAP18	-			
7456	-99.96	kd	CGS001-6251	RSU1	-			
7457	-99.96	kd	CGS001-10557	RPP38	-			
7458	-99.96	kd	CGS001-22944	KIN	-			
7459	-99.96	kd	CGS001-23028	KDM1A	Histone demethylase			
7460	-99.96	kd	CGS001-4616	GADD45B	-			
7461	-99.96	kd	CGS001-330	BIRC3	Inhibitors of apoptosis (IAP) protein family			
7462	-99.96	kd	CGS001-598	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7463	-99.96	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
7464	-99.98	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
7465	-99.98	kd	CGS001-5930	RBBP6	-			
7466	-99.98	kd	CGS001-4864	NPC1	-			
7467	-99.98	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
7468	-99.98	kd	CGS001-3895	KTN1	-			
7469	-99.98	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
7470	-100	cc		Ribosomal 40s Subunit LOF	-			
7471	-100	cc		Phospholipases LOF	-			
7472	-100	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
7473	-100	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
7474	-100	kd	CGS001-124626	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7475	-100	kd	CGS001-84527	ZNF559	Zinc fingers, C2H2-type			
7476	-100	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
7477	-100	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
7478	-100	kd	CGS001-7037	TFRC	CD molecules			
7479	-100	kd	CGS001-2030	SLC29A1	SLC29 family			
7480	-100	kd	CGS001-6499	SKIV2L	-			
7481	-100	kd	CGS001-205564	SENP5	-			
7482	-100	kd	CGS001-59343	SENP2	-			
7483	-100	kd	CGS001-6208	RPS14	S ribosomal proteins			
7484	-100	kd	CGS001-6117	RPA1	-			
7485	-100	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
7486	-100	kd	CGS001-10616	RBCK1	RING-type (C3HC4) zinc fingers			
7487	-100	kd	CGS001-5511	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7488	-100	kd	CGS001-5144	PDE4D	Phosphodiesterases			
7489	-100	kd	CGS001-55644	OSGEP	-			
7490	-100	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
7491	-100	kd	CGS001-4751	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
7492	-100	kd	CGS001-10161	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7493	-100	kd	CGS001-3932	LCK	Src family			
7494	-100	kd	CGS001-8942	KYNU	-			
7495	-100	kd	CGS001-3775	KCNK1	Two-P potassium channels			
7496	-100	kd	CGS001-151306	GPBAR1	Bile acid receptor			
7497	-100	kd	CGS001-2244	FGB	Endogenous ligands			
7498	-100	kd	CGS001-10447	FAM3C	-			
7499	-100	kd	CGS001-60528	ELAC2	-			
7500	-100	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
7501	-100	kd	CGS001-55526	DHTKD1	-			
7502	-100	kd	CGS001-56998	CTNNBIP1	Catenins			
7503	-100	kd	CGS001-1213	CLTC	-			
7504	-100	kd	CGS001-790	CAD	-			
7505	-100	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
7506	-100	kd	CGS001-8905	AP1S2	-			
