Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cc		Apolipoproteins LOF	-			
2	100	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
3	100	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
4	100	kd	CGS001-7187	TRAF3	-			
5	100	kd	CGS001-9344	TAOK2	TAO subfamily			
6	100	kd	CGS001-10617	STAMBP	-			
7	100	kd	CGS001-5345	SERPINF2	Serine (or cysteine) peptidase inhibitors			
8	100	kd	CGS001-6253	RTN2	-			
9	100	kd	CGS001-10287	RGS19	Regulators of G-protein signaling			
10	100	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
11	100	kd	CGS001-55163	PNPO	-			
12	100	kd	CGS001-5351	PLOD1	-			
13	100	kd	CGS001-54681	P4HTM	-			
14	100	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
15	100	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
16	100	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
17	100	kd	CGS001-94103	ORMDL3	-			
18	100	kd	CGS001-3225	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
19	100	kd	CGS001-23464	GCAT	-			
20	100	kd	CGS001-53834	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
21	100	kd	CGS001-84288	EFCAB2	EF-hand domain containing			
22	100	kd	CGS001-6387	CXCL12	Endogenous ligands			
23	100	kd	CGS001-23274	CLEC16A	C-type lectin domain containing			
24	100	kd	CGS001-55165	CEP55	-			
25	100	kd	CGS001-55832	CAND1	-			
26	100	kd	CGS001-116519	APOA5	Apolipoproteins			
27	99.98	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
28	99.98	kd	CGS001-118738	ZNF488	Zinc fingers, C2H2-type			
29	99.98	kd	CGS001-10494	STK25	YSK subfamily			
30	99.98	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
31	99.98	kd	CGS001-54442	KCTD5	-			
32	99.98	kd	CGS001-182	JAG1	CD molecules			
33	99.98	kd	CGS001-113878	DTX2	RING-type (C3HC4) zinc fingers			
34	99.98	kd	CGS001-7919	DDX39B	DEAD-boxes			
35	99.98	kd	CGS001-1488	CTBP2	-			
36	99.96	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
37	99.96	oe	ccsbBroad304_01699	TPD52L2	-			
38	99.96	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
39	99.96	oe	ccsbBroad304_02340	SORBS3	-			
40	99.96	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
41	99.96	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
42	99.96	oe	ccsbBroad304_04775	NTAN1	-			
43	99.96	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
44	99.96	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
45	99.96	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
46	99.96	oe	ccsbBroad304_06324	GPX7	-			
47	99.96	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
48	99.96	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
49	99.96	oe	ccsbBroad304_06290	GNA15	-			
50	99.96	oe	ccsbBroad304_02270	FAM20B	-			
51	99.96	oe	ccsbBroad304_03640	CEP72	-			
52	99.96	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
53	99.96	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
54	99.96	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
55	99.96	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
56	99.96	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
57	99.96	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
58	99.96	cp	BRD-K44094599	tacrolimus	Calcineurin inhibitor		FKBP1A, CYP3A5, CYP3A7	Calcineurin inhibitor
59	99.96	cp	BRD-K89708791	rifaximin	RNA synthesis inhibitor		NR1I2, CYP3A4	RNA synthesis inhibitor
60	99.96	cp	BRD-K23369905	oxiconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
61	99.96	cp	BRD-K32311154	nifekalant	Potassium channel blocker			Potassium channel blocker
62	99.96	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
63	99.96	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
64	99.96	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
65	99.96	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
66	99.96	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
67	99.96	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
68	99.96	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
69	99.96	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
70	99.96	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
71	99.96	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
72	99.96	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
73	99.96	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
74	99.96	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
75	99.96	kd	CGS001-6513	SLC2A1	Solute carriers			
76	99.96	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
77	99.96	kd	CGS001-4817	NIT1	-			
78	99.96	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
79	99.93	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
80	99.93	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
81	99.93	oe	ccsbBroad304_01560	SNAPC1	-			
82	99.93	oe	ccsbBroad304_02668	PNKP	-			
83	99.93	oe	ccsbBroad304_05038	HORMAD2	-			
84	99.93	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
85	99.93	cp	BRD-K37516142	idebenone	Calcium channel modulator			Calcium channel modulator
86	99.93	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
87	99.93	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
88	99.93	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
89	99.93	kd	CGS001-3459	IFNGR1	Interferon receptor family			
90	99.93	kd	CGS001-25793	FBXO7	F-boxes / other			
91	99.91	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
92	99.91	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
93	99.91	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
94	99.91	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
95	99.91	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
96	99.91	kd	CGS001-5695	PSMB7	Proteasome subunits			
97	99.91	kd	CGS001-440387	CTRB2	-			
98	99.91	kd	CGS001-348	APOE	Apolipoproteins			
99	99.91	kd	CGS001-308	ANXA5	Annexins			
100	99.91	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
101	99.89	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
102	99.89	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
103	99.89	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
104	99.89	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
105	99.89	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
106	99.89	kd	CGS001-54386	TERF2IP	-			
107	99.89	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
108	99.87	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
109	99.87	oe	ccsbBroad304_00783	HPRT1	-			
110	99.87	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
111	99.87	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
112	99.87	cp	BRD-K00532621	midazolam	Benzodiazepine receptor agonist		CYP3A5, CYP3A7, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3	Benzodiazepine receptor agonist
113	99.87	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
114	99.87	kd	CGS001-7105	TSPAN6	Tetraspanins			
115	99.87	kd	CGS001-8463	TEAD2	-			
116	99.87	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
117	99.87	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
118	99.87	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
119	99.87	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
120	99.87	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
121	99.85	oe	ccsbBroad304_01371	RALA	-			
122	99.85	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
123	99.85	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
124	99.85	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
125	99.85	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
126	99.85	oe	ccsbBroad304_02553	BLCAP	-			
127	99.85	cp	BRD-K10961822	latanoprost	Prostanoid receptor agonist		PTGFR	Prostanoid receptor agonist
128	99.85	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
129	99.85	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
130	99.85	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
131	99.85	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
132	99.85	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
133	99.85	kd	CGS001-11168	PSIP1	-			
134	99.85	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
135	99.85	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
136	99.82	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
137	99.82	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
138	99.82	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
139	99.82	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
140	99.82	kd	CGS001-4245	MGAT1	-			
141	99.81	oe	ccsbBroad304_02115	PTTG1	-			
142	99.81	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
143	99.8	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
144	99.8	kd	CGS001-333929	SNAI3	Snail homologs			
145	99.8	kd	CGS001-8650	NUMB	-			
146	99.8	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
147	99.8	kd	CGS001-717	C2	Complement system			
148	99.8	kd	CGS001-644	BLVRA	-			
149	99.78	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
150	99.78	oe	ccsbBroad304_00072	ANXA7	Annexins			
151	99.78	kd	CGS001-9958	USP15	Ubiquitin-specific peptidases			
152	99.78	kd	CGS001-9200	PTPLA	-			
153	99.76	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
154	99.76	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
155	99.76	kd	CGS001-5575	PRKAR1B	Protein kinase A			
156	99.75	kd	CGS001-7358	UGDH	-			
157	99.74	cc		Targets of VEGFR inhibitors GOF	-			
158	99.74	cc		Proteasome Pathway LOF	-			
159	99.74	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
160	99.74	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
161	99.74	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
162	99.74	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
163	99.72	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
164	99.72	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
165	99.72	kd	CGS001-55634	ZNF673	-			
166	99.72	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
167	99.72	kd	CGS001-4953	ODC1	Decarboxylases			
168	99.72	kd	CGS001-2782	GNB1	WD repeat domain containing			
169	99.7	kd	CGS001-2678	GGT1	CD molecules			
170	99.69	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
171	99.69	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
172	99.69	kd	CGS001-3170	FOXA2	Forkhead boxes			
173	99.69	kd	CGS001-10632	ATP5L	ATPases / F-type			
174	99.66	kd	CGS001-8438	RAD54L	-			
175	99.66	kd	CGS001-10014	HDAC5	Histone deacetylases			
176	99.65	oe	ccsbBroad304_01186	PHB	-			
177	99.65	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
178	99.65	kd	CGS001-5707	PSMD1	Proteasome subunits			
179	99.65	kd	CGS001-571	BACH1	BTB/POZ domain containing			
180	99.64	kd	CGS001-439	ASNA1	-			
181	99.63	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
182	99.63	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
183	99.63	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
184	99.63	kd	CGS001-8692	HYAL2	-			
185	99.63	kd	CGS001-2664	GDI1	-			
186	99.61	cc		Protein phosphatase catalytic subunits LOF	-			
187	99.61	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
188	99.61	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
189	99.61	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
190	99.61	kd	CGS001-9797	TATDN2	-			
191	99.61	kd	CGS001-6304	SATB1	Homeoboxes / CUT class			
192	99.61	kd	CGS001-3397	ID1	Basic helix-loop-helix proteins			
193	99.61	kd	CGS001-843	CASP10	Caspases			
194	99.58	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
195	99.58	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
196	99.58	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
197	99.58	kd	CGS001-6009	RHEB	-			
198	99.58	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
199	99.57	kd	CGS001-2356	FPGS	-			
200	99.56	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
201	99.56	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
202	99.54	oe	ccsbBroad304_01327	PSPH	-			
203	99.54	kd	CGS001-5654	HTRA1	Serine peptidases / Serine peptidases			
204	99.52	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
205	99.5	cp	BRD-A24381660	zeranol	Estrogen receptor agonist			Estrogen receptor agonist
206	99.5	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
207	99.5	kd	CGS001-7165	TPD52L2	-			
208	99.5	kd	CGS001-8435	SOAT2	-			
209	99.5	kd	CGS001-5997	RGS2	Endogenous ligands			
210	99.49	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
211	99.47	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
212	99.47	kd	CGS001-10460	TACC3	-			
213	99.47	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
214	99.47	oe	ccsbBroad304_01974	RNASET2	-			
215	99.47	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
216	99.45	oe	ccsbBroad304_02446	TADA3	-			
217	99.45	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
218	99.45	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
219	99.44	oe	ccsbBroad304_03155	DHH	-			
220	99.43	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
221	99.41	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
222	99.41	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
223	99.37	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
224	99.35	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
225	99.34	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
226	99.34	cp	BRD-K94887716	TFMPP	Serotonin receptor agonist			Serotonin receptor agonist, Serotonin receptor antagonist
227	99.34	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
228	99.34	kd	CGS001-10237	SLC35B1	SLC35 family of nucleotide sugar transporters			
229	99.34	kd	CGS001-3572	IL6ST	IL-6 receptor family			
230	99.33	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
231	99.32	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
232	99.3	kd	CGS001-5693	PSMB5	Proteasome subunits			
233	99.29	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
234	99.27	oe	ccsbBroad304_07053	TFPI	-			
235	99.26	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
236	99.26	kd	CGS001-2115	ETV1	ETS Transcription Factors			
237	99.23	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
238	99.23	kd	CGS001-211	ALAS1	-			
239	99.22	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
240	99.21	oe	ccsbBroad304_04038	ELOVL6	-			
241	99.21	kd	CGS001-23369	PUM2	-			
242	99.2	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
243	99.19	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
244	99.19	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
245	99.15	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
246	99.15	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
247	99.15	kd	CGS001-80714	PBX4	Homeoboxes / TALE class			
248	99.15	kd	CGS001-3486	IGFBP3	insulin-like growth factor (IGF) binding proteins			
249	99.15	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
250	99.14	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
251	99.12	kd	CGS001-56675	NRIP3	-			
252	99.12	kd	CGS001-9813	KIAA0494	-			
253	99.12	kd	CGS001-11164	NUDT5	Nudix motif containing			
254	99.1	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
255	99.09	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
256	99.08	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
257	99.08	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
258	99.06	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
259	99.06	oe	ccsbBroad304_00469	DUT	-			
260	99.06	kd	CGS001-147686	ZNF418	Zinc fingers, C2H2-type			
261	99.05	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
262	99.05	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
263	99.05	kd	CGS001-342926	ZNF677	Zinc fingers, C2H2-type			
264	99.04	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
265	99.04	kd	CGS001-1499	CTNNB1	Catenins			
266	99.03	cc		Retinoid receptor agonist	-			
267	99.03	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
268	99.03	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
269	99.02	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
270	99.02	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
271	99.01	cp	BRD-A70083328	secnidazole	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Microtubule inhibitor, Antiprotozoal
272	98.97	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
273	98.97	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
274	98.96	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
275	98.95	oe	ccsbBroad304_10846	GGT1	CD molecules			
276	98.95	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
277	98.94	kd	CGS001-6832	SUPV3L1	-			
278	98.93	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
279	98.93	oe	ccsbBroad304_03874	UBL5	-			
280	98.93	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
281	98.93	oe	ccsbBroad304_03641	ASF1B	-			
282	98.93	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
283	98.93	kd	CGS001-5091	PC	Carboxylases			
284	98.93	kd	CGS001-2882	GPX7	-			
285	98.93	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
286	98.92	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
287	98.91	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
288	98.91	kd	CGS001-5018	OXA1L	-			
289	98.91	kd	CGS001-30836	DNTTIP2	-			
290	98.9	kd	CGS001-4758	NEU1	-			
291	98.88	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
292	98.85	kd	CGS001-23314	SATB2	Homeoboxes / CUT class			
293	98.84	oe	ccsbBroad304_03037	TMEM97	-			
294	98.84	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
295	98.83	cp	BRD-K60160658	tiagabine	GABA uptake inhibitor		SLC6A1, CYP2C19	GABA uptake inhibitor
296	98.82	oe	ccsbBroad304_04675	ATG4A	-			
297	98.82	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
298	98.82	kd	CGS001-191	AHCY	Adenosine turnover			
299	98.8	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
300	98.78	oe	ccsbBroad304_07374	PTPLA	-			
301	98.77	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
302	98.77	kd	CGS001-11073	TOPBP1	-			
303	98.75	oe	ccsbBroad304_03118	NRBP1	NRBP family			
304	98.75	oe	ccsbBroad304_03591	ETNK1	-			
305	98.75	kd	CGS001-51172	NAGPA	-			
306	98.71	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
307	98.7	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
308	98.69	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
309	98.67	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
310	98.67	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
311	98.67	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
312	98.66	kd	CGS001-6491	STIL	-			
313	98.65	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
314	98.65	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
315	98.64	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
316	98.64	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
317	98.64	kd	CGS001-8974	P4HA2	-			
318	98.62	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
319	98.62	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
320	98.62	kd	CGS001-51014	TMED7	-			
321	98.62	kd	CGS001-10180	RBM6	G patch domain containing			
322	98.6	kd	CGS001-5684	PSMA3	Proteasome subunits			
323	98.58	oe	ccsbBroad304_03980	DCLRE1B	-			
324	98.58	kd	CGS001-10010	TANK	-			
325	98.57	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
326	98.56	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
327	98.56	kd	CGS001-84811	BUD13	-			
328	98.53	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
329	98.53	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
330	98.52	kd	CGS001-51495	PTPLAD1	-			
331	98.51	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
332	98.5	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
333	98.47	kd	CGS001-7295	TXN	-			
334	98.45	kd	CGS001-1022	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
335	98.43	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
336	98.41	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
337	98.37	kd	CGS001-5688	PSMA7	Proteasome subunits			
338	98.36	kd	CGS001-7004	TEAD4	-			
339	98.36	kd	CGS001-3053	SERPIND1	Serine (or cysteine) peptidase inhibitors			
340	98.35	cp	BRD-A52282606	lacidipine	Calcium channel blocker		CACNA1C	Calcium channel blocker
341	98.34	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
342	98.32	kd	CGS001-6652	SORD	-			
343	98.32	kd	CGS001-183	AGT	Endogenous ligands			
344	98.32	kd	CGS001-9451	EIF2AK3	PEK subfamily			
345	98.31	oe	ccsbBroad304_00962	SMAD4	SMADs			
346	98.31	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
347	98.3	kd	CGS001-238	ALK	Leukocyte tyrosine kinase (LTK) receptor family			
348	98.29	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
349	98.29	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
350	98.27	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
351	98.26	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
352	98.25	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
353	98.24	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
354	98.23	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
355	98.23	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
356	98.23	kd	CGS001-54566	EPB41L4B	-			
357	98.23	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
358	98.21	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
359	98.21	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
360	98.2	kd	CGS001-3978	LIG1	-			
361	98.18	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
362	98.18	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
363	98.18	kd	CGS001-11112	HIBADH	-			
364	98.16	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
365	98.15	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
366	98.11	kd	CGS001-54821	ERCC6L	-			
367	98.1	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
368	98.09	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
369	98.08	oe	ccsbBroad304_05194	LIPH	-			
370	98.05	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
371	98.04	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
372	98.04	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
373	98.01	kd	CGS001-808	CALM3	EF-hand domain containing			
374	98	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
375	97.96	oe	ccsbBroad304_08596	EAPP	-			
376	97.94	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
377	97.94	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
378	97.94	kd	CGS001-5910	RAP1GDS1	Armadillo repeat containing			
379	97.93	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
380	97.92	kd	CGS001-5198	PFAS	-			
381	97.91	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
382	97.9	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
383	97.88	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
384	97.88	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
385	97.87	kd	CGS001-344	APOC2	Apolipoproteins			
386	97.86	oe	ccsbBroad304_03533	CDCA8	-			
387	97.86	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
388	97.86	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
389	97.85	kd	CGS001-7157	TP53	-			
390	97.85	kd	CGS001-10468	FST	-			
391	97.84	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
392	97.84	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
393	97.83	kd	CGS001-4893	NRAS	RAS subfamily			
394	97.82	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
395	97.81	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
396	97.81	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
397	97.81	kd	CGS001-5328	PLAU	Chymotrypsin			
398	97.8	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
399	97.8	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
400	97.78	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
401	97.77	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
402	97.77	kd	CGS001-5595	MAPK3	MAPK:ERK subfamily			
403	97.74	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
404	97.71	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
405	97.7	kd	CGS001-84969	TOX2	-			
406	97.7	kd	CGS001-7292	TNFSF4	CD molecules			
407	97.68	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
408	97.68	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
409	97.68	kd	CGS001-84619	ZGPAT	G patch domain containing			
410	97.68	kd	CGS001-9455	HOMER2	-			
411	97.66	kd	CGS001-11015	KDELR3	-			
412	97.65	oe	ccsbBroad304_08023	EIF2C1	-			
413	97.64	oe	ccsbBroad304_00941	LIG3	-			
414	97.64	kd	CGS001-8467	SMARCA5	-			
415	97.63	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
416	97.62	kd	CGS001-8508	NIPSNAP1	-			
417	97.6	kd	CGS001-4976	OPA1	-			
418	97.58	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
419	97.57	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
420	97.57	cp	BRD-K37798499	etoposide	Topoisomerase inhibitor		TOP2A, CYP2E1, CYP3A5, TOP2B	Topoisomerase inhibitor
421	97.56	kd	CGS001-22921	MSRB2	-			
422	97.55	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
423	97.54	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
424	97.52	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
425	97.5	kd	CGS001-6519	SLC3A1	SLC3 family			
426	97.49	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
427	97.48	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
428	97.46	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
429	97.41	kd	CGS001-6812	STXBP1	-			
430	97.38	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
431	97.36	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
432	97.36	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
433	97.35	kd	CGS001-11214	AKAP13	A-kinase anchor proteins			
434	97.33	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
435	97.33	oe	ccsbBroad304_02862	CCRN4L	-			
436	97.33	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
437	97.3	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
438	97.3	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
439	97.29	oe	ccsbBroad304_07197	PDHX	-			
440	97.29	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
441	97.28	kd	CGS001-375318	AQP12A	Ion channels / Aquaporins			
442	97.27	oe	ccsbBroad304_08093	DCPS	-			
443	97.23	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
444	97.21	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
445	97.2	kd	CGS001-90861	HN1L	-			
446	97.16	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
447	97.14	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
448	97.13	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
449	97.1	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
450	97.09	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
451	97.09	kd	CGS001-51027	BOLA1	-			
452	97.08	oe	ccsbBroad304_03121	NRBF2	-			
453	97.08	kd	CGS001-1906	EDN1	Endogenous ligands			
454	97.08	kd	CGS001-539	ATP5O	ATPases / F-type			
455	97.06	kd	CGS001-1457	CSNK2A1	Casein kinase 2 (CK2) family			
456	97.05	kd	CGS001-2243	FGA	Endogenous ligands			
457	97.04	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
458	97.03	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
459	97.03	kd	CGS001-4482	MSRA	-			
460	96.99	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
461	96.98	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
462	96.97	oe	ccsbBroad304_02964	TIMM9	-			
463	96.97	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
464	96.96	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
465	96.94	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
466	96.94	kd	CGS001-23509	POFUT1	Fucosyltransferases			
467	96.92	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
468	96.86	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
469	96.85	cc		DNA polymerase inhibitor	-			
470	96.85	kd	CGS001-2004	ELK3	ETS Transcription Factors			
471	96.84	kd	CGS001-9807	IP6K1	-			
472	96.76	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
473	96.76	kd	CGS001-10972	TMED10	-			
474	96.75	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
475	96.74	oe	ccsbBroad304_06671	OPA1	-			
476	96.72	cc		Tumor necrosis factor superfamily LOF	-			
477	96.7	kd	CGS001-2550	GABBR1	GABA receptors			
478	96.69	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
479	96.68	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
480	96.66	oe	ccsbBroad304_02526	POP4	-			
481	96.61	kd	CGS001-5810	RAD1	-			
482	96.61	kd	CGS001-1962	EHHADH	-			
483	96.61	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
484	96.6	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
485	96.6	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
486	96.59	oe	ccsbBroad304_00150	BAX	-			
487	96.57	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
488	96.55	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
489	96.53	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
490	96.51	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
491	96.5	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
492	96.5	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
493	96.49	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
494	96.49	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
495	96.49	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
496	96.45	oe	ccsbBroad304_03696	C19ORF10	-			
497	96.44	kd	CGS001-1386	ATF2	basic leucine zipper proteins			
498	96.43	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
499	96.38	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
500	96.37	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
501	96.37	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
502	96.32	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
503	96.29	kd	CGS001-84878	ZBTB45	BTB/POZ domain containing			
504	96.28	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
505	96.28	kd	CGS001-8870	IER3	-			
506	96.27	kd	CGS001-2260	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
507	96.25	oe	ccsbBroad304_08839	IFIH1	-			
508	96.25	kd	CGS001-8503	PIK3R3	Phosphatidylinositol kinases			
509	96.24	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
510	96.23	oe	ccsbBroad304_05907	BUB1B	Bub family			
511	96.2	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
512	96.15	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
513	96.14	kd	CGS001-8480	RAE1	WD repeat domain containing			
514	96.13	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
515	96.05	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
516	96.04	kd	CGS001-7001	PRDX2	-			
517	96.01	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
518	96.01	kd	CGS001-55781	RIOK2	RIO2 subfamily			
519	96	kd	CGS001-6601	SMARCC2	-			
520	96	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
521	95.98	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
522	95.94	oe	ccsbBroad304_06235	G6PD	-			
523	95.9	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
524	95.85	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
525	95.83	oe	ccsbBroad304_01066	NDUFA4	-			
526	95.83	kd	CGS001-23636	NUP62	-			
527	95.82	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
528	95.82	cp	BRD-A48261811	argatroban	Thrombin inhibitor		F2, CYP3A5	Thrombin inhibitor
529	95.82	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
530	95.82	kd	CGS001-2961	GTF2E2	General transcription factors			
531	95.81	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
532	95.8	oe	ccsbBroad304_00883	ISG20	-			
533	95.8	kd	CGS001-221895	JAZF1	Zinc fingers, C2H2-type			
534	95.77	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
535	95.75	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
536	95.72	kd	CGS001-89766	UMODL1	-			
537	95.71	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
538	95.71	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
539	95.71	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
540	95.69	oe	ccsbBroad304_02402	TMEM5	-			
541	95.69	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
542	95.67	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
543	95.65	oe	ccsbBroad304_07920	NUP62	-			
544	95.64	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
545	95.62	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
546	95.62	kd	CGS001-2869	GRK5	GRK1/3 subfamily			
547	95.6	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
548	95.59	kd	CGS001-51465	UBE2J1	Ubiquitin-conjugating enzymes E2			
549	95.54	kd	CGS001-5985	RFC5	ATPases / AAA-type			
550	95.53	cp	BRD-K51730347	diphencyprone	Immunostimulant			Immunostimulant
551	95.51	oe	ccsbBroad304_02581	ASCC3	-			
552	95.51	kd	CGS001-11319	ECD	-			
553	95.49	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
554	95.48	kd	CGS001-81533	ITFG1	-			
555	95.47	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
556	95.45	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
557	95.45	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
558	95.44	oe	ccsbBroad304_03773	CIAPIN1	-			
559	95.41	kd	CGS001-8553	BHLHE40	Basic helix-loop-helix proteins			
560	95.41	kd	CGS001-2	A2M	-			
561	95.36	kd	CGS001-677	ZFP36L1	RING-type (C3HC4) zinc fingers			
562	95.36	kd	CGS001-6196	RPS6KA2	RSK subfamily			
563	95.33	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
564	95.32	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
565	95.31	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
566	95.29	kd	CGS001-3460	IFNGR2	Interferon receptor family			
567	95.21	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
568	95.2	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
569	95.16	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
570	95.16	kd	CGS001-2264	FGFR4	Type V RTKs: FGF (fibroblast growth factor) receptor family			
571	95.13	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
572	95.12	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
573	95.1	cp	BRD-K32744045	disulfiram	Aldehyde dehydrogenase inhibitor		ALDH2, ALDH1A2, ALDH5A1, ALDH7A1, CYP2E1, DBH, DNMT1, TRPA1	Aldehyde dehydrogenase inhibitor, TRPV agonist, DNA methyltransferase inhibitor
574	95.09	kd	CGS001-2230	FDX1	-			
575	95.05	kd	CGS001-6934	TCF7L2	-			
576	95.04	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
577	95.02	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
578	94.98	kd	CGS001-39	ACAT2	Lanosterol biosynthesis pathway			
579	94.92	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
580	94.91	kd	CGS001-22949	PTGR1	-			
581	94.9	kd	CGS001-11182	SLC2A6	Solute carriers			
582	94.89	kd	CGS001-63874	ABHD4	Abhydrolase domain containing			
583	94.87	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
584	94.86	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
585	94.78	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
586	94.77	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
587	94.77	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
588	94.76	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
589	94.75	kd	CGS001-3708	ITPR1	Ion channels / Inositol triphosphate receptors			
590	94.74	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
591	94.72	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
592	94.71	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
593	94.68	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
594	94.67	cc		Benzodiazepine receptor agonist	-			
595	94.64	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
596	94.6	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
597	94.59	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
598	94.58	oe	ccsbBroad304_00221	CASP3	Caspases			
599	94.58	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
600	94.45	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
601	94.44	kd	CGS001-85480	TSLP	-			
602	94.43	kd	CGS001-54555	DDX49	DEAD-boxes			
603	94.43	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
604	94.39	kd	CGS001-3856	KRT8	Intermediate filaments type II, keratins (basic)			
605	94.38	kd	CGS001-3033	HADH	-			
606	94.38	kd	CGS001-1152	CKB	-			
607	94.34	oe	ccsbBroad304_05980	CDKN1B	-			
608	94.34	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
609	94.33	oe	ccsbBroad304_07080	TM7SF2	-			
610	94.32	kd	CGS001-5682	PSMA1	Proteasome subunits			
611	94.31	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
612	94.3	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
613	94.26	cc		DNA synthesis inhibitor	-			
614	94.24	kd	CGS001-9221	NOLC1	-			
615	94.23	kd	CGS001-7444	VRK2	Vaccina related kinase (VRK) family			
616	94.23	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
617	94.2	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
618	94.2	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
619	94.15	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
620	94.14	oe	ccsbBroad304_02554	TRAFD1	-			
621	94.09	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
622	94.05	kd	CGS001-1950	EGF	-			
623	94	cc		Cannabinoid receptor agonist	-			
624	93.9	kd	CGS001-7013	TERF1	-			
625	93.86	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
626	93.86	kd	CGS001-9784	SNX17	Sorting nexins			
627	93.82	kd	CGS001-10587	TXNRD2	-			
628	93.8	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
629	93.74	kd	CGS001-641	BLM	-			
630	93.72	oe	ccsbBroad304_09195	MCM8	-			
631	93.71	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
632	93.69	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
633	93.67	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
634	93.63	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
635	93.57	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
636	93.51	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
637	93.49	oe	ccsbBroad304_02484	PAICS	-			
638	93.49	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
639	93.48	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
640	93.46	kd	CGS001-54811	ZNF562	Zinc fingers, C2H2-type			
641	93.45	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
642	93.43	oe	ccsbBroad304_01054	GADD45B	-			
643	93.43	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
644	93.42	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
645	93.42	kd	CGS001-478	ATP1A3	ATPases / P-type			
646	93.4	cp	BRD-A16934955	nalbuphine	Opioid receptor agonist		OPRD1, OPRK1, OPRM1	Opioid receptor agonist, Opioid receptor antagonist
647	93.4	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
648	93.35	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
649	93.35	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
650	93.34	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
651	93.33	oe	ccsbBroad304_02890	SYF2	-			
652	93.33	kd	CGS001-50846	DHH	-			
653	93.32	oe	ccsbBroad304_00515	ERH	-			
654	93.32	kd	CGS001-83743	GRWD1	WD repeat domain containing			
655	93.29	oe	ccsbBroad304_02576	MLLT11	-			
656	93.28	oe	ccsbBroad304_06845	RARRES3	-			
657	93.28	kd	CGS001-2821	GPI	-			
658	93.25	kd	CGS001-821	CANX	-			
659	93.24	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
660	93.24	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
661	93.23	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
662	93.23	cp	BRD-K90733503	cefalexin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
663	93.22	cc		Ubiquitin-specific peptidases LOF	-			
664	93.22	kd	CGS001-64750	SMURF2	-			
665	93.06	kd	CGS001-11340	EXOSC8	-			
666	93.01	kd	CGS001-9014	TAF1B	-			
667	92.96	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
668	92.94	kd	CGS001-8027	STAM	-			
669	92.87	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
670	92.87	kd	CGS001-79143	MBOAT7	-			
671	92.86	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
672	92.83	kd	CGS001-5498	PPOX	-			
673	92.81	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
674	92.74	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
675	92.7	kd	CGS001-9788	MTSS1	-			
676	92.67	kd	CGS001-55120	FANCL	Fanconi anemia, complementation groups			
677	92.67	kd	CGS001-115	ADCY9	Adenylyl cyclases			
678	92.66	kd	CGS001-3482	IGF2R	CD molecules			
679	92.62	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
680	92.61	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
681	92.59	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
682	92.59	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
683	92.57	oe	ccsbBroad304_04490	RSPH1	-			
684	92.57	oe	ccsbBroad304_07724	KDELR2	-			
685	92.57	kd	CGS001-6364	CCL20	Chemokine ligands			
686	92.56	kd	CGS001-51001	MTERFD1	-			
687	92.52	kd	CGS001-8834	TMEM11	-			
688	92.48	kd	CGS001-286380	FOXD4L3	-			
689	92.47	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
690	92.47	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
691	92.42	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
692	92.38	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
693	92.38	kd	CGS001-2786	GNG4	-			
694	92.34	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
695	92.34	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
696	92.3	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
697	92.26	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
698	92.23	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
699	92.23	kd	CGS001-2837	UTS2R	Urotensin receptor			
700	92.2	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
701	92.18	oe	ccsbBroad304_06008	AP2M1	-			
702	92.16	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
703	92.15	kd	CGS001-1209	CLPTM1	-			
704	92.11	kd	CGS001-22794	CASC3	-			
705	92.08	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
706	92.06	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
707	92.02	oe	ccsbBroad304_00462	DR1	-			
708	91.98	oe	ccsbBroad304_07280	LAMTOR3	-			
709	91.97	oe	ccsbBroad304_07128	VHL	-			
710	91.97	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
711	91.94	kd	CGS001-7025	NR2F1	COUP-TF-like receptors			
712	91.93	kd	CGS001-6813	STXBP2	-			
713	91.91	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
714	91.89	oe	ccsbBroad304_02596	KDELR3	-			
715	91.88	cc		Cell Cycle Inhibition GOF	-			
716	91.84	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
717	91.84	kd	CGS001-4299	AFF1	-			
718	91.83	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
719	91.83	kd	CGS001-51128	SAR1B	-			
720	91.83	kd	CGS001-10901	DHRS4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
721	91.78	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
722	91.77	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
723	91.75	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
724	91.73	kd	CGS001-23102	TBC1D2B	-			
725	91.71	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
726	91.7	kd	CGS001-51466	EVL	-			
727	91.63	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
728	91.6	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
729	91.54	kd	CGS001-7727	ZNF174	Zinc fingers, C2H2-type			
730	91.54	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
731	91.52	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
732	91.49	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
733	91.43	kd	CGS001-29998	GLTSCR1	-			
734	91.38	kd	CGS001-51720	UIMC1	-			
735	91.33	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
736	91.32	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
737	91.32	kd	CGS001-5743	PTGS2	Cyclooxygenase			
738	91.31	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
739	91.31	kd	CGS001-84875	PARP10	Poly (ADP-ribose) polymerases			
740	91.3	kd	CGS001-1515	CTSL2	-			
741	91.25	kd	CGS001-4905	NSF	ATPases / AAA-type			
742	91.23	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
743	91.2	kd	CGS001-80237	ELL3	-			
744	91.18	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
745	91.17	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
746	91.12	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
747	91.12	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
748	91.04	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
749	90.95	oe	ccsbBroad304_06066	CTSL1	-			
750	90.95	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
751	90.94	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
752	90.88	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
753	90.87	kd	CGS001-2956	MSH6	-			
754	90.81	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
755	90.77	kd	CGS001-2280	FKBP1A	Cis-trans-isomerases			
756	90.7	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
757	90.68	oe	ccsbBroad304_00239	CCNG1	-			
758	90.67	cp	BRD-K15916496	clotrimazole	Cytochrome P450 inhibitor		KCNN4, CYP3A4, CYP51A1, NR1I2, NR1I3, TRPM2, TRPM4, TRPM8	Cytochrome P450 inhibitor, Imidazoline receptor ligand
759	90.64	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
760	90.63	oe	ccsbBroad304_01208	PITPNA	-			
761	90.61	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
762	90.61	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
763	90.6	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
764	90.49	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
765	90.46	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
766	90.39	oe	ccsbBroad304_00572	FKBP3	-			
767	90.38	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
768	90.38	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
769	90.37	kd	CGS001-121549	ASCL4	Basic helix-loop-helix proteins			
770	90.33	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
771	90.33	kd	CGS001-9854	C2CD2L	-			
772	90.25	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
773	90.25	kd	CGS001-944	TNFSF8	CD molecules			
774	90.16	kd	CGS001-6713	SQLE	Lanosterol biosynthesis pathway			
775	90.15	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
776	90.1	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
777	90.09	kd	CGS001-54851	ANKRD49	Ankyrin repeat domain containing			
778	90.07	kd	CGS001-2149	F2R	Protease activated receptors			
779	90.03	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
780	90	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
781	89.99	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
782	89.95	cp	BRD-K50938287	sumatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1A, HTR1F, HTR1E, HTR5A, HTR6, HTR7	Serotonin receptor agonist
783	89.91	oe	ccsbBroad304_10230	STK19	G11 family			
784	89.85	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
785	89.78	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
786	89.77	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
787	89.77	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
788	89.74	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
789	89.68	oe	ccsbBroad304_02298	DNM1L	-			
790	89.68	kd	CGS001-54498	SMOX	-			
791	89.65	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
792	89.61	kd	CGS001-8050	PDHX	-			
793	89.58	kd	CGS001-2159	F10	Chymotrypsin			
794	89.57	oe	ccsbBroad304_06095	DFFB	-			
795	89.55	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
796	89.51	cp	BRD-K81916719	triclabendazole	Microtubule inhibitor		DNMT1	Microtubule inhibitor
797	89.46	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
798	89.46	kd	CGS001-51375	SNX7	Sorting nexins			
799	89.44	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
800	89.43	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
801	89.41	kd	CGS001-26086	GPSM1	Tetratricopeptide (TTC) repeat domain containing			
802	89.39	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
803	89.35	kd	CGS001-3269	HRH1	Histamine receptors			
804	89.33	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
805	89.31	kd	CGS001-10975	UQCR11	Mitochondrial respiratory chain complex / Complex III			
806	89.28	kd	CGS001-3995	FADS3	Fatty acid desaturases			
807	89.26	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
808	89.23	kd	CGS001-435	ASL	-			
809	89.15	kd	CGS001-3659	IRF1	-			
810	89.14	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
811	89.11	kd	CGS001-58477	SRPRB	-			
812	89.07	kd	CGS001-5618	PRLR	Prolactin receptor family			
813	89.06	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
814	89.05	oe	ccsbBroad304_08104	MED4	-			
815	89.02	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
816	89.02	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
817	89.01	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
818	89.01	kd	CGS001-1650	DDOST	-			
819	88.99	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
820	88.99	kd	CGS001-54957	TXNL4B	-			
821	88.96	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
822	88.95	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
823	88.94	kd	CGS001-9354	UBE4A	U-box domain containing			
824	88.92	kd	CGS001-8807	IL18RAP	CD molecules			
825	88.91	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
826	88.91	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
827	88.88	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
828	88.85	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
829	88.79	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
830	88.79	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
831	88.78	oe	ccsbBroad304_02443	HAX1	-			
832	88.77	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
833	88.76	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
834	88.69	cc		Thymidylate synthase inhibitor	-			
835	88.68	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
836	88.49	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
837	88.47	oe	ccsbBroad304_05152	SSBP4	-			
838	88.42	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
839	88.39	oe	ccsbBroad304_01139	PA2G4	-			
840	88.39	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
841	88.38	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
842	88.38	kd	CGS001-7181	NR2C1	Testicular receptors			
843	88.34	kd	CGS001-253260	RICTOR	-			
844	88.32	kd	CGS001-9767	PHF16	-			
845	88.3	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
846	88.29	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
847	88.24	kd	CGS001-5253	PHF2	Histone demethylases			
848	88.19	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
849	88.17	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
850	88.12	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
851	88.12	kd	CGS001-9703	KIAA0100	-			
852	88.11	kd	CGS001-7316	UBC	-			
853	88.07	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
854	88	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
855	87.98	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
856	87.94	kd	CGS001-1841	DTYMK	-			
857	87.92	cc		NFKB Activation GOF	-			
858	87.81	cp	BRD-K04196797	oxcarbazepine	Sodium channel blocker		CYP2C19, CYP3A4, CYP3A5, SCN1A, SCN3A, SCN5A	Sodium channel blocker
859	87.79	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
860	87.78	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
861	87.73	kd	CGS001-54732	TMED9	-			
862	87.68	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
863	87.67	cc		IMPDH inhibitor	-			
864	87.66	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
865	87.65	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
866	87.63	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
867	87.61	kd	CGS001-23	ABCF1	ATP binding cassette transporters / subfamily F			
868	87.61	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
869	87.56	kd	CGS001-3242	HPD	Oxidoreductases			
870	87.54	kd	CGS001-5883	RAD9A	-			
871	87.54	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
872	87.53	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
873	87.52	kd	CGS001-83694	RPS6KL1	RSKL family			
874	87.52	kd	CGS001-1284	COL4A2	Collagens			
875	87.47	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
876	87.46	kd	CGS001-53347	UBASH3A	-			
877	87.46	kd	CGS001-2254	FGF9	Endogenous ligands			
878	87.45	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
879	87.38	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
880	87.38	kd	CGS001-10513	APPBP2	-			
881	87.36	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
882	87.32	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
883	87.24	kd	CGS001-9632	SEC24C	-			
884	87.21	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
885	87.19	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
886	87.17	kd	CGS001-4947	OAZ2	-			
887	87.14	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
888	87.13	oe	ccsbBroad304_01002	METTL1	-			
889	87.11	oe	ccsbBroad304_00225	CAT	-			
890	87.09	kd	CGS001-1468	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
891	87.09	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
892	87.09	kd	CGS001-873	CBR1	Prostaglandin synthases			
893	87.06	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
894	87.04	kd	CGS001-55206	SBNO1	-			
895	86.93	oe	ccsbBroad304_06789	PSEN2	Presenilin			
896	86.86	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
897	86.83	kd	CGS001-7251	TSG101	-			
898	86.79	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
899	86.78	cc		LIM class homeoboxes GOF	-			
900	86.78	kd	CGS001-9833	MELK	MELK subfamily			
901	86.75	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
902	86.67	kd	CGS001-4331	MNAT1	RING-type (C3HC4) zinc fingers			
903	86.53	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
904	86.51	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
905	86.49	oe	ccsbBroad304_00282	CDKN1A	-			
906	86.49	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
907	86.43	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
908	86.31	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
909	86.3	cc		Sterol demethylase inhibitor	-			
910	86.29	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
911	86.24	kd	CGS001-5915	RARB	Retinoic acid receptors			
912	86.22	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
913	86.17	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
914	86.12	kd	CGS001-1036	CDO1	-			
915	86.09	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
916	86.05	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
917	86.05	kd	CGS001-598	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
918	86.03	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
919	85.93	kd	CGS001-23030	KDM4B	Histone demethylases			
920	85.87	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
921	85.86	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
922	85.83	cc		Reverse transcriptase inhibitor	-			
923	85.82	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
924	85.8	cp	BRD-K81169441	cerivastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A5	HMGCR inhibitor
925	85.75	kd	CGS001-1198	CLK3	CDC-like kinases			
926	85.69	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
927	85.68	kd	CGS001-6611	SMS	-			
928	85.67	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
929	85.67	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
930	85.61	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
931	85.56	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
932	85.52	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
933	85.46	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
934	85.38	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
935	85.37	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
936	85.3	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
937	85.28	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
938	85.27	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
939	85.25	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
940	85.22	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
941	85.2	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
942	85.17	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
943	85.16	kd	CGS001-55311	ZNF444	Zinc fingers, C2H2-type			
944	85.15	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
945	85.14	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
946	85.12	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
947	85.1	kd	CGS001-6709	SPTAN1	EF-hand domain containing			
948	85.05	oe	ccsbBroad304_06458	IRF3	-			
949	85.04	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
950	84.99	oe	ccsbBroad304_00033	ADSS	-			
951	84.9	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
952	84.88	kd	CGS001-6434	TRA2B	RNA binding motif (RRM) containing			
953	84.79	kd	CGS001-57665	RDH14	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
954	84.78	cp	BRD-K43236057	piceid	ICAM1 inhibitor		GAA, XDH	ICAM1 inhibitor
955	84.77	kd	CGS001-5860	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
956	84.71	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
