Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	99.95	kd	CGS001-8428	STK24	YSK subfamily			
2	99.95	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
3	99.95	kd	CGS001-7027	TFDP1	-			
4	99.95	kd	CGS001-10019	SH2B3	Pleckstrin homology (PH) domain containing			
5	99.95	kd	CGS001-5734	PTGER4	GPCR / Class A : Prostanoid receptors			
6	99.95	kd	CGS001-57804	POLD4	DNA polymerases			
7	99.95	kd	CGS001-4942	OAT	-			
8	99.95	kd	CGS001-29982	NRBF2	-			
9	99.95	kd	CGS001-58508	MLL3	-			
10	99.95	kd	CGS001-3035	HARS	Aminoacyl tRNA synthetases / Class II			
11	99.95	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
12	99.95	kd	CGS001-113878	DTX2	RING-type (C3HC4) zinc fingers			
13	99.95	kd	CGS001-1387	CREBBP	Chromatin-modifying enzymes / K-acetyltransferases			
14	99.95	kd	CGS001-6347	CCL2	Chemokine ligands			
15	99.95	kd	CGS001-837	CASP4	Caspases			
16	99.95	kd	CGS001-662	BNIP1	-			
17	99.93	cp	BRD-K33483813	actarit	Interleukin receptor agonist			Interleukin receptor agonist
18	99.93	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
19	99.93	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
20	99.93	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
21	99.93	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
22	99.92	kd	CGS001-23012	STK38L	NDR family			
23	99.92	kd	CGS001-25925	ZNF521	Zinc fingers, C2H2-type			
24	99.92	kd	CGS001-333929	SNAI3	Snail homologs			
25	99.92	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
26	99.92	kd	CGS001-80714	PBX4	Homeoboxes / TALE class			
27	99.92	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
28	99.92	kd	CGS001-3930	LBR	Tudor domain containing			
29	99.92	kd	CGS001-3682	ITGAE	Integrins			
30	99.92	kd	CGS001-3162	HMOX1	Haem oxygenase			
31	99.91	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
32	99.91	oe	ccsbBroad304_01699	TPD52L2	-			
33	99.91	oe	ccsbBroad304_06291	GNAI1	-			
34	99.91	oe	ccsbBroad304_06278	GK	Glycerol kinases			
35	99.91	oe	ccsbBroad304_00268	CD81	CD molecules			
36	99.91	oe	ccsbBroad304_04675	ATG4A	-			
37	99.91	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
38	99.91	oe	ccsbBroad304_01651	TCF7L2	-			
39	99.91	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
40	99.91	oe	ccsbBroad304_02845	PRPF6	-			
41	99.91	oe	ccsbBroad304_03604	ENOSF1	-			
42	99.91	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
43	99.91	oe	ccsbBroad304_05547	TMEM110	-			
44	99.91	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
45	99.91	oe	ccsbBroad304_07688	FAM114A2	-			
46	99.91	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
47	99.91	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
48	99.91	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
49	99.91	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
50	99.89	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
51	99.89	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
52	99.89	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
53	99.89	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
54	99.89	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
55	99.89	kd	CGS001-9833	MELK	MELK subfamily			
56	99.89	kd	CGS001-51451	LCMT1	-			
57	99.89	kd	CGS001-4254	KITLG	-			
58	99.89	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
59	99.89	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
60	99.89	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
61	99.87	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
62	99.87	kd	CGS001-5564	PRKAB1	AMPK subfamily			
63	99.87	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
64	99.87	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
65	99.86	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
66	99.86	oe	ccsbBroad304_01257	PPOX	-			
67	99.86	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
68	99.86	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
69	99.86	oe	ccsbBroad304_06462	ITGAE	Integrins			
70	99.86	oe	ccsbBroad304_00036	AFP	-			
71	99.86	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
72	99.86	oe	ccsbBroad304_00964	SMAD7	SMADs			
73	99.86	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
74	99.86	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
75	99.84	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
76	99.84	kd	CGS001-57761	TRIB3	Trbl family			
77	99.84	kd	CGS001-10608	MXD4	Basic helix-loop-helix proteins			
78	99.84	kd	CGS001-26205	GMEB2	-			
79	99.82	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
80	99.82	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
81	99.82	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
82	99.81	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
83	99.81	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
84	99.81	oe	ccsbBroad304_01211	PKM2	-			
85	99.81	oe	ccsbBroad304_01661	TFCP2	-			
86	99.81	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
87	99.79	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
88	99.79	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
89	99.79	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
90	99.79	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
91	99.79	kd	CGS001-6285	S100B	EF-hand domain containing			
92	99.79	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
93	99.79	kd	CGS001-604	BCL6	BTB/POZ domain containing			
94	99.77	oe	ccsbBroad304_04457	TOX2	-			
95	99.77	oe	ccsbBroad304_02446	TADA3	-			
96	99.77	oe	ccsbBroad304_02270	FAM20B	-			
97	99.77	oe	ccsbBroad304_00060	AMBP	Lipocalins			
98	99.77	oe	ccsbBroad304_01271	PPT1	-			
99	99.76	kd	CGS001-7756	ZNF207	Zinc fingers, C2H2-type			
100	99.76	kd	CGS001-51569	UFM1	-			
101	99.76	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
102	99.75	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
103	99.75	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
104	99.75	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
105	99.75	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
106	99.74	kd	CGS001-10477	UBE2E3	Ubiquitin-conjugating enzymes E2			
107	99.74	kd	CGS001-6812	STXBP1	-			
108	99.74	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
109	99.74	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
110	99.74	kd	CGS001-9791	PTDSS1	-			
111	99.72	oe	ccsbBroad304_02402	TMEM5	-			
112	99.72	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
113	99.72	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
114	99.72	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
115	99.72	oe	ccsbBroad304_04891	TMEM174	-			
116	99.71	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
117	99.71	kd	CGS001-224	ALDH3A2	Aldehyde dehydrogenases			
118	99.71	kd	CGS001-25898	RCHY1	RING-type (C3HC4) zinc fingers			
119	99.71	kd	CGS001-9943	OXSR1	FRAY subfamily			
120	99.71	kd	CGS001-22889	KIAA0907	-			
121	99.71	kd	CGS001-79135	APOO	Apolipoproteins			
122	99.68	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
123	99.68	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
124	99.68	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
125	99.67	kd	CGS001-5641	LGMN	Legumain			
126	99.66	kd	CGS001-6817	SULT1A1	Sulfotransferases, cytosolic			
127	99.66	kd	CGS001-4094	MAF	-			
128	99.66	kd	CGS001-3800	KIF5C	Kinesins			
129	99.66	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
130	99.65	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
131	99.65	cp	BRD-K84566043	fenpiverinium	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
132	99.65	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
133	99.65	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
134	99.65	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
135	99.63	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
136	99.63	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
137	99.63	kd	CGS001-51547	SIRT7	Histone deacetylases (HDACs)			
138	99.63	kd	CGS001-3912	LAMB1	Laminins			
139	99.63	kd	CGS001-29940	DSE	-			
140	99.63	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
141	99.63	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
142	99.63	oe	ccsbBroad304_01845	RDBP	-			
143	99.63	oe	ccsbBroad304_06174	ERCC1	-			
144	99.61	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
145	99.61	kd	CGS001-79258	MMEL1	-			
146	99.61	oe	ccsbBroad304_05758	ACADSB	-			
147	99.58	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
148	99.58	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
149	99.58	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
150	99.58	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
151	99.58	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
152	99.58	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
153	99.58	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
154	99.58	kd	CGS001-11073	TOPBP1	-			
155	99.58	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
156	99.58	kd	CGS001-6198	RPS6KB1	p70 subfamily			
157	99.58	kd	CGS001-4352	MPL	Prolactin receptor family			
158	99.58	kd	CGS001-3297	HSF1	-			
159	99.58	kd	CGS001-1209	CLPTM1	-			
160	99.58	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
161	99.58	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
162	99.57	oe	ccsbBroad304_06718	PFN2	-			
163	99.55	kd	CGS001-11113	CIT	Other DMPK family kinases			
164	99.55	kd	CGS001-306	ANXA3	Annexins			
165	99.54	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
166	99.54	oe	ccsbBroad304_00164	BLMH	-			
167	99.54	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
168	99.54	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
169	99.54	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
170	99.54	oe	ccsbBroad304_01247	POU2AF1	-			
171	99.53	kd	CGS001-3976	LIF	-			
172	99.53	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
173	99.52	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
174	99.51	kd	CGS001-10451	VAV3	Rho guanine nucleotide exchange factors			
175	99.5	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
176	99.5	kd	CGS001-79071	ELOVL6	-			
177	99.49	cc		Sodium channel blocker	-			
178	99.49	oe	ccsbBroad304_02052	KYNU	-			
179	99.49	oe	ccsbBroad304_05756	ACAA1	-			
180	99.48	kd	CGS001-26292	MYCBP	-			
181	99.47	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
182	99.47	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
183	99.47	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
184	99.47	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
185	99.47	kd	CGS001-8777	MPDZ	-			
186	99.47	kd	CGS001-84811	BUD13	-			
187	99.45	kd	CGS001-3717	JAK2	Janus kinase (JakA) family			
188	99.44	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
189	99.44	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
190	99.44	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
191	99.44	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
192	99.43	kd	CGS001-83439	TCF7L1	-			
193	99.42	kd	CGS001-10007	GNPDA1	-			
194	99.42	kd	CGS001-2161	F12	Chymotrypsin			
195	99.4	oe	ccsbBroad304_06645	NQO2	-			
196	99.4	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
197	99.4	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
198	99.4	kd	CGS001-11319	ECD	-			
199	99.39	kd	CGS001-5445	PON2	Paraoxonases			
200	99.39	kd	CGS001-85315	PAQR8	-			
201	99.39	kd	CGS001-3169	FOXA1	Forkhead boxes			
202	99.39	kd	CGS001-10973	ASCC3	-			
203	99.37	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
204	99.37	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
205	99.37	kd	CGS001-2243	FGA	Endogenous ligands			
206	99.37	kd	CGS001-1810	DR1	-			
207	99.36	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
208	99.35	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
209	99.35	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
210	99.35	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
211	99.34	cp	BRD-A23637604	oxymetholone	Androgen receptor agonist		AR	Androgen receptor agonist
212	99.34	kd	CGS001-10613	ERLIN1	-			
213	99.33	cp	BRD-A01787639	naftopidil	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
214	99.33	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
215	99.31	oe	ccsbBroad304_03308	YTHDF2	-			
216	99.31	kd	CGS001-285267	ZNF619	Zinc fingers, C2H2-type			
217	99.31	kd	CGS001-55226	NAT10	-			
218	99.31	oe	ccsbBroad304_07598	PEMT	-			
219	99.31	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
220	99.3	kd	CGS001-4088	SMAD3	SMADs			
221	99.29	kd	CGS001-54805	CNNM2	-			
222	99.29	kd	CGS001-118738	ZNF488	Zinc fingers, C2H2-type			
223	99.29	kd	CGS001-10161	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
224	99.28	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
225	99.27	kd	CGS001-55723	ASF1B	-			
226	99.26	kd	CGS001-55311	ZNF444	Zinc fingers, C2H2-type			
227	99.26	kd	CGS001-11031	RAB31	RAB, member RAS oncogene			
228	99.26	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
229	99.26	oe	ccsbBroad304_00650	GNA11	-			
230	99.26	oe	ccsbBroad304_01143	PAFAH1B3	-			
231	99.26	oe	ccsbBroad304_02217	FEZ1	-			
232	99.26	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
233	99.24	kd	CGS001-8767	RIPK2	Receptor interacting protein kinase (RIPK) family			
234	99.24	kd	CGS001-164091	PAQR7	-			
235	99.24	kd	CGS001-717	C2	Complement system			
236	99.21	kd	CGS001-1659	DHX8	DEAH-boxes			
237	99.21	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
238	99.2	oe	ccsbBroad304_02110	VAPB	-			
239	99.19	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
240	99.19	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
241	99.19	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
242	99.19	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
243	99.19	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
244	99.18	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
245	99.18	kd	CGS001-199704	ZNF585A	Zinc fingers, C2H2-type			
246	99.18	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
247	99.17	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
248	99.17	oe	ccsbBroad304_06294	GNAZ	-			
249	99.17	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
250	99.17	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
251	99.16	cc		Cyclooxygenase inhibitor	-			
252	99.16	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
253	99.15	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
254	99.15	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
255	99.14	kd	CGS001-55033	FKBP14	EF-hand domain containing			
256	99.13	kd	CGS001-2057	EPOR	Prolactin receptor family			
257	99.13	kd	CGS001-116519	APOA5	Apolipoproteins			
258	99.12	oe	ccsbBroad304_08104	MED4	-			
259	99.12	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
260	99.12	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
261	99.11	kd	CGS001-476	ATP1A1	ATPases / P-type			
262	99.11	kd	CGS001-64219	PJA1	RING-type (C3HC4) zinc fingers			
263	99.11	kd	CGS001-10401	PIAS3	Zinc fingers, MIZ-type			
264	99.11	kd	CGS001-3956	LGALS1	Endogenous ligands			
265	99.1	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
266	99.08	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
267	99.08	kd	CGS001-51015	ISOC1	-			
268	99.08	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
269	99.08	kd	CGS001-10257	ABCC4	ATP binding cassette transporters / subfamily C			
270	99.07	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
271	99.06	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
272	99.06	oe	ccsbBroad304_01152	PCNA	-			
273	99.05	cc		CCK receptor antagonist	-			
274	99.05	cp	BRD-K37516142	idebenone	Calcium channel modulator			Calcium channel modulator
275	99.05	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
276	99.05	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
277	99.03	cp	BRD-K22009844	phenprobamate	Muscle relaxant			Muscle relaxant
278	99.03	kd	CGS001-11124	FAF1	UBX domain containing			
279	99.03	kd	CGS001-3995	FADS3	Fatty acid desaturases			
280	99.02	kd	CGS001-2159	F10	Chymotrypsin			
281	99.01	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
282	99.01	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
283	98.99	kd	CGS001-1910	EDNRB	Endothelin receptors			
284	98.98	oe	ccsbBroad304_02443	HAX1	-			
285	98.98	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
286	98.98	oe	ccsbBroad304_01923	UXT	-			
287	98.98	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
288	98.97	kd	CGS001-10412	NSA2	-			
289	98.97	kd	CGS001-9231	DLG5	-			
290	98.96	oe	ccsbBroad304_00509	EPHX1	-			
291	98.95	kd	CGS001-23240	KIAA0922	-			
292	98.95	kd	CGS001-8714	ABCC3	ATP binding cassette transporters / subfamily C			
293	98.94	oe	ccsbBroad304_00212	CAMLG	-			
294	98.94	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
295	98.94	oe	ccsbBroad304_05907	BUB1B	Bub family			
296	98.93	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
297	98.93	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
298	98.92	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
299	98.92	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
300	98.91	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
301	98.91	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
302	98.91	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
303	98.9	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
304	98.89	kd	CGS001-539	ATP5O	ATPases / F-type			
305	98.88	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
306	98.87	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
307	98.87	kd	CGS001-5987	TRIM27	-			
308	98.86	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
309	98.84	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
310	98.84	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
311	98.84	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
312	98.83	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
313	98.82	kd	CGS001-3576	IL8	-			
314	98.82	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
315	98.8	oe	ccsbBroad304_03357	RASD1	-			
316	98.8	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
317	98.8	oe	ccsbBroad304_08167	DNTTIP2	-			
318	98.79	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
319	98.78	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
320	98.77	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
321	98.77	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
322	98.75	kd	CGS001-6720	SREBF1	Basic helix-loop-helix proteins			
323	98.75	kd	CGS001-24140	FTSJ1	-			
324	98.74	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
325	98.74	kd	CGS001-3428	IFI16	-			
326	98.74	kd	CGS001-2580	GAK	Heat shock proteins / DNAJ (HSP40)			
327	98.74	kd	CGS001-2308	FOXO1	Forkhead boxes			
328	98.74	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
329	98.73	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
330	98.71	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
331	98.71	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
332	98.71	kd	CGS001-54107	POLE3	DNA polymerases			
333	98.7	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
334	98.7	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
335	98.7	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
336	98.68	kd	CGS001-6648	SOD2	-			
337	98.68	kd	CGS001-7108	TM7SF2	-			
338	98.68	kd	CGS001-10928	RALBP1	-			
339	98.68	kd	CGS001-1112	FOXN3	Forkhead boxes			
340	98.68	kd	CGS001-509	ATP5C1	ATPases / F-type			
341	98.67	kd	CGS001-9702	CEP57	-			
342	98.66	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
343	98.66	kd	CGS001-5428	POLG	DNA polymerases			
344	98.66	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
345	98.64	kd	CGS001-9360	PPIG	-			
346	98.63	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
347	98.63	kd	CGS001-79643	CHMP6	Charged multivesicular body proteins			
348	98.63	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
349	98.62	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
350	98.62	kd	CGS001-4946	OAZ1	-			
351	98.61	kd	CGS001-29946	SERTAD3	-			
352	98.59	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
353	98.59	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
354	98.59	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
355	98.58	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
356	98.58	kd	CGS001-5550	PREP	Prolyl oligopeptidase			
357	98.58	kd	CGS001-23142	DCUN1D4	-			
358	98.57	kd	CGS001-7172	TPMT	-			
359	98.57	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
360	98.56	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
361	98.56	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
362	98.56	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
363	98.56	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
364	98.56	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
365	98.56	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
366	98.54	kd	CGS001-1676	DFFA	-			
367	98.53	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
368	98.52	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
369	98.5	kd	CGS001-9898	UBAP2L	-			
370	98.5	kd	CGS001-7004	TEAD4	-			
371	98.47	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
372	98.45	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
373	98.45	kd	CGS001-25885	POLR1A	RNA polymerase subunits			
374	98.45	kd	CGS001-3691	ITGB4	Integrins			
375	98.44	kd	CGS001-114112	TXNRD3	-			
376	98.42	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
377	98.4	cc		HIV protease inhibitor	-			
378	98.4	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
379	98.4	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
380	98.39	kd	CGS001-23252	OTUD3	OTU domain containing			
381	98.38	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
382	98.37	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
383	98.37	kd	CGS001-1978	EIF4EBP1	-			
384	98.37	kd	CGS001-63874	ABHD4	Abhydrolase domain containing			
385	98.36	kd	CGS001-3397	ID1	Basic helix-loop-helix proteins			
386	98.34	cp	BRD-K29113274	ketoconazole	Sterol demethylase inhibitor		AR, CYP19A1, CYP21A2, CYP2C19, CYP3A5, CYP3A7, KCNA10	Sterol demethylase inhibitor
387	98.34	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
388	98.34	kd	CGS001-84108	PCGF6	Polycomb group ring fingers			
389	98.34	kd	CGS001-11137	PWP1	WD repeat domain containing			
390	98.34	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
391	98.33	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
392	98.33	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
393	98.33	oe	ccsbBroad304_01675	TK1	-			
394	98.31	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
395	98.31	oe	ccsbBroad304_02243	DLGAP5	-			
396	98.29	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
397	98.29	kd	CGS001-29937	NENF	-			
398	98.28	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
399	98.27	oe	ccsbBroad304_00617	GBA	-			
400	98.26	kd	CGS001-5320	PLA2G2A	Hydrolases			
401	98.26	kd	CGS001-4548	MTR	-			
402	98.25	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
403	98.25	kd	CGS001-26064	RAI14	Ankyrin repeat domain containing			
404	98.25	kd	CGS001-5450	POU2AF1	-			
405	98.24	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
406	98.24	kd	CGS001-1051	CEBPB	basic leucine zipper proteins			
407	98.24	oe	ccsbBroad304_02357	SSX3	-			
408	98.22	kd	CGS001-54442	KCTD5	-			
409	98.21	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
410	98.21	kd	CGS001-84539	MCHR2	GPCR / Class A : MCH receptors			
411	98.21	kd	CGS001-5594	MAPK1	MAPK:ERK subfamily			
412	98.2	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
413	98.2	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
414	98.2	kd	CGS001-2280	FKBP1A	Cis-trans-isomerases			
415	98.2	kd	CGS001-468	ATF4	basic leucine zipper proteins			
416	98.18	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
417	98.18	kd	CGS001-2731	GLDC	-			
418	98.16	kd	CGS001-25942	SIN3A	-			
419	98.16	kd	CGS001-79143	MBOAT7	-			
420	98.15	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
421	98.15	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
422	98.15	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
423	98.15	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
424	98.13	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
425	98.13	kd	CGS001-7424	VEGFC	-			
426	98.13	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
427	98.12	kd	CGS001-124583	CANT1	-			
428	98.11	kd	CGS001-328	APEX1	-			
429	98.1	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
430	98.09	oe	ccsbBroad304_00962	SMAD4	SMADs			
431	98.08	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
432	98.08	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
433	98.07	oe	ccsbBroad304_02741	PDS5A	-			
434	98.06	oe	ccsbBroad304_02133	CD83	CD molecules			
435	98.06	cp	BRD-A49172652	lansoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4, CYP3A5	ATPase inhibitor
436	98.06	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
437	98.06	oe	ccsbBroad304_01618	STXBP1	-			
438	98.05	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
439	98.03	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
440	98.03	kd	CGS001-6397	SEC14L1	-			
441	98.03	kd	CGS001-26523	EIF2C1	-			
442	98.03	kd	CGS001-83440	ADPGK	-			
443	98.01	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
444	98.01	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
445	98	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
446	98	kd	CGS001-55937	APOM	Apolipoproteins			
447	97.99	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
448	97.95	kd	CGS001-9788	MTSS1	-			
449	97.95	kd	CGS001-4363	ABCC1	ATP binding cassette transporters / subfamily C			
450	97.9	kd	CGS001-56848	SPHK2	Sphingosine kinase			
451	97.89	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
452	97.89	kd	CGS001-91137	SLC25A46	Miscellaneous SLC25 mitochondrial transporters			
453	97.88	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
454	97.88	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
455	97.87	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
456	97.87	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
457	97.87	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
458	97.87	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
459	97.86	kd	CGS001-159	ADSS	-			
460	97.85	cc		Phospholipases LOF	-			
461	97.85	kd	CGS001-8204	NRIP1	-			
462	97.85	kd	CGS001-624	BDKRB2	Bradykinin receptors			
463	97.85	kd	CGS001-55054	ATG16L1	WD repeat domain containing			
464	97.84	kd	CGS001-5328	PLAU	Chymotrypsin			
465	97.82	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
466	97.81	oe	ccsbBroad304_00811	ICAM1	CD molecules			
467	97.8	oe	ccsbBroad304_02058	PLOD3	-			
468	97.79	cc		Integrin subunits beta LOF	-			
469	97.79	kd	CGS001-8859	STK19	G11 family			
470	97.79	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
471	97.79	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
472	97.78	oe	ccsbBroad304_02287	GNPDA1	-			
473	97.78	kd	CGS001-9217	VAPB	-			
474	97.77	kd	CGS001-5899	RALB	-			
475	97.75	kd	CGS001-57192	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
476	97.74	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
477	97.74	kd	CGS001-122809	SOCS4	SH2 domain containing			
478	97.74	kd	CGS001-2690	GHR	Prolactin receptor family			
479	97.73	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
480	97.72	kd	CGS001-3298	HSF2	-			
481	97.72	kd	CGS001-3205	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
482	97.71	cc		S100 calcium binding proteins LOF	-			
483	97.71	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
484	97.71	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
485	97.71	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
486	97.7	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
487	97.69	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
488	97.69	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
489	97.68	kd	CGS001-50865	HEBP1	Endogenous ligands			
490	97.67	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
491	97.66	kd	CGS001-10018	BCL2L11	-			
492	97.66	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
493	97.65	kd	CGS001-10308	ZNF267	Zinc fingers, C2H2-type			
494	97.64	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
495	97.64	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
496	97.64	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
497	97.63	kd	CGS001-2264	FGFR4	Type V RTKs: FGF (fibroblast growth factor) receptor family			
498	97.62	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
499	97.62	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
500	97.62	kd	CGS001-1390	CREM	basic leucine zipper proteins			
501	97.61	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
502	97.6	cc		Serotonin receptor agonist	-			
503	97.6	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
504	97.6	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
505	97.58	kd	CGS001-6778	STAT6	SH2 domain containing			
506	97.57	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
507	97.56	kd	CGS001-4856	NOV	-			
508	97.55	oe	ccsbBroad304_10212	GRHL3	-			
509	97.53	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
510	97.52	kd	CGS001-55509	BATF3	basic leucine zipper proteins			
511	97.51	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
512	97.5	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
513	97.5	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
514	97.5	kd	CGS001-222	ALDH3B2	Aldehyde dehydrogenases			
515	97.5	kd	CGS001-185	AGTR1	Angiotensin receptors			
516	97.49	kd	CGS001-323	APBB2	-			
517	97.48	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
518	97.47	cp	BRD-K46435977	valaciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
519	97.46	oe	ccsbBroad304_06264	GBP2	-			
520	97.45	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
521	97.45	oe	ccsbBroad304_01102	NMT1	-			
522	97.44	kd	CGS001-10474	TADA3	-			
523	97.43	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
524	97.43	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
525	97.43	cp	BRD-K50938287	sumatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1A, HTR1F, HTR1E, HTR5A, HTR6, HTR7	Serotonin receptor agonist
526	97.42	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
527	97.42	kd	CGS001-162655	ZNF519	Zinc fingers, C2H2-type			
528	97.41	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
529	97.39	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
530	97.39	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
531	97.38	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
532	97.38	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
533	97.37	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
534	97.35	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
535	97.35	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
536	97.35	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
537	97.34	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
538	97.31	oe	ccsbBroad304_01576	SOAT1	-			
539	97.3	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
540	97.29	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
541	97.26	oe	ccsbBroad304_01205	PIN1	-			
542	97.25	kd	CGS001-4072	EPCAM	CD molecules			
543	97.24	kd	CGS001-56834	GPR137	GPCR / Unclassified : 7TM orphan receptors			
544	97.24	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
545	97.23	kd	CGS001-54901	CDKAL1	-			
546	97.18	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
547	97.18	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
548	97.17	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
549	97.16	kd	CGS001-84759	PCGF1	Polycomb group ring fingers			
550	97.15	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
551	97.15	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
552	97.15	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
553	97.15	kd	CGS001-149428	BNIPL	-			
554	97.14	kd	CGS001-445	ASS1	-			
555	97.13	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
556	97.13	kd	CGS001-5037	PEBP1	-			
557	97.13	kd	CGS001-4773	NFATC2	Nuclear factor of activated T-cells			
558	97.12	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
559	97.08	oe	ccsbBroad304_03934	LEPRE1	-			
560	97.08	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
561	97.08	kd	CGS001-23030	KDM4B	Histone demethylases			
562	97.06	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
563	97.04	cp	BRD-K57930253	nitrazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, SCN1A	Benzodiazepine receptor agonist
564	97.04	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
565	97.03	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
566	97.03	kd	CGS001-65057	ACD	-			
567	97.02	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
568	97.02	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
569	97.01	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
570	97	kd	CGS001-57787	MARK4	MARK subfamily			
571	97	kd	CGS001-2295	FOXF2	Forkhead boxes			
572	96.98	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
573	96.97	kd	CGS001-5576	PRKAR2A	Protein kinase A			
574	96.96	cp	BRD-A56892734	esomeprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
575	96.96	kd	CGS001-650	BMP2	Bone morphogenetic proteins			
576	96.95	kd	CGS001-2077	ERF	ETS Transcription Factors			
577	96.94	kd	CGS001-10423	CDIPT	-			
578	96.94	kd	CGS001-23	ABCF1	ATP binding cassette transporters / subfamily F			
579	96.94	kd	CGS001-89845	ABCC10	ATP binding cassette transporters / subfamily C			
580	96.94	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
581	96.94	oe	ccsbBroad304_00424	DBI	-			
582	96.92	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
583	96.9	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
584	96.88	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
585	96.86	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
586	96.85	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
587	96.83	kd	CGS001-10434	LYPLA1	-			
588	96.83	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
589	96.81	cc		Wnt family LOF	-			
590	96.81	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
591	96.79	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
592	96.79	kd	CGS001-546	ATRX	-			
593	96.78	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
594	96.76	oe	ccsbBroad304_06711	PFAS	-			
595	96.76	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
596	96.76	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
597	96.74	kd	CGS001-6434	TRA2B	RNA binding motif (RRM) containing			
598	96.74	kd	CGS001-23067	SETD1B	Histone methyltransferases (HMTs)			
599	96.73	oe	ccsbBroad304_07920	NUP62	-			
600	96.72	oe	ccsbBroad304_03405	CHRAC1	-			
601	96.72	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
602	96.7	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
603	96.69	kd	CGS001-6821	SUOX	-			
604	96.68	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
605	96.68	kd	CGS001-5571	PRKAG1	AMPK subfamily			
606	96.65	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
607	96.64	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
608	96.62	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
609	96.6	kd	CGS001-5335	PLCG1	Phosphoinositide-specific phospholipase C			
610	96.6	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
611	96.59	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
612	96.57	oe	ccsbBroad304_00836	IGF2	-			
613	96.55	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
614	96.55	kd	CGS001-51588	PIAS4	Zinc fingers, MIZ-type			
615	96.55	kd	CGS001-1356	CP	-			
616	96.55	kd	CGS001-975	CD81	CD molecules			
617	96.54	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
618	96.52	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
619	96.52	oe	ccsbBroad304_13952	SHMT2	-			
620	96.5	kd	CGS001-21	ABCA3	ATP binding cassette transporters / subfamily A			
621	96.5	oe	ccsbBroad304_07569	TRIB1	Trbl family			
622	96.49	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
623	96.47	kd	CGS001-835	CASP2	Caspases			
624	96.47	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
625	96.45	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
626	96.44	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
627	96.41	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
628	96.41	kd	CGS001-7423	VEGFB	-			
629	96.41	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
630	96.38	kd	CGS001-4016	LOXL1	-			
631	96.36	kd	CGS001-8985	PLOD3	-			
632	96.35	kd	CGS001-9128	PRPF4	WD repeat domain containing			
633	96.35	kd	CGS001-27336	HTATSF1	RNA binding motif (RRM) containing			
634	96.32	oe	ccsbBroad304_01013	MIF	-			
635	96.31	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
636	96.3	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
637	96.3	oe	ccsbBroad304_08481	CEP55	-			
638	96.29	kd	CGS001-9961	MVP	-			
639	96.28	cc		MEK inhibitor	-			
640	96.27	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
641	96.26	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
642	96.26	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
643	96.26	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
644	96.25	oe	ccsbBroad304_06237	GAA	Glycosidases			
645	96.24	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
646	96.23	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
647	96.22	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
648	96.22	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
649	96.22	kd	CGS001-3586	IL10	Interleukins and interleukin receptors			
650	96.19	oe	ccsbBroad304_06013	CLPTM1	-			
651	96.19	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
652	96.18	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
653	96.14	kd	CGS001-4779	NFE2L1	basic leucine zipper proteins			
654	96.12	cp	BRD-K81916719	triclabendazole	Microtubule inhibitor		DNMT1	Microtubule inhibitor
655	96.12	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
656	96.11	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
657	96.11	oe	ccsbBroad304_02047	AP1S2	-			
658	96.07	kd	CGS001-2976	GTF3C2	General transcription factors			
659	96.06	oe	ccsbBroad304_00221	CASP3	Caspases			
660	96.06	kd	CGS001-51719	CAB39	-			
661	96.05	kd	CGS001-6883	TAF12	-			
662	96.05	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
663	96.04	kd	CGS001-3431	SP110	Non-enzymatic BRD containing proteins			
664	96.02	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
665	96.01	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
666	96.01	kd	CGS001-1984	EIF5A	-			
667	96.01	kd	CGS001-10289	EIF1B	-			
668	96	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
669	95.99	kd	CGS001-1407	CRY1	-			
670	95.96	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
671	95.95	kd	CGS001-7371	UCK2	-			
672	95.94	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
673	95.94	kd	CGS001-116832	RPL39L	L ribosomal proteins			
674	95.94	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
675	95.92	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
676	95.91	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
677	95.91	kd	CGS001-5054	SERPINE1	Serine (or cysteine) peptidase inhibitors			
678	95.89	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
679	95.88	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
680	95.88	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
681	95.87	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
682	95.87	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
683	95.84	kd	CGS001-2806	GOT2	-			
684	95.82	kd	CGS001-4795	NFKBIL1	-			
685	95.81	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
686	95.81	kd	CGS001-3417	IDH1	-			
687	95.79	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
688	95.77	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
689	95.76	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
690	95.74	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
691	95.74	kd	CGS001-6658	SOX3	SRY (sex determining region Y)-boxes			
692	95.72	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
693	95.69	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
694	95.68	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
695	95.68	kd	CGS001-285676	ZNF454	Zinc fingers, C2H2-type			
696	95.63	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
697	95.6	cp	BRD-K89708791	rifaximin	RNA synthesis inhibitor		NR1I2, CYP3A4	RNA synthesis inhibitor
698	95.59	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
699	95.59	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
700	95.59	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
701	95.58	kd	CGS001-51176	LEF1	-			
702	95.58	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
703	95.58	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
704	95.54	oe	ccsbBroad304_04153	PHF17	-			
705	95.52	kd	CGS001-3416	IDE	Pitrilysin			
706	95.52	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
707	95.5	kd	CGS001-4688	NCF2	Tetratricopeptide (TTC) repeat domain containing			
708	95.5	kd	CGS001-8522	GAS7	-			
709	95.47	kd	CGS001-1488	CTBP2	-			
710	95.46	kd	CGS001-7852	CXCR4	Chemokine receptors			
711	95.45	kd	CGS001-81848	SPRY4	-			
712	95.45	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
713	95.45	oe	ccsbBroad304_02759	DICER1	-			
714	95.42	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
715	95.42	kd	CGS001-3456	IFNB1	Interferons			
716	95.41	kd	CGS001-4781	NFIB	-			
717	95.4	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
718	95.39	oe	ccsbBroad304_01066	NDUFA4	-			
719	95.37	kd	CGS001-134187	POU5F2	Homeoboxes / POU class			
720	95.34	kd	CGS001-5066	PAM	-			
721	95.32	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
722	95.31	kd	CGS001-3225	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
723	95.3	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
724	95.3	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
725	95.3	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
726	95.29	kd	CGS001-55423	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
727	95.29	kd	CGS001-4208	MEF2C	Myocyte enhancer factors			
728	95.27	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
729	95.27	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
730	95.27	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
731	95.24	kd	CGS001-6794	STK11	LKB subfamily			
732	95.23	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
733	95.17	kd	CGS001-1675	CFD	Complement system			
734	95.15	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
735	95.13	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
736	95.13	kd	CGS001-10214	SSX3	-			
737	95.12	kd	CGS001-10617	STAMBP	-			
738	95.12	kd	CGS001-2793	GNGT2	-			
739	95.11	cp	BRD-A35519318	benidipine	Calcium channel blocker		CACNA1C, CACNA1G, CYP3A5	Calcium channel blocker
740	95.1	kd	CGS001-22905	EPN2	-			
741	95.1	oe	ccsbBroad304_01019	MLH1	-			
742	95.09	kd	CGS001-2876	GPX1	-			
743	95.08	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
744	95.07	kd	CGS001-571	BACH1	BTB/POZ domain containing			
745	95.07	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
746	95.03	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
747	95	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
748	95	kd	CGS001-374291	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
749	94.99	kd	CGS001-26277	TINF2	-			
750	94.97	kd	CGS001-813	CALU	EF-hand domain containing			
751	94.96	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
752	94.96	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
753	94.96	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
754	94.96	kd	CGS001-9638	FEZ1	-			
755	94.91	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
756	94.89	cp	BRD-K99447003	enalaprilat	ACE inhibitor		ACE	ACE inhibitor
757	94.87	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
758	94.86	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
759	94.86	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
760	94.86	cp	BRD-A62890442	3-methyl-GABA	GABA aminotransferase activator			GABA aminotransferase activator
761	94.83	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
762	94.82	kd	CGS001-55893	ZNF395	Zinc fingers, C2H2-type			
763	94.81	kd	CGS001-10437	IFI30	-			
764	94.78	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
765	94.77	kd	CGS001-930	CD19	CD molecules			
766	94.76	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
767	94.75	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
768	94.75	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
769	94.74	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
770	94.74	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
771	94.73	oe	ccsbBroad304_00239	CCNG1	-			
772	94.71	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
773	94.71	oe	ccsbBroad304_08116	TBK1	IKK family			
774	94.71	kd	CGS001-8692	HYAL2	-			
775	94.71	kd	CGS001-6990	DYNLT3	Cytoplasmic dyneins			
776	94.7	cp	BRD-K34508425	KUC103898N	-666			-666
777	94.7	kd	CGS001-218	ALDH3A1	Aldehyde dehydrogenases			
778	94.69	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
779	94.69	oe	ccsbBroad304_08605	PBK	TOPK family			
780	94.67	kd	CGS001-8805	TRIM24	TIF1 family			
781	94.6	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
782	94.59	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
783	94.58	kd	CGS001-6895	TARBP2	-			
784	94.57	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
785	94.54	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
786	94.54	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
787	94.51	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
788	94.48	kd	CGS001-3486	IGFBP3	insulin-like growth factor (IGF) binding proteins			
789	94.47	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
790	94.42	kd	CGS001-23344	ESYT1	Synaptotagmins			
791	94.41	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
792	94.41	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
793	94.39	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
794	94.37	kd	CGS001-5451	POU2F1	Homeoboxes / POU class			
795	94.36	cp	BRD-K51485625	ritonavir	HIV protease inhibitor		CYP3A4, CYP1A2, CYP2B6, CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
796	94.36	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
797	94.36	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
798	94.34	kd	CGS001-25861	DFNB31	-			
799	94.31	kd	CGS001-7345	UCHL1	Ubiquitin C-terminal hydrolase			
800	94.28	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
801	94.26	oe	ccsbBroad304_07080	TM7SF2	-			
802	94.25	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
803	94.25	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
804	94.24	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
805	94.24	kd	CGS001-607	BCL9	-			
806	94.24	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
807	94.23	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
808	94.21	cp	BRD-K06878038	deferiprone	Chelating agent		CYP4F2	Chelating agent
809	94.2	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
810	94.19	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
811	94.19	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
812	94.18	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
813	94.17	cc		Bromodomain Inhibitor	-			
814	94.13	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
815	94.11	kd	CGS001-9500	MAGED1	-			
816	94.09	kd	CGS001-51027	BOLA1	-			
817	94.08	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
818	94.08	kd	CGS001-6251	RSU1	-			
819	94.08	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
820	94.04	oe	ccsbBroad304_06845	RARRES3	-			
821	94.04	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
822	94.04	kd	CGS001-171017	ZNF384	Zinc fingers, C2H2-type			
823	94	kd	CGS001-10776	ARPP19	-			
824	93.98	cc		Akt Signaling GOF	-			
825	93.98	kd	CGS001-8463	TEAD2	-			
826	93.97	kd	CGS001-337867	UBAC2	-			
827	93.97	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
828	93.95	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
829	93.95	kd	CGS001-10795	ZNF268	Zinc fingers, C2H2-type			
830	93.95	kd	CGS001-3177	SLC29A2	SLC29 family			
831	93.95	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
832	93.94	kd	CGS001-51292	GMPR2	-			
833	93.92	kd	CGS001-8573	CASK	CASK family			
834	93.91	kd	CGS001-3630	INS	-			
835	93.89	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
836	93.88	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
837	93.88	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
838	93.87	oe	ccsbBroad304_06188	F10	Chymotrypsin			
839	93.86	cp	BRD-K96134740	kitasamycin	Protein synthesis inhibitor			Protein synthesis inhibitor
840	93.85	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
841	93.85	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
842	93.84	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
843	93.84	kd	CGS001-6787	NEK4	NIMA (never in mitosis gene a)- related kinase (NEK) family			
844	93.83	kd	CGS001-22841	RAB11FIP2	-			
845	93.82	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
846	93.82	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
847	93.81	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
848	93.76	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
849	93.75	kd	CGS001-5584	PRKCI	Iota subfamily			
850	93.74	kd	CGS001-83729	INHBE	-			
851	93.73	cp	BRD-A52282606	lacidipine	Calcium channel blocker		CACNA1C	Calcium channel blocker
852	93.72	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
853	93.71	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
854	93.71	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
855	93.71	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
856	93.7	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
857	93.7	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
858	93.68	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
859	93.67	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
860	93.67	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
861	93.66	kd	CGS001-6727	SRP14	-			
862	93.66	kd	CGS001-5590	PRKCZ	Iota subfamily			
863	93.65	oe	ccsbBroad304_02203	MAD2L1BP	-			
864	93.65	oe	ccsbBroad304_03047	BZW2	-			
865	93.65	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
866	93.64	oe	ccsbBroad304_06008	AP2M1	-			
867	93.63	kd	CGS001-54490	UGT2B28	UDP glucuronosyltransferases			
868	93.62	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
869	93.6	kd	CGS001-5875	RABGGTA	Prenyltransferase alpha subunit repeat containing			
870	93.57	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
871	93.56	oe	ccsbBroad304_01002	METTL1	-			
872	93.56	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
873	93.56	kd	CGS001-8914	TIMELESS	-			
874	93.55	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
875	93.54	kd	CGS001-10919	EHMT2	Histone methyltransferases			
876	93.53	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
877	93.52	cp	BRD-A71009679	KUC103420N	-666			-666
878	93.52	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
879	93.51	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
880	93.5	kd	CGS001-5359	PLSCR1	-			
881	93.49	kd	CGS001-10554	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
882	93.48	kd	CGS001-4712	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
883	93.47	kd	CGS001-716	C1S	Complement system			
884	93.46	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
885	93.45	kd	CGS001-390	RND3	-			
886	93.45	kd	CGS001-9759	HDAC4	Histone deacetylases			
887	93.44	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
888	93.43	cc		Mitogen activated protein kinases LOF	-			
889	93.41	kd	CGS001-7866	IFRD2	-			
890	93.38	kd	CGS001-6799	SULT1A2	Sulfotransferases, cytosolic			
891	93.36	kd	CGS001-2952	GSTT1	Glutathione S-transferases / Soluble			
892	93.34	kd	CGS001-23659	PLA2G15	-			
893	93.33	kd	CGS001-7181	NR2C1	Testicular receptors			
894	93.31	kd	CGS001-9375	TM9SF2	-			
895	93.31	kd	CGS001-1806	DPYD	-			
896	93.29	kd	CGS001-2730	GCLM	-			
897	93.29	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
898	93.29	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
899	93.27	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
900	93.27	kd	CGS001-3615	IMPDH2	Oxidoreductases			
901	93.16	kd	CGS001-5928	RBBP4	WD repeat domain containing			
902	93.15	oe	ccsbBroad304_03268	GMPR2	-			
903	93.15	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
904	93.13	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
905	93.1	kd	CGS001-6257	RXRB	Retinoid X receptors			
906	93.1	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
907	93.06	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
908	93.06	kd	CGS001-132	ADK	Adenosine turnover			
909	93.03	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
910	93.02	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
911	93.02	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
912	93.01	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
913	93.01	kd	CGS001-1981	EIF4G1	Parkinson disease			
914	93	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
915	93	kd	CGS001-891	CCNB1	-			
916	92.98	oe	ccsbBroad304_01577	SOD1	-			
917	92.97	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
918	92.97	kd	CGS001-5699	PSMB10	Proteasome (prosome, macropain) subunits			
919	92.95	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
920	92.95	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
921	92.92	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
922	92.89	oe	ccsbBroad304_03266	ERGIC2	-			
923	92.89	kd	CGS001-3664	IRF6	-			
924	92.89	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
925	92.86	kd	CGS001-1154	CISH	SH2 domain containing			
926	92.85	kd	CGS001-8743	TNFSF10	CD molecules			
927	92.8	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
928	92.8	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
929	92.79	kd	CGS001-140685	ZBTB46	BTB/POZ domain containing			
930	92.78	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
931	92.78	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
932	92.77	oe	ccsbBroad304_07761	CORO1A	Coronins			
933	92.72	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
934	92.72	kd	CGS001-9218	VAPA	-			
935	92.72	kd	CGS001-58528	RRAGD	-			
936	92.69	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
937	92.68	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
938	92.67	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
939	92.67	oe	ccsbBroad304_02298	DNM1L	-			
940	92.65	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
941	92.65	kd	CGS001-5018	OXA1L	-			
942	92.65	kd	CGS001-2056	EPO	Endogenous ligands			
943	92.63	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
944	92.54	oe	ccsbBroad304_03023	CRCP	-			
945	92.52	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
946	92.52	kd	CGS001-2168	FABP1	Fatty acid-binding proteins			
947	92.51	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
948	92.49	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
949	92.46	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
950	92.45	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
951	92.41	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
952	92.38	kd	CGS001-523	ATP6V1A	ATPases / V-type			
953	92.37	kd	CGS001-2959	GTF2B	General transcription factors			
954	92.32	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
955	92.32	kd	CGS001-55869	HDAC8	Histone deacetylases			
956	92.3	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
957	92.26	kd	CGS001-10691	GMEB1	-			
958	92.22	kd	CGS001-9817	KEAP1	Kelch-like proteins			
959	92.22	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
960	92.21	kd	CGS001-57665	RDH14	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
961	92.21	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
962	92.18	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
963	92.17	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
964	92.15	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
965	92.14	kd	CGS001-7374	UNG	-			
966	92.12	kd	CGS001-84433	CARD11	-			
967	92.11	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
968	92.1	kd	CGS001-10810	WASF3	-			
969	92.1	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
970	92.08	kd	CGS001-9263	STK17A	Death-associated kinase (DAPK) family			
971	92.04	kd	CGS001-22850	ADNP2	Zinc fingers, C2H2-type			
972	92.04	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
973	92.03	oe	ccsbBroad304_14047	TACC3	-			
974	92.01	cp	BRD-K32744045	disulfiram	Aldehyde dehydrogenase inhibitor		ALDH2, ALDH1A2, ALDH5A1, ALDH7A1, CYP2E1, DBH, DNMT1, TRPA1	Aldehyde dehydrogenase inhibitor, TRPV agonist, DNA methyltransferase inhibitor
975	91.99	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
976	91.97	kd	CGS001-23387	SIK3	QIK subfamily			
977	91.96	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
978	91.95	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
979	91.92	kd	CGS001-10957	PNRC1	-			
980	91.85	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
981	91.85	kd	CGS001-2153	F5	Blood coagulation components			
982	91.83	kd	CGS001-7175	TPR	-			
983	91.8	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
984	91.79	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
985	91.76	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
986	91.75	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
987	91.73	cp	BRD-K88701661	dimercaptosuccinic-acid	Chelating agent		DNMT1	Chelating agent
988	91.71	oe	ccsbBroad304_01304	PSEN1	Presenilin			
989	91.71	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
990	91.7	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
991	91.7	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
992	91.69	kd	CGS001-22894	DIS3	-			
993	91.68	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
994	91.64	kd	CGS001-6611	SMS	-			
995	91.62	kd	CGS001-28512	NKIRAS1	-			
996	91.61	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
997	91.6	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
998	91.59	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
999	91.59	kd	CGS001-808	CALM3	EF-hand domain containing			
1000	91.56	oe	ccsbBroad304_06837	RAF1	RAF family			
1001	91.55	kd	CGS001-4707	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
1002	91.55	kd	CGS001-8870	IER3	-			
1003	91.48	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
1004	91.46	kd	CGS001-7504	XK	Blood group antigens			
1005	91.46	kd	CGS001-8148	TAF15	RNA binding motif (RRM) containing			
1006	91.46	kd	CGS001-51031	GLOD4	-			
1007	91.44	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
1008	91.43	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
1009	91.42	kd	CGS001-3203	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
1010	91.41	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
1011	91.36	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
1012	91.35	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
1013	91.33	kd	CGS001-587	BCAT2	-			
1014	91.32	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
1015	91.32	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
1016	91.31	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
1017	91.31	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
1018	91.28	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
1019	91.26	kd	CGS001-65123	INTS3	-			
1020	91.23	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
1021	91.21	kd	CGS001-10131	TRAP1	Heat shock proteins / HSPC			
1022	91.2	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
1023	91.2	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
1024	91.19	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
1025	91.19	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
1026	91.18	kd	CGS001-5918	RARRES1	-			
1027	91.17	kd	CGS001-151742	PPM1L	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1028	91.16	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
1029	91.15	kd	CGS001-8874	ARHGEF7	Rho guanine nucleotide exchange factors			
1030	91.14	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
1031	91.13	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1032	91.12	kd	CGS001-597	BCL2A1	-			
1033	91.07	kd	CGS001-6472	SHMT2	-			
1034	91.07	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
1035	91.06	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
1036	91.06	kd	CGS001-57661	PHRF1	Zinc fingers, PHD-type			
1037	91.03	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
1038	91.01	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
1039	91.01	kd	CGS001-10652	YKT6	-			
1040	90.98	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
1041	90.96	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
1042	90.93	kd	CGS001-5653	KLK6	Chymotrypsin			
1043	90.93	kd	CGS001-1891	ECH1	-			
1044	90.82	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1045	90.81	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
1046	90.8	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
1047	90.78	kd	CGS001-5228	PGF	-			
1048	90.74	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
1049	90.73	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
1050	90.71	kd	CGS001-58492	ZNF77	Zinc fingers, C2H2-type			
1051	90.7	cc		General transcription factors group 1 LOF	-			
1052	90.7	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
1053	90.7	kd	CGS001-2130	EWSR1	RNA binding motif (RRM) containing			
1054	90.68	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
1055	90.68	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
1056	90.68	kd	CGS001-8726	EED	Neutral sphingomyelinase coupling factors			
1057	90.64	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
1058	90.62	kd	CGS001-5962	RDX	-			
1059	90.52	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
1060	90.49	kd	CGS001-6513	SLC2A1	Solute carriers			
1061	90.48	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
1062	90.47	kd	CGS001-1513	CTSK	Cathepsins			
1063	90.45	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
1064	90.43	kd	CGS001-7020	TFAP2A	-			
1065	90.39	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
1066	90.38	kd	CGS001-3705	ITPK1	-			
1067	90.36	kd	CGS001-54407	SLC38A2	System A-like transporters			
1068	90.36	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
1069	90.34	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1070	90.34	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
1071	90.33	kd	CGS001-5583	PRKCH	Eta subfamily			
1072	90.32	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
1073	90.32	kd	CGS001-1131	CHRM3	Cholinergic receptors			
1074	90.3	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
1075	90.28	kd	CGS001-2053	EPHX2	-			
1076	90.27	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
1077	90.27	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
1078	90.21	cc		Serpin peptidase inhibitors LOF	-			
1079	90.21	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
1080	90.2	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
1081	90.19	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1082	90.17	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
1083	90.16	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