957	84.66	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
958	84.65	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
959	84.64	kd	CGS001-9868	TOMM70A	Tetratricopeptide (TTC) repeat domain containing			
960	84.63	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
961	84.61	oe	ccsbBroad304_04406	PLA2G12B	-			
962	84.61	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
963	84.6	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
964	84.6	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
965	84.55	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
966	84.53	oe	ccsbBroad304_07761	CORO1A	Coronins			
967	84.51	oe	ccsbBroad304_03555	PANK4	-			
968	84.48	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
969	84.44	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
970	84.43	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
971	84.43	kd	CGS001-2295	FOXF2	Forkhead boxes			
972	84.43	kd	CGS001-403	ARL3	ADP-ribosylation factors			
973	84.38	oe	ccsbBroad304_07326	EIF2B2	-			
974	84.37	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
975	84.36	kd	CGS001-286075	ZNF707	Zinc fingers, C2H2-type			
976	84.33	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
977	84.28	kd	CGS001-10670	RRAGA	-			
978	84.27	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
979	84.26	kd	CGS001-6599	SMARCC1	-			
980	84.26	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
981	84.22	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
982	84.21	kd	CGS001-10112	KIF20A	Kinesins			
983	84.11	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
984	84.1	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
985	84.09	kd	CGS001-5546	PRCC	-			
986	84.08	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
987	84.07	oe	ccsbBroad304_07827	STK38L	NDR family			
988	84.07	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
989	84.05	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
990	83.9	oe	ccsbBroad304_06174	ERCC1	-			
991	83.8	kd	CGS001-8738	CRADD	-			
992	83.79	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
993	83.75	kd	CGS001-65975	STK33	CAMK-unique family			
994	83.68	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
995	83.63	kd	CGS001-6774	STAT3	SH2 domain containing			
996	83.59	oe	ccsbBroad304_06237	GAA	Glycosidases			
997	83.57	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
998	83.55	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
999	83.51	kd	CGS001-10013	HDAC6	Histone deacetylases			
1000	83.5	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
1001	83.39	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
1002	83.31	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
1003	83.25	kd	CGS001-25	ABL1	Abl family			
1004	83.18	kd	CGS001-10084	PQBP1	-			
1005	83.1	oe	ccsbBroad304_00060	AMBP	Lipocalins			
1006	83.1	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
1007	83.08	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
1008	83.07	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
1009	83.03	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
1010	83.02	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1011	82.96	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
1012	82.96	kd	CGS001-2203	FBP1	-			
1013	82.95	cp	BRD-K46435977	valaciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
1014	82.91	kd	CGS001-1120	CHKB	-			
1015	82.9	kd	CGS001-5613	PRKX	Protein kinase A			
1016	82.89	kd	CGS001-6757	SSX2	-			
1017	82.86	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
1018	82.84	kd	CGS001-8837	CFLAR	Endogenous ligands			
1019	82.8	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
1020	82.8	kd	CGS001-6188	RPS3	S ribosomal proteins			
1021	82.73	kd	CGS001-23710	GABARAPL1	-			
1022	82.7	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
1023	82.68	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
1024	82.62	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
1025	82.57	oe	ccsbBroad304_00459	DPYD	-			
1026	82.53	kd	CGS001-347736	NME9	-			
1027	82.49	kd	CGS001-8464	SUPT3H	-			
1028	82.47	kd	CGS001-10607	TBL3	WD repeat domain containing			
1029	82.46	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
1030	82.41	kd	CGS001-117154	DACH2	-			
1031	82.39	oe	ccsbBroad304_06711	PFAS	-			
1032	82.39	kd	CGS001-122402	TDRD9	Tudor domain containing			
1033	82.36	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
1034	82.3	oe	ccsbBroad304_07766	RASSF1	-			
1035	82.29	cp	BRD-K83144676	olmesartan	Angiotensin antagonist		AGTR1	Angiotensin antagonist
1036	82.29	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
1037	82.26	kd	CGS001-8527	DGKD	Pleckstrin homology (PH) domain containing			
1038	82.24	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
1039	82.12	kd	CGS001-51593	SRRT	-			
1040	82.03	oe	ccsbBroad304_03850	TRIB3	Trbl family			
1041	81.97	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
1042	81.96	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
1043	81.95	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
1044	81.95	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
1045	81.89	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
1046	81.78	kd	CGS001-29984	RHOD	-			
1047	81.77	oe	ccsbBroad304_03615	ZNF673	-			
1048	81.72	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
1049	81.68	kd	CGS001-383	ARG1	Arginase			
1050	81.66	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
1051	81.64	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
1052	81.63	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
1053	81.63	kd	CGS001-7504	XK	Blood group antigens			
1054	81.61	oe	ccsbBroad304_04064	PRR15L	-			
1055	81.61	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
1056	81.61	kd	CGS001-338557	O3FAR1	-			
1057	81.59	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
1058	81.56	kd	CGS001-6723	SRM	-			
1059	81.53	oe	ccsbBroad304_05936	CASP2	Caspases			
1060	81.53	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
1061	81.41	oe	ccsbBroad304_02276	MVP	-			
1062	81.39	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
1063	81.36	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
1064	81.35	kd	CGS001-5887	RAD23B	-			
1065	81.34	kd	CGS001-2053	EPHX2	-			
1066	81.28	kd	CGS001-23075	SWAP70	EF-hand domain containing			
1067	81.25	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
1068	81.17	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
1069	81.14	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
1070	81.12	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
1071	81.09	oe	ccsbBroad304_02058	PLOD3	-			
1072	81.07	kd	CGS001-55226	NAT10	-			
1073	81.06	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
1074	81.05	cp	BRD-K57930253	nitrazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, SCN1A	Benzodiazepine receptor agonist
1075	81.04	oe	ccsbBroad304_02292	BCL2L11	-			
1076	80.98	kd	CGS001-169436	C9ORF96	-			
1077	80.96	kd	CGS001-84333	PCGF5	Polycomb group ring fingers			
1078	80.92	kd	CGS001-51005	AMDHD2	-			
1079	80.87	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
1080	80.87	kd	CGS001-2769	GNA15	-			
1081	80.86	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
1082	80.83	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
1083	80.82	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
1084	80.81	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1085	80.8	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
1086	80.78	oe	ccsbBroad304_02414	IRF9	-			
1087	80.74	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
1088	80.74	kd	CGS001-81611	ANP32E	ANP32 acidic nuclear phosphoproteins			
1089	80.72	oe	ccsbBroad304_02438	FAM3C	-			
1090	80.7	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
1091	80.63	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
1092	80.63	kd	CGS001-7486	WRN	-			
1093	80.62	kd	CGS001-6337	SCNN1A	Epithelial sodium channels (ENaC)			
1094	80.59	kd	CGS001-1119	CHKA	-			
1095	80.57	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
1096	80.57	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
1097	80.46	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
1098	80.43	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
1099	80.41	kd	CGS001-58533	SNX6	Sorting nexins			
1100	80.4	kd	CGS001-3383	ICAM1	CD molecules			
1101	80.36	kd	CGS001-29899	GPSM2	Tetratricopeptide (TTC) repeat domain containing			
1102	80.35	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
1103	80.27	kd	CGS001-55107	ANO1	Calcium activated chloride channel			
1104	80.25	kd	CGS001-9815	GIT2	Ankyrin repeat domain containing			
1105	80.24	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
1106	80.23	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
1107	80.09	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
1108	80.03	kd	CGS001-123803	NTAN1	-			
1109	79.98	oe	ccsbBroad304_02278	THRAP3	-			
1110	79.97	kd	CGS001-2161	F12	Chymotrypsin			
1111	79.95	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
1112	79.92	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
1113	79.82	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
1114	79.82	kd	CGS001-55872	PBK	TOPK family			
1115	79.81	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
1116	79.79	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
1117	79.75	kd	CGS001-80025	PANK2	-			
1118	79.73	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
1119	79.65	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
1120	79.64	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
1121	79.56	oe	ccsbBroad304_00183	C1S	Complement system			
1122	79.48	kd	CGS001-9531	BAG3	-			
1123	79.48	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
1124	79.45	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
1125	79.43	kd	CGS001-7535	ZAP70	Syk family			
1126	79.41	kd	CGS001-79094	CHAC1	-			
1127	79.4	kd	CGS001-9925	ZBTB5	BTB/POZ domain containing			
1128	79.38	cc		MTOR inhibitor	-			
1129	79.38	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
1130	79.37	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
1131	79.34	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
1132	79.33	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
1133	79.32	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
1134	79.27	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
1135	79.25	kd	CGS001-523	ATP6V1A	ATPases / V-type			
1136	79.23	kd	CGS001-2771	GNAI2	-			
1137	79.22	kd	CGS001-53340	SPA17	-			
1138	79.18	kd	CGS001-27336	HTATSF1	RNA binding motif (RRM) containing			
1139	79.16	kd	CGS001-6909	TBX2	T-boxes			
1140	79.16	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
1141	79.15	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
1142	79.13	kd	CGS001-51422	PRKAG2	AMPK subfamily			
1143	79.12	cp	BRD-A35519318	benidipine	Calcium channel blocker		CACNA1C, CACNA1G, CYP3A5	Calcium channel blocker
1144	79.1	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
1145	79.09	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
1146	79.08	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
1147	78.89	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
1148	78.88	kd	CGS001-1644	DDC	Catecholamine turnover			
1149	78.66	kd	CGS001-5930	RBBP6	-			
1150	78.66	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
1151	78.64	oe	ccsbBroad304_00949	LRPAP1	-			
1152	78.46	kd	CGS001-2114	ETS2	ETS Transcription Factors			
1153	78.44	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
1154	78.37	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
1155	78.35	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
1156	78.34	kd	CGS001-80347	COASY	-			
1157	78.3	kd	CGS001-79581	GPR172A	-			
1158	78.24	kd	CGS001-369	ARAF	RAF family			
1159	78.21	kd	CGS001-2335	FN1	Endogenous ligands			
1160	78.17	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
1161	78.15	oe	ccsbBroad304_00001	NAT1	-			
1162	78.1	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
1163	78.08	kd	CGS001-5315	PKM2	-			
1164	78.07	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
1165	78.05	oe	ccsbBroad304_07600	NSA2	-			
1166	78.05	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
1167	78.02	kd	CGS001-27125	AFF4	-			
1168	77.98	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
1169	77.95	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
1170	77.93	oe	ccsbBroad304_05098	MAGEB6	-			
1171	77.93	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
1172	77.88	oe	ccsbBroad304_03047	BZW2	-			
1173	77.88	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
1174	77.87	oe	ccsbBroad304_00231	CBFB	-			
1175	77.87	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
1176	77.81	kd	CGS001-7423	VEGFB	-			
1177	77.79	kd	CGS001-2730	GCLM	-			
1178	77.73	oe	ccsbBroad304_02386	EIF1B	-			
1179	77.68	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
1180	77.61	kd	CGS001-5058	PAK1	PAKA subfamily			
1181	77.57	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
1182	77.54	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
1183	77.53	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
1184	77.5	kd	CGS001-4773	NFATC2	Nuclear factor of activated T-cells			
1185	77.44	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
1186	77.38	kd	CGS001-10921	RNPS1	RNA binding motif (RRM) containing			
1187	77.35	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
1188	77.29	kd	CGS001-149233	IL23R	IL-12 receptor family			
1189	77.25	oe	ccsbBroad304_00650	GNA11	-			
1190	77.25	kd	CGS001-5446	PON3	Paraoxonases			
1191	77.2	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
1192	77.14	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
1193	77.14	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
1194	77.13	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
1195	77.09	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
1196	77.09	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
1197	77.09	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
1198	77.09	kd	CGS001-91392	ZNF502	Zinc fingers, C2H2-type			
1199	77.05	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
1200	77.02	kd	CGS001-538	ATP7A	ATPases / P-type			
1201	76.98	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
1202	76.91	kd	CGS001-64087	MCCC2	-			
1203	76.88	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
1204	76.87	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
1205	76.86	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
1206	76.76	kd	CGS001-6189	RPS3A	S ribosomal proteins			
1207	76.62	oe	ccsbBroad304_02002	RNMT	-			
1208	76.6	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
1209	76.56	kd	CGS001-2768	GNA12	-			
1210	76.53	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
1211	76.47	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
1212	76.44	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
1213	76.38	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
1214	76.37	kd	CGS001-629	CFB	Complement system			
1215	76.35	kd	CGS001-1879	EBF1	-			
1216	76.33	kd	CGS001-3660	IRF2	-			
1217	76.3	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
1218	76.26	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
1219	76.19	kd	CGS001-1737	DLAT	-			
1220	76.18	kd	CGS001-10401	PIAS3	Zinc fingers, MIZ-type			
1221	76.06	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
1222	76.05	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
1223	75.94	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
1224	75.85	kd	CGS001-857	CAV1	-			
1225	75.79	kd	CGS001-26993	AKAP8L	-			
1226	75.75	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
1227	75.71	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
1228	75.69	kd	CGS001-10538	BATF	basic leucine zipper proteins			
1229	75.65	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
1230	75.61	kd	CGS001-6778	STAT6	SH2 domain containing			
1231	75.54	oe	ccsbBroad304_06178	ERCC5	-			
1232	75.5	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
1233	75.48	cc		Calmodulin antagonist	-			
1234	75.43	oe	ccsbBroad304_01105	PNP	-			
1235	75.43	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
1236	75.42	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1237	75.33	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
1238	75.32	kd	CGS001-9961	MVP	-			
1239	75.3	kd	CGS001-5591	PRKDC	Other PIKK family kinases			
1240	75.29	kd	CGS001-63948	DMRTB1	-			
1241	75.25	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
1242	75.15	oe	ccsbBroad304_01832	PAX8	Paired boxes			
1243	75.12	kd	CGS001-1154	CISH	SH2 domain containing			
1244	75.11	oe	ccsbBroad304_06318	GPER	-			
1245	75.08	oe	ccsbBroad304_00841	IKBKB	IKK family			
1246	75.08	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
1247	75.07	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
1248	75.03	kd	CGS001-81577	GFOD2	-			
1249	75	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
1250	74.89	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
1251	74.88	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
1252	74.78	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
1253	74.78	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
1254	74.78	kd	CGS001-1493	CTLA4	CD molecules			
1255	74.77	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
1256	74.75	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
1257	74.67	cc		PKC activator	-			
1258	74.65	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
1259	74.65	kd	CGS001-4801	NFYB	-			
1260	74.6	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
1261	74.59	kd	CGS001-3297	HSF1	-			
1262	74.57	kd	CGS001-5184	PEPD	Methionyl aminopeptidase			
1263	74.52	kd	CGS001-57167	SALL4	Zinc fingers, C2H2-type			
1264	74.51	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
1265	74.46	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
1266	74.42	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
1267	74.4	kd	CGS001-2966	GTF2H2	General transcription factors			
1268	74.39	kd	CGS001-3775	KCNK1	Two-P potassium channels			
1269	74.34	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
1270	74.34	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
1271	74.3	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
1272	74.29	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
1273	74.27	kd	CGS001-9122	SLC16A4	SLC16 family of monocarboxylate transporters			
1274	74.21	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
1275	74.17	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
1276	74.12	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
1277	73.95	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1278	73.93	kd	CGS001-29116	MYLIP	-			
1279	73.85	kd	CGS001-6210	RPS15A	S ribosomal proteins			
1280	73.84	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
1281	73.78	kd	CGS001-57121	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
1282	73.73	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
1283	73.7	kd	CGS001-9512	PMPCB	-			
1284	73.66	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
1285	73.6	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1286	73.6	kd	CGS001-56882	CDC42SE1	-			
1287	73.5	kd	CGS001-54899	PXK	Slob family			
1288	73.49	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
1289	73.47	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
1290	73.42	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
1291	73.33	kd	CGS001-10725	NFAT5	Nuclear factor of activated T-cells			
1292	73.3	oe	ccsbBroad304_03479	YTHDF1	-			
1293	73.26	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
1294	73.16	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
1295	73.15	oe	ccsbBroad304_05931	CAPG	-			
1296	73.11	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
1297	73.1	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
1298	73.02	kd	CGS001-54490	UGT2B28	UDP glucuronosyltransferases			
1299	73.01	cc		General transcription factors group 1 LOF	-			
1300	73.01	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
1301	72.98	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
1302	72.94	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
1303	72.93	oe	ccsbBroad304_01114	NUP88	-			
1304	72.92	kd	CGS001-4836	NMT1	-			
1305	72.88	cc		Sigma receptor antagonist	-			
1306	72.86	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
1307	72.83	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
1308	72.78	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
1309	72.75	cp	BRD-K96134740	kitasamycin	Protein synthesis inhibitor			Protein synthesis inhibitor
1310	72.75	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
1311	72.75	kd	CGS001-22850	ADNP2	Zinc fingers, C2H2-type			
1312	72.74	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
1313	72.74	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
1314	72.73	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
1315	72.69	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
1316	72.65	oe	ccsbBroad304_02415	TUBB3	Tubulins			
1317	72.64	oe	ccsbBroad304_00032	ADSL	-			
1318	72.64	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
1319	72.57	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
1320	72.57	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
1321	72.55	cc		Phospholipases GOF	-			
1322	72.55	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
1323	72.51	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
1324	72.43	kd	CGS001-4664	NAB1	-			
1325	72.38	kd	CGS001-6857	SYT1	Synaptotagmins			
1326	72.34	kd	CGS001-23753	SDF2L1	-			
1327	72.29	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
1328	72.27	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
1329	72.22	oe	ccsbBroad304_02048	BCL10	-			
1330	72.2	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
1331	72.18	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
1332	72.13	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
1333	72.09	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
1334	72.01	oe	ccsbBroad304_06494	KLRC1	CD molecules			
1335	72	kd	CGS001-3693	ITGB5	Integrins			
1336	71.96	oe	ccsbBroad304_04465	RERG	-			
1337	71.94	cp	BRD-K09471561	levofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
1338	71.78	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
1339	71.77	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
1340	71.76	oe	ccsbBroad304_08322	UFM1	-			
1341	71.72	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
1342	71.72	kd	CGS001-1978	EIF4EBP1	-			
1343	71.7	kd	CGS001-58478	ENOPH1	-			
1344	71.66	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
1345	71.62	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
1346	71.57	kd	CGS001-3431	SP110	Non-enzymatic BRD containing proteins			
1347	71.56	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
1348	71.53	kd	CGS001-5073	PARN	-			
1349	71.5	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
1350	71.37	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
1351	71.31	kd	CGS001-11140	CDC37	-			
1352	71.29	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
1353	71.26	kd	CGS001-55765	C1ORF106	-			
1354	71.23	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
1355	71.23	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
1356	71.21	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
1357	71.2	oe	ccsbBroad304_00212	CAMLG	-			
1358	71.18	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
1359	71.08	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
1360	71.01	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
1361	70.99	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
1362	70.96	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
1363	70.92	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
1364	70.91	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
1365	70.84	oe	ccsbBroad304_06301	GOT2	-			
1366	70.83	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
1367	70.77	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1368	70.76	oe	ccsbBroad304_05758	ACADSB	-			
1369	70.75	kd	CGS001-5223	PGAM1	-			
1370	70.74	kd	CGS001-3665	IRF7	-			
1371	70.72	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
1372	70.72	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
1373	70.72	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
1374	70.63	cp	BRD-K82109576	vincristine	Tubulin inhibitor		TUBB, TUBA4A	Tubulin inhibitor
1375	70.58	oe	ccsbBroad304_02579	YWHAQ	-			
1376	70.58	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1377	70.53	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
1378	70.52	kd	CGS001-55500	ETNK1	-			
1379	70.47	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
1380	70.39	kd	CGS001-51451	LCMT1	-			
1381	70.39	oe	ccsbBroad304_00112	ASNA1	-			
1382	70.37	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
1383	70.36	kd	CGS001-26292	MYCBP	-			
1384	70.34	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
1385	70.33	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
1386	70.32	oe	ccsbBroad304_06350	HAL	-			
1387	70.32	kd	CGS001-10221	TRIB1	Trbl family			
1388	70.31	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
1389	70.29	kd	CGS001-4830	NME1	-			
1390	70.27	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
1391	70.27	cp	BRD-A24191444	ifenprodil	Adrenergic receptor antagonist		GRIN1, GRIN2B	Adrenergic receptor antagonist, Glutamate receptor antagonist
1392	70.24	oe	ccsbBroad304_00549	FDX1	-			
1393	70.21	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1394	70.21	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
1395	70.19	kd	CGS001-657	BMPR1A	Type I receptor serine/threonine kinases			
1396	70.17	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
1397	70.14	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
1398	70.11	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
1399	70.09	kd	CGS001-5962	RDX	-			
1400	70.09	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
1401	70.03	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
1402	70.02	oe	ccsbBroad304_00464	DTNA	-			
1403	70.01	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
1404	69.99	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
1405	69.96	cp	BRD-K56614220	clofazimine	GK0582 inhibitor			GK0582 inhibitor
1406	69.94	kd	CGS001-5134	PDCD2	Zinc fingers, MYND-type			
1407	69.94	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
1408	69.93	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
1409	69.91	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
1410	69.87	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
1411	69.87	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
1412	69.84	kd	CGS001-2355	FOSL2	basic leucine zipper proteins			
1413	69.82	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
1414	69.77	cp	BRD-K62374253	rufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
1415	69.77	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
1416	69.74	oe	ccsbBroad304_06992	SRC	Src family			
1417	69.74	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1418	69.73	oe	ccsbBroad304_05756	ACAA1	-			
1419	69.7	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
1420	69.7	kd	CGS001-4791	NFKB2	NFkappaB transcription factor family			
1421	69.69	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
1422	69.62	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
1423	69.6	kd	CGS001-10392	NOD1	Nucleotide-binding domain and leucine rich repeat containing			
1424	69.59	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1425	69.57	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
1426	69.54	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
1427	69.54	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
1428	69.52	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
1429	69.5	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
1430	69.49	kd	CGS001-9917	FAM20B	-			
1431	69.48	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
1432	69.43	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
1433	69.43	kd	CGS001-23196	FAM120A	-			
1434	69.41	oe	ccsbBroad304_04457	TOX2	-			
1435	69.37	oe	ccsbBroad304_01701	TPI1	-			
1436	69.35	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
1437	69.33	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
1438	69.32	oe	ccsbBroad304_06462	ITGAE	Integrins			
1439	69.32	kd	CGS001-22934	RPIA	-			
1440	69.25	oe	ccsbBroad304_03112	NENF	-			
1441	69.25	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
1442	69.23	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
1443	69.22	oe	ccsbBroad304_03951	NARFL	-			
1444	69.17	oe	ccsbBroad304_02287	GNPDA1	-			
1445	69.14	kd	CGS001-7389	UROD	-			
1446	69.14	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
1447	69.13	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
1448	69.08	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
1449	69.08	kd	CGS001-3416	IDE	Pitrilysin			
1450	69.04	oe	ccsbBroad304_00795	HSF2	-			
1451	69.02	oe	ccsbBroad304_06777	PRNP	CD molecules			
1452	68.98	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
1453	68.93	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
1454	68.89	kd	CGS001-84634	KISS1R	GPCR / Class A : RF amide peptide receptors			
1455	68.87	kd	CGS001-10434	LYPLA1	-			
1456	68.85	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
1457	68.84	oe	ccsbBroad304_03386	SPA17	-			
1458	68.84	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
1459	68.8	kd	CGS001-3663	IRF5	-			
1460	68.78	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
1461	68.73	kd	CGS001-4191	MDH2	-			
1462	68.71	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
1463	68.62	oe	ccsbBroad304_03848	METTL14	-			
1464	68.54	kd	CGS001-11329	STK38	NDR family			
1465	68.53	oe	ccsbBroad304_07798	EXOC3	-			
1466	68.53	kd	CGS001-7052	TGM2	Transglutaminases			
1467	68.42	oe	ccsbBroad304_07252	DGKZ	-			
1468	68.42	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
1469	68.38	kd	CGS001-4208	MEF2C	Myocyte enhancer factors			
1470	68.34	oe	ccsbBroad304_08292	IP6K2	-			
1471	68.32	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
1472	68.24	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
1473	68.24	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
1474	68.17	cp	BRD-K33226500	indinavir	HIV protease inhibitor		CYP3A5	HIV protease inhibitor
1475	68.16	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
1476	68.15	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
1477	68.15	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
1478	68.15	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
1479	68.15	kd	CGS001-23530	NNT	-			
1480	68.13	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
1481	68.11	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
1482	68.11	kd	CGS001-6919	TCEA2	-			
1483	68.04	kd	CGS001-285676	ZNF454	Zinc fingers, C2H2-type			
1484	67.88	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
1485	67.84	kd	CGS001-79071	ELOVL6	-			
1486	67.84	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
1487	67.81	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
1488	67.75	kd	CGS001-6799	SULT1A2	Sulfotransferases, cytosolic			
1489	67.75	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
1490	67.73	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
1491	67.71	kd	CGS001-84759	PCGF1	Polycomb group ring fingers			
1492	67.67	cp	BRD-K54316499	tolterodine	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRM1, CHRM4, CHRM5	Acetylcholine receptor antagonist
1493	67.64	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
1494	67.64	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
1495	67.61	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
1496	67.5	oe	ccsbBroad304_08684	CXCR7	-			
1497	67.44	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
1498	67.43	oe	ccsbBroad304_02922	TES	-			
1499	67.38	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
1500	67.28	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
1501	67.27	kd	CGS001-4671	NAIP	Inhibitors of apoptosis (IAP) protein family			
1502	67.23	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
1503	67.1	kd	CGS001-4638	MYLK	Myosin Light Chain Kinase (MLCK) family			
1504	67.09	kd	CGS001-6217	RPS16	S ribosomal proteins			
1505	67.05	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
1506	67.02	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
1507	67.01	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
1508	66.95	oe	ccsbBroad304_01659	TERF1	-			
1509	66.95	oe	ccsbBroad304_06255	LRRC32	-			
1510	66.93	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
1511	66.92	kd	CGS001-3203	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
1512	66.89	kd	CGS001-4072	EPCAM	CD molecules			
1513	66.88	kd	CGS001-64781	CERK	Ceramide kinase			
1514	66.85	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
1515	66.85	kd	CGS001-206358	SLC36A1	SLC36 family of proton-coupled amino acid transporters			
1516	66.85	kd	CGS001-976	CD97	Adhesion Class GPCRs			
1517	66.84	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
1518	66.82	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
1519	66.79	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
1520	66.78	oe	ccsbBroad304_01632	SYPL1	-			
1521	66.78	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
1522	66.78	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
1523	66.68	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
1524	66.64	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
1525	66.42	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
1526	66.42	kd	CGS001-1147	CHUK	IKK family			
1527	66.39	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1528	66.37	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
1529	66.37	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
1530	66.33	kd	CGS001-3456	IFNB1	Interferons			
1531	66.27	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
1532	66.23	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
1533	66.21	kd	CGS001-26523	EIF2C1	-			
1534	66.15	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
1535	66.15	kd	CGS001-23066	CAND2	-			
1536	66.13	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
1537	66.12	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
1538	66.12	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
1539	66.06	kd	CGS001-8446	DUSP11	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1540	66.04	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
1541	65.97	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
1542	65.97	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
1543	65.96	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
1544	65.95	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
1545	65.93	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
1546	65.9	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
1547	65.88	kd	CGS001-25925	ZNF521	Zinc fingers, C2H2-type			
1548	65.82	kd	CGS001-5052	PRDX1	-			
1549	65.81	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
1550	65.77	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
1551	65.72	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1552	65.71	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
1553	65.64	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
1554	65.63	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
1555	65.56	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
1556	65.47	oe	ccsbBroad304_02834	GABARAPL1	-			
1557	65.43	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1558	65.42	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
1559	65.42	kd	CGS001-55723	ASF1B	-			
1560	65.38	oe	ccsbBroad304_09281	TPD52L3	-			
1561	65.37	kd	CGS001-328	APEX1	-			
1562	65.34	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
1563	65.28	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
1564	65.26	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
1565	65.1	kd	CGS001-10923	SUB1	-			
1566	65.05	oe	ccsbBroad304_01576	SOAT1	-			
1567	65.02	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
1568	65.02	kd	CGS001-10312	TCIRG1	ATPases / V-type			
1569	65.01	kd	CGS001-286530	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
1570	65	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
1571	64.99	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
1572	64.99	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
1573	64.95	kd	CGS001-10765	KDM5B	Histone demethylases			
1574	64.92	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
1575	64.92	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
1576	64.92	kd	CGS001-2023	ENO1	-			
1577	64.89	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
1578	64.88	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
1579	64.86	kd	CGS001-8797	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
1580	64.82	kd	CGS001-6622	SNCA	Parkinson disease			
1581	64.77	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
1582	64.67	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
1583	64.64	oe	ccsbBroad304_01880	LAGE3	-			
1584	64.62	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
1585	64.59	kd	CGS001-8826	IQGAP1	-			
1586	64.54	cc		EGFR inhibitor	-			
1587	64.5	oe	ccsbBroad304_00747	HLF	-			
1588	64.49	kd	CGS001-2108	ETFA	-			
1589	64.4	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1590	64.4	kd	CGS001-213	ALB	-			
1591	64.39	cp	BRD-K53220666	trimetozine	Sedative			Sedative
1592	64.33	oe	ccsbBroad304_01180	PFKFB3	-			
1593	64.2	oe	ccsbBroad304_03372	CAB39	-			
1594	64.18	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1595	64.14	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
1596	64.14	kd	CGS001-11044	PAPD7	-			
1597	64.12	kd	CGS001-23786	BCL2L13	-			
1598	64.07	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
1599	64.07	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
1600	64.04	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
1601	63.99	oe	ccsbBroad304_01304	PSEN1	Presenilin			
1602	63.97	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
1603	63.95	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1604	63.92	oe	ccsbBroad304_07411	LPXN	-			
1605	63.91	kd	CGS001-7485	WRB	-			
1606	63.91	kd	CGS001-2957	GTF2A1	General transcription factors			
1607	63.83	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
1608	63.83	kd	CGS001-3939	LDHA	-			
1609	63.83	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
1610	63.82	kd	CGS001-4869	NPM1	-			
1611	63.82	kd	CGS001-109	ADCY3	Adenylyl cyclases			
1612	63.74	kd	CGS001-3799	KIF5B	Kinesins			
1613	63.73	oe	ccsbBroad304_03544	FAIM	-			
1614	63.73	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
1615	63.72	cp	BRD-A23359898	sibutramine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, CYP2B6, CYP2C19, CYP3A5	Serotonin reuptake inhibitor
1616	63.71	kd	CGS001-345	APOC3	Apolipoproteins			
1617	63.7	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
1618	63.69	kd	CGS001-3169	FOXA1	Forkhead boxes			
1619	63.68	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
1620	63.64	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
1621	63.62	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
1622	63.59	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
1623	63.5	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
1624	63.49	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
1625	63.46	oe	ccsbBroad304_06837	RAF1	RAF family			
1626	63.44	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
1627	63.39	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
1628	63.38	oe	ccsbBroad304_00471	E2F6	-			
1629	63.37	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1630	63.32	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
1631	63.29	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
1632	63.27	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
1633	63.22	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
1634	63.15	kd	CGS001-701	BUB1B	Bub family			
1635	63.12	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1636	63.1	cp	BRD-A07395371	esmolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
1637	63.1	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
1638	63.08	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
1639	63.03	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
1640	63.03	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
1641	63.01	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
1642	63	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
1643	62.98	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
1644	62.93	kd	CGS001-4927	NUP88	-			
1645	62.92	kd	CGS001-7263	TST	-			
1646	62.92	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
1647	62.68	kd	CGS001-11113	CIT	Other DMPK family kinases			
1648	62.58	kd	CGS001-4548	MTR	-			
1649	62.56	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
1650	62.5	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
1651	62.49	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
1652	62.41	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
1653	62.4	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
1654	62.36	oe	ccsbBroad304_05528	TICAM2	-			
1655	62.23	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
1656	62.19	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
1657	62.12	oe	ccsbBroad304_08386	SMOX	-			
1658	62.12	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
1659	62.12	kd	CGS001-27333	GOLIM4	-			
1660	62	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
1661	61.93	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
1662	61.93	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
1663	61.91	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
1664	61.88	oe	ccsbBroad304_06090	DDOST	-			
1665	61.86	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
1666	61.82	kd	CGS001-10523	CHERP	G patch domain containing			
1667	61.8	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
1668	61.8	kd	CGS001-23536	ADAT1	-			
1669	61.75	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1670	61.71	kd	CGS001-2717	GLA	-			
1671	61.58	kd	CGS001-7016	TESK1	TESK subfamily			
1672	61.54	kd	CGS001-7247	TSN	-			
1673	61.5	kd	CGS001-10608	MXD4	Basic helix-loop-helix proteins			
1674	61.44	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
1675	61.42	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
1676	61.4	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
1677	61.38	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
1678	61.25	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1679	61.2	oe	ccsbBroad304_01617	STX4	-			
1680	61.16	kd	CGS001-6822	SULT2A1	Sulfotransferases, cytosolic			
1681	61.12	kd	CGS001-27347	STK39	FRAY subfamily			
1682	61.12	kd	CGS001-5608	MAP2K6	MAPKK:STE7 family			
1683	61.06	oe	ccsbBroad304_00423	DAXX	-			
1684	61.03	cc		X linked mental retardation group 2 LOF	-			
1685	61.03	oe	ccsbBroad304_03269	CD320	CD molecules			
1686	61.01	kd	CGS001-79885	HDAC11	Histone deacetylases			
1687	60.95	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1688	60.9	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
1689	60.88	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
1690	60.87	kd	CGS001-1356	CP	-			
1691	60.86	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
1692	60.84	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
1693	60.84	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
1694	60.79	oe	ccsbBroad304_02738	RRS1	-			
1695	60.79	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1696	60.77	kd	CGS001-58508	MLL3	-			
1697	60.62	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
1698	60.61	kd	CGS001-27097	TAF5L	WD repeat domain containing			
1699	60.61	kd	CGS001-124535	HSF5	-			
1700	60.48	kd	CGS001-367	AR	Nuclear hormone receptors			
1701	60.47	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1702	60.45	kd	CGS001-22889	KIAA0907	-			
1703	60.37	kd	CGS001-5320	PLA2G2A	Hydrolases			
1704	60.37	kd	CGS001-662	BNIP1	-			
1705	60.36	kd	CGS001-57459	GATAD2B	GATA zinc finger domain containing			
1706	60.35	kd	CGS001-6804	STX1A	-			
1707	60.28	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
1708	60.25	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
1709	60.25	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
1710	60.22	kd	CGS001-8495	PPFIBP2	Sterile alpha motif (SAM) domain containing			
1711	59.97	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
1712	59.94	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
1713	59.89	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
1714	59.79	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
1715	59.75	kd	CGS001-11154	AP4S1	-			
1716	59.72	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
1717	59.72	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
1718	59.72	oe	ccsbBroad304_02452	NXF1	-			
1719	59.7	kd	CGS001-6595	SMARCA2	Non-enzymatic BRD containing proteins			
1720	59.64	cc		Kinase anchoring proteins LOF	-			
1721	59.61	kd	CGS001-5562	PRKAA1	AMPK subfamily			
1722	59.59	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
1723	59.5	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
1724	59.5	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
1725	59.43	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
1726	59.39	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
1727	59.38	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
1728	59.31	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
1729	59.31	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
1730	59.26	cp	BRD-K82795137	loratadine	Histamine receptor antagonist		HRH1, CYP2C19, CYP3A5	Histamine receptor antagonist
1731	59.12	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
1732	59.1	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
1733	59.06	kd	CGS001-6608	SMO	GPCR / Class F : Frizzled receptors			
1734	59.06	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
1735	58.99	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
1736	58.97	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
1737	58.96	kd	CGS001-10682	EBP	-			
1738	58.95	oe	ccsbBroad304_02109	XPR1	-			
1739	58.95	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
1740	58.93	kd	CGS001-23057	NMNAT2	-			
1741	58.88	cp	BRD-K96471533	nitazoxanide	Pyruvate ferredoxin oxidoreductase inhibitor			Pyruvate ferredoxin oxidoreductase inhibitor
1742	58.87	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1743	58.81	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
1744	58.78	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
1745	58.77	kd	CGS001-125919	ZNF543	Zinc fingers, C2H2-type			
1746	58.77	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
1747	58.76	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
1748	58.75	oe	ccsbBroad304_00226	CAV1	-			
1749	58.74	kd	CGS001-112812	FDX1L	-			
1750	58.63	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
1751	58.63	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
1752	58.62	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
1753	58.61	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
1754	58.58	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
1755	58.57	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
1756	58.56	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
1757	58.52	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
1758	58.49	kd	CGS001-5590	PRKCZ	Iota subfamily			
1759	58.47	kd	CGS001-892	CCNC	-			
1760	58.43	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
1761	58.39	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
1762	58.25	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
1763	58.25	kd	CGS001-1128	CHRM1	Cholinergic receptors			
1764	58.24	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
1765	58.24	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
1766	58.13	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
1767	58.06	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
1768	58.06	kd	CGS001-27148	STK36	Unc-51-like kinase (ULK) family			
1769	57.99	kd	CGS001-185	AGTR1	Angiotensin receptors			
1770	57.95	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
1771	57.85	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
1772	57.84	oe	ccsbBroad304_07088	TP53	-			
1773	57.82	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
1774	57.82	kd	CGS001-3032	HADHB	-			
1775	57.81	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
1776	57.77	kd	CGS001-57804	POLD4	DNA polymerases			
1777	57.76	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
1778	57.62	kd	CGS001-813	CALU	EF-hand domain containing			
1779	57.62	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
1780	57.59	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
1781	57.58	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
1782	57.51	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
1783	57.49	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
1784	57.48	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
1785	57.46	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
1786	57.4	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
1787	57.4	kd	CGS001-805	CALM2	EF-hand domain containing			
1788	57.39	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
1789	57.36	kd	CGS001-51564	HDAC7	Histone deacetylases			
1790	57.23	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
1791	57.23	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
1792	57.22	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
1793	57.18	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
1794	57.04	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
1795	57.02	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
1796	57	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
1797	56.98	kd	CGS001-7353	UFD1L	-			
1798	56.98	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
1799	56.95	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1800	56.93	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
1801	56.91	oe	ccsbBroad304_06226	FTL	-			
1802	56.9	oe	ccsbBroad304_00880	IRF2	-			
1803	56.86	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
1804	56.83	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
1805	56.78	kd	CGS001-11333	PDAP1	-			
1806	56.77	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
1807	56.74	kd	CGS001-81620	CDT1	-			
1808	56.72	kd	CGS001-389421	LIN28B	-			
1809	56.66	oe	ccsbBroad304_01651	TCF7L2	-			
1810	56.66	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
1811	56.64	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
1812	56.6	kd	CGS001-2810	SFN	-			
1813	56.6	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
1814	56.55	kd	CGS001-56139	PCDHA10	Cadherins / Protocadherins : Clustered			
1815	56.55	kd	CGS001-3909	LAMA3	Laminins			
1816	56.53	kd	CGS001-10153	CEBPZ	-			
1817	56.5	kd	CGS001-2523	FUT1	Fucosyltransferases			
1818	56.49	kd	CGS001-9447	AIM2	-			
1819	56.48	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
1820	56.48	kd	CGS001-995	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1821	56.46	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
1822	56.43	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
1823	56.42	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
1824	56.38	kd	CGS001-6925	TCF4	Basic helix-loop-helix proteins			
1825	56.37	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
1826	56.3	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
1827	56.21	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
1828	56.2	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
1829	56.14	kd	CGS001-5950	RBP4	Lipocalins			
1830	56.13	kd	CGS001-29102	DROSHA	-			
1831	56.12	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
1832	56.12	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
1833	56.12	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
1834	56.08	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
1835	55.97	kd	CGS001-5710	PSMD4	Proteasome (prosome, macropain) subunits			
1836	55.95	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
1837	55.9	kd	CGS001-516	ATP5G1	ATPases / F-type			
1838	55.88	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
1839	55.86	cp	BRD-K66412701	pazufloxacin	Topoisomerase inhibitor			Topoisomerase inhibitor
1840	55.81	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
1841	55.73	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
1842	55.72	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
1843	55.64	oe	ccsbBroad304_07145	ZFP161	-			
1844	55.6	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1845	55.56	kd	CGS001-64376	IKZF5	IKAROS zinc fingers			
1846	55.53	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
1847	55.53	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
1848	55.39	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
1849	55.38	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
1850	55.34	kd	CGS001-581	BAX	-			
1851	55.25	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
1852	55.24	kd	CGS001-6251	RSU1	-			
1853	55.18	cp	BRD-A87387433	cefpodoxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1854	55.17	oe	ccsbBroad304_00370	CS	-			
1855	55.02	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
1856	54.98	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1857	54.92	cp	BRD-K55034111	pefloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
1858	54.88	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
1859	54.88	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
1860	54.88	oe	ccsbBroad304_00501	EMD	-			
1861	54.88	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
1862	54.84	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
1863	54.81	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
1864	54.8	kd	CGS001-7965	AIMP2	-			
1865	54.76	oe	ccsbBroad304_02136	COPS2	-			
1866	54.76	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
1867	54.74	kd	CGS001-58492	ZNF77	Zinc fingers, C2H2-type			
1868	54.72	kd	CGS001-9232	PTTG1	-			
1869	54.7	kd	CGS001-10652	YKT6	-			
1870	54.69	kd	CGS001-6446	SGK1	SGK family			
1871	54.64	kd	CGS001-2348	FOLR1	-			
1872	54.62	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
1873	54.62	kd	CGS001-1545	CYP1B1	Cytochrome P450s			
1874	54.49	kd	CGS001-79109	MAPKAP1	-			
1875	54.44	oe	ccsbBroad304_02838	SDF2L1	-			
1876	54.37	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
1877	54.35	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
1878	54.34	kd	CGS001-23046	KIF21B	Kinesins			
1879	54.31	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
1880	54.31	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
1881	54.27	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
1882	54.27	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
1883	54.25	oe	ccsbBroad304_02677	PDAP1	-			
1884	54.24	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
1885	54.18	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
1886	54.18	kd	CGS001-5621	PRNP	CD molecules			
1887	54.18	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
1888	54.16	kd	CGS001-139135	PASD1	-			
1889	54.15	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1890	54.15	kd	CGS001-11040	PIM2	PIM family			
1891	54.11	oe	ccsbBroad304_00268	CD81	CD molecules			
1892	54.11	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
1893	54.11	kd	CGS001-9453	GGPS1	Lanosterol biosynthesis pathway			
1894	54.04	kd	CGS001-54815	GATAD2A	GATA zinc finger domain containing			
1895	54.02	kd	CGS001-374291	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
1896	54.02	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1897	53.98	kd	CGS001-2168	FABP1	Fatty acid-binding proteins			
1898	53.97	kd	CGS001-466	ATF1	basic leucine zipper proteins			
1899	53.96	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
1900	53.9	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
1901	53.9	oe	ccsbBroad304_08167	DNTTIP2	-			
1902	53.9	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
1903	53.73	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
1904	53.69	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
1905	53.67	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1906	53.66	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
1907	53.62	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
1908	53.6	kd	CGS001-6391	SDHC	Mitochondrial respiratory chain complex / Complex II			
1909	53.56	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
1910	53.51	oe	ccsbBroad304_01593	SRP14	-			
1911	53.5	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
1912	53.48	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
1913	53.4	kd	CGS001-204	AK2	Adenylate kinases			
1914	53.39	oe	ccsbBroad304_00085	APRT	-			
1915	53.36	cp	BRD-K85503079	perospirone	Dopamine receptor antagonist		DRD2, HTR2A, DRD3, DRD4, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
1916	53.34	oe	ccsbBroad304_08452	PIH1D1	-			
1917	53.33	kd	CGS001-23142	DCUN1D4	-			
1918	53.27	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
1919	53.15	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1920	53.09	cc		CCK receptor antagonist	-			
1921	53.08	kd	CGS001-10841	FTCD	-			
1922	53.07	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
1923	53.04	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
1924	53.03	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
1925	53.03	cp	BRD-A00520476	otenzepad	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
1926	53	oe	ccsbBroad304_03570	QRSL1	-			
1927	52.95	kd	CGS001-55509	BATF3	basic leucine zipper proteins			
1928	52.94	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
1929	52.91	kd	CGS001-6775	STAT4	SH2 domain containing			
1930	52.88	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1931	52.86	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
1932	52.83	kd	CGS001-1662	DDX10	DEAD-boxes			
1933	52.8	oe	ccsbBroad304_08481	CEP55	-			
1934	52.8	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
1935	52.74	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
1936	52.74	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
1937	52.72	cc		MDM inhibitor	-			
1938	52.66	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1939	52.56	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
1940	52.52	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
1941	52.48	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
1942	52.48	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
1943	52.44	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
1944	52.32	oe	ccsbBroad304_03450	TMED9	-			
1945	52.32	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
1946	52.26	kd	CGS001-79145	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
1947	52.2	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
1948	52.19	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
1949	52.18	kd	CGS001-53632	PRKAG3	AMPK subfamily			
1950	52.15	kd	CGS001-5432	POLR2C	RNA polymerase subunits			
1951	52.06	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
1952	52.01	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
1953	51.96	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
1954	51.96	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
1955	51.95	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
1956	51.92	kd	CGS001-10943	MSL3	-			
1957	51.91	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
1958	51.89	kd	CGS001-8681	JMJD7-PLA2G4B	-			
1959	51.88	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1960	51.84	cp	BRD-A39390670	rabeprazole	ATPase inhibitor		ATP4A, CYP2C19	ATPase inhibitor, Gastrin inhibitor
1961	51.76	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
1962	51.74	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
1963	51.73	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
1964	51.72	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
1965	51.72	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
1966	51.69	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
1967	51.69	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
1968	51.69	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
1969	51.66	oe	ccsbBroad304_02243	DLGAP5	-			
1970	51.65	oe	ccsbBroad304_02133	CD83	CD molecules			
1971	51.65	kd	CGS001-10628	TXNIP	-			
1972	51.64	kd	CGS001-57504	MTA3	GATA zinc finger domain containing			
1973	51.61	cc		Ribosomal 40s Subunit LOF	-			
1974	51.6	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
1975	51.58	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
1976	51.57	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
1977	51.54	kd	CGS001-9929	JOSD1	-			
1978	51.53	oe	ccsbBroad304_00966	MAFG	-			
1979	51.52	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
1980	51.49	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
1981	51.43	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
1982	51.42	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
1983	51.36	kd	CGS001-3455	IFNAR2	Interferon receptor family			
1984	51.3	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
1985	51.25	oe	ccsbBroad304_03405	CHRAC1	-			
1986	51.25	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
1987	51.25	kd	CGS001-6908	TBP	General transcription factors			
1988	51.23	kd	CGS001-117581	TWIST2	Basic helix-loop-helix proteins			
1989	51.19	kd	CGS001-6625	SNRNP70	RNA binding motif (RRM) containing			
1990	51.13	kd	CGS001-2172	FABP6	Fatty acid binding protein family			
1991	51.12	oe	ccsbBroad304_07875	SPECC1L	-			
1992	51.12	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
1993	51.11	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
1994	51.1	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
1995	51.1	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1996	51.07	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
1997	51.05	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
1998	51.04	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
1999	51.01	kd	CGS001-8204	NRIP1	-			
2000	50.97	kd	CGS001-283	ANG	Ribonucleases, RNase A			
2001	50.96	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
2002	50.94	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2003	50.92	kd	CGS001-5987	TRIM27	-			
2004	50.9	kd	CGS001-4779	NFE2L1	basic leucine zipper proteins			
2005	50.88	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
2006	50.8	kd	CGS001-10626	TRIM16	Tripartite motif containing			
2007	50.78	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
2008	50.75	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
2009	50.72	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
2010	50.65	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
2011	50.6	kd	CGS001-8453	CUL2	-			
2012	50.59	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
2013	50.58	oe	ccsbBroad304_06136	ECHS1	-			
2014	50.52	kd	CGS001-54536	EXOC6	-			
2015	50.48	kd	CGS001-140690	CTCFL	Zinc fingers, C2H2-type			
2016	50.47	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
2017	50.44	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
2018	50.32	cc		MEK inhibitor	-			
2019	50.32	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
2020	50.26	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
2021	50.24	kd	CGS001-57326	PBXIP1	-			
2022	50.24	kd	CGS001-2674	GFRA1	GDNF receptor family			
2023	50.14	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
2024	50.12	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
2025	50.1	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
2026	50.09	kd	CGS001-6990	DYNLT3	Cytoplasmic dyneins			
2027	50	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
2028	49.96	oe	ccsbBroad304_06287	GM2A	-			
2029	49.9	kd	CGS001-2770	GNAI1	-			
2030	49.88	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
2031	49.87	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
2032	49.85	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
2033	49.73	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
2034	49.71	kd	CGS001-10873	ME3	-			
2035	49.7	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
2036	49.7	kd	CGS001-203	AK1	Adenylate kinases			
2037	49.69	kd	CGS001-6591	SNAI2	Snail homologs			
2038	49.69	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
2039	49.63	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
2040	49.61	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
2041	49.59	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
2042	49.58	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
2043	49.58	kd	CGS001-10131	TRAP1	Heat shock proteins / HSPC			
2044	49.57	kd	CGS001-10795	ZNF268	Zinc fingers, C2H2-type			
2045	49.57	kd	CGS001-83729	INHBE	-			
2046	49.52	oe	ccsbBroad304_01748	UFD1L	-			
2047	49.52	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
2048	49.47	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
2049	49.46	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
2050	49.45	kd	CGS001-2098	ESD	-			
2051	49.43	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
2052	49.32	kd	CGS001-51545	ZNF581	Zinc fingers, C2H2-type			
2053	49.31	kd	CGS001-3932	LCK	Src family			
2054	49.3	oe	ccsbBroad304_08426	TEX10	-			
2055	49.28	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
2056	49.27	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
2057	49.22	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
2058	49.2	kd	CGS001-8531	CSDA	-			
2059	49.18	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
2060	49.16	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
2061	49.13	oe	ccsbBroad304_03311	EVL	-			
2062	49.12	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
2063	49.1	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
2064	49.05	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
2065	49	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
2066	49	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
2067	48.95	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
2068	48.94	kd	CGS001-11041	B3GNT1	-			
2069	48.9	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
2070	48.9	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
2071	48.87	oe	ccsbBroad304_06976	SMARCE1	-			
2072	48.87	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2073	48.84	kd	CGS001-4856	NOV	-			
2074	48.78	oe	ccsbBroad304_02372	SPRY1	-			
2075	48.78	kd	CGS001-7477	WNT7B	Endogenous ligands			
2076	48.73	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2077	48.72	kd	CGS001-6727	SRP14	-			
2078	48.69	kd	CGS001-154197	PNLDC1	-			
2079	48.64	kd	CGS001-7018	TF	-			
2080	48.63	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
2081	48.63	oe	ccsbBroad304_03853	LSM2	-			
2082	48.54	oe	ccsbBroad304_00995	MECP2	-			
2083	48.51	kd	CGS001-32	ACACB	Carboxylases			
2084	48.46	kd	CGS001-23077	MYCBP2	-			
2085	48.44	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
2086	48.43	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
2087	48.42	kd	CGS001-23466	CBX6	-			
2088	48.38	kd	CGS001-55556	ENOSF1	-			
2089	48.37	oe	ccsbBroad304_01662	TFDP2	-			
2090	48.33	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
2091	48.33	kd	CGS001-3717	JAK2	Janus kinase (JakA) family			
2092	48.32	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
2093	48.26	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
2094	48.23	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
2095	48.23	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
2096	48.21	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
2097	48.18	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
2098	48.16	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
2099	48.13	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
2100	48.12	kd	CGS001-11325	DDX42	DEAD-boxes			
2101	48.11	oe	ccsbBroad304_00551	FECH	-			
2102	48.1	kd	CGS001-114609	TIRAP	-			
2103	48.06	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
2104	48.05	kd	CGS001-4711	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
2105	48.01	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
2106	48	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
2107	47.98	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
2108	47.92	kd	CGS001-2197	FAU	S ribosomal proteins			
2109	47.91	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
2110	47.88	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
2111	47.86	kd	CGS001-10007	GNPDA1	-			
2112	47.82	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
2113	47.8	oe	ccsbBroad304_00832	IFNB1	Interferons			
2114	47.74	kd	CGS001-10613	ERLIN1	-			
2115	47.67	oe	ccsbBroad304_07466	VGLL4	-			
2116	47.67	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
2117	47.6	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
2118	47.58	cp	BRD-K51485625	ritonavir	HIV protease inhibitor		CYP3A4, CYP1A2, CYP2B6, CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
2119	47.58	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
2120	47.55	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
2121	47.5	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
2122	47.43	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
2123	47.41	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
2124	47.39	kd	CGS001-11198	SUPT16H	-			
2125	47.37	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
2126	47.37	kd	CGS001-50	ACO2	-			
2127	47.31	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
2128	47.29	kd	CGS001-6884	TAF13	-			
2129	47.25	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
2130	47.24	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
2131	47.23	kd	CGS001-199704	ZNF585A	Zinc fingers, C2H2-type			
2132	47.21	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
2133	47.21	kd	CGS001-664	BNIP3	-			
2134	47.19	kd	CGS001-84890	ADO	-			
2135	47.17	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
2136	47.15	kd	CGS001-7311	UBA52	L ribosomal proteins			
2137	47.13	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
2138	47.12	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2139	47.12	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
2140	47.08	oe	ccsbBroad304_02203	MAD2L1BP	-			
2141	47.04	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
2142	47.03	cc		Aminoacyl tRNA synthetases class II LOF	-			
2143	47.03	kd	CGS001-2878	GPX3	-			
2144	47.01	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
2145	46.92	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
2146	46.91	oe	ccsbBroad304_03182	GLOD4	-			
2147	46.89	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
2148	46.86	kd	CGS001-8878	SQSTM1	-			
2149	46.85	kd	CGS001-7852	CXCR4	Chemokine receptors			
2150	46.82	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
2151	46.81	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
2152	46.81	kd	CGS001-59286	UBL5	-			
2153	46.8	kd	CGS001-8777	MPDZ	-			
2154	46.76	kd	CGS001-3676	ITGA4	Integrins			
2155	46.76	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
2156	46.76	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
2157	46.73	kd	CGS001-147948	ZNF582	Zinc fingers, C2H2-type			
2158	46.64	kd	CGS001-3161	HMMR	CD molecules			
2159	46.6	kd	CGS001-9709	HERPUD1	-			
2160	46.59	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
2161	46.59	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
2162	46.57	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
2163	46.5	kd	CGS001-149428	BNIPL	-			
2164	46.42	kd	CGS001-3614	IMPDH1	Oxidoreductases			
2165	46.36	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
2166	46.33	kd	CGS001-7982	ST7	-			
2167	46.31	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
2168	46.29	oe	ccsbBroad304_00993	MDM4	-			
2169	46.29	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
2170	46.27	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
2171	46.2	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
2172	46.15	cc		BMP Signaling LOF	-			
2173	46.13	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
2174	46.13	kd	CGS001-3298	HSF2	-			
2175	46.11	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
2176	46.08	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
2177	46.04	kd	CGS001-10769	PLK2	Polo-like kinase (PLK) family			
2178	46.02	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2179	46.02	kd	CGS001-10018	BCL2L11	-			
2180	46.01	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
2181	46	kd	CGS001-5373	PMM2	-			
2182	45.94	kd	CGS001-64121	RRAGC	-			
2183	45.87	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
2184	45.85	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
2185	45.77	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
2186	45.75	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
2187	45.75	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
2188	45.7	oe	ccsbBroad304_05745	CD24	CD molecules			
2189	45.7	kd	CGS001-4067	LYN	Src family			
2190	45.69	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
2191	45.69	kd	CGS001-6257	RXRB	Retinoid X receptors			
2192	45.64	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
2193	45.62	kd	CGS001-55278	QRSL1	-			
2194	45.58	kd	CGS001-9616	RNF7	RING-type (C3HC4) zinc fingers			
2195	45.54	kd	CGS001-1314	COPA	Endogenous ligands			
2196	45.53	kd	CGS001-8536	CAMK1	CAMK1 family			
2197	45.52	kd	CGS001-3669	ISG20	-			
2198	45.45	kd	CGS001-7915	ALDH5A1	Aldehyde dehydrogenases			
2199	45.42	oe	ccsbBroad304_03186	GMNN	-			
2200	45.34	kd	CGS001-10138	YAF2	-			
2201	45.33	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
2202	45.31	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
2203	45.3	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
2204	45.27	kd	CGS001-100	ADA	Adenosine turnover			
2205	45.23	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
2206	45.22	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
2207	45.2	oe	ccsbBroad304_00054	ALDOC	-			
2208	45.14	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
2209	45.14	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
2210	45.14	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
2211	45.12	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
2212	45.12	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
2213	45.09	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
2214	45.06	kd	CGS001-57396	CLK4	CDC-like kinases			
2215	45	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
2216	44.98	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
2217	44.96	oe	ccsbBroad304_14011	PAPSS1	-			
2218	44.93	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
2219	44.86	kd	CGS001-4781	NFIB	-			
2220	44.82	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
2221	44.72	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
2222	44.71	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
2223	44.67	kd	CGS001-5535	PPP3R2	EF-hand domain containing			
2224	44.66	kd	CGS001-1513	CTSK	Cathepsins			
2225	44.59	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
2226	44.54	kd	CGS001-2787	GNG5	-			
2227	44.51	kd	CGS001-6605	SMARCE1	-			
2228	44.41	kd	CGS001-9519	TBPL1	-			
2229	44.37	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
2230	44.37	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
2231	44.34	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
2232	44.29	kd	CGS001-5734	PTGER4	GPCR / Class A : Prostanoid receptors			
2233	44.27	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
2234	44.26	oe	ccsbBroad304_10431	HADHB	-			
2235	44.25	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
2236	44.24	oe	ccsbBroad304_07140	XPC	-			
2237	44.23	oe	ccsbBroad304_01247	POU2AF1	-			
2238	44.18	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
2239	44.17	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
2240	44.17	kd	CGS001-10845	CLPX	ATPases / AAA-type			
2241	44.17	kd	CGS001-408	ARRB1	-			
2242	44.16	kd	CGS001-51292	GMPR2	-			
2243	44.07	oe	ccsbBroad304_08339	CMPK1	-			
2244	44.06	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
2245	44.06	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
2246	44.06	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
2247	44.05	kd	CGS001-7088	TLE1	WD repeat domain containing			
2248	44.03	kd	CGS001-4190	MDH1	-			
2249	44.02	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
2250	44.01	kd	CGS001-174	AFP	-			
2251	43.98	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
2252	43.9	kd	CGS001-4200	ME2	-			
2253	43.88	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
2254	43.88	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
2255	43.87	kd	CGS001-54901	CDKAL1	-			
2256	43.85	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2257	43.84	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
2258	43.8	kd	CGS001-140465	MYL6B	EF-hand domain containing			
2259	43.77	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
2260	43.74	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
2261	43.74	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
2262	43.74	kd	CGS001-151306	GPBAR1	Bile acid receptor			
2263	43.68	kd	CGS001-652	BMP4	Bone morphogenetic proteins			
2264	43.66	kd	CGS001-1997	ELF1	ETS Transcription Factors			
2265	43.66	kd	CGS001-1788	DNMT3A	Methyltransferases			
2266	43.65	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
2267	43.63	kd	CGS001-5479	PPIB	-			
2268	43.61	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
2269	43.6	kd	CGS001-9133	CCNB2	-			
2270	43.6	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
2271	43.56	kd	CGS001-10969	EBNA1BP2	-			
2272	43.54	cc		HIV protease inhibitor	-			
2273	43.54	kd	CGS001-10298	PAK4	PAKB subfamily			
2274	43.52	cc		P38 MAPK inhibitor	-			
2275	43.52	kd	CGS001-7343	UBTF	-			
2276	43.51	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
2277	43.5	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2278	43.37	kd	CGS001-2783	GNB2	WD repeat domain containing			
2279	43.36	kd	CGS001-1738	DLD	-			
2280	43.32	kd	CGS001-262	AMD1	Decarboxylases			
2281	43.3	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
2282	43.27	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
2283	43.15	oe	ccsbBroad304_00313	TBCB	-			
2284	43.15	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
2285	43.11	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
2286	43.07	kd	CGS001-10437	IFI30	-			
2287	43	oe	ccsbBroad304_07217	AXIN2	-			
2288	42.98	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
2289	42.96	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
2290	42.95	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
2291	42.92	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
2292	42.89	kd	CGS001-6046	BRD2	Bromodomain kinase (BRDK) family			
2293	42.87	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
2294	42.87	oe	ccsbBroad304_02143	CNOT8	-			
2295	42.85	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
2296	42.85	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
2297	42.82	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
2298	42.79	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
2299	42.77	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
2300	42.75	cc		Wnt family LOF	-			
2301	42.75	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
2302	42.72	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
2303	42.71	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
2304	42.6	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
2305	42.54	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
2306	42.47	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
2307	42.44	kd	CGS001-83737	ITCH	-			
2308	42.37	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
2309	42.36	kd	CGS001-162655	ZNF519	Zinc fingers, C2H2-type			
2310	42.35	oe	ccsbBroad304_14047	TACC3	-			
2311	42.29	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
2312	42.25	kd	CGS001-4316	MMP7	Matrix metallopeptidase			
2313	42.24	kd	CGS001-79733	E2F8	-			
2314	42.21	kd	CGS001-2876	GPX1	-			
2315	42.19	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2316	42.18	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
2317	42.17	kd	CGS001-5699	PSMB10	Proteasome (prosome, macropain) subunits			
2318	42.16	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
2319	42.11	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
2320	42.11	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
2321	42.08	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
2322	42.01	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
2323	42.01	kd	CGS001-3672	ITGA1	Integrins			
2324	42	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
2325	42	kd	CGS001-467	ATF3	basic leucine zipper proteins			
2326	41.96	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
2327	41.92	kd	CGS001-290	ANPEP	Aminopeptidase N			
2328	41.89	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
2329	41.89	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
2330	41.87	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
2331	41.87	kd	CGS001-11157	LSM6	-			
2332	41.86	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
2333	41.84	kd	CGS001-7528	YY1	INO80 complex subunits			
2334	41.82	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
2335	41.82	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2336	41.8	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
2337	41.79	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
2338	41.76	kd	CGS001-7337	UBE3A	-			
2339	41.75	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
2340	41.72	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
2341	41.7	oe	ccsbBroad304_05981	CDO1	-			
2342	41.63	oe	ccsbBroad304_03444	PAF1	-			
2343	41.62	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
2344	41.61	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2345	41.56	oe	ccsbBroad304_07097	TRAF1	-			
2346	41.53	kd	CGS001-8800	PEX11A	-			
2347	41.51	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
2348	41.49	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
2349	41.48	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
2350	41.47	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
2351	41.44	kd	CGS001-817	CAMK2D	CAMK2 family			
2352	41.4	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
2353	41.35	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
2354	41.35	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
2355	41.25	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
2356	41.23	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
2357	41.23	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
2358	41.23	kd	CGS001-11336	EXOC3	-			
2359	41.17	oe	ccsbBroad304_08325	LIPT1	-			
2360	41.16	kd	CGS001-11257	TP53TG1	-			
2361	41.08	kd	CGS001-3551	IKBKB	IKK family			
2362	41.06	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
2363	41.06	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
2364	41.05	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
2365	41.03	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
2366	41.02	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
2367	40.99	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
2368	40.98	kd	CGS001-29946	SERTAD3	-			
2369	40.97	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
2370	40.94	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
2371	40.81	oe	ccsbBroad304_00854	IL8	-			
2372	40.77	oe	ccsbBroad304_08045	NOX1	-			
2373	40.68	oe	ccsbBroad304_12008	NLK	nmo subfamily			
2374	40.68	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
2375	40.66	oe	ccsbBroad304_02845	PRPF6	-			
2376	40.65	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
2377	40.56	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
2378	40.56	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
2379	40.54	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
2380	40.53	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
2381	40.52	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
2382	40.51	kd	CGS001-4734	NEDD4	-			
2383	40.48	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
2384	40.46	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
2385	40.41	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
2386	40.38	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
2387	40.34	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
2388	40.26	kd	CGS001-1211	CLTA	-			
2389	40.25	kd	CGS001-10253	SPRY2	-			
2390	40.24	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
2391	40.23	kd	CGS001-624	BDKRB2	Bradykinin receptors			
2392	40.21	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
2393	40.21	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
2394	40.18	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
2395	40.15	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
2396	40.12	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
2397	40.11	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
2398	40.09	kd	CGS001-4616	GADD45B	-			
2399	40.05	kd	CGS001-3920	LAMP2	CD molecules			
2400	39.99	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
2401	39.99	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
2402	39.99	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
2403	39.98	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
2404	39.96	kd	CGS001-11315	PARK7	Parkinson disease			
2405	39.96	kd	CGS001-4707	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
2406	39.94	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
2407	39.93	kd	CGS001-8569	MKNK1	MKN subfamily			
2408	39.91	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
2409	39.89	kd	CGS001-5442	POLRMT	-			
2410	39.86	kd	CGS001-6883	TAF12	-			
2411	39.8	cp	BRD-K59753975	vindesine	Tubulin inhibitor		TUBB, TUBB1	Tubulin inhibitor
2412	39.79	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
2413	39.74	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
2414	39.72	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
2415	39.68	kd	CGS001-7428	VHL	-			
2416	39.65	kd	CGS001-90655	TGIF2LY	Homeoboxes / TALE class			
2417	39.64	kd	CGS001-10810	WASF3	-			
2418	39.63	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
2419	39.63	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
2420	39.62	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
2421	39.6	kd	CGS001-351	APP	Endogenous ligands			
2422	39.59	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
2423	39.59	oe	ccsbBroad304_10212	GRHL3	-			
2424	39.56	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
2425	39.56	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
2426	39.55	kd	CGS001-57661	PHRF1	Zinc fingers, PHD-type			
2427	39.55	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
2428	39.54	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
2429	39.5	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
2430	39.49	kd	CGS001-26277	TINF2	-			
2431	39.47	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
2432	39.45	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
2433	39.45	kd	CGS001-5986	RFNG	Beta 3-glycosyltransferases			
2434	39.44	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
2435	39.36	kd	CGS001-811	CALR	-			
2436	39.35	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
2437	39.29	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
2438	39.29	kd	CGS001-26271	FBXO5	F-boxes / other			
2439	39.29	kd	CGS001-718	C3	Endogenous ligands			
2440	39.27	oe	ccsbBroad304_01257	PPOX	-			
2441	39.27	oe	ccsbBroad304_00179	BTG1	-			
2442	39.26	kd	CGS001-5048	PAFAH1B1	WD repeat domain containing			
2443	39.25	kd	CGS001-257397	TAB3	-			
2444	39.25	kd	CGS001-4942	OAT	-			
2445	39.23	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
2446	39.23	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
2447	39.21	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
2448	39.19	oe	ccsbBroad304_02633	LSM6	-			
2449	39.18	kd	CGS001-10214	SSX3	-			
2450	39.17	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
2451	39.16	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
2452	39.15	kd	CGS001-822	CAPG	-			
2453	39.14	oe	ccsbBroad304_08802	ELAC2	-			
2454	39.07	kd	CGS001-23658	LSM5	-			
2455	39.04	kd	CGS001-727	C5	Endogenous ligands			
2456	39.03	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
2457	39.02	kd	CGS001-2976	GTF3C2	General transcription factors			
2458	38.99	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
2459	38.98	kd	CGS001-9474	ATG5	-			
2460	38.96	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
2461	38.93	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
2462	38.92	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
2463	38.91	kd	CGS001-5269	SERPINB6	Serine (or cysteine) peptidase inhibitors			
2464	38.91	kd	CGS001-3054	HCFC1	-			
2465	38.77	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
2466	38.71	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
2467	38.7	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
2468	38.67	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
2469	38.66	kd	CGS001-9761	MLEC	-			
2470	38.65	oe	ccsbBroad304_06292	GNAI2	-			
2471	38.61	oe	ccsbBroad304_05590	NOTCH2NL	-			
2472	38.6	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
2473	38.6	kd	CGS001-6514	SLC2A2	Solute carriers			
2474	38.58	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
2475	38.53	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
2476	38.52	kd	CGS001-673	BRAF	RAF family			
2477	38.5	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
2478	38.48	kd	CGS001-81848	SPRY4	-			
2479	38.47	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
2480	38.45	oe	ccsbBroad304_11405	UBE3C	-			
2481	38.44	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
2482	38.42	kd	CGS001-891	CCNB1	-			
2483	38.41	kd	CGS001-10651	MTX2	-			
2484	38.4	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
2485	38.4	kd	CGS001-10284	SAP18	-			
2486	38.39	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
2487	38.38	kd	CGS001-6658	SOX3	SRY (sex determining region Y)-boxes			
2488	38.38	kd	CGS001-51022	GLRX2	-			
2489	38.37	kd	CGS001-1632	ECI1	-			
2490	38.35	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
2491	38.33	kd	CGS001-5744	PTHLH	Endogenous ligands			
2492	38.33	kd	CGS001-275	AMT	-			
2493	38.28	kd	CGS001-472	ATM	Other PIKK family kinases			
2494	38.27	cc		Bacterial DNA gyrase inhibitor	-			
2495	38.26	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
2496	38.23	kd	CGS001-5202	PFDN2	-			
2497	38.18	oe	ccsbBroad304_02217	FEZ1	-			
2498	38.14	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
2499	38.07	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
2500	38.07	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2501	38.06	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
2502	38.02	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
2503	37.99	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
2504	37.99	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
2505	37.96	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
2506	37.95	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
2507	37.94	kd	CGS001-2101	ESRRA	Estrogen-related receptors			
2508	37.93	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
2509	37.92	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
2510	37.92	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
2511	37.83	oe	ccsbBroad304_00447	DLD	-			
2512	37.82	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
2513	37.82	kd	CGS001-4594	MUT	-			
2514	37.82	kd	CGS001-2077	ERF	ETS Transcription Factors			
2515	37.81	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
2516	37.8	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
2517	37.77	cp	BRD-A49172652	lansoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4, CYP3A5	ATPase inhibitor
2518	37.67	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
2519	37.62	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
2520	37.61	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
2521	37.57	kd	CGS001-3776	KCNK2	Two-P potassium channels			
2522	37.53	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
2523	37.51	kd	CGS001-2710	GK	Glycerol kinases			
2524	37.5	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
2525	37.43	kd	CGS001-210	ALAD	-			
2526	37.34	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
2527	37.33	kd	CGS001-6932	TCF7	-			
2528	37.27	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
2529	37.27	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
2530	37.27	kd	CGS001-4234	METTL1	-			
2531	37.24	kd	CGS001-54205	CYCS	-			
2532	37.21	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
2533	37.2	kd	CGS001-9988	DMTF1	-			
2534	37.14	kd	CGS001-4860	PNP	-			
2535	37.13	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2536	37.13	kd	CGS001-2184	FAH	-			
2537	37.12	kd	CGS001-3066	HDAC2	Histone deacetylases			
2538	37.11	kd	CGS001-8655	DYNLL1	Cytoplasmic dyneins			
2539	37.07	oe	ccsbBroad304_00036	AFP	-			
2540	37.05	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
2541	37.04	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
2542	37.03	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
2543	36.99	oe	ccsbBroad304_06420	ICAM3	CD molecules			
2544	36.99	oe	ccsbBroad304_04655	TRIM9	-			
2545	36.99	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
2546	36.99	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
2547	36.98	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
2548	36.97	cp	BRD-A11990600	lorazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, TSPO	Benzodiazepine receptor agonist
2549	36.92	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
2550	36.92	kd	CGS001-57657	HCN3	Cyclic nucleotide-regulated channels			
2551	36.92	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
2552	36.9	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
2553	36.89	oe	ccsbBroad304_02869	ASF1A	-			
2554	36.88	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
2555	36.86	kd	CGS001-11142	PKIG	-			
2556	36.82	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
2557	36.81	kd	CGS001-7374	UNG	-			
2558	36.79	oe	ccsbBroad304_00615	GAPDH	-			
2559	36.74	kd	CGS001-10755	GIPC1	-			
2560	36.73	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
2561	36.73	kd	CGS001-3176	HNMT	-			
2562	36.7	oe	ccsbBroad304_00106	ARRB1	-			
2563	36.69	cc		V type ATPases LOF	-			
2564	36.68	kd	CGS001-64858	DCLRE1B	-			
2565	36.66	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
2566	36.59	oe	ccsbBroad304_00550	FDXR	-			
2567	36.57	kd	CGS001-708	C1QBP	-			
2568	36.49	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
2569	36.43	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
2570	36.43	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
2571	36.42	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
2572	36.39	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
2573	36.38	oe	ccsbBroad304_02837	BHMT2	-			
2574	36.36	oe	ccsbBroad304_04153	PHF17	-			
2575	36.36	kd	CGS001-2729	GCLC	-			
2576	36.35	kd	CGS001-83593	RASSF5	-			
2577	36.33	kd	CGS001-2277	FIGF	-			
2578	36.26	oe	ccsbBroad304_00164	BLMH	-			
2579	36.21	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
2580	36.21	kd	CGS001-1756	DMD	-			
2581	36.18	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
2582	36.16	kd	CGS001-8900	CCNA1	-			
2583	36.12	kd	CGS001-23242	COBL	-			
2584	36.06	kd	CGS001-11151	CORO1A	Coronins			
2585	36.05	kd	CGS001-150094	SIK1	QIK subfamily			
2586	36.05	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
2587	35.99	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
2588	35.93	kd	CGS001-898	CCNE1	-			
2589	35.92	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
2590	35.91	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
2591	35.91	kd	CGS001-54472	TOLLIP	-			
2592	35.91	kd	CGS001-8505	PARG	-			
2593	35.9	kd	CGS001-9697	TRAM2	-			
2594	35.85	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
2595	35.85	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
2596	35.82	kd	CGS001-5361	PLXNA1	Plexins			
2597	35.76	oe	ccsbBroad304_00624	GCK	Hexokinases			
2598	35.76	kd	CGS001-54881	TEX10	-			
2599	35.72	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
2600	35.69	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
2601	35.68	kd	CGS001-1070	CETN3	EF-hand domain containing			
2602	35.6	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2603	35.58	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2604	35.56	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
2605	35.51	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
2606	35.43	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
2607	35.41	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
2608	35.39	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
2609	35.37	kd	CGS001-4700	NDUFA6	LYR motif containing			
2610	35.32	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
2611	35.31	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
2612	35.3	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
2613	35.3	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
2614	35.25	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
2615	35.25	kd	CGS001-2987	GUK1	-			
2616	35.24	kd	CGS001-8522	GAS7	-			
2617	35.21	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
2618	35.21	kd	CGS001-5004	ORM1	Lipocalins			
2619	35.2	kd	CGS001-3685	ITGAV	Integrins			
2620	35.19	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2621	35.18	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
2622	35.17	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
2623	35.15	kd	CGS001-5624	PROC	Endogenous ligands			
2624	35.13	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
2625	35.09	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
2626	35.05	kd	CGS001-5515	PPP2CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2627	35.04	kd	CGS001-5576	PRKAR2A	Protein kinase A			
2628	35.03	kd	CGS001-118442	GPR62	GPCR / Class A : Orphans			
2629	35.02	kd	CGS001-2767	GNA11	-			
2630	35.01	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
2631	34.95	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
2632	34.9	oe	ccsbBroad304_12106	PXK	Slob family			
2633	34.89	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
2634	34.87	kd	CGS001-51070	NOSIP	-			
2635	34.85	oe	ccsbBroad304_06435	RBPJ	-			
2636	34.85	kd	CGS001-2778	GNAS	-			
2637	34.82	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
2638	34.81	kd	CGS001-4946	OAZ1	-			
2639	34.78	kd	CGS001-2542	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
2640	34.75	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
2641	34.73	kd	CGS001-164091	PAQR7	-			
2642	34.69	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2643	34.69	kd	CGS001-7484	WNT9B	Wingless-type MMTV integration sites			
2644	34.61	kd	CGS001-3376	IARS	Aminoacyl tRNA synthetases / Class I			
2645	34.55	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2646	34.54	kd	CGS001-1869	E2F1	-			
2647	34.52	cp	BRD-K06878038	deferiprone	Chelating agent		CYP4F2	Chelating agent
2648	34.51	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
2649	34.5	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
2650	34.48	oe	ccsbBroad304_02653	PRAF2	-			
2651	34.46	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
2652	34.42	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
2653	34.39	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
2654	34.38	kd	CGS001-5723	PSPH	-			
2655	34.37	cp	BRD-K66206289	lobeline	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist
2656	34.36	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
2657	34.35	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
2658	34.25	cp	BRD-K82357231	desloratadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2659	34.24	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
2660	34.22	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
2661	34.21	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
2662	34.17	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
2663	34.15	oe	ccsbBroad304_06386	HNMT	-			
2664	34.13	kd	CGS001-2565	GABRG1	GABA receptors			
2665	34.05	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
2666	34.04	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
2667	34.02	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
2668	34.01	kd	CGS001-8148	TAF15	RNA binding motif (RRM) containing			
2669	33.99	kd	CGS001-2828	GPR4	GPCR / Class A : Orphans			
2670	33.98	kd	CGS001-8634	RTCD1	-			
2671	33.93	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
2672	33.92	kd	CGS001-11284	PNKP	-			
2673	33.92	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
2674	33.91	kd	CGS001-23743	BHMT2	-			
2675	33.9	oe	ccsbBroad304_00645	GCLM	-			
2676	33.85	oe	ccsbBroad304_00665	GOT1	-			
2677	33.81	kd	CGS001-1977	EIF4E	Translation Initiation Factor 4E			
2678	33.79	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2679	33.79	kd	CGS001-2512	FTL	-			
2680	33.78	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
2681	33.76	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
2682	33.75	oe	ccsbBroad304_07569	TRIB1	Trbl family			
2683	33.75	kd	CGS001-230	ALDOC	-			
2684	33.74	kd	CGS001-4193	MDM2	-			
2685	33.71	cc		Aurora kinase inhibitor	-			
2686	33.71	kd	CGS001-23192	ATG4B	Aut2 peptidase			
2687	33.7	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
2688	33.68	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
2689	33.68	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
2690	33.68	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
2691	33.67	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2692	33.66	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
2693	33.66	kd	CGS001-133690	CAPSL	EF-hand domain containing			
2694	33.65	kd	CGS001-8767	RIPK2	Receptor interacting protein kinase (RIPK) family			
2695	33.63	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
2696	33.59	kd	CGS001-10991	SLC38A3	System N-like transporters			
2697	33.56	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
2698	33.55	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
2699	33.52	kd	CGS001-9891	NUAK1	NuaK subfamily			
2700	33.51	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
2701	33.48	oe	ccsbBroad304_06720	PHYH	-			
2702	33.46	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
2703	33.45	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
2704	33.43	kd	CGS001-1287	COL4A5	Collagens			
2705	33.41	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
2706	33.41	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
2707	33.41	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
2708	33.34	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
2709	33.31	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
2710	33.26	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
2711	33.25	kd	CGS001-50865	HEBP1	Endogenous ligands			
2712	33.19	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
2713	33.18	kd	CGS001-9898	UBAP2L	-			
2714	33.15	kd	CGS001-597	BCL2A1	-			
2715	33.1	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
2716	33.04	kd	CGS001-4795	NFKBIL1	-			
2717	33.02	kd	CGS001-7421	VDR	Vitamin D receptors			
2718	32.96	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
2719	32.93	oe	ccsbBroad304_03129	ERO1L	-			
2720	32.93	oe	ccsbBroad304_01960	CASK	CASK family			
2721	32.92	cc		Lysine acetyltransferases LOF	-			
2722	32.91	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
2723	32.9	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
2724	32.88	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
2725	32.84	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
2726	32.84	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
2727	32.83	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
2728	32.77	oe	ccsbBroad304_03122	RHOD	-			
2729	32.77	kd	CGS001-7297	TYK2	Janus kinase (JakA) family			
2730	32.76	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2731	32.75	kd	CGS001-148327	CREB3L4	basic leucine zipper proteins			
2732	32.65	kd	CGS001-2145	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
2733	32.64	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
2734	32.64	kd	CGS001-23635	SSBP2	-			
2735	32.64	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
2736	32.63	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2737	32.63	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
2738	32.54	kd	CGS001-392	ARHGAP1	Rho GTPase activating proteins			
2739	32.53	kd	CGS001-4837	NNMT	-			
2740	32.52	kd	CGS001-6829	SUPT5H	-			
2741	32.51	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
2742	32.48	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
2743	32.48	kd	CGS001-6461	SHB	SH2 domain containing			
2744	32.48	kd	CGS001-114785	MBD6	-			
2745	32.45	oe	ccsbBroad304_06870	RNH1	-			
2746	32.44	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
2747	32.42	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
2748	32.42	kd	CGS001-3638	INSIG1	-			
2749	32.39	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
2750	32.38	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2751	32.33	oe	ccsbBroad304_00147	BAG1	-			
2752	32.27	kd	CGS001-5932	RBBP8	-			
2753	32.24	kd	CGS001-7879	RAB7A	RAB, member RAS oncogene			
2754	32.24	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
2755	32.21	kd	CGS001-115201	ATG4A	-			
2756	32.2	kd	CGS001-9213	XPR1	-			
2757	32.18	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
2758	32.16	cc		SRY LOF	-			
2759	32.15	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
2760	32.1	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
2761	32.1	kd	CGS001-6285	S100B	EF-hand domain containing			
2762	32.05	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
2763	32.05	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
2764	32.04	kd	CGS001-1903	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
2765	32.03	oe	ccsbBroad304_03357	RASD1	-			
2766	32.01	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
2767	32.01	kd	CGS001-6199	RPS6KB2	p70 subfamily			
2768	32.01	kd	CGS001-5194	PEX13	-			
2769	32	kd	CGS001-10135	NAMPT	-			
2770	31.99	cc		Norepinephrine reuptake inhibitor	-			
2771	31.99	kd	CGS001-1212	CLTB	-			
2772	31.92	kd	CGS001-6663	SOX10	SRY (sex determining region Y)-boxes			
2773	31.92	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
2774	31.91	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
2775	31.91	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
2776	31.91	kd	CGS001-3046	HBE1	-			
2777	31.87	kd	CGS001-3675	ITGA3	Integrins			
2778	31.86	kd	CGS001-336	APOA2	Apolipoproteins			
2779	31.84	kd	CGS001-1399	CRKL	SH2 domain containing			
2780	31.82	kd	CGS001-7345	UCHL1	Ubiquitin C-terminal hydrolase			
2781	31.79	kd	CGS001-6720	SREBF1	Basic helix-loop-helix proteins			
2782	31.78	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
2783	31.75	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
2784	31.7	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
2785	31.69	kd	CGS001-9443	MED7	-			
2786	31.69	kd	CGS001-57007	CXCR7	-			
2787	31.66	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
2788	31.65	oe	ccsbBroad304_07727	LIAS	-			
2789	31.65	oe	ccsbBroad304_06535	LPL	-			
2790	31.6	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
2791	31.59	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
2792	31.57	kd	CGS001-1659	DHX8	DEAH-boxes			
2793	31.55	oe	ccsbBroad304_02502	GNA13	-			
2794	31.54	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
2795	31.52	kd	CGS001-6286	S100P	EF-hand domain containing			
2796	31.52	kd	CGS001-5689	PSMB1	Proteasome subunits			
2797	31.51	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
2798	31.5	kd	CGS001-171017	ZNF384	Zinc fingers, C2H2-type			
2799	31.42	oe	ccsbBroad304_02884	POT1	-			
2800	31.35	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
2801	31.35	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2802	31.31	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
2803	31.3	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2804	31.25	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
2805	31.2	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
2806	31.19	kd	CGS001-390980	ZNF805	Zinc fingers, C2H2-type			
2807	31.16	oe	ccsbBroad304_02501	DCTN6	-			
2808	31.16	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
2809	31.11	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
2810	31.05	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
2811	31.05	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
2812	31.05	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
2813	31	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
2814	31	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
2815	31	kd	CGS001-4668	NAGA	-			
2816	30.99	kd	CGS001-94234	FOXQ1	Forkhead boxes			
2817	30.98	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
2818	30.98	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
2819	30.97	kd	CGS001-3690	ITGB3	Integrins			
2820	30.97	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2821	30.95	kd	CGS001-7431	VIM	Intermediate filaments type III			
2822	30.93	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
2823	30.93	kd	CGS001-1028	CDKN1C	-			
2824	30.93	kd	CGS001-901	CCNG2	-			
2825	30.92	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
2826	30.91	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
2827	30.89	kd	CGS001-399664	MEX3D	Mex-3 homologs			
2828	30.87	oe	ccsbBroad304_09615	LACC1	-			
2829	30.87	kd	CGS001-23013	SPEN	RNA binding motif (RRM) containing			
2830	30.86	kd	CGS001-7159	TP53BP2	Ankyrin repeat domain containing			
2831	30.85	cc		Cyclooxygenase inhibitor	-			
2832	30.83	kd	CGS001-22938	SNW1	-			
2833	30.81	kd	CGS001-6887	TAL2	Basic helix-loop-helix proteins			
2834	30.8	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
2835	30.78	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
2836	30.76	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
2837	30.75	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
2838	30.74	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
2839	30.72	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
2840	30.63	kd	CGS001-10295	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
2841	30.61	kd	CGS001-5336	PLCG2	Phosphoinositide-specific phospholipase C			
2842	30.59	oe	ccsbBroad304_06862	RGS3	-			
2843	30.58	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
2844	30.54	cc		TGF beta receptor inhibitor	-			
2845	30.49	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
2846	30.48	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
2847	30.46	kd	CGS001-6632	SNRPD1	-			
2848	30.44	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
2849	30.42	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
2850	30.42	kd	CGS001-2597	GAPDH	-			
2851	30.41	oe	ccsbBroad304_00155	CCND1	-			
2852	30.36	cc		FLT3 inhibitor	-			
2853	30.3	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
2854	30.29	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
2855	30.28	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
2856	30.28	kd	CGS001-2806	GOT2	-			
2857	30.26	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
2858	30.25	oe	ccsbBroad304_02231	USP6NL	-			
2859	30.22	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2860	30.21	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
2861	30.21	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
2862	30.21	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
2863	30.16	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