1084	90.16	kd	CGS001-1389	CREBL2	basic leucine zipper proteins			
1085	90.13	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
1086	90.13	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
1087	90.13	kd	CGS001-23314	SATB2	Homeoboxes / CUT class			
1088	90.12	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
1089	90.12	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
1090	90.09	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
1091	90.07	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
1092	90.07	kd	CGS001-408	ARRB1	-			
1093	90	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
1094	89.95	oe	ccsbBroad304_00398	CTSL2	-			
1095	89.92	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
1096	89.91	cc		FXR antagonist	-			
1097	89.9	cp	BRD-K44094599	tacrolimus	Calcineurin inhibitor		FKBP1A, CYP3A5, CYP3A7	Calcineurin inhibitor
1098	89.9	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
1099	89.83	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
1100	89.82	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
1101	89.82	oe	ccsbBroad304_06739	PLOD1	-			
1102	89.81	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
1103	89.8	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
1104	89.8	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
1105	89.77	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
1106	89.77	kd	CGS001-168374	ZNF92	Zinc fingers, C2H2-type			
1107	89.7	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
1108	89.63	cc		Leucine rich repeat kinase inhibitor	-			
1109	89.63	oe	ccsbBroad304_07097	TRAF1	-			
1110	89.6	kd	CGS001-9	NAT1	-			
1111	89.55	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
1112	89.55	oe	ccsbBroad304_02220	MTFR1	-			
1113	89.54	kd	CGS001-8835	SOCS2	SH2 domain containing			
1114	89.5	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
1115	89.48	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
1116	89.44	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
1117	89.42	kd	CGS001-3665	IRF7	-			
1118	89.32	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
1119	89.31	oe	ccsbBroad304_09035	COASY	-			
1120	89.29	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
1121	89.29	kd	CGS001-9459	ARHGEF6	Rho guanine nucleotide exchange factors			
1122	89.27	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
1123	89.26	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
1124	89.24	oe	ccsbBroad304_01880	LAGE3	-			
1125	89.23	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
1126	89.23	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
1127	89.22	oe	ccsbBroad304_00390	CTGF	-			
1128	89.2	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
1129	89.2	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
1130	89.19	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1131	89.13	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
1132	89.11	kd	CGS001-7025	NR2F1	COUP-TF-like receptors			
1133	89.09	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
1134	89.08	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
1135	89.06	kd	CGS001-23131	GPATCH8	G patch domain containing			
1136	89.05	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
1137	89.04	kd	CGS001-1843	DUSP1	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1138	89.04	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
1139	88.97	kd	CGS001-6046	BRD2	Bromodomain kinase (BRDK) family			
1140	88.9	oe	ccsbBroad304_01139	PA2G4	-			
1141	88.88	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
1142	88.87	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
1143	88.82	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
1144	88.8	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
1145	88.75	kd	CGS001-8220	DGCR14	-			
1146	88.74	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
1147	88.71	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
1148	88.7	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
1149	88.67	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
1150	88.64	kd	CGS001-2072	ERCC4	-			
1151	88.62	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
1152	88.62	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
1153	88.62	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
1154	88.6	kd	CGS001-3131	HLF	-			
1155	88.56	kd	CGS001-10513	APPBP2	-			
1156	88.52	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
1157	88.51	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
1158	88.51	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
1159	88.49	kd	CGS001-6884	TAF13	-			
1160	88.49	kd	CGS001-5909	RAP1GAP	-			
1161	88.48	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1162	88.48	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
1163	88.48	kd	CGS001-5921	RASA1	Pleckstrin homology (PH) domain containing			
1164	88.47	kd	CGS001-1892	ECHS1	-			
1165	88.44	cc		MDM inhibitor	-			
1166	88.42	kd	CGS001-22954	TRIM32	-			
1167	88.41	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
1168	88.4	kd	CGS001-6519	SLC3A1	SLC3 family			
1169	88.38	kd	CGS001-80758	PRR7	-			
1170	88.37	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
1171	88.37	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
1172	88.36	kd	CGS001-6713	SQLE	Lanosterol biosynthesis pathway			
1173	88.35	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
1174	88.35	kd	CGS001-10991	SLC38A3	System N-like transporters			
1175	88.33	kd	CGS001-317705	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
1176	88.33	kd	CGS001-5688	PSMA7	Proteasome subunits			
1177	88.31	kd	CGS001-694	BTG1	-			
1178	88.3	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
1179	88.25	kd	CGS001-4069	LYZ	-			
1180	88.22	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
1181	88.18	kd	CGS001-51564	HDAC7	Histone deacetylases			
1182	88.15	kd	CGS001-2776	GNAQ	-			
1183	88.14	kd	CGS001-203	AK1	Adenylate kinases			
1184	88.12	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
1185	88.1	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
1186	88.09	kd	CGS001-9926	LPGAT1	-			
1187	88.08	kd	CGS001-10950	BTG3	-			
1188	88.06	kd	CGS001-4194	MDM4	-			
1189	88.01	kd	CGS001-9181	ARHGEF2	Rho guanine nucleotide exchange factors			
1190	87.98	oe	ccsbBroad304_01960	CASK	CASK family			
1191	87.95	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
1192	87.89	kd	CGS001-80212	CCDC92	-			
1193	87.88	cp	BRD-A48261811	argatroban	Thrombin inhibitor		F2, CYP3A5	Thrombin inhibitor
1194	87.81	kd	CGS001-23636	NUP62	-			
1195	87.81	kd	CGS001-375318	AQP12A	Ion channels / Aquaporins			
1196	87.79	cp	BRD-K81855038	roxatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
1197	87.78	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
1198	87.76	kd	CGS001-84109	QRFPR	GPCR / Class A : RF amide peptide receptors			
1199	87.75	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
1200	87.73	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
1201	87.73	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1202	87.7	kd	CGS001-55958	KLHL9	BTB/POZ domain containing			
1203	87.64	kd	CGS001-599	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1204	87.6	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
1205	87.59	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
1206	87.59	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
1207	87.58	kd	CGS001-8651	SOCS1	SH2 domain containing			
1208	87.57	kd	CGS001-9928	KIF14	Kinesins			
1209	87.56	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
1210	87.55	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
1211	87.53	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
1212	87.5	oe	ccsbBroad304_01519	SET	-			
1213	87.49	oe	ccsbBroad304_01392	TRIM27	-			
1214	87.49	kd	CGS001-4312	MMP1	Matrix metallopeptidase			
1215	87.46	kd	CGS001-1788	DNMT3A	Methyltransferases			
1216	87.44	kd	CGS001-6117	RPA1	-			
1217	87.43	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
1218	87.42	oe	ccsbBroad304_03269	CD320	CD molecules			
1219	87.41	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1220	87.4	kd	CGS001-5771	PTPN2	Protein tyrosine phosphatases			
1221	87.39	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
1222	87.37	kd	CGS001-1635	DCTD	-			
1223	87.37	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
1224	87.33	kd	CGS001-115727	RASGRP4	EF-hand domain containing			
1225	87.32	kd	CGS001-2747	GLUD2	-			
1226	87.31	oe	ccsbBroad304_02340	SORBS3	-			
1227	87.31	oe	ccsbBroad304_08840	KIF9	Kinesins			
1228	87.27	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
1229	87.27	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
1230	87.26	kd	CGS001-201799	TMEM154	-			
1231	87.26	kd	CGS001-63948	DMRTB1	-			
1232	87.24	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
1233	87.22	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
1234	87.22	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
1235	87.2	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
1236	87.2	kd	CGS001-471	ATIC	-			
1237	87.16	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
1238	87.15	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
1239	87.15	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
1240	87.09	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
1241	87.06	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
1242	87.03	kd	CGS001-80135	RPF1	-			
1243	87	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
1244	87	kd	CGS001-4282	MIF	-			
1245	86.95	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
1246	86.94	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
1247	86.92	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
1248	86.86	kd	CGS001-5091	PC	Carboxylases			
1249	86.84	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
1250	86.84	kd	CGS001-1876	E2F6	-			
1251	86.8	kd	CGS001-10553	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
1252	86.78	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
1253	86.76	oe	ccsbBroad304_09281	TPD52L3	-			
1254	86.76	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
1255	86.72	cc		PRD class homeoboxes and psudogenes LOF	-			
1256	86.72	kd	CGS001-5831	PYCR1	-			
1257	86.7	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
1258	86.7	kd	CGS001-51335	NGRN	-			
1259	86.68	kd	CGS001-1840	DTX1	-			
1260	86.64	cp	BRD-K56450366	NSC-94258	Antineoplastic		AKR1B1, CYP19A1, HSD17B1	Antineoplastic
1261	86.64	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
1262	86.63	oe	ccsbBroad304_01617	STX4	-			
1263	86.62	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
1264	86.62	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
1265	86.58	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1266	86.57	oe	ccsbBroad304_00614	GAMT	-			
1267	86.56	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
1268	86.53	kd	CGS001-3614	IMPDH1	Oxidoreductases			
1269	86.52	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
1270	86.51	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
1271	86.49	kd	CGS001-79006	METRN	-			
1272	86.45	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
1273	86.42	kd	CGS001-55214	LEPREL1	-			
1274	86.41	kd	CGS001-23649	POLA2	DNA polymerases			
1275	86.38	cc		PI3K Signaling LOF	-			
1276	86.38	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
1277	86.35	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
1278	86.34	kd	CGS001-2568	GABRP	GABA receptors			
1279	86.3	kd	CGS001-255877	BCL6B	BTB/POZ domain containing			
1280	86.25	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1281	86.22	cc		Bile acid	-			
1282	86.21	kd	CGS001-5824	PEX19	-			
1283	86.2	kd	CGS001-6925	TCF4	Basic helix-loop-helix proteins			
1284	86.19	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
1285	86.18	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
1286	86.13	kd	CGS001-23038	WDTC1	DDB1 and CUL4 associated factors			
1287	86.11	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
1288	86.1	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
1289	86.1	kd	CGS001-126208	ZNF787	Zinc fingers, C2H2-type			
1290	86.04	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1291	86.03	kd	CGS001-23039	XPO7	Exportins			
1292	86.03	kd	CGS001-2950	GSTP1	Glutathione S-transferases			
1293	86.02	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
1294	86.01	kd	CGS001-85377	MICALL1	-			
1295	86	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
1296	85.95	kd	CGS001-22891	ZNF365	Zinc fingers, C2H2-type			
1297	85.92	oe	ccsbBroad304_02668	PNKP	-			
1298	85.91	kd	CGS001-6886	TAL1	Basic helix-loop-helix proteins			
1299	85.88	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
1300	85.87	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1301	85.85	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
1302	85.85	kd	CGS001-55290	BRF2	-			
1303	85.84	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
1304	85.8	kd	CGS001-4190	MDH1	-			
1305	85.78	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
1306	85.76	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
1307	85.72	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
1308	85.72	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
1309	85.64	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
1310	85.63	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
1311	85.61	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
1312	85.59	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
1313	85.57	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
1314	85.55	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
1315	85.55	oe	ccsbBroad304_00883	ISG20	-			
1316	85.54	oe	ccsbBroad304_03444	PAF1	-			
1317	85.54	kd	CGS001-3688	ITGB1	Integrins			
1318	85.53	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
1319	85.5	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
1320	85.5	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
1321	85.44	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
1322	85.4	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
1323	85.39	oe	ccsbBroad304_02349	MPHOSPH9	-			
1324	85.38	kd	CGS001-3385	ICAM3	CD molecules			
1325	85.37	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
1326	85.35	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
1327	85.35	kd	CGS001-29899	GPSM2	Tetratricopeptide (TTC) repeat domain containing			
1328	85.33	kd	CGS001-23405	DICER1	-			
1329	85.3	kd	CGS001-9925	ZBTB5	BTB/POZ domain containing			
1330	85.28	kd	CGS001-211	ALAS1	-			
1331	85.21	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
1332	85.2	kd	CGS001-10046	MAMLD1	-			
1333	85.16	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
1334	85.15	oe	ccsbBroad304_02592	KIF2C	Kinesins			
1335	85.11	kd	CGS001-55654	TMEM127	-			
1336	85.1	kd	CGS001-2119	ETV5	ETS Transcription Factors			
1337	85.02	kd	CGS001-9531	BAG3	-			
1338	85.01	kd	CGS001-8896	BUD31	-			
1339	84.87	kd	CGS001-2048	EPHB2	Type XIII RTKs: Ephrin receptor family			
1340	84.86	kd	CGS001-90655	TGIF2LY	Homeoboxes / TALE class			
1341	84.86	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
1342	84.78	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
1343	84.76	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
1344	84.76	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
1345	84.75	kd	CGS001-29984	RHOD	-			
1346	84.74	kd	CGS001-51655	RASD1	-			
1347	84.71	kd	CGS001-6253	RTN2	-			
1348	84.66	kd	CGS001-5915	RARB	Retinoic acid receptors			
1349	84.65	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
1350	84.65	oe	ccsbBroad304_00183	C1S	Complement system			
1351	84.61	kd	CGS001-10221	TRIB1	Trbl family			
1352	84.61	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
1353	84.6	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
1354	84.55	kd	CGS001-147837	ZNF563	Zinc fingers, C2H2-type			
1355	84.54	oe	ccsbBroad304_00469	DUT	-			
1356	84.51	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
1357	84.51	kd	CGS001-10476	ATP5H	ATPases / F-type			
1358	84.51	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
1359	84.48	kd	CGS001-1386	ATF2	basic leucine zipper proteins			
1360	84.47	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
1361	84.46	kd	CGS001-5595	MAPK3	MAPK:ERK subfamily			
1362	84.43	kd	CGS001-10845	CLPX	ATPases / AAA-type			
1363	84.39	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
1364	84.33	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
1365	84.31	cp	BRD-K82143716	flucytosine	Antifungal		DNMT1	Antifungal
1366	84.31	kd	CGS001-286075	ZNF707	Zinc fingers, C2H2-type			
1367	84.28	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
1368	84.27	kd	CGS001-10237	SLC35B1	SLC35 family of nucleotide sugar transporters			
1369	84.27	kd	CGS001-50846	DHH	-			
1370	84.25	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
1371	84.24	cp	BRD-A24191444	ifenprodil	Adrenergic receptor antagonist		GRIN1, GRIN2B	Adrenergic receptor antagonist, Glutamate receptor antagonist
1372	84.24	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
1373	84.22	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
1374	84.22	kd	CGS001-8508	NIPSNAP1	-			
1375	84.21	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
1376	84.19	kd	CGS001-1948	EFNB2	Ephrins			
1377	84.02	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
1378	84.01	kd	CGS001-1719	DHFR	Oxidoreductases			
1379	83.99	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
1380	83.99	kd	CGS001-2098	ESD	-			
1381	83.93	kd	CGS001-10657	KHDRBS1	-			
1382	83.93	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
1383	83.92	kd	CGS001-23463	ICMT	-			
1384	83.88	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
1385	83.87	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
1386	83.85	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
1387	83.84	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
1388	83.8	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
1389	83.77	kd	CGS001-3176	HNMT	-			
1390	83.72	kd	CGS001-389421	LIN28B	-			
1391	83.65	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
1392	83.65	kd	CGS001-3690	ITGB3	Integrins			
1393	83.61	kd	CGS001-79733	E2F8	-			
1394	83.57	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
1395	83.57	kd	CGS001-4841	NONO	RNA binding motif (RRM) containing			
1396	83.56	oe	ccsbBroad304_02756	RRP8	-			
1397	83.56	kd	CGS001-55179	FAIM	-			
1398	83.55	kd	CGS001-6775	STAT4	SH2 domain containing			
1399	83.54	kd	CGS001-51441	YTHDF2	-			
1400	83.52	kd	CGS001-10153	CEBPZ	-			
1401	83.5	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
1402	83.48	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
1403	83.47	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
1404	83.45	kd	CGS001-6908	TBP	General transcription factors			
1405	83.43	oe	ccsbBroad304_06098	DHCR24	-			
1406	83.39	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
1407	83.38	cc		Bacterial 30S ribosomal subunit inhibitor	-			
1408	83.36	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
1409	83.35	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
1410	83.33	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
1411	83.28	cp	BRD-K82795137	loratadine	Histamine receptor antagonist		HRH1, CYP2C19, CYP3A5	Histamine receptor antagonist
1412	83.28	kd	CGS001-10755	GIPC1	-			
1413	83.25	kd	CGS001-9061	PAPSS1	-			
1414	83.21	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
1415	83.18	kd	CGS001-1468	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
1416	83.12	kd	CGS001-54732	TMED9	-			
1417	83.06	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
1418	83.06	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
1419	83.03	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
1420	83.02	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
1421	82.98	kd	CGS001-439	ASNA1	-			
1422	82.96	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
1423	82.89	kd	CGS001-3689	ITGB2	Integrins			
1424	82.87	oe	ccsbBroad304_03237	LEF1	-			
1425	82.84	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
1426	82.84	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
1427	82.83	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1428	82.75	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
1429	82.65	oe	ccsbBroad304_02239	RASSF2	-			
1430	82.65	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
1431	82.6	oe	ccsbBroad304_02596	KDELR3	-			
1432	82.59	kd	CGS001-80025	PANK2	-			
1433	82.57	kd	CGS001-6478	SIAH2	-			
1434	82.51	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
1435	82.51	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
1436	82.5	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
1437	82.47	kd	CGS001-55328	RNLS	-			
1438	82.45	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
1439	82.43	kd	CGS001-1951	CELSR3	Cadherins / Major cadherins			
1440	82.4	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
1441	82.4	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1442	82.37	kd	CGS001-6678	SPARC	-			
1443	82.35	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1444	82.33	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
1445	82.32	oe	ccsbBroad304_02579	YWHAQ	-			
1446	82.31	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
1447	82.31	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
1448	82.29	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
1449	82.28	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
1450	82.24	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
1451	82.16	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
1452	82.15	kd	CGS001-6722	SRF	-			
1453	82.15	kd	CGS001-2356	FPGS	-			
1454	82.13	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
1455	82.11	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
1456	82.1	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
1457	82.07	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
1458	82.03	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
1459	82.02	kd	CGS001-8318	CDC45	-			
1460	81.95	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
1461	81.94	kd	CGS001-58497	PRUNE	-			
1462	81.85	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
1463	81.81	kd	CGS001-83593	RASSF5	-			
1464	81.79	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
1465	81.75	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1466	81.69	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
1467	81.65	oe	ccsbBroad304_01163	PDHA1	-			
1468	81.61	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1469	81.6	oe	ccsbBroad304_05823	ANXA2	Annexins			
1470	81.52	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
1471	81.33	kd	CGS001-11257	TP53TG1	-			
1472	81.32	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
1473	81.31	oe	ccsbBroad304_00529	F3	CD molecules			
1474	81.3	kd	CGS001-55120	FANCL	Fanconi anemia, complementation groups			
1475	81.3	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
1476	81.29	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1477	81.28	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
1478	81.28	kd	CGS001-27097	TAF5L	WD repeat domain containing			
1479	81.25	oe	ccsbBroad304_00170	BNIP1	-			
1480	81.23	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
1481	81.2	kd	CGS001-23274	CLEC16A	C-type lectin domain containing			
1482	81.18	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
1483	81.16	kd	CGS001-5860	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
1484	81.16	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
1485	81.09	kd	CGS001-516	ATP5G1	ATPases / F-type			
1486	81.08	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1487	81.08	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
1488	81.03	oe	ccsbBroad304_02276	MVP	-			
1489	80.98	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
1490	80.98	kd	CGS001-6608	SMO	GPCR / Class F : Frizzled receptors			
1491	80.97	kd	CGS001-23077	MYCBP2	-			
1492	80.93	kd	CGS001-9767	PHF16	-			
1493	80.9	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
1494	80.88	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
1495	80.82	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
1496	80.77	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
1497	80.7	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
1498	80.69	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
1499	80.68	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
1500	80.67	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
1501	80.67	oe	ccsbBroad304_03089	PACSIN3	-			
1502	80.66	kd	CGS001-629	CFB	Complement system			
1503	80.64	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
1504	80.62	cp	BRD-K43236057	piceid	ICAM1 inhibitor		GAA, XDH	ICAM1 inhibitor
1505	80.61	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
1506	80.55	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
1507	80.54	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
1508	80.52	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
1509	80.49	oe	ccsbBroad304_02026	NRP1	CD molecules			
1510	80.45	kd	CGS001-23576	DDAH1	Dimethylarginine dimethylaminohydrolases			
1511	80.39	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
1512	80.36	oe	ccsbBroad304_06458	IRF3	-			
1513	80.35	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1514	80.34	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
1515	80.32	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
1516	80.27	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1517	80.27	oe	ccsbBroad304_06301	GOT2	-			
1518	80.26	kd	CGS001-3920	LAMP2	CD molecules			
1519	80.17	kd	CGS001-6601	SMARCC2	-			
1520	80.15	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
1521	80.13	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
1522	80.13	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
1523	80.13	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
1524	80.01	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
1525	80.01	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
1526	79.99	kd	CGS001-25793	FBXO7	F-boxes / other			
1527	79.98	kd	CGS001-1983	EIF5	-			
1528	79.96	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
1529	79.92	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
1530	79.92	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
1531	79.92	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
1532	79.92	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
1533	79.91	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
1534	79.87	kd	CGS001-27102	EIF2AK1	Other PEK family kinases			
1535	79.83	kd	CGS001-23492	CBX7	-			
1536	79.81	kd	CGS001-25987	TSKU	-			
1537	79.79	kd	CGS001-5563	PRKAA2	AMPK subfamily			
1538	79.76	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
1539	79.71	kd	CGS001-10888	GPR83	GPCR / Class A : Orphans			
1540	79.7	cc		Dihydrofolate reductase inhibitor	-			
1541	79.7	kd	CGS001-130497	OSR1	Zinc fingers, C2H2-type			
1542	79.68	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
1543	79.63	kd	CGS001-6272	SORT1	-			
1544	79.62	cp	BRD-K49404994	levetiracetam	Calcium channel blocker		SV2A, CACNA1B, SCN1A	Calcium channel blocker
1545	79.55	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
1546	79.55	kd	CGS001-5048	PAFAH1B1	WD repeat domain containing			
1547	79.54	oe	ccsbBroad304_08709	SCYL3	-			
1548	79.53	kd	CGS001-25888	ZNF473	Zinc fingers, C2H2-type			
1549	79.5	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
1550	79.48	kd	CGS001-8974	P4HA2	-			
1551	79.44	kd	CGS001-79600	TCTN1	Tectonic proteins			
1552	79.43	kd	CGS001-5805	PTS	-			
1553	79.4	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
1554	79.37	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
1555	79.34	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
1556	79.34	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
1557	79.34	kd	CGS001-415116	PIM3	PIM family			
1558	79.32	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
1559	79.3	kd	CGS001-9917	FAM20B	-			
1560	79.21	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
1561	79.18	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
1562	79.15	kd	CGS001-9918	NCAPD2	-			
1563	79.13	oe	ccsbBroad304_00150	BAX	-			
1564	79.13	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
1565	79.09	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
1566	79.05	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
1567	79.03	kd	CGS001-5645	PRSS2	Serine peptidases			
1568	79.01	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
1569	79.01	kd	CGS001-5352	PLOD2	-			
1570	78.98	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
1571	78.96	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
1572	78.88	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
1573	78.83	kd	CGS001-5236	PGM1	-			
1574	78.79	kd	CGS001-56654	NPDC1	-			
1575	78.76	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
1576	78.72	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
1577	78.71	kd	CGS001-7297	TYK2	Janus kinase (JakA) family			
1578	78.7	kd	CGS001-8895	CPNE3	-			
1579	78.7	oe	ccsbBroad304_00464	DTNA	-			
1580	78.64	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
1581	78.63	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
1582	78.62	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
1583	78.59	kd	CGS001-8535	CBX4	-			
1584	78.51	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1585	78.51	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
1586	78.51	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
1587	78.39	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
1588	78.38	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
1589	78.33	oe	ccsbBroad304_01208	PITPNA	-			
1590	78.21	kd	CGS001-6850	SYK	Syk family			
1591	78.21	kd	CGS001-338557	O3FAR1	-			
1592	78.19	oe	ccsbBroad304_06695	PCK2	-			
1593	78.15	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
1594	78.1	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
1595	78.08	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
1596	78.01	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
1597	77.98	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
1598	77.95	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1599	77.94	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
1600	77.88	kd	CGS001-842	CASP9	Caspases			
1601	77.86	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
1602	77.85	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
1603	77.82	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
1604	77.82	kd	CGS001-57680	CHD8	-			
1605	77.8	kd	CGS001-23211	ZC3H4	Zinc fingers, CCCH-type domain containing			
1606	77.79	kd	CGS001-23657	SLC7A11	Solute carriers			
1607	77.76	kd	CGS001-8772	FADD	-			
1608	77.76	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
1609	77.74	kd	CGS001-10269	ZMPSTE24	-			
1610	77.72	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
1611	77.69	kd	CGS001-8804	CREG1	-			
1612	77.68	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
1613	77.66	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
1614	77.63	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
1615	77.58	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
1616	77.57	oe	ccsbBroad304_03640	CEP72	-			
1617	77.56	kd	CGS001-5933	RBL1	-			
1618	77.55	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
1619	77.53	oe	ccsbBroad304_08045	NOX1	-			
1620	77.5	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
1621	77.45	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
1622	77.43	kd	CGS001-7249	TSC2	-			
1623	77.43	oe	ccsbBroad304_06048	CRYZ	-			
1624	77.41	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
1625	77.39	cc		Aurora kinase inhibitor	-			
1626	77.38	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
1627	77.38	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
1628	77.35	kd	CGS001-5306	PITPNA	-			
1629	77.3	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
1630	77.27	oe	ccsbBroad304_07326	EIF2B2	-			
1631	77.26	oe	ccsbBroad304_07118	UGDH	-			
1632	77.24	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
1633	77.14	oe	ccsbBroad304_00969	MAGEA10	-			
1634	77.09	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
1635	77.07	kd	CGS001-1305	COL13A1	Collagens			
1636	77.05	oe	ccsbBroad304_00001	NAT1	-			
1637	77.04	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
1638	76.91	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
1639	76.9	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
1640	76.84	kd	CGS001-286530	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
1641	76.81	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
1642	76.72	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
1643	76.7	kd	CGS001-1763	DNA2	-			
1644	76.7	kd	CGS001-10904	BLCAP	-			
1645	76.69	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
1646	76.67	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
1647	76.62	kd	CGS001-1509	CTSD	Cathepsins			
1648	76.57	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
1649	76.51	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
1650	76.49	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
1651	76.46	kd	CGS001-5618	PRLR	Prolactin receptor family			
1652	76.43	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
1653	76.4	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
1654	76.33	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
1655	76.32	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
1656	76.31	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
1657	76.3	kd	CGS001-2071	ERCC3	General transcription factors			
1658	76.19	kd	CGS001-7625	ZNF74	Zinc fingers, C2H2-type			
1659	76.16	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
1660	76.14	oe	ccsbBroad304_06420	ICAM3	CD molecules			
1661	76.06	kd	CGS001-10447	FAM3C	-			
1662	76.03	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
1663	75.99	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
1664	75.98	kd	CGS001-6625	SNRNP70	RNA binding motif (RRM) containing			
1665	75.98	kd	CGS001-7272	TTK	TTK family			
1666	75.98	kd	CGS001-2495	FTH1	-			
1667	75.97	kd	CGS001-79094	CHAC1	-			
1668	75.95	cc		Thymidylate synthase inhibitor	-			
1669	75.9	kd	CGS001-10887	PROKR1	GPCR / Class A : Prokineticin receptors			
1670	75.9	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
1671	75.86	kd	CGS001-80762	NDFIP1	-			
1672	75.84	kd	CGS001-991	CDC20	WD repeat domain containing			
1673	75.77	cp	BRD-K04196797	oxcarbazepine	Sodium channel blocker		CYP2C19, CYP3A4, CYP3A5, SCN1A, SCN3A, SCN5A	Sodium channel blocker
1674	75.75	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
1675	75.65	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
1676	75.65	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
1677	75.64	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
1678	75.56	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
1679	75.51	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
1680	75.48	kd	CGS001-1027	CDKN1B	-			
1681	75.44	kd	CGS001-3170	FOXA2	Forkhead boxes			
1682	75.44	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
1683	75.39	kd	CGS001-57157	PHTF2	-			
1684	75.37	kd	CGS001-3458	IFNG	Interferons			
1685	75.35	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
1686	75.34	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1687	75.32	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1688	75.32	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1689	75.31	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
1690	75.3	oe	ccsbBroad304_07238	STK24	YSK subfamily			
1691	75.17	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
1692	75.14	kd	CGS001-23461	ABCA5	ATP binding cassette transporters / subfamily A			
1693	75.1	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
1694	75.09	oe	ccsbBroad304_04619	GNG8	-			
1695	75.08	kd	CGS001-64781	CERK	Ceramide kinase			
1696	75.07	kd	CGS001-9261	MAPKAPK2	MAPKAPK subfamily			
1697	75.06	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
1698	75.03	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
1699	74.98	kd	CGS001-29998	GLTSCR1	-			
1700	74.95	kd	CGS001-55536	CDCA7L	-			
1701	74.89	oe	ccsbBroad304_01787	YES1	Src family			
1702	74.87	kd	CGS001-9955	HS3ST3A1	Sulfotransferases, membrane-bound			
1703	74.86	kd	CGS001-200734	SPRED2	-			
1704	74.86	kd	CGS001-64921	CASD1	-			
1705	74.84	kd	CGS001-598	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1706	74.81	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1707	74.79	kd	CGS001-5696	PSMB8	Proteasome (prosome, macropain) subunits			
1708	74.79	kd	CGS001-1031	CDKN2C	Ankyrin repeat domain containing			
1709	74.76	kd	CGS001-23401	FRAT2	-			
1710	74.76	kd	CGS001-55810	FOXJ2	Forkhead boxes			
1711	74.73	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
1712	74.69	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
1713	74.64	kd	CGS001-6813	STXBP2	-			
1714	74.61	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
1715	74.57	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
1716	74.56	cc		LIM class homeoboxes GOF	-			
1717	74.55	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
1718	74.54	oe	ccsbBroad304_13903	MTAP	-			
1719	74.53	kd	CGS001-29775	CARD10	-			
1720	74.42	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
1721	74.4	oe	ccsbBroad304_07280	LAMTOR3	-			
1722	74.39	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
1723	74.35	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
1724	74.31	kd	CGS001-25805	BAMBI	-			
1725	74.3	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
1726	74.11	cp	BRD-K32311154	nifekalant	Potassium channel blocker			Potassium channel blocker
1727	74.09	oe	ccsbBroad304_01933	TEAD2	-			
1728	74.07	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
1729	74.06	kd	CGS001-4170	MCL1	-			
1730	74.04	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
1731	73.97	kd	CGS001-54499	TMCO1	-			
1732	73.91	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
1733	73.91	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
1734	73.88	kd	CGS001-6286	S100P	EF-hand domain containing			
1735	73.87	kd	CGS001-3821	KLRC1	CD molecules			
1736	73.82	cp	BRD-K41051431	mecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1737	73.81	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
1738	73.8	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
1739	73.75	oe	ccsbBroad304_07561	YAF2	-			
1740	73.75	kd	CGS001-51172	NAGPA	-			
1741	73.69	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
1742	73.68	oe	ccsbBroad304_00876	INSIG1	-			
1743	73.64	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1744	73.61	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
1745	73.6	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
1746	73.54	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
1747	73.5	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
1748	73.49	kd	CGS001-9052	GPRC5A	GPCR / Class C : Orphans			
1749	73.42	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
1750	73.41	kd	CGS001-79960	PHF17	-			
1751	73.35	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1752	73.31	oe	ccsbBroad304_07050	TFAP2A	-			
1753	73.3	kd	CGS001-57222	ERGIC1	-			
1754	73.3	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
1755	73.27	oe	ccsbBroad304_00661	GNGT2	-			
1756	73.27	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
1757	73.25	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1758	73.23	kd	CGS001-2348	FOLR1	-			
1759	73.21	kd	CGS001-26136	TES	-			
1760	73.2	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
1761	73.18	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
1762	73.12	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
1763	73.07	kd	CGS001-25874	BRP44	-			
1764	73.02	kd	CGS001-10427	SEC24B	-			
1765	72.99	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
1766	72.92	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
1767	72.9	kd	CGS001-51701	NLK	nmo subfamily			
1768	72.88	kd	CGS001-8449	DHX16	DEAH-boxes			
1769	72.84	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
1770	72.82	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
1771	72.79	kd	CGS001-6757	SSX2	-			
1772	72.78	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
1773	72.75	oe	ccsbBroad304_01701	TPI1	-			
1774	72.74	kd	CGS001-664	BNIP3	-			
1775	72.71	oe	ccsbBroad304_02368	TIMM17B	-			
1776	72.59	kd	CGS001-29978	UBQLN2	Ubiquilin family			
1777	72.58	kd	CGS001-11188	NISCH	-			
1778	72.58	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
1779	72.54	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
1780	72.51	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
1781	72.5	kd	CGS001-8270	LAGE3	-			
1782	72.42	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
1783	72.41	kd	CGS001-163688	CALML6	EF-hand domain containing			
1784	72.39	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
1785	72.38	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
1786	72.26	cc		Benzodiazepine receptor agonist	-			
1787	72.17	oe	ccsbBroad304_07478	CCP110	-			
1788	72.13	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
1789	72.11	kd	CGS001-2834	PRLHR	GPCR / Class A : RF amide peptide receptors			
1790	72.1	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
1791	72.09	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
1792	72.09	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
1793	72.08	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
1794	72.08	kd	CGS001-10672	GNA13	-			
1795	72.08	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
1796	72.02	kd	CGS001-6676	SPAG4	-			
1797	71.97	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
1798	71.91	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
1799	71.9	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
1800	71.85	kd	CGS001-55604	LRRC16A	-			
1801	71.75	kd	CGS001-10673	TNFSF13B	CD molecules			
1802	71.75	kd	CGS001-9183	ZW10	-			
1803	71.74	kd	CGS001-367	AR	Nuclear hormone receptors			
1804	71.72	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
1805	71.7	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
1806	71.69	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
1807	71.68	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
1808	71.67	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
1809	71.66	kd	CGS001-283	ANG	Ribonucleases, RNase A			
1810	71.59	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
1811	71.54	cc		HDAC inhibitor	-			
1812	71.51	kd	CGS001-57819	LSM2	-			
1813	71.48	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
1814	71.48	kd	CGS001-466	ATF1	basic leucine zipper proteins			
1815	71.47	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1816	71.32	kd	CGS001-9854	C2CD2L	-			
1817	71.31	kd	CGS001-57007	CXCR7	-			
1818	71.3	kd	CGS001-3376	IARS	Aminoacyl tRNA synthetases / Class I			
1819	71.3	kd	CGS001-57459	GATAD2B	GATA zinc finger domain containing			
1820	71.29	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
1821	71.27	kd	CGS001-55324	ABCF3	ATP binding cassette transporters / subfamily F			
1822	71.24	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
1823	71.23	cp	BRD-A79314293	cephalosporanic-acid	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1824	71.2	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
1825	71.17	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
1826	71.14	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1827	71.12	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1828	71.09	kd	CGS001-54566	EPB41L4B	-			
1829	71.09	kd	CGS001-1147	CHUK	IKK family			
1830	71.07	oe	ccsbBroad304_01371	RALA	-			
1831	71.06	kd	CGS001-6675	UAP1	-			
1832	71.02	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
1833	70.99	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
1834	70.86	kd	CGS001-2920	CXCL2	Endogenous ligands			
1835	70.84	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
1836	70.83	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
1837	70.77	oe	ccsbBroad304_06745	PNN	-			
1838	70.74	kd	CGS001-10135	NAMPT	-			
1839	70.74	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
1840	70.67	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
1841	70.59	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1842	70.58	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
1843	70.57	kd	CGS001-10392	NOD1	Nucleotide-binding domain and leucine rich repeat containing			
1844	70.56	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
1845	70.53	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
1846	70.53	kd	CGS001-192669	EIF2C3	-			
1847	70.52	kd	CGS001-4292	MLH1	-			
1848	70.44	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
1849	70.42	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
1850	70.42	kd	CGS001-9815	GIT2	Ankyrin repeat domain containing			
1851	70.41	oe	ccsbBroad304_01560	SNAPC1	-			
1852	70.4	kd	CGS001-11129	CLASRP	-			
1853	70.36	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
1854	70.29	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
1855	70.25	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
1856	70.24	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
1857	70.22	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
1858	70.21	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
1859	70.17	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
1860	70.17	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
1861	70.16	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
1862	70.15	kd	CGS001-4927	NUP88	-			
1863	70.13	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
1864	70.12	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
1865	69.97	oe	ccsbBroad304_02414	IRF9	-			
1866	69.97	kd	CGS001-11112	HIBADH	-			
1867	69.95	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
1868	69.93	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
1869	69.83	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
1870	69.79	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
1871	69.78	kd	CGS001-9034	CCRL2	Chemokine receptors			
1872	69.77	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
1873	69.76	kd	CGS001-5813	PURA	-			
1874	69.73	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
1875	69.71	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
1876	69.7	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
1877	69.69	kd	CGS001-23530	NNT	-			
1878	69.66	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
1879	69.62	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
1880	69.51	kd	CGS001-8864	PER2	-			
1881	69.46	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1882	69.43	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
1883	69.42	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
1884	69.41	kd	CGS001-5442	POLRMT	-			
1885	69.41	kd	CGS001-4798	NFRKB	INO80 complex subunits			
1886	69.36	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
1887	69.27	cc		Sterol demethylase inhibitor	-			
1888	69.25	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
1889	69.23	kd	CGS001-84647	PLA2G12B	-			
1890	69.13	kd	CGS001-1545	CYP1B1	Cytochrome P450s			
1891	69.11	kd	CGS001-10971	YWHAQ	-			
1892	69.08	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
1893	69.07	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
1894	69.05	oe	ccsbBroad304_04775	NTAN1	-			
1895	69.04	kd	CGS001-6793	STK10	SLK subfamily			
1896	69.03	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
1897	69.03	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
1898	68.94	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
1899	68.81	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
1900	68.76	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
1901	68.76	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1902	68.73	kd	CGS001-80347	COASY	-			
1903	68.68	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1904	68.64	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
1905	68.55	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
1906	68.54	kd	CGS001-253260	RICTOR	-			
1907	68.54	kd	CGS001-2882	GPX7	-			
1908	68.48	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
1909	68.46	kd	CGS001-2817	GPC1	Proteoglycans / Cell Surface : Glypicans			
1910	68.34	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
1911	68.33	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
1912	68.28	kd	CGS001-5469	MED1	-			
1913	68.25	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
1914	68.22	oe	ccsbBroad304_00231	CBFB	-			
1915	68.18	kd	CGS001-572	BAD	-			
1916	68.18	kd	CGS001-573	BAG1	-			
1917	68.16	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
1918	68.14	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
1919	68.06	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
1920	67.89	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
1921	67.82	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
1922	67.81	kd	CGS001-169841	ZNF169	Zinc fingers, C2H2-type			
1923	67.8	kd	CGS001-10745	PHTF1	-			
1924	67.78	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
1925	67.74	oe	ccsbBroad304_06975	SMARCC2	-			
1926	67.66	oe	ccsbBroad304_03191	NOSIP	-			
1927	67.64	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
1928	67.59	cc		C2 domain containing protein kinases LOF	-			
1929	67.59	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
1930	67.58	kd	CGS001-6767	ST13	Tetratricopeptide (TTC) repeat domain containing			
1931	67.5	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
1932	67.49	kd	CGS001-3373	HYAL1	-			
1933	67.48	oe	ccsbBroad304_07511	KIF14	Kinesins			
1934	67.47	kd	CGS001-169792	GLIS3	Zinc fingers, C2H2-type			
1935	67.46	oe	ccsbBroad304_06350	HAL	-			
1936	67.4	cc		PKC activator	-			
1937	67.4	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
1938	67.4	kd	CGS001-27109	ATP5S	-			
1939	67.38	oe	ccsbBroad304_02416	TUBB4B	-			
1940	67.34	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
1941	67.33	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
1942	67.29	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
1943	67.29	kd	CGS001-54807	ZNF586	Zinc fingers, C2H2-type			
1944	67.28	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
1945	67.24	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
1946	67.15	oe	ccsbBroad304_01374	RAP1A	-			
1947	67.14	kd	CGS001-57657	HCN3	Cyclic nucleotide-regulated channels			
1948	67.12	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
1949	67.12	kd	CGS001-6197	RPS6KA3	RSK subfamily			
1950	67.1	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
1951	67.04	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
1952	67.01	kd	CGS001-23149	FCHO1	-			
1953	66.98	kd	CGS001-4316	MMP7	Matrix metallopeptidase			
1954	66.93	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
1955	66.9	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
1956	66.9	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1957	66.89	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
1958	66.88	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
1959	66.88	oe	ccsbBroad304_01672	TIMP2	-			
1960	66.84	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
1961	66.84	kd	CGS001-2244	FGB	Endogenous ligands			
1962	66.75	kd	CGS001-10397	NDRG1	-			
1963	66.66	kd	CGS001-6926	TBX3	T-boxes			
1964	66.66	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
1965	66.65	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
1966	66.6	kd	CGS001-3778	KCNMA1	Calcium-activated potassium channels			
1967	66.6	kd	CGS001-427	ASAH1	Acid ceramidase			
1968	66.59	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
1969	66.55	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
1970	66.51	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
1971	66.48	kd	CGS001-9847	KIAA0528	-			
1972	66.48	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1973	66.44	kd	CGS001-57326	PBXIP1	-			
1974	66.44	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
1975	66.44	kd	CGS001-3693	ITGB5	Integrins			
1976	66.44	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
1977	66.36	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
1978	66.32	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
1979	66.32	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
1980	66.28	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
1981	66.26	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
1982	66.23	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
1983	66.15	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
1984	66.08	kd	CGS001-6342	SCP2	-			
1985	66.08	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
1986	66.05	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
1987	66.03	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
1988	65.98	kd	CGS001-56139	PCDHA10	Cadherins / Protocadherins : Clustered			
1989	65.97	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
1990	65.97	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
1991	65.92	kd	CGS001-1493	CTLA4	CD molecules			
1992	65.87	kd	CGS001-58533	SNX6	Sorting nexins			
1993	65.85	kd	CGS001-1736	DKC1	-			
1994	65.83	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
1995	65.82	oe	ccsbBroad304_03415	GFOD1	-			
1996	65.81	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
1997	65.75	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
1998	65.74	kd	CGS001-3593	IL12B	Interleukins and interleukin receptors			
1999	65.7	oe	ccsbBroad304_02534	UTP14A	-			
2000	65.7	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
2001	65.64	kd	CGS001-51495	PTPLAD1	-			
2002	65.62	kd	CGS001-9429	ABCG2	ATP binding cassette transporters / subfamily G			
2003	65.54	kd	CGS001-7353	UFD1L	-			
2004	65.52	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
2005	65.4	kd	CGS001-5446	PON3	Paraoxonases			
2006	65.39	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
2007	65.36	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
2008	65.3	cp	BRD-K00532621	midazolam	Benzodiazepine receptor agonist		CYP3A5, CYP3A7, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3	Benzodiazepine receptor agonist
2009	65.3	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
2010	65.26	kd	CGS001-6304	SATB1	Homeoboxes / CUT class			
2011	65.26	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
2012	65.25	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
2013	65.21	cp	BRD-K01649396	indatraline	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine transporter inhibitor
2014	65.16	kd	CGS001-11154	AP4S1	-			
2015	65.13	kd	CGS001-1737	DLAT	-			
2016	65.12	kd	CGS001-1874	E2F4	-			
2017	65.11	kd	CGS001-2592	GALT	-			
2018	65.06	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
2019	65.06	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
2020	65.05	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
2021	64.94	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
2022	64.94	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
2023	64.91	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
2024	64.89	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
2025	64.88	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
2026	64.85	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
2027	64.78	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
2028	64.75	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
2029	64.65	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
2030	64.62	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
2031	64.57	kd	CGS001-3998	LMAN1	-			
2032	64.54	cp	BRD-K10670311	sulfasalazine	Antirheumatic		PTGS1, PTGS2, ACAT1, ALOX5, CHUK, IKBKB, PLA2G1B, PPARG, SLC46A1, SLC7A11, TBXAS1	Antirheumatic, NFkB pathway inhibitor
2033	64.52	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2034	64.5	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
2035	64.49	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
2036	64.46	oe	ccsbBroad304_03850	TRIB3	Trbl family			
2037	64.46	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
2038	64.45	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
2039	64.44	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
2040	64.43	oe	ccsbBroad304_06235	G6PD	-			
2041	64.43	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
2042	64.36	kd	CGS001-150094	SIK1	QIK subfamily			
2043	64.31	kd	CGS001-7155	TOP2B	DNA Topoisomerases			
2044	64.27	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
2045	64.26	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
2046	64.22	kd	CGS001-8453	CUL2	-			
2047	64.21	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
2048	64.2	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
2049	64.12	oe	ccsbBroad304_03618	OSGEP	-			
2050	64.11	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
2051	64.08	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
2052	64.04	cc		GPCR Subset GOF	-			
2053	64.04	oe	ccsbBroad304_01748	UFD1L	-			
2054	64.02	kd	CGS001-7052	TGM2	Transglutaminases			
2055	63.97	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2056	63.9	kd	CGS001-7343	UBTF	-			
2057	63.88	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
2058	63.87	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
2059	63.8	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
2060	63.8	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
2061	63.68	kd	CGS001-563	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
2062	63.67	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
2063	63.66	oe	ccsbBroad304_09708	PNLDC1	-			
2064	63.65	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
2065	63.65	kd	CGS001-3032	HADHB	-			
2066	63.63	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
2067	63.59	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
2068	63.59	oe	ccsbBroad304_06172	EPS8	-			
2069	63.48	kd	CGS001-83694	RPS6KL1	RSKL family			
2070	63.46	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
2071	63.38	kd	CGS001-3455	IFNAR2	Interferon receptor family			
2072	63.31	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
2073	63.28	oe	ccsbBroad304_02115	PTTG1	-			
2074	63.26	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
2075	63.25	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
2076	63.21	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
2077	63.21	kd	CGS001-467	ATF3	basic leucine zipper proteins			
2078	63.14	kd	CGS001-6832	SUPV3L1	-			
2079	63.13	kd	CGS001-11343	MGLL	Endocannabinoid turnover			
2080	63.09	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
2081	63.07	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
2082	63.02	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
2083	63.01	kd	CGS001-1950	EGF	-			
2084	63	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
2085	62.92	cp	BRD-A70083328	secnidazole	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Microtubule inhibitor, Antiprotozoal
2086	62.88	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
2087	62.85	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
2088	62.85	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
2089	62.84	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
2090	62.83	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
2091	62.81	oe	ccsbBroad304_00250	CD19	CD molecules			
2092	62.81	oe	ccsbBroad304_00795	HSF2	-			
2093	62.81	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2094	62.79	oe	ccsbBroad304_06820	PTS	-			
2095	62.75	oe	ccsbBroad304_05194	LIPH	-			
2096	62.74	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
2097	62.74	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
2098	62.68	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
2099	62.66	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
2100	62.66	kd	CGS001-10765	KDM5B	Histone demethylases			
2101	62.65	kd	CGS001-6595	SMARCA2	Non-enzymatic BRD containing proteins			
2102	62.63	kd	CGS001-7727	ZNF174	Zinc fingers, C2H2-type			
2103	62.61	kd	CGS001-64376	IKZF5	IKAROS zinc fingers			
2104	62.58	kd	CGS001-648	BMI1	Polycomb group ring fingers			
2105	62.55	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
2106	62.52	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
2107	62.43	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
2108	62.35	kd	CGS001-5108	PCM1	-			
2109	62.29	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2110	62.25	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
2111	62.22	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
2112	62.22	kd	CGS001-7728	ZNF175	Zinc fingers, C2H2-type			
2113	62.13	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
2114	62.11	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
2115	62.06	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
2116	62.03	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
2117	61.95	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
2118	61.94	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
2119	61.93	kd	CGS001-6732	SRPK1	SRPK family			
2120	61.9	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
2121	61.89	kd	CGS001-79001	VKORC1	Oxidoreductases			
2122	61.83	kd	CGS001-54957	TXNL4B	-			
2123	61.78	kd	CGS001-999	CDH1	CD molecules			
2124	61.77	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
2125	61.7	kd	CGS001-3939	LDHA	-			
2126	61.67	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
2127	61.67	kd	CGS001-8193	DPF1	Zinc fingers, PHD-type			
2128	61.66	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
2129	61.63	kd	CGS001-23242	COBL	-			
2130	61.61	kd	CGS001-2172	FABP6	Fatty acid binding protein family			
2131	61.56	cp	BRD-K70883034	nimetazepam	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA receptor agonist
2132	61.46	kd	CGS001-87	ACTN1	EF-hand domain containing			
2133	61.4	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
2134	61.39	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
2135	61.36	oe	ccsbBroad304_03767	TOMM22	-			
2136	61.31	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
2137	61.28	oe	ccsbBroad304_06292	GNAI2	-			
2138	61.25	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
2139	61.2	kd	CGS001-57019	CIAPIN1	-			
2140	61.13	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
2141	61.12	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
2142	61.09	oe	ccsbBroad304_08898	TRAK2	-			
2143	61.07	kd	CGS001-4232	MEST	-			
2144	61.03	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
2145	61.02	kd	CGS001-6050	RNH1	-			
2146	61.01	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
2147	60.98	kd	CGS001-5338	PLD2	Hydrolases			
2148	60.97	cc		X linked mental retardation group 2 LOF	-			
2149	60.97	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
2150	60.95	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
2151	60.92	kd	CGS001-51002	TPRKB	-			
2152	60.91	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
2153	60.9	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
2154	60.89	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
2155	60.85	kd	CGS001-5096	PCCB	Carboxylases			