2864	30.15	kd	CGS001-57521	RPTOR	WD repeat domain containing			
2865	30.14	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
2866	30.11	kd	CGS001-670	BPHL	-			
2867	30.1	kd	CGS001-27034	ACAD8	-			
2868	30.09	oe	ccsbBroad304_00174	BRAF	RAF family			
2869	30.06	kd	CGS001-7466	WFS1	-			
2870	30.05	kd	CGS001-11343	MGLL	Endocannabinoid turnover			
2871	30.04	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
2872	30.04	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
2873	29.94	kd	CGS001-10554	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
2874	29.87	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
2875	29.82	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
2876	29.78	kd	CGS001-4172	MCM3	-			
2877	29.77	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
2878	29.74	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2879	29.72	oe	ccsbBroad304_02497	YKT6	-			
2880	29.72	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
2881	29.72	kd	CGS001-7089	TLE2	WD repeat domain containing			
2882	29.62	cc		Imidazoline ligand	-			
2883	29.61	kd	CGS001-170591	S100Z	EF-hand domain containing			
2884	29.58	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
2885	29.58	kd	CGS001-776	CACNA1D	Calcium channel subunits			
2886	29.53	kd	CGS001-5966	REL	NFkappaB transcription factor family			
2887	29.52	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
2888	29.51	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
2889	29.47	oe	ccsbBroad304_07208	NRIP1	-			
2890	29.47	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
2891	29.45	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
2892	29.45	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
2893	29.4	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
2894	29.4	kd	CGS001-64175	LEPRE1	-			
2895	29.39	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
2896	29.34	kd	CGS001-4090	SMAD5	SMADs			
2897	29.29	cc		HRH1 antagonist	-			
2898	29.27	kd	CGS001-2073	ERCC5	-			
2899	29.24	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
2900	29.22	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
2901	29.21	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
2902	29.19	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
2903	29.18	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
2904	29.14	oe	ccsbBroad304_04786	CANT1	-			
2905	29.14	kd	CGS001-4552	MTRR	-			
2906	29.13	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2907	29.11	kd	CGS001-89765	RSPH1	-			
2908	29.05	kd	CGS001-10472	ZNF238	-			
2909	29.05	kd	CGS001-30	ACAA1	-			
2910	28.99	kd	CGS001-4048	LTA4H	Hydrolases			
2911	28.96	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
2912	28.94	oe	ccsbBroad304_07605	LYPLA1	-			
2913	28.93	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
2914	28.93	kd	CGS001-4282	MIF	-			
2915	28.92	oe	ccsbBroad304_07890	CBX7	-			
2916	28.87	cc		Sirtuins GOF	-			
2917	28.84	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
2918	28.83	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
2919	28.81	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
2920	28.81	oe	ccsbBroad304_02425	CDIPT	-			
2921	28.8	kd	CGS001-8859	STK19	G11 family			
2922	28.76	kd	CGS001-4708	NDUFB2	Mitochondrial respiratory chain complex / Complex I			
2923	28.75	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
2924	28.75	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
2925	28.74	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
2926	28.72	cc		NFkB pathway inhibitor	-			
2927	28.72	kd	CGS001-23384	SPECC1L	-			
2928	28.69	cc		General transcription factors group 2 LOF	-			
2929	28.64	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
2930	28.62	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
2931	28.59	kd	CGS001-10059	DNM1L	-			
2932	28.58	kd	CGS001-310	ANXA7	Annexins			
2933	28.56	kd	CGS001-5264	PHYH	-			
2934	28.54	kd	CGS001-2138	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2935	28.53	oe	ccsbBroad304_08645	BCCIP	-			
2936	28.52	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
2937	28.51	kd	CGS001-79960	PHF17	-			
2938	28.48	kd	CGS001-4811	NID1	-			
2939	28.48	kd	CGS001-3488	IGFBP5	insulin-like growth factor (IGF) binding proteins			
2940	28.48	kd	CGS001-2747	GLUD2	-			
2941	28.42	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
2942	28.42	kd	CGS001-11007	CCDC85B	-			
2943	28.23	kd	CGS001-444	ASPH	-			
2944	28.22	kd	CGS001-55718	POLR3E	RNA polymerase subunits			
2945	28.2	kd	CGS001-64219	PJA1	RING-type (C3HC4) zinc fingers			
2946	28.19	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
2947	28.19	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
2948	28.17	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
2949	28.16	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
2950	28.16	kd	CGS001-9252	RPS6KA5	MSK subfamily			
2951	28.09	kd	CGS001-1026	CDKN1A	-			
2952	28.02	kd	CGS001-10123	ARL4C	ADP-ribosylation factors			
2953	28	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
2954	28	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
2955	27.98	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
2956	27.97	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
2957	27.86	kd	CGS001-8573	CASK	CASK family			
2958	27.78	kd	CGS001-5025	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
2959	27.77	cc		Interleukins GOF	-			
2960	27.76	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
2961	27.72	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
2962	27.71	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
2963	27.7	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
2964	27.66	kd	CGS001-2963	GTF2F2	General transcription factors			
2965	27.58	kd	CGS001-2872	MKNK2	MKN subfamily			
2966	27.55	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
2967	27.52	kd	CGS001-6732	SRPK1	SRPK family			
2968	27.51	kd	CGS001-84775	ZNF607	Zinc fingers, C2H2-type			
2969	27.5	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
2970	27.5	kd	CGS001-283450	C12ORF51	-			
2971	27.42	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
2972	27.38	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
2973	27.36	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
2974	27.33	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
2975	27.33	kd	CGS001-883	CCBL1	Hydrogen sulphide synthesis			
2976	27.31	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
2977	27.31	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
2978	27.3	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
2979	27.29	kd	CGS001-388	RHOB	-			
2980	27.26	cp	BRD-A94543220	bifonazole	Sterol demethylase inhibitor		CYP2B6	Sterol demethylase inhibitor
2981	27.25	kd	CGS001-65263	PYCRL	-			
2982	27.2	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
2983	27.17	kd	CGS001-10476	ATP5H	ATPases / F-type			
2984	27.05	kd	CGS001-1861	TOR1A	-			
2985	27.04	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2986	27.04	oe	ccsbBroad304_02578	EBNA1BP2	-			
2987	27.03	oe	ccsbBroad304_08888	ACD	-			
2988	27.02	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
2989	27	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
2990	26.97	kd	CGS001-25898	RCHY1	RING-type (C3HC4) zinc fingers			
2991	26.97	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
2992	26.93	kd	CGS001-10308	ZNF267	Zinc fingers, C2H2-type			
2993	26.93	kd	CGS001-400	ARL1	ADP-ribosylation factors			
2994	26.91	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
2995	26.91	kd	CGS001-5538	PPT1	-			
2996	26.9	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
2997	26.85	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
2998	26.82	kd	CGS001-515	ATP5F1	ATPases / F-type			
2999	26.78	kd	CGS001-9967	THRAP3	-			
3000	26.77	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
3001	26.76	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
3002	26.76	oe	ccsbBroad304_04752	IKBIP	-			
3003	26.76	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
3004	26.76	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
3005	26.75	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
3006	26.72	oe	ccsbBroad304_03113	DSE	-			
3007	26.69	cc		Cyclins LOF	-			
3008	26.68	oe	ccsbBroad304_07362	NMI	-			
3009	26.64	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
3010	26.63	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
3011	26.58	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
3012	26.56	kd	CGS001-51290	ERGIC2	-			
3013	26.55	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
3014	26.54	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
3015	26.54	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
3016	26.53	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3017	26.52	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
3018	26.51	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
3019	26.51	kd	CGS001-5110	PCMT1	-			
3020	26.49	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
3021	26.49	kd	CGS001-29982	NRBF2	-			
3022	26.44	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
3023	26.42	kd	CGS001-7003	TEAD1	-			
3024	26.41	oe	ccsbBroad304_01519	SET	-			
3025	26.41	kd	CGS001-9231	DLG5	-			
3026	26.31	kd	CGS001-64094	SMOC2	EF-hand domain containing			
3027	26.3	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3028	26.3	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
3029	26.21	kd	CGS001-9441	MED26	-			
3030	26.15	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
3031	26.15	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
3032	26.14	kd	CGS001-350	APOH	Apolipoproteins			
3033	26.02	cp	BRD-K88304388	dextrorphan	Glutamate receptor antagonist		OPRM1, OPRK1, OPRD1, GRIN1, HTR1A, SLC6A2	Glutamate receptor antagonist
3034	25.99	kd	CGS001-51447	IP6K2	-			
3035	25.97	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
3036	25.96	kd	CGS001-378	ARF4	ADP-ribosylation factors			
3037	25.95	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
3038	25.92	kd	CGS001-80762	NDFIP1	-			
3039	25.91	kd	CGS001-9869	SETDB1	Histone methyltransferases (HMTs)			
3040	25.87	kd	CGS001-3127	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
3041	25.86	oe	ccsbBroad304_07337	TAF1B	-			
3042	25.86	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
3043	25.84	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
3044	25.84	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
3045	25.84	kd	CGS001-3664	IRF6	-			
3046	25.81	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
3047	25.8	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
3048	25.79	oe	ccsbBroad304_06264	GBP2	-			
3049	25.77	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
3050	25.74	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
3051	25.71	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
3052	25.7	kd	CGS001-10775	POP4	-			
3053	25.69	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
3054	25.67	kd	CGS001-170463	SSBP4	-			
3055	25.64	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
3056	25.64	kd	CGS001-1376	CPT2	-			
3057	25.64	kd	CGS001-826	CAPNS1	EF-hand domain containing			
3058	25.62	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
3059	25.62	kd	CGS001-3718	JAK3	Janus kinase (JakA) family			
3060	25.61	kd	CGS001-5573	PRKAR1A	Protein kinase A			
3061	25.53	kd	CGS001-533	ATP6V0B	ATPases / V-type			
3062	25.49	kd	CGS001-2100	ESR2	Estrogen receptors			
3063	25.48	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
3064	25.46	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
3065	25.45	oe	ccsbBroad304_06639	NFYB	-			
3066	25.42	oe	ccsbBroad304_02534	UTP14A	-			
3067	25.41	kd	CGS001-6307	MSMO1	Fatty acid hydroxylase domain containing			
3068	25.4	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
3069	25.4	kd	CGS001-9319	TRIP13	ATPases / AAA-type			
3070	25.39	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
3071	25.39	kd	CGS001-80777	CYB5B	-			
3072	25.29	kd	CGS001-7342	UBP1	-			
3073	25.29	kd	CGS001-10254	STAM2	-			
3074	25.27	kd	CGS001-4665	NAB2	-			
3075	25.2	kd	CGS001-116113	FOXP4	Forkhead boxes			
3076	25.19	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
3077	25.17	kd	CGS001-2353	FOS	basic leucine zipper proteins			
3078	25.16	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
3079	25.16	kd	CGS001-6259	RYK	Type XV RTKs: RYK			
3080	25.1	oe	ccsbBroad304_03415	GFOD1	-			
3081	25.08	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
3082	25.06	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
3083	25.05	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
3084	25.04	kd	CGS001-5982	RFC2	ATPases / AAA-type			
3085	25	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
3086	24.99	kd	CGS001-56848	SPHK2	Sphingosine kinase			
3087	24.98	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
3088	24.97	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
3089	24.9	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
3090	24.88	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
3091	24.84	kd	CGS001-10325	RRAGB	-			
3092	24.81	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
3093	24.79	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
3094	24.74	kd	CGS001-6520	SLC3A2	SLC3 family			
3095	24.72	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
3096	24.68	kd	CGS001-9638	FEZ1	-			
3097	24.67	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
3098	24.62	kd	CGS001-57787	MARK4	MARK subfamily			
3099	24.55	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
3100	24.55	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
3101	24.48	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
3102	24.41	kd	CGS001-7039	TGFA	-			
3103	24.31	kd	CGS001-6648	SOD2	-			
3104	24.29	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
3105	24.23	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
3106	24.22	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
3107	24.15	oe	ccsbBroad304_00648	GLRX	-			
3108	24.13	kd	CGS001-163688	CALML6	EF-hand domain containing			
3109	24.1	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
3110	24.04	kd	CGS001-255738	PCSK9	Subtilisin			
3111	24	cp	BRD-K13800121	parecoxib	Cyclooxygenase inhibitor		LTF, PTGS2	Cyclooxygenase inhibitor
3112	23.94	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
3113	23.86	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
3114	23.86	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
3115	23.82	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
3116	23.79	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
3117	23.76	kd	CGS001-8525	DGKZ	-			
3118	23.74	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
3119	23.73	kd	CGS001-3565	IL4	Interleukins and interleukin receptors			
3120	23.73	kd	CGS001-375	ARF1	ADP-ribosylation factors			
3121	23.66	kd	CGS001-103	ADAR	-			
3122	23.65	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3123	23.65	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
3124	23.6	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
3125	23.56	kd	CGS001-58528	RRAGD	-			
3126	23.55	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
3127	23.55	kd	CGS001-6118	RPA2	-			
3128	23.55	kd	CGS001-2773	GNAI3	-			
3129	23.5	kd	CGS001-4255	MGMT	-			
3130	23.49	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
3131	23.41	kd	CGS001-5571	PRKAG1	AMPK subfamily			
3132	23.4	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
3133	23.32	kd	CGS001-6821	SUOX	-			
3134	23.3	oe	ccsbBroad304_00532	F11	Chymotrypsin			
3135	23.3	kd	CGS001-111	ADCY5	Adenylate cyclases			
3136	23.29	kd	CGS001-55612	FERMT1	Fermitins			
3137	23.28	kd	CGS001-4199	ME1	-			
3138	23.23	kd	CGS001-6696	SPP1	Endogenous ligands			
3139	23.21	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
3140	23.13	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
3141	23.1	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
3142	23.08	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
3143	23.04	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
3144	23.04	kd	CGS001-5763	PTMS	-			
3145	23.01	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
3146	22.99	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
3147	22.96	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
3148	22.92	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
3149	22.89	kd	CGS001-1955	MEGF9	-			
3150	22.86	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
3151	22.86	kd	CGS001-158	ADSL	-			
3152	22.84	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
3153	22.75	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
3154	22.75	cp	BRD-K94649603	taxifolin	Opioid receptor antagonist		APOB, APP, HMGCR	Opioid receptor antagonist
3155	22.6	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
3156	22.58	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
3157	22.56	kd	CGS001-607	BCL9	-			
3158	22.55	kd	CGS001-6897	TARS	Aminoacyl tRNA synthetases / Class II			
3159	22.53	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
3160	22.51	kd	CGS001-1062	CENPE	Kinesins			
3161	22.44	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
3162	22.42	kd	CGS001-126208	ZNF787	Zinc fingers, C2H2-type			
3163	22.41	kd	CGS001-9146	HGS	Zinc fingers, FYVE domain containing			
3164	22.4	kd	CGS001-1503	CTPS	-			
3165	22.36	kd	CGS001-545	ATR	ATR subfamily			
3166	22.34	kd	CGS001-10381	TUBB3	Tubulins			
3167	22.31	kd	CGS001-23597	ACOT9	Acyl CoA thioesterases			
3168	22.26	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
3169	22.23	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
3170	22.11	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
3171	22.05	kd	CGS001-965	CD58	CD molecules			
3172	22.01	kd	CGS001-55837	EAPP	-			
3173	22	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
3174	21.99	cp	BRD-K47780086	penciclovir	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor
3175	21.96	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
3176	21.96	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
3177	21.92	cp	BRD-K29113274	ketoconazole	Sterol demethylase inhibitor		AR, CYP19A1, CYP21A2, CYP2C19, CYP3A5, CYP3A7, KCNA10	Sterol demethylase inhibitor
3178	21.88	kd	CGS001-27161	EIF2C2	-			
3179	21.84	kd	CGS001-10589	DRAP1	-			
3180	21.79	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
3181	21.77	oe	ccsbBroad304_03310	LCMT1	-			
3182	21.76	cc		Serpin peptidase inhibitors LOF	-			
3183	21.7	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
3184	21.64	cc		Integrin subunits alpha LOF	-			
3185	21.64	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
3186	21.64	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
3187	21.64	kd	CGS001-54884	RETSAT	-			
3188	21.62	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
3189	21.61	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
3190	21.61	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
3191	21.59	kd	CGS001-23244	PDS5A	-			
3192	21.56	oe	ccsbBroad304_00472	EBF1	-			
3193	21.56	kd	CGS001-9700	ESPL1	-			
3194	21.55	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
3195	21.5	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
3196	21.48	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
3197	21.4	kd	CGS001-50808	AK3	-			
3198	21.39	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
3199	21.33	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
3200	21.26	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
3201	21.26	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
3202	21.25	kd	CGS001-8678	BECN1	-			
3203	21.14	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
3204	21.05	kd	CGS001-9318	COPS2	-			
3205	21	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
3206	20.98	oe	ccsbBroad304_00568	FHL2	-			
3207	20.92	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
3208	20.81	kd	CGS001-55312	RFK	-			
3209	20.76	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
3210	20.72	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
3211	20.65	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
3212	20.56	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
3213	20.53	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
3214	20.48	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3215	20.43	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
3216	20.43	kd	CGS001-56616	DIABLO	-			
3217	20.39	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
3218	20.37	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
3219	20.31	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
3220	20.28	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
3221	20.25	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
3222	20.24	kd	CGS001-3177	SLC29A2	SLC29 family			
3223	20.2	kd	CGS001-83448	PUS7L	-			
3224	20.15	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
3225	20.13	kd	CGS001-51586	MED15	-			
3226	20.12	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
3227	20.11	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
3228	20.09	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
3229	20.04	kd	CGS001-116535	MRGPRF	GPCR / Class A : Orphans			
3230	19.97	cc		GATA Zinc finger domain containing LOF	-			
3231	19.9	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
3232	19.9	kd	CGS001-10105	PPIF	-			
3233	19.84	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
3234	19.81	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
3235	19.76	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
3236	19.76	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
3237	19.68	cc		Adenosine receptor agonist	-			
3238	19.67	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3239	19.62	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
3240	19.51	cp	BRD-K49404994	levetiracetam	Calcium channel blocker		SV2A, CACNA1B, SCN1A	Calcium channel blocker
3241	19.44	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
3242	19.43	kd	CGS001-64223	MLST8	WD repeat domain containing			
3243	19.4	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3244	19.36	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
3245	19.27	cc		Mitogen activated protein kinases LOF	-			
3246	19.19	kd	CGS001-11129	CLASRP	-			
3247	19.11	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
3248	19.1	kd	CGS001-5578	PRKCA	Delta subfamily			
3249	18.9	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
3250	18.81	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
3251	18.73	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
3252	18.66	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
3253	18.66	kd	CGS001-9712	USP6NL	-			
3254	18.39	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
3255	18.31	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
3256	18.29	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3257	18.18	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
3258	18.03	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
3259	17.9	cp	BRD-K18523449	mestanolone	Androgenic steroid			Androgenic steroid
3260	17.89	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
3261	17.88	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
3262	17.75	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
3263	17.65	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
3264	17.63	kd	CGS001-8535	CBX4	-			
3265	17.52	kd	CGS001-55239	OGFOD1	-			
3266	17.47	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
3267	17.41	kd	CGS001-5594	MAPK1	MAPK:ERK subfamily			
3268	17.31	cc		Bacterial 30S ribosomal subunit inhibitor	-			
3269	17.18	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
3270	17.15	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3271	17.14	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
3272	17.11	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
3273	16.96	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
3274	16.74	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3275	16.72	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
3276	16.6	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3277	16.57	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3278	16.5	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
3279	16.48	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
3280	16.45	oe	ccsbBroad304_00738	HINT1	-			
3281	16.37	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
3282	16.34	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3283	16.29	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
3284	16.21	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
3285	16.16	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
3286	16.12	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
3287	16.08	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
3288	15.99	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
3289	15.91	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
3290	15.89	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
3291	15.88	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3292	15.79	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
3293	15.77	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
3294	15.68	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
3295	15.58	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
3296	15.55	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
3297	15.5	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
3298	15.48	cc		AHSP Pathway LOF	-			
3299	15.35	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
3300	15.3	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
3301	15.17	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
3302	15.15	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
3303	15.03	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
3304	15.01	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
3305	14.99	cc		Ribonucleotide reductase inhibitor	-			
3306	14.85	cp	BRD-K11630072	carmofur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
3307	14.81	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
3308	14.66	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
3309	14.63	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
3310	14.61	kd	CGS001-1384	CRAT	-			
3311	14.55	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
3312	14.5	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
3313	14.38	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
3314	14.34	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
3315	14.34	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3316	14.33	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
3317	14.31	cp	BRD-K59456551	methotrexate	Dihydrofolate reductase inhibitor		DHFR, AOX1, FOLR1, TYMS	Dihydrofolate reductase inhibitor
3318	14.12	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
3319	14.05	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
3320	14.02	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
3321	13.93	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
3322	13.89	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
3323	13.74	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
3324	13.67	cp	BRD-K22009844	phenprobamate	Muscle relaxant			Muscle relaxant
3325	13.67	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
3326	13.53	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
3327	13.53	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
3328	13.44	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
3329	13.38	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
3330	13.27	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
3331	13.19	cc		Progesterone receptor agonist	-			
3332	13.14	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
3333	13.04	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3334	12.99	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
3335	12.97	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3336	12.95	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
3337	12.83	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
3338	12.68	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
3339	12.6	cp	BRD-K82143716	flucytosine	Antifungal		DNMT1	Antifungal
3340	12.44	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
3341	12.43	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
3342	12.42	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
3343	12.41	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
3344	12.4	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
3345	12.29	kd	CGS001-1452	CSNK1A1	Casein kinase 1 (CK1) family			
3346	12.28	cc		Zinc fingers RanBP2 type LOF	-			
3347	12.22	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
3348	12.13	cc		Dihydrofolate reductase inhibitor	-			
3349	12.1	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3350	12.08	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
3351	11.73	cp	BRD-K21806131	tegaserod	Serotonin receptor partial agonist		HTR4, HTR2B, HTR2A, HTR2C	Serotonin receptor partial agonist
3352	11.64	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
3353	11.3	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
3354	11.29	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
3355	11.25	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
3356	11.23	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
3357	11.2	cp	BRD-K65910366	KUC103904N	-666			-666
3358	10.83	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
3359	10.72	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
3360	10.68	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
3361	10.39	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
3362	10.36	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3363	10.35	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
3364	10.24	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
3365	10.22	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
3366	10.15	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
3367	10.06	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
3368	10.06	cp	BRD-K34508425	KUC103898N	-666			-666
3369	10.05	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
3370	9.95	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
3371	9.81	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
3372	9.73	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
3373	9.71	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
3374	9.64	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
3375	9.52	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
3376	9.47	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
3377	9.22	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
3378	9	cp	BRD-K44779798	miglitol	Glucosidase inhibitor		GAA, MGAM, GANAB, GANC, SLC5A4	Glucosidase inhibitor
3379	8.97	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
3380	8.92	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3381	8.8	cp	BRD-K47278471	diphenhydramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3382	8.78	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3383	8.71	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
3384	8.7	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
3385	8.68	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
3386	8.64	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
3387	8.6	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
3388	8.51	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
3389	8.42	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
3390	8.21	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
3391	7.94	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
3392	7.93	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
3393	7.82	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
3394	7.58	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
3395	7.38	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
3396	7.27	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
3397	7.24	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
3398	7.21	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
3399	6.79	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
3400	6.43	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
3401	6.31	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
3402	6.19	cp	BRD-A42423104	benproperine	Antitussive			Antitussive
3403	6.1	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
3404	6.1	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
3405	5.89	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3406	5.86	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
3407	5.75	cc		Bacterial cell wall synthesis inhibitor	-			
3408	5.37	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3409	5.21	cp	BRD-A68589262	troxipide	Glucosamine synthetase stimulant			Glucosamine synthetase stimulant
3410	5.16	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
3411	5.09	cc		Rho associated kinase inhibitor	-			
3412	4.46	cp	BRD-K13664374	dichloroacetic-acid	Pyruvate dehydrogenase kinase inhibitor		PDK1	Pyruvate dehydrogenase kinase inhibitor
3413	-2.27	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
3414	-2.31	cc		VEGFR inhibitor	-			
3415	-3.63	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
3416	-4.29	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
3417	-4.77	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
3418	-5.72	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
3419	-6.3	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
3420	-6.67	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
3421	-6.84	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
3422	-7	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
3423	-7.18	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
3424	-7.23	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
3425	-7.29	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
3426	-7.31	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
3427	-7.38	kd	CGS001-2931	GSK3A	GSK subfamily			
3428	-7.42	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
3429	-7.53	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
3430	-7.55	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
3431	-7.59	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
3432	-7.77	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
3433	-8.02	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
3434	-8.05	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
3435	-8.07	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
3436	-8.18	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
3437	-8.33	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
3438	-8.38	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
3439	-8.6	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
3440	-8.75	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
3441	-8.83	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
3442	-8.96	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
3443	-8.99	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
3444	-9.03	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3445	-9.1	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
3446	-9.42	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
3447	-9.45	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
3448	-9.58	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
3449	-9.61	cc		DNA Replication LOF	-			
3450	-9.72	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
3451	-9.8	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
3452	-10.1	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
3453	-10.11	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
3454	-10.29	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
3455	-10.43	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
3456	-10.5	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
3457	-10.6	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
3458	-10.66	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
3459	-10.7	cp	BRD-K73991644	isoquercetin	Aldose reductase inhibitor		AKR1B1, ACE	Aldose reductase inhibitor
3460	-10.78	cc		Tricyclic antidepressant	-			
3461	-10.83	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
3462	-10.95	cc		Androgen receptor modulator	-			
3463	-11.02	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
3464	-11.03	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
3465	-11.11	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
3466	-11.18	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3467	-11.28	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
3468	-11.31	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
3469	-11.31	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
3470	-11.33	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
3471	-11.37	cp	BRD-K62858456	lomerizine	Calcium channel blocker		ABCB1, CACNA1B, SCN5A	Calcium channel blocker
3472	-11.57	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
3473	-11.62	kd	CGS001-51268	PIPOX	-			
3474	-11.79	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
3475	-11.86	kd	CGS001-3265	HRAS	RAS subfamily			
3476	-11.95	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
3477	-11.97	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3478	-12.07	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
3479	-12.24	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
3480	-12.29	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3481	-12.29	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
3482	-12.4	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
3483	-12.46	kd	CGS001-7525	YES1	Src family			
3484	-12.49	cp	BRD-A88254928	salbutamol	Adrenergic receptor agonist		ADRB2, ADRB1	Adrenergic receptor agonist
3485	-12.55	cp	BRD-K39983086	loteprednol	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Phospholipase inhibitor
3486	-12.64	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
3487	-12.99	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
3488	-13.28	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
3489	-13.34	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
3490	-13.45	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
3491	-13.49	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
3492	-13.52	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
3493	-13.61	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
3494	-13.63	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
3495	-13.66	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
3496	-13.66	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
3497	-13.78	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
3498	-13.8	cc		Aldehyde dehydrogenases LOF	-			
3499	-13.89	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
3500	-13.9	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3501	-13.96	cp	BRD-K22227508	targinine	Nitric oxide synthase inhibitor		NOS2, NOS3	Nitric oxide synthase inhibitor
3502	-14.28	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
3503	-14.32	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
3504	-14.42	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
3505	-14.47	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
3506	-14.49	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
3507	-14.73	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
3508	-14.92	cc		SRC inhibitor	-			
3509	-14.96	oe	ccsbBroad304_00658	GNG5	-			
3510	-15.01	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
3511	-15.08	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
3512	-15.09	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
3513	-15.35	cc		RAF inhibitor	-			
3514	-15.36	kd	CGS001-2475	MTOR	FRAP subfamily			
3515	-15.39	kd	CGS001-8317	CDC7	CDC7 family			
3516	-15.43	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
3517	-15.44	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
3518	-15.44	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
3519	-15.5	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
3520	-15.51	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
3521	-15.74	cp	BRD-K88679075	methandriol	Androgenic steroid			Androgenic steroid
3522	-15.91	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
3523	-15.92	cp	BRD-K41051431	mecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3524	-16.08	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
3525	-16.08	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
3526	-16.1	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
3527	-16.15	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
3528	-16.27	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
3529	-16.48	kd	CGS001-4929	NR4A2	Nerve growth factor IB-like receptors			
3530	-16.56	cp	BRD-K51671335	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
3531	-16.59	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
3532	-16.59	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
3533	-16.63	cc		Nucleoside reverse transcriptase inhibitor	-			
3534	-16.65	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
3535	-16.71	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3536	-17.04	kd	CGS001-54541	DDIT4	-			
3537	-17.07	cc		IGF-1 inhibitor	-			
3538	-17.07	kd	CGS001-1362	CPD	Carboxypeptidase A			
3539	-17.09	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
3540	-17.12	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
3541	-17.12	kd	CGS001-1675	CFD	Complement system			
3542	-17.29	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
3543	-17.38	kd	CGS001-84722	PSRC1	-			
3544	-17.43	kd	CGS001-10400	PEMT	-			
3545	-17.46	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
3546	-17.55	kd	CGS001-1305	COL13A1	Collagens			
3547	-17.7	cp	BRD-K40758068	efavirenz	HIV protease inhibitor		CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5	HIV protease inhibitor
3548	-17.7	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
3549	-17.71	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
3550	-17.72	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
3551	-17.78	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
3552	-17.78	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
3553	-17.88	cc		BCL inhibitor	-			
3554	-17.9	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
3555	-17.93	cp	BRD-K06388322	pramipexole	Dopamine receptor agonist		DRD3, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3556	-17.95	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
3557	-17.99	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3558	-17.99	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
3559	-18.02	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
3560	-18.07	kd	CGS001-2731	GLDC	-			
3561	-18.12	kd	CGS001-4329	ALDH6A1	Aldehyde dehydrogenases			
3562	-18.13	kd	CGS001-955	ENTPD6	-			
3563	-18.26	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
3564	-18.28	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
3565	-18.34	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
3566	-18.39	cp	BRD-K85925969	zalcitabine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
3567	-18.4	kd	CGS001-5777	PTPN6	Protein tyrosine phosphatases			
3568	-18.42	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
3569	-18.5	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
3570	-18.59	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
3571	-18.61	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
3572	-18.64	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
3573	-18.67	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
3574	-18.73	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
3575	-18.76	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
3576	-18.78	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
3577	-18.85	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
3578	-18.88	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
3579	-18.95	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
3580	-18.99	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
3581	-19.01	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
3582	-19.04	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
3583	-19.06	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
3584	-19.06	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
3585	-19.1	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
3586	-19.16	kd	CGS001-35	ACADS	-			
3587	-19.19	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3588	-19.26	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
3589	-19.28	oe	ccsbBroad304_02313	ACTR3	-			
3590	-19.3	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
3591	-19.42	kd	CGS001-7030	TFE3	Basic helix-loop-helix proteins			
3592	-19.45	kd	CGS001-53836	GPR87	GPCR / Class A : Orphans			
3593	-19.46	kd	CGS001-4602	MYB	-			
3594	-19.5	cp	BRD-K34437622	BRD-K34437622	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
3595	-19.52	kd	CGS001-1859	DYRK1A	Dyrk1 subfamily			
3596	-19.53	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
3597	-19.57	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
3598	-19.66	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
3599	-19.67	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
3600	-19.74	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
3601	-19.77	kd	CGS001-4143	MAT1A	-			
3602	-19.82	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
3603	-19.85	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
3604	-19.88	kd	CGS001-2950	GSTP1	Glutathione S-transferases			
3605	-19.89	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
3606	-19.89	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
3607	-19.94	kd	CGS001-6119	RPA3	-			
3608	-19.95	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
3609	-19.95	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
3610	-20.02	oe	ccsbBroad304_03858	SRPRB	-			
3611	-20.05	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
3612	-20.06	kd	CGS001-9643	MORF4L2	-			
3613	-20.08	kd	CGS001-9341	VAMP3	Vesicle-associated membrane proteins			
3614	-20.11	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
3615	-20.14	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
3616	-20.17	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
3617	-20.21	kd	CGS001-3123	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
3618	-20.28	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
3619	-20.29	oe	ccsbBroad304_00833	IFNG	Interferons			
3620	-20.32	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
3621	-20.32	kd	CGS001-8669	EIF3J	-			
3622	-20.32	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
3623	-20.36	kd	CGS001-5217	PFN2	-			
3624	-20.37	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3625	-20.39	kd	CGS001-26149	ZNF658	Zinc fingers, C2H2-type			
3626	-20.43	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
3627	-20.48	cp	BRD-K00673382	famotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
3628	-20.64	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
3629	-20.65	oe	ccsbBroad304_03497	TXNL4B	-			
3630	-20.67	kd	CGS001-1445	CSK	Csk family			
3631	-20.71	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
3632	-20.72	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
3633	-20.8	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
3634	-20.87	kd	CGS001-4763	NF1	-			
3635	-20.91	kd	CGS001-3980	LIG3	-			
3636	-20.94	kd	CGS001-79258	MMEL1	-			
3637	-20.96	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
3638	-20.96	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
3639	-20.98	cc		Potassium channel blocker	-			
3640	-20.99	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
3641	-21	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
3642	-21	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
3643	-21.01	cc		Glucocorticoid receptor agonist	-			
3644	-21.03	kd	CGS001-546	ATRX	-			
3645	-21.07	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
3646	-21.25	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
3647	-21.25	kd	CGS001-2021	ENDOG	-			
3648	-21.26	kd	CGS001-1195	CLK1	CDC-like kinases			
3649	-21.29	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
3650	-21.35	kd	CGS001-94235	GNG8	-			
3651	-21.4	kd	CGS001-7276	TTR	-			
3652	-21.4	kd	CGS001-93487	MAPK1IP1L	-			
3653	-21.42	cp	BRD-K50866992	tropisetron	Serotonin receptor antagonist		HTR3A, GLRA1, GLRA2, GLRB, HTR4	Serotonin receptor antagonist
3654	-21.44	kd	CGS001-637	BID	Endogenous ligands			
3655	-21.45	kd	CGS001-65123	INTS3	-			
3656	-21.54	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
3657	-21.55	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
3658	-21.55	kd	CGS001-6443	SGCB	-			
3659	-21.57	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
3660	-21.63	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
3661	-21.64	cc		C2 domain containing protein kinases LOF	-			
3662	-21.64	kd	CGS001-10489	LRRC41	-			
3663	-21.65	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
3664	-21.66	kd	CGS001-6810	STX4	-			
3665	-21.67	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
3666	-21.68	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
3667	-21.7	kd	CGS001-51026	GOLT1B	-			
3668	-21.74	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
3669	-21.79	oe	ccsbBroad304_07017	SUOX	-			
3670	-21.81	kd	CGS001-501	ALDH7A1	Aldehyde dehydrogenases			
3671	-21.83	kd	CGS001-5300	PIN1	-			
3672	-21.92	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
3673	-21.94	oe	ccsbBroad304_07592	CEPT1	-			
3674	-21.96	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
3675	-22	kd	CGS001-23378	RRP8	-			
3676	-22.02	kd	CGS001-8022	LHX3	Homeoboxes / LIM class			
3677	-22.03	oe	ccsbBroad304_07768	NISCH	-			
3678	-22.05	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
3679	-22.06	kd	CGS001-9871	SEC24D	-			
3680	-22.09	cc		HMGCR inhibitor	-			
3681	-22.14	kd	CGS001-5829	PXN	-			
3682	-22.17	kd	CGS001-7471	WNT1	Endogenous ligands			
3683	-22.18	cp	BRD-K39621635	artemether	Antimalarial		ATP1A1, CYP2B6, CYP2C19, CYP3A5	Antimalarial
3684	-22.21	kd	CGS001-3226	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
3685	-22.25	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
3686	-22.29	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
3687	-22.3	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
3688	-22.36	kd	CGS001-166793	ZBTB49	BTB/POZ domain containing			
3689	-22.37	cc		Kruppel like transcription factors LOF	-			
3690	-22.38	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
3691	-22.4	oe	ccsbBroad304_10487	BPHL	-			
3692	-22.49	oe	ccsbBroad304_09881	RFX6	-			
3693	-22.49	kd	CGS001-1066	CES1	Carboxylesterases			
3694	-22.5	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
3695	-22.6	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
3696	-22.67	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
3697	-22.75	kd	CGS001-1374	CPT1A	-			
3698	-22.76	kd	CGS001-5362	PLXNA2	Plexins			
3699	-22.77	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
3700	-22.78	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
3701	-22.81	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
3702	-22.81	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3703	-22.81	kd	CGS001-6788	STK3	MST subfamily			
3704	-22.84	cc		HOXL subclass homeoboxes LOF	-			
3705	-22.85	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
3706	-22.86	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
3707	-22.91	cc		Proteasome inhibitor	-			
3708	-22.97	kd	CGS001-5293	PIK3CD	Phosphatidylinositol kinases			
3709	-23	oe	ccsbBroad304_06952	SKP1	-			
3710	-23.05	kd	CGS001-29978	UBQLN2	Ubiquilin family			
3711	-23.06	kd	CGS001-4697	NDUFA4	-			
3712	-23.1	kd	CGS001-23386	NUDCD3	-			
3713	-23.12	kd	CGS001-91949	COG7	Components of oligomeric golgi complex			
3714	-23.17	kd	CGS001-5567	PRKACB	Protein kinase A			
3715	-23.17	kd	CGS001-4967	OGDH	-			
3716	-23.17	oe	ccsbBroad304_07220	CDC45	-			
3717	-23.22	oe	ccsbBroad304_00376	CSK	Csk family			
3718	-23.23	kd	CGS001-2182	ACSL4	Acyl-CoA synthetase family			
3719	-23.25	kd	CGS001-5925	RB1	Endogenous ligands			
3720	-23.28	kd	CGS001-4904	YBX1	-			
3721	-23.3	kd	CGS001-81550	TDRD3	Tudor domain containing			
3722	-23.3	kd	CGS001-9928	KIF14	Kinesins			
3723	-23.32	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
3724	-23.34	kd	CGS001-7468	WHSC1	Zinc fingers, PHD-type			
3725	-23.39	oe	ccsbBroad304_00446	DKC1	-			
3726	-23.41	oe	ccsbBroad304_00960	SMAD1	SMADs			
3727	-23.42	oe	ccsbBroad304_07832	XPO7	Exportins			
3728	-23.44	kd	CGS001-5108	PCM1	-			
3729	-23.45	kd	CGS001-665	BNIP3L	-			
3730	-23.47	kd	CGS001-59343	SENP2	-			
3731	-23.49	kd	CGS001-25937	WWTR1	Hippo Signaling			
3732	-23.49	kd	CGS001-5928	RBBP4	WD repeat domain containing			
3733	-23.5	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
3734	-23.5	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
3735	-23.5	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
3736	-23.52	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
3737	-23.52	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
3738	-23.54	kd	CGS001-340371	NRBP2	NRBP family			
3739	-23.54	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
3740	-23.55	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
3741	-23.56	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
3742	-23.57	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
3743	-23.57	kd	CGS001-23499	MACF1	EF-hand domain containing			
3744	-23.61	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
3745	-23.62	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
3746	-23.63	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
3747	-23.65	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
3748	-23.66	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
3749	-23.69	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
3750	-23.77	oe	ccsbBroad304_00626	GDI1	-			
3751	-23.8	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
3752	-23.8	kd	CGS001-11014	KDELR2	-			
3753	-23.83	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
3754	-23.86	kd	CGS001-3119	HLA-DQB1	Immunoglobulin superfamily / C1-set domain containing			
3755	-23.87	cc		Homeobox Gene GOF	-			
3756	-23.87	kd	CGS001-8996	NOL3	-			
3757	-23.91	oe	ccsbBroad304_03658	DCP1A	-			
3758	-23.96	cc		G2 M Checkpoint LOF	-			
3759	-23.99	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
3760	-23.99	oe	ccsbBroad304_00789	HSBP1	-			
3761	-23.99	kd	CGS001-5092	PCBD1	-			
3762	-24.01	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
3763	-24.02	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
3764	-24.04	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
3765	-24.04	kd	CGS001-11243	PMF1	-			
3766	-24.05	oe	ccsbBroad304_09006	RPF1	-			
3767	-24.06	oe	ccsbBroad304_01640	TAF12	-			
3768	-24.07	kd	CGS001-27109	ATP5S	-			
3769	-24.08	kd	CGS001-5245	PHB	-			
3770	-24.09	oe	ccsbBroad304_02804	KLHDC2	-			
3771	-24.09	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3772	-24.12	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
3773	-24.12	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
3774	-24.12	kd	CGS001-306	ANXA3	Annexins			
3775	-24.12	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
3776	-24.13	cc		FOS transcription factor family GOF	-			
3777	-24.13	kd	CGS001-2690	GHR	Prolactin receptor family			
3778	-24.14	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
3779	-24.16	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
3780	-24.18	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
3781	-24.18	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
3782	-24.2	oe	ccsbBroad304_07178	ZFP112	-			
3783	-24.21	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