2156	60.85	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
2157	60.79	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
2158	60.76	oe	ccsbBroad304_04170	PANK2	-			
2159	60.76	kd	CGS001-3281	HSBP1	-			
2160	60.75	kd	CGS001-5627	PROS1	-			
2161	60.72	kd	CGS001-81611	ANP32E	ANP32 acidic nuclear phosphoproteins			
2162	60.68	kd	CGS001-7484	WNT9B	Wingless-type MMTV integration sites			
2163	60.63	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
2164	60.6	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
2165	60.57	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
2166	60.54	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
2167	60.51	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
2168	60.51	kd	CGS001-391013	PLA2G2C	-			
2169	60.5	kd	CGS001-3927	LASP1	-			
2170	60.43	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
2171	60.41	kd	CGS001-79862	ZNF669	Zinc fingers, C2H2-type			
2172	60.39	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
2173	60.39	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
2174	60.38	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
2175	60.36	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
2176	60.35	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
2177	60.31	oe	ccsbBroad304_00147	BAG1	-			
2178	60.3	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
2179	60.22	kd	CGS001-140612	ZFP28	Zinc fingers, C2H2-type			
2180	60.09	oe	ccsbBroad304_02484	PAICS	-			
2181	59.97	kd	CGS001-5613	PRKX	Protein kinase A			
2182	59.94	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
2183	59.91	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
2184	59.88	kd	CGS001-3579	CXCR2	Chemokine receptors			
2185	59.87	kd	CGS001-538	ATP7A	ATPases / P-type			
2186	59.87	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
2187	59.86	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
2188	59.85	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
2189	59.84	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
2190	59.83	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
2191	59.75	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2192	59.67	kd	CGS001-5036	PA2G4	-			
2193	59.63	kd	CGS001-51079	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
2194	59.63	kd	CGS001-29947	DNMT3L	-			
2195	59.57	oe	ccsbBroad304_01203	PIM1	PIM family			
2196	59.56	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
2197	59.56	kd	CGS001-688	KLF5	Kruppel-like transcription factors			
2198	59.53	kd	CGS001-5105	PCK1	-			
2199	59.5	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
2200	59.49	kd	CGS001-1345	COX6C	Mitochondrial respiratory chain complex			
2201	59.45	kd	CGS001-23139	MAST2	MAST family			
2202	59.45	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
2203	59.41	kd	CGS001-11315	PARK7	Parkinson disease			
2204	59.38	kd	CGS001-8905	AP1S2	-			
2205	59.32	oe	ccsbBroad304_02955	MYCBP	-			
2206	59.27	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
2207	59.21	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
2208	59.2	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
2209	59.13	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
2210	59.11	kd	CGS001-9870	KIAA0317	-			
2211	59.06	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
2212	59.05	cc		Cannabinoid receptor agonist	-			
2213	59.05	kd	CGS001-4507	MTAP	-			
2214	59.05	kd	CGS001-51601	LIPT1	-			
2215	59	kd	CGS001-397	ARHGDIB	Endogenous ligands			
2216	58.97	cp	BRD-A80928489	1-monopalmitin	P-glycoprotein inhibitor		ABCB1	P-glycoprotein inhibitor
2217	58.96	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
2218	58.9	oe	ccsbBroad304_06671	OPA1	-			
2219	58.89	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
2220	58.8	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
2221	58.79	kd	CGS001-3958	LGALS3	Endogenous ligands			
2222	58.72	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
2223	58.7	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2224	58.58	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
2225	58.57	kd	CGS001-6277	S100A6	EF-hand domain containing			
2226	58.57	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2227	58.54	kd	CGS001-22908	SACM1L	-			
2228	58.53	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
2229	58.52	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
2230	58.51	cc		Targets of VEGFR inhibitors GOF	-			
2231	58.49	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
2232	58.48	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
2233	58.48	kd	CGS001-23161	SNX13	Sorting nexins			
2234	58.26	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
2235	58.25	oe	ccsbBroad304_07275	PSMG1	-			
2236	58.21	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
2237	58.16	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
2238	58.14	kd	CGS001-10670	RRAGA	-			
2239	58.06	kd	CGS001-375449	MAST4	MAST family			
2240	58.04	kd	CGS001-23534	TNPO3	Importins			
2241	58.03	kd	CGS001-10400	PEMT	-			
2242	58.01	kd	CGS001-6621	SNAPC4	-			
2243	57.91	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
2244	57.89	cp	BRD-K85925969	zalcitabine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
2245	57.79	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
2246	57.66	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
2247	57.6	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
2248	57.59	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
2249	57.57	kd	CGS001-5460	POU5F1	Homeoboxes / POU class			
2250	57.56	kd	CGS001-10606	PAICS	-			
2251	57.5	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
2252	57.42	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
2253	57.41	oe	ccsbBroad304_02432	IFI30	-			
2254	57.4	oe	ccsbBroad304_03433	DDIT4	-			
2255	57.31	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
2256	57.31	oe	ccsbBroad304_02501	DCTN6	-			
2257	57.13	kd	CGS001-163486	DENND1B	DENN/MADD domain containing			
2258	57.01	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
2259	56.99	oe	ccsbBroad304_04257	SPRY4	-			
2260	56.99	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
2261	56.97	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
2262	56.95	oe	ccsbBroad304_04292	INHBE	-			
2263	56.93	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
2264	56.85	kd	CGS001-10123	ARL4C	ADP-ribosylation factors			
2265	56.84	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
2266	56.79	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
2267	56.73	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
2268	56.72	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
2269	56.64	oe	ccsbBroad304_00783	HPRT1	-			
2270	56.61	oe	ccsbBroad304_01527	SGK1	SGK family			
2271	56.55	kd	CGS001-10295	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
2272	56.54	oe	ccsbBroad304_06777	PRNP	CD molecules			
2273	56.52	oe	ccsbBroad304_09284	UBE3B	-			
2274	56.51	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
2275	56.51	oe	ccsbBroad304_04471	C5ORF62	-			
2276	56.45	kd	CGS001-283450	C12ORF51	-			
2277	56.42	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
2278	56.4	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2279	56.36	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
2280	56.3	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
2281	56.29	cc		NADH ubiquinone oxidoreductase supernumerary subunits LOF	-			
2282	56.26	kd	CGS001-7158	TP53BP1	-			
2283	56.24	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
2284	56.2	oe	ccsbBroad304_01034	MSH2	-			
2285	56.2	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
2286	56.2	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2287	56.16	oe	ccsbBroad304_10846	GGT1	CD molecules			
2288	56.07	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
2289	56.05	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
2290	56.03	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
2291	55.99	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
2292	55.96	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
2293	55.89	kd	CGS001-80351	TNKS2	Ankyrin repeat domain containing			
2294	55.82	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
2295	55.78	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
2296	55.75	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
2297	55.73	kd	CGS001-6453	ITSN1	Rho guanine nucleotide exchange factors			
2298	55.72	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2299	55.64	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
2300	55.58	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
2301	55.56	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
2302	55.56	kd	CGS001-2717	GLA	-			
2303	55.54	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
2304	55.54	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
2305	55.4	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2306	55.35	kd	CGS001-4724	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
2307	55.31	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
2308	55.3	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
2309	55.25	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
2310	55.21	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
2311	55.19	kd	CGS001-29916	SNX11	Sorting nexins			
2312	55.15	kd	CGS001-91433	RCCD1	-			
2313	55.12	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
2314	55.1	kd	CGS001-115201	ATG4A	-			
2315	55.06	kd	CGS001-116535	MRGPRF	GPCR / Class A : Orphans			
2316	54.97	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
2317	54.92	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
2318	54.92	kd	CGS001-29763	PACSIN3	-			
2319	54.91	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
2320	54.88	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
2321	54.85	kd	CGS001-5925	RB1	Endogenous ligands			
2322	54.83	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
2323	54.83	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
2324	54.82	kd	CGS001-4610	MYCL1	-			
2325	54.81	kd	CGS001-1201	CLN3	-			
2326	54.78	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
2327	54.66	oe	ccsbBroad304_06992	SRC	Src family			
2328	54.65	kd	CGS001-699	BUB1	Bub family			
2329	54.64	kd	CGS001-200081	TXLNA	-			
2330	54.63	kd	CGS001-79174	CRELD2	-			
2331	54.57	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
2332	54.53	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
2333	54.53	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
2334	54.5	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2335	54.46	kd	CGS001-4671	NAIP	Inhibitors of apoptosis (IAP) protein family			
2336	54.43	kd	CGS001-1820	ARID3A	-			
2337	54.4	oe	ccsbBroad304_00658	GNG5	-			
2338	54.38	kd	CGS001-399664	MEX3D	Mex-3 homologs			
2339	54.36	oe	ccsbBroad304_01623	SUPT4H1	-			
2340	54.36	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
2341	54.33	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
2342	54.25	kd	CGS001-995	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2343	54.16	oe	ccsbBroad304_01723	TTK	TTK family			
2344	54.14	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
2345	54.09	kd	CGS001-5194	PEX13	-			
2346	54.08	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
2347	54.05	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
2348	53.94	oe	ccsbBroad304_07217	AXIN2	-			
2349	53.86	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
2350	53.82	kd	CGS001-10626	TRIM16	Tripartite motif containing			
2351	53.64	oe	ccsbBroad304_07727	LIAS	-			
2352	53.62	kd	CGS001-5106	PCK2	-			
2353	53.62	kd	CGS001-51742	ARID4B	-			
2354	53.6	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
2355	53.51	kd	CGS001-9189	ZBED1	Pseudoautosomal regions / PAR1			
2356	53.45	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
2357	53.42	kd	CGS001-2237	FEN1	-			
2358	53.4	kd	CGS001-2203	FBP1	-			
2359	53.38	kd	CGS001-30001	ERO1L	-			
2360	53.16	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
2361	53.16	oe	ccsbBroad304_06998	SRPK1	SRPK family			
2362	53.01	cp	BRD-K11630072	carmofur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
2363	53.01	kd	CGS001-7032	TFF2	-			
2364	52.85	kd	CGS001-253430	IPMK	-			
2365	52.75	oe	ccsbBroad304_03848	METTL14	-			
2366	52.72	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
2367	52.68	kd	CGS001-475	ATOX1	-			
2368	52.61	kd	CGS001-4904	YBX1	-			
2369	52.52	kd	CGS001-53834	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
2370	52.47	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
2371	52.44	kd	CGS001-10112	KIF20A	Kinesins			
2372	52.43	kd	CGS001-55770	EXOC2	-			
2373	52.37	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
2374	52.25	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
2375	52.18	kd	CGS001-6827	SUPT4H1	-			
2376	52.1	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
2377	52.05	kd	CGS001-6917	TCEA1	General transcription factors			
2378	52.05	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
2379	51.99	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
2380	51.97	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
2381	51.96	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
2382	51.91	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
2383	51.85	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
2384	51.82	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
2385	51.79	kd	CGS001-25948	KBTBD2	BTB/POZ domain containing			
2386	51.78	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
2387	51.68	kd	CGS001-7247	TSN	-			
2388	51.63	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
2389	51.57	oe	ccsbBroad304_07851	FAM120A	-			
2390	51.54	oe	ccsbBroad304_06654	NPM1	-			
2391	51.53	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
2392	51.48	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
2393	51.44	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
2394	51.41	oe	ccsbBroad304_07884	RYBP	-			
2395	51.41	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
2396	51.39	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
2397	51.31	kd	CGS001-2745	GLRX	-			
2398	51.3	kd	CGS001-7342	UBP1	-			
2399	51.3	kd	CGS001-2805	GOT1	-			
2400	51.29	kd	CGS001-9975	NR1D2	Rev-Erb receptors			
2401	51.27	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
2402	51.24	oe	ccsbBroad304_00161	BID	Endogenous ligands			
2403	51.22	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
2404	51.22	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
2405	51.2	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
2406	51.12	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
2407	51.11	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
2408	51.01	oe	ccsbBroad304_06367	HK1	-			
2409	50.91	cc		FOS transcription factor family GOF	-			
2410	50.89	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2411	50.84	kd	CGS001-8569	MKNK1	MKN subfamily			
2412	50.83	kd	CGS001-2562	GABRB3	GABA receptors			
2413	50.81	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
2414	50.76	kd	CGS001-2550	GABBR1	GABA receptors			
2415	50.75	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2416	50.72	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
2417	50.64	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
2418	50.6	kd	CGS001-29928	TIMM22	-			
2419	50.53	oe	ccsbBroad304_03554	NAT10	-			
2420	50.51	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
2421	50.48	kd	CGS001-54677	CROT	-			
2422	50.45	kd	CGS001-122402	TDRD9	Tudor domain containing			
2423	50.44	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
2424	50.36	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2425	50.31	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
2426	50.28	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
2427	50.25	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
2428	50.23	kd	CGS001-8566	PDXK	-			
2429	50.22	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
2430	50.18	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
2431	50.17	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
2432	50.08	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
2433	50.08	kd	CGS001-23378	RRP8	-			
2434	50.06	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
2435	50.01	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
2436	49.95	kd	CGS001-55139	ANKZF1	Ankyrin repeat domain containing			
2437	49.91	kd	CGS001-7090	TLE3	WD repeat domain containing			
2438	49.9	kd	CGS001-1827	RCAN1	-			
2439	49.88	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
2440	49.69	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2441	49.69	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
2442	49.66	kd	CGS001-1362	CPD	Carboxypeptidase A			
2443	49.57	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
2444	49.56	cc		FGFR inhibitor	-			
2445	49.56	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
2446	49.54	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
2447	49.52	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
2448	49.48	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
2449	49.45	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
2450	49.41	kd	CGS001-6461	SHB	SH2 domain containing			
2451	49.37	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
2452	49.3	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
2453	49.29	kd	CGS001-4121	MAN1A1	-			
2454	49.18	oe	ccsbBroad304_00033	ADSS	-			
2455	49.16	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
2456	49.13	kd	CGS001-79080	CCDC86	-			
2457	49.12	oe	ccsbBroad304_03874	UBL5	-			
2458	49.03	kd	CGS001-51447	IP6K2	-			
2459	49	oe	ccsbBroad304_08322	UFM1	-			
2460	48.95	oe	ccsbBroad304_02578	EBNA1BP2	-			
2461	48.94	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
2462	48.93	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
2463	48.92	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
2464	48.85	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
2465	48.85	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
2466	48.83	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
2467	48.83	kd	CGS001-24138	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
2468	48.82	kd	CGS001-65243	ZNF643	-			
2469	48.76	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
2470	48.76	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
2471	48.7	kd	CGS001-29116	MYLIP	-			
2472	48.69	oe	ccsbBroad304_08684	CXCR7	-			
2473	48.65	oe	ccsbBroad304_07506	UBAP2L	-			
2474	48.61	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
2475	48.59	kd	CGS001-10059	DNM1L	-			
2476	48.54	kd	CGS001-440387	CTRB2	-			
2477	48.43	kd	CGS001-28985	MCTS1	-			
2478	48.41	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
2479	48.34	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
2480	48.31	kd	CGS001-117581	TWIST2	Basic helix-loop-helix proteins			
2481	48.23	kd	CGS001-10128	LRPPRC	-			
2482	48.15	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2483	48.1	oe	ccsbBroad304_02589	COPS5	-			
2484	48.1	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
2485	48.04	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
2486	48	oe	ccsbBroad304_03450	TMED9	-			
2487	47.99	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
2488	47.96	kd	CGS001-79712	GTDC1	Glycosyltransferase group 1 domain containing			
2489	47.92	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
2490	47.92	kd	CGS001-6541	SLC7A1	SLC7 family			
2491	47.84	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
2492	47.83	kd	CGS001-1445	CSK	Csk family			
2493	47.81	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
2494	47.79	oe	ccsbBroad304_02738	RRS1	-			
2495	47.75	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
2496	47.71	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
2497	47.49	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
2498	47.49	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
2499	47.44	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
2500	47.36	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
2501	47.32	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
2502	47.31	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
2503	47.29	oe	ccsbBroad304_00418	CD55	CD molecules			
2504	47.29	kd	CGS001-57720	GPR107	GPCR / Unclassified : 7TM orphan receptors			
2505	47.28	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
2506	47.27	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
2507	47.23	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
2508	47.13	kd	CGS001-861	RUNX1	-			
2509	47.11	oe	ccsbBroad304_04387	MKI67IP	-			
2510	47.09	kd	CGS001-9380	GRHPR	-			
2511	46.82	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2512	46.79	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
2513	46.78	kd	CGS001-5053	PAH	Amino acid hydroxylases			
2514	46.77	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
2515	46.73	kd	CGS001-11182	SLC2A6	Solute carriers			
2516	46.7	kd	CGS001-2629	GBA	-			
2517	46.66	kd	CGS001-3094	HINT1	-			
2518	46.63	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
2519	46.62	kd	CGS001-8829	NRP1	CD molecules			
2520	46.61	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
2521	46.6	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
2522	46.6	kd	CGS001-5277	PIGA	Glycosyltransferase group 1 domain containing			
2523	46.58	kd	CGS001-55634	ZNF673	-			
2524	46.55	kd	CGS001-23536	ADAT1	-			
2525	46.49	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
2526	46.47	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
2527	46.43	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
2528	46.42	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
2529	46.4	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
2530	46.38	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
2531	46.34	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
2532	46.34	oe	ccsbBroad304_06494	KLRC1	CD molecules			
2533	46.26	oe	ccsbBroad304_03113	DSE	-			
2534	46.25	kd	CGS001-64319	FBRS	-			
2535	46.19	kd	CGS001-5577	PRKAR2B	Protein kinase A			
2536	46.18	kd	CGS001-7105	TSPAN6	Tetraspanins			
2537	46.17	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
2538	46.13	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
2539	46.1	kd	CGS001-5366	PMAIP1	-			
2540	46.1	kd	CGS001-5223	PGAM1	-			
2541	46.01	oe	ccsbBroad304_00572	FKBP3	-			
2542	45.99	kd	CGS001-51128	SAR1B	-			
2543	45.94	oe	ccsbBroad304_00510	EPHX2	-			
2544	45.93	kd	CGS001-51014	TMED7	-			
2545	45.89	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2546	45.8	oe	ccsbBroad304_07531	TANK	-			
2547	45.76	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
2548	45.71	kd	CGS001-5087	PBX1	Homeoboxes / TALE class			
2549	45.7	kd	CGS001-1855	DVL1	Dishevelled homologs			
2550	45.69	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
2551	45.68	kd	CGS001-102	ADAM10	ADAM metallopeptidase domain containing			
2552	45.66	cc		C2 domain containing LOF	-			
2553	45.6	kd	CGS001-6822	SULT2A1	Sulfotransferases, cytosolic			
2554	45.59	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
2555	45.57	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
2556	45.55	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
2557	45.54	kd	CGS001-1490	CTGF	-			
2558	45.52	kd	CGS001-23013	SPEN	RNA binding motif (RRM) containing			
2559	45.46	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
2560	45.39	kd	CGS001-79902	NUP85	-			
2561	45.38	kd	CGS001-5796	PTPRK	Receptor tyrosine phosphatases (RTP)			
2562	45.35	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
2563	45.35	kd	CGS001-4811	NID1	-			
2564	45.33	kd	CGS001-10096	ACTR3	-			
2565	45.27	oe	ccsbBroad304_00818	IDH3A	-			
2566	45.26	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2567	45.13	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
2568	45.11	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
2569	45.09	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
2570	45.04	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
2571	44.98	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
2572	44.98	kd	CGS001-896	CCND3	-			
2573	44.89	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
2574	44.89	kd	CGS001-51022	GLRX2	-			
2575	44.88	oe	ccsbBroad304_03853	LSM2	-			
2576	44.88	kd	CGS001-10398	MYL9	EF-hand domain containing			
2577	44.73	kd	CGS001-976	CD97	Adhesion Class GPCRs			
2578	44.65	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
2579	44.6	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
2580	44.55	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
2581	44.49	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
2582	44.48	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
2583	44.47	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
2584	44.47	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
2585	44.45	kd	CGS001-8878	SQSTM1	-			
2586	44.39	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
2587	44.39	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
2588	44.33	kd	CGS001-80274	SCUBE1	-			
2589	44.13	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
2590	44.1	oe	ccsbBroad304_09054	EGFL8	-			
2591	44.06	kd	CGS001-9541	CIR1	-			
2592	44.01	oe	ccsbBroad304_13813	ARAF	RAF family			
2593	43.99	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
2594	43.82	kd	CGS001-2	A2M	-			
2595	43.77	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
2596	43.77	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
2597	43.72	cp	BRD-K85503079	perospirone	Dopamine receptor antagonist		DRD2, HTR2A, DRD3, DRD4, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
2598	43.62	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
2599	43.62	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
2600	43.61	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
2601	43.59	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
2602	43.56	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
2603	43.55	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
2604	43.53	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2605	43.44	kd	CGS001-898	CCNE1	-			
2606	43.38	kd	CGS001-326	AIRE	Zinc fingers, PHD-type			
2607	43.3	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
2608	43.29	oe	ccsbBroad304_07923	LSM5	-			
2609	43.29	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
2610	43.27	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
2611	43.18	kd	CGS001-23621	BACE1	Pepsin			
2612	43.16	kd	CGS001-1376	CPT2	-			
2613	43.13	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
2614	43.13	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
2615	43.1	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
2616	43.05	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
2617	43	kd	CGS001-843	CASP10	Caspases			
2618	42.97	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2619	42.96	kd	CGS001-8233	ZRSR2	RNA binding motif (RRM) containing			
2620	42.83	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
2621	42.83	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
2622	42.79	oe	ccsbBroad304_03625	HIF1AN	-			
2623	42.78	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
2624	42.77	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
2625	42.75	oe	ccsbBroad304_06889	RPN2	-			
2626	42.67	kd	CGS001-3559	IL2RA	IL-2 receptor family			
2627	42.66	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
2628	42.65	kd	CGS001-5515	PPP2CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2629	42.59	cp	BRD-K63784565	BRD-K63784565	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
2630	42.5	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
2631	42.48	kd	CGS001-26036	ZNF451	Zinc fingers, C2H2-type			
2632	42.48	kd	CGS001-1879	EBF1	-			
2633	42.38	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
2634	42.33	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
2635	42.31	kd	CGS001-7323	UBE2D3	Ubiquitin-conjugating enzymes E2			
2636	42.29	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
2637	42.29	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
2638	42.28	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
2639	42.25	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
2640	42.21	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
2641	42.21	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
2642	42.05	kd	CGS001-10014	HDAC5	Histone deacetylases			
2643	42.03	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
2644	41.98	kd	CGS001-64087	MCCC2	-			
2645	41.97	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
2646	41.96	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
2647	41.95	kd	CGS001-10180	RBM6	G patch domain containing			
2648	41.93	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
2649	41.89	kd	CGS001-7157	TP53	-			
2650	41.73	kd	CGS001-1786	DNMT1	Methyltransferases			
2651	41.68	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
2652	41.65	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
2653	41.65	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
2654	41.59	kd	CGS001-8446	DUSP11	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2655	41.56	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
2656	41.55	kd	CGS001-26959	HBP1	-			
2657	41.52	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
2658	41.5	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
2659	41.48	kd	CGS001-5565	PRKAB2	AMPK subfamily			
2660	41.46	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
2661	41.42	kd	CGS001-10721	POLQ	DNA polymerases			
2662	41.39	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
2663	41.23	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
2664	41.21	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
2665	41.12	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
2666	41.11	oe	ccsbBroad304_00809	HUS1	-			
2667	41.06	kd	CGS001-1903	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
2668	41.03	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2669	40.92	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2670	40.9	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
2671	40.83	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
2672	40.73	kd	CGS001-57167	SALL4	Zinc fingers, C2H2-type			
2673	40.68	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
2674	40.58	oe	ccsbBroad304_05757	ACADS	-			
2675	40.53	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
2676	40.5	kd	CGS001-2138	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2677	40.4	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
2678	40.39	kd	CGS001-1605	DAG1	-			
2679	40.37	kd	CGS001-3053	SERPIND1	Serine (or cysteine) peptidase inhibitors			
2680	40.33	kd	CGS001-6773	STAT2	SH2 domain containing			
2681	40.32	oe	ccsbBroad304_06789	PSEN2	Presenilin			
2682	40.29	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
2683	40.26	kd	CGS001-25913	POT1	-			
2684	40.25	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
2685	40.23	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
2686	40.22	oe	ccsbBroad304_01624	SUPV3L1	-			
2687	40.22	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
2688	40.21	kd	CGS001-11179	ZNF277	-			
2689	40.17	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
2690	40.11	oe	ccsbBroad304_03739	NRIP3	-			
2691	40.11	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
2692	40.08	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
2693	40.02	oe	ccsbBroad304_02361	MFSD10	-			
2694	40	oe	ccsbBroad304_01131	OXCT1	-			
2695	39.98	kd	CGS001-10456	HAX1	-			
2696	39.95	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
2697	39.94	cc		Poly ADP ribose polymerases LOF	-			
2698	39.92	kd	CGS001-10969	EBNA1BP2	-			
2699	39.89	kd	CGS001-9587	MAD2L1BP	-			
2700	39.75	kd	CGS001-5581	PRKCE	Eta subfamily			
2701	39.72	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2702	39.68	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
2703	39.66	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
2704	39.61	kd	CGS001-10001	MED6	-			
2705	39.56	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
2706	39.44	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
2707	39.44	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
2708	39.41	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
2709	39.4	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
2710	39.39	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
2711	39.37	kd	CGS001-5479	PPIB	-			
2712	39.32	oe	ccsbBroad304_04202	MED28	-			
2713	39.22	kd	CGS001-1644	DDC	Catecholamine turnover			
2714	39.22	oe	ccsbBroad304_07119	UGP2	-			
2715	39.21	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
2716	39.06	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
2717	39.05	oe	ccsbBroad304_02566	MORF4L1	-			
2718	38.97	kd	CGS001-3659	IRF1	-			
2719	38.87	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
2720	38.83	kd	CGS001-2710	GK	Glycerol kinases			
2721	38.76	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
2722	38.75	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
2723	38.73	kd	CGS001-2770	GNAI1	-			
2724	38.72	kd	CGS001-4299	AFF1	-			
2725	38.67	kd	CGS001-3065	HDAC1	Histone deacetylases			
2726	38.64	cp	BRD-K59456551	methotrexate	Dihydrofolate reductase inhibitor		DHFR, AOX1, FOLR1, TYMS	Dihydrofolate reductase inhibitor
2727	38.56	kd	CGS001-8438	RAD54L	-			
2728	38.47	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
2729	38.42	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
2730	38.4	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
2731	38.39	cc		EMSY complex LOF	-			
2732	38.32	kd	CGS001-3799	KIF5B	Kinesins			
2733	38.27	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
2734	38.23	kd	CGS001-55012	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2735	38.19	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
2736	38.17	cp	BRD-A39390670	rabeprazole	ATPase inhibitor		ATP4A, CYP2C19	ATPase inhibitor, Gastrin inhibitor
2737	38.15	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
2738	38.04	kd	CGS001-8797	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
2739	38	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
2740	37.94	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
2741	37.9	kd	CGS001-5654	HTRA1	Serine peptidases / Serine peptidases			
2742	37.84	cp	BRD-A23359898	sibutramine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, CYP2B6, CYP2C19, CYP3A5	Serotonin reuptake inhibitor
2743	37.83	oe	ccsbBroad304_03533	CDCA8	-			
2744	37.82	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
2745	37.8	kd	CGS001-8802	SUCLG1	-			
2746	37.79	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
2747	37.78	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
2748	37.77	kd	CGS001-2184	FAH	-			
2749	37.75	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
2750	37.72	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
2751	37.43	kd	CGS001-5188	PET112	-			
2752	37.4	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
2753	37.39	kd	CGS001-1534	CYB561	Cytochrome b genes			
2754	37.35	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
2755	37.35	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2756	37.33	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
2757	37.27	kd	CGS001-259	AMBP	Lipocalins			
2758	37.2	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
2759	37.19	kd	CGS001-91392	ZNF502	Zinc fingers, C2H2-type			
2760	37.18	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
2761	37.14	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
2762	37.01	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
2763	36.89	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
2764	36.88	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
2765	36.88	cp	BRD-K18523449	mestanolone	Androgenic steroid			Androgenic steroid
2766	36.8	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
2767	36.71	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
2768	36.7	oe	ccsbBroad304_02838	SDF2L1	-			
2769	36.68	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2770	36.66	cp	BRD-K93618743	ipriflavone	Bone resorption inhibitor			Bone resorption inhibitor
2771	36.66	kd	CGS001-6887	TAL2	Basic helix-loop-helix proteins			
2772	36.65	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
2773	36.65	cp	BRD-A42423104	benproperine	Antitussive			Antitussive
2774	36.62	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
2775	36.62	kd	CGS001-9945	GFPT2	-			
2776	36.6	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
2777	36.54	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
2778	36.52	cc		Histone deacetylases LOF	-			
2779	36.52	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
2780	36.48	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
2781	36.42	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
2782	36.41	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2783	36.38	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
2784	36.35	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
2785	36.28	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
2786	36.26	kd	CGS001-23429	RYBP	-			
2787	36.21	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
2788	36.2	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
2789	36.19	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
2790	36.18	kd	CGS001-5049	PAFAH1B2	-			
2791	36.05	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2792	36	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
2793	35.95	kd	CGS001-7040	TGFB1	Endogenous ligands			
2794	35.94	kd	CGS001-55715	DOK4	Pleckstrin homology (PH) domain containing			
2795	35.91	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
2796	35.89	oe	ccsbBroad304_07704	SUB1	-			
2797	35.78	kd	CGS001-9447	AIM2	-			
2798	35.76	kd	CGS001-3251	HPRT1	-			
2799	35.7	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
2800	35.62	oe	ccsbBroad304_07875	SPECC1L	-			
2801	35.61	kd	CGS001-4267	CD99	CD molecules			
2802	35.53	oe	ccsbBroad304_06382	HMGCL	-			
2803	35.49	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
2804	35.45	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
2805	35.38	kd	CGS001-883	CCBL1	Hydrogen sulphide synthesis			
2806	35.31	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
2807	35.27	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
2808	35.27	kd	CGS001-9784	SNX17	Sorting nexins			
2809	35.23	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
2810	35.19	kd	CGS001-9559	VPS26A	-			
2811	35.16	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
2812	35.15	kd	CGS001-53836	GPR87	GPCR / Class A : Orphans			
2813	35.08	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
2814	35.06	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
2815	35.04	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
2816	34.97	kd	CGS001-2017	CTTN	-			
2817	34.81	kd	CGS001-5966	REL	NFkappaB transcription factor family			
2818	34.78	oe	ccsbBroad304_13891	LCK	Src family			
2819	34.76	kd	CGS001-1606	DGKA	EF-hand domain containing			
2820	34.58	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2821	34.58	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
2822	34.54	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
2823	34.49	kd	CGS001-873	CBR1	Prostaglandin synthases			
2824	34.39	oe	ccsbBroad304_08461	CDCA4	-			
2825	34.37	kd	CGS001-5887	RAD23B	-			
2826	34.32	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
2827	34.31	oe	ccsbBroad304_02576	MLLT11	-			
2828	34.23	cp	BRD-K50866992	tropisetron	Serotonin receptor antagonist		HTR3A, GLRA1, GLRA2, GLRB, HTR4	Serotonin receptor antagonist
2829	34.22	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
2830	34.22	kd	CGS001-5447	POR	-			
2831	34.17	kd	CGS001-89765	RSPH1	-			
2832	34.13	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
2833	34.12	oe	ccsbBroad304_07362	NMI	-			
2834	34.1	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
2835	34.09	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
2836	34.06	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
2837	34.03	oe	ccsbBroad304_00710	GUSB	-			
2838	34.02	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
2839	33.98	oe	ccsbBroad304_06720	PHYH	-			
2840	33.98	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
2841	33.98	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
2842	33.91	oe	ccsbBroad304_01398	RHEB	-			
2843	33.9	kd	CGS001-4090	SMAD5	SMADs			
2844	33.87	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
2845	33.86	cp	BRD-A16444946	acarbose	Glucosidase inhibitor		GAA, MGAM, AMY2A, SI	Glucosidase inhibitor
2846	33.84	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
2847	33.67	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
2848	33.63	kd	CGS001-5579	PRKCB	Alpha subfamily			
2849	33.54	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
2850	33.44	oe	ccsbBroad304_06290	GNA15	-			
2851	33.44	kd	CGS001-10196	PRMT3	Protein arginine N-methyltransferases			
2852	33.43	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
2853	33.42	oe	ccsbBroad304_03182	GLOD4	-			
2854	33.4	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
2855	33.39	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
2856	33.36	kd	CGS001-2729	GCLC	-			
2857	33.34	kd	CGS001-2932	GSK3B	GSK subfamily			
2858	33.28	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
2859	33.28	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
2860	33.23	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2861	33.22	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
2862	33.2	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
2863	33.2	kd	CGS001-51727	CMPK1	-			
2864	33.14	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
2865	33.14	kd	CGS001-5992	RFX4	-			
2866	33.06	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
2867	33.06	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
2868	33.06	kd	CGS001-3692	EIF6	-			
2869	33.03	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
2870	33	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
2871	32.98	kd	CGS001-11329	STK38	NDR family			
2872	32.97	kd	CGS001-2004	ELK3	ETS Transcription Factors			
2873	32.97	kd	CGS001-64077	LHPP	-			
2874	32.95	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
2875	32.94	kd	CGS001-60493	FASTKD5	-			
2876	32.92	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
2877	32.85	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
2878	32.77	kd	CGS001-25819	CCRN4L	-			
2879	32.73	kd	CGS001-2857	GPR34	GPCR / Class A : Orphans			
2880	32.69	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
2881	32.68	kd	CGS001-4129	MAOB	Catecholamine turnover			
2882	32.63	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
2883	32.57	kd	CGS001-11168	PSIP1	-			
2884	32.52	oe	ccsbBroad304_05931	CAPG	-			
2885	32.5	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2886	32.46	cp	BRD-K83144676	olmesartan	Angiotensin antagonist		AGTR1	Angiotensin antagonist
2887	32.35	kd	CGS001-10058	ABCB6	ATP binding cassette transporters / subfamily B			
2888	32.33	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
2889	32.25	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
2890	32.23	kd	CGS001-663	BNIP2	-			
2891	32.2	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
2892	32.13	cc		Mediator complex LOF	-			
2893	32.13	oe	ccsbBroad304_02964	TIMM9	-			
2894	32.12	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
2895	32.09	kd	CGS001-5004	ORM1	Lipocalins			
2896	32.06	kd	CGS001-3776	KCNK2	Two-P potassium channels			
2897	32.02	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
2898	31.99	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
2899	31.99	kd	CGS001-83933	HDAC10	Histone deacetylases			
2900	31.95	cp	BRD-A92630576	trimebutine	Opioid receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Opioid receptor agonist
2901	31.93	oe	ccsbBroad304_02884	POT1	-			
2902	31.89	kd	CGS001-58478	ENOPH1	-			
2903	31.85	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
2904	31.78	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
2905	31.77	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
2906	31.76	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
2907	31.7	kd	CGS001-5927	KDM5A	Histone demethylases			
2908	31.63	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
2909	31.61	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
2910	31.58	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
2911	31.56	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
2912	31.55	kd	CGS001-3570	IL6R	IL-6 receptor family			
2913	31.49	kd	CGS001-55127	HEATR1	-			
2914	31.44	kd	CGS001-23210	JMJD6	-			
2915	31.39	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
2916	31.39	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
2917	31.38	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
2918	31.35	oe	ccsbBroad304_00532	F11	Chymotrypsin			
2919	31.33	kd	CGS001-22934	RPIA	-			
2920	31.31	oe	ccsbBroad304_07605	LYPLA1	-			
2921	31.29	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
2922	31.26	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
2923	31.17	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
2924	31.17	kd	CGS001-57121	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2925	31.13	kd	CGS001-3676	ITGA4	Integrins			
2926	31.12	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
2927	31.11	kd	CGS001-4193	MDM2	-			
2928	31.04	kd	CGS001-10589	DRAP1	-			
2929	30.95	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
2930	30.93	oe	ccsbBroad304_03573	BRF2	-			
2931	30.92	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
2932	30.91	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
2933	30.86	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
2934	30.84	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
2935	30.83	kd	CGS001-3364	HUS1	-			
2936	30.78	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
2937	30.78	kd	CGS001-81539	SLC38A1	System A-like transporters			
2938	30.76	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
2939	30.73	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
2940	30.72	oe	ccsbBroad304_02737	JMJD6	-			
2941	30.71	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2942	30.65	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
2943	30.61	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
2944	30.61	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
2945	30.59	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
2946	30.58	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
2947	30.53	kd	CGS001-84878	ZBTB45	BTB/POZ domain containing			
2948	30.53	kd	CGS001-1802	DPH2	-			
2949	30.42	kd	CGS001-9903	KLHL21	BTB/POZ domain containing			
2950	30.39	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
2951	30.39	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
2952	30.36	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
2953	30.36	oe	ccsbBroad304_02551	CPSF4	-			
2954	30.31	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
2955	30.3	kd	CGS001-25836	NIPBL	-			
2956	30.2	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
2957	30.18	kd	CGS001-6199	RPS6KB2	p70 subfamily			
2958	30.15	kd	CGS001-1195	CLK1	CDC-like kinases			
2959	30.13	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
2960	30.09	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
2961	30.08	kd	CGS001-51071	DERA	-			
2962	30.07	kd	CGS001-64175	LEPRE1	-			
2963	30.07	kd	CGS001-8536	CAMK1	CAMK1 family			
2964	30.05	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
2965	30.04	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
2966	30.02	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
2967	30.01	oe	ccsbBroad304_07140	XPC	-			
2968	29.99	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
2969	29.95	kd	CGS001-2355	FOSL2	basic leucine zipper proteins			
2970	29.93	kd	CGS001-8649	LAMTOR3	-			
2971	29.93	kd	CGS001-64858	DCLRE1B	-			
2972	29.75	kd	CGS001-5269	SERPINB6	Serine (or cysteine) peptidase inhibitors			
2973	29.68	cc		Cyclin dependent kinases LOF	-			
2974	29.68	oe	ccsbBroad304_00038	AGL	-			
2975	29.63	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
2976	29.61	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
2977	29.56	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
2978	29.49	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
2979	29.44	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
2980	29.43	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
2981	29.4	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
2982	29.37	oe	ccsbBroad304_01215	PLAUR	CD molecules			
2983	29.35	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
2984	29.33	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
2985	29.33	kd	CGS001-1030	CDKN2B	-			
2986	29.31	oe	ccsbBroad304_08775	SQRDL	-			
2987	29.15	kd	CGS001-5906	RAP1A	-			
2988	29.15	kd	CGS001-5134	PDCD2	Zinc fingers, MYND-type			
2989	29.11	kd	CGS001-27113	BBC3	-			
2990	29.1	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
2991	29.08	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
2992	29.06	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
2993	29.01	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
2994	28.92	kd	CGS001-51530	ZC3HC1	Zinc fingers, C3HC-type			
2995	28.91	kd	CGS001-4125	MAN2B1	-			
2996	28.9	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
2997	28.9	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
2998	28.87	kd	CGS001-23635	SSBP2	-			
2999	28.8	kd	CGS001-1349	COX7B	Mitochondrial respiratory chain complex			
3000	28.76	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
3001	28.76	oe	ccsbBroad304_03122	RHOD	-			
3002	28.71	oe	ccsbBroad304_03129	ERO1L	-			
3003	28.65	kd	CGS001-167826	OLIG3	Basic helix-loop-helix proteins			
3004	28.64	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
3005	28.56	kd	CGS001-4144	MAT2A	-			
3006	28.56	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
3007	28.55	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
3008	28.48	kd	CGS001-55644	OSGEP	-			
3009	28.47	oe	ccsbBroad304_02002	RNMT	-			
3010	28.39	oe	ccsbBroad304_00725	HADHA	-			
3011	28.33	kd	CGS001-348	APOE	Apolipoproteins			
3012	28.23	kd	CGS001-7535	ZAP70	Syk family			
3013	28.21	cp	BRD-A94543220	bifonazole	Sterol demethylase inhibitor		CYP2B6	Sterol demethylase inhibitor
3014	28.2	oe	ccsbBroad304_03372	CAB39	-			
3015	28.14	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
3016	28.13	kd	CGS001-10975	UQCR11	Mitochondrial respiratory chain complex / Complex III			
3017	28.13	oe	ccsbBroad304_10431	HADHB	-			
3018	28.1	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
3019	28.03	kd	CGS001-162	AP1B1	-			
3020	28	oe	ccsbBroad304_02195	SPAG7	-			
3021	27.99	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
3022	27.98	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
3023	27.96	kd	CGS001-6804	STX1A	-			
3024	27.92	kd	CGS001-23710	GABARAPL1	-			
3025	27.91	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
3026	27.89	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
3027	27.81	kd	CGS001-7086	TKT	-			
3028	27.77	kd	CGS001-8893	EIF2B5	-			
3029	27.75	cp	BRD-K06817181	BRD-K06817181	JAK inhibitor		JAK2	JAK inhibitor
3030	27.67	kd	CGS001-28511	NKIRAS2	-			
3031	27.62	kd	CGS001-6196	RPS6KA2	RSK subfamily			
3032	27.6	kd	CGS001-4176	MCM7	-			
3033	27.58	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
3034	27.58	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
3035	27.57	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
3036	27.56	oe	ccsbBroad304_08386	SMOX	-			
3037	27.55	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
3038	27.51	kd	CGS001-1622	DBI	-			
3039	27.5	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
3040	27.39	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
3041	27.31	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
3042	27.3	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3043	27.25	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
3044	27.24	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
3045	27.24	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
3046	27.23	oe	ccsbBroad304_02502	GNA13	-			
3047	27.22	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
3048	27.19	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
3049	27.19	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
3050	27.14	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
3051	27.1	oe	ccsbBroad304_06140	EEF1D	-			
3052	27.09	kd	CGS001-5575	PRKAR1B	Protein kinase A			
3053	26.93	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
3054	26.89	kd	CGS001-9988	DMTF1	-			
3055	26.88	cc		Adenosine receptor agonist	-			
3056	26.8	oe	ccsbBroad304_12226	NAGK	-			
3057	26.8	kd	CGS001-22937	SCAP	WD repeat domain containing			
3058	26.8	kd	CGS001-32	ACACB	Carboxylases			
3059	26.75	kd	CGS001-27297	CRCP	-			
3060	26.73	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
3061	26.7	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3062	26.7	kd	CGS001-5467	PPARD	Nuclear hormone receptors			
3063	26.62	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
3064	26.62	oe	ccsbBroad304_02708	TRIM32	-			
3065	26.59	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
3066	26.59	oe	ccsbBroad304_06435	RBPJ	-			
3067	26.58	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
3068	26.56	oe	ccsbBroad304_00397	CTSK	Cathepsins			
3069	26.51	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
3070	26.49	oe	ccsbBroad304_07349	MAP7	-			
3071	26.47	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
3072	26.46	kd	CGS001-2773	GNAI3	-			
3073	26.39	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
3074	26.37	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
3075	26.33	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
3076	26.31	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
3077	26.31	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
3078	26.28	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
3079	26.28	kd	CGS001-4717	NDUFC1	Mitochondrial respiratory chain complex / Complex I			
3080	26.28	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
3081	26.23	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
3082	26.21	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
3083	26.14	kd	CGS001-7248	TSC1	-			
3084	26.09	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3085	26.09	kd	CGS001-5422	POLA1	DNA polymerases			
3086	26.07	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
3087	26.07	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
3088	26.07	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
3089	26.02	kd	CGS001-2261	FGFR3	Type V RTKs: FGF (fibroblast growth factor) receptor family			
3090	26.01	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
3091	25.97	kd	CGS001-10247	HRSP12	-			
3092	25.92	oe	ccsbBroad304_01008	KITLG	-			
3093	25.84	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
3094	25.83	kd	CGS001-4091	SMAD6	SMADs			
3095	25.81	kd	CGS001-10241	CALCOCO2	-			
3096	25.72	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
3097	25.71	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3098	25.55	kd	CGS001-7466	WFS1	-			
3099	25.52	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
3100	25.5	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
3101	25.45	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
3102	25.32	cp	BRD-K32398298	alprazolam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, CYP3A5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
3103	25.31	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
3104	25.31	kd	CGS001-139135	PASD1	-			
3105	25.25	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
3106	25.24	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
3107	25.24	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
3108	25.18	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
3109	25.16	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
3110	25.16	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
3111	25.14	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
3112	25.07	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
3113	25.07	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
3114	25	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
3115	24.96	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
3116	24.93	kd	CGS001-7106	TSPAN4	Tetraspanins			
3117	24.91	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
3118	24.87	kd	CGS001-8531	CSDA	-			
3119	24.85	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
3120	24.83	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
3121	24.82	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
3122	24.82	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
3123	24.76	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
3124	24.76	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
3125	24.76	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
3126	24.72	oe	ccsbBroad304_09756	PAQR7	-			
3127	24.69	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
3128	24.66	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
3129	24.66	kd	CGS001-339403	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
3130	24.57	oe	ccsbBroad304_07411	LPXN	-			
3131	24.56	kd	CGS001-8334	HIST1H2AC	Histones / Replication-dependent			
3132	24.53	kd	CGS001-8659	ALDH4A1	Aldehyde dehydrogenases			
3133	24.52	kd	CGS001-29083	GTPBP8	-			
3134	24.5	oe	ccsbBroad304_00986	MCM2	-			
3135	24.49	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
3136	24.49	oe	ccsbBroad304_10437	STMN1	-			
3137	24.46	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3138	24.45	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3139	24.44	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
3140	24.44	kd	CGS001-64783	RBM15	RNA binding motif (RRM) containing			
3141	24.42	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
3142	24.42	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
3143	24.3	kd	CGS001-3660	IRF2	-			
3144	24.27	oe	ccsbBroad304_00222	CASP6	Caspases			
3145	24.27	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
3146	24.27	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
3147	24.25	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3148	24.23	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
3149	24.16	kd	CGS001-1440	CSF3	Endogenous ligands			
3150	24.13	oe	ccsbBroad304_02399	TNIP1	-			
3151	24.1	oe	ccsbBroad304_00648	GLRX	-			
3152	24.02	oe	ccsbBroad304_03121	NRBF2	-			
3153	24.02	kd	CGS001-9221	NOLC1	-			
3154	24.01	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
3155	24.01	oe	ccsbBroad304_04064	PRR15L	-			
3156	23.99	kd	CGS001-116443	GRIN3A	Glutamate receptors			
3157	23.95	kd	CGS001-2010	EMD	-			
3158	23.89	oe	ccsbBroad304_00392	CTLA4	CD molecules			
3159	23.85	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
3160	23.83	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
3161	23.82	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
3162	23.82	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
3163	23.8	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
3164	23.79	kd	CGS001-23066	CAND2	-			
3165	23.76	kd	CGS001-79139	DERL1	-			
3166	23.75	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
3167	23.74	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
3168	23.73	kd	CGS001-161725	OTUD7A	OTU domain containing			
3169	23.64	kd	CGS001-23224	SYNE2	-			
3170	23.61	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
3171	23.6	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
3172	23.59	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3173	23.57	kd	CGS001-54884	RETSAT	-			
3174	23.55	oe	ccsbBroad304_08426	TEX10	-			
3175	23.53	kd	CGS001-1841	DTYMK	-			
3176	23.45	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
3177	23.42	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
3178	23.39	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
3179	23.39	kd	CGS001-10395	DLC1	Rho GTPase activating proteins			
3180	23.38	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
3181	23.34	kd	CGS001-9643	MORF4L2	-			
3182	23.31	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
3183	23.22	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
3184	23.17	oe	ccsbBroad304_03179	BOLA1	-			
3185	23.14	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
3186	23.14	oe	ccsbBroad304_00112	ASNA1	-			
3187	23.14	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
3188	23.09	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
3189	23.08	kd	CGS001-822	CAPG	-			
3190	23.07	kd	CGS001-4436	MSH2	-			
3191	23.06	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
3192	22.98	oe	ccsbBroad304_09195	MCM8	-			
3193	22.96	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
3194	22.93	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
3195	22.92	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
3196	22.84	oe	ccsbBroad304_01114	NUP88	-			
3197	22.83	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
3198	22.83	kd	CGS001-3487	IGFBP4	insulin-like growth factor (IGF) binding proteins			
3199	22.81	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
3200	22.79	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
3201	22.76	kd	CGS001-6810	STX4	-			
3202	22.74	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
3203	22.69	kd	CGS001-8624	PSMG1	-			
3204	22.65	kd	CGS001-23335	WDR7	WD repeat domain containing			
3205	22.63	kd	CGS001-54899	PXK	Slob family			
3206	22.62	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
3207	22.57	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
3208	22.57	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
3209	22.53	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
3210	22.52	kd	CGS001-5361	PLXNA1	Plexins			
3211	22.5	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
3212	22.49	cc		Glucocorticoid receptor agonist	-			
3213	22.4	oe	ccsbBroad304_01841	BAG6	-			
3214	22.39	cp	BRD-K46742498	alosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
3215	22.39	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3216	22.39	kd	CGS001-55608	ANKRD10	Ankyrin repeat domain containing			
3217	22.33	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3218	22.25	oe	ccsbBroad304_03118	NRBP1	NRBP family			
3219	22.14	oe	ccsbBroad304_00179	BTG1	-			
3220	22.13	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
3221	22.1	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
3222	22.1	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
3223	22.09	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
3224	22.08	kd	CGS001-60528	ELAC2	-			
3225	22.03	oe	ccsbBroad304_06670	OGG1	-			
3226	22.02	cp	BRD-K29653726	topiramate	Carbonic anhydrase inhibitor		CA2, CA4, GRIK1, CA1, CA12, CA7, CYP2C19, CYP3A4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA1, SCN1A, SCN5A	Carbonic anhydrase inhibitor, Glutamate receptor antagonist, Kainate receptor antagonist
3227	22.01	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3228	21.99	oe	ccsbBroad304_00102	RND3	-			
3229	21.97	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
3230	21.9	oe	ccsbBroad304_07808	RAB11FIP2	-			
3231	21.89	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
3232	21.89	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
3233	21.89	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
3234	21.88	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
3235	21.86	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
3236	21.86	oe	ccsbBroad304_03264	UBAP1	-			
3237	21.84	oe	ccsbBroad304_08093	DCPS	-			
3238	21.84	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
3239	21.68	kd	CGS001-9258	MFHAS1	-			
3240	21.67	kd	CGS001-7001	PRDX2	-			
3241	21.66	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
3242	21.62	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3243	21.61	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
3244	21.51	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
3245	21.51	kd	CGS001-8850	KAT2B	Histone acetyltransferases (HATs)			
3246	21.48	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
3247	21.44	cc		Aromatase inhibitor	-			
3248	21.44	kd	CGS001-5357	PLS1	EF-hand domain containing			
3249	21.34	kd	CGS001-1105	CHD1	-			
3250	21.29	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
3251	21.21	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
3252	21.2	kd	CGS001-4706	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
3253	21.17	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
3254	21.17	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
3255	21.16	kd	CGS001-2828	GPR4	GPCR / Class A : Orphans			
3256	21.09	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
3257	21.09	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
3258	21.05	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
3259	21.04	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
3260	21.03	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
3261	20.99	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3262	20.9	kd	CGS001-8678	BECN1	-			
3263	20.88	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
3264	20.88	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3265	20.88	kd	CGS001-10472	ZNF238	-			
3266	20.83	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
3267	20.74	oe	ccsbBroad304_12106	PXK	Slob family			
3268	20.66	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
3269	20.65	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
3270	20.63	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
3271	20.6	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3272	20.55	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
3273	20.54	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
3274	20.52	cc		Norepinephrine reuptake inhibitor	-			
3275	20.48	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
3276	20.48	kd	CGS001-57406	ABHD6	Abhydrolase domain containing			
3277	20.47	oe	ccsbBroad304_07018	SUPT5H	-			
3278	20.45	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
3279	20.44	kd	CGS001-2769	GNA15	-			
3280	20.39	kd	CGS001-55437	STRADB	STLK subfamily			
3281	20.37	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
3282	20.36	kd	CGS001-23585	TMEM50A	-			
3283	20.33	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
3284	20.27	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
3285	20.25	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
3286	20.25	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
3287	20.23	kd	CGS001-3957	LGALS2	Lectins, galactoside-binding			
3288	20.16	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
3289	20.16	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
3290	20.15	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
3291	20.12	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
3292	20.11	kd	CGS001-5092	PCBD1	-			
3293	20.09	kd	CGS001-478	ATP1A3	ATPases / P-type			
3294	20.04	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
3295	20.03	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
3296	20.03	kd	CGS001-8669	EIF3J	-			
3297	19.95	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
3298	19.94	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
3299	19.88	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
3300	19.88	kd	CGS001-3638	INSIG1	-			
3301	19.78	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
3302	19.74	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3303	19.68	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
3304	19.68	kd	CGS001-9415	FADS2	Fatty acid desaturases			
3305	19.66	cc		IMPDH inhibitor	-			
3306	19.63	kd	CGS001-6652	SORD	-			
3307	19.63	oe	ccsbBroad304_05192	SPRED2	-			
3308	19.62	oe	ccsbBroad304_13633	PI4KAP2	-			
3309	19.56	cp	BRD-K39983086	loteprednol	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Phospholipase inhibitor
3310	19.51	oe	ccsbBroad304_08553	STAP2	-			
3311	19.48	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
3312	19.47	cc		Imidazoline ligand	-			
3313	19.47	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
3314	19.42	kd	CGS001-23062	GGA2	-			
3315	19.38	oe	ccsbBroad304_00570	FIGF	-			
3316	19.37	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
3317	19.28	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
3318	19.22	kd	CGS001-3783	KCNN4	Calcium-activated potassium channels			
3319	19.22	kd	CGS001-3418	IDH2	-			
3320	19.21	kd	CGS001-8525	DGKZ	-			
3321	19.2	kd	CGS001-4594	MUT	-			
3322	19.19	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
3323	19.18	kd	CGS001-29968	PSAT1	-			
3324	19.15	kd	CGS001-10165	SLC25A13	Mitochondrial amino acid transporter subfamily			
3325	19.15	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
3326	19.07	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
3327	19.07	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
3328	18.96	kd	CGS001-3589	IL11	Endogenous ligands			
3329	18.94	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
3330	18.92	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
3331	18.9	kd	CGS001-4331	MNAT1	RING-type (C3HC4) zinc fingers			
3332	18.89	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
3333	18.84	kd	CGS001-51776	ZAK	MLK subfamily			
3334	18.84	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
3335	18.84	kd	CGS001-11007	CCDC85B	-			
3336	18.82	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
3337	18.69	oe	ccsbBroad304_00420	DAP	-			
3338	18.62	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
3339	18.59	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
3340	18.56	cc		Estrogen receptor antagonist	-			
3341	18.55	kd	CGS001-93349	SP140L	Zinc fingers, PHD-type			
3342	18.53	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
3343	18.53	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
3344	18.52	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
3345	18.5	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3346	18.48	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
3347	18.45	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
3348	18.44	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
3349	18.38	oe	ccsbBroad304_02633	LSM6	-			
3350	18.37	oe	ccsbBroad304_02862	CCRN4L	-			
3351	18.34	kd	CGS001-3460	IFNGR2	Interferon receptor family			
3352	18.33	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
3353	18.33	kd	CGS001-7030	TFE3	Basic helix-loop-helix proteins			
3354	18.31	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
3355	18.31	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
3356	18.22	oe	ccsbBroad304_02231	USP6NL	-			
3357	18.22	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
3358	18.18	kd	CGS001-54925	ZNF434	-			
3359	18.14	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
3360	18.11	kd	CGS001-3054	HCFC1	-			
3361	18.08	kd	CGS001-10481	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
3362	18.07	oe	ccsbBroad304_02345	TXNDC9	-			
3363	18.01	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3364	17.99	kd	CGS001-4734	NEDD4	-			
3365	17.99	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
3366	17.99	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
3367	17.97	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
3368	17.88	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
3369	17.88	kd	CGS001-6309	SC5DL	-			
3370	17.87	kd	CGS001-7534	YWHAZ	-			
3371	17.85	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3372	17.84	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
3373	17.83	cc		Androgen receptor modulator	-			
3374	17.79	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
3375	17.79	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
3376	17.79	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
3377	17.76	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
3378	17.74	kd	CGS001-5588	PRKCQ	Delta subfamily			
3379	17.71	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
3380	17.7	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
3381	17.69	kd	CGS001-823	CAPN1	EF-hand domain containing			
3382	17.66	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
3383	17.64	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
3384	17.63	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
3385	17.61	cp	BRD-K47278471	diphenhydramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
3386	17.61	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
3387	17.56	kd	CGS001-8853	ASAP2	Ankyrin repeat domain containing			
3388	17.55	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
3389	17.54	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
3390	17.5	kd	CGS001-10099	TSPAN3	Tetraspanins			
3391	17.48	kd	CGS001-9131	AIFM1	-			
3392	17.47	kd	CGS001-8505	PARG	-			
3393	17.46	cc		Nucleoside reverse transcriptase inhibitor	-			
3394	17.46	oe	ccsbBroad304_06324	GPX7	-			
3395	17.46	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
3396	17.42	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
3397	17.4	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
3398	17.39	kd	CGS001-537	ATP6AP1	-			
3399	17.38	kd	CGS001-8527	DGKD	Pleckstrin homology (PH) domain containing			
3400	17.36	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
3401	17.36	oe	ccsbBroad304_01148	PCBD1	-			
3402	17.36	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
3403	17.32	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3404	17.32	oe	ccsbBroad304_05948	CCND2	-			
3405	17.31	oe	ccsbBroad304_00949	LRPAP1	-			
3406	17.3	kd	CGS001-727	C5	Endogenous ligands			
3407	17.29	oe	ccsbBroad304_02834	GABARAPL1	-			
3408	17.27	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
3409	17.26	cc		Beta-adrenergic receptor agonist	-			
3410	17.25	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
3411	17.25	kd	CGS001-6709	SPTAN1	EF-hand domain containing			
3412	17.16	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
3413	17.05	cp	BRD-K44442813	pidotimod	Interferon receptor agonist			Interferon receptor agonist, Interleukin receptor agonist
3414	17.04	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
3415	16.98	kd	CGS001-2260	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
3416	16.95	kd	CGS001-1500	CTNND1	Catenins			
3417	16.94	kd	CGS001-1036	CDO1	-			
3418	16.92	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
3419	16.91	kd	CGS001-100133941	CD24	CD molecules			
3420	16.88	kd	CGS001-6009	RHEB	-			
3421	16.87	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
3422	16.83	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
3423	16.8	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
3424	16.79	oe	ccsbBroad304_00550	FDXR	-			
3425	16.78	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
3426	16.75	kd	CGS001-2523	FUT1	Fucosyltransferases			
3427	16.75	kd	CGS001-1499	CTNNB1	Catenins			
3428	16.73	kd	CGS001-8312	AXIN1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3429	16.72	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
3430	16.72	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
3431	16.68	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
3432	16.62	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
3433	16.6	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
3434	16.58	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
3435	16.56	kd	CGS001-4287	ATXN3	Ataxins			
3436	16.52	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
3437	16.51	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
3438	16.51	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
3439	16.46	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3440	16.42	oe	ccsbBroad304_05038	HORMAD2	-			
3441	16.39	kd	CGS001-255738	PCSK9	Subtilisin			
3442	16.38	kd	CGS001-7295	TXN	-			
3443	16.38	kd	CGS001-462	SERPINC1	Serine (or cysteine) peptidase inhibitors			
3444	16.36	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
3445	16.35	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
3446	16.35	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
3447	16.29	oe	ccsbBroad304_04490	RSPH1	-			
3448	16.27	kd	CGS001-9891	NUAK1	NuaK subfamily			
3449	16.18	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
3450	16.18	oe	ccsbBroad304_00359	CPT1A	-			
3451	16.16	kd	CGS001-53632	PRKAG3	AMPK subfamily			
3452	16.1	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
3453	16.1	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
3454	16.09	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
3455	16.08	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3456	16.04	kd	CGS001-205	AK4	Adenylate kinases			
3457	16.01	kd	CGS001-221391	OPN5	GPCR / Class A : Opsin receptors			
3458	15.98	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
3459	15.97	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
3460	15.95	oe	ccsbBroad304_07798	EXOC3	-			
3461	15.94	kd	CGS001-51001	MTERFD1	-			
3462	15.9	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
3463	15.87	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
3464	15.86	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
3465	15.86	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
3466	15.8	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
3467	15.77	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
3468	15.76	kd	CGS001-5781	PTPN11	Protein tyrosine phosphatases			
3469	15.74	kd	CGS001-642	BLMH	-			
3470	15.65	kd	CGS001-8548	BLZF1	-			
3471	15.6	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3472	15.59	kd	CGS001-4023	LPL	-			
3473	15.59	kd	CGS001-302	ANXA2	Annexins			
3474	15.55	kd	CGS001-9232	PTTG1	-			
3475	15.54	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
3476	15.51	oe	ccsbBroad304_06318	GPER	-			
3477	15.46	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
3478	15.44	oe	ccsbBroad304_05135	PARP15	-			
3479	15.44	kd	CGS001-2617	GARS	Aminoacyl tRNA synthetases / Class II			
3480	15.42	kd	CGS001-7168	TPM1	Tropomyosins			
3481	15.41	kd	CGS001-831	CAST	-			
3482	15.39	kd	CGS001-3675	ITGA3	Integrins			
3483	15.32	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
3484	15.31	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
3485	15.31	kd	CGS001-5931	RBBP7	WD repeat domain containing			
3486	15.29	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
3487	15.24	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
3488	15.19	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
3489	15.18	kd	CGS001-1997	ELF1	ETS Transcription Factors			
3490	15.17	kd	CGS001-51684	SUFU	-			
3491	15.15	oe	ccsbBroad304_01373	RAN	-			
3492	15.14	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
3493	15.12	kd	CGS001-51734	SEPX1	-			
3494	15.08	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
3495	15.07	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
3496	15.03	oe	ccsbBroad304_02922	TES	-			
3497	14.99	kd	CGS001-23192	ATG4B	Aut2 peptidase			
3498	14.99	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
3499	14.97	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
3500	14.97	oe	ccsbBroad304_01395	RFX5	-			
3501	14.93	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
3502	14.9	kd	CGS001-7405	UVRAG	-			
3503	14.88	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3504	14.87	oe	ccsbBroad304_00471	E2F6	-			
3505	14.85	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
3506	14.78	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
3507	14.68	kd	CGS001-23597	ACOT9	Acyl CoA thioesterases			
3508	14.63	oe	ccsbBroad304_03961	SMURF2	-			
3509	14.6	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
3510	14.55	oe	ccsbBroad304_08055	ATP5S	-			
3511	14.55	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
3512	14.54	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
3513	14.49	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
3514	14.47	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
3515	14.47	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
3516	14.46	oe	ccsbBroad304_07094	TPMT	-			
3517	14.45	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
3518	14.4	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
3519	14.35	kd	CGS001-23753	SDF2L1	-			
3520	14.34	kd	CGS001-2335	FN1	Endogenous ligands			
3521	14.31	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
3522	14.26	kd	CGS001-1173	AP2M1	-			
3523	14.24	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
3524	14.19	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
3525	14.18	kd	CGS001-9616	RNF7	RING-type (C3HC4) zinc fingers			
3526	14.13	kd	CGS001-2956	MSH6	-			
3527	14.11	kd	CGS001-7099	TLR4	Toll-like receptor family			
3528	14.11	kd	CGS001-85027	C5ORF62	-			
3529	14.1	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
3530	14.08	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
3531	13.98	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
3532	13.97	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
3533	13.95	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
3534	13.94	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
3535	13.94	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
3536	13.93	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
3537	13.91	cp	BRD-A15914070	4-hydroxy-2-nonenal	Cytotoxic lipid peroxidation product		IKBKB	Cytotoxic lipid peroxidation product
3538	13.89	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
3539	13.88	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
3540	13.84	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
3541	13.79	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
3542	13.79	kd	CGS001-94235	GNG8	-			
3543	13.76	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
3544	13.74	kd	CGS001-80306	MED28	-			
3545	13.73	cp	BRD-K23369905	oxiconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3546	13.68	kd	CGS001-10325	RRAGB	-			
3547	13.67	kd	CGS001-64943	NT5DC2	-			
3548	13.64	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
3549	13.62	kd	CGS001-10493	VAT1	-			
3550	13.55	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
3551	13.53	kd	CGS001-59286	UBL5	-			
3552	13.51	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
3553	13.44	kd	CGS001-5950	RBP4	Lipocalins			
3554	13.44	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
3555	13.43	kd	CGS001-51720	UIMC1	-			
3556	13.41	cc		Wnt family GOF	-			
3557	13.4	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
3558	13.38	oe	ccsbBroad304_00225	CAT	-			
3559	13.37	kd	CGS001-5345	SERPINF2	Serine (or cysteine) peptidase inhibitors			
3560	13.34	kd	CGS001-1045	CDX2	Homeoboxes / ANTP class : HOXL subclass			
3561	13.28	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
3562	13.27	kd	CGS001-84875	PARP10	Poly (ADP-ribose) polymerases			
3563	13.26	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
3564	13.26	oe	ccsbBroad304_00313	TBCB	-			
3565	13.25	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
3566	13.25	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
3567	13.25	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
3568	13.25	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
3569	13.23	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
3570	13.23	kd	CGS001-3459	IFNGR1	Interferon receptor family			
3571	13.17	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
3572	13.14	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
3573	13.11	oe	ccsbBroad304_01091	NFIB	-			
3574	13.11	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
3575	13.09	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3576	13.06	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
3577	13.02	cc		FLT3 inhibitor	-			
3578	13.02	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
3579	13	kd	CGS001-6605	SMARCE1	-			
3580	12.99	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
3581	12.97	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
3582	12.97	kd	CGS001-1844	DUSP2	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3583	12.96	kd	CGS001-51375	SNX7	Sorting nexins			
3584	12.9	kd	CGS001-3029	HAGH	-			
3585	12.86	kd	CGS001-23223	RRP12	-			
3586	12.84	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
3587	12.84	kd	CGS001-10632	ATP5L	ATPases / F-type			
3588	12.83	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
3589	12.83	kd	CGS001-55143	CDCA8	-			
3590	12.73	kd	CGS001-1647	GADD45A	-			
3591	12.7	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
3592	12.68	oe	ccsbBroad304_06226	FTL	-			
3593	12.66	kd	CGS001-9670	IPO13	Importins			
3594	12.65	kd	CGS001-23408	SIRT5	Histone deacetylases			
3595	12.63	oe	ccsbBroad304_07252	DGKZ	-			
3596	12.61	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
3597	12.59	kd	CGS001-11243	PMF1	-			
3598	12.58	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
3599	12.58	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
3600	12.54	kd	CGS001-1211	CLTA	-			
3601	12.52	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
3602	12.5	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
3603	12.48	oe	ccsbBroad304_07766	RASSF1	-			
3604	12.47	kd	CGS001-6446	SGK1	SGK family			
3605	12.47	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
3606	12.39	oe	ccsbBroad304_07890	CBX7	-			
3607	12.39	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
3608	12.38	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
3609	12.34	kd	CGS001-444	ASPH	-			
3610	12.31	oe	ccsbBroad304_02157	MED21	-			
3611	12.3	kd	CGS001-1287	COL4A5	Collagens			
3612	12.28	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
3613	12.26	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
3614	12.22	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
3615	12.21	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
3616	12.14	oe	ccsbBroad304_00155	CCND1	-			
3617	12.12	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
3618	12.1	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3619	12.03	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
3620	11.94	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
3621	11.91	oe	ccsbBroad304_03878	SENP2	-			
3622	11.89	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
3623	11.79	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
3624	11.76	kd	CGS001-2230	FDX1	-			
3625	11.69	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
3626	11.66	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
3627	11.64	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
3628	11.64	kd	CGS001-160	AP2A1	-			
3629	11.61	oe	ccsbBroad304_02136	COPS2	-			
3630	11.59	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
3631	11.56	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
3632	11.53	kd	CGS001-2786	GNG4	-			
3633	11.43	oe	ccsbBroad304_02569	BTG3	-			
3634	11.42	kd	CGS001-2963	GTF2F2	General transcription factors			
3635	11.4	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
3636	11.39	oe	ccsbBroad304_13939	MOK	RCK family			
3637	11.31	kd	CGS001-84288	EFCAB2	EF-hand domain containing			
3638	11.29	kd	CGS001-55632	G2E3	Zinc fingers, PHD-type			
3639	11.28	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
3640	11.26	kd	CGS001-1594	CYP27B1	Cytochrome P450s			
3641	11.17	kd	CGS001-8681	JMJD7-PLA2G4B	-			
3642	11.15	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
3643	11.13	kd	CGS001-5300	PIN1	-			
3644	11.07	kd	CGS001-9318	COPS2	-			
3645	11.05	kd	CGS001-5817	PVR	Immunoglobulin superfamily / C2-set domain containing			
3646	11	kd	CGS001-51271	UBAP1	-			
3647	10.99	cp	BRD-K62858456	lomerizine	Calcium channel blocker		ABCB1, CACNA1B, SCN5A	Calcium channel blocker
3648	10.98	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
3649	10.98	kd	CGS001-965	CD58	CD molecules			
3650	10.97	kd	CGS001-10494	STK25	YSK subfamily			
3651	10.92	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
3652	10.88	oe	ccsbBroad304_00941	LIG3	-			
3653	10.88	kd	CGS001-7965	AIMP2	-			
3654	10.86	kd	CGS001-83743	GRWD1	WD repeat domain containing			
3655	10.81	oe	ccsbBroad304_01674	TIMP4	-			
3656	10.81	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
3657	10.81	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
3658	10.75	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3659	10.73	kd	CGS001-2288	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
3660	10.73	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
3661	10.67	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
3662	10.67	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
3663	10.66	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
3664	10.65	oe	ccsbBroad304_02875	BRP44	-			
3665	10.65	oe	ccsbBroad304_00447	DLD	-			
3666	10.65	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
3667	10.61	kd	CGS001-8634	RTCD1	-			
3668	10.59	kd	CGS001-3856	KRT8	Intermediate filaments type II, keratins (basic)			
3669	10.58	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
3670	10.56	oe	ccsbBroad304_02229	TRAM2	-			
3671	10.42	kd	CGS001-5327	PLAT	Chymotrypsin			
3672	10.39	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
3673	10.29	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
3674	10.29	kd	CGS001-1869	E2F1	-			
3675	10.27	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
3676	10.23	kd	CGS001-85480	TSLP	-			
3677	10.21	kd	CGS001-10475	TRIM38	-			
3678	10.2	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
3679	10.18	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
3680	10.14	kd	CGS001-84527	ZNF559	Zinc fingers, C2H2-type			
3681	10.13	kd	CGS001-2615	LRRC32	-			
3682	10.12	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3683	10.11	kd	CGS001-1384	CRAT	-			
3684	10.09	oe	ccsbBroad304_02500	RRAGA	-			
3685	10.08	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
3686	10.06	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
3687	10.05	oe	ccsbBroad304_02686	COPZ1	-			
3688	10.04	kd	CGS001-51545	ZNF581	Zinc fingers, C2H2-type			
3689	10.01	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
3690	9.94	kd	CGS001-256364	EML3	WD repeat domain containing			
3691	9.86	oe	ccsbBroad304_01930	CUL2	-			
3692	9.85	oe	ccsbBroad304_08596	EAPP	-			
3693	9.84	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
3694	9.83	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
3695	9.82	kd	CGS001-271	AMPD2	-			
3696	9.76	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
3697	9.74	kd	CGS001-10891	PPARGC1A	RNA binding motif (RRM) containing			
3698	9.71	kd	CGS001-472	ATM	Other PIKK family kinases			
3699	9.7	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
3700	9.68	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
3701	9.68	oe	ccsbBroad304_07827	STK38L	NDR family			
3702	9.64	kd	CGS001-5881	RAC3	Endogenous ligands			
3703	9.61	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
3704	9.58	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
3705	9.55	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
3706	9.55	oe	ccsbBroad304_05745	CD24	CD molecules			
3707	9.53	oe	ccsbBroad304_00954	LYN	Src family			
3708	9.51	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
3709	9.48	oe	ccsbBroad304_04616	ORMDL3	-			
3710	9.46	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
3711	9.43	oe	ccsbBroad304_02553	BLCAP	-			
3712	9.43	oe	ccsbBroad304_06855	RDX	-			
3713	9.42	kd	CGS001-64094	SMOC2	EF-hand domain containing			
3714	9.4	oe	ccsbBroad304_09821	TMEM154	-			
3715	9.4	oe	ccsbBroad304_06349	HAGH	-			
3716	9.3	kd	CGS001-23523	CABIN1	-			
3717	9.25	kd	CGS001-80349	WDR61	WD repeat domain containing			
3718	9.19	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
3719	9.14	kd	CGS001-154197	PNLDC1	-			
3720	9.13	kd	CGS001-25937	WWTR1	Hippo Signaling			
3721	9.08	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
3722	9.04	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
3723	8.99	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
3724	8.95	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
3725	8.95	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
3726	8.92	oe	ccsbBroad304_03910	CCDC90A	-			
3727	8.92	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
3728	8.87	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
3729	8.84	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
3730	8.84	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
3731	8.78	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
3732	8.74	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
3733	8.73	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
3734	8.67	oe	ccsbBroad304_02278	THRAP3	-			
3735	8.67	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
3736	8.51	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3737	8.5	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
3738	8.48	kd	CGS001-1460	CSNK2B	Casein kinase 2 (CK2) family			
3739	8.44	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
3740	8.4	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
3741	8.4	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
3742	8.32	oe	ccsbBroad304_00854	IL8	-			
3743	8.28	kd	CGS001-10413	YAP1	Hippo Signaling			
3744	8.27	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
3745	8.24	kd	CGS001-23047	PDS5B	-			
3746	8.21	kd	CGS001-84969	TOX2	-			
3747	8.18	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
3748	8.12	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
3749	8.1	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
3750	8.09	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
3751	8.09	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
3752	8.05	kd	CGS001-718	C3	Endogenous ligands			
3753	8.03	kd	CGS001-10538	BATF	basic leucine zipper proteins			
3754	8.02	kd	CGS001-56889	TM9SF3	-			
3755	7.95	kd	CGS001-9441	MED26	-			
3756	7.95	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
3757	7.9	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
3758	7.9	oe	ccsbBroad304_02506	EBP	-			
3759	7.88	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
3760	7.88	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3761	7.87	oe	ccsbBroad304_02485	STAMBP	-			
3762	7.84	kd	CGS001-1066	CES1	Carboxylesterases			
3763	7.81	kd	CGS001-23464	GCAT	-			
3764	7.81	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
3765	7.8	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
3766	7.78	oe	ccsbBroad304_02017	PEX11A	-			
3767	7.76	kd	CGS001-7917	BAG6	-			
3768	7.74	kd	CGS001-5916	RARG	Retinoic acid receptors			
3769	7.72	kd	CGS001-8764	TNFRSF14	Tumour necrosis factor (TNF) receptor family			
3770	7.68	oe	ccsbBroad304_00747	HLF	-			
3771	7.68	kd	CGS001-1212	CLTB	-			
3772	7.64	oe	ccsbBroad304_08694	TBX20	T-boxes			
3773	7.63	oe	ccsbBroad304_05152	SSBP4	-			
3774	7.63	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
3775	7.62	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
3776	7.61	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
3777	7.6	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
3778	7.48	oe	ccsbBroad304_02890	SYF2	-			
3779	7.43	kd	CGS001-6643	SNX2	Sorting nexins			
3780	7.36	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
3781	7.36	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
3782	7.36	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
3783	7.32	oe	ccsbBroad304_06095	DFFB	-			
3784	7.29	kd	CGS001-9807	IP6K1	-			
3785	7.28	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
3786	7.26	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3787	7.22	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
3788	7.21	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
3789	7.18	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
3790	7.16	kd	CGS001-345	APOC3	Apolipoproteins			
3791	7.12	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
3792	7.11	oe	ccsbBroad304_05937	CASP7	Caspases			
3793	7.1	cp	BRD-K96740444	itopride	Dopamine receptor antagonist		DRD2, ACHE, CHRM3	Dopamine receptor antagonist
3794	7.07	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
3795	7.03	kd	CGS001-23509	POFUT1	Fucosyltransferases			
3796	6.98	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
3797	6.95	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
3798	6.94	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3799	6.93	cp	BRD-K51730347	diphencyprone	Immunostimulant			Immunostimulant
3800	6.9	kd	CGS001-6776	STAT5A	SH2 domain containing			
3801	6.9	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
3802	6.88	oe	ccsbBroad304_01962	STK16	NAK family			
3803	6.87	kd	CGS001-6364	CCL20	Chemokine ligands			
3804	6.86	oe	ccsbBroad304_03859	ENOPH1	-			
3805	6.84	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
3806	6.83	kd	CGS001-1977	EIF4E	Translation Initiation Factor 4E			
3807	6.82	kd	CGS001-51347	TAOK3	TAO subfamily			
3808	6.78	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
3809	6.76	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
3810	6.75	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
3811	6.71	kd	CGS001-170463	SSBP4	-			
3812	6.65	cc		Topoisomerase inhibitor	-			
3813	6.64	cc		G2 M Checkpoint LOF	-			
3814	6.62	kd	CGS001-593	BCKDHA	-			
3815	6.61	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
3816	6.57	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3817	6.51	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3818	6.5	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
3819	6.4	kd	CGS001-3066	HDAC2	Histone deacetylases			
3820	6.4	kd	CGS001-55802	DCP1A	-			
3821	6.38	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
3822	6.38	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3823	6.34	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
3824	6.31	oe	ccsbBroad304_07800	EXOSC8	-			
3825	6.29	kd	CGS001-9319	TRIP13	ATPases / AAA-type			
3826	6.2	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
3827	6.12	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
3828	6.08	kd	CGS001-344	APOC2	Apolipoproteins			
3829	6.07	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
3830	6.07	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
3831	6.06	oe	ccsbBroad304_00865	ILF2	-			
3832	6.02	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
3833	5.92	kd	CGS001-5052	PRDX1	-			
3834	5.92	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
3835	5.91	cp	BRD-A79903587	tegafur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
3836	5.9	kd	CGS001-3269	HRH1	Histamine receptors			
3837	5.88	kd	CGS001-5660	PSAP	Endogenous ligands			
3838	5.82	cc		Protein phosphatase catalytic subunits LOF	-			
3839	5.69	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
3840	5.69	oe	ccsbBroad304_03072	GTPBP8	-			
3841	5.61	kd	CGS001-4711	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
3842	5.6	cc		VEGFR inhibitor	-			
3843	5.59	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
3844	5.58	kd	CGS001-4817	NIT1	-			
3845	5.58	kd	CGS001-4668	NAGA	-			
3846	5.58	kd	CGS001-9184	BUB3	WD repeat domain containing			
3847	5.57	kd	CGS001-26086	GPSM1	Tetratricopeptide (TTC) repeat domain containing			
3848	5.56	oe	ccsbBroad304_08339	CMPK1	-			
3849	5.55	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
3850	5.51	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
3851	5.47	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
3852	5.47	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
3853	5.44	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
3854	5.41	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
3855	5.39	kd	CGS001-51222	ZNF219	Zinc fingers, C2H2-type			
3856	5.34	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
3857	5.32	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
3858	5.29	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
3859	5.25	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
3860	5.09	oe	ccsbBroad304_07768	NISCH	-			
3861	5.03	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
3862	5.02	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
3863	5	kd	CGS001-117154	DACH2	-			
3864	4.98	oe	ccsbBroad304_06518	LDHA	-			
3865	4.95	kd	CGS001-901	CCNG2	-			
3866	4.91	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
3867	4.86	oe	ccsbBroad304_05590	NOTCH2NL	-			
3868	4.82	kd	CGS001-2618	GART	Ribosyl transferases			
3869	4.81	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
3870	4.81	kd	CGS001-4638	MYLK	Myosin Light Chain Kinase (MLCK) family			
3871	4.81	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
3872	4.79	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
3873	4.77	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3874	4.74	kd	CGS001-4708	NDUFB2	Mitochondrial respiratory chain complex / Complex I			
3875	4.58	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
3876	4.53	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
3877	4.51	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
3878	4.47	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
3879	4.44	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
3880	4.44	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
3881	4.44	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
3882	4.38	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
3883	4.37	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
3884	4.32	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
3885	4.21	oe	ccsbBroad304_03641	ASF1B	-			
3886	4.17	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
3887	4.14	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
3888	4.1	oe	ccsbBroad304_02554	TRAFD1	-			
3889	4.07	oe	ccsbBroad304_04786	CANT1	-			
3890	4.07	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
3891	4.07	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
3892	4.03	oe	ccsbBroad304_07662	NPRL2	-			
3893	4.03	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
3894	3.98	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
3895	3.97	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3896	3.81	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
3897	3.8	kd	CGS001-8467	SMARCA5	-			
3898	3.8	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
3899	3.8	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
3900	3.74	oe	ccsbBroad304_06004	CKB	-			
3901	3.71	kd	CGS001-7057	THBS1	-			
3902	3.69	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
3903	3.64	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
3904	3.63	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
3905	3.61	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
3906	3.52	oe	ccsbBroad304_00632	GGCX	Carboxylases			
3907	3.47	cc		Apolipoproteins LOF	-			
3908	3.4	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
3909	3.4	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
3910	3.38	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
3911	3.35	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
3912	3.28	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
3913	3.25	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
3914	3.24	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
3915	3.22	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
3916	3.22	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
3917	3.18	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
3918	3.18	kd	CGS001-581	BAX	-			
3919	3.16	kd	CGS001-5727	PTCH1	-			
3920	3.1	oe	ccsbBroad304_13880	IDH3G	-			
3921	2.98	oe	ccsbBroad304_05749	A2M	-			
3922	2.92	kd	CGS001-5164	PDK2	PDHK family			
3923	2.87	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
3924	2.66	kd	CGS001-4245	MGAT1	-			
3925	2.64	oe	ccsbBroad304_01485	SC5DL	-			
3926	2.59	oe	ccsbBroad304_03112	NENF	-			
3927	2.59	oe	ccsbBroad304_02306	PQBP1	-			
3928	2.58	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
3929	2.54	oe	ccsbBroad304_01613	STK11	LKB subfamily			
3930	2.49	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
3931	2.36	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
3932	2.32	kd	CGS001-57149	LYRM1	LYR motif containing			
3933	2.22	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3934	2.18	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
3935	2.08	oe	ccsbBroad304_04649	ADC	-			
3936	1.76	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
3937	1.57	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
3938	1.57	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
3939	1.53	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
3940	1.39	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
3941	1.39	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
3942	1.39	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
3943	1.39	oe	ccsbBroad304_01035	MSH5	-			
3944	1.25	oe	ccsbBroad304_07219	CDC7	CDC7 family			
3945	0.97	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
3946	0.83	oe	ccsbBroad304_02452	NXF1	-			
3947	0.8	oe	ccsbBroad304_06178	ERCC5	-			
3948	0.67	cc		Potassium channel blocker	-			
3949	0.42	kd	CGS001-2931	GSK3A	GSK subfamily			
3950	-0.51	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3951	-0.96	kd	CGS001-11200	CHEK2	CHK1 subfamily			
3952	-1.25	oe	ccsbBroad304_00162	BIK	-			
3953	-1.26	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
3954	-1.3	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
3955	-1.3	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
3956	-1.34	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
3957	-1.37	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
3958	-1.52	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
3959	-1.57	oe	ccsbBroad304_03565	ADI1	-			
3960	-1.59	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
3961	-1.6	oe	ccsbBroad304_00644	GCLC	-			
3962	-1.71	oe	ccsbBroad304_06765	PRCC	-			
3963	-1.74	kd	CGS001-2957	GTF2A1	General transcription factors			
3964	-1.9	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
3965	-1.91	oe	ccsbBroad304_00054	ALDOC	-			
3966	-1.94	oe	ccsbBroad304_00446	DKC1	-			
3967	-1.94	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
3968	-2.08	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
3969	-2.15	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
3970	-2.17	oe	ccsbBroad304_05821	ANXA1	Annexins			
3971	-2.22	oe	ccsbBroad304_07557	NAMPT	-			
3972	-2.27	oe	ccsbBroad304_06870	RNH1	-			
3973	-2.27	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
3974	-2.36	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
3975	-2.42	oe	ccsbBroad304_01105	PNP	-			
3976	-2.45	oe	ccsbBroad304_02831	SGK3	SGK family			
3977	-2.54	cp	BRD-K52080565	rilmenidine	Imidazoline receptor agonist		NISCH	Imidazoline receptor agonist
3978	-2.54	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
3979	-2.63	kd	CGS001-4790	NFKB1	NFkappaB transcription factor family			
3980	-2.73	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
3981	-2.73	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
3982	-2.78	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
3983	-2.78	oe	ccsbBroad304_14242	MCCC2	-			
3984	-2.84	kd	CGS001-6622	SNCA	Parkinson disease			
3985	-2.9	oe	ccsbBroad304_09354	IGSF8	CD molecules			
3986	-2.92	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
3987	-2.92	oe	ccsbBroad304_01641	TAF13	-			
3988	-2.93	oe	ccsbBroad304_00993	MDM4	-			
3989	-3	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
3990	-3.01	oe	ccsbBroad304_03386	SPA17	-			
3991	-3.01	oe	ccsbBroad304_01724	TTR	-			
3992	-3.02	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
3993	-3.03	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
3994	-3.06	cc		Phospholipases GOF	-			
3995	-3.06	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
3996	-3.08	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
3997	-3.1	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
3998	-3.14	oe	ccsbBroad304_00933	LDHB	-			
3999	-3.15	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
4000	-3.16	kd	CGS001-1495	CTNNA1	Catenins			
4001	-3.24	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
4002	-3.29	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
4003	-3.29	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
4004	-3.4	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
4005	-3.43	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
4006	-3.43	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4007	-3.56	oe	ccsbBroad304_02496	MTX2	-			
4008	-3.61	kd	CGS001-2837	UTS2R	Urotensin receptor			
4009	-3.68	kd	CGS001-4172	MCM3	-			
4010	-3.74	kd	CGS001-8848	TSC22D1	-			
4011	-3.76	kd	CGS001-678	ZFP36L2	RING-type (C3HC4) zinc fingers			
4012	-3.84	oe	ccsbBroad304_07401	TXNL1	-			
4013	-3.84	kd	CGS001-57026	PDXP	-			
4014	-3.89	kd	CGS001-55832	CAND1	-			
4015	-3.97	kd	CGS001-586	BCAT1	-			
4016	-3.99	oe	ccsbBroad304_00006	ACADM	-			
4017	-4.1	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
4018	-4.11	kd	CGS001-55234	SMU1	WD repeat domain containing			
4019	-4.19	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
4020	-4.21	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
4021	-4.24	kd	CGS001-7477	WNT7B	Endogenous ligands			
4022	-4.25	kd	CGS001-10390	CEPT1	-			
4023	-4.28	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
4024	-4.35	oe	ccsbBroad304_03950	ATG3	-			
4025	-4.37	kd	CGS001-776	CACNA1D	Calcium channel subunits			
4026	-4.4	kd	CGS001-3725	JUN	basic leucine zipper proteins			
4027	-4.43	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
4028	-4.47	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
4029	-4.48	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
4030	-4.51	cp	BRD-K53220666	trimetozine	Sedative			Sedative
4031	-4.54	oe	ccsbBroad304_03428	EXOSC4	-			
4032	-4.58	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
4033	-4.58	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
4034	-4.62	oe	ccsbBroad304_01084	NEU1	-			
4035	-4.68	oe	ccsbBroad304_07012	STK3	MST subfamily			
4036	-4.69	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4037	-4.77	oe	ccsbBroad304_04406	PLA2G12B	-			
4038	-4.77	oe	ccsbBroad304_12008	NLK	nmo subfamily			
4039	-4.78	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
4040	-4.85	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
4041	-4.86	oe	ccsbBroad304_00963	SMAD5	SMADs			
4042	-4.89	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
4043	-4.92	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
4044	-4.95	oe	ccsbBroad304_09954	PTRF	-			
4045	-4.95	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4046	-4.95	oe	ccsbBroad304_06836	RAD23B	-			
4047	-4.96	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
4048	-5	oe	ccsbBroad304_09615	LACC1	-			
4049	-5.03	oe	ccsbBroad304_06538	LSP1	-			
4050	-5.06	oe	ccsbBroad304_07045	TEAD4	-			
4051	-5.09	kd	CGS001-10252	SPRY1	-			
4052	-5.1	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
4053	-5.11	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
4054	-5.14	oe	ccsbBroad304_03173	TMED7	-			
4055	-5.16	kd	CGS001-10955	SERINC3	-			
4056	-5.16	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
4057	-5.16	oe	ccsbBroad304_01054	GADD45B	-			
4058	-5.17	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
4059	-5.19	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
4060	-5.19	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
4061	-5.2	kd	CGS001-1026	CDKN1A	-			
4062	-5.25	kd	CGS001-10587	TXNRD2	-			
4063	-5.26	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
4064	-5.26	kd	CGS001-22887	FOXJ3	Forkhead boxes			
4065	-5.28	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
4066	-5.32	kd	CGS001-5744	PTHLH	Endogenous ligands			
4067	-5.38	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
4068	-5.42	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
4069	-5.42	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
4070	-5.43	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
4071	-5.44	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
4072	-5.46	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
4073	-5.46	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
4074	-5.47	kd	CGS001-701	BUB1B	Bub family			
4075	-5.48	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
4076	-5.53	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
4077	-5.54	kd	CGS001-51548	SIRT6	Histone deacetylases (HDACs)			
4078	-5.6	kd	CGS001-7572	ZNF24	Zinc fingers, C2H2-type			
4079	-5.63	kd	CGS001-7533	YWHAH	-			
4080	-5.69	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
4081	-5.69	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
4082	-5.7	oe	ccsbBroad304_00098	ARG1	Arginase			
4083	-5.76	kd	CGS001-7389	UROD	-			
4084	-5.76	kd	CGS001-29079	MED4	-			
4085	-5.78	cp	BRD-K55034111	pefloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4086	-5.78	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
4087	-5.79	kd	CGS001-79947	DHDDS	-			
4088	-5.82	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
4089	-5.84	kd	CGS001-23369	PUM2	-			
4090	-5.88	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
4091	-5.9	kd	CGS001-515	ATP5F1	ATPases / F-type			
4092	-5.92	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
4093	-5.93	kd	CGS001-5573	PRKAR1A	Protein kinase A			
4094	-6.02	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
4095	-6.02	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
4096	-6.04	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
4097	-6.08	kd	CGS001-4929	NR4A2	Nerve growth factor IB-like receptors			
4098	-6.11	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
4099	-6.13	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
4100	-6.16	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
4101	-6.16	kd	CGS001-6491	STIL	-			
4102	-6.18	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
4103	-6.19	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
4104	-6.28	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
4105	-6.3	oe	ccsbBroad304_03311	EVL	-			
4106	-6.3	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4107	-6.33	oe	ccsbBroad304_04544	RCCD1	-			
4108	-6.33	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4109	-6.33	oe	ccsbBroad304_02497	YKT6	-			
4110	-6.34	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
4111	-6.34	kd	CGS001-1906	EDN1	Endogenous ligands			
4112	-6.39	oe	ccsbBroad304_01605	SSX2	-			
4113	-6.41	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4114	-6.44	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
4115	-6.45	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
4116	-6.45	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
4117	-6.46	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
4118	-6.48	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
4119	-6.5	kd	CGS001-22883	CLSTN1	Cadherins / Cadherin-related			
4120	-6.52	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
4121	-6.53	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
4122	-6.54	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
4123	-6.57	kd	CGS001-84930	MASTL	MAST family			
4124	-6.57	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
4125	-6.59	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4126	-6.6	kd	CGS001-55082	ARGLU1	-			
4127	-6.64	kd	CGS001-1111	CHEK1	CHK1 subfamily			
4128	-6.66	kd	CGS001-966	CD59	CD molecules			
4129	-6.69	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
4130	-6.7	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
4131	-6.75	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
4132	-6.78	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
4133	-6.79	kd	CGS001-55191	NADSYN1	-			
4134	-6.85	oe	ccsbBroad304_03615	ZNF673	-			
4135	-6.87	kd	CGS001-4864	NPC1	-			
4136	-6.88	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
4137	-6.89	kd	CGS001-3421	IDH3G	-			
4138	-6.9	kd	CGS001-144811	LACC1	-			
4139	-6.9	kd	CGS001-9290	GPR55	GPCR / Class A : Orphans			
4140	-6.92	kd	CGS001-5019	OXCT1	-			
4141	-6.98	kd	CGS001-5708	PSMD2	Proteasome subunits			
4142	-6.99	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
4143	-7.05	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
4144	-7.12	kd	CGS001-55165	CEP55	-			
4145	-7.17	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
4146	-7.21	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
4147	-7.26	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
4148	-7.27	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
4149	-7.27	oe	ccsbBroad304_00501	EMD	-			
4150	-7.27	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
4151	-7.31	oe	ccsbBroad304_02425	CDIPT	-			
4152	-7.31	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
4153	-7.36	oe	ccsbBroad304_08993	DHDDS	-			
4154	-7.37	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
4155	-7.41	kd	CGS001-5226	PGD	-			
4156	-7.45	oe	ccsbBroad304_08888	ACD	-			
4157	-7.51	cp	BRD-K60690191	MPEP	Glutamate receptor antagonist		GRM5, GRM1, GRM4	Glutamate receptor antagonist
4158	-7.56	oe	ccsbBroad304_06976	SMARCE1	-			
4159	-7.59	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
4160	-7.64	oe	ccsbBroad304_02869	ASF1A	-			
4161	-7.64	oe	ccsbBroad304_01673	TIMP3	-			
4162	-7.66	oe	ccsbBroad304_00115	ASPH	-			
4163	-7.7	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
4164	-7.72	kd	CGS001-665	BNIP3L	-			
4165	-7.72	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4166	-7.73	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
4167	-7.75	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
4168	-7.75	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
4169	-7.76	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
4170	-7.78	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
4171	-7.81	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
4172	-7.81	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4173	-7.86	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
4174	-7.87	oe	ccsbBroad304_06648	CNOT3	-			
4175	-7.9	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
4176	-7.9	oe	ccsbBroad304_03037	TMEM97	-			
4177	-7.91	kd	CGS001-5411	PNN	-			
4178	-7.91	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
4179	-7.92	oe	ccsbBroad304_06952	SKP1	-			
4180	-7.92	kd	CGS001-7029	TFDP2	-			
4181	-7.95	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
4182	-8.01	oe	ccsbBroad304_01948	GAS7	-			
4183	-8.01	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
4184	-8.08	kd	CGS001-10250	SRRM1	-			
4185	-8.09	kd	CGS001-23786	BCL2L13	-			
4186	-8.1	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
4187	-8.12	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
4188	-8.13	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
4189	-8.14	kd	CGS001-3663	IRF5	-			
4190	-8.15	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
4191	-8.19	kd	CGS001-5167	ENPP1	-			
4192	-8.19	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
4193	-8.2	oe	ccsbBroad304_05528	TICAM2	-			
4194	-8.21	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
4195	-8.27	kd	CGS001-283150	FOXR1	Forkhead boxes			
4196	-8.27	oe	ccsbBroad304_06225	FTH1	-			
4197	-8.33	kd	CGS001-7263	TST	-			
4198	-8.36	cc		TGF beta receptor inhibitor	-			
4199	-8.39	kd	CGS001-139760	GPR119	GPCR / Class A : Orphans			
4200	-8.4	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
4201	-8.42	kd	CGS001-5257	PHKB	-			
4202	-8.44	kd	CGS001-11336	EXOC3	-			
4203	-8.47	kd	CGS001-6857	SYT1	Synaptotagmins			
4204	-8.52	kd	CGS001-30	ACAA1	-			
4205	-8.52	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
4206	-8.53	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4207	-8.53	kd	CGS001-10198	MPHOSPH9	-			
4208	-8.55	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
4209	-8.56	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
4210	-8.59	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
4211	-8.59	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
4212	-8.66	kd	CGS001-238	ALK	Leukocyte tyrosine kinase (LTK) receptor family			
4213	-8.68	kd	CGS001-51593	SRRT	-			
4214	-8.7	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
4215	-8.71	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
4216	-8.71	kd	CGS001-93185	IGSF8	CD molecules			
4217	-8.71	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
4218	-8.74	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
4219	-8.76	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
4220	-8.77	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
4221	-8.79	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
4222	-8.79	oe	ccsbBroad304_00665	GOT1	-			
4223	-8.79	cp	BRD-K27184429	levocetirizine	Histamine receptor antagonist		HRH1, CXCL8	Histamine receptor antagonist
4224	-8.8	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
4225	-8.8	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4226	-8.82	kd	CGS001-9014	TAF1B	-			
4227	-8.82	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4228	-8.9	oe	ccsbBroad304_02086	PDLIM1	-			
4229	-8.96	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
4230	-8.99	kd	CGS001-9412	MED21	-			
4231	-9	kd	CGS001-10013	HDAC6	Histone deacetylases			
4232	-9.04	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
4233	-9.06	kd	CGS001-182	JAG1	CD molecules			
4234	-9.08	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
4235	-9.1	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
4236	-9.18	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
4237	-9.26	kd	CGS001-55256	ADI1	-			
4238	-9.29	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
4239	-9.31	oe	ccsbBroad304_04038	ELOVL6	-			
4240	-9.32	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
4241	-9.34	kd	CGS001-147179	WIPF2	-			
4242	-9.35	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
4243	-9.37	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
4244	-9.39	kd	CGS001-11164	NUDT5	Nudix motif containing			
4245	-9.41	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
4246	-9.42	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
4247	-9.44	kd	CGS001-5159	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
4248	-9.45	kd	CGS001-4179	CD46	CD molecules			
4249	-9.46	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
4250	-9.46	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
4251	-9.46	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
4252	-9.5	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
4253	-9.52	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
4254	-9.54	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
4255	-9.55	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
4256	-9.55	kd	CGS001-54881	TEX10	-			
4257	-9.59	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
4258	-9.61	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
4259	-9.63	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
4260	-9.67	oe	ccsbBroad304_00931	LCN2	Lipocalins			
4261	-9.75	kd	CGS001-2099	ESR1	Estrogen receptors			
4262	-9.75	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4263	-9.78	kd	CGS001-4860	PNP	-			
4264	-9.78	kd	CGS001-10681	GNB5	WD repeat domain containing			
4265	-9.78	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
4266	-9.8	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
4267	-9.85	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
4268	-9.85	kd	CGS001-5621	PRNP	CD molecules			
4269	-9.87	kd	CGS001-10943	MSL3	-			
4270	-9.92	kd	CGS001-9158	FIBP	-			
4271	-9.94	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
4272	-9.95	kd	CGS001-6271	S100A1	EF-hand domain containing			
4273	-9.97	kd	CGS001-4782	NFIC	-			
4274	-9.99	kd	CGS001-5689	PSMB1	Proteasome subunits			
4275	-10.01	oe	ccsbBroad304_03186	GMNN	-			
4276	-10.05	oe	ccsbBroad304_07337	TAF1B	-			
4277	-10.05	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
4278	-10.09	kd	CGS001-10010	TANK	-			
4279	-10.09	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
4280	-10.2	cp	BRD-K56614220	clofazimine	GK0582 inhibitor			GK0582 inhibitor
4281	-10.21	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
4282	-10.21	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
4283	-10.23	oe	ccsbBroad304_07515	GFPT2	-			
4284	-10.25	oe	ccsbBroad304_00423	DAXX	-			
4285	-10.25	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
4286	-10.31	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
4287	-10.39	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
4288	-10.41	kd	CGS001-2990	GUSB	-			
4289	-10.42	kd	CGS001-10921	RNPS1	RNA binding motif (RRM) containing			
4290	-10.44	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
4291	-10.44	kd	CGS001-7031	TFF1	-			
4292	-10.46	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
4293	-10.48	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
4294	-10.52	cp	BRD-K81169441	cerivastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A5	HMGCR inhibitor
4295	-10.58	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
4296	-10.62	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
4297	-10.63	kd	CGS001-4700	NDUFA6	LYR motif containing			
4298	-10.63	oe	ccsbBroad304_09358	MAPK1IP1L	-			
4299	-10.66	kd	CGS001-147948	ZNF582	Zinc fingers, C2H2-type			
4300	-10.68	oe	ccsbBroad304_04053	DERL1	-			
4301	-10.7	kd	CGS001-81577	GFOD2	-			
4302	-10.75	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
4303	-10.76	oe	ccsbBroad304_07843	FCHO1	-			
4304	-10.81	oe	ccsbBroad304_01754	UCK2	-			
4305	-10.87	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
4306	-10.87	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
4307	-10.9	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
4308	-10.92	cp	BRD-K34437622	BRD-K34437622	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
4309	-10.99	kd	CGS001-22938	SNW1	-			
4310	-10.99	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
4311	-11.07	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
4312	-11.11	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
4313	-11.17	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
4314	-11.2	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
4315	-11.23	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
4316	-11.25	kd	CGS001-84775	ZNF607	Zinc fingers, C2H2-type			