3784	-24.22	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
3785	-24.27	kd	CGS001-7465	WEE1	WEE family			
3786	-24.3	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
3787	-24.31	kd	CGS001-506	ATP5B	ATPases / F-type			
3788	-24.36	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
3789	-24.37	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
3790	-24.39	kd	CGS001-25949	SYF2	-			
3791	-24.41	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
3792	-24.42	kd	CGS001-5577	PRKAR2B	Protein kinase A			
3793	-24.42	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
3794	-24.48	kd	CGS001-6309	SC5DL	-			
3795	-24.5	oe	ccsbBroad304_00961	SMAD2	SMADs			
3796	-24.5	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
3797	-24.52	oe	ccsbBroad304_00963	SMAD5	SMADs			
3798	-24.57	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
3799	-24.58	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
3800	-24.61	kd	CGS001-91433	RCCD1	-			
3801	-24.62	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
3802	-24.62	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
3803	-24.63	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
3804	-24.64	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
3805	-24.67	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
3806	-24.69	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
3807	-24.72	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
3808	-24.72	kd	CGS001-5588	PRKCQ	Delta subfamily			
3809	-24.74	kd	CGS001-1112	FOXN3	Forkhead boxes			
3810	-24.79	kd	CGS001-2919	CXCL1	Endogenous ligands			
3811	-24.81	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
3812	-24.84	kd	CGS001-1534	CYB561	Cytochrome b genes			
3813	-24.9	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
3814	-24.94	kd	CGS001-801	CALM1	EF-hand domain containing			
3815	-24.95	kd	CGS001-51750	RTEL1	-			
3816	-24.97	kd	CGS001-391013	PLA2G2C	-			
3817	-24.97	kd	CGS001-2274	FHL2	-			
3818	-24.98	kd	CGS001-5566	PRKACA	Protein kinase A			
3819	-25	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
3820	-25.01	kd	CGS001-64080	RBKS	-			
3821	-25.03	kd	CGS001-57222	ERGIC1	-			
3822	-25.05	kd	CGS001-4683	NBN	-			
3823	-25.06	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
3824	-25.07	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
3825	-25.08	kd	CGS001-8772	FADD	-			
3826	-25.1	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
3827	-25.11	kd	CGS001-861	RUNX1	-			
3828	-25.11	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3829	-25.12	kd	CGS001-3065	HDAC1	Histone deacetylases			
3830	-25.16	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
3831	-25.16	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
3832	-25.17	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
3833	-25.19	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
3834	-25.2	kd	CGS001-6207	RPS13	S ribosomal proteins			
3835	-25.23	kd	CGS001-151126	ZNF385B	-			
3836	-25.24	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
3837	-25.27	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
3838	-25.27	kd	CGS001-10046	MAMLD1	-			
3839	-25.29	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
3840	-25.3	kd	CGS001-8639	AOC3	Oxidoreductases			
3841	-25.31	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
3842	-25.31	kd	CGS001-51655	RASD1	-			
3843	-25.32	oe	ccsbBroad304_02822	ARFIP2	-			
3844	-25.34	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
3845	-25.37	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
3846	-25.37	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
3847	-25.39	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
3848	-25.44	kd	CGS001-1509	CTSD	Cathepsins			
3849	-25.44	kd	CGS001-27	ABL2	Abl family			
3850	-25.49	kd	CGS001-11267	SNF8	-			
3851	-25.51	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
3852	-25.54	cp	BRD-K92413528	thiazolidinecarboxylic-acid	Reducing agent			Reducing agent
3853	-25.54	kd	CGS001-29880	ALG5	Glycosyltransferase family 2 domain containing			
3854	-25.55	oe	ccsbBroad304_08694	TBX20	T-boxes			
3855	-25.57	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
3856	-25.58	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
3857	-25.58	kd	CGS001-2629	GBA	-			
3858	-25.6	oe	ccsbBroad304_02163	MED7	-			
3859	-25.63	kd	CGS001-79139	DERL1	-			
3860	-25.64	kd	CGS001-25797	QPCT	Aminopeptidase Y			
3861	-25.65	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
3862	-25.66	oe	ccsbBroad304_03040	NKIRAS2	-			
3863	-25.66	kd	CGS001-10928	RALBP1	-			
3864	-25.66	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
3865	-25.69	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
3866	-25.71	oe	ccsbBroad304_02686	COPZ1	-			
3867	-25.73	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
3868	-25.74	kd	CGS001-8667	EIF3H	-			
3869	-25.75	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
3870	-25.75	kd	CGS001-55234	SMU1	WD repeat domain containing			
3871	-25.75	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
3872	-25.76	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
3873	-25.77	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
3874	-25.81	kd	CGS001-7357	UGCG	Glycosyltransferase family 2 domain containing			
3875	-25.83	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
3876	-25.83	kd	CGS001-5894	RAF1	RAF family			
3877	-25.85	kd	CGS001-23670	TMEM2	-			
3878	-25.86	kd	CGS001-5019	OXCT1	-			
3879	-25.87	kd	CGS001-23118	TAB2	-			
3880	-25.9	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3881	-25.91	kd	CGS001-6421	SFPQ	RNA binding motif (RRM) containing			
3882	-25.93	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
3883	-25.95	cp	BRD-A71009679	KUC103420N	-666			-666
3884	-25.97	kd	CGS001-23047	PDS5B	-			
3885	-25.99	kd	CGS001-2266	FGG	Endogenous ligands			
3886	-26.02	kd	CGS001-23335	WDR7	WD repeat domain containing			
3887	-26.03	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
3888	-26.03	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
3889	-26.08	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
3890	-26.08	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
3891	-26.09	kd	CGS001-5423	POLB	DNA polymerases			
3892	-26.1	oe	ccsbBroad304_06836	RAD23B	-			
3893	-26.11	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
3894	-26.11	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
3895	-26.11	kd	CGS001-23566	LPAR3	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
3896	-26.13	kd	CGS001-324	APC	Armadillo repeat containing			
3897	-26.15	kd	CGS001-26036	ZNF451	Zinc fingers, C2H2-type			
3898	-26.17	kd	CGS001-55176	SEC61A2	-			
3899	-26.18	oe	ccsbBroad304_06695	PCK2	-			
3900	-26.18	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
3901	-26.19	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
3902	-26.21	kd	CGS001-5579	PRKCB	Alpha subfamily			
3903	-26.23	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
3904	-26.27	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
3905	-26.3	oe	ccsbBroad304_09821	TMEM154	-			
3906	-26.36	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
3907	-26.36	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
3908	-26.38	kd	CGS001-3479	IGF1	Endogenous ligands			
3909	-26.38	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
3910	-26.39	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3911	-26.39	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
3912	-26.44	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
3913	-26.47	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
3914	-26.5	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
3915	-26.52	kd	CGS001-5565	PRKAB2	AMPK subfamily			
3916	-26.52	kd	CGS001-50943	FOXP3	Forkhead boxes			
3917	-26.54	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
3918	-26.54	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
3919	-26.54	kd	CGS001-57154	SMURF1	-			
3920	-26.55	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
3921	-26.55	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
3922	-26.56	kd	CGS001-5881	RAC3	Endogenous ligands			
3923	-26.56	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
3924	-26.58	kd	CGS001-55193	PBRM1	Non-enzymatic BRD containing proteins			
3925	-26.6	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
3926	-26.62	kd	CGS001-1196	CLK2	CDC-like kinases			
3927	-26.65	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
3928	-26.65	kd	CGS001-1843	DUSP1	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3929	-26.67	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3930	-26.68	cc		PKC inhibitor	-			
3931	-26.7	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3932	-26.71	kd	CGS001-9131	AIFM1	-			
3933	-26.76	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3934	-26.81	kd	CGS001-3992	FADS1	Fatty acid desaturases			
3935	-26.82	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
3936	-26.82	kd	CGS001-8841	HDAC3	Histone deacetylases			
3937	-26.84	oe	ccsbBroad304_05948	CCND2	-			
3938	-26.85	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
3939	-26.89	oe	ccsbBroad304_07704	SUB1	-			
3940	-26.9	oe	ccsbBroad304_02741	PDS5A	-			
3941	-26.9	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
3942	-26.92	oe	ccsbBroad304_03928	RRAGC	-			
3943	-26.95	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
3944	-26.97	oe	ccsbBroad304_08993	DHDDS	-			
3945	-26.97	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
3946	-26.98	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
3947	-27.04	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
3948	-27.05	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
3949	-27.06	oe	ccsbBroad304_00098	ARG1	Arginase			
3950	-27.07	kd	CGS001-85004	RERG	-			
3951	-27.07	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
3952	-27.08	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
3953	-27.09	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
3954	-27.09	kd	CGS001-10695	CNPY3	Trinucleotide (CAG) repeat containing			
3955	-27.09	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
3956	-27.11	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
3957	-27.13	kd	CGS001-10250	SRRM1	-			
3958	-27.15	kd	CGS001-139760	GPR119	GPCR / Class A : Orphans			
3959	-27.17	oe	ccsbBroad304_00542	FBP1	-			
3960	-27.17	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
3961	-27.17	kd	CGS001-3481	IGF2	-			
3962	-27.17	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
3963	-27.17	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
3964	-27.18	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
3965	-27.19	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
3966	-27.2	kd	CGS001-1001	CDH3	Cadherins / Major cadherins			
3967	-27.21	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
3968	-27.23	oe	ccsbBroad304_07124	UROD	-			
3969	-27.23	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
3970	-27.25	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
3971	-27.29	kd	CGS001-5663	PSEN1	Presenilin			
3972	-27.3	kd	CGS001-2153	F5	Blood coagulation components			
3973	-27.31	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
3974	-27.31	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
3975	-27.34	kd	CGS001-51174	TUBD1	Tubulins			
3976	-27.35	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
3977	-27.35	kd	CGS001-4176	MCM7	-			
3978	-27.38	kd	CGS001-8720	MBTPS1	Subtilisin			
3979	-27.39	kd	CGS001-4174	MCM5	-			
3980	-27.41	kd	CGS001-8220	DGCR14	-			
3981	-27.43	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
3982	-27.43	kd	CGS001-1810	DR1	-			
3983	-27.45	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
3984	-27.48	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
3985	-27.5	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
3986	-27.53	kd	CGS001-58497	PRUNE	-			
3987	-27.54	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
3988	-27.54	kd	CGS001-26298	EHF	-			
3989	-27.57	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
3990	-27.61	kd	CGS001-55437	STRADB	STLK subfamily			
3991	-27.62	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
3992	-27.64	kd	CGS001-51203	NUSAP1	-			
3993	-27.65	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
3994	-27.65	kd	CGS001-1512	CTSH	Cathepsins			
3995	-27.66	oe	ccsbBroad304_02605	PAPD7	-			
3996	-27.66	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
3997	-27.68	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
3998	-27.68	kd	CGS001-823	CAPN1	EF-hand domain containing			
3999	-27.73	kd	CGS001-130497	OSR1	Zinc fingers, C2H2-type			
4000	-27.77	kd	CGS001-1045	CDX2	Homeoboxes / ANTP class : HOXL subclass			
4001	-27.78	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
4002	-27.78	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
4003	-27.83	oe	ccsbBroad304_00250	CD19	CD molecules			
4004	-27.83	kd	CGS001-9374	PPT2	-			
4005	-27.83	kd	CGS001-79722	ANKRD55	Ankyrin repeat domain containing			
4006	-27.84	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
4007	-27.85	kd	CGS001-54861	SNRK	SNRK subfamily			
4008	-27.86	kd	CGS001-397	ARHGDIB	Endogenous ligands			
4009	-27.87	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
4010	-27.88	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
4011	-27.89	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
4012	-27.91	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
4013	-27.97	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
4014	-27.99	kd	CGS001-2967	GTF2H3	General transcription factors			
4015	-28.02	kd	CGS001-55214	LEPREL1	-			
4016	-28.03	kd	CGS001-66008	TRAK2	-			
4017	-28.04	kd	CGS001-10957	PNRC1	-			
4018	-28.05	kd	CGS001-3579	CXCR2	Chemokine receptors			
4019	-28.09	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
4020	-28.09	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
4021	-28.09	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
4022	-28.11	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
4023	-28.11	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
4024	-28.13	oe	ccsbBroad304_04379	LZIC	-			
4025	-28.13	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
4026	-28.14	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
4027	-28.16	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
4028	-28.19	kd	CGS001-259	AMBP	Lipocalins			
4029	-28.23	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
4030	-28.23	kd	CGS001-79947	DHDDS	-			
4031	-28.26	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
4032	-28.26	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
4033	-28.27	kd	CGS001-84109	QRFPR	GPCR / Class A : RF amide peptide receptors			
4034	-28.29	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
4035	-28.29	kd	CGS001-475	ATOX1	-			
4036	-28.3	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
4037	-28.31	oe	ccsbBroad304_13939	MOK	RCK family			
4038	-28.31	kd	CGS001-10452	TOMM40	-			
4039	-28.33	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
4040	-28.34	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
4041	-28.34	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
4042	-28.4	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
4043	-28.4	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
4044	-28.4	kd	CGS001-5050	PAFAH1B3	-			
4045	-28.4	kd	CGS001-8874	ARHGEF7	Rho guanine nucleotide exchange factors			
4046	-28.42	oe	ccsbBroad304_00397	CTSK	Cathepsins			
4047	-28.46	oe	ccsbBroad304_02271	LPGAT1	-			
4048	-28.46	cp	BRD-K16336526	capsaicin	TRPV agonist		TRPV1, CFTR, ENOX2	TRPV agonist
4049	-28.47	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
4050	-28.48	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
4051	-28.48	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
4052	-28.52	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
4053	-28.55	kd	CGS001-7076	TIMP1	-			
4054	-28.57	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
4055	-28.59	oe	ccsbBroad304_06449	ILF3	-			
4056	-28.62	oe	ccsbBroad304_08879	CASD1	-			
4057	-28.66	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
4058	-28.66	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
4059	-28.68	kd	CGS001-10493	VAT1	-			
4060	-28.7	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
4061	-28.72	oe	ccsbBroad304_06159	CTTN	-			
4062	-28.76	kd	CGS001-51079	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
4063	-28.82	kd	CGS001-161725	OTUD7A	OTU domain containing			
4064	-28.83	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
4065	-28.86	oe	ccsbBroad304_00009	ACLY	-			
4066	-28.87	kd	CGS001-8892	EIF2B2	-			
4067	-28.88	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
4068	-28.88	kd	CGS001-5586	PKN2	Protein kinase N (PKN) family			
4069	-28.89	kd	CGS001-3149	HMGB3	High-mobility group / Canonical			
4070	-28.92	oe	ccsbBroad304_00316	CKS1B	-			
4071	-28.95	kd	CGS001-3673	ITGA2	Integrins			
4072	-28.95	kd	CGS001-55082	ARGLU1	-			
4073	-28.96	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
4074	-28.97	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
4075	-29	kd	CGS001-6277	S100A6	EF-hand domain containing			
4076	-29.01	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
4077	-29.02	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
4078	-29.1	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
4079	-29.12	kd	CGS001-26520	TIMM9	-			
4080	-29.17	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
4081	-29.19	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
4082	-29.2	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
4083	-29.23	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
4084	-29.24	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
4085	-29.28	kd	CGS001-10477	UBE2E3	Ubiquitin-conjugating enzymes E2			
4086	-29.28	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
4087	-29.29	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
4088	-29.29	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
4089	-29.29	kd	CGS001-5106	PCK2	-			
4090	-29.33	kd	CGS001-5036	PA2G4	-			
4091	-29.35	cc		FXR antagonist	-			
4092	-29.36	kd	CGS001-1030	CDKN2B	-			
4093	-29.38	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
4094	-29.38	oe	ccsbBroad304_06574	MDH2	-			
4095	-29.48	kd	CGS001-2852	GPER	-			
4096	-29.49	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
4097	-29.51	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
4098	-29.54	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
4099	-29.58	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
4100	-29.65	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
4101	-29.68	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
4102	-29.68	kd	CGS001-5427	POLE2	DNA polymerases			
4103	-29.71	kd	CGS001-10645	CAMKK2	Meta subfamily			
4104	-29.71	kd	CGS001-4088	SMAD3	SMADs			
4105	-29.71	kd	CGS001-1763	DNA2	-			
4106	-29.74	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
4107	-29.75	oe	ccsbBroad304_01787	YES1	Src family			
4108	-29.75	oe	ccsbBroad304_01624	SUPV3L1	-			
4109	-29.77	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
4110	-29.8	kd	CGS001-27102	EIF2AK1	Other PEK family kinases			
4111	-29.82	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
4112	-29.88	kd	CGS001-51271	UBAP1	-			
4113	-29.91	oe	ccsbBroad304_06889	RPN2	-			
4114	-29.91	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
4115	-29.93	kd	CGS001-5696	PSMB8	Proteasome (prosome, macropain) subunits			
4116	-29.94	cc		S100 calcium binding proteins LOF	-			
4117	-29.95	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
4118	-29.96	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4119	-29.97	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
4120	-29.97	oe	ccsbBroad304_01061	NAB2	-			
4121	-29.97	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
4122	-29.98	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
4123	-30	cc		Akt Signaling LOF	-			
4124	-30	kd	CGS001-10252	SPRY1	-			
4125	-30.03	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
4126	-30.03	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
4127	-30.06	oe	ccsbBroad304_00600	FYN	Src family			
4128	-30.07	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
4129	-30.08	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
4130	-30.09	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
4131	-30.1	oe	ccsbBroad304_00964	SMAD7	SMADs			
4132	-30.14	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
4133	-30.16	kd	CGS001-84290	CAPNS2	EF-hand domain containing			
4134	-30.17	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
4135	-30.23	kd	CGS001-23475	QPRT	-			
4136	-30.26	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
4137	-30.27	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
4138	-30.29	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
4139	-30.3	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
4140	-30.31	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
4141	-30.31	kd	CGS001-2079	ERH	-			
4142	-30.32	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
4143	-30.44	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
4144	-30.45	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
4145	-30.46	kd	CGS001-3566	IL4R	IL-2 receptor family			
4146	-30.49	oe	ccsbBroad304_01754	UCK2	-			
4147	-30.5	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
4148	-30.53	kd	CGS001-9308	CD83	CD molecules			
4149	-30.54	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
4150	-30.56	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4151	-30.58	kd	CGS001-7079	TIMP4	-			
4152	-30.6	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
4153	-30.61	oe	ccsbBroad304_00519	ETFB	-			
4154	-30.61	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
4155	-30.63	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4156	-30.63	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
4157	-30.64	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
4158	-30.65	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
4159	-30.69	oe	ccsbBroad304_07478	CCP110	-			
4160	-30.71	oe	ccsbBroad304_03933	CARD9	-			
4161	-30.72	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
4162	-30.73	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
4163	-30.74	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
4164	-30.77	kd	CGS001-8702	B4GALT4	Beta 4-glycosyltransferases			
4165	-30.78	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
4166	-30.78	kd	CGS001-6741	SSB	La ribonucleoprotein domain containing			
4167	-30.8	kd	CGS001-5451	POU2F1	Homeoboxes / POU class			
4168	-30.82	oe	ccsbBroad304_04257	SPRY4	-			
4169	-30.82	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
4170	-30.84	cp	BRD-K29653726	topiramate	Carbonic anhydrase inhibitor		CA2, CA4, GRIK1, CA1, CA12, CA7, CYP2C19, CYP3A4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA1, SCN1A, SCN5A	Carbonic anhydrase inhibitor, Glutamate receptor antagonist, Kainate receptor antagonist
4171	-30.86	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4172	-30.87	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
4173	-30.88	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
4174	-30.89	cc		Tubulin inhibitor	-			
4175	-30.89	kd	CGS001-10987	COPS5	-			
4176	-30.91	oe	ccsbBroad304_00888	ITPK1	-			
4177	-30.95	kd	CGS001-3596	IL13	Interleukins and interleukin receptors			
4178	-30.97	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
4179	-30.97	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
4180	-30.98	oe	ccsbBroad304_06765	PRCC	-			
4181	-30.98	kd	CGS001-6233	RPS27A	S ribosomal proteins			
4182	-31.01	cp	BRD-K41903098	diphenoxylate	Opioid receptor agonist		OPRM1, OPRD1	Opioid receptor agonist
4183	-31.05	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
4184	-31.08	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
4185	-31.11	kd	CGS001-23588	KLHDC2	-			
4186	-31.12	kd	CGS001-4023	LPL	-			
4187	-31.13	oe	ccsbBroad304_02569	BTG3	-			
4188	-31.19	kd	CGS001-57215	THAP11	THAP (C2CH-type zinc finger) domain containing			
4189	-31.2	kd	CGS001-9787	DLGAP5	-			
4190	-31.28	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
4191	-31.28	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
4192	-31.31	kd	CGS001-57147	SCYL3	-			
4193	-31.36	kd	CGS001-7849	PAX8	Paired boxes			
4194	-31.41	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
4195	-31.42	kd	CGS001-51547	SIRT7	Histone deacetylases (HDACs)			
4196	-31.43	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
4197	-31.44	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
4198	-31.45	kd	CGS001-3998	LMAN1	-			
4199	-31.46	oe	ccsbBroad304_00329	CLTA	-			
4200	-31.47	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
4201	-31.47	kd	CGS001-2235	FECH	-			
4202	-31.5	cp	BRD-K96740444	itopride	Dopamine receptor antagonist		DRD2, ACHE, CHRM3	Dopamine receptor antagonist
4203	-31.51	cp	BRD-K33106058	cytarabine	Ribonucleotide reductase inhibitor		POLB, POLA1	Ribonucleotide reductase inhibitor
4204	-31.54	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
4205	-31.55	kd	CGS001-4097	MAFG	-			
4206	-31.57	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
4207	-31.58	kd	CGS001-4907	NT5E	Adenosine turnover			
4208	-31.59	oe	ccsbBroad304_00146	BAD	-			
4209	-31.59	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
4210	-31.61	oe	ccsbBroad304_07808	RAB11FIP2	-			
4211	-31.61	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
4212	-31.63	kd	CGS001-6944	VPS72	-			
4213	-31.64	kd	CGS001-9406	ZRANB2	Zinc fingers, RAN-binding domain containing			
4214	-31.69	oe	ccsbBroad304_00957	M6PR	-			
4215	-31.7	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
4216	-31.71	kd	CGS001-5371	PML	RING-type (C3HC4) zinc fingers			
4217	-31.73	kd	CGS001-1184	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
4218	-31.76	kd	CGS001-7533	YWHAH	-			
4219	-31.78	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
4220	-31.79	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
4221	-31.8	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
4222	-31.84	kd	CGS001-10058	ABCB6	ATP binding cassette transporters / subfamily B			
4223	-31.86	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
4224	-31.86	kd	CGS001-840	CASP7	Caspases			
4225	-31.9	oe	ccsbBroad304_06820	PTS	-			
4226	-31.97	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
4227	-31.97	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
4228	-31.98	kd	CGS001-6098	ROS1	Type XVII RTKs: ROS receptors			
4229	-31.98	kd	CGS001-51734	SEPX1	-			
4230	-31.98	kd	CGS001-2287	FKBP3	-			
4231	-32.02	kd	CGS001-5612	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
4232	-32.03	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
4233	-32.05	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
4234	-32.05	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
4235	-32.07	kd	CGS001-1528	CYB5A	Cytochrome b genes			
4236	-32.08	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4237	-32.14	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
4238	-32.15	kd	CGS001-6794	STK11	LKB subfamily			
4239	-32.18	cp	BRD-K99063460	didanosine	Nucleoside reverse transcriptase inhibitor		PNP	Nucleoside reverse transcriptase inhibitor
4240	-32.18	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
4241	-32.19	kd	CGS001-8334	HIST1H2AC	Histones / Replication-dependent			
4242	-32.2	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
4243	-32.21	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
4244	-32.22	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
4245	-32.27	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
4246	-32.28	cc		Serotonin receptor antagonist	-			
4247	-32.28	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
4248	-32.29	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
4249	-32.29	kd	CGS001-384	ARG2	Arginase			
4250	-32.35	kd	CGS001-1827	RCAN1	-			
4251	-32.37	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
4252	-32.39	oe	ccsbBroad304_00510	EPHX2	-			
4253	-32.4	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
4254	-32.4	kd	CGS001-6715	SRD5A1	-			
4255	-32.44	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
4256	-32.48	oe	ccsbBroad304_01205	PIN1	-			
4257	-32.48	kd	CGS001-7086	TKT	-			
4258	-32.48	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4259	-32.48	oe	ccsbBroad304_01613	STK11	LKB subfamily			
4260	-32.49	cc		Cyclin dependent kinases LOF	-			
4261	-32.5	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
4262	-32.53	kd	CGS001-7167	TPI1	-			
4263	-32.54	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
4264	-32.55	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
4265	-32.64	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
4266	-32.65	kd	CGS001-2776	GNAQ	-			
4267	-32.67	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
4268	-32.67	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
4269	-32.72	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
4270	-32.74	oe	ccsbBroad304_03177	FIS1	-			
4271	-32.75	kd	CGS001-222546	RFX6	-			
4272	-32.75	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
4273	-32.76	cp	BRD-K33483813	actarit	Interleukin receptor agonist			Interleukin receptor agonist
4274	-32.79	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
4275	-32.81	oe	ccsbBroad304_02875	BRP44	-			
4276	-32.82	kd	CGS001-9290	GPR55	GPCR / Class A : Orphans			
4277	-32.83	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
4278	-32.85	kd	CGS001-9134	CCNE2	-			
4279	-32.89	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
4280	-32.9	kd	CGS001-55818	KDM3A	Histone demethylases			
4281	-32.96	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
4282	-32.99	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
4283	-33	oe	ccsbBroad304_07561	YAF2	-			
4284	-33.03	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
4285	-33.03	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
4286	-33.04	kd	CGS001-2015	EMR1	Adhesion Class GPCRs			
4287	-33.06	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
4288	-33.07	kd	CGS001-152	ADRA2C	GPCR / Class A : Adrenoceptors : alpha			
4289	-33.11	oe	ccsbBroad304_00709	GUK1	-			
4290	-33.11	kd	CGS001-8659	ALDH4A1	Aldehyde dehydrogenases			
4291	-33.12	kd	CGS001-11200	CHEK2	CHK1 subfamily			
4292	-33.13	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
4293	-33.14	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
4294	-33.16	kd	CGS001-23266	LPHN2	Adhesion Class GPCRs			
4295	-33.17	kd	CGS001-5645	PRSS2	Serine peptidases			
4296	-33.18	kd	CGS001-595	CCND1	-			
4297	-33.19	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
4298	-33.19	kd	CGS001-6303	SAT1	-			
4299	-33.21	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
4300	-33.27	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
4301	-33.28	kd	CGS001-3420	IDH3B	-			
4302	-33.3	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
4303	-33.31	kd	CGS001-121599	SPIC	ETS Transcription Factors			
4304	-33.35	kd	CGS001-9140	ATG12	-			
4305	-33.38	kd	CGS001-55632	G2E3	Zinc fingers, PHD-type			
4306	-33.39	oe	ccsbBroad304_06294	GNAZ	-			
4307	-33.41	kd	CGS001-29079	MED4	-			
4308	-33.42	oe	ccsbBroad304_01052	MYB	-			
4309	-33.42	oe	ccsbBroad304_02052	KYNU	-			
4310	-33.43	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
4311	-33.44	oe	ccsbBroad304_01084	NEU1	-			
4312	-33.44	kd	CGS001-178	AGL	-			
4313	-33.45	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
4314	-33.46	oe	ccsbBroad304_02349	MPHOSPH9	-			
4315	-33.48	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
4316	-33.48	oe	ccsbBroad304_06089	DDIT3	-			
4317	-33.49	oe	ccsbBroad304_02086	PDLIM1	-			
4318	-33.53	kd	CGS001-5257	PHKB	-			
4319	-33.54	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
4320	-33.54	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
4321	-33.58	kd	CGS001-10390	CEPT1	-			
4322	-33.59	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
4323	-33.59	kd	CGS001-4069	LYZ	-			
4324	-33.63	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
4325	-33.64	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
4326	-33.65	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
4327	-33.7	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
4328	-33.73	oe	ccsbBroad304_00818	IDH3A	-			
4329	-33.77	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
4330	-33.79	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
4331	-33.83	kd	CGS001-2864	FFAR1	Fatty acid receptors			
4332	-33.84	kd	CGS001-29915	HCFC2	-			
4333	-33.85	kd	CGS001-3957	LGALS2	Lectins, galactoside-binding			
4334	-33.88	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
4335	-33.92	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
4336	-33.95	kd	CGS001-10641	NPRL2	-			
4337	-33.96	kd	CGS001-10447	FAM3C	-			
4338	-33.98	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
4339	-34.01	oe	ccsbBroad304_02671	ECD	-			
4340	-34.05	kd	CGS001-27035	NOX1	-			
4341	-34.08	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
4342	-34.08	kd	CGS001-9412	MED21	-			
4343	-34.08	kd	CGS001-6790	AURKA	Aurora kinase			
4344	-34.09	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
4345	-34.17	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
4346	-34.18	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
4347	-34.2	kd	CGS001-839	CASP6	Caspases			
4348	-34.23	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
4349	-34.26	kd	CGS001-8848	TSC22D1	-			
4350	-34.26	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
4351	-34.28	oe	ccsbBroad304_01222	PLP2	-			
4352	-34.28	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
4353	-34.34	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
4354	-34.34	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
4355	-34.35	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
4356	-34.39	cc		Mediator complex LOF	-			
4357	-34.42	kd	CGS001-25913	POT1	-			
4358	-34.43	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
4359	-34.48	kd	CGS001-7534	YWHAZ	-			
4360	-34.5	kd	CGS001-147837	ZNF563	Zinc fingers, C2H2-type			
4361	-34.51	kd	CGS001-5335	PLCG1	Phosphoinositide-specific phospholipase C			
4362	-34.57	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
4363	-34.58	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
4364	-34.59	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
4365	-34.59	kd	CGS001-5891	MOK	RCK family			
4366	-34.6	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4367	-34.6	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
4368	-34.64	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
4369	-34.65	kd	CGS001-57026	PDXP	-			
4370	-34.66	oe	ccsbBroad304_09284	UBE3B	-			
4371	-34.74	kd	CGS001-58472	SQRDL	-			
4372	-34.76	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
4373	-34.77	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
4374	-34.78	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
4375	-34.79	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
4376	-34.82	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
4377	-34.83	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
4378	-34.88	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
4379	-34.9	oe	ccsbBroad304_03266	ERGIC2	-			
4380	-34.91	kd	CGS001-22930	RAB3GAP1	-			
4381	-34.92	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
4382	-34.94	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
4383	-34.96	kd	CGS001-5387	PMS2P3	-			
4384	-34.96	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
4385	-34.97	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
4386	-34.98	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
4387	-34.98	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4388	-35	kd	CGS001-51002	TPRKB	-			
4389	-35.01	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
4390	-35.06	kd	CGS001-9870	KIAA0317	-			
4391	-35.08	kd	CGS001-7371	UCK2	-			
4392	-35.13	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
4393	-35.14	oe	ccsbBroad304_01951	BLZF1	-			
4394	-35.14	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
4395	-35.15	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4396	-35.16	kd	CGS001-25966	C2CD2	-			
4397	-35.19	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
4398	-35.21	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
4399	-35.22	cc		FGFR inhibitor	-			
4400	-35.22	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
4401	-35.23	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
4402	-35.24	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
4403	-35.24	cp	BRD-K70358946	aripiprazole	Serotonin receptor agonist		DRD2, HTR1A, HTR2A, HRH1, HTR1B, HTR1D, HTR2C, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR1E, HTR3A, HTR6, HTR7	Serotonin receptor agonist, Serotonin receptor antagonist
4404	-35.27	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
4405	-35.31	kd	CGS001-80135	RPF1	-			
4406	-35.33	oe	ccsbBroad304_07851	FAM120A	-			
4407	-35.37	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
4408	-35.38	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4409	-35.42	kd	CGS001-6722	SRF	-			
4410	-35.43	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
4411	-35.44	oe	ccsbBroad304_02589	COPS5	-			
4412	-35.45	oe	ccsbBroad304_01034	MSH2	-			
4413	-35.46	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
4414	-35.47	kd	CGS001-4724	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
4415	-35.49	oe	ccsbBroad304_00836	IGF2	-			
4416	-35.5	kd	CGS001-9377	COX5A	Mitochondrial respiratory chain complex			
4417	-35.59	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
4418	-35.61	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
4419	-35.63	kd	CGS001-25942	SIN3A	-			
4420	-35.65	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
4421	-35.65	oe	ccsbBroad304_09358	MAPK1IP1L	-			
4422	-35.67	kd	CGS001-2568	GABRP	GABA receptors			
4423	-35.68	kd	CGS001-9670	IPO13	Importins			
4424	-35.7	oe	ccsbBroad304_00237	CCND3	-			
4425	-35.7	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
4426	-35.71	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
4427	-35.72	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
4428	-35.72	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4429	-35.73	oe	ccsbBroad304_01091	NFIB	-			
4430	-35.74	kd	CGS001-894	CCND2	-			
4431	-35.75	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
4432	-35.77	oe	ccsbBroad304_08365	CYCS	-			
4433	-35.78	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
4434	-35.79	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4435	-35.81	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4436	-35.83	kd	CGS001-5306	PITPNA	-			
4437	-35.85	kd	CGS001-6016	RIT1	-			
4438	-35.85	kd	CGS001-4798	NFRKB	INO80 complex subunits			
4439	-35.87	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
4440	-35.89	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
4441	-35.92	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
4442	-35.92	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
4443	-35.93	kd	CGS001-4323	MMP14	Matrix metallopeptidase			
4444	-35.95	kd	CGS001-1949	EFNB3	Ephrins			
4445	-35.96	oe	ccsbBroad304_06523	LIG1	-			
4446	-35.96	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
4447	-35.97	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
4448	-36.01	kd	CGS001-6621	SNAPC4	-			
4449	-36.02	kd	CGS001-7272	TTK	TTK family			
4450	-36.03	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
4451	-36.03	kd	CGS001-8233	ZRSR2	RNA binding motif (RRM) containing			
4452	-36.05	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
4453	-36.06	kd	CGS001-10465	PPIH	-			
4454	-36.06	kd	CGS001-34	ACADM	-			
4455	-36.11	kd	CGS001-7175	TPR	-			
4456	-36.11	kd	CGS001-5359	PLSCR1	-			
4457	-36.13	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
4458	-36.16	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
4459	-36.2	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
4460	-36.23	kd	CGS001-2896	GRN	-			
4461	-36.26	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
4462	-36.26	kd	CGS001-837	CASP4	Caspases			
4463	-36.27	oe	ccsbBroad304_08840	KIF9	Kinesins			
4464	-36.27	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
4465	-36.28	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
4466	-36.29	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
4467	-36.29	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
4468	-36.3	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
4469	-36.36	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
4470	-36.36	kd	CGS001-23429	RYBP	-			
4471	-36.38	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
4472	-36.44	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
4473	-36.47	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4474	-36.47	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
4475	-36.47	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
4476	-36.48	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
4477	-36.49	oe	ccsbBroad304_03164	MTERFD1	-			
4478	-36.49	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
4479	-36.52	kd	CGS001-2194	FASN	Short chain dehydrogenase/reductase superfamily / Atypical members			
4480	-36.53	oe	ccsbBroad304_01164	PDHB	-			
4481	-36.54	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
4482	-36.57	kd	CGS001-6502	SKP2	F-boxes / Leucine-rich repeats			
4483	-36.58	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
4484	-36.59	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
4485	-36.66	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
4486	-36.71	kd	CGS001-5037	PEBP1	-			
4487	-36.74	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
4488	-36.75	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
4489	-36.8	oe	ccsbBroad304_03089	PACSIN3	-			
4490	-36.85	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
4491	-36.86	kd	CGS001-29105	C16ORF80	-			
4492	-36.9	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
4493	-36.92	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
4494	-36.94	kd	CGS001-8313	AXIN2	-			
4495	-36.97	kd	CGS001-2002	ELK1	ETS Transcription Factors			
4496	-36.98	cc		IL4 Pathway LOF	-			
4497	-36.98	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
4498	-37.02	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
4499	-37.02	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
4500	-37.02	kd	CGS001-9404	LPXN	-			
4501	-37.02	kd	CGS001-4680	CEACAM6	CD molecules			
4502	-37.03	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
4503	-37.04	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
4504	-37.04	kd	CGS001-79073	TMEM109	-			
4505	-37.05	kd	CGS001-5411	PNN	-			
4506	-37.06	kd	CGS001-129685	TAF8	-			
4507	-37.07	kd	CGS001-10142	AKAP9	A-kinase anchor proteins			
4508	-37.09	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
4509	-37.11	cp	BRD-A12560204	nitrendipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1H, CACNA1S, CACNA2D2, CACNB2, CACNG1, KCNN4	Calcium channel blocker
4510	-37.13	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
4511	-37.13	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
4512	-37.13	kd	CGS001-462	SERPINC1	Serine (or cysteine) peptidase inhibitors			
4513	-37.14	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
4514	-37.14	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
4515	-37.14	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
4516	-37.17	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
4517	-37.19	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
4518	-37.22	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
4519	-37.23	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
4520	-37.24	kd	CGS001-29763	PACSIN3	-			
4521	-37.25	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4522	-37.27	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
4523	-37.27	kd	CGS001-2958	GTF2A2	General transcription factors			
4524	-37.31	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
4525	-37.33	cc		Vitamin D receptor agonist	-			
4526	-37.36	oe	ccsbBroad304_06367	HK1	-			
4527	-37.36	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
4528	-37.41	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
4529	-37.45	kd	CGS001-978	CDA	-			
4530	-37.49	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
4531	-37.52	oe	ccsbBroad304_02772	ICMT	-			
4532	-37.54	kd	CGS001-84647	PLA2G12B	-			
4533	-37.56	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
4534	-37.58	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
4535	-37.6	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
4536	-37.61	kd	CGS001-9263	STK17A	Death-associated kinase (DAPK) family			
4537	-37.62	kd	CGS001-8192	CLPP	ATPases / AAA-type			
4538	-37.63	oe	ccsbBroad304_08825	LHPP	-			
4539	-37.63	cp	BRD-A75935363	atracurium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
4540	-37.63	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
4541	-37.64	kd	CGS001-29968	PSAT1	-			
4542	-37.65	kd	CGS001-9326	ZNHIT3	Zinc fingers, HIT-type			
4543	-37.66	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
4544	-37.69	oe	ccsbBroad304_03746	CDC42SE1	-			
4545	-37.69	kd	CGS001-23211	ZC3H4	Zinc fingers, CCCH-type domain containing			
4546	-37.71	kd	CGS001-3601	IL15RA	IL-2 receptor family			
4547	-37.72	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
4548	-37.73	kd	CGS001-405	ARNT	Basic helix-loop-helix proteins			
4549	-37.81	cc		EMSY complex LOF	-			
4550	-37.82	kd	CGS001-3927	LASP1	-			
4551	-37.86	cc		Histone deacetylases LOF	-			
4552	-37.86	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
4553	-37.88	kd	CGS001-54106	TLR9	Toll-like receptor family			
4554	-37.9	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
4555	-37.91	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
4556	-37.94	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
4557	-37.96	kd	CGS001-29110	TBK1	IKK family			
4558	-38.04	kd	CGS001-1633	DCK	-			
4559	-38.05	oe	ccsbBroad304_13598	NRBP2	NRBP family			
4560	-38.11	oe	ccsbBroad304_08709	SCYL3	-			
4561	-38.11	oe	ccsbBroad304_06278	GK	Glycerol kinases			
4562	-38.12	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
4563	-38.14	oe	ccsbBroad304_01102	NMT1	-			
4564	-38.18	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
4565	-38.2	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
4566	-38.2	oe	ccsbBroad304_00632	GGCX	Carboxylases			
4567	-38.2	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
4568	-38.23	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
4569	-38.25	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
4570	-38.26	oe	ccsbBroad304_00161	BID	Endogenous ligands			
4571	-38.28	kd	CGS001-10906	TRAFD1	-			
4572	-38.32	oe	ccsbBroad304_02416	TUBB4B	-			
4573	-38.33	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4574	-38.34	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
4575	-38.35	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
4576	-38.37	oe	ccsbBroad304_00509	EPHX1	-			
4577	-38.38	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
4578	-38.39	kd	CGS001-9380	GRHPR	-			
4579	-38.43	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
4580	-38.45	oe	ccsbBroad304_01654	TCTA	-			
4581	-38.49	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
4582	-38.5	kd	CGS001-3421	IDH3G	-			
4583	-38.51	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
4584	-38.52	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
4585	-38.53	oe	ccsbBroad304_00564	FGR	Src family			
4586	-38.54	kd	CGS001-3476	IGBP1	-			
4587	-38.55	oe	ccsbBroad304_04170	PANK2	-			
4588	-38.6	oe	ccsbBroad304_09708	PNLDC1	-			
4589	-38.63	oe	ccsbBroad304_01147	PC	Carboxylases			
4590	-38.66	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
4591	-38.72	oe	ccsbBroad304_02708	TRIM32	-			
4592	-38.74	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
4593	-38.77	kd	CGS001-3682	ITGAE	Integrins			
4594	-38.78	kd	CGS001-3725	JUN	basic leucine zipper proteins			
4595	-38.78	kd	CGS001-9867	PJA2	RING-type (C3HC4) zinc fingers			
4596	-38.83	kd	CGS001-55699	IARS2	Aminoacyl tRNA synthetases / Class I			
4597	-38.84	kd	CGS001-6347	CCL2	Chemokine ligands			
4598	-38.87	kd	CGS001-9687	GREB1	-			
4599	-38.89	kd	CGS001-6275	S100A4	EF-hand domain containing			
4600	-38.89	kd	CGS001-29937	NENF	-			
4601	-38.91	cp	BRD-K07237224	moclobemide	Monoamine oxidase inhibitor		MAOA, CYP2C19, MAOB	Monoamine oxidase inhibitor
4602	-38.92	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
4603	-38.96	oe	ccsbBroad304_06518	LDHA	-			
4604	-38.96	kd	CGS001-122809	SOCS4	SH2 domain containing			
4605	-38.97	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
4606	-38.97	oe	ccsbBroad304_02197	VPS26A	-			
4607	-38.99	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
4608	-39.01	oe	ccsbBroad304_00985	MCL1	-			
4609	-39.02	oe	ccsbBroad304_06134	ECH1	-			
4610	-39.06	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
4611	-39.11	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
4612	-39.11	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
4613	-39.14	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
4614	-39.14	oe	ccsbBroad304_01146	PARN	-			
4615	-39.14	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
4616	-39.16	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
4617	-39.16	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
4618	-39.18	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4619	-39.21	kd	CGS001-56889	TM9SF3	-			
4620	-39.24	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
4621	-39.27	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
4622	-39.28	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
4623	-39.29	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
4624	-39.33	oe	ccsbBroad304_00418	CD55	CD molecules			
4625	-39.33	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
4626	-39.34	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
4627	-39.36	oe	ccsbBroad304_05192	SPRED2	-			
4628	-39.37	kd	CGS001-3559	IL2RA	IL-2 receptor family			
4629	-39.46	kd	CGS001-10557	RPP38	-			
4630	-39.47	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
4631	-39.49	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
4632	-39.52	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
4633	-39.58	kd	CGS001-4144	MAT2A	-			
4634	-39.58	kd	CGS001-25948	KBTBD2	BTB/POZ domain containing			
4635	-39.59	kd	CGS001-7846	TUBA1A	Tubulins			
4636	-39.6	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
4637	-39.6	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4638	-39.61	oe	ccsbBroad304_08152	PSAT1	-			
4639	-39.62	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
4640	-39.63	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
4641	-39.64	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
4642	-39.64	kd	CGS001-4129	MAOB	Catecholamine turnover			
4643	-39.65	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
4644	-39.65	kd	CGS001-10681	GNB5	WD repeat domain containing			
4645	-39.66	kd	CGS001-5445	PON2	Paraoxonases			
4646	-39.77	kd	CGS001-6271	S100A1	EF-hand domain containing			
4647	-39.78	kd	CGS001-5355	PLP2	-			
4648	-39.8	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
4649	-39.82	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
4650	-39.82	oe	ccsbBroad304_08461	CDCA4	-			
4651	-39.83	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
4652	-39.84	kd	CGS001-1312	COMT	Catecholamine turnover			
4653	-39.85	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
4654	-39.86	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
4655	-39.87	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
4656	-39.87	kd	CGS001-2010	EMD	-			
4657	-39.89	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
4658	-39.93	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
4659	-39.94	cc		EIF Proteins LOF	-			
4660	-39.94	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4661	-39.95	oe	ccsbBroad304_03080	C16ORF80	-			
4662	-39.95	kd	CGS001-54512	EXOSC4	-			
4663	-39.96	oe	ccsbBroad304_02840	PISD	Decarboxylases			
4664	-39.98	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
4665	-39.98	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
4666	-40.06	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
4667	-40.07	kd	CGS001-2017	CTTN	-			
4668	-40.09	kd	CGS001-9903	KLHL21	BTB/POZ domain containing			
4669	-40.1	kd	CGS001-960	CD44	CD molecules			
4670	-40.11	oe	ccsbBroad304_13633	PI4KAP2	-			
4671	-40.11	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
4672	-40.14	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
4673	-40.14	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
4674	-40.16	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
4675	-40.17	kd	CGS001-9184	BUB3	WD repeat domain containing			
4676	-40.28	kd	CGS001-205	AK4	Adenylate kinases			
4677	-40.3	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
4678	-40.32	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
4679	-40.33	kd	CGS001-51181	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4680	-40.38	kd	CGS001-10553	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
4681	-40.4	kd	CGS001-2048	EPHB2	Type XIII RTKs: Ephrin receptor family			
4682	-40.4	oe	ccsbBroad304_06383	HMMR	CD molecules			
4683	-40.41	cp	BRD-K18895904	olanzapine	Dopamine receptor antagonist		DRD2, HTR2A, HTR2C, DRD1, DRD3, DRD4, HRH1, HTR1A, HTR1B, HTR1D, HTR1E, HTR6, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C8, DRD5, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH2, HRH4, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
4684	-40.43	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
4685	-40.5	kd	CGS001-8743	TNFSF10	CD molecules			
4686	-40.5	kd	CGS001-29959	NRBP1	NRBP family			
4687	-40.52	kd	CGS001-19	ABCA1	ATP binding cassette transporters / subfamily A			
4688	-40.55	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
4689	-40.56	oe	ccsbBroad304_02012	FADD	-			
4690	-40.6	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
4691	-40.64	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
4692	-40.68	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
4693	-40.7	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
4694	-40.72	kd	CGS001-10797	MTHFD2	-			
4695	-40.73	cc		PI3K inhibitor	-			
4696	-40.73	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
4697	-40.73	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
4698	-40.82	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4699	-40.83	oe	ccsbBroad304_02956	EHF	-			
4700	-40.85	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
4701	-40.86	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
4702	-40.88	cp	BRD-K29530284	amlexanox	Histamine receptor modulator		FGF1, IL3, S100A12, S100A13	Histamine receptor modulator
4703	-40.92	oe	ccsbBroad304_02361	MFSD10	-			
4704	-40.93	cp	BRD-K48932581	cetraxate	Mucus protecting agent		GAST	Mucus protecting agent
4705	-40.99	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
4706	-41.02	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
4707	-41.03	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
4708	-41.03	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
4709	-41.04	cc		Vesicular Transport LOF	-			
4710	-41.05	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
4711	-41.06	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
4712	-41.06	kd	CGS001-6194	RPS6	S ribosomal proteins			
4713	-41.07	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
4714	-41.11	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4715	-41.11	kd	CGS001-3109	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
4716	-41.13	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
4717	-41.16	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