4317	-11.27	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
4318	-11.29	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
4319	-11.31	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4320	-11.34	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
4321	-11.35	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4322	-11.36	oe	ccsbBroad304_00987	MCM3	-			
4323	-11.37	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4324	-11.39	kd	CGS001-222546	RFX6	-			
4325	-11.41	kd	CGS001-140465	MYL6B	EF-hand domain containing			
4326	-11.41	kd	CGS001-29105	C16ORF80	-			
4327	-11.44	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
4328	-11.46	kd	CGS001-2145	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
4329	-11.48	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
4330	-11.48	oe	ccsbBroad304_08511	RFK	-			
4331	-11.49	kd	CGS001-1072	CFL1	-			
4332	-11.55	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
4333	-11.56	kd	CGS001-5982	RFC2	ATPases / AAA-type			
4334	-11.62	kd	CGS001-9967	THRAP3	-			
4335	-11.65	kd	CGS001-29880	ALG5	Glycosyltransferase family 2 domain containing			
4336	-11.67	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
4337	-11.68	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
4338	-11.69	oe	ccsbBroad304_00053	ALDOA	-			
4339	-11.71	oe	ccsbBroad304_02815	SSBP2	-			
4340	-11.72	cc		Supressors of cytokine signaling GOF	-			
4341	-11.83	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
4342	-11.83	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
4343	-11.87	kd	CGS001-5498	PPOX	-			
4344	-11.91	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
4345	-11.95	kd	CGS001-140690	CTCFL	Zinc fingers, C2H2-type			
4346	-11.95	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
4347	-12.05	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
4348	-12.06	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
4349	-12.1	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
4350	-12.14	cc		Reverse transcriptase inhibitor	-			
4351	-12.14	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
4352	-12.18	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
4353	-12.18	kd	CGS001-9655	SOCS5	SH2 domain containing			
4354	-12.2	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
4355	-12.25	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
4356	-12.31	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
4357	-12.34	kd	CGS001-7251	TSG101	-			
4358	-12.35	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
4359	-12.35	kd	CGS001-27346	TMEM97	-			
4360	-12.35	kd	CGS001-3123	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
4361	-12.4	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
4362	-12.43	kd	CGS001-11232	POLG2	DNA polymerases			
4363	-12.43	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
4364	-12.5	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
4365	-12.51	oe	ccsbBroad304_03696	C19ORF10	-			
4366	-12.53	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
4367	-12.54	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
4368	-12.55	oe	ccsbBroad304_02653	PRAF2	-			
4369	-12.6	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
4370	-12.64	kd	CGS001-836	CASP3	Caspases			
4371	-12.65	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4372	-12.65	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
4373	-12.65	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4374	-12.69	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
4375	-12.71	oe	ccsbBroad304_03933	CARD9	-			
4376	-12.73	kd	CGS001-390980	ZNF805	Zinc fingers, C2H2-type			
4377	-12.73	kd	CGS001-10906	TRAFD1	-			
4378	-12.74	kd	CGS001-1314	COPA	Endogenous ligands			
4379	-12.75	kd	CGS001-10227	MFSD10	-			
4380	-12.81	kd	CGS001-10489	LRRC41	-			
4381	-12.81	kd	CGS001-840	CASP7	Caspases			
4382	-12.82	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
4383	-12.84	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
4384	-12.84	kd	CGS001-1514	CTSL1	-			
4385	-12.87	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4386	-12.87	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
4387	-12.88	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
4388	-12.89	kd	CGS001-25797	QPCT	Aminopeptidase Y			
4389	-12.92	kd	CGS001-1128	CHRM1	Cholinergic receptors			
4390	-12.94	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
4391	-12.95	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
4392	-12.98	oe	ccsbBroad304_00223	CASP9	Caspases			
4393	-12.99	kd	CGS001-5062	PAK2	PAKA subfamily			
4394	-13	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
4395	-13.02	oe	ccsbBroad304_10207	ERLIN1	-			
4396	-13.03	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
4397	-13.04	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
4398	-13.11	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
4399	-13.13	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
4400	-13.16	kd	CGS001-2872	MKNK2	MKN subfamily			
4401	-13.18	kd	CGS001-1515	CTSL2	-			
4402	-13.19	kd	CGS001-51466	EVL	-			
4403	-13.2	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
4404	-13.23	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
4405	-13.23	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
4406	-13.24	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
4407	-13.24	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
4408	-13.28	oe	ccsbBroad304_00880	IRF2	-			
4409	-13.3	kd	CGS001-262	AMD1	Decarboxylases			
4410	-13.3	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
4411	-13.33	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
4412	-13.36	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
4413	-13.41	kd	CGS001-4683	NBN	-			
4414	-13.41	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
4415	-13.42	kd	CGS001-6118	RPA2	-			
4416	-13.44	oe	ccsbBroad304_01142	PAFAH1B2	-			
4417	-13.47	kd	CGS001-5378	PMS1	-			
4418	-13.49	kd	CGS001-55107	ANO1	Calcium activated chloride channel			
4419	-13.49	kd	CGS001-158	ADSL	-			
4420	-13.51	kd	CGS001-10138	YAF2	-			
4421	-13.51	kd	CGS001-5710	PSMD4	Proteasome (prosome, macropain) subunits			
4422	-13.52	oe	ccsbBroad304_07124	UROD	-			
4423	-13.53	kd	CGS001-2664	GDI1	-			
4424	-13.55	kd	CGS001-256281	NUDT14	Nudix motif containing			
4425	-13.56	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
4426	-13.59	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
4427	-13.6	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
4428	-13.61	kd	CGS001-2149	F2R	Protease activated receptors			
4429	-13.66	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
4430	-13.66	kd	CGS001-7077	TIMP2	-			
4431	-13.67	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
4432	-13.72	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
4433	-13.72	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
4434	-13.73	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
4435	-13.78	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
4436	-13.88	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
4437	-13.93	kd	CGS001-4704	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4438	-13.96	kd	CGS001-23266	LPHN2	Adhesion Class GPCRs			
4439	-13.98	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4440	-14.05	kd	CGS001-93134	ZNF561	Zinc fingers, C2H2-type			
4441	-14.06	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
4442	-14.09	oe	ccsbBroad304_02367	CALCOCO2	-			
4443	-14.23	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
4444	-14.24	oe	ccsbBroad304_06424	IFI16	-			
4445	-14.25	kd	CGS001-3329	HSPD1	Heat Shock Proteins / Chaperonins			
4446	-14.29	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
4447	-14.36	cc		Lipocalins GOF	-			
4448	-14.4	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
4449	-14.41	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
4450	-14.49	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
4451	-14.52	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4452	-14.52	kd	CGS001-5567	PRKACB	Protein kinase A			
4453	-14.55	kd	CGS001-25989	ULK3	Unc-51-like kinase (ULK) family			
4454	-14.6	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
4455	-14.62	kd	CGS001-8495	PPFIBP2	Sterile alpha motif (SAM) domain containing			
4456	-14.63	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
4457	-14.65	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
4458	-14.67	kd	CGS001-9455	HOMER2	-			
4459	-14.68	oe	ccsbBroad304_02772	ICMT	-			
4460	-14.68	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
4461	-14.71	kd	CGS001-24148	PRPF6	-			
4462	-14.72	kd	CGS001-4869	NPM1	-			
4463	-14.78	kd	CGS001-116113	FOXP4	Forkhead boxes			
4464	-14.79	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
4465	-14.82	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
4466	-14.85	oe	ccsbBroad304_00626	GDI1	-			
4467	-14.89	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
4468	-14.91	oe	ccsbBroad304_05981	CDO1	-			
4469	-14.95	kd	CGS001-29965	C16ORF5	-			
4470	-14.97	kd	CGS001-57521	RPTOR	WD repeat domain containing			
4471	-14.99	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
4472	-15	cc		HRH1 antagonist	-			
4473	-15.01	kd	CGS001-4791	NFKB2	NFkappaB transcription factor family			
4474	-15.06	kd	CGS001-8837	CFLAR	Endogenous ligands			
4475	-15.07	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
4476	-15.07	kd	CGS001-661	POLR3D	RNA polymerase subunits			
4477	-15.12	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
4478	-15.13	kd	CGS001-11157	LSM6	-			
4479	-15.13	oe	ccsbBroad304_06180	ESD	-			
4480	-15.18	kd	CGS001-10939	AFG3L2	ATPases / AAA-type			
4481	-15.18	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
4482	-15.19	kd	CGS001-9869	SETDB1	Histone methyltransferases (HMTs)			
4483	-15.22	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
4484	-15.23	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
4485	-15.24	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
4486	-15.27	cc		Nucleophosmin inhibitor	-			
4487	-15.28	kd	CGS001-2548	GAA	Glycosidases			
4488	-15.29	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
4489	-15.29	kd	CGS001-10084	PQBP1	-			
4490	-15.3	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
4491	-15.32	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
4492	-15.34	kd	CGS001-213	ALB	-			
4493	-15.37	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
4494	-15.38	kd	CGS001-1504	CTRB1	-			
4495	-15.39	kd	CGS001-7846	TUBA1A	Tubulins			
4496	-15.42	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
4497	-15.42	kd	CGS001-81621	KAZALD1	Immunoglobulin superfamily / I-set domain containing			
4498	-15.44	oe	ccsbBroad304_07374	PTPLA	-			
4499	-15.44	kd	CGS001-230	ALDOC	-			
4500	-15.46	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
4501	-15.47	kd	CGS001-2744	GLS	Ankyrin repeat domain containing			
4502	-15.55	kd	CGS001-55111	PLEKHJ1	Pleckstrin homology (PH) domain containing			
4503	-15.58	kd	CGS001-5198	PFAS	-			
4504	-15.58	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
4505	-15.6	kd	CGS001-3109	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
4506	-15.67	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
4507	-15.68	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
4508	-15.74	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
4509	-15.76	kd	CGS001-55500	ETNK1	-			
4510	-15.78	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
4511	-15.78	kd	CGS001-5163	PDK1	-			
4512	-15.81	kd	CGS001-949	SCARB1	-			
4513	-15.83	kd	CGS001-1725	DHPS	-			
4514	-15.88	cp	BRD-K16336526	capsaicin	TRPV agonist		TRPV1, CFTR, ENOX2	TRPV agonist
4515	-15.88	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
4516	-15.89	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
4517	-15.9	kd	CGS001-54498	SMOX	-			
4518	-15.93	oe	ccsbBroad304_02804	KLHDC2	-			
4519	-15.93	oe	ccsbBroad304_06287	GM2A	-			
4520	-15.94	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
4521	-15.96	kd	CGS001-9842	PLEKHM1	Pleckstrin homology (PH) domain containing			
4522	-15.96	kd	CGS001-174	AFP	-			
4523	-15.97	kd	CGS001-8022	LHX3	Homeoboxes / LIM class			
4524	-15.98	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
4525	-16.01	cp	BRD-K02227374	milnacipran	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Serotonin reuptake inhibitor
4526	-16.01	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
4527	-16.05	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
4528	-16.08	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
4529	-16.08	oe	ccsbBroad304_07754	FGFR1OP	-			
4530	-16.1	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
4531	-16.11	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
4532	-16.13	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4533	-16.19	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
4534	-16.2	kd	CGS001-4143	MAT1A	-			
4535	-16.26	kd	CGS001-58472	SQRDL	-			
4536	-16.27	oe	ccsbBroad304_00009	ACLY	-			
4537	-16.28	kd	CGS001-22933	SIRT2	Histone deacetylases			
4538	-16.36	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
4539	-16.38	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
4540	-16.38	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
4541	-16.38	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
4542	-16.38	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
4543	-16.39	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
4544	-16.41	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
4545	-16.44	kd	CGS001-10725	NFAT5	Nuclear factor of activated T-cells			
4546	-16.49	kd	CGS001-375346	TMEM110	-			
4547	-16.5	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
4548	-16.51	oe	ccsbBroad304_06665	OAT	-			
4549	-16.51	kd	CGS001-4221	MEN1	-			
4550	-16.58	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
4551	-16.58	oe	ccsbBroad304_02674	STK38	NDR family			
4552	-16.62	oe	ccsbBroad304_02373	SPRY2	-			
4553	-16.64	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
4554	-16.67	kd	CGS001-27333	GOLIM4	-			
4555	-16.69	oe	ccsbBroad304_04294	ATG10	-			
4556	-16.72	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
4557	-16.75	kd	CGS001-54584	GNB1L	WD repeat domain containing			
4558	-16.79	kd	CGS001-5910	RAP1GDS1	Armadillo repeat containing			
4559	-16.82	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
4560	-16.83	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
4561	-16.83	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
4562	-16.84	kd	CGS001-342926	ZNF677	Zinc fingers, C2H2-type			
4563	-16.87	kd	CGS001-817	CAMK2D	CAMK2 family			
4564	-16.88	oe	ccsbBroad304_00690	GRN	-			
4565	-16.96	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
4566	-17	kd	CGS001-51293	CD320	CD molecules			
4567	-17.03	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
4568	-17.06	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
4569	-17.08	kd	CGS001-7693	ZNF134	Zinc fingers, C2H2-type			
4570	-17.15	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
4571	-17.17	kd	CGS001-51026	GOLT1B	-			
4572	-17.26	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
4573	-17.3	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
4574	-17.31	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
4575	-17.32	oe	ccsbBroad304_06985	SORD	-			
4576	-17.32	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
4577	-17.32	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
4578	-17.37	kd	CGS001-10857	PGRMC1	-			
4579	-17.42	kd	CGS001-23510	KCTD2	-			
4580	-17.44	kd	CGS001-4976	OPA1	-			
4581	-17.48	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
4582	-17.61	oe	ccsbBroad304_04194	ELL3	-			
4583	-17.62	kd	CGS001-27125	AFF4	-			
4584	-17.62	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
4585	-17.64	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
4586	-17.64	kd	CGS001-10287	RGS19	Regulators of G-protein signaling			
4587	-17.66	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
4588	-17.67	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
4589	-17.67	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
4590	-17.68	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
4591	-17.68	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
4592	-17.73	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
4593	-17.73	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
4594	-17.75	kd	CGS001-2645	GCK	Hexokinases			
4595	-17.76	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
4596	-17.84	kd	CGS001-28969	BZW2	-			
4597	-17.87	kd	CGS001-5591	PRKDC	Other PIKK family kinases			
4598	-17.89	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4599	-17.92	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
4600	-17.94	kd	CGS001-6387	CXCL12	Endogenous ligands			
4601	-18	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
4602	-18.02	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
4603	-18.04	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
4604	-18.12	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
4605	-18.14	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
4606	-18.16	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
4607	-18.16	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
4608	-18.17	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
4609	-18.17	oe	ccsbBroad304_10491	PFKL	-			
4610	-18.2	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
4611	-18.22	kd	CGS001-1512	CTSH	Cathepsins			
4612	-18.26	kd	CGS001-3119	HLA-DQB1	Immunoglobulin superfamily / C1-set domain containing			
4613	-18.29	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
4614	-18.31	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
4615	-18.33	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
4616	-18.38	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
4617	-18.44	oe	ccsbBroad304_00152	BCAT2	-			
4618	-18.45	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
4619	-18.45	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
4620	-18.51	kd	CGS001-1632	ECI1	-			
4621	-18.52	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
4622	-18.52	kd	CGS001-190	NR0B1	DAX-like receptors			
4623	-18.53	kd	CGS001-7915	ALDH5A1	Aldehyde dehydrogenases			
4624	-18.63	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
4625	-18.64	oe	ccsbBroad304_09881	RFX6	-			
4626	-18.68	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
4627	-18.69	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
4628	-18.7	cp	BRD-A87387433	cefpodoxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4629	-18.7	kd	CGS001-399694	SHC4	SH2 domain containing			
4630	-18.76	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
4631	-18.78	kd	CGS001-2787	GNG5	-			
4632	-18.83	kd	CGS001-335	APOA1	Apolipoproteins			
4633	-18.83	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
4634	-18.84	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
4635	-18.86	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
4636	-18.88	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
4637	-18.9	oe	ccsbBroad304_07208	NRIP1	-			
4638	-18.91	kd	CGS001-2639	GCDH	-			
4639	-18.97	kd	CGS001-310	ANXA7	Annexins			
4640	-18.99	kd	CGS001-4680	CEACAM6	CD molecules			
4641	-19.02	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
4642	-19.04	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
4643	-19.12	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
4644	-19.14	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
4645	-19.18	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
4646	-19.22	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
4647	-19.23	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
4648	-19.26	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
4649	-19.27	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
4650	-19.27	kd	CGS001-5684	PSMA3	Proteasome subunits			
4651	-19.28	oe	ccsbBroad304_09254	PAQR8	-			
4652	-19.32	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
4653	-19.37	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
4654	-19.37	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
4655	-19.4	kd	CGS001-4758	NEU1	-			
4656	-19.41	kd	CGS001-4947	OAZ2	-			
4657	-19.43	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
4658	-19.44	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
4659	-19.47	oe	ccsbBroad304_06094	DFFA	-			
4660	-19.55	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
4661	-19.6	oe	ccsbBroad304_03746	CDC42SE1	-			
4662	-19.61	kd	CGS001-8409	UXT	-			
4663	-19.7	oe	ccsbBroad304_00282	CDKN1A	-			
4664	-19.72	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
4665	-19.74	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
4666	-19.74	kd	CGS001-1374	CPT1A	-			
4667	-19.76	oe	ccsbBroad304_01862	YEATS4	-			
4668	-19.79	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
4669	-19.8	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
4670	-19.81	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
4671	-19.81	kd	CGS001-2115	ETV1	ETS Transcription Factors			
4672	-19.82	kd	CGS001-351	APP	Endogenous ligands			
4673	-19.82	oe	ccsbBroad304_06683	FURIN	Subtilisin			
4674	-19.85	kd	CGS001-6894	TARBP1	-			
4675	-19.9	cp	BRD-M41783010	acamprosate	Glutamate receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B, GRM5	Glutamate receptor antagonist
4676	-19.97	kd	CGS001-8655	DYNLL1	Cytoplasmic dyneins			
4677	-19.97	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
4678	-19.97	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
4679	-20.01	kd	CGS001-29890	RBM15B	RNA binding motif (RRM) containing			
4680	-20.02	oe	ccsbBroad304_03080	C16ORF80	-			
4681	-20.03	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
4682	-20.04	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
4683	-20.06	oe	ccsbBroad304_01150	PCCB	Carboxylases			
4684	-20.07	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
4685	-20.08	kd	CGS001-133690	CAPSL	EF-hand domain containing			
4686	-20.11	oe	ccsbBroad304_00020	ACY1	-			
4687	-20.11	kd	CGS001-2783	GNB2	WD repeat domain containing			
4688	-20.14	oe	ccsbBroad304_00519	ETFB	-			
4689	-20.17	kd	CGS001-5050	PAFAH1B3	-			
4690	-20.24	kd	CGS001-10097	ACTR2	-			
4691	-20.25	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
4692	-20.31	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
4693	-20.33	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
4694	-20.35	kd	CGS001-10421	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4695	-20.38	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
4696	-20.4	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
4697	-20.44	kd	CGS001-150962	PUS10	-			
4698	-20.45	oe	ccsbBroad304_00072	ANXA7	Annexins			
4699	-20.48	oe	ccsbBroad304_02716	NMNAT2	-			
4700	-20.5	kd	CGS001-10972	TMED10	-			
4701	-20.53	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
4702	-20.53	kd	CGS001-4012	LNPEP	Aminopeptidase N			
4703	-20.55	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
4704	-20.61	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
4705	-20.65	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
4706	-20.65	kd	CGS001-4086	SMAD1	SMADs			
4707	-20.65	kd	CGS001-7905	REEP5	Receptor accessory proteins			
4708	-20.68	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
4709	-20.75	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
4710	-20.82	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4711	-20.82	kd	CGS001-2242	FES	Fer family			
4712	-20.86	kd	CGS001-55312	RFK	-			
4713	-20.87	kd	CGS001-257397	TAB3	-			
4714	-20.9	kd	CGS001-2108	ETFA	-			
4715	-20.91	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
4716	-21.03	kd	CGS001-133522	PPARGC1B	RNA binding motif (RRM) containing			
4717	-21.04	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
4718	-21.04	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
4719	-21.04	kd	CGS001-36	ACADSB	-			
4720	-21.05	kd	CGS001-677	ZFP36L1	RING-type (C3HC4) zinc fingers			
4721	-21.05	kd	CGS001-2534	FYN	Src family			
4722	-21.05	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
4723	-21.06	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
4724	-21.06	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
4725	-21.1	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
4726	-21.11	kd	CGS001-2155	F7	Chymotrypsin			
4727	-21.11	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
4728	-21.12	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
4729	-21.16	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
4730	-21.17	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
4731	-21.19	kd	CGS001-8576	STK16	NAK family			
4732	-21.35	kd	CGS001-388677	NOTCH2NL	-			
4733	-21.36	kd	CGS001-8872	CDC123	-			
4734	-21.37	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
4735	-21.37	kd	CGS001-84328	LZIC	-			
4736	-21.37	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
4737	-21.39	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4738	-21.4	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
4739	-21.4	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
4740	-21.42	oe	ccsbBroad304_11405	UBE3C	-			
4741	-21.44	oe	ccsbBroad304_01662	TFDP2	-			
4742	-21.44	oe	ccsbBroad304_03591	ETNK1	-			
4743	-21.45	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
4744	-21.47	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
4745	-21.47	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
4746	-21.51	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
4747	-21.54	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
4748	-21.57	kd	CGS001-54108	CHRAC1	-			
4749	-21.58	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
4750	-21.6	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
4751	-21.67	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
4752	-21.71	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
4753	-21.74	oe	ccsbBroad304_06862	RGS3	-			
4754	-21.82	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
4755	-21.88	kd	CGS001-5063	PAK3	PAKA subfamily			
4756	-21.89	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
4757	-21.93	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
4758	-21.94	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4759	-21.95	kd	CGS001-11151	CORO1A	Coronins			
4760	-21.96	oe	ccsbBroad304_06549	SMAD3	SMADs			
4761	-21.99	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
4762	-22.05	kd	CGS001-4938	OAS1	-			
4763	-22.11	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
4764	-22.16	cc		Interleukins GOF	-			
4765	-22.21	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
4766	-22.21	kd	CGS001-8140	SLC7A5	SLC7 family			
4767	-22.25	kd	CGS001-4303	FOXO4	Forkhead boxes			
4768	-22.32	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4769	-22.36	kd	CGS001-125965	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
4770	-22.39	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
4771	-22.39	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
4772	-22.4	kd	CGS001-6934	TCF7L2	-			
4773	-22.42	kd	CGS001-114785	MBD6	-			
4774	-22.43	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
4775	-22.54	kd	CGS001-84971	ATG4D	-			
4776	-22.55	oe	ccsbBroad304_13998	PDXK	-			
4777	-22.55	kd	CGS001-6469	SHH	-			
4778	-22.55	kd	CGS001-4763	NF1	-			
4779	-22.56	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4780	-22.58	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
4781	-22.59	kd	CGS001-22794	CASC3	-			
4782	-22.62	kd	CGS001-3669	ISG20	-			
4783	-22.64	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
4784	-22.65	kd	CGS001-57822	GRHL3	-			
4785	-22.7	cc		Kruppel like transcription factors LOF	-			
4786	-22.71	kd	CGS001-2597	GAPDH	-			
4787	-22.74	kd	CGS001-2887	GRB10	Pleckstrin homology (PH) domain containing			
4788	-22.76	kd	CGS001-7013	TERF1	-			
4789	-22.77	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
4790	-22.8	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
4791	-22.87	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
4792	-22.89	oe	ccsbBroad304_02386	EIF1B	-			
4793	-22.9	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
4794	-22.9	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
4795	-22.91	kd	CGS001-2254	FGF9	Endogenous ligands			
4796	-22.93	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
4797	-22.94	kd	CGS001-79073	TMEM109	-			
4798	-22.95	kd	CGS001-7415	VCP	ATPases / AAA-type			
4799	-22.96	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
4800	-22.96	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
4801	-23	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
4802	-23.01	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
4803	-23.03	kd	CGS001-222894	FERD3L	Basic helix-loop-helix proteins			
4804	-23.03	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
4805	-23.05	oe	ccsbBroad304_03506	AURKAIP1	-			
4806	-23.06	kd	CGS001-5245	PHB	-			
4807	-23.1	oe	ccsbBroad304_00489	EHHADH	-			
4808	-23.15	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
4809	-23.18	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
4810	-23.19	kd	CGS001-64754	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
4811	-23.2	cp	BRD-K70358946	aripiprazole	Serotonin receptor agonist		DRD2, HTR1A, HTR2A, HRH1, HTR1B, HTR1D, HTR2C, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR1E, HTR3A, HTR6, HTR7	Serotonin receptor agonist, Serotonin receptor antagonist
4812	-23.21	oe	ccsbBroad304_08802	ELAC2	-			
4813	-23.22	kd	CGS001-54536	EXOC6	-			
4814	-23.27	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
4815	-23.28	kd	CGS001-8575	PRKRA	-			
4816	-23.29	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
4817	-23.33	cp	BRD-A87125127	3-matida	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4818	-23.36	cp	BRD-A24381660	zeranol	Estrogen receptor agonist			Estrogen receptor agonist
4819	-23.39	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
4820	-23.41	kd	CGS001-51290	ERGIC2	-			
4821	-23.42	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
4822	-23.51	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
4823	-23.57	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
4824	-23.57	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
4825	-23.57	kd	CGS001-10362	HMG20B	High mobility group / Non-canonical			
4826	-23.58	oe	ccsbBroad304_02676	PHB2	-			
4827	-23.6	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
4828	-23.6	kd	CGS001-64147	KIF9	Kinesins			
4829	-23.62	kd	CGS001-4043	LRPAP1	-			
4830	-23.63	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
4831	-23.63	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
4832	-23.64	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
4833	-23.66	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
4834	-23.69	kd	CGS001-9868	TOMM70A	Tetratricopeptide (TTC) repeat domain containing			
4835	-23.7	kd	CGS001-64121	RRAGC	-			
4836	-23.73	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
4837	-23.73	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
4838	-23.73	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
4839	-23.75	kd	CGS001-10628	TXNIP	-			
4840	-23.78	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
4841	-23.82	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
4842	-23.82	oe	ccsbBroad304_02837	BHMT2	-			
4843	-23.83	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
4844	-23.83	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4845	-23.84	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
4846	-23.86	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
4847	-23.89	kd	CGS001-51005	AMDHD2	-			
4848	-23.91	kd	CGS001-170591	S100Z	EF-hand domain containing			
4849	-23.94	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
4850	-23.97	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
4851	-24.02	kd	CGS001-85004	RERG	-			
4852	-24.03	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
4853	-24.03	kd	CGS001-4067	LYN	Src family			
4854	-24.03	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
4855	-24.05	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
4856	-24.12	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
4857	-24.15	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
4858	-24.16	kd	CGS001-3608	ILF2	-			
4859	-24.23	cp	BRD-K33312228	halometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4860	-24.23	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
4861	-24.24	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
4862	-24.3	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
4863	-24.32	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
4864	-24.33	cp	BRD-K66896231	BRD-K66896231	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
4865	-24.33	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4866	-24.36	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
4867	-24.37	cc		Aldehyde dehydrogenases LOF	-			
4868	-24.37	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
4869	-24.41	oe	ccsbBroad304_00568	FHL2	-			
4870	-24.41	kd	CGS001-3033	HADH	-			
4871	-24.43	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
4872	-24.43	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
4873	-24.44	kd	CGS001-6185	RPN2	-			
4874	-24.46	oe	ccsbBroad304_02822	ARFIP2	-			
4875	-24.5	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
4876	-24.52	kd	CGS001-4173	MCM4	-			
4877	-24.57	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
4878	-24.57	oe	ccsbBroad304_00881	IRF5	-			
4879	-24.58	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
4880	-24.65	kd	CGS001-9352	TXNL1	-			
4881	-24.65	kd	CGS001-894	CCND2	-			
4882	-24.66	kd	CGS001-890	CCNA2	-			
4883	-24.71	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
4884	-24.72	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
4885	-24.75	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
4886	-24.79	oe	ccsbBroad304_02230	HERPUD1	-			
4887	-24.81	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
4888	-24.88	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
4889	-24.88	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
4890	-24.89	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
4891	-24.98	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
4892	-24.98	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
4893	-25.01	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
4894	-25.06	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
4895	-25.06	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
4896	-25.15	oe	ccsbBroad304_02533	NOXA1	-			
4897	-25.15	kd	CGS001-558	AXL	Fibronectin type III domain containing			
4898	-25.19	oe	ccsbBroad304_08325	LIPT1	-			
4899	-25.2	oe	ccsbBroad304_00146	BAD	-			
4900	-25.22	kd	CGS001-3551	IKBKB	IKK family			
4901	-25.24	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
4902	-25.26	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
4903	-25.28	kd	CGS001-308	ANXA5	Annexins			
4904	-25.33	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
4905	-25.35	kd	CGS001-801	CALM1	EF-hand domain containing			
4906	-25.36	kd	CGS001-1738	DLD	-			
4907	-25.4	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
4908	-25.43	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
4909	-25.44	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
4910	-25.45	kd	CGS001-3718	JAK3	Janus kinase (JakA) family			
4911	-25.47	kd	CGS001-1604	CD55	CD molecules			
4912	-25.52	cc		HMGCR inhibitor	-			
4913	-25.52	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
4914	-25.54	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
4915	-25.54	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
4916	-25.63	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
4917	-25.64	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
4918	-25.65	kd	CGS001-11212	PROSC	-			
4919	-25.67	kd	CGS001-7982	ST7	-			
4920	-25.71	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
4921	-25.71	oe	ccsbBroad304_03652	EXOC2	-			
4922	-25.74	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
4923	-25.76	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
4924	-25.78	kd	CGS001-124641	OVCA2	-			
4925	-25.78	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
4926	-25.79	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
4927	-25.83	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
4928	-25.84	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
4929	-25.84	kd	CGS001-345611	IRGM	-			
4930	-25.85	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
4931	-25.86	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
4932	-25.87	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
4933	-25.91	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4934	-25.96	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
4935	-25.98	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
4936	-25.99	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
4937	-26.02	kd	CGS001-2778	GNAS	-			
4938	-26.02	kd	CGS001-1457	CSNK2A1	Casein kinase 2 (CK2) family			
4939	-26.02	kd	CGS001-19	ABCA1	ATP binding cassette transporters / subfamily A			
4940	-26.05	kd	CGS001-392	ARHGAP1	Rho GTPase activating proteins			
4941	-26.12	kd	CGS001-11320	MGAT4A	-			
4942	-26.12	oe	ccsbBroad304_01556	SMARCB1	-			
4943	-26.17	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
4944	-26.2	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
4945	-26.2	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
4946	-26.25	kd	CGS001-6715	SRD5A1	-			
4947	-26.31	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
4948	-26.33	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
4949	-26.37	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
4950	-26.37	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
4951	-26.37	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
4952	-26.4	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
4953	-26.42	oe	ccsbBroad304_14020	SH3BP5	-			
4954	-26.46	kd	CGS001-5981	RFC1	ATPases / AAA-type			
4955	-26.46	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
4956	-26.47	kd	CGS001-151126	ZNF385B	-			
4957	-26.5	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
4958	-26.52	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
4959	-26.55	kd	CGS001-9111	NMI	-			
4960	-26.59	kd	CGS001-290	ANPEP	Aminopeptidase N			
4961	-26.74	kd	CGS001-7541	ZFP161	-			
4962	-26.76	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
4963	-26.8	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
4964	-26.8	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
4965	-26.99	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
4966	-27	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
4967	-27.02	kd	CGS001-51203	NUSAP1	-			
4968	-27.06	kd	CGS001-57215	THAP11	THAP (C2CH-type zinc finger) domain containing			
4969	-27.09	kd	CGS001-3980	LIG3	-			
4970	-27.1	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
4971	-27.18	oe	ccsbBroad304_00819	IDH3B	-			
4972	-27.24	kd	CGS001-5144	PDE4D	Phosphodiesterases			
4973	-27.25	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
4974	-27.28	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
4975	-27.29	kd	CGS001-10468	FST	-			
4976	-27.33	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
4977	-27.37	kd	CGS001-1152	CKB	-			
4978	-27.4	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
4979	-27.43	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
4980	-27.45	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
4981	-27.54	oe	ccsbBroad304_03773	CIAPIN1	-			
4982	-27.6	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
4983	-27.63	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
4984	-27.65	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
4985	-27.66	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
4986	-27.68	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
4987	-27.75	kd	CGS001-8833	GMPS	-			
4988	-27.78	kd	CGS001-23014	FBXO21	F-boxes / other			
4989	-27.79	kd	CGS001-4893	NRAS	RAS subfamily			
4990	-27.84	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
4991	-27.84	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4992	-27.86	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
4993	-27.86	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
4994	-27.87	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
4995	-27.89	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
4996	-27.93	kd	CGS001-4830	NME1	-			
4997	-27.98	kd	CGS001-5682	PSMA1	Proteasome subunits			
4998	-27.99	oe	ccsbBroad304_00600	FYN	Src family			
4999	-28	cc		General transcription factors group 2 LOF	-			
5000	-28	oe	ccsbBroad304_00552	FEN1	-			
5001	-28.01	kd	CGS001-284	ANGPT1	Fibrinogen C domain containing			
5002	-28.02	kd	CGS001-55612	FERMT1	Fermitins			
5003	-28.08	oe	ccsbBroad304_07145	ZFP161	-			
5004	-28.14	kd	CGS001-109	ADCY3	Adenylyl cyclases			
5005	-28.21	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
5006	-28.22	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
5007	-28.31	kd	CGS001-55206	SBNO1	-			
5008	-28.38	kd	CGS001-165082	GPR113	Adhesion Class GPCRs			
5009	-28.39	kd	CGS001-892	CCNC	-			
5010	-28.41	kd	CGS001-64425	POLR1E	RNA polymerase subunits			
5011	-28.44	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
5012	-28.49	kd	CGS001-2782	GNB1	WD repeat domain containing			
5013	-28.52	kd	CGS001-8996	NOL3	-			
5014	-28.58	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
5015	-28.61	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
5016	-28.66	kd	CGS001-8572	PDLIM4	-			
5017	-28.67	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
5018	-28.71	kd	CGS001-3163	HMOX2	Haem oxygenase			
5019	-28.72	kd	CGS001-23043	TNIK	MSN subfamily			
5020	-28.73	kd	CGS001-7270	TTF1	-			
5021	-28.75	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5022	-28.77	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
5023	-28.77	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
5024	-28.83	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
5025	-28.84	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
5026	-28.85	oe	ccsbBroad304_00728	HBE1	-			
5027	-28.9	kd	CGS001-635	BHMT	-			
5028	-28.95	cc		RAF inhibitor	-			
5029	-29.02	oe	ccsbBroad304_01483	SAT1	-			
5030	-29.03	cp	BRD-K18895904	olanzapine	Dopamine receptor antagonist		DRD2, HTR2A, HTR2C, DRD1, DRD3, DRD4, HRH1, HTR1A, HTR1B, HTR1D, HTR1E, HTR6, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C8, DRD5, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH2, HRH4, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
5031	-29.03	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
5032	-29.09	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
5033	-29.09	kd	CGS001-5562	PRKAA1	AMPK subfamily			
5034	-29.1	oe	ccsbBroad304_07017	SUOX	-			
5035	-29.12	kd	CGS001-56916	SMARCAD1	-			
5036	-29.15	kd	CGS001-9344	TAOK2	TAO subfamily			
5037	-29.29	oe	ccsbBroad304_06449	ILF3	-			
5038	-29.31	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
5039	-29.31	kd	CGS001-375	ARF1	ADP-ribosylation factors			
5040	-29.36	kd	CGS001-5184	PEPD	Methionyl aminopeptidase			
5041	-29.37	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
5042	-29.42	kd	CGS001-89766	UMODL1	-			
5043	-29.47	kd	CGS001-5693	PSMB5	Proteasome subunits			
5044	-29.48	kd	CGS001-9134	CCNE2	-			
5045	-29.49	kd	CGS001-8639	AOC3	Oxidoreductases			
5046	-29.5	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
5047	-29.5	oe	ccsbBroad304_06134	ECH1	-			
5048	-29.54	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
5049	-29.55	kd	CGS001-6195	RPS6KA1	RSK subfamily			
5050	-29.6	kd	CGS001-91949	COG7	Components of oligomeric golgi complex			
5051	-29.61	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
5052	-29.62	kd	CGS001-8050	PDHX	-			
5053	-29.71	oe	ccsbBroad304_00459	DPYD	-			
5054	-29.73	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
5055	-29.73	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
5056	-29.75	kd	CGS001-330	BIRC3	Inhibitors of apoptosis (IAP) protein family			
5057	-29.77	kd	CGS001-3934	LCN2	Lipocalins			
5058	-29.83	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
5059	-29.87	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
5060	-29.87	kd	CGS001-3171	FOXA3	Forkhead boxes			
5061	-29.88	kd	CGS001-84936	ZFYVE19	Zinc fingers, FYVE domain containing			
5062	-29.93	kd	CGS001-54623	PAF1	-			
5063	-29.96	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
5064	-29.96	oe	ccsbBroad304_06159	CTTN	-			
5065	-29.97	kd	CGS001-55526	DHTKD1	-			
5066	-29.99	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
5067	-30.03	oe	ccsbBroad304_02092	SYNGR3	-			
5068	-30.14	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
5069	-30.18	kd	CGS001-11284	PNKP	-			
5070	-30.19	kd	CGS001-1677	DFFB	-			
5071	-30.24	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
5072	-30.28	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
5073	-30.29	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
5074	-30.29	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
5075	-30.34	kd	CGS001-3590	IL11RA	IL-6 receptor family			
5076	-30.4	kd	CGS001-338	APOB	Apolipoproteins			
5077	-30.41	kd	CGS001-27076	LYPD3	-			
5078	-30.41	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
5079	-30.43	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5080	-30.45	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
5081	-30.47	oe	ccsbBroad304_02438	FAM3C	-			
5082	-30.51	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
5083	-30.54	kd	CGS001-5663	PSEN1	Presenilin			
5084	-30.61	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
5085	-30.66	cp	BRD-K88679075	methandriol	Androgenic steroid			Androgenic steroid
5086	-30.66	kd	CGS001-340371	NRBP2	NRBP family			
5087	-30.71	kd	CGS001-2247	FGF2	Endogenous ligands			
5088	-30.72	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
5089	-30.75	kd	CGS001-5110	PCMT1	-			
5090	-30.75	kd	CGS001-8738	CRADD	-			
5091	-30.79	kd	CGS001-9146	HGS	Zinc fingers, FYVE domain containing			
5092	-30.92	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
5093	-31.15	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
5094	-31.17	kd	CGS001-7597	ZBTB25	BTB/POZ domain containing			
5095	-31.21	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
5096	-31.22	oe	ccsbBroad304_02671	ECD	-			
5097	-31.25	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
5098	-31.26	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
5099	-31.28	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
5100	-31.28	kd	CGS001-8553	BHLHE40	Basic helix-loop-helix proteins			
5101	-31.29	kd	CGS001-3601	IL15RA	IL-2 receptor family			
5102	-31.39	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
5103	-31.4	kd	CGS001-8780	RIOK3	RIO3 subfamily			
5104	-31.48	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
5105	-31.5	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
5106	-31.54	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
5107	-31.57	cc		Proteasome Pathway LOF	-			
5108	-31.63	oe	ccsbBroad304_01974	RNASET2	-			
5109	-31.65	kd	CGS001-10253	SPRY2	-			
5110	-31.65	kd	CGS001-9887	SMG7	-			
5111	-31.65	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
5112	-31.66	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
5113	-31.67	kd	CGS001-1069	CETN2	EF-hand domain containing			
5114	-31.68	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
5115	-31.7	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
5116	-31.72	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
5117	-31.8	kd	CGS001-5986	RFNG	Beta 3-glycosyltransferases			
5118	-31.81	kd	CGS001-2852	GPER	-			
5119	-31.82	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
5120	-31.83	cp	BRD-K29530284	amlexanox	Histamine receptor modulator		FGF1, IL3, S100A12, S100A13	Histamine receptor modulator
5121	-31.86	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5122	-31.89	cp	BRD-K31491153	1-phenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
5123	-31.98	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
5124	-32.03	oe	ccsbBroad304_00171	BNIP3L	-			
5125	-32.04	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
5126	-32.04	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
5127	-32.05	kd	CGS001-7360	UGP2	-			
5128	-32.05	kd	CGS001-760	CA2	Carbonic anhydrases			
5129	-32.06	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
5130	-32.07	kd	CGS001-1528	CYB5A	Cytochrome b genes			
5131	-32.1	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5132	-32.1	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
5133	-32.15	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
5134	-32.16	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
5135	-32.17	kd	CGS001-103	ADAR	-			
5136	-32.21	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
5137	-32.22	kd	CGS001-6988	TCTA	-			
5138	-32.23	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
5139	-32.24	kd	CGS001-64080	RBKS	-			
5140	-32.25	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
5141	-32.28	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
5142	-32.28	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
5143	-32.3	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
5144	-32.35	kd	CGS001-481	ATP1B1	ATPases / P-type			
5145	-32.38	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
5146	-32.4	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
5147	-32.43	kd	CGS001-8795	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
5148	-32.44	kd	CGS001-10841	FTCD	-			
5149	-32.48	kd	CGS001-7421	VDR	Vitamin D receptors			
5150	-32.57	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
5151	-32.61	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5152	-32.61	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
5153	-32.65	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
5154	-32.67	cp	BRD-A80383043	BRD-A80383043	Glutamate receptor agonist		GRM1, GRM2	Glutamate receptor agonist, Glutamate receptor antagonist
5155	-32.67	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5156	-32.68	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
5157	-32.68	oe	ccsbBroad304_06535	LPL	-			
5158	-32.68	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
5159	-32.71	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
5160	-32.74	kd	CGS001-51586	MED15	-			
5161	-32.77	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
5162	-32.77	kd	CGS001-3575	IL7R	IL-2 receptor family			
5163	-32.82	oe	ccsbBroad304_07724	KDELR2	-			
5164	-32.83	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
5165	-32.86	kd	CGS001-23384	SPECC1L	-			
5166	-32.93	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
5167	-32.95	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
5168	-32.95	kd	CGS001-2896	GRN	-			
5169	-32.99	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
5170	-33.06	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
5171	-33.06	kd	CGS001-3909	LAMA3	Laminins			
5172	-33.08	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
5173	-33.08	kd	CGS001-221393	GPR115	Adhesion Class GPCRs			
5174	-33.14	cp	BRD-K19462402	buflomedil	Adrenergic receptor antagonist		CACNA1C	Adrenergic receptor antagonist, Calcium channel blocker
5175	-33.14	kd	CGS001-51181	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5176	-33.14	oe	ccsbBroad304_06089	DDIT3	-			
5177	-33.17	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
5178	-33.22	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
5179	-33.23	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
5180	-33.37	kd	CGS001-1861	TOR1A	-			
5181	-33.41	kd	CGS001-29883	CNOT7	-			
5182	-33.42	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
5183	-33.48	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
5184	-33.49	kd	CGS001-8408	ULK1	Unc-51-like kinase (ULK) family			
5185	-33.51	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
5186	-33.51	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
5187	-33.56	oe	ccsbBroad304_00615	GAPDH	-			
5188	-33.56	kd	CGS001-7919	DDX39B	DEAD-boxes			
5189	-33.56	oe	ccsbBroad304_08660	SMARCAD1	-			
5190	-33.61	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
5191	-33.61	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
5192	-33.72	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
5193	-33.75	kd	CGS001-7165	TPD52L2	-			
5194	-33.76	kd	CGS001-64863	METTL4	-			
5195	-33.77	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
5196	-33.77	kd	CGS001-64422	ATG3	-			
5197	-33.83	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
5198	-33.88	oe	ccsbBroad304_02313	ACTR3	-			
5199	-33.91	kd	CGS001-55008	HERC6	-			
5200	-33.91	kd	CGS001-55722	CEP72	-			
5201	-33.93	kd	CGS001-26298	EHF	-			
5202	-33.96	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
5203	-33.97	kd	CGS001-150280	HORMAD2	-			
5204	-33.99	kd	CGS001-841	CASP8	Caspases			
5205	-34.02	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
5206	-34.06	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
5207	-34.07	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
5208	-34.08	oe	ccsbBroad304_07088	TP53	-			
5209	-34.11	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
5210	-34.17	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
5211	-34.18	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
5212	-34.2	kd	CGS001-2109	ETFB	-			
5213	-34.3	kd	CGS001-81544	GDPD5	-			
5214	-34.32	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
5215	-34.32	kd	CGS001-10491	CRTAP	-			
5216	-34.33	kd	CGS001-5535	PPP3R2	EF-hand domain containing			
5217	-34.36	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
5218	-34.38	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
5219	-34.4	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
5220	-34.42	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
5221	-34.44	kd	CGS001-64710	NUCKS1	-			
5222	-34.48	oe	ccsbBroad304_03040	NKIRAS2	-			
5223	-34.5	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
5224	-34.5	kd	CGS001-3420	IDH3B	-			
5225	-34.52	kd	CGS001-388650	FAM69A	-			
5226	-34.53	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
5227	-34.56	kd	CGS001-10105	PPIF	-			
5228	-34.57	kd	CGS001-4602	MYB	-			
5229	-34.6	kd	CGS001-80237	ELL3	-			
5230	-34.64	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
5231	-34.65	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
5232	-34.75	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
5233	-34.77	oe	ccsbBroad304_00370	CS	-			
5234	-34.77	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
5235	-34.79	kd	CGS001-2182	ACSL4	Acyl-CoA synthetase family			
5236	-34.86	kd	CGS001-10813	UTP14A	-			
5237	-34.98	oe	ccsbBroad304_07616	ZNF238	-			
5238	-34.98	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
5239	-35	oe	ccsbBroad304_02857	BAMBI	-			
5240	-35.05	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
5241	-35.1	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
5242	-35.14	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
5243	-35.27	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
5244	-35.29	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5245	-35.3	kd	CGS001-1198	CLK3	CDC-like kinases			
5246	-35.31	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
5247	-35.34	kd	CGS001-26993	AKAP8L	-			
5248	-35.41	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
5249	-35.43	oe	ccsbBroad304_06085	DCK	-			
5250	-35.43	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
5251	-35.45	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
5252	-35.54	oe	ccsbBroad304_09006	RPF1	-			
5253	-35.54	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
5254	-35.66	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
5255	-35.77	kd	CGS001-1363	CPE	Carboxypeptidase A			
5256	-35.8	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
5257	-35.82	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
5258	-35.82	kd	CGS001-5894	RAF1	RAF family			
5259	-35.87	kd	CGS001-3569	IL6	Interferons			
5260	-35.88	oe	ccsbBroad304_07287	HYAL2	-			
5261	-35.88	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
5262	-35.96	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
5263	-35.96	cp	BRD-A02189320	met-leu-phe	-666			-666
5264	-35.98	kd	CGS001-10682	EBP	-			
5265	-35.99	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
5266	-36.11	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
5267	-36.16	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
5268	-36.18	oe	ccsbBroad304_08825	LHPP	-			
5269	-36.21	cp	BRD-A07395371	esmolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
5270	-36.25	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
5271	-36.31	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
5272	-36.35	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
5273	-36.38	cp	BRD-M47937986	cefatrizine	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5274	-36.4	kd	CGS001-54815	GATAD2A	GATA zinc finger domain containing			
5275	-36.47	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
5276	-36.48	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
5277	-36.48	kd	CGS001-9650	MTFR1	-			
5278	-36.48	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
5279	-36.55	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
5280	-36.59	oe	ccsbBroad304_07528	DMTF1	-			
5281	-36.62	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
5282	-36.65	oe	ccsbBroad304_02487	TXNIP	-			
5283	-36.67	oe	ccsbBroad304_03497	TXNL4B	-			
5284	-36.7	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
5285	-36.7	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
5286	-36.71	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
5287	-36.72	oe	ccsbBroad304_01664	TGFA	-			
5288	-36.79	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
5289	-36.79	kd	CGS001-3046	HBE1	-			
5290	-36.85	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
5291	-36.92	kd	CGS001-22796	COG2	Components of oligomeric golgi complex			
5292	-36.97	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
5293	-36.99	kd	CGS001-9354	UBE4A	U-box domain containing			
5294	-36.99	kd	CGS001-5217	PFN2	-			
5295	-36.99	oe	ccsbBroad304_01659	TERF1	-			
5296	-36.99	oe	ccsbBroad304_01165	PDK1	-			
5297	-37.05	oe	ccsbBroad304_07029	TADA2A	-			
5298	-37.05	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
5299	-37.06	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
5300	-37.07	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
5301	-37.07	kd	CGS001-116931	MED12L	-			
5302	-37.11	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
5303	-37.12	kd	CGS001-2274	FHL2	-			
5304	-37.15	kd	CGS001-51097	SCCPDH	-			
5305	-37.18	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
5306	-37.18	kd	CGS001-79796	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
5307	-37.2	kd	CGS001-58477	SRPRB	-			
5308	-37.2	kd	CGS001-1854	DUT	-			
5309	-37.23	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5310	-37.31	kd	CGS001-6603	SMARCD2	-			
5311	-37.32	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
5312	-37.34	cp	BRD-K69650333	idarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
5313	-37.41	oe	ccsbBroad304_06523	LIG1	-			
5314	-37.44	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
5315	-37.52	kd	CGS001-9488	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
5316	-37.54	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
5317	-37.63	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
5318	-37.68	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
5319	-37.69	oe	ccsbBroad304_07128	VHL	-			
5320	-37.73	kd	CGS001-9252	RPS6KA5	MSK subfamily			
5321	-37.73	kd	CGS001-10023	FRAT1	-			
5322	-37.73	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
5323	-37.74	kd	CGS001-4047	LSS	Lanosterol biosynthesis pathway			
5324	-37.75	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
5325	-37.8	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
5326	-37.86	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
5327	-37.87	kd	CGS001-7079	TIMP4	-			
5328	-37.88	kd	CGS001-23076	RRP1B	-			
5329	-37.91	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
5330	-37.94	cc		Estrogen receptor agonist	-			
5331	-37.96	kd	CGS001-2674	GFRA1	GDNF receptor family			
5332	-38.05	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
5333	-38.05	kd	CGS001-324	APC	Armadillo repeat containing			
5334	-38.16	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
5335	-38.16	kd	CGS001-3612	IMPA1	Inositol monophosphatase			
5336	-38.26	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
5337	-38.29	kd	CGS001-210	ALAD	-			
5338	-38.3	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
5339	-38.34	oe	ccsbBroad304_07491	IP6K1	-			
5340	-38.34	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
5341	-38.38	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
5342	-38.39	oe	ccsbBroad304_05902	BNIP3	-			
5343	-38.39	oe	ccsbBroad304_08662	MCCC1	-			
5344	-38.42	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
5345	-38.44	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
5346	-38.45	kd	CGS001-26520	TIMM9	-			
5347	-38.56	oe	ccsbBroad304_05947	CCNC	-			
5348	-38.56	kd	CGS001-55556	ENOSF1	-			
5349	-38.58	kd	CGS001-220	ALDH1A3	Aldehyde dehydrogenases			
5350	-38.6	kd	CGS001-4171	MCM2	-			
5351	-38.61	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
5352	-38.69	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
5353	-38.7	kd	CGS001-56731	SLC2A4RG	-			
5354	-38.75	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
5355	-38.77	kd	CGS001-390212	GPR152	GPCR / Class A : Orphans			
5356	-38.78	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
5357	-38.82	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
5358	-38.83	cc		CDK inhibitor	-			
5359	-38.83	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
5360	-38.83	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
5361	-38.84	kd	CGS001-839	CASP6	Caspases			
5362	-38.9	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
5363	-38.91	kd	CGS001-23588	KLHDC2	-			
5364	-38.94	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
5365	-38.94	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
5366	-38.96	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
5367	-39	kd	CGS001-18	ABAT	GABA turnover			
5368	-39.01	kd	CGS001-375133	PI4KAP2	-			
5369	-39.03	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
5370	-39.04	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
5371	-39.05	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
5372	-39.06	kd	CGS001-545	ATR	ATR subfamily			
5373	-39.08	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
5374	-39.08	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
5375	-39.08	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
5376	-39.12	cc		AHSP Pathway LOF	-			
5377	-39.13	cc		Rho GTPase activating proteins LOF	-			
5378	-39.13	kd	CGS001-2878	GPX3	-			
5379	-39.16	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
5380	-39.17	kd	CGS001-275	AMT	-			