4718	-41.17	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
4719	-41.18	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
4720	-41.2	kd	CGS001-4170	MCL1	-			
4721	-41.21	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
4722	-41.27	cp	BRD-A24543851	nornicotine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
4723	-41.32	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4724	-41.37	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
4725	-41.4	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
4726	-41.4	kd	CGS001-415116	PIM3	PIM family			
4727	-41.49	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
4728	-41.55	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
4729	-41.56	oe	ccsbBroad304_13998	PDXK	-			
4730	-41.56	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
4731	-41.58	kd	CGS001-8896	BUD31	-			
4732	-41.61	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
4733	-41.63	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
4734	-41.68	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
4735	-41.69	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
4736	-41.72	kd	CGS001-771	CA12	Carbonic anhydrases			
4737	-41.73	kd	CGS001-2853	GPR31	GPCR / Class A : Orphans			
4738	-41.82	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
4739	-41.82	kd	CGS001-10891	PPARGC1A	RNA binding motif (RRM) containing			
4740	-41.87	oe	ccsbBroad304_07662	NPRL2	-			
4741	-41.88	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
4742	-41.92	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
4743	-41.95	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
4744	-41.96	oe	ccsbBroad304_06286	GLUL	-			
4745	-42	kd	CGS001-4300	MLLT3	-			
4746	-42.03	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
4747	-42.05	oe	ccsbBroad304_07843	FCHO1	-			
4748	-42.05	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
4749	-42.08	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
4750	-42.11	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
4751	-42.14	kd	CGS001-6827	SUPT4H1	-			
4752	-42.2	kd	CGS001-23387	SIK3	QIK subfamily			
4753	-42.22	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
4754	-42.27	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
4755	-42.28	oe	ccsbBroad304_07506	UBAP2L	-			
4756	-42.3	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
4757	-42.32	oe	ccsbBroad304_00420	DAP	-			
4758	-42.32	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
4759	-42.33	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
4760	-42.36	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
4761	-42.41	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
4762	-42.43	kd	CGS001-2877	GPX2	-			
4763	-42.44	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4764	-42.47	oe	ccsbBroad304_05823	ANXA2	Annexins			
4765	-42.48	kd	CGS001-83637	ZMIZ2	Zinc fingers, MIZ-type			
4766	-42.49	kd	CGS001-7100	TLR5	Toll-like receptor family			
4767	-42.52	oe	ccsbBroad304_06126	TSC22D3	-			
4768	-42.58	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
4769	-42.58	kd	CGS001-10898	CPSF4	-			
4770	-42.6	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
4771	-42.6	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
4772	-42.61	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
4773	-42.65	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
4774	-42.65	kd	CGS001-51160	VPS28	-			
4775	-42.65	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
4776	-42.7	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
4777	-42.75	kd	CGS001-55662	HIF1AN	-			
4778	-42.8	kd	CGS001-65243	ZNF643	-			
4779	-42.8	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
4780	-42.82	kd	CGS001-1642	DDB1	-			
4781	-42.83	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
4782	-42.92	kd	CGS001-3832	KIF11	Kinesins			
4783	-42.96	cp	BRD-K33312228	halometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4784	-43.04	oe	ccsbBroad304_07834	GGA2	-			
4785	-43.09	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
4786	-43.09	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4787	-43.16	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
4788	-43.22	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
4789	-43.22	kd	CGS001-3373	HYAL1	-			
4790	-43.23	kd	CGS001-1616	DAXX	-			
4791	-43.24	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
4792	-43.24	oe	ccsbBroad304_02566	MORF4L1	-			
4793	-43.28	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
4794	-43.28	oe	ccsbBroad304_00529	F3	CD molecules			
4795	-43.28	kd	CGS001-3575	IL7R	IL-2 receptor family			
4796	-43.29	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
4797	-43.3	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
4798	-43.32	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
4799	-43.37	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
4800	-43.4	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
4801	-43.41	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4802	-43.41	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
4803	-43.42	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
4804	-43.43	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
4805	-43.44	cc		Aromatase inhibitor	-			
4806	-43.45	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
4807	-43.46	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
4808	-43.46	kd	CGS001-1407	CRY1	-			
4809	-43.47	cp	BRD-K69650333	idarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4810	-43.48	kd	CGS001-3034	HAL	-			
4811	-43.55	kd	CGS001-5898	RALA	-			
4812	-43.56	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
4813	-43.57	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
4814	-43.65	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
4815	-43.67	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
4816	-43.75	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
4817	-43.81	oe	ccsbBroad304_07515	GFPT2	-			
4818	-43.83	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
4819	-43.83	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
4820	-43.83	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
4821	-43.85	kd	CGS001-8764	TNFRSF14	Tumour necrosis factor (TNF) receptor family			
4822	-43.86	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
4823	-43.86	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
4824	-43.88	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
4825	-43.89	kd	CGS001-23062	GGA2	-			
4826	-43.9	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
4827	-43.91	kd	CGS001-9748	SLK	SLK subfamily			
4828	-43.95	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
4829	-43.97	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
4830	-44	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
4831	-44.01	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
4832	-44.02	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
4833	-44.03	kd	CGS001-9541	CIR1	-			
4834	-44.06	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
4835	-44.07	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
4836	-44.18	kd	CGS001-53343	NUDT9	Nudix motif containing			
4837	-44.23	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
4838	-44.23	kd	CGS001-634	CEACAM1	CD molecules			
4839	-44.26	kd	CGS001-51548	SIRT6	Histone deacetylases (HDACs)			
4840	-44.29	kd	CGS001-2030	SLC29A1	SLC29 family			
4841	-44.41	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
4842	-44.42	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
4843	-44.45	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
4844	-44.47	oe	ccsbBroad304_01672	TIMP2	-			
4845	-44.48	oe	ccsbBroad304_01398	RHEB	-			
4846	-44.56	kd	CGS001-25989	ULK3	Unc-51-like kinase (ULK) family			
4847	-44.58	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
4848	-44.59	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4849	-44.6	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
4850	-44.6	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
4851	-44.6	kd	CGS001-55577	NAGK	-			
4852	-44.6	kd	CGS001-8895	CPNE3	-			
4853	-44.65	kd	CGS001-80274	SCUBE1	-			
4854	-44.72	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
4855	-44.73	oe	ccsbBroad304_09503	KLHDC9	-			
4856	-44.76	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4857	-44.76	kd	CGS001-55012	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4858	-44.82	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
4859	-44.85	kd	CGS001-5292	PIM1	PIM family			
4860	-44.86	cc		Nucleoporin LOF	-			
4861	-44.89	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
4862	-44.9	kd	CGS001-84669	USP32	EF-hand domain containing			
4863	-44.97	kd	CGS001-10525	HYOU1	Heat shock proteins / HSP70			
4864	-44.98	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
4865	-44.98	kd	CGS001-10285	SMNDC1	Tudor domain containing			
4866	-44.99	kd	CGS001-9791	PTDSS1	-			
4867	-45.06	kd	CGS001-9817	KEAP1	Kelch-like proteins			
4868	-45.07	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
4869	-45.11	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
4870	-45.12	oe	ccsbBroad304_03934	LEPRE1	-			
4871	-45.15	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4872	-45.15	oe	ccsbBroad304_09756	PAQR7	-			
4873	-45.15	kd	CGS001-4436	MSH2	-			
4874	-45.22	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
4875	-45.22	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
4876	-45.29	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4877	-45.29	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
4878	-45.31	oe	ccsbBroad304_01674	TIMP4	-			
4879	-45.31	kd	CGS001-55526	DHTKD1	-			
4880	-45.32	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
4881	-45.32	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
4882	-45.33	kd	CGS001-6195	RPS6KA1	RSK subfamily			
4883	-45.38	oe	ccsbBroad304_09954	PTRF	-			
4884	-45.39	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
4885	-45.43	kd	CGS001-124641	OVCA2	-			
4886	-45.45	kd	CGS001-22818	COPZ1	-			
4887	-45.52	kd	CGS001-6871	TADA2A	-			
4888	-45.53	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
4889	-45.56	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
4890	-45.62	kd	CGS001-3281	HSBP1	-			
4891	-45.64	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
4892	-45.67	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
4893	-45.71	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
4894	-45.72	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
4895	-45.73	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
4896	-45.75	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
4897	-45.76	kd	CGS001-84328	LZIC	-			
4898	-45.77	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
4899	-45.79	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
4900	-45.8	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
4901	-45.83	kd	CGS001-1514	CTSL1	-			
4902	-45.85	kd	CGS001-5422	POLA1	DNA polymerases			
4903	-45.87	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
4904	-45.89	kd	CGS001-23139	MAST2	MAST family			
4905	-45.96	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
4906	-45.99	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
4907	-46.01	oe	ccsbBroad304_04544	RCCD1	-			
4908	-46.02	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
4909	-46.02	kd	CGS001-79862	ZNF669	Zinc fingers, C2H2-type			
4910	-46.04	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4911	-46.09	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
4912	-46.12	kd	CGS001-57720	GPR107	GPCR / Unclassified : 7TM orphan receptors			
4913	-46.12	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
4914	-46.15	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
4915	-46.15	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
4916	-46.17	kd	CGS001-89882	TPD52L3	-			
4917	-46.19	oe	ccsbBroad304_03950	ATG3	-			
4918	-46.21	cp	BRD-A79903587	tegafur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
4919	-46.24	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
4920	-46.26	cp	BRD-K94144010	cotinine	Nicotine metabolite			Nicotine metabolite
4921	-46.27	kd	CGS001-929	CD14	CD molecules			
4922	-46.29	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
4923	-46.31	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
4924	-46.38	oe	ccsbBroad304_02230	HERPUD1	-			
4925	-46.4	kd	CGS001-6721	SREBF2	Basic helix-loop-helix proteins			
4926	-46.4	kd	CGS001-1429	CRYZ	-			
4927	-46.41	oe	ccsbBroad304_06745	PNN	-			
4928	-46.45	oe	ccsbBroad304_07887	GCAT	-			
4929	-46.46	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4930	-46.49	oe	ccsbBroad304_00552	FEN1	-			
4931	-46.54	kd	CGS001-537	ATP6AP1	-			
4932	-46.66	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
4933	-46.67	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
4934	-46.68	cp	BRD-K02227374	milnacipran	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Serotonin reuptake inhibitor
4935	-46.71	kd	CGS001-10048	RANBP9	-			
4936	-46.72	kd	CGS001-8295	TRRAP	TRRAP subfamily			
4937	-46.72	kd	CGS001-83440	ADPGK	-			
4938	-46.75	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
4939	-46.75	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
4940	-46.8	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
4941	-46.8	kd	CGS001-23463	ICMT	-			
4942	-46.85	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
4943	-46.87	kd	CGS001-831	CAST	-			
4944	-46.91	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
4945	-46.96	kd	CGS001-9061	PAPSS1	-			
4946	-47.01	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
4947	-47.04	kd	CGS001-51222	ZNF219	Zinc fingers, C2H2-type			
4948	-47.05	kd	CGS001-2534	FYN	Src family			
4949	-47.06	kd	CGS001-9258	MFHAS1	-			
4950	-47.1	cp	BRD-K63265447	docetaxel	Tubulin inhibitor		TUBB, BCL2, MAP2, MAP4, MAPT, NR1I2, TUBB1	Tubulin inhibitor
4951	-47.1	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
4952	-47.12	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
4953	-47.15	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
4954	-47.17	kd	CGS001-1999	ELF3	ETS Transcription Factors			
4955	-47.19	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
4956	-47.19	kd	CGS001-2109	ETFB	-			
4957	-47.21	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
4958	-47.22	cc		Topoisomerase inhibitor	-			
4959	-47.22	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
4960	-47.22	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
4961	-47.26	kd	CGS001-3560	IL2RB	IL-2 receptor family			
4962	-47.27	kd	CGS001-29775	CARD10	-			
4963	-47.28	cp	BRD-K25310650	ormetoprim	Bacterial antifolate			Bacterial antifolate
4964	-47.33	oe	ccsbBroad304_04471	C5ORF62	-			
4965	-47.33	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
4966	-47.33	kd	CGS001-80212	CCDC92	-			
4967	-47.35	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
4968	-47.35	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
4969	-47.36	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
4970	-47.39	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
4971	-47.43	kd	CGS001-6895	TARBP2	-			
4972	-47.43	kd	CGS001-375133	PI4KAP2	-			
4973	-47.44	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
4974	-47.46	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
4975	-47.51	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
4976	-47.51	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
4977	-47.54	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
4978	-47.59	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
4979	-47.67	kd	CGS001-9738	CCP110	-			
4980	-47.69	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
4981	-47.69	kd	CGS001-4016	LOXL1	-			
4982	-47.76	kd	CGS001-7572	ZNF24	Zinc fingers, C2H2-type			
4983	-47.79	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4984	-47.88	kd	CGS001-23210	JMJD6	-			
4985	-47.94	kd	CGS001-335	APOA1	Apolipoproteins			
4986	-47.94	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
4987	-47.96	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
4988	-47.97	oe	ccsbBroad304_09354	IGSF8	CD molecules			
4989	-47.99	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
4990	-48	oe	ccsbBroad304_00614	GAMT	-			
4991	-48	kd	CGS001-9034	CCRL2	Chemokine receptors			
4992	-48.03	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
4993	-48.05	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
4994	-48.05	kd	CGS001-55038	CDCA4	-			
4995	-48.06	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
4996	-48.1	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
4997	-48.1	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
4998	-48.14	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
4999	-48.18	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
5000	-48.22	oe	ccsbBroad304_08775	SQRDL	-			
5001	-48.23	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
5002	-48.23	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
5003	-48.24	oe	ccsbBroad304_08878	METTL4	-			
5004	-48.25	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
5005	-48.26	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
5006	-48.26	kd	CGS001-55191	NADSYN1	-			
5007	-48.27	kd	CGS001-3985	LIMK2	LIMK subfamily			
5008	-48.31	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
5009	-48.35	oe	ccsbBroad304_07923	LSM5	-			
5010	-48.36	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
5011	-48.37	oe	ccsbBroad304_03056	MCTS1	-			
5012	-48.4	oe	ccsbBroad304_09578	PASD1	-			
5013	-48.47	kd	CGS001-5920	RARRES3	-			
5014	-48.48	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
5015	-48.49	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
5016	-48.49	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
5017	-48.55	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
5018	-48.59	kd	CGS001-9212	AURKB	Aurora kinase			
5019	-48.59	kd	CGS001-56916	SMARCAD1	-			
5020	-48.63	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
5021	-48.71	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
5022	-48.76	kd	CGS001-7057	THBS1	-			
5023	-48.79	oe	ccsbBroad304_00038	AGL	-			
5024	-48.79	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5025	-48.8	kd	CGS001-84547	PGBD1	-			
5026	-48.81	kd	CGS001-5906	RAP1A	-			
5027	-48.84	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
5028	-48.87	oe	ccsbBroad304_00816	IDE	Pitrilysin			
5029	-48.89	oe	ccsbBroad304_04294	ATG10	-			
5030	-48.92	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
5031	-48.98	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
5032	-48.99	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
5033	-49	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
5034	-49.02	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
5035	-49.02	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
5036	-49.06	kd	CGS001-23576	DDAH1	Dimethylarginine dimethylaminohydrolases			
5037	-49.14	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
5038	-49.19	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
5039	-49.22	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
5040	-49.23	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
5041	-49.25	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
5042	-49.27	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
5043	-49.29	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
5044	-49.29	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
5045	-49.31	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
5046	-49.32	oe	ccsbBroad304_02487	TXNIP	-			
5047	-49.32	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5048	-49.38	kd	CGS001-1856	DVL2	Dishevelled homologs			
5049	-49.4	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
5050	-49.4	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
5051	-49.42	oe	ccsbBroad304_09035	COASY	-			
5052	-49.42	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
5053	-49.43	oe	ccsbBroad304_01203	PIM1	PIM family			
5054	-49.46	oe	ccsbBroad304_01008	KITLG	-			
5055	-49.46	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
5056	-49.53	kd	CGS001-1605	DAG1	-			
5057	-49.56	kd	CGS001-10933	MORF4L1	-			
5058	-49.59	kd	CGS001-133522	PPARGC1B	RNA binding motif (RRM) containing			
5059	-49.61	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
5060	-49.62	cp	BRD-K84955386	hyperoside	Glucosidase inhibitor		ACE, AKR1B1, GAA	Glucosidase inhibitor
5061	-49.63	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
5062	-49.65	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
5063	-49.7	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
5064	-49.71	kd	CGS001-10314	LANCL1	-			
5065	-49.74	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
5066	-49.75	kd	CGS001-1465	CSRP1	-			
5067	-49.76	kd	CGS001-124583	CANT1	-			
5068	-49.81	kd	CGS001-5817	PVR	Immunoglobulin superfamily / C2-set domain containing			
5069	-49.84	kd	CGS001-301	ANXA1	Annexins			
5070	-49.89	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
5071	-49.9	kd	CGS001-7541	ZFP161	-			
5072	-49.9	kd	CGS001-8985	PLOD3	-			
5073	-49.91	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
5074	-49.96	kd	CGS001-9375	TM9SF2	-			
5075	-49.96	kd	CGS001-6617	SNAPC1	-			
5076	-49.97	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
5077	-50.02	cp	BRD-K86887724	dofetilide	Potassium channel blocker		KCNH2, KCNH1, KCNJ12, KCNK2	Potassium channel blocker
5078	-50.07	kd	CGS001-9641	IKBKE	IKK family			
5079	-50.1	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
5080	-50.14	oe	ccsbBroad304_07861	COBL	-			
5081	-50.14	kd	CGS001-47	ACLY	-			
5082	-50.16	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
5083	-50.16	kd	CGS001-23408	SIRT5	Histone deacetylases			
5084	-50.25	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5085	-50.25	kd	CGS001-1072	CFL1	-			
5086	-50.26	cc		GABA receptor antagonist	-			
5087	-50.26	kd	CGS001-24148	PRPF6	-			
5088	-50.27	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
5089	-50.31	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
5090	-50.32	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
5091	-50.37	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
5092	-50.44	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
5093	-50.48	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
5094	-50.48	kd	CGS001-23647	ARFIP2	-			
5095	-50.54	kd	CGS001-1840	DTX1	-			
5096	-50.57	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
5097	-50.58	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
5098	-50.59	oe	ccsbBroad304_03420	TOLLIP	-			
5099	-50.63	kd	CGS001-10020	GNE	-			
5100	-50.64	kd	CGS001-23492	CBX7	-			
5101	-50.66	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
5102	-50.68	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
5103	-50.69	oe	ccsbBroad304_02045	BUD31	-			
5104	-50.7	cp	BRD-K44442813	pidotimod	Interferon receptor agonist			Interferon receptor agonist, Interleukin receptor agonist
5105	-50.74	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
5106	-50.75	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
5107	-50.86	kd	CGS001-5900	RALGDS	-			
5108	-50.86	kd	CGS001-79712	GTDC1	Glycosyltransferase group 1 domain containing			
5109	-50.87	oe	ccsbBroad304_00652	GNAS	-			
5110	-50.89	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
5111	-50.91	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
5112	-50.91	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
5113	-50.95	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
5114	-50.96	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
5115	-50.96	kd	CGS001-2673	GFPT1	-			
5116	-50.99	kd	CGS001-9887	SMG7	-			
5117	-51	kd	CGS001-2147	F2	Endogenous ligands			
5118	-51	kd	CGS001-835	CASP2	Caspases			
5119	-51.02	oe	ccsbBroad304_07238	STK24	YSK subfamily			
5120	-51.04	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
5121	-51.05	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
5122	-51.12	kd	CGS001-162	AP1B1	-			
5123	-51.13	oe	ccsbBroad304_00115	ASPH	-			
5124	-51.19	kd	CGS001-5045	FURIN	Subtilisin			
5125	-51.23	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
5126	-51.24	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
5127	-51.25	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
5128	-51.27	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5129	-51.34	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
5130	-51.35	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
5131	-51.37	kd	CGS001-1611	DAP	-			
5132	-51.38	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
5133	-51.4	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
5134	-51.41	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
5135	-51.45	kd	CGS001-54505	DHX29	DEAH-boxes			
5136	-51.48	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
5137	-51.53	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
5138	-51.54	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
5139	-51.54	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
5140	-51.54	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
5141	-51.55	oe	ccsbBroad304_07018	SUPT5H	-			
5142	-51.55	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
5143	-51.62	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
5144	-51.64	kd	CGS001-699	BUB1	Bub family			
5145	-51.65	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
5146	-51.7	kd	CGS001-91304	C19ORF6	-			
5147	-51.71	kd	CGS001-9978	RBX1	RING-type (C3HC4) zinc fingers			
5148	-51.76	kd	CGS001-9897	KIAA0196	-			
5149	-51.8	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
5150	-51.81	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
5151	-51.84	kd	CGS001-54584	GNB1L	WD repeat domain containing			
5152	-51.92	oe	ccsbBroad304_08553	STAP2	-			
5153	-51.95	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
5154	-52.01	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
5155	-52.01	kd	CGS001-1111	CHEK1	CHK1 subfamily			
5156	-52.05	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
5157	-52.05	kd	CGS001-8649	LAMTOR3	-			
5158	-52.07	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
5159	-52.1	kd	CGS001-115650	TNFRSF13C	Tumour necrosis factor (TNF) receptor family			
5160	-52.14	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
5161	-52.14	kd	CGS001-4507	MTAP	-			
5162	-52.15	kd	CGS001-4221	MEN1	-			
5163	-52.18	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
5164	-52.2	kd	CGS001-5660	PSAP	Endogenous ligands			
5165	-52.21	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
5166	-52.22	kd	CGS001-31	ACACA	Carboxylases			
5167	-52.28	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
5168	-52.29	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
5169	-52.31	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
5170	-52.35	kd	CGS001-3155	HMGCL	-			
5171	-52.37	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5172	-52.38	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
5173	-52.43	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
5174	-52.45	oe	ccsbBroad304_02219	MORF4L2	-			
5175	-52.5	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
5176	-52.52	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5177	-52.53	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
5178	-52.53	kd	CGS001-9475	ROCK2	Pleckstrin homology (PH) domain containing			
5179	-52.55	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
5180	-52.63	kd	CGS001-3074	HEXB	-			
5181	-52.64	oe	ccsbBroad304_03264	UBAP1	-			
5182	-52.67	kd	CGS001-4637	MYL6	EF-hand domain containing			
5183	-52.68	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
5184	-52.68	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
5185	-52.69	kd	CGS001-50604	IL20	Interleukins and interleukin receptors			
5186	-52.7	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
5187	-52.7	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
5188	-52.74	kd	CGS001-3925	STMN1	-			
5189	-52.74	kd	CGS001-1163	CKS1B	-			
5190	-52.83	oe	ccsbBroad304_02533	NOXA1	-			
5191	-52.86	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
5192	-52.86	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
5193	-52.88	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
5194	-52.88	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
5195	-52.9	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
5196	-52.9	kd	CGS001-8193	DPF1	Zinc fingers, PHD-type			
5197	-52.92	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
5198	-52.93	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
5199	-52.94	kd	CGS001-10544	PROCR	CD molecules			
5200	-52.97	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
5201	-52.98	oe	ccsbBroad304_00392	CTLA4	CD molecules			
5202	-52.98	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
5203	-52.99	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
5204	-53	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
5205	-53.02	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
5206	-53.03	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
5207	-53.04	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
5208	-53.07	cc		Gamma secretase inhibitor	-			
5209	-53.11	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
5210	-53.12	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
5211	-53.17	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5212	-53.17	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
5213	-53.23	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
5214	-53.32	kd	CGS001-64863	METTL4	-			
5215	-53.35	kd	CGS001-9360	PPIG	-			
5216	-53.47	oe	ccsbBroad304_03772	CCNL1	-			
5217	-53.47	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
5218	-53.48	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5219	-53.49	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
5220	-53.5	kd	CGS001-9020	MAP3K14	MAPKKK:STE-unique family			
5221	-53.51	kd	CGS001-25888	ZNF473	Zinc fingers, C2H2-type			
5222	-53.57	kd	CGS001-83439	TCF7L1	-			
5223	-53.58	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
5224	-53.59	oe	ccsbBroad304_03191	NOSIP	-			
5225	-53.61	oe	ccsbBroad304_02249	KIAA0494	-			
5226	-53.63	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
5227	-53.66	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
5228	-53.66	kd	CGS001-26574	AATF	-			
5229	-53.7	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
5230	-53.74	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
5231	-53.75	kd	CGS001-7280	TUBB2A	Tubulins			
5232	-53.76	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
5233	-53.79	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
5234	-53.91	oe	ccsbBroad304_01001	MEST	-			
5235	-53.94	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
5236	-53.98	kd	CGS001-2099	ESR1	Estrogen receptors			
5237	-54	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5238	-54.01	cc		Tachykinin antagonist	-			
5239	-54.02	oe	ccsbBroad304_02094	FIBP	-			
5240	-54.06	cc		T-type calcium channel blocker	-			
5241	-54.07	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
5242	-54.08	kd	CGS001-4012	LNPEP	Aminopeptidase N			
5243	-54.09	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
5244	-54.1	kd	CGS001-79187	FSD1	Fibronectin type III domain containing			
5245	-54.16	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
5246	-54.21	kd	CGS001-2309	FOXO3	Forkhead boxes			
5247	-54.22	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
5248	-54.26	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
5249	-54.33	kd	CGS001-4351	MPI	-			
5250	-54.46	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
5251	-54.46	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
5252	-54.48	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
5253	-54.5	kd	CGS001-8935	SKAP2	Pleckstrin homology (PH) domain containing			
5254	-54.54	kd	CGS001-9276	COPB2	WD repeat domain containing			
5255	-54.56	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
5256	-54.57	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
5257	-54.59	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
5258	-54.65	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
5259	-54.68	kd	CGS001-9218	VAPA	-			
5260	-54.71	kd	CGS001-55907	CMAS	-			
5261	-54.72	oe	ccsbBroad304_00118	ATIC	-			
5262	-54.79	kd	CGS001-29888	STRN4	WD repeat domain containing			
5263	-54.79	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
5264	-54.8	oe	ccsbBroad304_02398	LANCL1	-			
5265	-54.81	oe	ccsbBroad304_03554	NAT10	-			
5266	-54.81	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
5267	-54.86	oe	ccsbBroad304_07800	EXOSC8	-			
5268	-54.86	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
5269	-54.87	kd	CGS001-51601	LIPT1	-			
5270	-54.95	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
5271	-54.96	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
5272	-54.98	kd	CGS001-28511	NKIRAS2	-			
5273	-54.99	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
5274	-55.03	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
5275	-55.04	cp	BRD-K92870997	pterostilbene	Cyclooxygenase inhibitor		FAAH, PPARA, PTGS1, PTGS2	Cyclooxygenase inhibitor, PPAR receptor agonist
5276	-55.09	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
5277	-55.09	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
5278	-55.13	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
5279	-55.17	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
5280	-55.19	cc		Bile acid	-			
5281	-55.22	oe	ccsbBroad304_07219	CDC7	CDC7 family			
5282	-55.23	oe	ccsbBroad304_09225	BUD13	-			
5283	-55.24	kd	CGS001-162699	TCEB3C	-			
5284	-55.24	kd	CGS001-221188	GPR114	Adhesion Class GPCRs			
5285	-55.26	kd	CGS001-1440	CSF3	Endogenous ligands			
5286	-55.27	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
5287	-55.29	cc		KCNJ11 modulator	-			
5288	-55.32	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
5289	-55.36	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
5290	-55.41	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
5291	-55.43	kd	CGS001-51684	SUFU	-			
5292	-55.44	kd	CGS001-79902	NUP85	-			
5293	-55.47	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
5294	-55.52	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
5295	-55.64	oe	ccsbBroad304_00810	HYAL1	-			
5296	-55.65	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
5297	-55.66	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
5298	-55.69	kd	CGS001-7314	UBB	-			
5299	-55.69	kd	CGS001-9695	EDEM1	-			
5300	-55.7	kd	CGS001-3958	LGALS3	Endogenous ligands			
5301	-55.71	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
5302	-55.73	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
5303	-55.74	oe	ccsbBroad304_08055	ATP5S	-			
5304	-55.75	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5305	-55.81	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
5306	-55.85	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
5307	-55.86	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
5308	-55.88	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
5309	-55.92	oe	ccsbBroad304_10207	ERLIN1	-			
5310	-55.92	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
5311	-55.95	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
5312	-55.98	cc		Estrogen receptor antagonist	-			
5313	-56	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
5314	-56.02	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5315	-56.04	kd	CGS001-9459	ARHGEF6	Rho guanine nucleotide exchange factors			
5316	-56.09	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
5317	-56.11	oe	ccsbBroad304_02500	RRAGA	-			
5318	-56.13	kd	CGS001-11186	RASSF1	-			
5319	-56.14	kd	CGS001-30001	ERO1L	-			
5320	-56.14	kd	CGS001-1495	CTNNA1	Catenins			
5321	-56.15	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
5322	-56.15	kd	CGS001-10427	SEC24B	-			
5323	-56.16	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
5324	-56.16	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
5325	-56.19	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
5326	-56.2	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
5327	-56.2	oe	ccsbBroad304_01372	RALB	-			
5328	-56.21	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
5329	-56.28	cc		Dopamine receptor antagonist	-			
5330	-56.31	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
5331	-56.35	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
5332	-56.36	kd	CGS001-2645	GCK	Hexokinases			
5333	-56.37	kd	CGS001-85027	C5ORF62	-			
5334	-56.43	oe	ccsbBroad304_01394	RFX4	-			
5335	-56.44	oe	ccsbBroad304_01184	PGK1	-			
5336	-56.44	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
5337	-56.44	kd	CGS001-5167	ENPP1	-			
5338	-56.44	kd	CGS001-60	ACTB	-			
5339	-56.48	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
5340	-56.51	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
5341	-56.54	kd	CGS001-1719	DHFR	Oxidoreductases			
5342	-56.6	oe	ccsbBroad304_08346	COQ3	-			
5343	-56.63	oe	ccsbBroad304_05749	A2M	-			
5344	-56.64	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
5345	-56.65	oe	ccsbBroad304_07814	SACM1L	-			
5346	-56.67	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
5347	-56.68	kd	CGS001-8853	ASAP2	Ankyrin repeat domain containing			
5348	-56.75	oe	ccsbBroad304_10437	STMN1	-			
5349	-56.76	kd	CGS001-3845	KRAS	RAS subfamily			
5350	-56.77	kd	CGS001-6927	HNF1A	Homeoboxes / HNF class			
5351	-56.86	kd	CGS001-7296	TXNRD1	-			
5352	-56.89	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
5353	-56.9	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
5354	-56.93	kd	CGS001-481	ATP1B1	ATPases / P-type			
5355	-56.94	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
5356	-56.99	kd	CGS001-2167	FABP4	Fatty acid binding protein family			
5357	-57.03	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
5358	-57.03	kd	CGS001-5228	PGF	-			
5359	-57.14	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
5360	-57.15	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
5361	-57.17	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
5362	-57.24	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
5363	-57.24	kd	CGS001-51727	CMPK1	-			
5364	-57.25	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
5365	-57.27	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
5366	-57.27	kd	CGS001-3029	HAGH	-			
5367	-57.31	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
5368	-57.33	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
5369	-57.36	oe	ccsbBroad304_03433	DDIT4	-			
5370	-57.38	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
5371	-57.41	oe	ccsbBroad304_06349	HAGH	-			
5372	-57.43	kd	CGS001-6929	TCF3	Basic helix-loop-helix proteins			
5373	-57.45	kd	CGS001-6773	STAT2	SH2 domain containing			
5374	-57.47	kd	CGS001-2735	GLI1	Zinc fingers, C2H2-type			
5375	-57.49	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
5376	-57.51	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
5377	-57.58	oe	ccsbBroad304_00617	GBA	-			
5378	-57.62	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
5379	-57.75	oe	ccsbBroad304_02017	PEX11A	-			
5380	-57.78	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
5381	-57.79	oe	ccsbBroad304_12226	NAGK	-			
5382	-57.8	oe	ccsbBroad304_00651	GNAI3	-			
5383	-57.8	oe	ccsbBroad304_07888	CBX6	-			
5384	-57.84	cp	BRD-K86003836	flubendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
5385	-57.85	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
5386	-57.87	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
5387	-57.93	kd	CGS001-558	AXL	Fibronectin type III domain containing			
5388	-57.94	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
5389	-57.96	oe	ccsbBroad304_00819	IDH3B	-			
5390	-57.98	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
5391	-58.08	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
5392	-58.1	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
5393	-58.1	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
5394	-58.1	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
5395	-58.13	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
5396	-58.16	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
5397	-58.18	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
5398	-58.23	oe	ccsbBroad304_02306	PQBP1	-			
5399	-58.23	kd	CGS001-79135	APOO	Apolipoproteins			
5400	-58.27	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
5401	-58.3	oe	ccsbBroad304_04616	ORMDL3	-			
5402	-58.37	kd	CGS001-8802	SUCLG1	-			
5403	-58.38	cp	BRD-K27184429	levocetirizine	Histamine receptor antagonist		HRH1, CXCL8	Histamine receptor antagonist
5404	-58.42	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5405	-58.43	oe	ccsbBroad304_06253	GALT	-			
5406	-58.43	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
5407	-58.51	kd	CGS001-83933	HDAC10	Histone deacetylases			
5408	-58.53	cp	BRD-K84566043	fenpiverinium	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
5409	-58.56	kd	CGS001-283455	KSR2	RAF family			
5410	-58.57	oe	ccsbBroad304_01215	PLAUR	CD molecules			
5411	-58.58	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
5412	-58.59	kd	CGS001-433	ASGR2	C-type lectin domain containing			
5413	-58.6	kd	CGS001-29883	CNOT7	-			
5414	-58.61	kd	CGS001-3608	ILF2	-			
5415	-58.66	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
5416	-58.69	kd	CGS001-284	ANGPT1	Fibrinogen C domain containing			
5417	-58.72	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
5418	-58.75	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
5419	-58.75	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
5420	-58.77	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
5421	-58.81	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
5422	-58.82	oe	ccsbBroad304_03573	BRF2	-			
5423	-58.87	kd	CGS001-56647	BCCIP	-			
5424	-58.91	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
5425	-58.92	kd	CGS001-8449	DHX16	DEAH-boxes			
5426	-58.94	cp	BRD-K70883034	nimetazepam	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA receptor agonist
5427	-59.03	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
5428	-59.07	kd	CGS001-8804	CREG1	-			
5429	-59.13	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
5430	-59.13	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
5431	-59.17	oe	ccsbBroad304_02509	GMEB1	-			
5432	-59.22	kd	CGS001-10111	RAD50	-			
5433	-59.26	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
5434	-59.31	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
5435	-59.33	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
5436	-59.34	kd	CGS001-900	CCNG1	-			
5437	-59.4	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
5438	-59.4	kd	CGS001-8829	NRP1	CD molecules			
5439	-59.41	kd	CGS001-167826	OLIG3	Basic helix-loop-helix proteins			
5440	-59.43	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
5441	-59.43	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
5442	-59.44	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
5443	-59.46	oe	ccsbBroad304_00491	EIF4EBP2	-			
5444	-59.46	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
5445	-59.48	kd	CGS001-6598	SMARCB1	-			
5446	-59.48	kd	CGS001-51176	LEF1	-			
5447	-59.53	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
5448	-59.54	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
5449	-59.54	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
5450	-59.55	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
5451	-59.59	kd	CGS001-3339	HSPG2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5452	-59.61	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
5453	-59.62	kd	CGS001-143187	VTI1A	-			
5454	-59.63	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
5455	-59.7	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
5456	-59.72	kd	CGS001-5170	PDPK1	PDK1 family			
5457	-59.73	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
5458	-59.75	cc		HIF activator	-			
5459	-59.76	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
5460	-59.79	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5461	-59.83	kd	CGS001-56654	NPDC1	-			
5462	-59.88	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
5463	-59.88	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
5464	-59.89	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
5465	-59.9	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
5466	-59.92	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
5467	-59.95	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
5468	-59.96	kd	CGS001-399694	SHC4	SH2 domain containing			
5469	-59.99	kd	CGS001-23043	TNIK	MSN subfamily			
5470	-60.01	cc		Progesterone receptor antagonist	-			
5471	-60.03	kd	CGS001-563	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
5472	-60.07	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
5473	-60.07	kd	CGS001-50813	COPS7A	-			
5474	-60.1	kd	CGS001-23650	TRIM29	-			
5475	-60.16	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
5476	-60.2	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
5477	-60.22	oe	ccsbBroad304_01962	STK16	NAK family			
5478	-60.22	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
5479	-60.24	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
5480	-60.3	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
5481	-60.32	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
5482	-60.34	oe	ccsbBroad304_00120	ATOX1	-			
5483	-60.41	kd	CGS001-26959	HBP1	-			
5484	-60.47	kd	CGS001-638	BIK	-			
5485	-60.47	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
5486	-60.5	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
5487	-60.54	kd	CGS001-54658	UGT1A1	UDP glucuronosyltransferases			
5488	-60.58	kd	CGS001-256281	NUDT14	Nudix motif containing			
5489	-60.59	oe	ccsbBroad304_02864	PRDX5	-			
5490	-60.6	oe	ccsbBroad304_00661	GNGT2	-			
5491	-60.6	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
5492	-60.61	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
5493	-60.64	cc		PRD class homeoboxes and psudogenes LOF	-			
5494	-60.65	oe	ccsbBroad304_01183	PGD	-			
5495	-60.65	kd	CGS001-10939	AFG3L2	ATPases / AAA-type			
5496	-60.66	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
5497	-60.68	oe	ccsbBroad304_00986	MCM2	-			
5498	-60.7	kd	CGS001-113451	ADC	-			
5499	-60.72	kd	CGS001-7862	BRPF1	Non-enzymatic BRD containing proteins			
5500	-60.76	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
5501	-60.78	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
5502	-60.8	kd	CGS001-7360	UGP2	-			
5503	-60.82	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
5504	-60.85	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
5505	-60.86	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
5506	-60.96	kd	CGS001-5327	PLAT	Chymotrypsin			
5507	-61.05	kd	CGS001-23534	TNPO3	Importins			
5508	-61.09	kd	CGS001-23012	STK38L	NDR family			
5509	-61.12	kd	CGS001-3593	IL12B	Interleukins and interleukin receptors			
5510	-61.16	kd	CGS001-56993	TOMM22	-			
5511	-61.18	kd	CGS001-4171	MCM2	-			
5512	-61.24	oe	ccsbBroad304_08511	RFK	-			
5513	-61.33	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
5514	-61.33	kd	CGS001-1020	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
5515	-61.34	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
5516	-61.34	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
5517	-61.35	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
5518	-61.35	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
5519	-61.37	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
5520	-61.41	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
5521	-61.42	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
5522	-61.49	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
5523	-61.51	kd	CGS001-140612	ZFP28	Zinc fingers, C2H2-type			
5524	-61.55	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
5525	-61.57	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5526	-61.61	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
5527	-61.62	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
5528	-61.62	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
5529	-61.71	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
5530	-61.76	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
5531	-61.78	oe	ccsbBroad304_01948	GAS7	-			
5532	-61.78	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
5533	-61.82	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
5534	-61.85	kd	CGS001-836	CASP3	Caspases			
5535	-61.9	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
5536	-61.93	kd	CGS001-3458	IFNG	Interferons			
5537	-61.97	kd	CGS001-2539	G6PD	-			
5538	-61.98	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
5539	-62	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
5540	-62.08	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
5541	-62.08	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
5542	-62.12	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
5543	-62.12	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
5544	-62.14	kd	CGS001-7054	TH	Amino acid hydroxylases			
5545	-62.14	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
5546	-62.14	kd	CGS001-10128	LRPPRC	-			
5547	-62.16	kd	CGS001-2879	GPX4	-			
5548	-62.18	oe	ccsbBroad304_03859	ENOPH1	-			
5549	-62.19	oe	ccsbBroad304_02018	SUCLA2	-			
5550	-62.19	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
5551	-62.22	kd	CGS001-2805	GOT1	-			
5552	-62.24	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
5553	-62.24	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
5554	-62.28	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5555	-62.31	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
5556	-62.32	oe	ccsbBroad304_01101	NME1	-			
5557	-62.36	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
5558	-62.39	kd	CGS001-9759	HDAC4	Histone deacetylases			
5559	-62.53	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
5560	-62.64	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
5561	-62.64	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
5562	-62.64	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
5563	-62.68	kd	CGS001-160	AP2A1	-			
5564	-62.7	oe	ccsbBroad304_02458	STK25	YSK subfamily			
5565	-62.7	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
5566	-62.72	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
5567	-62.8	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
5568	-62.8	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
5569	-62.8	kd	CGS001-23028	KDM1A	Histone demethylase			
5570	-62.82	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
5571	-62.82	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
5572	-62.82	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
5573	-62.83	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
5574	-62.83	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
5575	-62.85	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
5576	-62.85	kd	CGS001-1201	CLN3	-			
5577	-62.88	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
5578	-62.91	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
5579	-62.92	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
5580	-62.97	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
5581	-62.98	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
5582	-63.03	kd	CGS001-3419	IDH3A	-			
5583	-63.08	kd	CGS001-190	NR0B1	DAX-like receptors			
5584	-63.09	kd	CGS001-11320	MGAT4A	-			
5585	-63.09	kd	CGS001-9415	FADS2	Fatty acid desaturases			
5586	-63.13	oe	ccsbBroad304_00113	ASNS	-			
5587	-63.14	kd	CGS001-4835	NQO2	-			
5588	-63.17	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
5589	-63.18	oe	ccsbBroad304_01038	MSRA	-			
5590	-63.22	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
5591	-63.23	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
5592	-63.28	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
5593	-63.29	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5594	-63.3	oe	ccsbBroad304_03506	AURKAIP1	-			
5595	-63.31	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
5596	-63.35	kd	CGS001-84971	ATG4D	-			
5597	-63.36	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
5598	-63.39	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
5599	-63.41	kd	CGS001-6793	STK10	SLK subfamily			
5600	-63.43	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
5601	-63.51	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
5602	-63.56	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
5603	-63.56	kd	CGS001-6117	RPA1	-			
5604	-63.61	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
5605	-63.61	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
5606	-63.64	oe	ccsbBroad304_02801	CASP14	Caspases			
5607	-63.66	cp	BRD-K93618743	ipriflavone	Bone resorption inhibitor			Bone resorption inhibitor
5608	-63.68	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
5609	-63.69	kd	CGS001-5378	PMS1	-			
5610	-63.7	kd	CGS001-7020	TFAP2A	-			
5611	-63.72	kd	CGS001-5450	POU2AF1	-			
5612	-63.73	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
5613	-63.75	cc		Sodium channel blocker	-			
5614	-63.76	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
5615	-63.81	kd	CGS001-353	APRT	-			
5616	-63.84	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
5617	-63.85	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
5618	-63.87	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
5619	-63.88	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
5620	-63.92	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
5621	-63.95	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
5622	-63.95	cp	BRD-K97752965	nicorandil	Nitric oxide donor		ABCC9, KCNJ11, KCNJ8	Nitric oxide donor, Potassium channel activator
5623	-63.95	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
5624	-64.01	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
5625	-64.02	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
5626	-64.03	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
5627	-64.05	kd	CGS001-5053	PAH	Amino acid hydroxylases			
5628	-64.06	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
5629	-64.1	kd	CGS001-1892	ECHS1	-			
5630	-64.15	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
5631	-64.15	kd	CGS001-126823	KLHDC9	-			
5632	-64.18	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
5633	-64.22	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
5634	-64.23	kd	CGS001-1984	EIF5A	-			
5635	-64.26	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5636	-64.28	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
5637	-64.3	kd	CGS001-1844	DUSP2	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
5638	-64.33	kd	CGS001-6894	TARBP1	-			
5639	-64.35	kd	CGS001-2119	ETV5	ETS Transcription Factors			
5640	-64.37	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
5641	-64.39	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
5642	-64.39	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5643	-64.44	kd	CGS001-218	ALDH3A1	Aldehyde dehydrogenases			
5644	-64.45	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
5645	-64.5	kd	CGS001-10671	DCTN6	-			
5646	-64.53	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
5647	-64.56	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
5648	-64.58	kd	CGS001-29940	DSE	-			
5649	-64.6	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
5650	-64.64	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
5651	-64.64	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
5652	-64.65	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
5653	-64.66	kd	CGS001-1718	DHCR24	-			
5654	-64.7	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
5655	-64.76	kd	CGS001-7077	TIMP2	-			
5656	-64.77	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
5657	-64.84	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
5658	-64.9	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