5381	-39.19	cp	BRD-K73991644	isoquercetin	Aldose reductase inhibitor		AKR1B1, ACE	Aldose reductase inhibitor
5382	-39.3	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
5383	-39.3	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
5384	-39.32	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
5385	-39.37	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
5386	-39.38	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
5387	-39.38	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
5388	-39.42	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
5389	-39.45	kd	CGS001-126823	KLHDC9	-			
5390	-39.46	kd	CGS001-9122	SLC16A4	SLC16 family of monocarboxylate transporters			
5391	-39.46	oe	ccsbBroad304_01394	RFX4	-			
5392	-39.47	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
5393	-39.5	kd	CGS001-55818	KDM3A	Histone demethylases			
5394	-39.53	kd	CGS001-7849	PAX8	Paired boxes			
5395	-39.56	kd	CGS001-31	ACACA	Carboxylases			
5396	-39.57	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
5397	-39.58	kd	CGS001-369	ARAF	RAF family			
5398	-39.59	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
5399	-39.59	kd	CGS001-54106	TLR9	Toll-like receptor family			
5400	-39.6	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
5401	-39.62	cc		Potassium channel activator	-			
5402	-39.73	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
5403	-39.77	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
5404	-39.83	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
5405	-39.83	kd	CGS001-84890	ADO	-			
5406	-39.84	kd	CGS001-1859	DYRK1A	Dyrk1 subfamily			
5407	-39.85	cc		Sigma receptor antagonist	-			
5408	-39.87	oe	ccsbBroad304_03858	SRPRB	-			
5409	-39.88	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
5410	-39.96	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
5411	-39.96	kd	CGS001-9958	USP15	Ubiquitin-specific peptidases			
5412	-39.99	oe	ccsbBroad304_06828	PYCR1	-			
5413	-40.01	kd	CGS001-6663	SOX10	SRY (sex determining region Y)-boxes			
5414	-40.03	oe	ccsbBroad304_00394	CTSD	Cathepsins			
5415	-40.06	kd	CGS001-23196	FAM120A	-			
5416	-40.06	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
5417	-40.09	cc		Tricyclic antidepressant	-			
5418	-40.19	kd	CGS001-4837	NNMT	-			
5419	-40.19	kd	CGS001-9374	PPT2	-			
5420	-40.21	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
5421	-40.28	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
5422	-40.29	kd	CGS001-54659	UGT1A3	UDP glucuronosyltransferases			
5423	-40.3	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
5424	-40.3	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
5425	-40.31	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
5426	-40.33	kd	CGS001-57504	MTA3	GATA zinc finger domain containing			
5427	-40.33	oe	ccsbBroad304_03479	YTHDF1	-			
5428	-40.34	kd	CGS001-4482	MSRA	-			
5429	-40.35	kd	CGS001-1120	CHKB	-			
5430	-40.35	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
5431	-40.36	oe	ccsbBroad304_06569	MCM5	-			
5432	-40.38	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
5433	-40.39	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
5434	-40.42	kd	CGS001-183	AGT	Endogenous ligands			
5435	-40.42	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
5436	-40.43	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
5437	-40.44	oe	ccsbBroad304_07053	TFPI	-			
5438	-40.44	kd	CGS001-1398	CRK	SH2 domain containing			
5439	-40.47	oe	ccsbBroad304_07024	SYK	Syk family			
5440	-40.47	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
5441	-40.49	kd	CGS001-6455	SH3GL1	-			
5442	-40.52	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
5443	-40.54	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
5444	-40.6	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
5445	-40.65	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5446	-40.71	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
5447	-40.77	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
5448	-40.8	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
5449	-40.83	kd	CGS001-960	CD44	CD molecules			
5450	-40.84	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
5451	-40.84	kd	CGS001-9612	NCOR2	-			
5452	-40.85	kd	CGS001-10987	COPS5	-			
5453	-40.94	kd	CGS001-2853	GPR31	GPCR / Class A : Orphans			
5454	-40.95	kd	CGS001-5329	PLAUR	CD molecules			
5455	-40.96	kd	CGS001-8543	LMO4	-			
5456	-41	kd	CGS001-57154	SMURF1	-			
5457	-41	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
5458	-41.09	kd	CGS001-771	CA12	Carbonic anhydrases			
5459	-41.1	oe	ccsbBroad304_06090	DDOST	-			
5460	-41.15	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
5461	-41.16	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
5462	-41.23	kd	CGS001-7508	XPC	-			
5463	-41.25	oe	ccsbBroad304_01654	TCTA	-			
5464	-41.26	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
5465	-41.26	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
5466	-41.28	kd	CGS001-6098	ROS1	Type XVII RTKs: ROS receptors			
5467	-41.29	cp	BRD-K98493452	honokiol	AKT inhibitor		ALOX5, PTGS1, PTGS2	AKT inhibitor
5468	-41.32	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
5469	-41.34	kd	CGS001-10314	LANCL1	-			
5470	-41.34	kd	CGS001-51805	COQ3	-			
5471	-41.43	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
5472	-41.45	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
5473	-41.47	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
5474	-41.47	kd	CGS001-3553	IL1B	Interleukins and interleukin receptors			
5475	-41.48	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
5476	-41.53	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
5477	-41.67	kd	CGS001-118442	GPR62	GPCR / Class A : Orphans			
5478	-41.69	cc		X linked mental retardation group 1 LOF	-			
5479	-41.79	kd	CGS001-7097	TLR2	Toll-like receptor family			
5480	-41.83	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
5481	-41.84	kd	CGS001-50943	FOXP3	Forkhead boxes			
5482	-41.94	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5483	-41.96	oe	ccsbBroad304_01640	TAF12	-			
5484	-42	kd	CGS001-152	ADRA2C	GPCR / Class A : Adrenoceptors : alpha			
5485	-42.05	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
5486	-42.06	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
5487	-42.12	kd	CGS001-6714	SRC	Src family			
5488	-42.13	kd	CGS001-5230	PGK1	-			
5489	-42.17	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
5490	-42.2	kd	CGS001-4329	ALDH6A1	Aldehyde dehydrogenases			
5491	-42.23	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
5492	-42.25	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
5493	-42.28	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
5494	-42.29	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
5495	-42.32	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
5496	-42.32	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
5497	-42.34	kd	CGS001-9159	PCSK7	Subtilisin			
5498	-42.36	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
5499	-42.38	kd	CGS001-3199	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
5500	-42.46	kd	CGS001-8295	TRRAP	TRRAP subfamily			
5501	-42.47	kd	CGS001-3098	HK1	-			
5502	-42.52	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
5503	-42.63	oe	ccsbBroad304_05985	CFL1	-			
5504	-42.67	kd	CGS001-55577	NAGK	-			
5505	-42.7	oe	ccsbBroad304_08266	PIPOX	-			
5506	-42.71	kd	CGS001-50808	AK3	-			
5507	-42.82	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5508	-42.87	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
5509	-42.9	kd	CGS001-1643	DDB2	WD repeat domain containing			
5510	-42.96	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
5511	-42.97	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
5512	-42.97	kd	CGS001-3654	IRAK1	Interleukin-1 receptor-associated kinase (IRAK) family			
5513	-43.01	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
5514	-43.11	kd	CGS001-8192	CLPP	ATPases / AAA-type			
5515	-43.16	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
5516	-43.21	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
5517	-43.23	kd	CGS001-56882	CDC42SE1	-			
5518	-43.34	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
5519	-43.35	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
5520	-43.36	kd	CGS001-5891	MOK	RCK family			
5521	-43.4	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
5522	-43.4	oe	ccsbBroad304_01183	PGD	-			
5523	-43.41	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
5524	-43.41	kd	CGS001-3030	HADHA	-			
5525	-43.42	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
5526	-43.44	cp	BRD-K54316499	tolterodine	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRM1, CHRM4, CHRM5	Acetylcholine receptor antagonist
5527	-43.46	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
5528	-43.47	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
5529	-43.51	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
5530	-43.54	oe	ccsbBroad304_00118	ATIC	-			
5531	-43.55	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
5532	-43.63	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
5533	-43.68	oe	ccsbBroad304_00975	MAT2A	-			
5534	-43.69	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
5535	-43.78	kd	CGS001-4751	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5536	-43.78	oe	ccsbBroad304_00960	SMAD1	SMADs			
5537	-43.79	kd	CGS001-6856	SYPL1	-			
5538	-43.84	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
5539	-43.87	cp	BRD-K82357231	desloratadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5540	-43.89	kd	CGS001-6119	RPA3	-			
5541	-43.89	kd	CGS001-25801	GCA	EF-hand domain containing			
5542	-43.9	kd	CGS001-327	APEH	Prolyl oligopeptidase			
5543	-43.93	kd	CGS001-5743	PTGS2	Cyclooxygenase			
5544	-43.97	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
5545	-44.06	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
5546	-44.07	kd	CGS001-353	APRT	-			
5547	-44.08	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
5548	-44.1	kd	CGS001-4637	MYL6	EF-hand domain containing			
5549	-44.13	kd	CGS001-81550	TDRD3	Tudor domain containing			
5550	-44.18	kd	CGS001-634	CEACAM1	CD molecules			
5551	-44.32	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
5552	-44.34	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
5553	-44.34	kd	CGS001-7132	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
5554	-44.34	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
5555	-44.37	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
5556	-44.39	kd	CGS001-4801	NFYB	-			
5557	-44.43	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
5558	-44.48	kd	CGS001-55837	EAPP	-			
5559	-44.49	kd	CGS001-10465	PPIH	-			
5560	-44.5	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
5561	-44.52	kd	CGS001-149233	IL23R	IL-12 receptor family			
5562	-44.65	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
5563	-44.66	cp	BRD-K94144010	cotinine	Nicotine metabolite			Nicotine metabolite
5564	-44.66	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
5565	-44.68	cp	BRD-K06388322	pramipexole	Dopamine receptor agonist		DRD3, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
5566	-44.7	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
5567	-44.74	oe	ccsbBroad304_02173	ATG5	-			
5568	-44.74	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
5569	-44.75	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
5570	-44.77	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
5571	-44.79	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
5572	-44.79	kd	CGS001-865	CBFB	-			
5573	-44.83	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5574	-44.85	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
5575	-44.85	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
5576	-44.86	kd	CGS001-7468	WHSC1	Zinc fingers, PHD-type			
5577	-44.89	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
5578	-44.89	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
5579	-44.89	kd	CGS001-11015	KDELR3	-			
5580	-44.93	kd	CGS001-28964	GIT1	Ankyrin repeat domain containing			
5581	-44.94	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
5582	-44.95	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
5583	-44.96	kd	CGS001-2475	MTOR	FRAP subfamily			
5584	-44.98	cp	BRD-K00673382	famotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
5585	-44.98	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
5586	-45.04	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
5587	-45.05	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
5588	-45.06	kd	CGS001-2538	G6PC	-			
5589	-45.07	kd	CGS001-533	ATP6V0B	ATPases / V-type			
5590	-45.14	kd	CGS001-26128	KIAA1279	-			
5591	-45.15	kd	CGS001-56616	DIABLO	-			
5592	-45.19	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
5593	-45.24	kd	CGS001-148103	ZNF599	Zinc fingers, C2H2-type			
5594	-45.27	kd	CGS001-2760	GM2A	-			
5595	-45.28	kd	CGS001-54541	DDIT4	-			
5596	-45.34	kd	CGS001-23271	CAMSAP2	-			
5597	-45.36	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
5598	-45.42	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
5599	-45.43	kd	CGS001-857	CAV1	-			
5600	-45.51	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
5601	-45.52	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
5602	-45.53	kd	CGS001-7316	UBC	-			
5603	-45.54	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
5604	-45.55	kd	CGS001-435	ASL	-			
5605	-45.55	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
5606	-45.57	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
5607	-45.58	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
5608	-45.64	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
5609	-45.65	cc		Ribonucleotide reductase inhibitor	-			
5610	-45.67	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
5611	-45.68	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
5612	-45.7	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
5613	-45.71	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
5614	-45.71	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
5615	-45.74	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
5616	-45.76	kd	CGS001-50813	COPS7A	-			
5617	-45.77	kd	CGS001-1717	DHCR7	-			
5618	-45.81	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
5619	-45.83	cp	BRD-K28849549	mesalazine	Cyclooxygenase inhibitor		PTGS1, PPARG, PTGS2, ALOX5, CHUK, CTNNB1, IKBKB, MPO, NAT1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor, Prostanoid receptor antagonist
5620	-45.88	kd	CGS001-124535	HSF5	-			
5621	-45.89	oe	ccsbBroad304_01061	NAB2	-			
5622	-46	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
5623	-46.07	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
5624	-46.09	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
5625	-46.09	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
5626	-46.12	kd	CGS001-8464	SUPT3H	-			
5627	-46.12	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
5628	-46.12	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
5629	-46.15	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
5630	-46.2	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
5631	-46.22	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
5632	-46.23	oe	ccsbBroad304_02109	XPR1	-			
5633	-46.26	kd	CGS001-7078	TIMP3	-			
5634	-46.29	kd	CGS001-22921	MSRB2	-			
5635	-46.32	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
5636	-46.33	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
5637	-46.33	kd	CGS001-3566	IL4R	IL-2 receptor family			
5638	-46.35	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
5639	-46.35	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5640	-46.35	kd	CGS001-59343	SENP2	-			
5641	-46.37	cp	BRD-A00520476	otenzepad	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
5642	-46.4	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
5643	-46.5	oe	ccsbBroad304_00003	ABAT	GABA turnover			
5644	-46.55	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
5645	-46.57	kd	CGS001-4605	MYBL2	-			
5646	-46.58	kd	CGS001-4300	MLLT3	-			
5647	-46.59	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
5648	-46.6	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
5649	-46.63	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
5650	-46.63	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
5651	-46.65	kd	CGS001-4074	M6PR	-			
5652	-46.66	kd	CGS001-3672	ITGA1	Integrins			
5653	-46.67	kd	CGS001-11267	SNF8	-			
5654	-46.68	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
5655	-46.76	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
5656	-46.77	kd	CGS001-4664	NAB1	-			
5657	-46.79	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
5658	-46.8	kd	CGS001-9813	KIAA0494	-			
5659	-46.81	oe	ccsbBroad304_02057	P4HA2	-			
5660	-46.81	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
5661	-46.81	kd	CGS001-4849	CNOT3	-			
5662	-46.83	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
5663	-46.84	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
5664	-46.84	kd	CGS001-11040	PIM2	PIM family			
5665	-46.89	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
5666	-46.9	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
5667	-46.9	oe	ccsbBroad304_06562	MAT1A	-			
5668	-46.99	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
5669	-47.02	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
5670	-47.02	kd	CGS001-8945	BTRC	F-boxes / WD-40 domains			
5671	-47.04	oe	ccsbBroad304_01832	PAX8	Paired boxes			
5672	-47.05	kd	CGS001-5695	PSMB7	Proteasome subunits			
5673	-47.07	kd	CGS001-27161	EIF2C2	-			
5674	-47.08	oe	ccsbBroad304_00841	IKBKB	IKK family			
5675	-47.11	cc		Rho associated kinase inhibitor	-			
5676	-47.14	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
5677	-47.15	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
5678	-47.16	kd	CGS001-51182	HSPA14	Heat shock proteins / HSP70			
5679	-47.2	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
5680	-47.22	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
5681	-47.25	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
5682	-47.28	kd	CGS001-6258	RXRG	Retinoid X receptors			
5683	-47.3	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
5684	-47.33	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
5685	-47.37	kd	CGS001-10452	TOMM40	-			
5686	-47.37	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
5687	-47.42	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
5688	-47.46	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
5689	-47.47	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
5690	-47.47	kd	CGS001-2937	GSS	-			
5691	-47.47	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
5692	-47.52	oe	ccsbBroad304_00316	CKS1B	-			
5693	-47.59	kd	CGS001-5336	PLCG2	Phosphoinositide-specific phospholipase C			
5694	-47.63	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5695	-47.63	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
5696	-47.64	kd	CGS001-6885	MAP3K7	MAPKKK:TAK1 subfamily			
5697	-47.7	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
5698	-47.78	kd	CGS001-2621	GAS6	-			
5699	-47.81	kd	CGS001-4151	MB	-			
5700	-47.85	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5701	-47.86	kd	CGS001-51096	UTP18	WD repeat domain containing			
5702	-47.96	kd	CGS001-5315	PKM2	-			
5703	-47.97	kd	CGS001-27148	STK36	Unc-51-like kinase (ULK) family			
5704	-48.1	kd	CGS001-10544	PROCR	CD molecules			
5705	-48.15	kd	CGS001-25825	BACE2	Pepsin			
5706	-48.25	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
5707	-48.3	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
5708	-48.31	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
5709	-48.33	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
5710	-48.34	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
5711	-48.35	kd	CGS001-353345	GPR141	GPCR / Class A : Orphans			
5712	-48.38	kd	CGS001-5427	POLE2	DNA polymerases			
5713	-48.4	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
5714	-48.44	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
5715	-48.5	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
5716	-48.53	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5717	-48.54	kd	CGS001-55631	LRRC40	-			
5718	-48.56	kd	CGS001-775	CACNA1C	Calcium channel subunits			
5719	-48.57	kd	CGS001-8800	PEX11A	-			
5720	-48.59	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
5721	-48.61	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
5722	-48.62	cc		Homeobox Gene GOF	-			
5723	-48.63	kd	CGS001-221188	GPR114	Adhesion Class GPCRs			
5724	-48.64	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
5725	-48.65	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
5726	-48.67	kd	CGS001-8935	SKAP2	Pleckstrin homology (PH) domain containing			
5727	-48.72	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
5728	-48.73	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
5729	-48.76	kd	CGS001-8942	KYNU	-			
5730	-48.76	oe	ccsbBroad304_01716	TSN	-			
5731	-48.82	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
5732	-48.83	oe	ccsbBroad304_01379	RBBP6	-			
5733	-48.84	oe	ccsbBroad304_01985	EIF3H	-			
5734	-48.91	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
5735	-48.92	cp	BRD-K04710043	hexamethylenebisacetamide	AKT inhibitor			AKT inhibitor, Differentiation inducer, NFkB pathway inhibitor
5736	-48.96	kd	CGS001-23386	NUDCD3	-			
5737	-49	kd	CGS001-11186	RASSF1	-			
5738	-49.01	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
5739	-49.05	kd	CGS001-4833	NME4	-			
5740	-49.17	kd	CGS001-1955	MEGF9	-			
5741	-49.2	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
5742	-49.2	kd	CGS001-7016	TESK1	TESK subfamily			
5743	-49.25	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
5744	-49.27	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
5745	-49.31	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
5746	-49.33	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
5747	-49.37	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
5748	-49.46	cp	BRD-K94887716	TFMPP	Serotonin receptor agonist			Serotonin receptor agonist, Serotonin receptor antagonist
5749	-49.48	kd	CGS001-5985	RFC5	ATPases / AAA-type			
5750	-49.48	kd	CGS001-1429	CRYZ	-			
5751	-49.57	kd	CGS001-84722	PSRC1	-			
5752	-49.58	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
5753	-49.58	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
5754	-49.58	kd	CGS001-2678	GGT1	CD molecules			
5755	-49.59	kd	CGS001-64223	MLST8	WD repeat domain containing			
5756	-49.69	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
5757	-49.69	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
5758	-49.73	kd	CGS001-136	ADORA2B	GPCR / Class A : Adenosine receptors			
5759	-49.75	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
5760	-49.76	kd	CGS001-11004	KIF2C	Kinesins			
5761	-49.77	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
5762	-49.79	cp	BRD-K37798499	etoposide	Topoisomerase inhibitor		TOP2A, CYP2E1, CYP3A5, TOP2B	Topoisomerase inhibitor
5763	-49.79	kd	CGS001-10078	TSSC4	-			
5764	-49.8	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
5765	-49.81	kd	CGS001-166793	ZBTB49	BTB/POZ domain containing			
5766	-49.82	cc		SRY LOF	-			
5767	-49.88	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
5768	-49.9	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
5769	-49.91	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
5770	-49.92	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
5771	-49.93	kd	CGS001-6924	TCEB3	-			
5772	-49.96	kd	CGS001-2877	GPX2	-			
5773	-49.97	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
5774	-49.97	kd	CGS001-8834	TMEM11	-			
5775	-49.98	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
5776	-50	kd	CGS001-9053	MAP7	-			
5777	-50.01	cp	BRD-K09471561	levofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
5778	-50.01	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
5779	-50.02	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
5780	-50.02	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
5781	-50.02	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
5782	-50.04	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
5783	-50.05	kd	CGS001-7054	TH	Amino acid hydroxylases			
5784	-50.06	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
5785	-50.1	kd	CGS001-10923	SUB1	-			
5786	-50.14	kd	CGS001-1020	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
5787	-50.15	kd	CGS001-7159	TP53BP2	Ankyrin repeat domain containing			
5788	-50.18	kd	CGS001-2212	FCGR2A	CD molecules			
5789	-50.19	kd	CGS001-10174	SORBS3	-			
5790	-50.25	kd	CGS001-7010	TEK	Type XII RTKs: TIE family of angiopoietin receptors			
5791	-50.26	oe	ccsbBroad304_08023	EIF2C1	-			
5792	-50.33	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
5793	-50.39	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
5794	-50.46	kd	CGS001-55907	CMAS	-			
5795	-50.46	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
5796	-50.5	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5797	-50.52	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
5798	-50.55	kd	CGS001-4255	MGMT	-			
5799	-50.57	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
5800	-50.58	kd	CGS001-8741	TNFSF13	CD molecules			
5801	-50.61	kd	CGS001-54749	EPDR1	-			
5802	-50.61	kd	CGS001-125919	ZNF543	Zinc fingers, C2H2-type			
5803	-50.61	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
5804	-50.63	kd	CGS001-5351	PLOD1	-			
5805	-50.65	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
5806	-50.67	kd	CGS001-1465	CSRP1	-			
5807	-50.69	cp	BRD-K84955386	hyperoside	Glucosidase inhibitor		ACE, AKR1B1, GAA	Glucosidase inhibitor
5808	-50.71	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5809	-50.79	kd	CGS001-5362	PLXNA2	Plexins			
5810	-50.79	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
5811	-50.84	kd	CGS001-2969	GTF2I	General transcription factors			
5812	-50.88	kd	CGS001-2015	EMR1	Adhesion Class GPCRs			
5813	-51.05	kd	CGS001-2869	GRK5	GRK1/3 subfamily			
5814	-51.05	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
5815	-51.06	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
5816	-51.19	kd	CGS001-1999	ELF3	ETS Transcription Factors			
5817	-51.2	kd	CGS001-5025	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
5818	-51.21	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
5819	-51.3	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
5820	-51.33	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
5821	-51.33	oe	ccsbBroad304_06852	RBP4	Lipocalins			
5822	-51.36	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
5823	-51.37	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
5824	-51.4	kd	CGS001-2752	GLUL	-			
5825	-51.41	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5826	-51.42	oe	ccsbBroad304_03232	VPS28	-			
5827	-51.43	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
5828	-51.47	kd	CGS001-1431	CS	-			
5829	-51.48	kd	CGS001-2289	FKBP5	Tetratricopeptide (TTC) repeat domain containing			
5830	-51.5	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
5831	-51.53	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
5832	-51.57	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
5833	-51.57	kd	CGS001-23355	VPS8	-			
5834	-51.57	kd	CGS001-9276	COPB2	WD repeat domain containing			
5835	-51.63	kd	CGS001-216	ALDH1A1	Aldehyde dehydrogenases			
5836	-51.69	kd	CGS001-121599	SPIC	ETS Transcription Factors			
5837	-51.7	cc		PPAR receptor agonist	-			
5838	-51.72	kd	CGS001-7003	TEAD1	-			
5839	-51.73	kd	CGS001-4836	NMT1	-			
5840	-51.75	kd	CGS001-23451	SF3B1	-			
5841	-51.78	kd	CGS001-84617	TUBB6	Tubulins			
5842	-51.81	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
5843	-51.84	kd	CGS001-54386	TERF2IP	-			
5844	-51.85	kd	CGS001-5624	PROC	Endogenous ligands			
5845	-51.95	cp	BRD-K15842202	eudesmic-acid	-666			-666
5846	-51.96	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
5847	-52.02	oe	ccsbBroad304_02143	CNOT8	-			
5848	-52.08	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
5849	-52.08	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
5850	-52.11	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
5851	-52.11	kd	CGS001-1028	CDKN1C	-			
5852	-52.11	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
5853	-52.12	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
5854	-52.12	kd	CGS001-3481	IGF2	-			
5855	-52.12	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
5856	-52.16	kd	CGS001-23678	SGK3	SGK family			
5857	-52.19	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
5858	-52.2	oe	ccsbBroad304_03980	DCLRE1B	-			
5859	-52.24	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
5860	-52.27	kd	CGS001-56647	BCCIP	-			
5861	-52.28	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
5862	-52.32	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
5863	-52.33	kd	CGS001-5373	PMM2	-			
5864	-52.34	cp	BRD-K44779798	miglitol	Glucosidase inhibitor		GAA, MGAM, GANAB, GANC, SLC5A4	Glucosidase inhibitor
5865	-52.36	kd	CGS001-2746	GLUD1	-			
5866	-52.38	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
5867	-52.4	cp	BRD-K86003836	flubendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
5868	-52.42	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
5869	-52.46	cc		V type ATPases LOF	-			
5870	-52.46	kd	CGS001-1650	DDOST	-			
5871	-52.54	kd	CGS001-805	CALM2	EF-hand domain containing			
5872	-52.59	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
5873	-52.59	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
5874	-52.61	kd	CGS001-29888	STRN4	WD repeat domain containing			
5875	-52.65	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
5876	-52.7	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
5877	-52.73	kd	CGS001-29911	HOOK2	-			
5878	-52.73	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
5879	-52.75	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5880	-52.79	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
5881	-52.8	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
5882	-52.87	kd	CGS001-9552	SPAG7	-			
5883	-52.89	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
5884	-52.9	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
5885	-52.91	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
5886	-52.92	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
5887	-53.02	cc		EGFR inhibitor	-			
5888	-53.03	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
5889	-53.05	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
5890	-53.05	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
5891	-53.06	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
5892	-53.08	kd	CGS001-57057	TBX20	T-boxes			
5893	-53.1	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
5894	-53.1	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
5895	-53.11	kd	CGS001-4199	ME1	-			
5896	-53.11	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
5897	-53.13	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
5898	-53.14	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
5899	-53.14	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
5900	-53.19	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
5901	-53.25	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
5902	-53.26	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
5903	-53.28	kd	CGS001-94103	ORMDL3	-			
5904	-53.28	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
5905	-53.29	kd	CGS001-5501	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5906	-53.35	kd	CGS001-26149	ZNF658	Zinc fingers, C2H2-type			
5907	-53.39	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
5908	-53.43	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
5909	-53.44	oe	ccsbBroad304_07592	CEPT1	-			
5910	-53.47	kd	CGS001-3488	IGFBP5	insulin-like growth factor (IGF) binding proteins			
5911	-53.51	kd	CGS001-79885	HDAC11	Histone deacetylases			
5912	-53.52	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
5913	-53.54	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
5914	-53.56	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
5915	-53.59	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
5916	-53.62	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
5917	-53.62	kd	CGS001-54788	DNAJB12	Heat shock proteins / DNAJ (HSP40)			
5918	-53.64	kd	CGS001-1974	EIF4A2	DEAD-boxes			
5919	-53.65	kd	CGS001-2197	FAU	S ribosomal proteins			
5920	-53.73	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
5921	-53.81	kd	CGS001-169436	C9ORF96	-			
5922	-53.82	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
5923	-53.82	kd	CGS001-4925	NUCB2	EF-hand domain containing			
5924	-53.85	kd	CGS001-7431	VIM	Intermediate filaments type III			
5925	-53.87	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
5926	-53.87	oe	ccsbBroad304_07651	HEXIM1	-			
5927	-53.88	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
5928	-53.9	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
5929	-53.9	kd	CGS001-2593	GAMT	-			
5930	-53.92	oe	ccsbBroad304_08365	CYCS	-			
5931	-53.92	kd	CGS001-7035	TFPI	-			
5932	-54	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
5933	-54.01	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
5934	-54.02	kd	CGS001-336	APOA2	Apolipoproteins			
5935	-54.05	kd	CGS001-11014	KDELR2	-			
5936	-54.22	kd	CGS001-25966	C2CD2	-			
5937	-54.25	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
5938	-54.25	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
5939	-54.25	kd	CGS001-55038	CDCA4	-			
5940	-54.27	kd	CGS001-7862	BRPF1	Non-enzymatic BRD containing proteins			
5941	-54.31	kd	CGS001-2101	ESRRA	Estrogen-related receptors			
5942	-54.45	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
5943	-54.46	kd	CGS001-23028	KDM1A	Histone demethylase			
5944	-54.46	kd	CGS001-60	ACTB	-			
5945	-54.49	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
5946	-54.57	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
5947	-54.63	kd	CGS001-578	BAK1	-			
5948	-54.68	kd	CGS001-9690	UBE3C	-			
5949	-54.69	kd	CGS001-6520	SLC3A2	SLC3 family			
5950	-54.7	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
5951	-54.71	kd	CGS001-51380	CSAD	-			
5952	-54.76	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
5953	-54.76	kd	CGS001-4953	ODC1	Decarboxylases			
5954	-54.78	kd	CGS001-27035	NOX1	-			
5955	-54.78	kd	CGS001-8826	IQGAP1	-			
5956	-54.82	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
5957	-54.84	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
5958	-54.87	cc		HOXL subclass homeoboxes LOF	-			
5959	-54.9	kd	CGS001-10651	MTX2	-			
5960	-54.91	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
5961	-54.94	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
5962	-54.96	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
5963	-54.96	kd	CGS001-11140	CDC37	-			
5964	-54.98	kd	CGS001-6774	STAT3	SH2 domain containing			
5965	-54.99	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
5966	-55.04	cc		DNA polymerase inhibitor	-			
5967	-55.07	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
5968	-55.09	kd	CGS001-2147	F2	Endogenous ligands			
5969	-55.2	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
5970	-55.21	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
5971	-55.23	kd	CGS001-8803	SUCLA2	-			
5972	-55.31	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
5973	-55.36	kd	CGS001-7039	TGFA	-			
5974	-55.38	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
5975	-55.43	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
5976	-55.48	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
5977	-55.51	kd	CGS001-3516	RBPJ	-			
5978	-55.51	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
5979	-55.54	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5980	-55.56	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5981	-55.59	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
5982	-55.62	kd	CGS001-50604	IL20	Interleukins and interleukin receptors			
5983	-55.69	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
5984	-55.69	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5985	-55.7	kd	CGS001-7337	UBE3A	-			
5986	-55.71	cp	BRD-K33106058	cytarabine	Ribonucleotide reductase inhibitor		POLB, POLA1	Ribonucleotide reductase inhibitor
5987	-55.76	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
5988	-55.78	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5989	-55.82	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
5990	-55.85	oe	ccsbBroad304_01347	RAD1	-			
5991	-55.85	kd	CGS001-56993	TOMM22	-			
5992	-55.85	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
5993	-55.93	kd	CGS001-6929	TCF3	Basic helix-loop-helix proteins			
5994	-56.01	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
5995	-56.05	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
5996	-56.06	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
5997	-56.08	kd	CGS001-3309	HSPA5	Heat shock proteins / HSP70			
5998	-56.08	kd	CGS001-2683	B4GALT1	Beta 4-glycosyltransferases			
5999	-56.09	oe	ccsbBroad304_03155	DHH	-			
6000	-56.12	kd	CGS001-283455	KSR2	RAF family			
6001	-56.16	kd	CGS001-29102	DROSHA	-			
6002	-56.22	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
6003	-56.23	oe	ccsbBroad304_06996	SRM	-			
6004	-56.25	kd	CGS001-4552	MTRR	-			
6005	-56.27	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6006	-56.28	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
6007	-56.28	kd	CGS001-6598	SMARCB1	-			
6008	-56.3	kd	CGS001-3315	HSPB1	Heat shock proteins / HSPB			
6009	-56.31	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
6010	-56.31	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
6011	-56.35	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
6012	-56.37	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
6013	-56.38	kd	CGS001-1155	TBCB	-			
6014	-56.41	oe	ccsbBroad304_01372	RALB	-			
6015	-56.43	oe	ccsbBroad304_08346	COQ3	-			
6016	-56.44	oe	ccsbBroad304_03812	PBXIP1	-			
6017	-56.45	kd	CGS001-151306	GPBAR1	Bile acid receptor			
6018	-56.49	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
6019	-56.5	kd	CGS001-84365	MKI67IP	-			
6020	-56.51	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
6021	-56.52	oe	ccsbBroad304_14174	CDKAL1	-			
6022	-56.58	oe	ccsbBroad304_13499	KSR2	RAF family			
6023	-56.58	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
6024	-56.59	kd	CGS001-51174	TUBD1	Tubulins			
6025	-56.59	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
6026	-56.61	kd	CGS001-8635	RNASET2	-			
6027	-56.61	kd	CGS001-3988	LIPA	-			
6028	-56.65	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
6029	-56.65	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
6030	-56.68	kd	CGS001-65975	STK33	CAMK-unique family			
6031	-56.68	kd	CGS001-826	CAPNS1	EF-hand domain containing			
6032	-56.72	cc		P38 MAPK inhibitor	-			
6033	-56.75	kd	CGS001-9133	CCNB2	-			
6034	-56.78	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
6035	-56.79	kd	CGS001-221895	JAZF1	Zinc fingers, C2H2-type			
6036	-56.84	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
6037	-56.85	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
6038	-56.91	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
6039	-56.91	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
6040	-56.92	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
6041	-56.92	kd	CGS001-94234	FOXQ1	Forkhead boxes			
6042	-56.99	cp	BRD-A20589515	dihydroxyphenylglycine	Glutamate receptor agonist		GRM1	Glutamate receptor agonist
6043	-57.02	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
6044	-57.07	kd	CGS001-100	ADA	Adenosine turnover			
6045	-57.12	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
6046	-57.12	oe	ccsbBroad304_14011	PAPSS1	-			
6047	-57.17	oe	ccsbBroad304_00389	CTBP1	-			
6048	-57.19	cp	BRD-K44353683	nateglinide	Insulin secretagogue		ABCC8, KCNJ11, CYP3A4, INS, KCNJ10, PPARG	Insulin secretagogue
6049	-57.19	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
6050	-57.27	kd	CGS001-7474	WNT5A	Endogenous ligands			
6051	-57.27	oe	ccsbBroad304_08797	FASTKD5	-			
6052	-57.32	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
6053	-57.34	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
6054	-57.35	kd	CGS001-30836	DNTTIP2	-			
6055	-57.38	kd	CGS001-9474	ATG5	-			
6056	-57.39	kd	CGS001-670	BPHL	-			
6057	-57.43	oe	ccsbBroad304_07888	CBX6	-			
6058	-57.44	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
6059	-57.46	kd	CGS001-10444	ZER1	ZYG11 cell cycle regulator family			
6060	-57.49	kd	CGS001-10557	RPP38	-			
6061	-57.49	oe	ccsbBroad304_01184	PGK1	-			
6062	-57.54	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
6063	-57.62	kd	CGS001-4191	MDH2	-			
6064	-57.67	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6065	-57.71	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
6066	-57.73	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
6067	-57.8	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
6068	-57.81	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
6069	-57.85	kd	CGS001-5827	PXMP2	-			
6070	-57.9	kd	CGS001-8480	RAE1	WD repeat domain containing			
6071	-57.91	oe	ccsbBroad304_02415	TUBB3	Tubulins			
6072	-57.97	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
6073	-58.03	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
6074	-58.03	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
6075	-58.05	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
6076	-58.06	kd	CGS001-8317	CDC7	CDC7 family			
6077	-58.13	kd	CGS001-50810	HDGFRP3	-			
6078	-58.17	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6079	-58.18	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
6080	-58.18	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
6081	-58.2	kd	CGS001-115	ADCY9	Adenylyl cyclases			
6082	-58.26	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
6083	-58.27	kd	CGS001-51160	VPS28	-			
6084	-58.28	cc		Lysine acetyltransferases LOF	-			
6085	-58.3	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
6086	-58.31	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
6087	-58.33	oe	ccsbBroad304_06642	NIT1	-			
6088	-58.37	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
6089	-58.45	kd	CGS001-10329	TMEM5	-			
6090	-58.47	kd	CGS001-3339	HSPG2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6091	-58.49	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
6092	-58.51	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6093	-58.55	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
6094	-58.55	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
6095	-58.56	kd	CGS001-55968	NSFL1C	UBX domain containing			
6096	-58.65	kd	CGS001-54681	P4HTM	-			
6097	-58.66	kd	CGS001-3897	L1CAM	CD molecules			
6098	-58.67	oe	ccsbBroad304_00738	HINT1	-			
6099	-58.74	oe	ccsbBroad304_06651	NOV	-			
6100	-58.74	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
6101	-58.85	kd	CGS001-10914	PAPOLA	-			
6102	-58.93	oe	ccsbBroad304_00789	HSBP1	-			
6103	-58.96	oe	ccsbBroad304_05890	BHMT	-			
6104	-58.98	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6105	-59.09	kd	CGS001-9200	PTPLA	-			
6106	-59.12	kd	CGS001-7296	TXNRD1	-			
6107	-59.14	kd	CGS001-51135	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
6108	-59.18	kd	CGS001-1837	DTNA	-			
6109	-59.2	kd	CGS001-10901	DHRS4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6110	-59.21	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
6111	-59.21	kd	CGS001-7276	TTR	-			
6112	-59.25	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
6113	-59.28	kd	CGS001-5888	RAD51	-			
6114	-59.28	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
6115	-59.3	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
6116	-59.34	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
6117	-59.34	kd	CGS001-9443	MED7	-			
6118	-59.35	oe	ccsbBroad304_07490	SCRN1	-			
6119	-59.38	kd	CGS001-10607	TBL3	WD repeat domain containing			
6120	-59.51	kd	CGS001-90861	HN1L	-			
6121	-59.53	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
6122	-59.53	kd	CGS001-9170	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6123	-59.55	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
6124	-59.55	kd	CGS001-5970	RELA	NFkappaB transcription factor family			
6125	-59.57	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
6126	-59.59	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
6127	-59.62	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
6128	-59.62	kd	CGS001-5578	PRKCA	Delta subfamily			
6129	-59.62	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6130	-59.63	kd	CGS001-5586	PKN2	Protein kinase N (PKN) family			
6131	-59.67	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
6132	-59.69	kd	CGS001-135	ADORA2A	GPCR / Class A : Adenosine receptors			
6133	-59.7	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
6134	-59.73	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
6135	-59.73	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6136	-59.76	oe	ccsbBroad304_03164	MTERFD1	-			
6137	-59.85	oe	ccsbBroad304_03056	MCTS1	-			
6138	-59.85	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
6139	-59.86	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
6140	-59.87	cp	BRD-K90733503	cefalexin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6141	-59.94	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
6142	-59.95	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
6143	-59.98	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
6144	-60	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
6145	-60.06	kd	CGS001-54505	DHX29	DEAH-boxes			
6146	-60.07	oe	ccsbBroad304_03951	NARFL	-			
6147	-60.17	kd	CGS001-84923	FAM104A	-			
6148	-60.18	oe	ccsbBroad304_06286	GLUL	-			
6149	-60.19	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
6150	-60.21	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
6151	-60.27	kd	CGS001-5686	PSMA5	Proteasome subunits			
6152	-60.27	oe	ccsbBroad304_02045	BUD31	-			
6153	-60.28	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
6154	-60.28	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
6155	-60.28	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
6156	-60.34	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
6157	-60.35	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6158	-60.36	kd	CGS001-64343	AZI2	-			
6159	-60.38	kd	CGS001-1718	DHCR24	-			
6160	-60.4	kd	CGS001-1756	DMD	-			
6161	-60.41	kd	CGS001-3845	KRAS	RAS subfamily			
6162	-60.42	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
6163	-60.43	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6164	-60.45	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
6165	-60.46	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
6166	-60.48	kd	CGS001-26191	PTPN22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6167	-60.48	kd	CGS001-378	ARF4	ADP-ribosylation factors			
6168	-60.51	kd	CGS001-129685	TAF8	-			
6169	-60.52	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
6170	-60.55	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
6171	-60.58	kd	CGS001-1649	DDIT3	-			
6172	-60.58	kd	CGS001-1284	COL4A2	Collagens			
6173	-60.59	kd	CGS001-286380	FOXD4L3	-			
6174	-60.62	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
6175	-60.72	kd	CGS001-3482	IGF2R	CD molecules			
6176	-60.72	kd	CGS001-111	ADCY5	Adenylate cyclases			
6177	-60.74	oe	ccsbBroad304_14143	NUSAP1	-			
6178	-60.76	oe	ccsbBroad304_00652	GNAS	-			
6179	-60.78	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6180	-60.79	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
6181	-60.79	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
6182	-60.82	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
6183	-60.85	kd	CGS001-4522	MTHFD1	-			
6184	-60.89	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
6185	-60.91	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
6186	-60.94	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
6187	-61.01	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
6188	-61.03	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
6189	-61.05	oe	ccsbBroad304_07834	GGA2	-			
6190	-61.05	kd	CGS001-3565	IL4	Interleukins and interleukin receptors			
6191	-61.07	kd	CGS001-34	ACADM	-			
6192	-61.12	kd	CGS001-9709	HERPUD1	-			
6193	-61.15	oe	ccsbBroad304_10758	CTBP2	-			
6194	-61.17	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
6195	-61.21	cp	BRD-K41903098	diphenoxylate	Opioid receptor agonist		OPRM1, OPRD1	Opioid receptor agonist
6196	-61.24	cc		DNA Replication LOF	-			
6197	-61.24	oe	ccsbBroad304_00888	ITPK1	-			
6198	-61.32	oe	ccsbBroad304_02175	MAGED1	-			
6199	-61.32	kd	CGS001-10048	RANBP9	-			
6200	-61.36	cp	BRD-A09495397	bicuculline	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, KCNN1	GABA receptor antagonist
6201	-61.4	kd	CGS001-8731	RNMT	-			
6202	-61.43	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
6203	-61.43	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
6204	-61.44	cc		Tubulin inhibitor	-			
6205	-61.45	kd	CGS001-5900	RALGDS	-			
6206	-61.47	cc		JAK inhibitor	-			
6207	-61.49	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
6208	-61.51	kd	CGS001-5355	PLP2	-			
6209	-61.55	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
6210	-61.56	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6211	-61.59	oe	ccsbBroad304_09225	BUD13	-			
6212	-61.65	oe	ccsbBroad304_01632	SYPL1	-			
6213	-61.66	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
6214	-61.66	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6215	-61.7	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
6216	-61.71	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
6217	-61.73	cc		ATPase inhibitor	-			
6218	-61.73	kd	CGS001-4323	MMP14	Matrix metallopeptidase			
6219	-61.74	kd	CGS001-7525	YES1	Src family			
6220	-61.74	kd	CGS001-64333	ARHGAP9	Rho GTPase activating proteins			
6221	-61.74	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
6222	-61.77	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
6223	-61.78	kd	CGS001-5432	POLR2C	RNA polymerase subunits			
6224	-61.79	kd	CGS001-2810	SFN	-			
6225	-61.8	cp	BRD-A68589262	troxipide	Glucosamine synthetase stimulant			Glucosamine synthetase stimulant
6226	-61.84	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
6227	-61.89	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
6228	-61.9	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
6229	-61.91	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
6230	-61.91	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
6231	-61.98	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
6232	-62.01	oe	ccsbBroad304_00816	IDE	Pitrilysin			
6233	-62.01	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
6234	-62.04	kd	CGS001-147686	ZNF418	Zinc fingers, C2H2-type			
6235	-62.05	kd	CGS001-6829	SUPT5H	-			
6236	-62.05	kd	CGS001-1001	CDH3	Cadherins / Major cadherins			
6237	-62.1	oe	ccsbBroad304_07363	AIFM1	-			
6238	-62.11	kd	CGS001-4846	NOS3	Nitric oxide synthases			
6239	-62.14	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6240	-62.15	cc		Proteasome inhibitor	-			
6241	-62.15	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6242	-62.19	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
6243	-62.29	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
6244	-62.36	kd	CGS001-5253	PHF2	Histone demethylases			
6245	-62.37	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
6246	-62.43	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
6247	-62.44	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
6248	-62.44	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
6249	-62.45	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
6250	-62.49	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
6251	-62.49	kd	CGS001-80314	EPC1	-			
6252	-62.51	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
6253	-62.53	kd	CGS001-27034	ACAD8	-			
6254	-62.72	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6255	-62.72	kd	CGS001-2000	ELF4	ETS Transcription Factors			
6256	-62.81	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
6257	-62.82	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
6258	-62.82	kd	CGS001-57616	TSHZ3	Teashirt zinc fingers			
6259	-62.88	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
6260	-62.89	kd	CGS001-6189	RPS3A	S ribosomal proteins			
6261	-62.91	oe	ccsbBroad304_01147	PC	Carboxylases			
6262	-62.95	oe	ccsbBroad304_05439	O3FAR1	-			
6263	-62.96	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
6264	-62.99	kd	CGS001-5580	PRKCD	Delta subfamily			
6265	-62.99	oe	ccsbBroad304_02218	IKBKE	IKK family			
6266	-63.09	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
6267	-63.11	oe	ccsbBroad304_03555	PANK4	-			
6268	-63.12	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
6269	-63.26	kd	CGS001-55793	FAM63A	-			
6270	-63.29	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
6271	-63.33	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
6272	-63.34	kd	CGS001-9900	SV2A	Major facilitator superfamily (MFS) of transporters			
6273	-63.36	kd	CGS001-2781	GNAZ	-			
6274	-63.39	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
6275	-63.41	kd	CGS001-5193	PEX12	-			
6276	-63.41	kd	CGS001-55229	PANK4	-			
6277	-63.41	kd	CGS001-9738	CCP110	-			
6278	-63.45	kd	CGS001-2859	GPR35	GPCR / Class A : Orphans			
6279	-63.45	kd	CGS001-25	ABL1	Abl family			
6280	-63.46	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
6281	-63.47	cp	BRD-A16934955	nalbuphine	Opioid receptor agonist		OPRD1, OPRK1, OPRM1	Opioid receptor agonist, Opioid receptor antagonist
6282	-63.47	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
6283	-63.47	kd	CGS001-84634	KISS1R	GPCR / Class A : RF amide peptide receptors			
6284	-63.53	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
6285	-63.53	kd	CGS001-3155	HMGCL	-			
6286	-63.56	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
6287	-63.58	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
6288	-63.6	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
6289	-63.61	oe	ccsbBroad304_00226	CAV1	-			
6290	-63.61	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
6291	-63.68	oe	ccsbBroad304_02526	POP4	-			
6292	-63.69	kd	CGS001-4097	MAFG	-			
6293	-63.75	kd	CGS001-29110	TBK1	IKK family			
6294	-63.76	kd	CGS001-114609	TIRAP	-			
6295	-63.77	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
6296	-63.81	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
6297	-63.82	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
6298	-63.84	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
6299	-63.87	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6300	-63.88	kd	CGS001-54556	ING3	Zinc fingers, PHD-type			
6301	-63.92	oe	ccsbBroad304_06255	LRRC32	-			
6302	-64	kd	CGS001-9519	TBPL1	-			
6303	-64.05	cc		IGF-1 inhibitor	-			
6304	-64.06	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
6305	-64.07	kd	CGS001-11162	NUDT6	Nudix motif containing			
6306	-64.11	kd	CGS001-2909	ARHGAP35	Rho GTPase activating proteins			
6307	-64.15	kd	CGS001-3670	ISL1	Homeoboxes / LIM class			
6308	-64.15	kd	CGS001-488	ATP2A2	Calcium-ATPases			
6309	-64.2	cp	BRD-K65910366	KUC103904N	-666			-666
6310	-64.24	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
6311	-64.26	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
6312	-64.27	kd	CGS001-3609	ILF3	-			
6313	-64.27	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
6314	-64.32	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
6315	-64.33	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
6316	-64.33	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
6317	-64.34	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
6318	-64.35	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
6319	-64.38	oe	ccsbBroad304_02509	GMEB1	-			
6320	-64.39	kd	CGS001-486	FXYD2	Ion transport regulator			
6321	-64.42	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
6322	-64.43	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
6323	-64.47	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
6324	-64.47	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
6325	-64.49	kd	CGS001-23549	DNPEP	Aminopeptidase I			
6326	-64.52	kd	CGS001-2558	GABRA5	GABA receptors			
6327	-64.56	oe	ccsbBroad304_00991	MDH1	-			
6328	-64.61	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
6329	-64.63	oe	ccsbBroad304_08839	IFIH1	-			
6330	-64.65	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
6331	-64.66	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
6332	-64.66	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
6333	-64.68	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
6334	-64.68	kd	CGS001-2735	GLI1	Zinc fingers, C2H2-type			
6335	-64.68	kd	CGS001-811	CALR	-			
6336	-64.72	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
6337	-64.72	kd	CGS001-6502	SKP2	F-boxes / Leucine-rich repeats			
6338	-64.73	kd	CGS001-9637	FEZ2	-			
6339	-64.74	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
6340	-64.75	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
6341	-64.77	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
6342	-64.89	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
6343	-64.91	cc		PDGFR/KIT inhibitor	-			
6344	-64.91	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
6345	-64.92	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
6346	-64.93	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
6347	-64.93	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
6348	-64.96	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
6349	-64.98	kd	CGS001-5538	PPT1	-			
6350	-65.03	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
6351	-65.03	kd	CGS001-65263	PYCRL	-			
6352	-65.04	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
6353	-65.05	kd	CGS001-79618	HMBOX1	Homeoboxes / HNF class			
6354	-65.07	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
6355	-65.08	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
6356	-65.12	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6357	-65.21	kd	CGS001-56922	MCCC1	-			
6358	-65.21	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
6359	-65.22	kd	CGS001-506	ATP5B	ATPases / F-type			
6360	-65.28	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
6361	-65.28	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
6362	-65.39	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
6363	-65.41	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
6364	-65.44	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
6365	-65.44	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
6366	-65.47	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
6367	-65.48	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
6368	-65.49	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
6369	-65.51	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
6370	-65.54	oe	ccsbBroad304_00329	CLTA	-			
6371	-65.54	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
6372	-65.55	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
6373	-65.57	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
6374	-65.57	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
6375	-65.58	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
6376	-65.62	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
6377	-65.62	kd	CGS001-55379	LRRC59	-			
6378	-65.76	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
6379	-65.79	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
6380	-65.86	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
6381	-65.93	kd	CGS001-7076	TIMP1	-			
6382	-65.94	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
6383	-66	cc		SRC inhibitor	-			
6384	-66.01	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
6385	-66.04	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
6386	-66.06	kd	CGS001-2936	GSR	Oxidoreductases			
6387	-66.09	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
6388	-66.13	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
6389	-66.17	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
6390	-66.18	kd	CGS001-23081	KDM4C	Histone demethylases			
6391	-66.19	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
6392	-66.21	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
6393	-66.29	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
6394	-66.41	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
6395	-66.42	kd	CGS001-1399	CRKL	SH2 domain containing			
6396	-66.51	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
6397	-66.52	kd	CGS001-5723	PSPH	-			
6398	-66.54	kd	CGS001-1642	DDB1	-			
6399	-66.55	kd	CGS001-1213	CLTC	-			
6400	-66.59	kd	CGS001-3476	IGBP1	-			
6401	-66.74	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
6402	-66.74	kd	CGS001-5433	POLR2D	RNA polymerase subunits			
6403	-66.77	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
6404	-66.78	kd	CGS001-9143	SYNGR3	-			
6405	-66.82	kd	CGS001-23118	TAB2	-			
6406	-66.83	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
6407	-66.86	kd	CGS001-10318	TNIP1	-			
6408	-66.88	oe	ccsbBroad304_08480	PNPO	-			
6409	-66.93	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
6410	-66.99	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
6411	-67.07	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6412	-67.08	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
6413	-67.08	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
6414	-67.09	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
6415	-67.11	kd	CGS001-23075	SWAP70	EF-hand domain containing			
6416	-67.14	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
6417	-67.17	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
6418	-67.2	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
6419	-67.22	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
6420	-67.23	kd	CGS001-23239	PHLPP1	Pleckstrin homology (PH) domain containing			
6421	-67.26	kd	CGS001-9212	AURKB	Aurora kinase			
6422	-67.28	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
6423	-67.34	cp	BRD-K25310650	ormetoprim	Bacterial antifolate			Bacterial antifolate
6424	-67.35	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
6425	-67.4	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
6426	-67.43	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
6427	-67.47	cp	BRD-K66206289	lobeline	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist
6428	-67.48	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
6429	-67.48	kd	CGS001-6932	TCF7	-			
6430	-67.56	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
6431	-67.61	kd	CGS001-123803	NTAN1	-			
6432	-67.63	cp	BRD-K50384076	7,4'-dihydroxyflavone	Opioid receptor antagonist		CYP19A1	Opioid receptor antagonist
6433	-67.66	kd	CGS001-51311	TLR8	Toll-like receptor family			
6434	-67.7	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
6435	-67.7	kd	CGS001-5566	PRKACA	Protein kinase A			
6436	-67.73	kd	CGS001-7321	UBE2D1	Ubiquitin-conjugating enzymes E2			
6437	-67.73	kd	CGS001-9695	EDEM1	-			
6438	-67.76	oe	ccsbBroad304_07277	RTCD1	-			
6439	-67.82	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
6440	-67.83	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
6441	-67.84	cp	BRD-K59753975	vindesine	Tubulin inhibitor		TUBB, TUBB1	Tubulin inhibitor
6442	-67.84	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
6443	-67.88	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
6444	-67.89	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
6445	-67.9	oe	ccsbBroad304_00549	FDX1	-			
6446	-67.92	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
6447	-67.93	kd	CGS001-4439	MSH5	-			
6448	-67.97	cc		PKC inhibitor	-			
6449	-68.01	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
6450	-68.01	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
6451	-68.02	oe	ccsbBroad304_02219	MORF4L2	-			
6452	-68.02	oe	ccsbBroad304_04626	EGLN3	-			
6453	-68.09	oe	ccsbBroad304_09095	PUS7L	-			
6454	-68.12	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
6455	-68.12	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6456	-68.14	kd	CGS001-9512	PMPCB	-			
6457	-68.14	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
6458	-68.17	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
6459	-68.18	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6460	-68.2	kd	CGS001-387	RHOA	-			
6461	-68.23	kd	CGS001-6241	RRM2	Ribonucleoside-diphosphate reductases			
6462	-68.24	kd	CGS001-2821	GPI	-			
6463	-68.31	kd	CGS001-2542	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
6464	-68.31	oe	ccsbBroad304_05098	MAGEB6	-			
6465	-68.33	kd	CGS001-203523	ZNF449	Zinc fingers, C2H2-type			
6466	-68.36	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
6467	-68.37	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
6468	-68.37	kd	CGS001-1633	DCK	-			
6469	-68.41	oe	ccsbBroad304_01951	BLZF1	-			
6470	-68.41	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
6471	-68.42	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
6472	-68.43	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
6473	-68.43	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
6474	-68.44	kd	CGS001-2864	FFAR1	Fatty acid receptors			
6475	-68.51	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
6476	-68.52	cc		HSP inhibitor	-			
6477	-68.56	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
6478	-68.56	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
6479	-68.6	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
6480	-68.63	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
6481	-68.69	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
6482	-68.69	kd	CGS001-657	BMPR1A	Type I receptor serine/threonine kinases			
6483	-68.72	kd	CGS001-7088	TLE1	WD repeat domain containing			
6484	-68.73	oe	ccsbBroad304_07178	ZFP112	-			
6485	-68.74	kd	CGS001-6443	SGCB	-			
6486	-68.77	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
6487	-68.77	oe	ccsbBroad304_02565	RALBP1	-			
6488	-68.82	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6489	-68.83	oe	ccsbBroad304_06464	ITGB2	Integrins			
6490	-68.86	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
6491	-68.88	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
6492	-68.89	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
6493	-68.91	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
6494	-68.92	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6495	-68.93	kd	CGS001-5979	RET	Type XIV RTKs: RET			
6496	-68.94	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
6497	-68.97	kd	CGS001-7750	ZMYM2	Zinc fingers, MYM type			
6498	-69.02	oe	ccsbBroad304_02677	PDAP1	-			
6499	-69.02	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
6500	-69.05	oe	ccsbBroad304_10230	STK19	G11 family			
6501	-69.06	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
6502	-69.06	kd	CGS001-5045	FURIN	Subtilisin			
6503	-69.07	cp	BRD-A95696820	acadesine	AMPK activator			AMPK activator
6504	-69.08	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
6505	-69.09	cp	BRD-K63343048	orlistat	Lipase inhibitor		PNLIP, DAGLA, FASN, LIPF, CNR1, DAGLB	Lipase inhibitor
6506	-69.09	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
6507	-69.09	kd	CGS001-3895	KTN1	-			
6508	-69.11	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
6509	-69.12	oe	ccsbBroad304_06133	TOR1A	-			
6510	-69.2	kd	CGS001-6282	S100A11	EF-hand domain containing			
6511	-69.21	kd	CGS001-1163	CKS1B	-			
6512	-69.23	kd	CGS001-23361	ZNF629	Zinc fingers, C2H2-type			
6513	-69.24	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
6514	-69.25	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
6515	-69.34	kd	CGS001-4967	OGDH	-			
6516	-69.36	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
6517	-69.43	kd	CGS001-7485	WRB	-			
6518	-69.47	kd	CGS001-5612	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
6519	-69.48	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
6520	-69.48	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
6521	-69.51	cp	BRD-A11990600	lorazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, TSPO	Benzodiazepine receptor agonist
6522	-69.58	kd	CGS001-11198	SUPT16H	-			
6523	-69.59	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
6524	-69.6	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
6525	-69.6	kd	CGS001-7298	TYMS	Methyltransferases			
6526	-69.62	kd	CGS001-79581	GPR172A	-			
6527	-69.67	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
6528	-69.69	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
6529	-69.69	kd	CGS001-57721	METTL14	-			
6530	-69.71	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
6531	-69.74	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
6532	-69.74	kd	CGS001-5160	PDHA1	-			
6533	-69.75	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
6534	-69.75	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
6535	-69.77	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
6536	-69.8	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
6537	-69.87	oe	ccsbBroad304_00651	GNAI3	-			
6538	-70.01	oe	ccsbBroad304_06234	G6PC	-			
6539	-70.01	kd	CGS001-8720	MBTPS1	Subtilisin			
6540	-70.02	kd	CGS001-10523	CHERP	G patch domain containing			
6541	-70.04	cp	BRD-K82109576	vincristine	Tubulin inhibitor		TUBB, TUBA4A	Tubulin inhibitor
6542	-70.08	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
6543	-70.08	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
6544	-70.11	kd	CGS001-2073	ERCC5	-			
6545	-70.12	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
6546	-70.14	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
6547	-70.19	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
6548	-70.22	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
6549	-70.24	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
6550	-70.31	kd	CGS001-51520	LARS	Aminoacyl tRNA synthetases / Class I			
6551	-70.32	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
6552	-70.32	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
6553	-70.41	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
6554	-70.42	oe	ccsbBroad304_03728	DIABLO	-			
6555	-70.44	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
6556	-70.47	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
6557	-70.51	cp	BRD-K30563334	rifabutin	Protein synthesis inhibitor		CYP3A4, HSP90AA1, HSP90B1	Protein synthesis inhibitor
6558	-70.56	oe	ccsbBroad304_01532	SIAH1	-			
6559	-70.6	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
6560	-70.6	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
6561	-70.61	kd	CGS001-998	CDC42	-			
6562	-70.65	kd	CGS001-23647	ARFIP2	-			
6563	-70.72	kd	CGS001-6514	SLC2A2	Solute carriers			
6564	-70.72	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
6565	-70.77	kd	CGS001-11344	TWF2	Twinfilin subfamily			
6566	-70.83	kd	CGS001-7185	TRAF1	-			
6567	-70.88	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
6568	-70.94	cp	BRD-K51671335	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
6569	-70.95	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
6570	-70.97	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
6571	-71.01	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
6572	-71.02	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
6573	-71.12	kd	CGS001-2849	GPR26	GPCR / Class A : Orphans			
6574	-71.15	oe	ccsbBroad304_06144	EFNB3	Ephrins			
6575	-71.17	kd	CGS001-55662	HIF1AN	-			
6576	-71.18	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
6577	-71.19	kd	CGS001-1452	CSNK1A1	Casein kinase 1 (CK1) family			
6578	-71.2	kd	CGS001-53340	SPA17	-			
6579	-71.22	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
6580	-71.26	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
6581	-71.32	kd	CGS001-498	ATP5A1	ATPases / F-type			
6582	-71.36	kd	CGS001-5914	RARA	Retinoic acid receptors			
6583	-71.36	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
6584	-71.36	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
6585	-71.4	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
6586	-71.42	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
6587	-71.55	kd	CGS001-29959	NRBP1	NRBP family			
6588	-71.58	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
6589	-71.6	oe	ccsbBroad304_03177	FIS1	-			
6590	-71.62	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
6591	-71.68	oe	ccsbBroad304_00985	MCL1	-			
6592	-71.69	kd	CGS001-84333	PCGF5	Polycomb group ring fingers			
6593	-71.85	kd	CGS001-9978	RBX1	RING-type (C3HC4) zinc fingers			
6594	-71.85	kd	CGS001-11116	FGFR1OP	-			
6595	-71.87	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6596	-71.88	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
6597	-71.89	kd	CGS001-93487	MAPK1IP1L	-			
6598	-71.92	kd	CGS001-23499	MACF1	EF-hand domain containing			
6599	-71.94	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
6600	-71.95	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
6601	-71.99	kd	CGS001-1936	EEF1D	-			
6602	-72	kd	CGS001-4665	NAB2	-			
6603	-72	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
6604	-72.03	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
6605	-72.03	kd	CGS001-8807	IL18RAP	CD molecules			
6606	-72.04	kd	CGS001-57147	SCYL3	-			
6607	-72.05	oe	ccsbBroad304_00492	EIF5A	-			
6608	-72.11	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
6609	-72.16	oe	ccsbBroad304_02864	PRDX5	-			
6610	-72.17	kd	CGS001-8477	GPR65	GPCR / Class A : Orphans			
6611	-72.19	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
6612	-72.19	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
6613	-72.26	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
6614	-72.27	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
6615	-72.27	oe	ccsbBroad304_02605	PAPD7	-			
6616	-72.35	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
6617	-72.42	kd	CGS001-5690	PSMB2	Proteasome subunits			
6618	-72.56	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
6619	-72.58	kd	CGS001-5898	RALA	-			
6620	-72.69	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6621	-72.7	kd	CGS001-3685	ITGAV	Integrins			
6622	-72.7	kd	CGS001-2287	FKBP3	-			
6623	-72.71	kd	CGS001-10298	PAK4	PAKB subfamily			
6624	-72.73	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
6625	-72.73	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6626	-72.74	kd	CGS001-8435	SOAT2	-			
6627	-72.81	oe	ccsbBroad304_05887	CFB	Complement system			
6628	-72.83	kd	CGS001-2059	EPS8	-			
6629	-72.83	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
6630	-72.86	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
6631	-72.87	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
6632	-72.9	kd	CGS001-35	ACADS	-			
6633	-72.91	kd	CGS001-5810	RAD1	-			
6634	-73.01	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
6635	-73.06	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
6636	-73.07	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
6637	-73.11	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
6638	-73.14	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
6639	-73.14	kd	CGS001-122618	PLD4	-			
6640	-73.16	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
6641	-73.22	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
6642	-73.24	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
6643	-73.27	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
6644	-73.33	kd	CGS001-6500	SKP1	-			
6645	-73.34	kd	CGS001-7771	ZFP112	-			
6646	-73.35	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
6647	-73.38	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
6648	-73.41	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
6649	-73.43	cp	BRD-A68888262	azelastine	Histamine receptor antagonist		HRH1, CYP2C19	Histamine receptor antagonist
6650	-73.45	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
6651	-73.48	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
6652	-73.49	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6653	-73.7	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
6654	-73.73	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
6655	-73.73	oe	ccsbBroad304_00174	BRAF	RAF family			
6656	-73.76	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
6657	-73.76	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
6658	-73.77	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
6659	-73.78	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
6660	-73.79	oe	ccsbBroad304_09503	KLHDC9	-			
6661	-73.8	kd	CGS001-4122	MAN2A2	-			
6662	-73.8	kd	CGS001-23365	ARHGEF12	Rho guanine nucleotide exchange factors			
6663	-73.91	kd	CGS001-81894	SLC25A28	Miscellaneous SLC25 mitochondrial transporters			
6664	-73.93	kd	CGS001-64135	IFIH1	-			
6665	-73.94	kd	CGS001-191	AHCY	Adenosine turnover			
6666	-73.96	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
6667	-73.97	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
6668	-73.99	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
6669	-74.02	kd	CGS001-9213	XPR1	-			
6670	-74.02	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
6671	-74.04	kd	CGS001-4174	MCM5	-			
6672	-74.06	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
6673	-74.07	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
6674	-74.09	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
6675	-74.09	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
6676	-74.1	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6677	-74.16	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
6678	-74.17	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
6679	-74.18	kd	CGS001-154	ADRB2	GPCR / Class A : Adrenoceptors : beta			
6680	-74.2	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
6681	-74.22	kd	CGS001-8841	HDAC3	Histone deacetylases			
6682	-74.27	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
6683	-74.39	oe	ccsbBroad304_00032	ADSL	-			
6684	-74.48	oe	ccsbBroad304_00116	ASS1	-			
6685	-74.49	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
6686	-74.5	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
6687	-74.51	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
6688	-74.52	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
6689	-74.53	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
6690	-74.53	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
6691	-74.54	oe	ccsbBroad304_03772	CCNL1	-			
6692	-74.55	cp	BRD-K96471533	nitazoxanide	Pyruvate ferredoxin oxidoreductase inhibitor			Pyruvate ferredoxin oxidoreductase inhibitor
6693	-74.59	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
6694	-74.63	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
6695	-74.63	kd	CGS001-84619	ZGPAT	G patch domain containing			
6696	-74.63	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
6697	-74.64	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
6698	-74.66	kd	CGS001-2673	GFPT1	-			
6699	-74.68	kd	CGS001-9700	ESPL1	-			
6700	-74.71	kd	CGS001-83448	PUS7L	-			
6701	-74.71	oe	ccsbBroad304_00794	HSF1	-			
6702	-74.73	kd	CGS001-25949	SYF2	-			
6703	-74.74	kd	CGS001-10094	ARPC3	Actin related protein 2/3 complex subunits			
6704	-74.75	kd	CGS001-55239	OGFOD1	-			
6705	-74.75	kd	CGS001-2643	GCH1	-			
6706	-74.77	kd	CGS001-2309	FOXO3	Forkhead boxes			
6707	-74.77	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
6708	-74.79	cc		Trace amine receptors LOF	-			
6709	-74.82	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
6710	-74.83	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
6711	-74.84	oe	ccsbBroad304_01052	MYB	-			
6712	-74.85	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
6713	-74.86	cp	BRD-K63265447	docetaxel	Tubulin inhibitor		TUBB, BCL2, MAP2, MAP4, MAPT, NR1I2, TUBB1	Tubulin inhibitor
6714	-74.93	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
6715	-74.93	kd	CGS001-84515	MCM8	-			
6716	-75.02	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
6717	-75.03	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
6718	-75.04	kd	CGS001-8836	GGH	Gamma-glutamyl hydrolase			
6719	-75.04	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
6720	-75.06	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
6721	-75.13	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
6722	-75.14	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
6723	-75.17	kd	CGS001-23658	LSM5	-			
6724	-75.18	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
6725	-75.21	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6726	-75.29	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
6727	-75.34	oe	ccsbBroad304_05963	CD44	CD molecules			
6728	-75.35	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
6729	-75.48	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
6730	-75.52	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
6731	-75.54	kd	CGS001-2277	FIGF	-			
6732	-75.54	oe	ccsbBroad304_08878	METTL4	-			
6733	-75.56	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
6734	-75.58	kd	CGS001-3596	IL13	Interleukins and interleukin receptors			
6735	-75.59	oe	ccsbBroad304_00491	EIF4EBP2	-			
6736	-75.61	kd	CGS001-7311	UBA52	L ribosomal proteins			
6737	-75.64	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
6738	-75.65	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
6739	-75.65	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
6740	-75.68	kd	CGS001-23650	TRIM29	-			
6741	-75.7	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
6742	-75.72	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
6743	-75.76	kd	CGS001-350	APOH	Apolipoproteins			
6744	-75.77	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
6745	-75.83	oe	ccsbBroad304_02163	MED7	-			
6746	-75.83	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
6747	-75.88	kd	CGS001-821	CANX	-			
6748	-75.89	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
6749	-75.9	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
6750	-75.91	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
6751	-75.92	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
6752	-75.93	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
6753	-75.99	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
6754	-76.02	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
6755	-76.05	kd	CGS001-3661	IRF3	-			
6756	-76.07	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
6757	-76.07	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
6758	-76.1	kd	CGS001-55699	IARS2	Aminoacyl tRNA synthetases / Class I			
6759	-76.1	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
6760	-76.16	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
6761	-76.17	cc		Gamma secretase inhibitor	-			
6762	-76.22	kd	CGS001-2588	GALNS	Arylsulfatase family			
6763	-76.26	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
6764	-76.32	cp	BRD-K60160658	tiagabine	GABA uptake inhibitor		SLC6A1, CYP2C19	GABA uptake inhibitor
6765	-76.34	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
6766	-76.42	kd	CGS001-2771	GNAI2	-			
6767	-76.42	kd	CGS001-2052	EPHX1	-			
6768	-76.44	kd	CGS001-1312	COMT	Catecholamine turnover			
6769	-76.44	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
6770	-76.46	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6771	-76.47	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
6772	-76.47	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
6773	-76.49	kd	CGS001-790	CAD	-			
6774	-76.51	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
6775	-76.53	kd	CGS001-347736	NME9	-			
6776	-76.54	kd	CGS001-51268	PIPOX	-			
6777	-76.55	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
6778	-76.58	kd	CGS001-2565	GABRG1	GABA receptors			
6779	-76.63	kd	CGS001-79921	TCEAL4	-			
6780	-76.63	kd	CGS001-5934	RBL2	-			
6781	-76.64	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
6782	-76.65	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
6783	-76.65	kd	CGS001-125950	RAVER1	RNA binding motif (RRM) containing			
6784	-76.65	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
6785	-76.67	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
6786	-76.67	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
6787	-76.7	kd	CGS001-10645	CAMKK2	Meta subfamily			
6788	-76.72	kd	CGS001-5869	RAB5B	RAB, member RAS oncogene			
6789	-76.75	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
6790	-76.76	oe	ccsbBroad304_02956	EHF	-			
6791	-76.76	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
6792	-76.77	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
6793	-76.78	kd	CGS001-162699	TCEB3C	-			
6794	-76.78	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
6795	-76.8	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
6796	-76.8	kd	CGS001-9712	USP6NL	-			
6797	-76.84	kd	CGS001-6499	SKIV2L	-			
6798	-76.92	cp	BRD-K82147103	lofepramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
6799	-76.95	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
6800	-76.96	kd	CGS001-2958	GTF2A2	General transcription factors			
6801	-76.98	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
6802	-76.99	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
6803	-77.08	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
6804	-77.09	cc		NFkB pathway inhibitor	-			
6805	-77.11	kd	CGS001-2079	ERH	-			
6806	-77.14	kd	CGS001-5292	PIM1	PIM family			
6807	-77.26	kd	CGS001-64428	NARFL	-			
6808	-77.3	oe	ccsbBroad304_07861	COBL	-			
6809	-77.31	kd	CGS001-3248	HPGD	Prostaglandin synthases			
6810	-77.4	kd	CGS001-28960	DCPS	-			
6811	-77.45	kd	CGS001-4087	SMAD2	SMADs			
6812	-77.53	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
6813	-77.54	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
6814	-77.58	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
6815	-77.67	kd	CGS001-53343	NUDT9	Nudix motif containing			
6816	-77.68	oe	ccsbBroad304_08217	SCCPDH	-			
6817	-77.7	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
6818	-77.75	kd	CGS001-5649	RELN	-			
6819	-77.79	cc		Calmodulin antagonist	-			
6820	-77.8	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
6821	-77.81	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
6822	-77.87	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
6823	-77.91	kd	CGS001-9919	SEC16A	-			
6824	-77.91	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
6825	-77.93	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
6826	-77.99	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6827	-78.04	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
6828	-78.04	kd	CGS001-5883	RAD9A	-			
6829	-78.07	kd	CGS001-6909	TBX2	T-boxes			
6830	-78.08	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
6831	-78.09	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
6832	-78.17	cc		Na-K-Cl transporter inhibitor	-			
6833	-78.17	cp	BRD-A43082555	loxoprofen	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
6834	-78.19	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
6835	-78.23	oe	ccsbBroad304_00184	C2	Complement system			
6836	-78.23	kd	CGS001-23338	PHF15	-			
6837	-78.24	kd	CGS001-6204	RPS10	S ribosomal proteins			
6838	-78.27	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
6839	-78.29	kd	CGS001-9851	KIAA0753	-			
6840	-78.33	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
6841	-78.42	kd	CGS001-25824	PRDX5	-			
6842	-78.42	oe	ccsbBroad304_05936	CASP2	Caspases			
6843	-78.49	kd	CGS001-5930	RBBP6	-			
6844	-78.49	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
6845	-78.51	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
6846	-78.53	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
6847	-78.54	kd	CGS001-4615	MYD88	-			
6848	-78.55	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
6849	-78.57	kd	CGS001-2581	GALC	-			
6850	-78.6	cc		BCL inhibitor	-			
6851	-78.6	oe	ccsbBroad304_03570	QRSL1	-			
6852	-78.63	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
6853	-78.67	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
6854	-78.71	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
6855	-78.75	kd	CGS001-143187	VTI1A	-			
6856	-78.78	kd	CGS001-5608	MAP2K6	MAPKK:STE7 family			
6857	-78.8	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
6858	-78.9	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
6859	-78.9	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
6860	-78.94	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
6861	-78.94	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
6862	-78.96	oe	ccsbBroad304_07220	CDC45	-			
6863	-78.97	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
6864	-79	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
6865	-79.1	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
6866	-79.1	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6867	-79.1	kd	CGS001-23743	BHMT2	-			
6868	-79.13	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
6869	-79.22	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
6870	-79.22	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
6871	-79.23	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6872	-79.26	kd	CGS001-10616	RBCK1	RING-type (C3HC4) zinc fingers			
6873	-79.26	kd	CGS001-1497	CTNS	-			
6874	-79.26	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
6875	-79.27	oe	ccsbBroad304_01413	RPA2	-			
6876	-79.3	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
6877	-79.32	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6878	-79.32	kd	CGS001-2078	ERG	ETS Transcription Factors			
6879	-79.33	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
6880	-79.34	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6881	-79.52	kd	CGS001-8894	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6882	-79.54	kd	CGS001-9897	KIAA0196	-			
6883	-79.58	kd	CGS001-5511	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6884	-79.6	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
6885	-79.63	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
6886	-79.66	kd	CGS001-27241	BBS9	-			
6887	-79.66	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
6888	-79.69	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
6889	-79.7	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
6890	-79.71	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
6891	-79.75	kd	CGS001-929	CD14	CD molecules			
6892	-79.78	oe	ccsbBroad304_00624	GCK	Hexokinases			
6893	-79.8	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
6894	-79.84	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
6895	-79.86	cc		Vitamin D receptor agonist	-			
6896	-79.87	kd	CGS001-5997	RGS2	Endogenous ligands			
6897	-79.87	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
6898	-79.88	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
6899	-79.88	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
6900	-79.89	kd	CGS001-3932	LCK	Src family			
6901	-79.95	kd	CGS001-63933	CCDC90A	-			
6902	-80	kd	CGS001-22949	PTGR1	-			
6903	-80.03	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6904	-80.08	kd	CGS001-5371	PML	RING-type (C3HC4) zinc fingers			
6905	-80.09	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
6906	-80.18	oe	ccsbBroad304_08536	PARL	-			
6907	-80.18	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6908	-80.18	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
6909	-80.18	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
6910	-80.18	kd	CGS001-6184	RPN1	-			
6911	-80.2	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
6912	-80.21	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
6913	-80.25	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
6914	-80.27	cp	BRD-K17705806	JTC-801	Opioid receptor antagonist		OPRL1	Opioid receptor antagonist
6915	-80.29	kd	CGS001-11331	PHB2	-			
6916	-80.32	kd	CGS001-10614	HEXIM1	-			
6917	-80.32	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
6918	-80.33	kd	CGS001-641	BLM	-			
6919	-80.34	cp	BRD-A84134924	pancuronium	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRNA1, CHRNA2	Acetylcholine receptor antagonist
6920	-80.39	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
6921	-80.43	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
6922	-80.44	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
6923	-80.47	cc		Progesterone receptor antagonist	-			
6924	-80.48	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
6925	-80.53	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
6926	-80.56	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
6927	-80.56	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
6928	-80.58	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
6929	-80.62	kd	CGS001-200879	LIPH	-			
6930	-80.64	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6931	-80.64	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6932	-80.68	cc		DNA synthesis inhibitor	-			
6933	-80.69	kd	CGS001-9270	ITGB1BP1	-			
6934	-80.8	kd	CGS001-440	ASNS	-			
6935	-80.8	oe	ccsbBroad304_06253	GALT	-			
6936	-80.82	kd	CGS001-5993	RFX5	-			
6937	-80.95	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
6938	-80.95	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
6939	-81.01	kd	CGS001-5387	PMS2P3	-			
6940	-81.05	cc		Glycogen synthase kinase inhibitor	-			
6941	-81.07	kd	CGS001-7024	TFCP2	-			
6942	-81.08	cp	BRD-K85090592	pilocarpine	Acetylcholine receptor agonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor agonist
6943	-81.1	kd	CGS001-388	RHOB	-			
6944	-81.11	kd	CGS001-51282	SCAND1	-			
6945	-81.18	cc		Interleukin receptors LOF	-			
6946	-81.2	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
6947	-81.21	kd	CGS001-83637	ZMIZ2	Zinc fingers, MIZ-type			
6948	-81.21	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
6949	-81.21	kd	CGS001-161	AP2A2	-			
6950	-81.21	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
6951	-81.23	kd	CGS001-47	ACLY	-			
6952	-81.24	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
6953	-81.29	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
6954	-81.3	oe	ccsbBroad304_00995	MECP2	-			
6955	-81.31	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
6956	-81.33	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
6957	-81.33	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
6958	-81.37	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
6959	-81.43	kd	CGS001-2100	ESR2	Estrogen receptors			
6960	-81.45	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
6961	-81.45	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
6962	-81.47	kd	CGS001-5162	PDHB	-			
6963	-81.49	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
6964	-81.5	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
6965	-81.5	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
6966	-81.52	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
6967	-81.55	oe	ccsbBroad304_02580	TMED10	-			
6968	-81.57	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
6969	-81.57	kd	CGS001-84159	ARID5B	-			
6970	-81.59	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
6971	-81.59	kd	CGS001-382	ARF6	ADP-ribosylation factors			
6972	-81.62	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
6973	-81.64	oe	ccsbBroad304_06525	LIPA	-			
6974	-81.65	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
6975	-81.69	kd	CGS001-54512	EXOSC4	-			
6976	-81.7	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
6977	-81.7	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
6978	-81.71	cp	BRD-K10961822	latanoprost	Prostanoid receptor agonist		PTGFR	Prostanoid receptor agonist
6979	-81.72	oe	ccsbBroad304_00515	ERH	-			
6980	-81.73	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
6981	-81.74	oe	ccsbBroad304_00542	FBP1	-			
6982	-81.75	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
6983	-81.78	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
6984	-81.78	kd	CGS001-112858	TP53RK	Bud32 family			
6985	-81.78	kd	CGS001-955	ENTPD6	-			
6986	-81.79	kd	CGS001-10285	SMNDC1	Tudor domain containing			
6987	-81.79	kd	CGS001-9774	BCLAF1	-			
6988	-81.81	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
6989	-81.82	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
6990	-81.82	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
6991	-81.84	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
6992	-81.87	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
6993	-81.87	kd	CGS001-10284	SAP18	-			
6994	-81.88	kd	CGS001-9453	GGPS1	Lanosterol biosynthesis pathway			
6995	-81.9	kd	CGS001-6919	TCEA2	-			
6996	-81.92	kd	CGS001-10641	NPRL2	-			
6997	-81.94	cc		Toll like receptors LOF	-			
6998	-81.95	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6999	-81.95	kd	CGS001-4175	MCM6	-			
7000	-81.99	oe	ccsbBroad304_06888	RPN1	-			
7001	-82.01	cc		Cell Cycle Inhibition GOF	-			
7002	-82.02	kd	CGS001-3479	IGF1	Endogenous ligands			
7003	-82.02	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
7004	-82.04	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
7005	-82.11	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
7006	-82.12	kd	CGS001-8431	NR0B2	DAX-like receptors			
7007	-82.12	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
7008	-82.14	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
7009	-82.22	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
7010	-82.24	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
7011	-82.25	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
7012	-82.3	kd	CGS001-22944	KIN	-			
7013	-82.3	kd	CGS001-2512	FTL	-			
7014	-82.35	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
7015	-82.42	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
7016	-82.42	kd	CGS001-91304	C19ORF6	-			
7017	-82.47	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
7018	-82.47	kd	CGS001-7292	TNFSF4	CD molecules			
7019	-82.48	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
7020	-82.49	kd	CGS001-6646	SOAT1	-			
7021	-82.5	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
7022	-82.54	kd	CGS001-3242	HPD	Oxidoreductases			
7023	-82.57	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
7024	-82.58	cp	BRD-A39172021	ampiroxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
7025	-82.59	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
7026	-82.63	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
7027	-82.63	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
7028	-82.69	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
7029	-82.74	oe	ccsbBroad304_00249	CD14	CD molecules			
7030	-82.74	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
7031	-82.77	kd	CGS001-2634	GBP2	-			
7032	-82.78	kd	CGS001-79090	TRAPPC6A	Trafficking protein particle complex			
7033	-82.81	kd	CGS001-3708	ITPR1	Ion channels / Inositol triphosphate receptors			
7034	-82.83	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
7035	-82.83	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
7036	-82.9	kd	CGS001-2767	GNA11	-			
7037	-82.91	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
7038	-82.93	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
7039	-82.93	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
7040	-82.96	cp	BRD-A96107863	nisoldipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNB2, CYP3A5	Calcium channel blocker
7041	-82.96	kd	CGS001-23670	TMEM2	-			
7042	-82.98	kd	CGS001-84669	USP32	EF-hand domain containing			
7043	-83	oe	ccsbBroad304_00709	GUK1	-			
7044	-83	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
7045	-83.02	kd	CGS001-54851	ANKRD49	Ankyrin repeat domain containing			
7046	-83.03	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
7047	-83.03	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
7048	-83.07	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
7049	-83.08	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
7050	-83.11	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
7051	-83.2	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
7052	-83.22	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
7053	-83.22	kd	CGS001-10827	FAM114A2	-			
7054	-83.24	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
7055	-83.27	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
7056	-83.29	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
7057	-83.33	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
7058	-83.33	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
7059	-83.35	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
7060	-83.42	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
7061	-83.46	oe	ccsbBroad304_00620	GCDH	-			
7062	-83.46	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
7063	-83.49	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
7064	-83.51	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
7065	-83.52	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7066	-83.52	kd	CGS001-501	ALDH7A1	Aldehyde dehydrogenases			
7067	-83.55	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
7068	-83.55	kd	CGS001-54658	UGT1A1	UDP glucuronosyltransferases			
7069	-83.57	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
7070	-83.6	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
7071	-83.62	kd	CGS001-405	ARNT	Basic helix-loop-helix proteins			
7072	-83.64	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
7073	-83.69	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
7074	-83.72	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
7075	-83.72	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
7076	-83.75	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
7077	-83.77	kd	CGS001-4907	NT5E	Adenosine turnover			
7078	-83.82	kd	CGS001-2919	CXCL1	Endogenous ligands			
7079	-83.89	kd	CGS001-7528	YY1	INO80 complex subunits			
7080	-83.92	kd	CGS001-51422	PRKAG2	AMPK subfamily			
7081	-83.92	kd	CGS001-11340	EXOSC8	-			
7082	-83.93	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
7083	-83.97	kd	CGS001-5879	RAC1	Endogenous ligands			
7084	-83.98	oe	ccsbBroad304_06126	TSC22D3	-			
7085	-83.99	oe	ccsbBroad304_04752	IKBIP	-			
7086	-84	kd	CGS001-25842	ASF1A	-			
7087	-84.01	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
7088	-84.05	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
7089	-84.09	cc		Purinergic receptors P2Y GOF	-			
7090	-84.1	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
7091	-84.16	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
7092	-84.17	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
7093	-84.2	kd	CGS001-403	ARL3	ADP-ribosylation factors			
7094	-84.22	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
7095	-84.22	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
7096	-84.23	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
7097	-84.23	oe	ccsbBroad304_05763	ACTB	-			
7098	-84.27	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
7099	-84.27	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
7100	-84.27	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
7101	-84.3	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
7102	-84.33	oe	ccsbBroad304_00376	CSK	Csk family			
7103	-84.33	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
7104	-84.35	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
7105	-84.35	oe	ccsbBroad304_02138	TRIP10	-			
7106	-84.36	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
7107	-84.37	kd	CGS001-22930	RAB3GAP1	-			
7108	-84.39	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
7109	-84.39	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
7110	-84.4	kd	CGS001-11019	LIAS	-			
7111	-84.42	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
7112	-84.46	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
7113	-84.53	kd	CGS001-89910	UBE3B	-			
7114	-84.56	kd	CGS001-5707	PSMD1	Proteasome subunits			
7115	-84.57	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
7116	-84.57	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
7117	-84.59	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
7118	-84.61	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7119	-84.68	kd	CGS001-11142	PKIG	-			
7120	-84.71	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
7121	-84.75	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
7122	-84.78	kd	CGS001-1962	EHHADH	-			
7123	-84.79	kd	CGS001-9322	TRIP10	-			
7124	-84.82	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
7125	-84.84	oe	ccsbBroad304_09833	SENP5	-			
7126	-84.87	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
7127	-84.87	oe	ccsbBroad304_00210	CALR	-			
7128	-84.88	kd	CGS001-1508	CTSB	Cathepsins			
7129	-84.88	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
7130	-84.91	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
7131	-84.91	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
7132	-84.92	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
7133	-84.94	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
7134	-84.96	oe	ccsbBroad304_09578	PASD1	-			
7135	-84.98	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
7136	-84.99	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
7137	-85	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
7138	-85.04	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
7139	-85.09	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
7140	-85.12	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
7141	-85.15	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
7142	-85.2	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
7143	-85.22	kd	CGS001-3560	IL2RB	IL-2 receptor family			
7144	-85.22	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
7145	-85.25	cp	BRD-K40758068	efavirenz	HIV protease inhibitor		CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5	HIV protease inhibitor
7146	-85.25	kd	CGS001-2768	GNA12	-			
7147	-85.28	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
7148	-85.3	kd	CGS001-64750	SMURF2	-			
7149	-85.34	kd	CGS001-847	CAT	-			
7150	-85.36	oe	ccsbBroad304_07548	TSSC4	-			
7151	-85.36	kd	CGS001-3992	FADS1	Fatty acid desaturases			
7152	-85.37	kd	CGS001-7486	WRN	-			
7153	-85.37	kd	CGS001-5471	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
7154	-85.38	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
7155	-85.39	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
7156	-85.41	oe	ccsbBroad304_00106	ARRB1	-			
7157	-85.49	kd	CGS001-6871	TADA2A	-			
7158	-85.49	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
7159	-85.51	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
7160	-85.52	oe	ccsbBroad304_02285	MED6	-			
7161	-85.54	cp	BRD-K49668410	clarithromycin	Bacterial 50S ribosomal subunit inhibitor		CYP2C19, CYP3A4, CYP3A5, CYP3A7	Bacterial 50S ribosomal subunit inhibitor
7162	-85.55	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
7163	-85.57	kd	CGS001-3383	ICAM1	CD molecules			
7164	-85.59	kd	CGS001-79109	MAPKAP1	-			
7165	-85.61	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
7166	-85.61	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
7167	-85.64	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
7168	-85.65	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7169	-85.66	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
7170	-85.71	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
7171	-85.71	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
7172	-85.74	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
7173	-85.77	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
7174	-85.78	kd	CGS001-3149	HMGB3	High-mobility group / Canonical			
7175	-85.8	cc		MCM family LOF	-			
7176	-85.82	kd	CGS001-1616	DAXX	-			
7177	-85.83	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
7178	-85.84	kd	CGS001-644	BLVRA	-			
7179	-85.85	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
7180	-85.89	cc		Calcium channel blocker	-			
7181	-85.91	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
7182	-85.96	oe	ccsbBroad304_01180	PFKFB3	-			
7183	-85.97	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
7184	-85.98	oe	ccsbBroad304_07832	XPO7	Exportins			
7185	-86.03	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
7186	-86.06	kd	CGS001-9797	TATDN2	-			
7187	-86.06	kd	CGS001-11136	SLC7A9	SLC7 family			
7188	-86.1	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
7189	-86.12	cc		Serotonin receptor antagonist	-			
7190	-86.13	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
7191	-86.17	kd	CGS001-11230	PRAF2	-			
7192	-86.18	cc		GABA receptor antagonist	-			
7193	-86.18	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
7194	-86.24	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
7195	-86.24	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
7196	-86.27	kd	CGS001-9180	OSMR	IL-6 receptor family			
7197	-86.29	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
7198	-86.29	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
7199	-86.3	kd	CGS001-1655	DDX5	DEAD-boxes			
7200	-86.36	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
7201	-86.38	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
7202	-86.41	kd	CGS001-9686	VGLL4	-			
7203	-86.41	oe	ccsbBroad304_01469	RSU1	-			
7204	-86.42	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
7205	-86.45	oe	ccsbBroad304_06066	CTSL1	-			
7206	-86.45	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
7207	-86.46	oe	ccsbBroad304_08137	HOOK2	-			
7208	-86.47	cc		GATA Zinc finger domain containing LOF	-			
7209	-86.47	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
7210	-86.47	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
7211	-86.48	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
7212	-86.49	kd	CGS001-2885	GRB2	SH2 domain containing			
7213	-86.49	oe	ccsbBroad304_00085	APRT	-			
7214	-86.51	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
7215	-86.52	oe	ccsbBroad304_06565	MB	-			
7216	-86.52	kd	CGS001-833	CARS	Aminoacyl tRNA synthetases / Class I			
7217	-86.53	cp	BRD-K39391626	ethylestrenol	Progesterone receptor agonist		AR	Progesterone receptor agonist
7218	-86.57	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
7219	-86.61	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
7220	-86.61	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
7221	-86.63	oe	ccsbBroad304_03658	DCP1A	-			
7222	-86.63	oe	ccsbBroad304_02990	LYPD3	-			
7223	-86.65	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
7224	-86.67	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
7225	-86.7	oe	ccsbBroad304_02419	NDRG1	-			
7226	-86.72	oe	ccsbBroad304_06282	GLDC	-			
7227	-86.73	oe	ccsbBroad304_02398	LANCL1	-			
7228	-86.74	kd	CGS001-9632	SEC24C	-			
7229	-86.74	kd	CGS001-2118	ETV4	ETS Transcription Factors			
7230	-86.76	kd	CGS001-3945	LDHB	-			
7231	-86.78	kd	CGS001-6654	SOS1	Rho guanine nucleotide exchange factors			
7232	-86.79	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
7233	-86.8	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
7234	-86.81	kd	CGS001-5111	PCNA	-			
7235	-86.81	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
7236	-86.82	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
7237	-86.83	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
7238	-86.84	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
7239	-86.86	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
7240	-86.95	cp	BRD-K97752965	nicorandil	Nitric oxide donor		ABCC9, KCNJ11, KCNJ8	Nitric oxide donor, Potassium channel activator
7241	-86.96	oe	ccsbBroad304_00099	ARG2	Arginase			
7242	-86.96	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
7243	-86.98	kd	CGS001-2114	ETS2	ETS Transcription Factors			
7244	-87.03	cc		Dopamine receptor antagonist	-			
7245	-87.06	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
7246	-87.09	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
7247	-87.1	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
7248	-87.15	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
7249	-87.18	kd	CGS001-79170	PRR15L	-			
7250	-87.18	oe	ccsbBroad304_07632	PROCR	CD molecules			
7251	-87.19	oe	ccsbBroad304_00564	FGR	Src family			
7252	-87.23	kd	CGS001-2263	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
7253	-87.29	kd	CGS001-819	CAMLG	-			
7254	-87.32	kd	CGS001-22832	KIAA1009	-			
7255	-87.33	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
7256	-87.36	kd	CGS001-84547	PGBD1	-			
7257	-87.36	oe	ccsbBroad304_01872	DGCR14	-			
7258	-87.37	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
7259	-87.38	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
7260	-87.39	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
7261	-87.39	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
7262	-87.4	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
7263	-87.45	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
7264	-87.45	kd	CGS001-2023	ENO1	-			
7265	-87.46	oe	ccsbBroad304_02318	KIF20A	Kinesins			
7266	-87.48	kd	CGS001-10460	TACC3	-			
7267	-87.5	oe	ccsbBroad304_00486	EFNB2	Ephrins			
7268	-87.51	kd	CGS001-55176	SEC61A2	-			
7269	-87.53	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
7270	-87.53	oe	ccsbBroad304_00063	AMPD2	-			
7271	-87.55	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
7272	-87.56	kd	CGS001-9761	MLEC	-			
7273	-87.57	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
7274	-87.59	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
7275	-87.6	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
7276	-87.6	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
7277	-87.6	kd	CGS001-9687	GREB1	-			
7278	-87.6	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
7279	-87.65	oe	ccsbBroad304_07101	TSC2	-			
7280	-87.66	kd	CGS001-7444	VRK2	Vaccina related kinase (VRK) family			
7281	-87.66	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
7282	-87.67	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
7283	-87.68	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
7284	-87.68	kd	CGS001-9337	CNOT8	-			
7285	-87.71	kd	CGS001-26227	PHGDH	-			
7286	-87.71	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
7287	-87.72	cc		Baculoviral IAP repeat domain containing LOF	-			
7288	-87.78	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
7289	-87.79	cc		Tachykinin antagonist	-			
7290	-87.79	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
7291	-87.8	kd	CGS001-11044	PAPD7	-			
7292	-87.81	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
7293	-87.87	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
7294	-87.87	kd	CGS001-9748	SLK	SLK subfamily			
7295	-87.87	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7296	-87.9	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
7297	-87.91	kd	CGS001-51750	RTEL1	-			
7298	-87.93	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
7299	-87.94	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
7300	-87.95	kd	CGS001-121549	ASCL4	Basic helix-loop-helix proteins			
7301	-87.96	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
7302	-87.97	oe	ccsbBroad304_07102	TSG101	-			
7303	-87.98	cp	BRD-K66412701	pazufloxacin	Topoisomerase inhibitor			Topoisomerase inhibitor
7304	-88	kd	CGS001-115650	TNFRSF13C	Tumour necrosis factor (TNF) receptor family			
7305	-88.01	oe	ccsbBroad304_03097	CNOT7	-			
7306	-88.01	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
7307	-88.02	cc		Retinoid receptor agonist	-			
7308	-88.02	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
7309	-88.02	kd	CGS001-6193	RPS5	S ribosomal proteins			
7310	-88.07	cc		DNA dependent protein kinase inhibitor	-			
7311	-88.09	kd	CGS001-64167	ERAP2	Aminopeptidase N			
7312	-88.1	kd	CGS001-2966	GTF2H2	General transcription factors			
7313	-88.11	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
7314	-88.14	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
7315	-88.14	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
7316	-88.17	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
7317	-88.18	cc		Serine proteases GOF	-			
7318	-88.18	kd	CGS001-5202	PFDN2	-			
7319	-88.18	kd	CGS001-85442	KNDC1	-			
7320	-88.19	kd	CGS001-10202	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7321	-88.2	kd	CGS001-51053	GMNN	-			
7322	-88.21	kd	CGS001-527	ATP6V0C	ATPases / V-type			
7323	-88.22	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
7324	-88.25	kd	CGS001-1503	CTPS	-			
7325	-88.28	kd	CGS001-4205	MEF2A	Myocyte enhancer factors			
7326	-88.29	oe	ccsbBroad304_00957	M6PR	-			
7327	-88.3	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
7328	-88.31	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
7329	-88.31	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
7330	-88.32	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
7331	-88.32	oe	ccsbBroad304_04465	RERG	-			
7332	-88.34	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
7333	-88.35	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
7334	-88.36	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
7335	-88.38	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
7336	-88.38	kd	CGS001-8650	NUMB	-			
7337	-88.38	kd	CGS001-79145	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
7338	-88.4	oe	ccsbBroad304_07071	TKT	-			
7339	-88.44	cp	BRD-K52020312	metronidazole	DNA inhibitor		CYP2C8, CYP2E1, CYP3A5, CYP3A7	DNA inhibitor, Antiprotozoal
7340	-88.45	kd	CGS001-1119	CHKA	-			
7341	-88.45	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
7342	-88.48	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
7343	-88.49	kd	CGS001-8892	EIF2B2	-			
7344	-88.5	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
7345	-88.51	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
7346	-88.52	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
7347	-88.53	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
7348	-88.54	oe	ccsbBroad304_01663	TFF2	-			
7349	-88.55	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
7350	-88.58	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
7351	-88.58	kd	CGS001-8061	FOSL1	basic leucine zipper proteins			
7352	-88.59	kd	CGS001-2002	ELK1	ETS Transcription Factors			
7353	-88.6	kd	CGS001-7764	ZNF217	Zinc fingers, C2H2-type			
7354	-88.64	cc		Vesicular Transport LOF	-			
7355	-88.64	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
7356	-88.66	oe	ccsbBroad304_00262	CD59	CD molecules			
7357	-88.67	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
7358	-88.67	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
7359	-88.68	oe	ccsbBroad304_07922	TRIM29	-			
7360	-88.68	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
7361	-88.72	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7362	-88.72	cp	BRD-K33226500	indinavir	HIV protease inhibitor		CYP3A5	HIV protease inhibitor
7363	-88.73	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
7364	-88.75	oe	ccsbBroad304_04190	CCDC92	-			
7365	-88.76	oe	ccsbBroad304_00966	MAFG	-			
7366	-88.78	kd	CGS001-4234	METTL1	-			
7367	-88.81	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
7368	-88.82	kd	CGS001-7840	ALMS1	-			
7369	-88.84	kd	CGS001-54438	GFOD1	-			
7370	-88.86	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
7371	-88.87	kd	CGS001-9867	PJA2	RING-type (C3HC4) zinc fingers			
7372	-88.88	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
7373	-88.91	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
7374	-88.93	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
7375	-88.94	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
7376	-88.94	kd	CGS001-1070	CETN3	EF-hand domain containing			
7377	-88.96	kd	CGS001-1949	EFNB3	Ephrins			
7378	-88.97	cc		Bacterial DNA gyrase inhibitor	-			
7379	-88.98	kd	CGS001-513	ATP5D	ATPases / F-type			
7380	-88.99	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
7381	-89.01	cc		HIF activator	-			
7382	-89.05	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
7383	-89.08	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
7384	-89.08	kd	CGS001-8900	CCNA1	-			
7385	-89.12	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
7386	-89.13	kd	CGS001-4204	MECP2	-			
7387	-89.18	kd	CGS001-8027	STAM	-			
7388	-89.21	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
7389	-89.22	kd	CGS001-79850	FAM57A	-			
7390	-89.23	kd	CGS001-1871	E2F3	-			
7391	-89.26	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
7392	-89.26	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
7393	-89.31	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
7394	-89.32	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
7395	-89.34	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
7396	-89.36	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
7397	-89.37	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
7398	-89.38	oe	ccsbBroad304_06136	ECHS1	-			
7399	-89.38	kd	CGS001-55620	STAP2	-			
7400	-89.42	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
7401	-89.42	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
7402	-89.46	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
7403	-89.46	cp	BRD-K21806131	tegaserod	Serotonin receptor partial agonist		HTR4, HTR2B, HTR2A, HTR2C	Serotonin receptor partial agonist
7404	-89.47	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
7405	-89.47	kd	CGS001-26271	FBXO5	F-boxes / other			
7406	-89.48	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
7407	-89.51	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
7408	-89.52	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
7409	-89.54	kd	CGS001-22	ABCB7	ATP binding cassette transporters / subfamily B			
7410	-89.54	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
7411	-89.57	oe	ccsbBroad304_01001	MEST	-			
7412	-89.6	kd	CGS001-6790	AURKA	Aurora kinase			
7413	-89.62	kd	CGS001-23102	TBC1D2B	-			
7414	-89.63	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
7415	-89.64	kd	CGS001-944	TNFSF8	CD molecules			
7416	-89.64	kd	CGS001-27244	SESN1	-			
7417	-89.65	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
7418	-89.68	kd	CGS001-6259	RYK	Type XV RTKs: RYK			
7419	-89.68	kd	CGS001-54821	ERCC6L	-			
7420	-89.68	kd	CGS001-1611	DAP	-			
7421	-89.68	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
7422	-89.7	kd	CGS001-2037	EPB41L2	-			
7423	-89.71	kd	CGS001-66008	TRAK2	-			
7424	-89.72	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
7425	-89.72	oe	ccsbBroad304_04404	TUBB6	Tubulins			
7426	-89.73	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
7427	-89.73	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
7428	-89.74	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
7429	-89.77	kd	CGS001-3880	KRT19	Intermediate filaments type I, keratins (acidic)			
7430	-89.78	cp	BRD-K10065684	dantron	Laxative			Laxative
7431	-89.79	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
7432	-89.84	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
7433	-89.9	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
7434	-89.9	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7435	-89.92	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
7436	-89.93	kd	CGS001-23411	SIRT1	Histone deacetylases			
7437	-89.93	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
7438	-89.99	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
7439	-90.01	kd	CGS001-9451	EIF2AK3	PEK subfamily			
7440	-90.01	oe	ccsbBroad304_03235	TUBD1	Tubulins			
7441	-90.01	oe	ccsbBroad304_00961	SMAD2	SMADs			
7442	-90.02	kd	CGS001-64241	ABCG8	ATP binding cassette transporters / subfamily G			
7443	-90.06	cc		Tumor necrosis factor superfamily LOF	-			
7444	-90.09	cc		BMP Signaling LOF	-			
7445	-90.09	kd	CGS001-3127	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
7446	-90.1	cp	BRD-A12560204	nitrendipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1H, CACNA1S, CACNA2D2, CACNB2, CACNG1, KCNN4	Calcium channel blocker
7447	-90.12	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7448	-90.12	cp	BRD-K62374253	rufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
7449	-90.15	kd	CGS001-1327	COX4I1	Mitochondrial respiratory chain complex			
7450	-90.18	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
7451	-90.21	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
7452	-90.22	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
7453	-90.22	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
7454	-90.24	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
7455	-90.25	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
7456	-90.29	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
7457	-90.31	oe	ccsbBroad304_07466	VGLL4	-			
7458	-90.31	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
7459	-90.33	cp	BRD-K48932581	cetraxate	Mucus protecting agent		GAST	Mucus protecting agent
7460	-90.34	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
7461	-90.34	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
7462	-90.35	kd	CGS001-4077	NBR1	-			
7463	-90.35	oe	ccsbBroad304_02249	KIAA0494	-			
7464	-90.36	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
7465	-90.38	kd	CGS001-2697	GJA1	Ion channels / Gap junction proteins (connexins)			
7466	-90.38	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
7467	-90.38	kd	CGS001-23244	PDS5A	-			
7468	-90.4	kd	CGS001-83737	ITCH	-			
7469	-90.41	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
7470	-90.42	oe	ccsbBroad304_00100	RHOA	-			
7471	-90.42	kd	CGS001-978	CDA	-			
7472	-90.43	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
7473	-90.45	kd	CGS001-4547	MTTP	-			
7474	-90.47	oe	ccsbBroad304_03798	PHTF2	-			
7475	-90.55	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
7476	-90.55	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
7477	-90.58	oe	ccsbBroad304_01855	NCOA4	-			
7478	-90.64	kd	CGS001-602	BCL3	Ankyrin repeat domain containing			
7479	-90.65	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
7480	-90.68	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
7481	-90.7	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
7482	-90.7	kd	CGS001-148327	CREB3L4	basic leucine zipper proteins			
7483	-90.71	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
7484	-90.73	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
7485	-90.74	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
7486	-90.75	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
7487	-90.76	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