5659	-64.91	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5660	-64.97	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
5661	-64.98	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
5662	-65.04	kd	CGS001-9181	ARHGEF2	Rho guanine nucleotide exchange factors			
5663	-65.05	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
5664	-65.08	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
5665	-65.1	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
5666	-65.12	cc		Akt Signaling GOF	-			
5667	-65.12	kd	CGS001-509	ATP5C1	ATPases / F-type			
5668	-65.13	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
5669	-65.14	cp	BRD-A37052580	physostigmine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Cholinesterase inhibitor
5670	-65.16	oe	ccsbBroad304_04190	CCDC92	-			
5671	-65.19	cp	BRD-K05350981	oligomycin-c	ATPase inhibitor		ATP5A1	ATPase inhibitor, ATP synthase inhibitor
5672	-65.19	kd	CGS001-3017	HIST1H2BD	Histones / Replication-dependent			
5673	-65.19	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5674	-65.2	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
5675	-65.21	kd	CGS001-1647	GADD45A	-			
5676	-65.23	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
5677	-65.29	cc		JAK inhibitor	-			
5678	-65.3	kd	CGS001-57822	GRHL3	-			
5679	-65.3	kd	CGS001-338	APOB	Apolipoproteins			
5680	-65.31	kd	CGS001-221393	GPR115	Adhesion Class GPCRs			
5681	-65.32	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
5682	-65.43	oe	ccsbBroad304_06642	NIT1	-			
5683	-65.5	oe	ccsbBroad304_07490	SCRN1	-			
5684	-65.5	cp	BRD-K98493452	honokiol	AKT inhibitor		ALOX5, PTGS1, PTGS2	AKT inhibitor
5685	-65.53	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
5686	-65.54	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
5687	-65.56	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
5688	-65.58	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
5689	-65.6	kd	CGS001-57057	TBX20	T-boxes			
5690	-65.69	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
5691	-65.7	kd	CGS001-5584	PRKCI	Iota subfamily			
5692	-65.72	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
5693	-65.75	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
5694	-65.82	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
5695	-65.84	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
5696	-65.85	oe	ccsbBroad304_07029	TADA2A	-			
5697	-65.85	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
5698	-65.86	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5699	-65.94	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
5700	-65.96	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
5701	-65.96	kd	CGS001-5159	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5702	-65.96	kd	CGS001-23549	DNPEP	Aminopeptidase I			
5703	-66	oe	ccsbBroad304_00489	EHHADH	-			
5704	-66.04	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
5705	-66.06	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
5706	-66.09	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
5707	-66.09	kd	CGS001-23239	PHLPP1	Pleckstrin homology (PH) domain containing			
5708	-66.13	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
5709	-66.2	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
5710	-66.21	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
5711	-66.22	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
5712	-66.22	kd	CGS001-2263	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
5713	-66.23	oe	ccsbBroad304_02990	LYPD3	-			
5714	-66.23	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
5715	-66.26	kd	CGS001-55536	CDCA7L	-			
5716	-66.28	cc		Beta-adrenergic receptor agonist	-			
5717	-66.29	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
5718	-66.3	oe	ccsbBroad304_07363	AIFM1	-			
5719	-66.36	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
5720	-66.41	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
5721	-66.42	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
5722	-66.45	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
5723	-66.45	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
5724	-66.48	kd	CGS001-1677	DFFB	-			
5725	-66.53	kd	CGS001-84108	PCGF6	Polycomb group ring fingers			
5726	-66.54	kd	CGS001-23451	SF3B1	-			
5727	-66.55	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
5728	-66.56	oe	ccsbBroad304_04619	GNG8	-			
5729	-66.56	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
5730	-66.57	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5731	-66.58	kd	CGS001-10421	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5732	-66.61	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
5733	-66.64	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
5734	-66.64	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
5735	-66.65	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
5736	-66.69	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
5737	-66.69	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5738	-66.78	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
5739	-66.79	kd	CGS001-8833	GMPS	-			
5740	-66.98	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
5741	-67.02	oe	ccsbBroad304_00210	CALR	-			
5742	-67.03	kd	CGS001-5033	P4HA1	-			
5743	-67.11	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
5744	-67.24	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
5745	-67.24	kd	CGS001-5708	PSMD2	Proteasome subunits			
5746	-67.29	kd	CGS001-54623	PAF1	-			
5747	-67.31	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
5748	-67.34	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
5749	-67.35	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
5750	-67.38	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5751	-67.4	kd	CGS001-25819	CCRN4L	-			
5752	-67.41	kd	CGS001-5105	PCK1	-			
5753	-67.41	oe	ccsbBroad304_01841	BAG6	-			
5754	-67.45	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
5755	-67.46	kd	CGS001-3956	LGALS1	Endogenous ligands			
5756	-67.48	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
5757	-67.5	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
5758	-67.52	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
5759	-67.53	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
5760	-67.56	cc		PI3K Signaling LOF	-			
5761	-67.63	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
5762	-67.65	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
5763	-67.67	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
5764	-67.67	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
5765	-67.69	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
5766	-67.76	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
5767	-67.81	oe	ccsbBroad304_01379	RBBP6	-			
5768	-67.81	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
5769	-67.82	cp	BRD-K82147103	lofepramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
5770	-67.91	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
5771	-67.98	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
5772	-68.07	kd	CGS001-27297	CRCP	-			
5773	-68.11	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
5774	-68.13	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
5775	-68.15	cp	BRD-K04710043	hexamethylenebisacetamide	AKT inhibitor			AKT inhibitor, Differentiation inducer, NFkB pathway inhibitor
5776	-68.16	kd	CGS001-55229	PANK4	-			
5777	-68.17	oe	ccsbBroad304_00170	BNIP1	-			
5778	-68.21	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
5779	-68.22	kd	CGS001-818	CAMK2G	CAMK2 family			
5780	-68.29	cc		Non Homologous End Joining LOF	-			
5781	-68.3	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
5782	-68.32	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
5783	-68.36	oe	ccsbBroad304_01532	SIAH1	-			
5784	-68.36	kd	CGS001-890	CCNA2	-			
5785	-68.38	kd	CGS001-4077	NBR1	-			
5786	-68.42	kd	CGS001-7103	TSPAN8	Tetraspanins			
5787	-68.46	oe	ccsbBroad304_04626	EGLN3	-			
5788	-68.51	oe	ccsbBroad304_14242	MCCC2	-			
5789	-68.54	oe	ccsbBroad304_10240	CROT	-			
5790	-68.54	cp	BRD-A43082555	loxoprofen	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
5791	-68.56	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
5792	-68.73	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
5793	-68.74	oe	ccsbBroad304_05757	ACADS	-			
5794	-68.88	kd	CGS001-6714	SRC	Src family			
5795	-68.91	kd	CGS001-9568	GABBR2	GABA receptors			
5796	-68.93	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5797	-68.94	cp	BRD-K66896231	BRD-K66896231	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5798	-69.04	oe	ccsbBroad304_06188	F10	Chymotrypsin			
5799	-69.04	kd	CGS001-5901	RAN	-			
5800	-69.04	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
5801	-69.09	kd	CGS001-4122	MAN2A2	-			
5802	-69.1	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
5803	-69.11	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
5804	-69.13	oe	ccsbBroad304_00222	CASP6	Caspases			
5805	-69.13	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
5806	-69.21	kd	CGS001-54925	ZNF434	-			
5807	-69.23	oe	ccsbBroad304_06048	CRYZ	-			
5808	-69.27	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
5809	-69.32	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
5810	-69.36	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
5811	-69.36	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
5812	-69.39	kd	CGS001-9180	OSMR	IL-6 receptor family			
5813	-69.4	kd	CGS001-57616	TSHZ3	Teashirt zinc fingers			
5814	-69.41	kd	CGS001-4938	OAS1	-			
5815	-69.48	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
5816	-69.5	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
5817	-69.5	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
5818	-69.53	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
5819	-69.54	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
5820	-69.59	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
5821	-69.64	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
5822	-69.65	oe	ccsbBroad304_02175	MAGED1	-			
5823	-69.67	oe	ccsbBroad304_00991	MDH1	-			
5824	-69.72	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
5825	-69.72	oe	ccsbBroad304_02345	TXNDC9	-			
5826	-69.76	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
5827	-69.76	kd	CGS001-5933	RBL1	-			
5828	-69.78	kd	CGS001-57721	METTL14	-			
5829	-69.79	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
5830	-69.84	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
5831	-69.93	kd	CGS001-6464	SHC1	SH2 domain containing			
5832	-69.95	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
5833	-69.97	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
5834	-70	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
5835	-70.04	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
5836	-70.06	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
5837	-70.1	kd	CGS001-4926	NUMA1	-			
5838	-70.24	kd	CGS001-7771	ZFP112	-			
5839	-70.25	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
5840	-70.25	oe	ccsbBroad304_06852	RBP4	Lipocalins			
5841	-70.29	oe	ccsbBroad304_01985	EIF3H	-			
5842	-70.29	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
5843	-70.32	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
5844	-70.36	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
5845	-70.37	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
5846	-70.45	cc		PDGFR/KIT inhibitor	-			
5847	-70.46	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
5848	-70.47	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
5849	-70.47	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
5850	-70.47	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
5851	-70.48	kd	CGS001-5511	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5852	-70.49	kd	CGS001-486	FXYD2	Ion transport regulator			
5853	-70.5	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
5854	-70.51	oe	ccsbBroad304_00100	RHOA	-			
5855	-70.54	kd	CGS001-7024	TFCP2	-			
5856	-70.57	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
5857	-70.58	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
5858	-70.58	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
5859	-70.59	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
5860	-70.61	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
5861	-70.61	kd	CGS001-7029	TFDP2	-			
5862	-70.62	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
5863	-70.63	kd	CGS001-23161	SNX13	Sorting nexins			
5864	-70.64	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
5865	-70.65	oe	ccsbBroad304_02756	RRP8	-			
5866	-70.69	kd	CGS001-4047	LSS	Lanosterol biosynthesis pathway			
5867	-70.72	oe	ccsbBroad304_06098	DHCR24	-			
5868	-70.75	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
5869	-70.79	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
5870	-70.8	kd	CGS001-7128	TNFAIP3	OTU domain containing			
5871	-70.8	oe	ccsbBroad304_00933	LDHB	-			
5872	-70.85	kd	CGS001-2937	GSS	-			
5873	-70.89	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
5874	-70.93	kd	CGS001-488	ATP2A2	Calcium-ATPases			
5875	-70.97	kd	CGS001-221391	OPN5	GPCR / Class A : Opsin receptors			
5876	-70.98	kd	CGS001-6197	RPS6KA3	RSK subfamily			
5877	-70.99	kd	CGS001-3098	HK1	-			
5878	-71.07	oe	ccsbBroad304_03652	EXOC2	-			
5879	-71.11	kd	CGS001-8576	STK16	NAK family			
5880	-71.14	kd	CGS001-7248	TSC1	-			
5881	-71.19	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
5882	-71.24	cc		Bromodomain Inhibitor	-			
5883	-71.3	kd	CGS001-949	SCARB1	-			
5884	-71.31	kd	CGS001-54788	DNAJB12	Heat shock proteins / DNAJ (HSP40)			
5885	-71.35	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
5886	-71.38	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5887	-71.39	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
5888	-71.4	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
5889	-71.42	kd	CGS001-4089	SMAD4	SMADs			
5890	-71.42	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
5891	-71.47	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
5892	-71.48	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
5893	-71.48	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
5894	-71.5	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
5895	-71.5	kd	CGS001-8872	CDC123	-			
5896	-71.51	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
5897	-71.53	kd	CGS001-3163	HMOX2	Haem oxygenase			
5898	-71.54	kd	CGS001-7032	TFF2	-			
5899	-71.54	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
5900	-71.59	oe	ccsbBroad304_02195	SPAG7	-			
5901	-71.61	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
5902	-71.62	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
5903	-71.69	cc		Interleukin receptors LOF	-			
5904	-71.69	kd	CGS001-200879	LIPH	-			
5905	-71.71	kd	CGS001-8780	RIOK3	RIO3 subfamily			
5906	-71.78	kd	CGS001-222894	FERD3L	Basic helix-loop-helix proteins			
5907	-71.82	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
5908	-71.84	cc		HDAC inhibitor	-			
5909	-71.86	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
5910	-71.95	kd	CGS001-9637	FEZ2	-			
5911	-71.96	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
5912	-72.01	kd	CGS001-5160	PDHA1	-			
5913	-72.04	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
5914	-72.06	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
5915	-72.08	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
5916	-72.13	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
5917	-72.13	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
5918	-72.14	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
5919	-72.16	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
5920	-72.2	kd	CGS001-5564	PRKAB1	AMPK subfamily			
5921	-72.22	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
5922	-72.22	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
5923	-72.23	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
5924	-72.24	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
5925	-72.25	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
5926	-72.27	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
5927	-72.31	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
5928	-72.32	oe	ccsbBroad304_01165	PDK1	-			
5929	-72.33	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
5930	-72.35	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
5931	-72.39	kd	CGS001-3171	FOXA3	Forkhead boxes			
5932	-72.4	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
5933	-72.42	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
5934	-72.42	kd	CGS001-57018	CCNL1	-			
5935	-72.43	kd	CGS001-4717	NDUFC1	Mitochondrial respiratory chain complex / Complex I			
5936	-72.58	kd	CGS001-5294	PIK3CG	Phosphatidylinositol kinases			
5937	-72.65	oe	ccsbBroad304_01234	POLB	DNA polymerases			
5938	-72.66	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
5939	-72.67	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
5940	-72.68	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
5941	-72.68	kd	CGS001-2959	GTF2B	General transcription factors			
5942	-72.7	oe	ccsbBroad304_06670	OGG1	-			
5943	-72.71	kd	CGS001-678	ZFP36L2	RING-type (C3HC4) zinc fingers			
5944	-72.73	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
5945	-72.75	oe	ccsbBroad304_06004	CKB	-			
5946	-72.79	kd	CGS001-327	APEH	Prolyl oligopeptidase			
5947	-72.81	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
5948	-72.83	oe	ccsbBroad304_06651	NOV	-			
5949	-72.83	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5950	-72.84	oe	ccsbBroad304_00817	IDH2	-			
5951	-72.88	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
5952	-72.9	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
5953	-72.94	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
5954	-72.95	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
5955	-73.04	kd	CGS001-2849	GPR26	GPCR / Class A : Orphans			
5956	-73.1	oe	ccsbBroad304_06234	G6PC	-			
5957	-73.11	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
5958	-73.13	kd	CGS001-64710	NUCKS1	-			
5959	-73.16	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
5960	-73.19	cc		NADH ubiquinone oxidoreductase supernumerary subunits LOF	-			
5961	-73.23	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
5962	-73.29	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
5963	-73.32	oe	ccsbBroad304_01174	PEX13	-			
5964	-73.33	kd	CGS001-2056	EPO	Endogenous ligands			
5965	-73.35	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
5966	-73.39	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
5967	-73.39	cp	BRD-K46742498	alosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5968	-73.4	kd	CGS001-3428	IFI16	-			
5969	-73.43	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
5970	-73.49	oe	ccsbBroad304_01577	SOD1	-			
5971	-73.56	kd	CGS001-991	CDC20	WD repeat domain containing			
5972	-73.56	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
5973	-73.57	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
5974	-73.59	oe	ccsbBroad304_02626	PKIG	-			
5975	-73.59	kd	CGS001-5162	PDHB	-			
5976	-73.63	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5977	-73.65	kd	CGS001-3692	EIF6	-			
5978	-73.74	kd	CGS001-3248	HPGD	Prostaglandin synthases			
5979	-73.75	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
5980	-73.84	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
5981	-73.85	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
5982	-73.86	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
5983	-73.88	kd	CGS001-2593	GAMT	-			
5984	-73.89	kd	CGS001-8575	PRKRA	-			
5985	-73.94	kd	CGS001-10887	PROKR1	GPCR / Class A : Prokineticin receptors			
5986	-73.97	kd	CGS001-124626	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5987	-74.01	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
5988	-74.01	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5989	-74.06	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
5990	-74.07	kd	CGS001-5163	PDK1	-			
5991	-74.11	kd	CGS001-3030	HADHA	-			
5992	-74.14	oe	ccsbBroad304_14143	NUSAP1	-			
5993	-74.27	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
5994	-74.28	kd	CGS001-85442	KNDC1	-			
5995	-74.31	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5996	-74.34	kd	CGS001-79006	METRN	-			
5997	-74.35	kd	CGS001-6643	SNX2	Sorting nexins			
5998	-74.35	kd	CGS001-6282	S100A11	EF-hand domain containing			
5999	-74.38	kd	CGS001-4094	MAF	-			
6000	-74.38	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
6001	-74.39	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
6002	-74.44	kd	CGS001-4849	CNOT3	-			
6003	-74.57	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
6004	-74.57	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
6005	-74.6	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
6006	-74.71	oe	ccsbBroad304_06783	LGMN	Legumain			
6007	-74.74	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
6008	-74.74	kd	CGS001-55631	LRRC40	-			
6009	-74.75	kd	CGS001-9467	SH3BP5	-			
6010	-74.76	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
6011	-74.76	oe	ccsbBroad304_05821	ANXA1	Annexins			
6012	-74.85	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
6013	-74.85	kd	CGS001-1975	EIF4B	RNA binding motif (RRM) containing			
6014	-74.92	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
6015	-74.94	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
6016	-74.96	kd	CGS001-10456	HAX1	-			
6017	-74.99	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
6018	-75.05	cc		ATP synthase inhibitor	-			
6019	-75.05	kd	CGS001-6223	RPS19	S ribosomal proteins			
6020	-75.1	kd	CGS001-79618	HMBOX1	Homeoboxes / HNF class			
6021	-75.17	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
6022	-75.17	kd	CGS001-6198	RPS6KB1	p70 subfamily			
6023	-75.17	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
6024	-75.2	kd	CGS001-5664	PSEN2	Presenilin			
6025	-75.29	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
6026	-75.3	oe	ccsbBroad304_02173	ATG5	-			
6027	-75.31	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
6028	-75.33	kd	CGS001-2634	GBP2	-			
6029	-75.35	kd	CGS001-4121	MAN1A1	-			
6030	-75.35	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
6031	-75.4	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
6032	-75.44	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
6033	-75.46	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
6034	-75.55	kd	CGS001-2936	GSR	Oxidoreductases			
6035	-75.59	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
6036	-75.59	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
6037	-75.6	cp	BRD-K73196317	urapidil	Adrenergic receptor antagonist		HTR1A	Adrenergic receptor antagonist
6038	-75.6	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
6039	-75.6	kd	CGS001-2588	GALNS	Arylsulfatase family			
6040	-75.78	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
6041	-75.78	kd	CGS001-6050	RNH1	-			
6042	-75.79	kd	CGS001-284119	PTRF	-			
6043	-75.8	cc		Supressors of cytokine signaling GOF	-			
6044	-75.8	kd	CGS001-55011	PIH1D1	-			
6045	-75.92	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
6046	-76.02	kd	CGS001-26128	KIAA1279	-			
6047	-76.02	kd	CGS001-3670	ISL1	Homeoboxes / LIM class			
6048	-76.22	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
6049	-76.24	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
6050	-76.29	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6051	-76.34	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
6052	-76.35	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
6053	-76.37	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
6054	-76.38	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
6055	-76.39	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
6056	-76.47	oe	ccsbBroad304_01347	RAD1	-			
6057	-76.48	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
6058	-76.49	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
6059	-76.55	cp	BRD-K32398298	alprazolam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, CYP3A5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
6060	-76.63	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
6061	-76.65	cc		SMAD family LOF	-			
6062	-76.71	kd	CGS001-3912	LAMB1	Laminins			
6063	-76.71	kd	CGS001-7917	BAG6	-			
6064	-76.76	kd	CGS001-114112	TXNRD3	-			
6065	-76.8	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
6066	-76.81	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
6067	-76.83	kd	CGS001-4718	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
6068	-76.83	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
6069	-76.91	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
6070	-76.93	oe	ccsbBroad304_07557	NAMPT	-			
6071	-76.98	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
6072	-77	oe	ccsbBroad304_06144	EFNB3	Ephrins			
6073	-77	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
6074	-77.04	cp	BRD-K85090592	pilocarpine	Acetylcholine receptor agonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor agonist
6075	-77.08	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
6076	-77.11	kd	CGS001-10078	TSSC4	-			
6077	-77.12	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
6078	-77.15	cc		Lipocalins GOF	-			
6079	-77.2	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
6080	-77.23	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
6081	-77.25	kd	CGS001-54438	GFOD1	-			
6082	-77.26	kd	CGS001-8864	PER2	-			
6083	-77.27	kd	CGS001-5927	KDM5A	Histone demethylases			
6084	-77.31	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
6085	-77.34	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
6086	-77.39	oe	ccsbBroad304_07632	PROCR	CD molecules			
6087	-77.4	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6088	-77.46	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6089	-77.52	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
6090	-77.54	oe	ccsbBroad304_02057	P4HA2	-			
6091	-77.55	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
6092	-77.55	kd	CGS001-7078	TIMP3	-			
6093	-77.56	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
6094	-77.59	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
6095	-77.61	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
6096	-77.62	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
6097	-77.63	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
6098	-77.64	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
6099	-77.66	oe	ccsbBroad304_00006	ACADM	-			
6100	-77.7	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
6101	-77.75	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
6102	-77.76	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6103	-77.78	cc		GPCR Subset GOF	-			
6104	-77.82	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
6105	-77.83	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
6106	-77.83	kd	CGS001-11019	LIAS	-			
6107	-77.86	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
6108	-77.96	kd	CGS001-4706	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
6109	-78.02	kd	CGS001-390	RND3	-			
6110	-78.03	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
6111	-78.04	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6112	-78.04	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
6113	-78.05	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
6114	-78.07	kd	CGS001-10745	PHTF1	-			
6115	-78.1	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
6116	-78.14	kd	CGS001-1490	CTGF	-			
6117	-78.18	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
6118	-78.27	cp	BRD-A41450521	tosufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6119	-78.27	kd	CGS001-11179	ZNF277	-			
6120	-78.31	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
6121	-78.32	kd	CGS001-8428	STK24	YSK subfamily			
6122	-78.37	oe	ccsbBroad304_01872	DGCR14	-			
6123	-78.39	kd	CGS001-9337	CNOT8	-			
6124	-78.4	kd	CGS001-5581	PRKCE	Eta subfamily			
6125	-78.43	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
6126	-78.43	oe	ccsbBroad304_00956	LYZ	-			
6127	-78.53	kd	CGS001-83999	KREMEN1	-			
6128	-78.55	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
6129	-78.55	oe	ccsbBroad304_08605	PBK	TOPK family			
6130	-78.59	oe	ccsbBroad304_00020	ACY1	-			
6131	-78.62	kd	CGS001-54108	CHRAC1	-			
6132	-78.64	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
6133	-78.7	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
6134	-78.71	kd	CGS001-51752	ERAP1	Aminopeptidase N			
6135	-78.73	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
6136	-78.76	kd	CGS001-7097	TLR2	Toll-like receptor family			
6137	-78.77	kd	CGS001-4179	CD46	CD molecules			
6138	-78.78	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
6139	-78.79	oe	ccsbBroad304_01556	SMARCB1	-			
6140	-78.92	oe	ccsbBroad304_14174	CDKAL1	-			
6141	-78.92	kd	CGS001-2212	FCGR2A	CD molecules			
6142	-78.93	kd	CGS001-7693	ZNF134	Zinc fingers, C2H2-type			
6143	-78.94	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
6144	-78.97	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
6145	-78.97	kd	CGS001-2224	FDPS	Lanosterol biosynthesis pathway			
6146	-78.98	kd	CGS001-406	ARNTL	Basic helix-loop-helix proteins			
6147	-79.03	kd	CGS001-3689	ITGB2	Integrins			
6148	-79.05	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
6149	-79.08	oe	ccsbBroad304_04194	ELL3	-			
6150	-79.29	kd	CGS001-4704	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6151	-79.35	oe	ccsbBroad304_02506	EBP	-			
6152	-79.49	kd	CGS001-84365	MKI67IP	-			
6153	-79.52	kd	CGS001-10198	MPHOSPH9	-			
6154	-79.54	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
6155	-79.61	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
6156	-79.63	kd	CGS001-7832	BTG2	-			
6157	-79.66	cc		Leucine rich repeat kinase inhibitor	-			
6158	-79.67	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
6159	-79.67	cp	BRD-A68888262	azelastine	Histamine receptor antagonist		HRH1, CYP2C19	Histamine receptor antagonist
6160	-79.7	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
6161	-79.79	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
6162	-79.8	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
6163	-79.84	oe	ccsbBroad304_00070	ANXA5	Annexins			
6164	-79.88	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
6165	-79.93	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
6166	-79.97	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
6167	-79.98	kd	CGS001-55644	OSGEP	-			
6168	-80	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
6169	-80.01	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
6170	-80.02	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
6171	-80.05	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
6172	-80.05	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6173	-80.07	kd	CGS001-572	BAD	-			
6174	-80.08	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
6175	-80.11	oe	ccsbBroad304_05439	O3FAR1	-			
6176	-80.13	kd	CGS001-6678	SPARC	-			
6177	-80.2	kd	CGS001-5164	PDK2	PDHK family			
6178	-80.24	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
6179	-80.25	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
6180	-80.36	oe	ccsbBroad304_00262	CD59	CD molecules			
6181	-80.44	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
6182	-80.49	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
6183	-80.5	oe	ccsbBroad304_02218	IKBKE	IKK family			
6184	-80.54	cc		DNA dependent protein kinase inhibitor	-			
6185	-80.55	kd	CGS001-6670	SP3	Specificity protein transcription factors			
6186	-80.55	kd	CGS001-64077	LHPP	-			
6187	-80.57	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
6188	-80.62	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
6189	-80.63	kd	CGS001-23621	BACE1	Pepsin			
6190	-80.66	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6191	-80.7	oe	ccsbBroad304_03604	ENOSF1	-			
6192	-80.81	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
6193	-80.86	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
6194	-80.9	kd	CGS001-116931	MED12L	-			
6195	-80.95	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
6196	-80.96	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
6197	-80.96	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
6198	-81.02	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
6199	-81.03	kd	CGS001-3251	HPRT1	-			
6200	-81.04	kd	CGS001-9352	TXNL1	-			
6201	-81.06	kd	CGS001-663	BNIP2	-			
6202	-81.14	kd	CGS001-5550	PREP	Prolyl oligopeptidase			
6203	-81.15	cp	BRD-A23637604	oxymetholone	Androgen receptor agonist		AR	Androgen receptor agonist
6204	-81.16	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
6205	-81.17	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
6206	-81.17	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
6207	-81.18	kd	CGS001-9322	TRIP10	-			
6208	-81.21	kd	CGS001-84515	MCM8	-			
6209	-81.22	kd	CGS001-51588	PIAS4	Zinc fingers, MIZ-type			
6210	-81.24	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
6211	-81.24	kd	CGS001-10955	SERINC3	-			
6212	-81.25	oe	ccsbBroad304_07528	DMTF1	-			
6213	-81.26	cc		Wnt family GOF	-			
6214	-81.27	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
6215	-81.31	kd	CGS001-36	ACADSB	-			
6216	-81.33	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
6217	-81.4	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
6218	-81.42	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
6219	-81.43	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
6220	-81.44	kd	CGS001-8431	NR0B2	DAX-like receptors			
6221	-81.53	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
6222	-81.53	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
6223	-81.54	kd	CGS001-9275	BCL7B	-			
6224	-81.55	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
6225	-81.59	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
6226	-81.62	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6227	-81.66	kd	CGS001-5563	PRKAA2	AMPK subfamily			
6228	-81.68	kd	CGS001-9943	OXSR1	FRAY subfamily			
6229	-81.76	kd	CGS001-10673	TNFSF13B	CD molecules			
6230	-81.8	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
6231	-81.84	kd	CGS001-5879	RAC1	Endogenous ligands			
6232	-81.85	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
6233	-81.86	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
6234	-81.88	oe	ccsbBroad304_00238	CCNE1	-			
6235	-81.89	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
6236	-81.91	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
6237	-81.93	cc		Toll like receptors LOF	-			
6238	-81.94	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
6239	-81.94	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6240	-81.95	kd	CGS001-5727	PTCH1	-			
6241	-81.97	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
6242	-81.98	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6243	-82.03	oe	ccsbBroad304_00152	BCAT2	-			
6244	-82.03	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
6245	-82.04	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
6246	-82.1	cp	BRD-A16444946	acarbose	Glucosidase inhibitor		GAA, MGAM, AMY2A, SI	Glucosidase inhibitor
6247	-82.18	oe	ccsbBroad304_00486	EFNB2	Ephrins			
6248	-82.29	kd	CGS001-2244	FGB	Endogenous ligands			
6249	-82.36	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
6250	-82.47	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
6251	-82.52	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
6252	-82.54	cc		Angiotensin receptor antagonist	-			
6253	-82.59	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
6254	-82.6	kd	CGS001-760	CA2	Carbonic anhydrases			
6255	-82.62	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
6256	-82.63	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
6257	-82.65	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6258	-82.66	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
6259	-82.66	kd	CGS001-6856	SYPL1	-			
6260	-82.66	kd	CGS001-11188	NISCH	-			
6261	-82.68	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
6262	-82.72	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
6263	-82.73	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
6264	-82.74	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
6265	-82.75	kd	CGS001-54807	ZNF586	Zinc fingers, C2H2-type			
6266	-82.75	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
6267	-82.78	oe	ccsbBroad304_06683	FURIN	Subtilisin			
6268	-82.79	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
6269	-82.79	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
6270	-82.82	oe	ccsbBroad304_06538	LSP1	-			
6271	-82.82	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
6272	-82.85	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
6273	-82.86	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
6274	-82.87	oe	ccsbBroad304_03910	CCDC90A	-			
6275	-82.89	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
6276	-82.94	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
6277	-82.94	kd	CGS001-578	BAK1	-			
6278	-82.97	oe	ccsbBroad304_03961	SMURF2	-			
6279	-82.99	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
6280	-83.02	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
6281	-83.03	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
6282	-83.04	kd	CGS001-6675	UAP1	-			
6283	-83.07	cc		RNA Polymerase Enzymes LOF	-			
6284	-83.08	oe	ccsbBroad304_02496	MTX2	-			
6285	-83.1	kd	CGS001-498	ATP5A1	ATPases / F-type			
6286	-83.11	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
6287	-83.21	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
6288	-83.23	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
6289	-83.29	kd	CGS001-165082	GPR113	Adhesion Class GPCRs			
6290	-83.31	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
6291	-83.38	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
6292	-83.42	oe	ccsbBroad304_08266	PIPOX	-			
6293	-83.45	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
6294	-83.47	kd	CGS001-5580	PRKCD	Delta subfamily			
6295	-83.48	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
6296	-83.54	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
6297	-83.56	oe	ccsbBroad304_02026	NRP1	CD molecules			
6298	-83.57	kd	CGS001-2859	GPR35	GPCR / Class A : Orphans			
6299	-83.65	kd	CGS001-3821	KLRC1	CD molecules			
6300	-83.66	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
6301	-83.71	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
6302	-83.73	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
6303	-83.73	kd	CGS001-81544	GDPD5	-			
6304	-83.75	cp	BRD-A02189320	met-leu-phe	-666			-666
6305	-83.76	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
6306	-83.82	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
6307	-83.85	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
6308	-83.9	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
6309	-84	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
6310	-84.04	kd	CGS001-9589	WTAP	-			
6311	-84.06	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6312	-84.07	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
6313	-84.09	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
6314	-84.09	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
6315	-84.12	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
6316	-84.16	kd	CGS001-87	ACTN1	EF-hand domain containing			
6317	-84.2	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
6318	-84.22	kd	CGS001-7150	TOP1	DNA Topoisomerases			
6319	-84.23	oe	ccsbBroad304_00975	MAT2A	-			
6320	-84.27	kd	CGS001-2909	ARHGAP35	Rho GTPase activating proteins			
6321	-84.32	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
6322	-84.35	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
6323	-84.36	oe	ccsbBroad304_00931	LCN2	Lipocalins			
6324	-84.36	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
6325	-84.36	cp	BRD-K99447003	enalaprilat	ACE inhibitor		ACE	ACE inhibitor
6326	-84.37	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
6327	-84.4	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
6328	-84.41	oe	ccsbBroad304_05985	CFL1	-			
6329	-84.42	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
6330	-84.43	kd	CGS001-57761	TRIB3	Trbl family			
6331	-84.45	kd	CGS001-136	ADORA2B	GPCR / Class A : Adenosine receptors			
6332	-84.54	oe	ccsbBroad304_05902	BNIP3	-			
6333	-84.54	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
6334	-84.55	kd	CGS001-661	POLR3D	RNA polymerase subunits			
6335	-84.56	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
6336	-84.58	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
6337	-84.59	kd	CGS001-2639	GCDH	-			
6338	-84.61	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
6339	-84.61	kd	CGS001-2160	F11	Chymotrypsin			
6340	-84.62	oe	ccsbBroad304_13813	ARAF	RAF family			
6341	-84.63	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
6342	-84.66	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
6343	-84.72	oe	ccsbBroad304_00954	LYN	Src family			
6344	-84.73	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
6345	-84.74	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
6346	-84.76	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
6347	-84.77	kd	CGS001-2538	G6PC	-			
6348	-84.79	kd	CGS001-4175	MCM6	-			
6349	-84.79	kd	CGS001-4287	ATXN3	Ataxins			
6350	-84.8	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
6351	-84.8	kd	CGS001-7083	TK1	-			
6352	-84.8	kd	CGS001-3199	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
6353	-84.8	kd	CGS001-2078	ERG	ETS Transcription Factors			
6354	-84.88	oe	ccsbBroad304_02239	RASSF2	-			
6355	-84.91	kd	CGS001-5255	PHKA1	-			
6356	-84.92	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
6357	-84.94	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
6358	-84.94	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
6359	-84.95	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
6360	-85.03	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
6361	-85.04	kd	CGS001-6258	RXRG	Retinoid X receptors			
6362	-85.08	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6363	-85.09	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
6364	-85.09	kd	CGS001-57157	PHTF2	-			
6365	-85.15	oe	ccsbBroad304_03268	GMPR2	-			
6366	-85.18	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
6367	-85.2	cc		Serotonin receptor agonist	-			
6368	-85.2	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
6369	-85.2	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
6370	-85.21	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
6371	-85.29	oe	ccsbBroad304_02318	KIF20A	Kinesins			
6372	-85.4	oe	ccsbBroad304_00053	ALDOA	-			
6373	-85.4	kd	CGS001-203523	ZNF449	Zinc fingers, C2H2-type			
6374	-85.44	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
6375	-85.46	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
6376	-85.48	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
6377	-85.56	kd	CGS001-11136	SLC7A9	SLC7 family			
6378	-85.62	kd	CGS001-10001	MED6	-			
6379	-85.64	kd	CGS001-23523	CABIN1	-			
6380	-85.68	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
6381	-85.68	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
6382	-85.74	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
6383	-85.76	kd	CGS001-3485	IGFBP2	insulin-like growth factor (IGF) binding proteins			
6384	-85.78	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
6385	-85.79	kd	CGS001-10051	SMC4	Structural maintenance of chromosomes proteins			
6386	-85.83	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
6387	-85.87	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
6388	-85.99	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
6389	-86.01	kd	CGS001-55810	FOXJ2	Forkhead boxes			
6390	-86.02	kd	CGS001-4087	SMAD2	SMADs			
6391	-86.06	oe	ccsbBroad304_06085	DCK	-			
6392	-86.06	kd	CGS001-7172	TPMT	-			
6393	-86.07	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
6394	-86.11	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
6395	-86.13	kd	CGS001-7155	TOP2B	DNA Topoisomerases			
6396	-86.16	kd	CGS001-4439	MSH5	-			
6397	-86.17	kd	CGS001-64343	AZI2	-			
6398	-86.18	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
6399	-86.23	kd	CGS001-4522	MTHFD1	-			
6400	-86.26	kd	CGS001-5277	PIGA	Glycosyltransferase group 1 domain containing			
6401	-86.28	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
6402	-86.41	oe	ccsbBroad304_07820	SNW1	-			
6403	-86.43	kd	CGS001-527	ATP6V0C	ATPases / V-type			
6404	-86.52	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
6405	-86.53	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
6406	-86.55	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
6407	-86.58	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
6408	-86.6	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
6409	-86.6	kd	CGS001-55770	EXOC2	-			
6410	-86.65	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
6411	-86.66	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
6412	-86.69	oe	ccsbBroad304_02092	SYNGR3	-			
6413	-86.71	oe	ccsbBroad304_01664	TGFA	-			
6414	-86.72	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
6415	-86.72	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
6416	-86.73	kd	CGS001-10857	PGRMC1	-			
6417	-86.74	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6418	-86.75	oe	ccsbBroad304_06739	PLOD1	-			
6419	-86.77	kd	CGS001-10614	HEXIM1	-			
6420	-86.8	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
6421	-86.84	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
6422	-86.85	cc		MCM family LOF	-			
6423	-86.92	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6424	-86.92	kd	CGS001-6850	SYK	Syk family			
6425	-86.94	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
6426	-86.95	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
6427	-86.97	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
6428	-86.98	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
6429	-87.04	kd	CGS001-116443	GRIN3A	Glutamate receptors			
6430	-87.14	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
6431	-87.18	kd	CGS001-11344	TWF2	Twinfilin subfamily			
6432	-87.2	oe	ccsbBroad304_02815	SSBP2	-			
6433	-87.2	kd	CGS001-256364	EML3	WD repeat domain containing			
6434	-87.21	kd	CGS001-586	BCAT1	-			
6435	-87.22	kd	CGS001-5230	PGK1	-			
6436	-87.23	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
6437	-87.27	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
6438	-87.28	kd	CGS001-4615	MYD88	-			
6439	-87.29	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
6440	-87.3	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
6441	-87.31	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
6442	-87.31	kd	CGS001-84433	CARD11	-			
6443	-87.32	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
6444	-87.32	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
6445	-87.4	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
6446	-87.43	kd	CGS001-5352	PLOD2	-			
6447	-87.44	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
6448	-87.44	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6449	-87.46	oe	ccsbBroad304_03072	GTPBP8	-			
6450	-87.51	kd	CGS001-10023	FRAT1	-			
6451	-87.52	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
6452	-87.56	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
6453	-87.56	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
6454	-87.56	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
6455	-87.59	oe	ccsbBroad304_06382	HMGCL	-			
6456	-87.61	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
6457	-87.65	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
6458	-87.66	kd	CGS001-5934	RBL2	-			
6459	-87.69	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
6460	-87.71	oe	ccsbBroad304_06282	GLDC	-			
6461	-87.72	kd	CGS001-112858	TP53RK	Bud32 family			
6462	-87.76	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
6463	-87.77	kd	CGS001-285267	ZNF619	Zinc fingers, C2H2-type			
6464	-87.78	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
6465	-87.81	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
6466	-87.83	cp	BRD-K19462402	buflomedil	Adrenergic receptor antagonist		CACNA1C	Adrenergic receptor antagonist, Calcium channel blocker
6467	-87.91	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
6468	-87.91	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
6469	-87.91	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6470	-87.96	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
6471	-87.96	kd	CGS001-5433	POLR2D	RNA polymerase subunits			
6472	-88.01	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
6473	-88.04	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
6474	-88.09	kd	CGS001-26227	PHGDH	-			
6475	-88.16	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
6476	-88.22	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
6477	-88.24	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
6478	-88.25	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
6479	-88.28	cp	BRD-K17705806	JTC-801	Opioid receptor antagonist		OPRL1	Opioid receptor antagonist
6480	-88.3	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6481	-88.31	kd	CGS001-11004	KIF2C	Kinesins			
6482	-88.38	kd	CGS001-9655	SOCS5	SH2 domain containing			
6483	-88.4	oe	ccsbBroad304_03878	SENP2	-			
6484	-88.47	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
6485	-88.48	cp	BRD-K52080565	rilmenidine	Imidazoline receptor agonist		NISCH	Imidazoline receptor agonist
6486	-88.53	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
6487	-88.53	kd	CGS001-6924	TCEB3	-			
6488	-88.53	kd	CGS001-10174	SORBS3	-			
6489	-88.54	kd	CGS001-8741	TNFSF13	CD molecules			
6490	-88.63	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
6491	-88.65	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
6492	-88.69	kd	CGS001-4194	MDM4	-			
6493	-88.7	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
6494	-88.72	oe	ccsbBroad304_03173	TMED7	-			
6495	-88.74	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
6496	-88.74	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
6497	-88.75	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
6498	-88.78	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
6499	-88.8	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
6500	-88.83	kd	CGS001-10915	TCERG1	-			
6501	-88.84	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
6502	-88.85	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
6503	-88.86	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
6504	-88.88	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6505	-88.89	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6506	-88.92	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
6507	-88.92	cp	BRD-A64297288	amlodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, ABCG2, CA1, CACNA1B, CACNA1S, CACNA2D3, CACNB1, CACNB2, SMPD1	Calcium channel blocker
6508	-88.97	kd	CGS001-3516	RBPJ	-			
6509	-88.98	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
6510	-88.99	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
6511	-89.02	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
6512	-89.02	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
6513	-89.02	kd	CGS001-22954	TRIM32	-			
6514	-89.02	kd	CGS001-2745	GLRX	-			
6515	-89.04	cc		HSP inhibitor	-			
6516	-89.13	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
6517	-89.15	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6518	-89.17	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
6519	-89.18	kd	CGS001-51135	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
6520	-89.21	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
6521	-89.21	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6522	-89.24	oe	ccsbBroad304_08536	PARL	-			
6523	-89.24	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
6524	-89.24	kd	CGS001-60493	FASTKD5	-			
6525	-89.25	kd	CGS001-6647	SOD1	-			
6526	-89.31	kd	CGS001-10474	TADA3	-			
6527	-89.33	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
6528	-89.34	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
6529	-89.38	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
6530	-89.42	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
6531	-89.43	kd	CGS001-3654	IRAK1	Interleukin-1 receptor-associated kinase (IRAK) family			
6532	-89.43	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
6533	-89.45	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
6534	-89.45	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
6535	-89.49	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
6536	-89.5	kd	CGS001-650	BMP2	Bone morphogenetic proteins			
6537	-89.51	kd	CGS001-64147	KIF9	Kinesins			
6538	-89.52	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
6539	-89.53	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6540	-89.53	kd	CGS001-2232	FDXR	-			
6541	-89.53	kd	CGS001-23581	CASP14	Caspases			
6542	-89.56	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
6543	-89.62	kd	CGS001-4254	KITLG	-			
6544	-89.65	oe	ccsbBroad304_09095	PUS7L	-			
6545	-89.65	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
6546	-89.75	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
6547	-89.78	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
6548	-89.79	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
6549	-89.82	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
6550	-89.86	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
6551	-89.88	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
6552	-89.89	oe	ccsbBroad304_02373	SPRY2	-			
6553	-89.92	cc		ATPase inhibitor	-			
6554	-89.94	kd	CGS001-975	CD81	CD molecules			
6555	-89.97	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
6556	-89.99	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
6557	-90.03	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
6558	-90.08	kd	CGS001-10398	MYL9	EF-hand domain containing			
6559	-90.08	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
6560	-90.09	kd	CGS001-10914	PAPOLA	-			
6561	-90.1	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
6562	-90.15	kd	CGS001-1649	DDIT3	-			
6563	-90.16	oe	ccsbBroad304_07101	TSC2	-			
6564	-90.18	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
6565	-90.2	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
6566	-90.21	kd	CGS001-5641	LGMN	Legumain			
6567	-90.22	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
6568	-90.23	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
6569	-90.23	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
6570	-90.23	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
6571	-90.23	kd	CGS001-5063	PAK3	PAKA subfamily			
6572	-90.26	kd	CGS001-2760	GM2A	-			
6573	-90.27	kd	CGS001-1606	DGKA	EF-hand domain containing			
6574	-90.27	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
6575	-90.28	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
6576	-90.32	oe	ccsbBroad304_07531	TANK	-			
6577	-90.34	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
6578	-90.36	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
6579	-90.36	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
6580	-90.36	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
6581	-90.36	kd	CGS001-8850	KAT2B	Histone acetyltransferases (HATs)			
6582	-90.4	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
6583	-90.4	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
6584	-90.47	oe	ccsbBroad304_03119	C16ORF5	-			
6585	-90.47	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
6586	-90.48	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
6587	-90.55	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
6588	-90.55	kd	CGS001-8986	RPS6KA4	MSK subfamily			
6589	-90.59	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
6590	-90.61	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
6591	-90.63	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6592	-90.65	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
6593	-90.65	kd	CGS001-6500	SKP1	-			
6594	-90.69	kd	CGS001-6208	RPS14	S ribosomal proteins			
6595	-90.8	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
6596	-90.83	kd	CGS001-7056	THBD	CD molecules			
6597	-90.84	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
6598	-90.84	kd	CGS001-23761	PISD	Decarboxylases			
6599	-90.85	kd	CGS001-5211	PFKL	-			
6600	-90.85	oe	ccsbBroad304_00389	CTBP1	-			
6601	-90.85	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
6602	-90.86	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
6603	-90.86	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6604	-90.86	kd	CGS001-6603	SMARCD2	-			
6605	-90.87	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
6606	-90.88	kd	CGS001-345611	IRGM	-			
6607	-90.92	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
6608	-90.99	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
6609	-91.01	kd	CGS001-1173	AP2M1	-			
6610	-91.05	kd	CGS001-9	NAT1	-			
6611	-91.08	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6612	-91.09	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
6613	-91.1	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
6614	-91.13	kd	CGS001-84539	MCHR2	GPCR / Class A : MCH receptors			
6615	-91.13	kd	CGS001-84930	MASTL	MAST family			
6616	-91.15	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
6617	-91.15	kd	CGS001-132	ADK	Adenosine turnover			
6618	-91.16	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
6619	-91.17	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
6620	-91.17	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
6621	-91.2	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
6622	-91.2	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
6623	-91.22	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
6624	-91.23	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
6625	-91.27	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
6626	-91.3	cc		Canonical high mobility group proteins LOF	-			
6627	-91.3	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6628	-91.32	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6629	-91.36	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6630	-91.41	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
6631	-91.42	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
6632	-91.42	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
6633	-91.42	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
6634	-91.45	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
6635	-91.47	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6636	-91.48	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
6637	-91.49	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
6638	-91.53	oe	ccsbBroad304_03097	CNOT7	-			
6639	-91.56	kd	CGS001-440	ASNS	-			
6640	-91.57	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
6641	-91.61	kd	CGS001-5193	PEX12	-			
6642	-91.64	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
6643	-91.67	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
6644	-91.72	kd	CGS001-7424	VEGFC	-			
6645	-91.78	kd	CGS001-1676	DFFA	-			
6646	-91.79	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
6647	-91.8	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
6648	-91.81	kd	CGS001-10962	MLLT11	-			
6649	-91.82	kd	CGS001-147179	WIPF2	-			
6650	-91.83	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
6651	-91.85	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6652	-91.87	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
6653	-91.87	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
6654	-91.89	kd	CGS001-51520	LARS	Aminoacyl tRNA synthetases / Class I			
6655	-91.91	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6656	-91.93	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
6657	-91.97	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
6658	-91.97	kd	CGS001-8408	ULK1	Unc-51-like kinase (ULK) family			
6659	-91.98	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
6660	-92.01	oe	ccsbBroad304_02285	MED6	-			
6661	-92.03	oe	ccsbBroad304_02205	WTAP	-			
6662	-92.03	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
6663	-92.04	oe	ccsbBroad304_02737	JMJD6	-			
6664	-92.04	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
6665	-92.04	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
6666	-92.05	kd	CGS001-22796	COG2	Components of oligomeric golgi complex			
6667	-92.07	kd	CGS001-6193	RPS5	S ribosomal proteins			
6668	-92.1	kd	CGS001-51347	TAOK3	TAO subfamily			
6669	-92.1	kd	CGS001-85315	PAQR8	-			
6670	-92.12	kd	CGS001-1635	DCTD	-			
6671	-92.16	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
6672	-92.16	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
6673	-92.16	kd	CGS001-22978	NT5C2	Adenosine turnover			
6674	-92.19	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
6675	-92.2	kd	CGS001-23224	SYNE2	-			
6676	-92.26	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
6677	-92.26	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
6678	-92.29	oe	ccsbBroad304_01527	SGK1	SGK family			
6679	-92.32	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
6680	-92.36	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
6681	-92.37	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
6682	-92.41	kd	CGS001-23223	RRP12	-			
6683	-92.43	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
6684	-92.46	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
6685	-92.46	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
6686	-92.47	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
6687	-92.5	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
6688	-92.5	kd	CGS001-1831	TSC22D3	-			
6689	-92.5	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
6690	-92.5	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
6691	-92.52	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
6692	-92.59	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
6693	-92.6	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
6694	-92.6	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
6695	-92.6	kd	CGS001-7099	TLR4	Toll-like receptor family			
6696	-92.61	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
6697	-92.65	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
6698	-92.65	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
6699	-92.65	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
6700	-92.68	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
6701	-92.68	kd	CGS001-390212	GPR152	GPCR / Class A : Orphans			
6702	-92.72	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
6703	-92.73	oe	ccsbBroad304_05947	CCNC	-			
6704	-92.74	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
6705	-92.76	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
6706	-92.78	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
6707	-92.79	oe	ccsbBroad304_00490	EIF4EBP1	-			
6708	-92.82	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
6709	-92.85	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
6710	-92.86	kd	CGS001-4173	MCM4	-			
6711	-92.87	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
6712	-92.9	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
6713	-92.91	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
6714	-92.91	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
6715	-92.94	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
6716	-92.94	kd	CGS001-5981	RFC1	ATPases / AAA-type			
6717	-92.94	kd	CGS001-3827	KNG1	Endogenous ligands			
6718	-92.97	oe	ccsbBroad304_01769	VEGFB	-			
6719	-93.01	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
6720	-93.02	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
6721	-93.02	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
6722	-93.03	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
6723	-93.04	kd	CGS001-23212	RRS1	-			
6724	-93.07	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
6725	-93.09	kd	CGS001-2793	GNGT2	-			
6726	-93.12	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
6727	-93.12	kd	CGS001-4605	MYBL2	-			
6728	-93.12	kd	CGS001-8226	HDHD1	-			
6729	-93.2	kd	CGS001-7037	TFRC	CD molecules			
6730	-93.25	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
6731	-93.28	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
6732	-93.34	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
6733	-93.34	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
6734	-93.35	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
6735	-93.38	kd	CGS001-3897	L1CAM	CD molecules			
6736	-93.4	cc		Structural maintenance of chromosomes proteins LOF	-			
6737	-93.4	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
6738	-93.42	kd	CGS001-55937	APOM	Apolipoproteins			
6739	-93.43	cp	BRD-M47937986	cefatrizine	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6740	-93.45	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
6741	-93.46	cc		CDK inhibitor	-			
6742	-93.49	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
6743	-93.52	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
6744	-93.54	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
6745	-93.55	kd	CGS001-3880	KRT19	Intermediate filaments type I, keratins (acidic)			
6746	-93.57	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
6747	-93.57	kd	CGS001-5979	RET	Type XIV RTKs: RET			
6748	-93.58	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6749	-93.59	kd	CGS001-998	CDC42	-			
6750	-93.6	kd	CGS001-55869	HDAC8	Histone deacetylases			
6751	-93.65	cc		Estrogen receptor agonist	-			
6752	-93.68	kd	CGS001-3589	IL11	Endogenous ligands			
6753	-93.68	kd	CGS001-10481	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
6754	-93.68	kd	CGS001-283150	FOXR1	Forkhead boxes			
6755	-93.72	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
6756	-93.73	kd	CGS001-4751	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6757	-93.78	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
6758	-93.79	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
6759	-93.8	kd	CGS001-51569	UFM1	-			
6760	-93.82	kd	CGS001-3705	ITPK1	-			
6761	-93.85	kd	CGS001-8548	BLZF1	-			
6762	-93.86	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
6763	-93.86	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
6764	-93.86	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
6765	-93.89	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
6766	-93.89	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
6767	-93.9	oe	ccsbBroad304_00003	ABAT	GABA turnover			
6768	-93.91	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
6769	-93.92	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
6770	-93.94	cc		Potassium channel activator	-			
6771	-93.95	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
6772	-93.95	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
6773	-93.96	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
6774	-93.97	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
6775	-94	oe	ccsbBroad304_05135	PARP15	-			
6776	-94.03	kd	CGS001-205564	SENP5	-			
6777	-94.11	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
6778	-94.11	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
6779	-94.14	kd	CGS001-1736	DKC1	-			
6780	-94.17	cp	BRD-A92630576	trimebutine	Opioid receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Opioid receptor agonist
6781	-94.17	kd	CGS001-1643	DDB2	WD repeat domain containing			
6782	-94.18	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
6783	-94.2	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
6784	-94.21	kd	CGS001-3569	IL6	Interferons			
6785	-94.25	oe	ccsbBroad304_03808	ERGIC1	-			
6786	-94.25	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6787	-94.25	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
6788	-94.37	oe	ccsbBroad304_01723	TTK	TTK family			
6789	-94.37	kd	CGS001-899	CCNF	F-boxes / other			
6790	-94.38	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
6791	-94.42	kd	CGS001-63892	THADA	-			
6792	-94.44	oe	ccsbBroad304_02432	IFI30	-			
6793	-94.44	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
6794	-94.44	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
6795	-94.44	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6796	-94.46	oe	ccsbBroad304_06975	SMARCC2	-			
6797	-94.46	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
6798	-94.46	kd	CGS001-4968	OGG1	-			
6799	-94.47	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
6800	-94.5	oe	ccsbBroad304_02565	RALBP1	-			
6801	-94.51	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
6802	-94.51	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
6803	-94.54	cc		Glycogen synthase kinase inhibitor	-			
6804	-94.54	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
6805	-94.56	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
6806	-94.58	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
6807	-94.6	kd	CGS001-9261	MAPKAPK2	MAPKAPK subfamily			
6808	-94.62	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
6809	-94.63	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
6810	-94.64	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
6811	-94.64	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
6812	-94.64	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
6813	-94.67	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
6814	-94.69	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
6815	-94.72	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
6816	-94.73	kd	CGS001-1837	DTNA	-			
6817	-94.76	oe	ccsbBroad304_01148	PCBD1	-			
6818	-94.78	oe	ccsbBroad304_06828	PYCR1	-			
6819	-94.78	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
6820	-94.78	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
6821	-94.82	cp	BRD-A01787639	naftopidil	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
6822	-94.84	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
6823	-94.85	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
6824	-94.88	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
6825	-94.88	kd	CGS001-6541	SLC7A1	SLC7 family			
6826	-94.93	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
6827	-94.96	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
6828	-94.96	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
6829	-94.97	cp	BRD-K22947005	dexbrompheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6830	-94.97	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
6831	-95.02	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
6832	-95.02	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6833	-95.05	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
6834	-95.07	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
6835	-95.08	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6836	-95.09	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
6837	-95.1	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
6838	-95.11	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
6839	-95.14	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
6840	-95.14	kd	CGS001-9774	BCLAF1	-			
6841	-95.15	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
6842	-95.16	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
6843	-95.22	cc		Phospholipases LOF	-			
6844	-95.24	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
6845	-95.27	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
6846	-95.28	oe	ccsbBroad304_07889	QPRT	-			
6847	-95.3	oe	ccsbBroad304_04649	ADC	-			
6848	-95.32	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
6849	-95.33	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
6850	-95.34	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
6851	-95.34	cp	BRD-K30563334	rifabutin	Protein synthesis inhibitor		CYP3A4, HSP90AA1, HSP90B1	Protein synthesis inhibitor
6852	-95.35	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
6853	-95.37	oe	ccsbBroad304_02485	STAMBP	-			
6854	-95.37	kd	CGS001-4846	NOS3	Nitric oxide synthases			
6855	-95.39	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6856	-95.4	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
6857	-95.41	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
6858	-95.45	kd	CGS001-2261	FGFR3	Type V RTKs: FGF (fibroblast growth factor) receptor family			
6859	-95.46	oe	ccsbBroad304_02572	SERINC3	-			
6860	-95.47	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
6861	-95.53	cc		Na-K-Cl transporter inhibitor	-			
6862	-95.54	kd	CGS001-89910	UBE3B	-			
6863	-95.54	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
6864	-95.54	kd	CGS001-1497	CTNS	-			
6865	-95.57	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
6866	-95.61	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
6867	-95.67	cc		Protein synthesis inhibitor	-			
6868	-95.67	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
6869	-95.67	kd	CGS001-9690	UBE3C	-			
6870	-95.68	cc		Baculoviral IAP repeat domain containing LOF	-			
6871	-95.72	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
6872	-95.75	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
6873	-95.76	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
6874	-95.76	kd	CGS001-51284	TLR7	Toll-like receptor family			
6875	-95.78	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
6876	-95.78	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
6877	-95.8	cc		Calcium channel blocker	-			
6878	-95.82	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
6879	-95.86	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
6880	-95.87	kd	CGS001-1453	CSNK1D	Casein kinase 1 (CK1) family			
6881	-95.87	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
6882	-95.89	kd	CGS001-4547	MTTP	-			
6883	-95.89	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
6884	-95.9	kd	CGS001-4790	NFKB1	NFkappaB transcription factor family			
6885	-95.95	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
6886	-95.96	kd	CGS001-204851	HIPK1	HIPK subfamily			
6887	-95.96	kd	CGS001-10094	ARPC3	Actin related protein 2/3 complex subunits			
6888	-95.98	oe	ccsbBroad304_02702	MSRB2	-			
6889	-96.01	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
6890	-96.01	kd	CGS001-2618	GART	Ribosyl transferases			
6891	-96.02	oe	ccsbBroad304_00394	CTSD	Cathepsins			
6892	-96.04	kd	CGS001-54556	ING3	Zinc fingers, PHD-type			
6893	-96.04	kd	CGS001-51380	CSAD	-			
6894	-96.05	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
6895	-96.07	kd	CGS001-4204	MECP2	-			
6896	-96.12	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6897	-96.15	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
6898	-96.16	kd	CGS001-5428	POLG	DNA polymerases			
6899	-96.16	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6900	-96.17	oe	ccsbBroad304_07491	IP6K1	-			
6901	-96.17	kd	CGS001-8836	GGH	Gamma-glutamyl hydrolase			
6902	-96.17	kd	CGS001-10097	ACTR2	-			
6903	-96.21	oe	ccsbBroad304_06993	SRD5A1	-			
6904	-96.23	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
6905	-96.25	kd	CGS001-4092	SMAD7	SMADs			
6906	-96.26	kd	CGS001-26191	PTPN22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6907	-96.27	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
6908	-96.3	kd	CGS001-1213	CLTC	-			
6909	-96.32	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
6910	-96.32	kd	CGS001-2118	ETV4	ETS Transcription Factors			
6911	-96.36	cc		IKK inhibitor	-			
6912	-96.37	kd	CGS001-11212	PROSC	-			
6913	-96.39	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
6914	-96.4	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
6915	-96.41	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
6916	-96.42	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
6917	-96.42	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
6918	-96.42	kd	CGS001-150280	HORMAD2	-			
6919	-96.45	cc		Trace amine receptors LOF	-			
6920	-96.45	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
6921	-96.45	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
6922	-96.49	oe	ccsbBroad304_07275	PSMG1	-			
6923	-96.53	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
6924	-96.53	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
6925	-96.53	kd	CGS001-9900	SV2A	Major facilitator superfamily (MFS) of transporters			
6926	-96.54	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
6927	-96.54	kd	CGS001-3755	KCNG1	Voltage-gated potassium channels			
6928	-96.58	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
6929	-96.59	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
6930	-96.61	kd	CGS001-23325	KIAA1033	-			
6931	-96.62	kd	CGS001-5686	PSMA5	Proteasome subunits			
6932	-96.63	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
6933	-96.64	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
6934	-96.68	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
6935	-96.7	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
6936	-96.71	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
6937	-96.72	kd	CGS001-2990	GUSB	-			
6938	-96.74	kd	CGS001-716	C1S	Complement system			
6939	-96.75	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
6940	-96.76	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6941	-96.76	oe	ccsbBroad304_04399	PGBD1	-			
6942	-96.76	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
6943	-96.76	kd	CGS001-51053	GMNN	-			
6944	-96.78	kd	CGS001-5338	PLD2	Hydrolases			
6945	-96.78	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
6946	-96.82	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
6947	-96.83	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
6948	-96.83	kd	CGS001-54749	EPDR1	-			
6949	-96.85	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
6950	-96.87	kd	CGS001-5144	PDE4D	Phosphodiesterases			
6951	-96.87	kd	CGS001-6885	MAP3K7	MAPKKK:TAK1 subfamily			
6952	-96.91	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
6953	-96.91	kd	CGS001-1910	EDNRB	Endothelin receptors			
6954	-96.92	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
6955	-96.96	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
6956	-96.98	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
6957	-96.99	kd	CGS001-28985	MCTS1	-			
6958	-96.99	kd	CGS001-1622	DBI	-			
6959	-96.99	kd	CGS001-29965	C16ORF5	-			
6960	-97.03	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
6961	-97.03	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
6962	-97.06	kd	CGS001-3895	KTN1	-			
6963	-97.07	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6964	-97.07	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
6965	-97.08	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
6966	-97.1	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
6967	-97.11	kd	CGS001-1948	EFNB2	Ephrins			
6968	-97.13	cp	BRD-K63343048	orlistat	Lipase inhibitor		PNLIP, DAGLA, FASN, LIPF, CNR1, DAGLB	Lipase inhibitor
6969	-97.13	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
6970	-97.14	cp	BRD-K52020312	metronidazole	DNA inhibitor		CYP2C8, CYP2E1, CYP3A5, CYP3A7	DNA inhibitor, Antiprotozoal
6971	-97.16	cp	BRD-K28849549	mesalazine	Cyclooxygenase inhibitor		PTGS1, PPARG, PTGS2, ALOX5, CHUK, CTNNB1, IKBKB, MPO, NAT1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor, Prostanoid receptor antagonist
6972	-97.16	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
6973	-97.18	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6974	-97.19	kd	CGS001-6203	RPS9	S ribosomal proteins			
6975	-97.22	oe	ccsbBroad304_06665	OAT	-			
6976	-97.24	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
6977	-97.24	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
6978	-97.24	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
6979	-97.24	kd	CGS001-2932	GSK3B	GSK subfamily			
6980	-97.27	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
6981	-97.28	oe	ccsbBroad304_01373	RAN	-			
6982	-97.28	kd	CGS001-573	BAG1	-			
6983	-97.29	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
6984	-97.31	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
6985	-97.32	oe	ccsbBroad304_00101	RHOC	-			
6986	-97.34	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
6987	-97.39	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
6988	-97.39	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
6989	-97.39	kd	CGS001-1431	CS	-			
6990	-97.39	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
6991	-97.4	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
6992	-97.41	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
6993	-97.41	kd	CGS001-3783	KCNN4	Calcium-activated potassium channels			
6994	-97.42	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
6995	-97.44	oe	ccsbBroad304_06562	MAT1A	-			
6996	-97.44	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
6997	-97.44	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
6998	-97.45	kd	CGS001-28964	GIT1	Ankyrin repeat domain containing			
6999	-97.45	kd	CGS001-23365	ARHGEF12	Rho guanine nucleotide exchange factors			
7000	-97.46	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
7001	-97.48	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
7002	-97.5	cp	BRD-K39391626	ethylestrenol	Progesterone receptor agonist		AR	Progesterone receptor agonist
7003	-97.51	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
7004	-97.56	kd	CGS001-55379	LRRC59	-			
7005	-97.57	kd	CGS001-3590	IL11RA	IL-6 receptor family			
7006	-97.58	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
7007	-97.58	kd	CGS001-2289	FKBP5	Tetratricopeptide (TTC) repeat domain containing			
7008	-97.6	kd	CGS001-5209	PFKFB3	-			
7009	-97.62	oe	ccsbBroad304_07267	PDLIM4	-			
7010	-97.62	cp	BRD-K85030058	benactyzine	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
7011	-97.64	oe	ccsbBroad304_00644	GCLC	-			
7012	-97.64	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7013	-97.65	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
7014	-97.66	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
7015	-97.71	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
7016	-97.74	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
7017	-97.74	kd	CGS001-8543	LMO4	-			
7018	-97.75	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
7019	-97.77	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
7020	-97.78	kd	CGS001-271	AMPD2	-			
7021	-97.79	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
7022	-97.79	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
7023	-97.8	cp	BRD-K10065684	dantron	Laxative			Laxative
7024	-97.81	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
7025	-97.81	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
7026	-97.83	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
7027	-97.86	kd	CGS001-22933	SIRT2	Histone deacetylases			
7028	-97.86	kd	CGS001-5062	PAK2	PAKA subfamily			
7029	-97.88	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
7030	-97.89	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
7031	-97.91	oe	ccsbBroad304_01623	SUPT4H1	-			
7032	-97.92	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
7033	-97.96	kd	CGS001-9710	KIAA0355	-			
7034	-97.97	kd	CGS001-25801	GCA	EF-hand domain containing			
7035	-97.98	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
7036	-97.98	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
7037	-97.98	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
7038	-97.99	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
7039	-97.99	kd	CGS001-8477	GPR65	GPCR / Class A : Orphans			
7040	-97.99	kd	CGS001-2752	GLUL	-			
7041	-98.01	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7042	-98.01	kd	CGS001-56731	SLC2A4RG	-			
7043	-98.03	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
7044	-98.05	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
7045	-98.06	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
7046	-98.08	kd	CGS001-4292	MLH1	-			
7047	-98.1	oe	ccsbBroad304_01673	TIMP3	-			
7048	-98.11	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
7049	-98.14	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
7050	-98.15	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
7051	-98.16	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
7052	-98.16	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
7053	-98.16	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
7054	-98.17	kd	CGS001-7474	WNT5A	Endogenous ligands			
7055	-98.18	oe	ccsbBroad304_00249	CD14	CD molecules			
7056	-98.18	kd	CGS001-7511	XPNPEP1	Methionyl aminopeptidase			
7057	-98.18	kd	CGS001-2057	EPOR	Prolactin receptor family			
7058	-98.18	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
7059	-98.19	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
7060	-98.2	kd	CGS001-3988	LIPA	-			
7061	-98.21	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
7062	-98.21	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
7063	-98.24	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
7064	-98.25	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
7065	-98.27	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
7066	-98.27	kd	CGS001-5914	RARA	Retinoic acid receptors			
7067	-98.29	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
7068	-98.29	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
7069	-98.3	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
7070	-98.31	oe	ccsbBroad304_05183	TXLNA	-			
7071	-98.31	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
7072	-98.32	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
7073	-98.32	oe	ccsbBroad304_02604	B3GNT1	-			
7074	-98.32	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
7075	-98.34	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
7076	-98.36	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
7077	-98.36	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
7078	-98.38	oe	ccsbBroad304_00034	AES	-			
7079	-98.38	cp	BRD-A96107863	nisoldipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNB2, CYP3A5	Calcium channel blocker
7080	-98.38	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
7081	-98.39	kd	CGS001-10397	NDRG1	-			
7082	-98.4	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
7083	-98.4	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
7084	-98.45	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
7085	-98.47	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
7086	-98.47	kd	CGS001-7090	TLE3	WD repeat domain containing			
7087	-98.47	kd	CGS001-2495	FTH1	-			
7088	-98.47	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7089	-98.49	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
7090	-98.49	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
7091	-98.49	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
7092	-98.49	kd	CGS001-7298	TYMS	Methyltransferases			
7093	-98.51	oe	ccsbBroad304_09054	EGFL8	-			
7094	-98.51	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
7095	-98.51	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
7096	-98.51	kd	CGS001-64422	ATG3	-			
7097	-98.53	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7098	-98.54	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
7099	-98.56	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
7100	-98.58	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
7101	-98.58	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
7102	-98.59	cp	BRD-K10670311	sulfasalazine	Antirheumatic		PTGS1, PTGS2, ACAT1, ALOX5, CHUK, IKBKB, PLA2G1B, PPARG, SLC46A1, SLC7A11, TBXAS1	Antirheumatic, NFkB pathway inhibitor
7103	-98.59	kd	CGS001-5916	RARG	Retinoic acid receptors			
7104	-98.6	oe	ccsbBroad304_02367	CALCOCO2	-			
7105	-98.6	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
7106	-98.6	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
7107	-98.61	kd	CGS001-339403	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
7108	-98.62	kd	CGS001-64241	ABCG8	ATP binding cassette transporters / subfamily G			
7109	-98.64	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
7110	-98.64	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
7111	-98.65	oe	ccsbBroad304_00184	C2	Complement system			
7112	-98.67	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
7113	-98.67	oe	ccsbBroad304_00518	ETFA	-			
7114	-98.67	kd	CGS001-10616	RBCK1	RING-type (C3HC4) zinc fingers			
7115	-98.67	kd	CGS001-93185	IGSF8	CD molecules			
7116	-98.67	kd	CGS001-1594	CYP27B1	Cytochrome P450s			
7117	-98.69	oe	ccsbBroad304_01716	TSN	-			
7118	-98.69	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
7119	-98.69	kd	CGS001-6776	STAT5A	SH2 domain containing			
7120	-98.7	kd	CGS001-50814	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7121	-98.73	kd	CGS001-1460	CSNK2B	Casein kinase 2 (CK2) family			
7122	-98.75	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
7123	-98.75	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
7124	-98.75	kd	CGS001-51335	NGRN	-			
7125	-98.76	kd	CGS001-7010	TEK	Type XII RTKs: TIE family of angiopoietin receptors			
7126	-98.76	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
7127	-98.8	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
7128	-98.8	kd	CGS001-23585	TMEM50A	-			
7129	-98.8	kd	CGS001-8635	RNASET2	-			
7130	-98.81	oe	ccsbBroad304_07287	HYAL2	-			
7131	-98.81	kd	CGS001-18	ABAT	GABA turnover			
7132	-98.82	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
7133	-98.82	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
7134	-98.83	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
7135	-98.86	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
7136	-98.86	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7137	-98.86	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
7138	-98.87	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
7139	-98.88	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
7140	-98.88	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
7141	-98.88	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
7142	-98.88	kd	CGS001-3651	PDX1	Homeoboxes / ANTP class : HOXL subclass			
7143	-98.89	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
7144	-98.9	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
7145	-98.91	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
7146	-98.91	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
7147	-98.91	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
7148	-98.91	kd	CGS001-6499	SKIV2L	-			
7149	-98.91	kd	CGS001-6469	SHH	-			
7150	-98.91	kd	CGS001-2247	FGF2	Endogenous ligands			
7151	-98.91	kd	CGS001-79174	CRELD2	-			
7152	-98.95	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
7153	-98.95	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
7154	-98.95	kd	CGS001-645	BLVRB	Short chain dehydrogenase/reductase superfamily / Atypical members			
7155	-98.96	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
7156	-98.96	kd	CGS001-10318	TNIP1	-			
7157	-98.97	kd	CGS001-4864	NPC1	-			
7158	-98.98	kd	CGS001-1728	NQO1	-			
7159	-98.99	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
7160	-99	kd	CGS001-10672	GNA13	-			
7161	-99.02	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
7162	-99.04	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
7163	-99.04	oe	ccsbBroad304_00657	GNG4	-			
7164	-99.04	kd	CGS001-10329	TMEM5	-			
7165	-99.04	kd	CGS001-2152	F3	CD molecules			
7166	-99.04	kd	CGS001-54805	CNNM2	-			
7167	-99.05	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
7168	-99.06	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
7169	-99.06	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
7170	-99.06	kd	CGS001-84923	FAM104A	-			
7171	-99.08	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7172	-99.08	kd	CGS001-55876	GSDMB	-			
7173	-99.08	kd	CGS001-2237	FEN1	-			
7174	-99.09	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
7175	-99.1	cc		Serine proteases GOF	-			
7176	-99.1	cc		Minor histocompatibility antigens LOF	-			
7177	-99.1	cp	BRD-K01649396	indatraline	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine transporter inhibitor
7178	-99.1	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
7179	-99.11	kd	CGS001-84527	ZNF559	Zinc fingers, C2H2-type			
7180	-99.12	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
7181	-99.12	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
7182	-99.12	cp	BRD-K15842202	eudesmic-acid	-666			-666
7183	-99.12	kd	CGS001-11254	SLC6A14	Glycine transporter subfamily			
7184	-99.14	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
7185	-99.15	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
7186	-99.15	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
7187	-99.15	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
7188	-99.15	kd	CGS001-81539	SLC38A1	System A-like transporters			
7189	-99.15	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
7190	-99.17	oe	ccsbBroad304_07320	SQSTM1	-			
7191	-99.17	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
7192	-99.17	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
7193	-99.17	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
7194	-99.19	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
7195	-99.19	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
7196	-99.19	oe	ccsbBroad304_03732	NPDC1	-			
7197	-99.19	kd	CGS001-4916	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
7198	-99.2	oe	ccsbBroad304_01658	PRDX2	-			
7199	-99.2	oe	ccsbBroad304_00728	HBE1	-			
7200	-99.21	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
7201	-99.21	oe	ccsbBroad304_00099	ARG2	Arginase			
7202	-99.21	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
7203	-99.22	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
7204	-99.22	kd	CGS001-3586	IL10	Interleukins and interleukin receptors			
7205	-99.24	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
7206	-99.24	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
7207	-99.25	cc		X linked mental retardation group 1 LOF	-			
7208	-99.25	kd	CGS001-10451	VAV3	Rho guanine nucleotide exchange factors			
7209	-99.26	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
7210	-99.26	oe	ccsbBroad304_10758	CTBP2	-			
7211	-99.26	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
7212	-99.27	kd	CGS001-790	CAD	-			
7213	-99.28	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
7214	-99.28	kd	CGS001-55746	NUP133	-			
7215	-99.31	kd	CGS001-2037	EPB41L2	-			
7216	-99.32	oe	ccsbBroad304_07277	RTCD1	-			
7217	-99.32	oe	ccsbBroad304_03798	PHTF2	-			
7218	-99.32	oe	ccsbBroad304_13499	KSR2	RAF family			
7219	-99.32	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
7220	-99.32	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
7221	-99.33	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
7222	-99.34	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
7223	-99.34	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
7224	-99.34	kd	CGS001-5992	RFX4	-			
7225	-99.35	oe	ccsbBroad304_00874	INS	-			
7226	-99.35	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
7227	-99.36	kd	CGS001-8089	YEATS4	-			
7228	-99.37	oe	ccsbBroad304_02843	FTSJ1	-			
7229	-99.37	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
7230	-99.37	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
7231	-99.39	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
7232	-99.41	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
7233	-99.41	kd	CGS001-8905	AP1S2	-			
7234	-99.43	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
7235	-99.43	oe	ccsbBroad304_01166	PDK2	PDHK family			
7236	-99.43	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
7237	-99.43	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
7238	-99.43	kd	CGS001-23657	SLC7A11	Solute carriers			
7239	-99.43	kd	CGS001-382	ARF6	ADP-ribosylation factors			
7240	-99.43	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
7241	-99.45	cp	BRD-A56892734	esomeprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
7242	-99.45	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
7243	-99.47	oe	ccsbBroad304_06663	OAS1	-			
7244	-99.47	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
7245	-99.47	oe	ccsbBroad304_08217	SCCPDH	-			
7246	-99.47	oe	ccsbBroad304_02788	PRAME	-			
7247	-99.47	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
7248	-99.47	kd	CGS001-9945	GFPT2	-			
7249	-99.47	kd	CGS001-775	CACNA1C	Calcium channel subunits			
7250	-99.5	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
7251	-99.5	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
7252	-99.5	kd	CGS001-55256	ADI1	-			
7253	-99.52	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
7254	-99.52	oe	ccsbBroad304_01933	TEAD2	-			
7255	-99.52	kd	CGS001-23355	VPS8	-			
7256	-99.52	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
7257	-99.52	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
7258	-99.54	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
7259	-99.54	oe	ccsbBroad304_00620	GCDH	-			
7260	-99.54	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
7261	-99.54	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
7262	-99.54	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
7263	-99.55	kd	CGS001-64425	POLR1E	RNA polymerase subunits			
7264	-99.56	cc		PARP inhibitor	-			
7265	-99.56	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
7266	-99.57	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
7267	-99.61	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
7268	-99.61	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
7269	-99.62	kd	CGS001-388677	NOTCH2NL	-			
7270	-99.63	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
7271	-99.63	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
7272	-99.63	oe	ccsbBroad304_00492	EIF5A	-			
7273	-99.63	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
7274	-99.65	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
7275	-99.65	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7276	-99.65	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
7277	-99.65	kd	CGS001-93349	SP140L	Zinc fingers, PHD-type			
7278	-99.65	kd	CGS001-8945	BTRC	F-boxes / WD-40 domains			
7279	-99.67	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
7280	-99.67	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
7281	-99.67	kd	CGS001-84936	ZFYVE19	Zinc fingers, FYVE domain containing			
7282	-99.67	kd	CGS001-2580	GAK	Heat shock proteins / DNAJ (HSP40)			
7283	-99.67	kd	CGS001-847	CAT	-			
7284	-99.68	cc		PKA inhibitor	-			
7285	-99.69	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
7286	-99.69	cp	BRD-K81855038	roxatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
7287	-99.69	cp	BRD-K44353683	nateglinide	Insulin secretagogue		ABCC8, KCNJ11, CYP3A4, INS, KCNJ10, PPARG	Insulin secretagogue
7288	-99.69	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
7289	-99.69	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
7290	-99.69	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
7291	-99.69	kd	CGS001-1604	CD55	CD molecules			
7292	-99.71	kd	CGS001-24140	FTSJ1	-			
7293	-99.72	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
7294	-99.72	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
7295	-99.72	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
7296	-99.72	kd	CGS001-10482	NXF1	-			
7297	-99.72	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
7298	-99.73	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
7299	-99.74	oe	ccsbBroad304_00077	APEX1	-			
7300	-99.74	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
7301	-99.74	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
7302	-99.74	kd	CGS001-64921	CASD1	-			
7303	-99.76	oe	ccsbBroad304_02032	TSC22D1	-			
7304	-99.76	kd	CGS001-8805	TRIM24	TIF1 family			
7305	-99.76	kd	CGS001-55958	KLHL9	BTB/POZ domain containing			
7306	-99.76	kd	CGS001-2242	FES	Fer family			
7307	-99.76	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
7308	-99.78	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
7309	-99.78	oe	ccsbBroad304_07548	TSSC4	-			
7310	-99.78	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7311	-99.78	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
7312	-99.78	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
7313	-99.78	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
7314	-99.78	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
7315	-99.78	kd	CGS001-51701	NLK	nmo subfamily			
7316	-99.78	kd	CGS001-148103	ZNF599	Zinc fingers, C2H2-type			
7317	-99.78	kd	CGS001-10165	SLC25A13	Mitochondrial amino acid transporter subfamily			
7318	-99.78	kd	CGS001-2592	GALT	-			
7319	-99.78	kd	CGS001-966	CD59	CD molecules			
7320	-99.78	kd	CGS001-226	ALDOA	-			
7321	-99.8	oe	ccsbBroad304_02674	STK38	NDR family			
7322	-99.8	cp	BRD-A39172021	ampiroxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
7323	-99.8	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
7324	-99.8	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
7325	-99.8	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
7326	-99.8	kd	CGS001-57819	LSM2	-			
7327	-99.8	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
7328	-99.8	kd	CGS001-1345	COX6C	Mitochondrial respiratory chain complex			
7329	-99.8	kd	CGS001-930	CD19	CD molecules			
7330	-99.81	kd	CGS001-115727	RASGRP4	EF-hand domain containing			
7331	-99.82	cc		Thromboxane receptor antagonist	-			
7332	-99.82	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
7333	-99.82	oe	ccsbBroad304_02419	NDRG1	-			
7334	-99.82	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
7335	-99.82	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
7336	-99.82	kd	CGS001-4833	NME4	-			
7337	-99.82	kd	CGS001-2155	F7	Chymotrypsin			
7338	-99.82	kd	CGS001-1727	CYB5R3	-			
7339	-99.82	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
7340	-99.85	oe	ccsbBroad304_08480	PNPO	-			
7341	-99.85	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
7342	-99.85	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
7343	-99.85	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
7344	-99.85	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
7345	-99.85	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
7346	-99.85	kd	CGS001-6772	STAT1	SH2 domain containing			
7347	-99.85	kd	CGS001-9805	SCRN1	-			
7348	-99.85	kd	CGS001-57048	PLSCR3	-			
7349	-99.85	kd	CGS001-25861	DFNB31	-			
7350	-99.85	kd	CGS001-593	BCKDHA	-			
7351	-99.85	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
7352	-99.85	kd	CGS001-95	ACY1	-			
7353	-99.86	oe	ccsbBroad304_00223	CASP9	Caspases			
7354	-99.87	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
7355	-99.87	oe	ccsbBroad304_00398	CTSL2	-			
7356	-99.87	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
7357	-99.87	oe	ccsbBroad304_03565	ADI1	-			
7358	-99.87	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
7359	-99.87	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
7360	-99.87	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
7361	-99.87	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
7362	-99.87	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
7363	-99.87	kd	CGS001-5471	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
7364	-99.87	kd	CGS001-10606	PAICS	-			
7365	-99.87	kd	CGS001-79711	IPO4	Importins			
7366	-99.87	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7367	-99.89	oe	ccsbBroad304_14020	SH3BP5	-			
7368	-99.89	oe	ccsbBroad304_03618	OSGEP	-			
7369	-99.89	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
7370	-99.89	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
7371	-99.89	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
7372	-99.89	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
7373	-99.89	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
7374	-99.89	kd	CGS001-5993	RFX5	-			
7375	-99.89	kd	CGS001-56998	CTNNBIP1	Catenins			
7376	-99.89	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
7377	-99.9	oe	ccsbBroad304_01401	RIT1	-			
7378	-99.91	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
7379	-99.91	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
7380	-99.91	oe	ccsbBroad304_00116	ASS1	-			
7381	-99.91	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
7382	-99.91	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
7383	-99.91	cp	BRD-K49481516	galantamine	Acetylcholinesterase inhibitor		ACHE, BCHE, CHRNA1, CHRNA10, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNA9, CHRNB1, CHRNB2, CHRNB3, CHRNB4, CHRND, CHRNE, CHRNG	Acetylcholinesterase inhibitor
7384	-99.91	cp	BRD-K49668410	clarithromycin	Bacterial 50S ribosomal subunit inhibitor		CYP2C19, CYP3A4, CYP3A5, CYP3A7	Bacterial 50S ribosomal subunit inhibitor
7385	-99.91	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
7386	-99.91	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
7387	-99.91	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
7388	-99.91	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
7389	-99.91	kd	CGS001-319100	TAAR6	GPCR / Class A : Trace amine associated receptors			
7390	-99.91	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
7391	-99.91	kd	CGS001-6184	RPN1	-			
7392	-99.91	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
7393	-99.91	kd	CGS001-253430	IPMK	-			
7394	-99.91	kd	CGS001-94239	H2AFV	Histones / Replication-independent			
7395	-99.91	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
7396	-99.93	oe	ccsbBroad304_03308	YTHDF2	-			
7397	-99.93	oe	ccsbBroad304_07511	KIF14	Kinesins			
7398	-99.93	oe	ccsbBroad304_14291	GDPD5	-			
7399	-99.93	oe	ccsbBroad304_06094	DFFA	-			
7400	-99.93	cp	BRD-A84134924	pancuronium	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRNA1, CHRNA2	Acetylcholine receptor antagonist
7401	-99.93	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
7402	-99.93	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
7403	-99.93	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7404	-99.93	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
7405	-99.93	kd	CGS001-375449	MAST4	MAST family			
7406	-99.93	kd	CGS001-51776	ZAK	MLK subfamily			
7407	-99.93	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
7408	-99.93	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
7409	-99.93	kd	CGS001-55033	FKBP14	EF-hand domain containing			
7410	-99.93	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
7411	-99.96	oe	ccsbBroad304_03917	RBKS	-			
7412	-99.96	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
7413	-99.96	oe	ccsbBroad304_02759	DICER1	-			
7414	-99.96	oe	ccsbBroad304_00390	CTGF	-			
7415	-99.96	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
7416	-99.96	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
7417	-99.96	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
7418	-99.96	oe	ccsbBroad304_06888	RPN1	-			
7419	-99.96	oe	ccsbBroad304_06855	RDX	-			
7420	-99.96	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
7421	-99.96	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
7422	-99.96	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
7423	-99.96	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
7424	-99.96	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
7425	-99.96	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
7426	-99.96	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
7427	-99.96	oe	ccsbBroad304_08952	E2F8	-			
7428	-99.96	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
7429	-99.96	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
7430	-99.96	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
7431	-99.96	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
7432	-99.96	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
7433	-99.96	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
7434	-99.96	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
7435	-99.96	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
7436	-99.96	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
7437	-99.96	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
7438	-99.96	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
7439	-99.96	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
7440	-99.96	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
7441	-99.96	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
7442	-99.96	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
7443	-99.96	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
7444	-99.96	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
7445	-99.96	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
7446	-99.96	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
7447	-99.96	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
7448	-99.96	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
7449	-99.96	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
7450	-99.96	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7451	-99.96	kd	CGS001-2834	PRLHR	GPCR / Class A : RF amide peptide receptors			
7452	-99.96	kd	CGS001-5583	PRKCH	Eta subfamily			
7453	-99.96	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
7454	-99.96	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
7455	-99.96	kd	CGS001-8566	PDXK	-			
7456	-99.96	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
7457	-99.96	kd	CGS001-4709	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
7458	-99.96	kd	CGS001-22944	KIN	-			
7459	-99.96	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
7460	-99.96	kd	CGS001-25842	ASF1A	-			
7461	-99.96	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
7462	-99.96	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
7463	-99.98	cc		Purinergic receptors P2Y GOF	-			
7464	-99.98	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
7465	-99.98	kd	CGS001-5460	POU5F1	Homeoboxes / POU class			
7466	-99.98	kd	CGS001-9156	EXO1	-			
7467	-99.98	kd	CGS001-2000	ELF4	ETS Transcription Factors			
7468	-100	cc		PPAR receptor agonist	-			
7469	-100	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
7470	-100	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
7471	-100	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
7472	-100	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
7473	-100	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
7474	-100	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
7475	-100	kd	CGS001-7625	ZNF74	Zinc fingers, C2H2-type			
7476	-100	kd	CGS001-54659	UGT1A3	UDP glucuronosyltransferases			
7477	-100	kd	CGS001-337867	UBAC2	-			
7478	-100	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
7479	-100	kd	CGS001-6429	SRSF4	RNA binding motif (RRM) containing			
7480	-100	kd	CGS001-6272	SORT1	-			
7481	-100	kd	CGS001-6493	SIM2	Basic helix-loop-helix proteins			
7482	-100	kd	CGS001-23678	SGK3	SGK family			
7483	-100	kd	CGS001-51097	SCCPDH	-			
7484	-100	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
7485	-100	kd	CGS001-25824	PRDX5	-			
7486	-100	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
7487	-100	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
7488	-100	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
7489	-100	kd	CGS001-10161	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7490	-100	kd	CGS001-3934	LCN2	Lipocalins			
7491	-100	kd	CGS001-8942	KYNU	-			
7492	-100	kd	CGS001-10657	KHDRBS1	-			
7493	-100	kd	CGS001-2621	GAS6	-			
7494	-100	kd	CGS001-80314	EPC1	-			
7495	-100	kd	CGS001-60528	ELAC2	-			
7496	-100	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
7497	-100	kd	CGS001-1105	CHD1	-			
7498	-100	kd	CGS001-1029	CDKN2A	-			
7499	-100	kd	CGS001-833	CARS	Aminoacyl tRNA synthetases / Class I			
7500	-100	kd	CGS001-330	BIRC3	Inhibitors of apoptosis (IAP) protein family			
7501	-100	kd	CGS001-604	BCL6	BTB/POZ domain containing			
7502	-100	kd	CGS001-27113	BBC3	-			
7503	-100	kd	CGS001-302	ANXA2	Annexins			
7504	-100	kd	CGS001-135	ADORA2A	GPCR / Class A : Adenosine receptors			
7505	-100	kd	CGS001-2181	ACSL3	Acyl-CoA synthetase family			
7506	-100	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