7488	-90.77	kd	CGS001-134288	TMEM174	-			
7489	-90.77	kd	CGS001-5073	PARN	-			
7490	-90.77	kd	CGS001-3034	HAL	-			
7491	-90.78	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
7492	-90.79	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
7493	-90.79	oe	ccsbBroad304_06916	SCP2	-			
7494	-90.8	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
7495	-90.8	oe	ccsbBroad304_07887	GCAT	-			
7496	-90.82	cc		IKK inhibitor	-			
7497	-90.84	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
7498	-90.85	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
7499	-90.85	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
7500	-90.88	kd	CGS001-2235	FECH	-			
7501	-90.89	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
7502	-90.92	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
7503	-90.92	kd	CGS001-7465	WEE1	WEE family			
7504	-90.96	oe	ccsbBroad304_00034	AES	-			
7505	-91.06	kd	CGS001-22978	NT5C2	Adenosine turnover			
7506	-91.06	kd	CGS001-2113	ETS1	ETS Transcription Factors			
7507	-91.08	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
7508	-91.08	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
7509	-91.1	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
7510	-91.11	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
7511	-91.12	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
7512	-91.13	kd	CGS001-10873	ME3	-			
7513	-91.14	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
7514	-91.16	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
7515	-91.18	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
7516	-91.18	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
7517	-91.18	kd	CGS001-818	CAMK2G	CAMK2 family			
7518	-91.19	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
7519	-91.24	oe	ccsbBroad304_00874	INS	-			
7520	-91.24	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
7521	-91.24	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
7522	-91.25	kd	CGS001-93594	WDR67	-			
7523	-91.29	kd	CGS001-3572	IL6ST	IL-6 receptor family			
7524	-91.3	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
7525	-91.3	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
7526	-91.31	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
7527	-91.33	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
7528	-91.34	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
7529	-91.34	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
7530	-91.34	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
7531	-91.35	cp	BRD-K73196317	urapidil	Adrenergic receptor antagonist		HTR1A	Adrenergic receptor antagonist
7532	-91.36	kd	CGS001-6464	SHC1	SH2 domain containing			
7533	-91.38	kd	CGS001-2863	GPR39	GPCR / Class A : Orphans			
7534	-91.39	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
7535	-91.41	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
7536	-91.42	oe	ccsbBroad304_03928	RRAGC	-			
7537	-91.44	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
7538	-91.46	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
7539	-91.47	kd	CGS001-8915	BCL10	-			
7540	-91.48	kd	CGS001-6897	TARS	Aminoacyl tRNA synthetases / Class II			
7541	-91.5	oe	ccsbBroad304_02604	B3GNT1	-			
7542	-91.53	kd	CGS001-319100	TAAR6	GPCR / Class A : Trace amine associated receptors			
7543	-91.56	kd	CGS001-7511	XPNPEP1	Methionyl aminopeptidase			
7544	-91.57	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
7545	-91.59	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
7546	-91.6	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
7547	-91.62	kd	CGS001-4968	OGG1	-			
7548	-91.62	kd	CGS001-4485	MST1	-			
7549	-91.64	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
7550	-91.65	kd	CGS001-50814	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7551	-91.69	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
7552	-91.71	kd	CGS001-8824	CES2	Carboxylesterases			
7553	-91.73	cc		Zinc fingers RanBP2 type LOF	-			
7554	-91.73	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
7555	-91.75	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
7556	-91.75	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
7557	-91.77	kd	CGS001-9641	IKBKE	IKK family			
7558	-91.78	kd	CGS001-9020	MAP3K14	MAPKKK:STE-unique family			
7559	-91.8	kd	CGS001-4709	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
7560	-91.81	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
7561	-91.83	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
7562	-91.85	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
7563	-91.88	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
7564	-91.89	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
7565	-91.91	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
7566	-91.93	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
7567	-91.93	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
7568	-91.93	kd	CGS001-114904	C1QTNF6	-			
7569	-91.94	oe	ccsbBroad304_01038	MSRA	-			
7570	-91.95	oe	ccsbBroad304_07320	SQSTM1	-			
7571	-91.96	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
7572	-92	kd	CGS001-9140	ATG12	-			
7573	-92.02	cp	BRD-K49481516	galantamine	Acetylcholinesterase inhibitor		ACHE, BCHE, CHRNA1, CHRNA10, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNA9, CHRNB1, CHRNB2, CHRNB3, CHRNB4, CHRND, CHRNE, CHRNG	Acetylcholinesterase inhibitor
7574	-92.04	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
7575	-92.06	kd	CGS001-9929	JOSD1	-			
7576	-92.07	kd	CGS001-6303	SAT1	-			
7577	-92.1	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
7578	-92.11	oe	ccsbBroad304_01146	PARN	-			
7579	-92.17	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
7580	-92.18	oe	ccsbBroad304_02048	BCL10	-			
7581	-92.22	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
7582	-92.26	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
7583	-92.35	cc		Aminoacyl tRNA synthetases class II LOF	-			
7584	-92.36	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
7585	-92.37	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
7586	-92.38	kd	CGS001-10051	SMC4	Structural maintenance of chromosomes proteins			
7587	-92.44	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
7588	-92.47	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
7589	-92.47	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
7590	-92.48	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
7591	-92.48	oe	ccsbBroad304_13598	NRBP2	NRBP family			
7592	-92.52	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
7593	-92.53	oe	ccsbBroad304_02789	ADAT1	-			
7594	-92.53	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
7595	-92.57	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
7596	-92.58	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
7597	-92.59	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
7598	-92.63	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
7599	-92.63	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
7600	-92.64	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
7601	-92.66	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
7602	-92.69	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
7603	-92.7	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
7604	-92.73	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
7605	-92.75	kd	CGS001-2353	FOS	basic leucine zipper proteins			
7606	-92.78	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
7607	-92.79	kd	CGS001-5264	PHYH	-			
7608	-92.8	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
7609	-92.81	cc		Non Homologous End Joining LOF	-			
7610	-92.85	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
7611	-92.86	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
7612	-92.87	cp	BRD-A75935363	atracurium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
7613	-92.89	kd	CGS001-7167	TPI1	-			
7614	-92.92	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
7615	-92.92	oe	ccsbBroad304_02581	ASCC3	-			
7616	-92.95	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
7617	-92.95	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
7618	-92.96	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
7619	-92.96	kd	CGS001-23057	NMNAT2	-			
7620	-92.97	cc		Structural maintenance of chromosomes proteins LOF	-			
7621	-92.97	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
7622	-92.97	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
7623	-92.97	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
7624	-92.99	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
7625	-93	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
7626	-93.03	oe	ccsbBroad304_00430	GADD45A	-			
7627	-93.03	kd	CGS001-3651	PDX1	Homeoboxes / ANTP class : HOXL subclass			
7628	-93.05	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
7629	-93.05	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
7630	-93.05	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
7631	-93.06	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
7632	-93.06	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
7633	-93.06	kd	CGS001-7480	WNT10B	Wingless-type MMTV integration sites			
7634	-93.07	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
7635	-93.07	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
7636	-93.08	kd	CGS001-637	BID	Endogenous ligands			
7637	-93.11	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
7638	-93.11	oe	ccsbBroad304_02018	SUCLA2	-			
7639	-93.12	kd	CGS001-112812	FDX1L	-			
7640	-93.13	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
7641	-93.14	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
7642	-93.15	oe	ccsbBroad304_01769	VEGFB	-			
7643	-93.15	kd	CGS001-51070	NOSIP	-			
7644	-93.22	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
7645	-93.23	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
7646	-93.24	kd	CGS001-1831	TSC22D3	-			
7647	-93.27	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
7648	-93.28	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
7649	-93.29	kd	CGS001-10962	MLLT11	-			
7650	-93.29	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
7651	-93.31	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
7652	-93.32	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
7653	-93.32	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
7654	-93.33	oe	ccsbBroad304_01101	NME1	-			
7655	-93.35	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
7656	-93.37	kd	CGS001-51024	FIS1	-			
7657	-93.38	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
7658	-93.39	oe	ccsbBroad304_04655	TRIM9	-			
7659	-93.4	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
7660	-93.4	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
7661	-93.41	cc		NFKB Activation GOF	-			
7662	-93.41	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
7663	-93.42	cp	BRD-K22227508	targinine	Nitric oxide synthase inhibitor		NOS2, NOS3	Nitric oxide synthase inhibitor
7664	-93.42	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
7665	-93.44	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
7666	-93.44	kd	CGS001-6721	SREBF2	Basic helix-loop-helix proteins			
7667	-93.44	oe	ccsbBroad304_09396	TIRAP	-			
7668	-93.45	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
7669	-93.45	kd	CGS001-166	AES	-			
7670	-93.46	kd	CGS001-23046	KIF21B	Kinesins			
7671	-93.48	oe	ccsbBroad304_07197	PDHX	-			
7672	-93.49	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
7673	-93.51	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
7674	-93.51	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
7675	-93.54	oe	ccsbBroad304_03808	ERGIC1	-			
7676	-93.55	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
7677	-93.56	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
7678	-93.57	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
7679	-93.58	kd	CGS001-81533	ITFG1	-			
7680	-93.59	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
7681	-93.62	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
7682	-93.66	kd	CGS001-1856	DVL2	Dishevelled homologs			
7683	-93.66	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
7684	-93.67	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
7685	-93.67	kd	CGS001-6391	SDHC	Mitochondrial respiratory chain complex / Complex II			
7686	-93.68	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
7687	-93.7	kd	CGS001-7089	TLE2	WD repeat domain containing			
7688	-93.71	oe	ccsbBroad304_00077	APEX1	-			
7689	-93.71	cp	BRD-K86887724	dofetilide	Potassium channel blocker		KCNH2, KCNH1, KCNJ12, KCNK2	Potassium channel blocker
7690	-93.72	kd	CGS001-11325	DDX42	DEAD-boxes			
7691	-93.75	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
7692	-93.76	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
7693	-93.77	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
7694	-93.77	kd	CGS001-5293	PIK3CD	Phosphatidylinositol kinases			
7695	-93.8	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
7696	-93.83	kd	CGS001-9568	GABBR2	GABA receptors			
7697	-93.86	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
7698	-93.86	kd	CGS001-64786	TBC1D15	-			
7699	-93.87	kd	CGS001-64170	CARD9	-			
7700	-93.89	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
7701	-93.9	kd	CGS001-56005	C19ORF10	-			
7702	-93.91	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
7703	-93.92	kd	CGS001-10312	TCIRG1	ATPases / V-type			
7704	-93.94	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
7705	-93.95	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
7706	-93.96	oe	ccsbBroad304_01166	PDK2	PDHK family			
7707	-93.97	oe	ccsbBroad304_03420	TOLLIP	-			
7708	-94	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
7709	-94.03	cp	BRD-A37052580	physostigmine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Cholinesterase inhibitor
7710	-94.03	kd	CGS001-1662	DDX10	DEAD-boxes			
7711	-94.04	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
7712	-94.05	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
7713	-94.05	oe	ccsbBroad304_08452	PIH1D1	-			
7714	-94.08	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
7715	-94.09	kd	CGS001-8667	EIF3H	-			
7716	-94.1	oe	ccsbBroad304_00070	ANXA5	Annexins			
7717	-94.11	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
7718	-94.12	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
7719	-94.12	oe	ccsbBroad304_02572	SERINC3	-			
7720	-94.14	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
7721	-94.17	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
7722	-94.19	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
7723	-94.2	kd	CGS001-27	ABL2	Abl family			
7724	-94.23	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
7725	-94.23	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
7726	-94.28	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
7727	-94.3	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
7728	-94.33	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
7729	-94.33	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
7730	-94.33	kd	CGS001-10695	CNPY3	Trinucleotide (CAG) repeat containing			
7731	-94.35	oe	ccsbBroad304_02372	SPRY1	-			
7732	-94.35	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
7733	-94.38	kd	CGS001-1022	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
7734	-94.38	kd	CGS001-6129	RPL7	L ribosomal proteins			
7735	-94.39	cc		T-type calcium channel blocker	-			
7736	-94.39	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
7737	-94.4	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
7738	-94.4	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
7739	-94.42	kd	CGS001-1645	AKR1C1	Aldo-keto reductases			
7740	-94.43	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
7741	-94.45	kd	CGS001-638	BIK	-			
7742	-94.46	oe	ccsbBroad304_02801	CASP14	Caspases			
7743	-94.46	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
7744	-94.46	oe	ccsbBroad304_02012	FADD	-			
7745	-94.47	kd	CGS001-9404	LPXN	-			
7746	-94.48	kd	CGS001-4931	NVL	ATPases / AAA-type			
7747	-94.48	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
7748	-94.49	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
7749	-94.49	oe	ccsbBroad304_01401	RIT1	-			
7750	-94.5	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
7751	-94.5	kd	CGS001-89882	TPD52L3	-			
7752	-94.51	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
7753	-94.51	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
7754	-94.52	cc		Progesterone receptor agonist	-			
7755	-94.53	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
7756	-94.55	cp	BRD-K05350981	oligomycin-c	ATPase inhibitor		ATP5A1	ATPase inhibitor, ATP synthase inhibitor
7757	-94.56	kd	CGS001-55163	PNPO	-			
7758	-94.57	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
7759	-94.59	oe	ccsbBroad304_01584	SPARC	-			
7760	-94.6	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
7761	-94.6	kd	CGS001-7018	TF	-			
7762	-94.61	cc		Protein synthesis inhibitor	-			
7763	-94.61	kd	CGS001-652	BMP4	Bone morphogenetic proteins			
7764	-94.62	cc		ATP synthase inhibitor	-			
7765	-94.63	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
7766	-94.63	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
7767	-94.64	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
7768	-94.65	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
7769	-94.65	kd	CGS001-6741	SSB	La ribonucleoprotein domain containing			
7770	-94.69	kd	CGS001-4200	ME2	-			
7771	-94.71	kd	CGS001-23512	SUZ12	Zinc fingers, C2H2-type			
7772	-94.72	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
7773	-94.74	kd	CGS001-645	BLVRB	Short chain dehydrogenase/reductase superfamily / Atypical members			
7774	-94.79	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
7775	-94.79	kd	CGS001-7936	RDBP	-			
7776	-94.79	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
7777	-94.8	kd	CGS001-4297	MLL	-			
7778	-94.81	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7779	-94.81	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
7780	-94.82	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
7781	-94.84	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
7782	-94.84	kd	CGS001-9377	COX5A	Mitochondrial respiratory chain complex			
7783	-94.85	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
7784	-94.86	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
7785	-94.87	kd	CGS001-10933	MORF4L1	-			
7786	-94.89	kd	CGS001-6723	SRM	-			
7787	-94.9	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
7788	-94.91	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
7789	-94.91	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
7790	-94.93	oe	ccsbBroad304_08645	BCCIP	-			
7791	-94.94	kd	CGS001-2266	FGG	Endogenous ligands			
7792	-94.95	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
7793	-94.96	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
7794	-94.96	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
7795	-94.96	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
7796	-94.99	oe	ccsbBroad304_00101	RHOC	-			
7797	-94.99	kd	CGS001-2677	GGCX	Carboxylases			
7798	-95	oe	ccsbBroad304_00657	GNG4	-			
7799	-95	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
7800	-95	kd	CGS001-6599	SMARCC1	-			
7801	-95	kd	CGS001-5825	ABCD3	ATP binding cassette transporters / subfamily D			
7802	-95.01	kd	CGS001-6146	RPL22	L ribosomal proteins			
7803	-95.02	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7804	-95.02	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
7805	-95.03	cp	BRD-K15916496	clotrimazole	Cytochrome P450 inhibitor		KCNN4, CYP3A4, CYP51A1, NR1I2, NR1I3, TRPM2, TRPM4, TRPM8	Cytochrome P450 inhibitor, Imidazoline receptor ligand
7806	-95.05	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
7807	-95.06	cc		Mitochondrial complex IV LOF	-			
7808	-95.09	kd	CGS001-26511	CHIC2	-			
7809	-95.1	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
7810	-95.12	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
7811	-95.14	cc		PARP inhibitor	-			
7812	-95.15	kd	CGS001-8660	IRS2	Pleckstrin homology (PH) domain containing			
7813	-95.16	kd	CGS001-206358	SLC36A1	SLC36 family of proton-coupled amino acid transporters			
7814	-95.17	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
7815	-95.17	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
7816	-95.19	kd	CGS001-2160	F11	Chymotrypsin			
7817	-95.19	kd	CGS001-3485	IGFBP2	insulin-like growth factor (IGF) binding proteins			
7818	-95.19	oe	ccsbBroad304_04534	HN1L	-			
7819	-95.22	kd	CGS001-4905	NSF	ATPases / AAA-type			
7820	-95.24	oe	ccsbBroad304_02094	FIBP	-			
7821	-95.24	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
7822	-95.25	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
7823	-95.25	oe	ccsbBroad304_07820	SNW1	-			
7824	-95.27	kd	CGS001-11041	B3GNT1	-			
7825	-95.29	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
7826	-95.31	kd	CGS001-4718	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
7827	-95.31	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
7828	-95.34	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
7829	-95.35	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
7830	-95.42	kd	CGS001-23761	PISD	Decarboxylases			
7831	-95.42	kd	CGS001-899	CCNF	F-boxes / other			
7832	-95.45	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
7833	-95.46	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
7834	-95.47	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
7835	-95.48	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
7836	-95.49	cc		KCNJ11 modulator	-			
7837	-95.49	oe	ccsbBroad304_07600	NSA2	-			
7838	-95.49	kd	CGS001-10254	STAM2	-			
7839	-95.51	cp	BRD-A88254928	salbutamol	Adrenergic receptor agonist		ADRB2, ADRB1	Adrenergic receptor agonist
7840	-95.51	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
7841	-95.51	kd	CGS001-3161	HMMR	CD molecules			
7842	-95.55	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
7843	-95.55	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
7844	-95.56	oe	ccsbBroad304_00237	CCND3	-			
7845	-95.57	kd	CGS001-6307	MSMO1	Fatty acid hydroxylase domain containing			
7846	-95.58	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
7847	-95.61	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
7848	-95.62	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
7849	-95.62	kd	CGS001-91975	ZNF300	Zinc fingers, C2H2-type			
7850	-95.62	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
7851	-95.67	kd	CGS001-6696	SPP1	Endogenous ligands			
7852	-95.67	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
7853	-95.68	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
7854	-95.69	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
7855	-95.69	kd	CGS001-9787	DLGAP5	-			
7856	-95.69	kd	CGS001-400	ARL1	ADP-ribosylation factors			
7857	-95.7	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
7858	-95.7	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
7859	-95.7	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
7860	-95.7	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
7861	-95.72	kd	CGS001-7150	TOP1	DNA Topoisomerases			
7862	-95.73	kd	CGS001-708	C1QBP	-			
7863	-95.74	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
7864	-95.74	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
7865	-95.75	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
7866	-95.76	kd	CGS001-10020	GNE	-			
7867	-95.78	cc		Integrin subunits alpha LOF	-			
7868	-95.78	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
7869	-95.81	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
7870	-95.81	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
7871	-95.83	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
7872	-95.86	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
7873	-95.86	oe	ccsbBroad304_02843	FTSJ1	-			
7874	-95.87	kd	CGS001-1727	CYB5R3	-			
7875	-95.87	oe	ccsbBroad304_00472	EBF1	-			
7876	-95.88	oe	ccsbBroad304_03310	LCMT1	-			
7877	-95.91	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7878	-95.91	oe	ccsbBroad304_01327	PSPH	-			
7879	-95.91	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
7880	-95.92	cc		RNA Polymerase Enzymes LOF	-			
7881	-95.92	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
7882	-95.92	kd	CGS001-5423	POLB	DNA polymerases			
7883	-95.92	kd	CGS001-192286	HIGD2A	-			
7884	-95.93	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
7885	-95.95	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
7886	-95.97	oe	ccsbBroad304_01593	SRP14	-			
7887	-95.98	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
7888	-95.98	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
7889	-95.99	kd	CGS001-7267	TTC3	RING-type (C3HC4) zinc fingers			
7890	-95.99	kd	CGS001-2030	SLC29A1	SLC29 family			
7891	-96.01	cp	BRD-K88304388	dextrorphan	Glutamate receptor antagonist		OPRM1, OPRK1, OPRD1, GRIN1, HTR1A, SLC6A2	Glutamate receptor antagonist
7892	-96.01	kd	CGS001-5209	PFKFB3	-			
7893	-96.05	kd	CGS001-23212	RRS1	-			
7894	-96.07	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
7895	-96.1	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
7896	-96.12	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
7897	-96.12	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
7898	-96.13	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
7899	-96.15	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
7900	-96.17	cc		Canonical high mobility group proteins LOF	-			
7901	-96.18	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
7902	-96.2	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
7903	-96.2	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
7904	-96.21	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
7905	-96.21	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
7906	-96.22	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
7907	-96.23	kd	CGS001-23475	QPRT	-			
7908	-96.23	kd	CGS001-10671	DCTN6	-			
7909	-96.24	kd	CGS001-3925	STMN1	-			
7910	-96.25	kd	CGS001-4048	LTA4H	Hydrolases			
7911	-96.26	kd	CGS001-293	SLC25A6	Mitochondrial nucleotide transporter subfamily			
7912	-96.26	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
7913	-96.28	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
7914	-96.3	oe	ccsbBroad304_05183	TXLNA	-			
7915	-96.3	cp	BRD-K94649603	taxifolin	Opioid receptor antagonist		APOB, APP, HMGCR	Opioid receptor antagonist
7916	-96.3	oe	ccsbBroad304_06663	OAS1	-			
7917	-96.31	kd	CGS001-6337	SCNN1A	Epithelial sodium channels (ENaC)			
7918	-96.32	kd	CGS001-5829	PXN	-			
7919	-96.33	kd	CGS001-2194	FASN	Short chain dehydrogenase/reductase superfamily / Atypical members			
7920	-96.34	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
7921	-96.36	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
7922	-96.38	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
7923	-96.41	cp	BRD-K37814297	acepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
7924	-96.42	kd	CGS001-8031	NCOA4	-			
7925	-96.44	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
7926	-96.44	cp	BRD-K92413528	thiazolidinecarboxylic-acid	Reducing agent			Reducing agent
7927	-96.44	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
7928	-96.44	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
7929	-96.45	oe	ccsbBroad304_00551	FECH	-			
7930	-96.46	kd	CGS001-9688	NUP93	-			
7931	-96.47	oe	ccsbBroad304_14291	GDPD5	-			
7932	-96.48	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
7933	-96.5	kd	CGS001-5294	PIK3CG	Phosphatidylinositol kinases			
7934	-96.51	kd	CGS001-81620	CDT1	-			
7935	-96.54	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
7936	-96.55	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
7937	-96.55	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
7938	-96.56	oe	ccsbBroad304_00113	ASNS	-			
7939	-96.57	kd	CGS001-7471	WNT1	Endogenous ligands			
7940	-96.59	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
7941	-96.59	cp	BRD-K07237224	moclobemide	Monoamine oxidase inhibitor		MAOA, CYP2C19, MAOB	Monoamine oxidase inhibitor
7942	-96.62	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
7943	-96.62	cp	BRD-K92870997	pterostilbene	Cyclooxygenase inhibitor		FAAH, PPARA, PTGS1, PTGS2	Cyclooxygenase inhibitor, PPAR receptor agonist
7944	-96.63	kd	CGS001-301	ANXA1	Annexins			
7945	-96.63	kd	CGS001-9589	WTAP	-			
7946	-96.64	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
7947	-96.64	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
7948	-96.65	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
7949	-96.65	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
7950	-96.67	oe	ccsbBroad304_00645	GCLM	-			
7951	-96.67	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7952	-96.67	kd	CGS001-1196	CLK2	CDC-like kinases			
7953	-96.68	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
7954	-96.68	kd	CGS001-55718	POLR3E	RNA polymerase subunits			
7955	-96.68	kd	CGS001-11333	PDAP1	-			
7956	-96.69	kd	CGS001-4835	NQO2	-			
7957	-96.69	kd	CGS001-3827	KNG1	Endogenous ligands			
7958	-96.71	oe	ccsbBroad304_01174	PEX13	-			
7959	-96.71	kd	CGS001-10142	AKAP9	A-kinase anchor proteins			
7960	-96.72	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
7961	-96.73	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
7962	-96.73	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
7963	-96.74	kd	CGS001-9710	KIAA0355	-			
7964	-96.74	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
7965	-96.76	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
7966	-96.76	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
7967	-96.77	kd	CGS001-2737	GLI3	Zinc fingers, C2H2-type			
7968	-96.78	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
7969	-96.79	kd	CGS001-2961	GTF2E2	General transcription factors			
7970	-96.79	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
7971	-96.81	oe	ccsbBroad304_06993	SRD5A1	-			
7972	-96.81	oe	ccsbBroad304_02788	PRAME	-			
7973	-96.81	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
7974	-96.82	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
7975	-96.82	oe	ccsbBroad304_04788	OVCA2	-			
7976	-96.84	kd	CGS001-9467	SH3BP5	-			
7977	-96.85	cp	BRD-K85030058	benactyzine	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
7978	-96.86	kd	CGS001-9805	SCRN1	-			
7979	-96.86	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
7980	-96.87	kd	CGS001-3312	HSPA8	Heat shock proteins / HSP70			
7981	-96.88	kd	CGS001-124626	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7982	-96.89	kd	CGS001-11214	AKAP13	A-kinase anchor proteins			
7983	-96.9	kd	CGS001-9326	ZNHIT3	Zinc fingers, HIT-type			
7984	-96.92	kd	CGS001-6927	HNF1A	Homeoboxes / HNF class			
7985	-96.93	oe	ccsbBroad304_00832	IFNB1	Interferons			
7986	-96.93	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
7987	-96.93	kd	CGS001-57396	CLK4	CDC-like kinases			
7988	-96.94	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
7989	-96.94	oe	ccsbBroad304_02205	WTAP	-			
7990	-96.95	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
7991	-96.98	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
7992	-96.99	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
7993	-97	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
7994	-97	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
7995	-97.02	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
7996	-97.04	kd	CGS001-6591	SNAI2	Snail homologs			
7997	-97.06	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
7998	-97.06	kd	CGS001-8801	SUCLG2	-			
7999	-97.08	oe	ccsbBroad304_08152	PSAT1	-			
8000	-97.08	cp	BRD-K22947005	dexbrompheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
8001	-97.08	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
8002	-97.09	kd	CGS001-3017	HIST1H2BD	Histones / Replication-dependent			
8003	-97.09	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
8004	-97.12	kd	CGS001-1875	E2F5	-			
8005	-97.13	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
8006	-97.14	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
8007	-97.15	cc		EIF Proteins LOF	-			
8008	-97.15	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
8009	-97.18	oe	ccsbBroad304_10240	CROT	-			
8010	-97.18	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
8011	-97.19	kd	CGS001-595	CCND1	-			
8012	-97.19	kd	CGS001-5932	RBBP8	-			
8013	-97.2	oe	ccsbBroad304_00833	IFNG	Interferons			
8014	-97.2	kd	CGS001-204851	HIPK1	HIPK subfamily			
8015	-97.22	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
8016	-97.22	cp	BRD-K39621635	artemether	Antimalarial		ATP1A1, CYP2B6, CYP2C19, CYP3A5	Antimalarial
8017	-97.22	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
8018	-97.24	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
8019	-97.26	kd	CGS001-51460	SFMBT1	Sterile alpha motif (SAM) domain containing			
8020	-97.26	kd	CGS001-10482	NXF1	-			
8021	-97.27	kd	CGS001-7879	RAB7A	RAB, member RAS oncogene			
8022	-97.33	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
8023	-97.33	kd	CGS001-5058	PAK1	PAKA subfamily			
8024	-97.33	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
8025	-97.34	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
8026	-97.35	kd	CGS001-55422	ZNF331	Zinc fingers, C2H2-type			
8027	-97.36	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
8028	-97.36	kd	CGS001-26574	AATF	-			
8029	-97.39	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
8030	-97.4	cc		PI3K inhibitor	-			
8031	-97.4	kd	CGS001-7428	VHL	-			
8032	-97.41	kd	CGS001-53347	UBASH3A	-			
8033	-97.42	kd	CGS001-1029	CDKN2A	-			
8034	-97.43	kd	CGS001-55011	PIH1D1	-			
8035	-97.43	kd	CGS001-55193	PBRM1	Non-enzymatic BRD containing proteins			
8036	-97.43	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
8037	-97.44	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
8038	-97.45	oe	ccsbBroad304_00956	LYZ	-			
8039	-97.45	kd	CGS001-23581	CASP14	Caspases			
8040	-97.46	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
8041	-97.48	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
8042	-97.5	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
8043	-97.5	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
8044	-97.5	oe	ccsbBroad304_00462	DR1	-			
8045	-97.51	kd	CGS001-7357	UGCG	Glycosyltransferase family 2 domain containing			
8046	-97.55	oe	ccsbBroad304_04379	LZIC	-			
8047	-97.56	kd	CGS001-4092	SMAD7	SMADs			
8048	-97.56	kd	CGS001-673	BRAF	RAF family			
8049	-97.57	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
8050	-97.6	kd	CGS001-6936	C2ORF3	-			
8051	-97.61	oe	ccsbBroad304_06639	NFYB	-			
8052	-97.61	kd	CGS001-4046	LSP1	-			
8053	-97.64	cc		Minor histocompatibility antigens LOF	-			
8054	-97.64	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
8055	-97.66	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
8056	-97.67	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
8057	-97.67	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
8058	-97.69	kd	CGS001-10245	TIMM17B	-			
8059	-97.69	oe	ccsbBroad304_06574	MDH2	-			
8060	-97.7	kd	CGS001-6016	RIT1	-			
8061	-97.71	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
8062	-97.71	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
8063	-97.71	kd	CGS001-50	ACO2	-			
8064	-97.71	oe	ccsbBroad304_07814	SACM1L	-			
8065	-97.72	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
8066	-97.73	kd	CGS001-6207	RPS13	S ribosomal proteins			
8067	-97.73	kd	CGS001-3419	IDH3A	-			
8068	-97.73	kd	CGS001-2944	GSTM1	Glutathione S-transferases / Soluble			
8069	-97.74	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
8070	-97.75	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
8071	-97.76	kd	CGS001-7082	TJP1	-			
8072	-97.76	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
8073	-97.76	kd	CGS001-1453	CSNK1D	Casein kinase 1 (CK1) family			
8074	-97.77	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
8075	-97.77	kd	CGS001-6772	STAT1	SH2 domain containing			
8076	-97.78	cc		MTOR inhibitor	-			
8077	-97.78	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
8078	-97.78	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
8079	-97.82	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
8080	-97.82	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
8081	-97.84	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
8082	-97.84	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
8083	-97.84	kd	CGS001-9124	PDLIM1	-			
8084	-97.84	oe	ccsbBroad304_10487	BPHL	-			
8085	-97.85	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
8086	-97.85	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
8087	-97.85	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
8088	-97.86	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
8089	-97.87	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
8090	-97.87	oe	ccsbBroad304_08952	E2F8	-			
8091	-97.87	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
8092	-97.88	oe	ccsbBroad304_02458	STK25	YSK subfamily			
8093	-97.89	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
8094	-97.89	kd	CGS001-54861	SNRK	SNRK subfamily			
8095	-97.89	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
8096	-97.91	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
8097	-97.91	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
8098	-97.91	kd	CGS001-384	ARG2	Arginase			
8099	-97.91	oe	ccsbBroad304_02197	VPS26A	-			
8100	-97.92	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
8101	-97.92	kd	CGS001-7083	TK1	-			
8102	-97.93	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
8103	-97.94	oe	ccsbBroad304_01976	EIF4EBP3	-			
8104	-97.95	kd	CGS001-6617	SNAPC1	-			
8105	-97.96	oe	ccsbBroad304_02702	MSRB2	-			
8106	-97.96	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
8107	-97.96	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
8108	-97.96	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
8109	-97.97	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
8110	-97.97	kd	CGS001-1050	CEBPA	basic leucine zipper proteins			
8111	-97.98	kd	CGS001-5610	EIF2AK2	Other PEK family kinases			
8112	-98	cp	BRD-K15519488	CS-110266	Dopamine receptor agonist		SLC6A3	Dopamine receptor agonist
8113	-98	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
8114	-98	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
8115	-98	kd	CGS001-84290	CAPNS2	EF-hand domain containing			
8116	-98	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
8117	-98.03	cp	BRD-K47780086	penciclovir	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor
8118	-98.03	kd	CGS001-1184	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
8119	-98.05	kd	CGS001-55278	QRSL1	-			
8120	-98.06	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
8121	-98.06	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
8122	-98.08	kd	CGS001-11215	AKAP11	A-kinase anchor proteins			
8123	-98.1	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
8124	-98.13	cp	BRD-K13800121	parecoxib	Cyclooxygenase inhibitor		LTF, PTGS2	Cyclooxygenase inhibitor
8125	-98.13	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
8126	-98.13	kd	CGS001-7100	TLR5	Toll-like receptor family			
8127	-98.13	kd	CGS001-79722	ANKRD55	Ankyrin repeat domain containing			
8128	-98.15	kd	CGS001-10190	TXNDC9	-			
8129	-98.15	kd	CGS001-10381	TUBB3	Tubulins			
8130	-98.16	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
8131	-98.16	kd	CGS001-204	AK2	Adenylate kinases			
8132	-98.19	oe	ccsbBroad304_02626	PKIG	-			
8133	-98.19	oe	ccsbBroad304_06103	DMD	-			
8134	-98.19	kd	CGS001-57048	PLSCR3	-			
8135	-98.21	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
8136	-98.23	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
8137	-98.24	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
8138	-98.24	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
8139	-98.24	kd	CGS001-9156	EXO1	-			
8140	-98.24	oe	ccsbBroad304_08879	CASD1	-			
8141	-98.25	kd	CGS001-7184	HSP90B1	Heat shock proteins / HSPC			
8142	-98.26	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
8143	-98.27	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
8144	-98.28	oe	ccsbBroad304_00810	HYAL1	-			
8145	-98.29	kd	CGS001-55781	RIOK2	RIO2 subfamily			
8146	-98.3	kd	CGS001-8891	EIF2B3	-			
8147	-98.31	oe	ccsbBroad304_01164	PDHB	-			
8148	-98.32	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
8149	-98.32	kd	CGS001-8226	HDHD1	-			
8150	-98.33	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
8151	-98.33	kd	CGS001-6418	SET	-			
8152	-98.33	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
8153	-98.34	kd	CGS001-226	ALDOA	-			
8154	-98.36	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
8155	-98.36	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
8156	-98.36	kd	CGS001-54472	TOLLIP	-			
8157	-98.36	kd	CGS001-3755	KCNG1	Voltage-gated potassium channels			
8158	-98.38	oe	ccsbBroad304_02032	TSC22D1	-			
8159	-98.38	oe	ccsbBroad304_00817	IDH2	-			
8160	-98.38	kd	CGS001-55129	ANO10	Calcium activated chloride channel			
8161	-98.38	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
8162	-98.39	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
8163	-98.42	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
8164	-98.43	oe	ccsbBroad304_03732	NPDC1	-			
8165	-98.44	kd	CGS001-3313	HSPA9	Heat shock proteins / HSP70			
8166	-98.45	kd	CGS001-9697	TRAM2	-			
8167	-98.45	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
8168	-98.47	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
8169	-98.48	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
8170	-98.48	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
8171	-98.48	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
8172	-98.48	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
8173	-98.48	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
8174	-98.5	kd	CGS001-6670	SP3	Specificity protein transcription factors			
8175	-98.5	kd	CGS001-3985	LIMK2	LIMK subfamily			
8176	-98.51	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
8177	-98.52	oe	ccsbBroad304_06386	HNMT	-			
8178	-98.52	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
8179	-98.52	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
8180	-98.52	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
8181	-98.53	cp	BRD-A64297288	amlodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, ABCG2, CA1, CACNA1B, CACNA1S, CACNA2D3, CACNB1, CACNB2, SMPD1	Calcium channel blocker
8182	-98.53	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
8183	-98.56	cc		SMAD family LOF	-			
8184	-98.56	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
8185	-98.56	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
8186	-98.56	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
8187	-98.56	kd	CGS001-900	CCNG1	-			
8188	-98.58	kd	CGS001-79711	IPO4	Importins			
8189	-98.59	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
8190	-98.59	kd	CGS001-54205	CYCS	-			
8191	-98.59	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
8192	-98.59	kd	CGS001-7182	NR2C2	Testicular receptors			
8193	-98.59	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
8194	-98.6	cc		Bacterial cell wall synthesis inhibitor	-			
8195	-98.61	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
8196	-98.61	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
8197	-98.62	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
8198	-98.62	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
8199	-98.63	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
8200	-98.63	kd	CGS001-5920	RARRES3	-			
8201	-98.63	kd	CGS001-9703	KIAA0100	-			
8202	-98.63	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
8203	-98.65	kd	CGS001-9475	ROCK2	Pleckstrin homology (PH) domain containing			
8204	-98.67	oe	ccsbBroad304_06783	LGMN	Legumain			
8205	-98.68	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
8206	-98.69	kd	CGS001-6477	SIAH1	-			
8207	-98.69	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
8208	-98.7	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
8209	-98.7	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
8210	-98.7	kd	CGS001-6493	SIM2	Basic helix-loop-helix proteins			
8211	-98.7	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
8212	-98.72	kd	CGS001-2232	FDXR	-			
8213	-98.75	oe	ccsbBroad304_01186	PHB	-			
8214	-98.75	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
8215	-98.76	cp	BRD-A41450521	tosufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
8216	-98.76	kd	CGS001-6233	RPS27A	S ribosomal proteins			
8217	-98.77	cp	BRD-A24543851	nornicotine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
8218	-98.77	kd	CGS001-5664	PSEN2	Presenilin			
8219	-98.78	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
8220	-98.79	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
8221	-98.79	kd	CGS001-5901	RAN	-			
8222	-98.79	kd	CGS001-2879	GPX4	-			
8223	-98.79	kd	CGS001-6275	S100A4	EF-hand domain containing			
8224	-98.79	kd	CGS001-3265	HRAS	RAS subfamily			
8225	-98.8	oe	ccsbBroad304_05980	CDKN1B	-			
8226	-98.8	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
8227	-98.82	kd	CGS001-4697	NDUFA4	-			
8228	-98.83	cp	BRD-K99063460	didanosine	Nucleoside reverse transcriptase inhibitor		PNP	Nucleoside reverse transcriptase inhibitor
8229	-98.83	kd	CGS001-10111	RAD50	-			
8230	-98.83	kd	CGS001-4926	NUMA1	-			
8231	-98.84	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
8232	-98.84	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
8233	-98.84	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
8234	-98.85	kd	CGS001-10769	PLK2	Polo-like kinase (PLK) family			
8235	-98.86	kd	CGS001-6788	STK3	MST subfamily			
8236	-98.86	kd	CGS001-3673	ITGA2	Integrins			
8237	-98.87	kd	CGS001-10525	HYOU1	Heat shock proteins / HSP70			
8238	-98.87	kd	CGS001-1595	CYP51A1	Cytochrome P450s			
8239	-98.88	cc		Sirtuins GOF	-			
8240	-98.88	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
8241	-98.89	oe	ccsbBroad304_07889	QPRT	-			
8242	-98.89	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
8243	-98.89	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
8244	-98.91	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
8245	-98.91	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
8246	-98.92	kd	CGS001-2987	GUK1	-			
8247	-98.93	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
8248	-98.93	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
8249	-98.94	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
8250	-98.94	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
8251	-98.94	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
8252	-98.94	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
8253	-98.95	kd	CGS001-54998	AURKAIP1	-			
8254	-98.98	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
8255	-99	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
8256	-99	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
8257	-99	kd	CGS001-4771	NF2	A-kinase anchor proteins			
8258	-99	kd	CGS001-3226	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
8259	-99	kd	CGS001-10898	CPSF4	-			
8260	-99.01	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
8261	-99.01	kd	CGS001-79187	FSD1	Fibronectin type III domain containing			
8262	-99.03	cc		Kinase anchoring proteins LOF	-			
8263	-99.03	kd	CGS001-6208	RPS14	S ribosomal proteins			
8264	-99.03	oe	ccsbBroad304_06040	CRY1	-			
8265	-99.05	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
8266	-99.05	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
8267	-99.05	kd	CGS001-55746	NUP133	-			
8268	-99.05	kd	CGS001-39	ACAT2	Lanosterol biosynthesis pathway			
8269	-99.07	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
8270	-99.07	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
8271	-99.07	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
8272	-99.08	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
8273	-99.08	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
8274	-99.08	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
8275	-99.11	kd	CGS001-433	ASGR2	C-type lectin domain containing			
8276	-99.13	kd	CGS001-23566	LPAR3	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
8277	-99.13	kd	CGS001-2967	GTF2H3	General transcription factors			
8278	-99.13	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
8279	-99.15	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
8280	-99.16	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
8281	-99.16	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
8282	-99.17	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
8283	-99.17	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
8284	-99.17	oe	ccsbBroad304_06383	HMMR	CD molecules			
8285	-99.18	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
8286	-99.18	kd	CGS001-29915	HCFC2	-			
8287	-99.18	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
8288	-99.18	kd	CGS001-2167	FABP4	Fatty acid binding protein family			
8289	-99.19	cc		Heat shock 70kDa proteins LOF	-			
8290	-99.19	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
8291	-99.19	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
8292	-99.19	kd	CGS001-5033	P4HA1	-			
8293	-99.19	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
8294	-99.19	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
8295	-99.21	kd	CGS001-113451	ADC	-			
8296	-99.21	kd	CGS001-51741	WWOX	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
8297	-99.21	kd	CGS001-10342	TFG	-			
8298	-99.21	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
8299	-99.22	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
8300	-99.23	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
8301	-99.23	kd	CGS001-1975	EIF4B	RNA binding motif (RRM) containing			
8302	-99.24	kd	CGS001-11254	SLC6A14	Glycine transporter subfamily			
8303	-99.24	kd	CGS001-2524	FUT2	Fucosyltransferases			
8304	-99.25	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
8305	-99.25	kd	CGS001-8313	AXIN2	-			
8306	-99.26	oe	ccsbBroad304_03544	FAIM	-			
8307	-99.26	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
8308	-99.26	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
8309	-99.26	kd	CGS001-22818	COPZ1	-			
8310	-99.26	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
8311	-99.28	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
8312	-99.29	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
8313	-99.29	kd	CGS001-9341	VAMP3	Vesicle-associated membrane proteins			
8314	-99.3	kd	CGS001-4351	MPI	-			
8315	-99.31	oe	ccsbBroad304_03917	RBKS	-			
8316	-99.31	oe	ccsbBroad304_00238	CCNE1	-			
8317	-99.31	oe	ccsbBroad304_05894	BLVRA	-			
8318	-99.32	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
8319	-99.32	kd	CGS001-54915	YTHDF1	-			
8320	-99.32	kd	CGS001-6944	VPS72	-			
8321	-99.32	kd	CGS001-9770	RASSF2	-			
8322	-99.32	kd	CGS001-4998	ORC1	ATPases / AAA-type			
8323	-99.32	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
8324	-99.34	kd	CGS001-6201	RPS7	S ribosomal proteins			
8325	-99.34	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
8326	-99.35	kd	CGS001-10497	UNC13B	-			
8327	-99.35	kd	CGS001-7128	TNFAIP3	OTU domain containing			
8328	-99.37	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
8329	-99.37	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
8330	-99.37	kd	CGS001-6421	SFPQ	RNA binding motif (RRM) containing			
8331	-99.37	kd	CGS001-2067	ERCC1	-			
8332	-99.37	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
8333	-99.38	kd	CGS001-11180	WDR6	WD repeat domain containing			
8334	-99.38	kd	CGS001-10379	IRF9	-			
8335	-99.38	kd	CGS001-2152	F3	CD molecules			
8336	-99.38	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
8337	-99.39	cc		Akt Signaling LOF	-			
8338	-99.39	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
8339	-99.39	kd	CGS001-23466	CBX6	-			
8340	-99.4	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
8341	-99.4	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
8342	-99.4	kd	CGS001-7187	TRAF3	-			
8343	-99.4	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
8344	-99.4	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
8345	-99.41	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
8346	-99.42	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
8347	-99.42	kd	CGS001-205564	SENP5	-			
8348	-99.42	kd	CGS001-9275	BCL7B	-			
8349	-99.43	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
8350	-99.44	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
8351	-99.44	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
8352	-99.44	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
8353	-99.44	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
8354	-99.44	oe	ccsbBroad304_02370	HRSP12	-			
8355	-99.44	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
8356	-99.44	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
8357	-99.44	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
8358	-99.44	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
8359	-99.45	kd	CGS001-7103	TSPAN8	Tetraspanins			
8360	-99.45	kd	CGS001-5170	PDPK1	PDK1 family			
8361	-99.45	kd	CGS001-56998	CTNNBIP1	Catenins			
8362	-99.47	kd	CGS001-1487	CTBP1	-			
8363	-99.47	kd	CGS001-8717	TRADD	-			
8364	-99.47	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
8365	-99.47	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
8366	-99.48	kd	CGS001-5211	PFKL	-			
8367	-99.49	oe	ccsbBroad304_00120	ATOX1	-			
8368	-99.5	kd	CGS001-8503	PIK3R3	Phosphatidylinositol kinases			
8369	-99.5	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
8370	-99.5	kd	CGS001-4616	GADD45B	-			
8371	-99.51	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
8372	-99.51	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
8373	-99.51	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
8374	-99.51	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
8375	-99.51	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
8376	-99.51	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
8377	-99.53	kd	CGS001-2539	G6PD	-			
8378	-99.53	kd	CGS001-6223	RPS19	S ribosomal proteins			
8379	-99.53	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
8380	-99.54	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
8381	-99.54	kd	CGS001-26039	SS18L1	-			
8382	-99.54	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
8383	-99.54	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
8384	-99.55	kd	CGS001-51465	UBE2J1	Ubiquitin-conjugating enzymes E2			
8385	-99.55	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
8386	-99.55	kd	CGS001-10915	TCERG1	-			
8387	-99.55	kd	CGS001-6203	RPS9	S ribosomal proteins			
8388	-99.55	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
8389	-99.55	kd	CGS001-56675	NRIP3	-			
8390	-99.55	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
8391	-99.55	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
8392	-99.55	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
8393	-99.56	cc		Nucleoporin LOF	-			
8394	-99.56	kd	CGS001-2224	FDPS	Lanosterol biosynthesis pathway			
8395	-99.58	cc		Cyclins LOF	-			
8396	-99.58	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
8397	-99.58	kd	CGS001-5080	PAX6	Paired boxes			
8398	-99.58	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
8399	-99.58	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
8400	-99.58	kd	CGS001-9308	CD83	CD molecules			
8401	-99.58	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
8402	-99.58	kd	CGS001-383	ARG1	Arginase			
8403	-99.58	oe	ccsbBroad304_01658	PRDX2	-			
8404	-99.58	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
8405	-99.59	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
8406	-99.6	kd	CGS001-83999	KREMEN1	-			
8407	-99.61	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
8408	-99.61	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
8409	-99.61	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
8410	-99.61	kd	CGS001-6632	SNRPD1	-			
8411	-99.61	kd	CGS001-6210	RPS15A	S ribosomal proteins			
8412	-99.61	kd	CGS001-3978	LIG1	-			
8413	-99.61	kd	CGS001-57018	CCNL1	-			
8414	-99.63	kd	CGS001-6256	RXRA	Retinoid X receptors			
8415	-99.63	kd	CGS001-2021	ENDOG	-			
8416	-99.63	kd	CGS001-8727	CTNNAL1	Catenins			
8417	-99.63	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
8418	-99.63	oe	ccsbBroad304_00518	ETFA	-			
8419	-99.66	kd	CGS001-7280	TUBB2A	Tubulins			
8420	-99.66	kd	CGS001-80777	CYB5B	-			
8421	-99.66	kd	CGS001-7314	UBB	-			
8422	-99.66	kd	CGS001-7037	TFRC	CD molecules			
8423	-99.68	oe	ccsbBroad304_02840	PISD	Decarboxylases			
8424	-99.68	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
8425	-99.68	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
8426	-99.68	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
8427	-99.68	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
8428	-99.68	kd	CGS001-8089	YEATS4	-			
8429	-99.68	kd	CGS001-4089	SMAD4	SMADs			
8430	-99.68	kd	CGS001-7913	DEK	-			
8431	-99.68	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
8432	-99.68	oe	ccsbBroad304_01351	PEX19	-			
8433	-99.68	oe	ccsbBroad304_08392	EXOC6	-			
8434	-99.71	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
8435	-99.71	kd	CGS001-2181	ACSL3	Acyl-CoA synthetase family			
8436	-99.72	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
8437	-99.72	oe	ccsbBroad304_00490	EIF4EBP1	-			
8438	-99.72	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
8439	-99.72	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
8440	-99.73	cc		IL4 Pathway LOF	-			
8441	-99.74	kd	CGS001-8986	RPS6KA4	MSK subfamily			
8442	-99.74	kd	CGS001-6194	RPS6	S ribosomal proteins			
8443	-99.74	kd	CGS001-6217	RPS16	S ribosomal proteins			
8444	-99.74	kd	CGS001-55486	PARL	-			
8445	-99.75	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
8446	-99.75	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
8447	-99.75	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
8448	-99.75	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
8449	-99.75	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
8450	-99.75	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
8451	-99.76	kd	CGS001-7056	THBD	CD molecules			
8452	-99.76	kd	CGS001-6429	SRSF4	RNA binding motif (RRM) containing			
8453	-99.76	kd	CGS001-5763	PTMS	-			
8454	-99.77	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
8455	-99.77	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
8456	-99.77	oe	ccsbBroad304_02919	KIAA1279	-			
8457	-99.77	oe	ccsbBroad304_03119	C16ORF5	-			
8458	-99.77	oe	ccsbBroad304_07267	PDLIM4	-			
8459	-99.79	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
8460	-99.79	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
8461	-99.79	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
8462	-99.79	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
8463	-99.79	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
8464	-99.79	kd	CGS001-9871	SEC24D	-			
8465	-99.79	kd	CGS001-5777	PTPN6	Protein tyrosine phosphatases			
8466	-99.79	kd	CGS001-5255	PHKA1	-			
8467	-99.79	kd	CGS001-55765	C1ORF106	-			
8468	-99.79	oe	ccsbBroad304_02292	BCL2L11	-			
8469	-99.8	kd	CGS001-94239	H2AFV	Histones / Replication-independent			
8470	-99.81	kd	CGS001-51752	ERAP1	Aminopeptidase N			
8471	-99.81	oe	ccsbBroad304_02405	TFG	-			
8472	-99.81	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
8473	-99.82	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
8474	-99.82	cp	BRD-K13664374	dichloroacetic-acid	Pyruvate dehydrogenase kinase inhibitor		PDK1	Pyruvate dehydrogenase kinase inhibitor
8475	-99.82	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
8476	-99.82	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
8477	-99.82	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
8478	-99.82	kd	CGS001-143	PARP4	Poly (ADP-ribose) polymerases			
8479	-99.82	kd	CGS001-1062	CENPE	Kinesins			
8480	-99.82	kd	CGS001-406	ARNTL	Basic helix-loop-helix proteins			
8481	-99.83	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
8482	-99.84	cc		Ribosomal 40s Subunit LOF	-			
8483	-99.84	cc		PKA inhibitor	-			
8484	-99.84	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
8485	-99.84	kd	CGS001-6188	RPS3	S ribosomal proteins			
8486	-99.84	kd	CGS001-10775	POP4	-			
8487	-99.85	cc		Angiotensin receptor antagonist	-			
8488	-99.86	oe	ccsbBroad304_02271	LPGAT1	-			
8489	-99.86	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
8490	-99.86	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
8491	-99.86	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
8492	-99.86	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
8493	-99.86	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
8494	-99.86	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
8495	-99.86	oe	ccsbBroad304_04399	PGBD1	-			
8496	-99.86	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
8497	-99.87	kd	CGS001-219333	USP12	Ubiquitin-specific peptidases			
8498	-99.87	kd	CGS001-3832	KIF11	Kinesins			
8499	-99.87	kd	CGS001-6777	STAT5B	SH2 domain containing			
8500	-99.87	kd	CGS001-3588	IL10RB	IL-10 receptor family			
8501	-99.88	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
8502	-99.89	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
8503	-99.89	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
8504	-99.89	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
8505	-99.89	kd	CGS001-8644	AKR1C3	Prostaglandin synthases			
8506	-99.89	kd	CGS001-10383	TUBB2C	Tubulins			
8507	-99.89	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
8508	-99.89	kd	CGS001-5546	PRCC	-			
8509	-99.89	kd	CGS001-23325	KIAA1033	-			
8510	-99.89	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
8511	-99.89	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
8512	-99.89	kd	CGS001-80150	ASRGL1	-			
8513	-99.91	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
8514	-99.91	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
8515	-99.91	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
8516	-99.91	oe	ccsbBroad304_01234	POLB	DNA polymerases			
8517	-99.91	oe	ccsbBroad304_01222	PLP2	-			
8518	-99.91	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
8519	-99.91	oe	ccsbBroad304_08292	IP6K2	-			
8520	-99.91	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
8521	-99.91	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
8522	-99.92	kd	CGS001-6647	SOD1	-			
8523	-99.92	kd	CGS001-54811	ZNF562	Zinc fingers, C2H2-type			
8524	-99.92	kd	CGS001-7358	UGDH	-			
8525	-99.92	kd	CGS001-51284	TLR7	Toll-like receptor family			
8526	-99.92	kd	CGS001-63892	THADA	-			
8527	-99.92	kd	CGS001-5636	PRPSAP2	-			
8528	-99.92	kd	CGS001-55872	PBK	TOPK family			
8529	-99.92	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
8530	-99.92	kd	CGS001-474354	LRRC18	-			
8531	-99.92	kd	CGS001-3775	KCNK1	Two-P potassium channels			
8532	-99.92	kd	CGS001-3074	HEXB	-			
8533	-99.92	kd	CGS001-2313	FLI1	ETS Transcription Factors			
8534	-99.92	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
8535	-99.92	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
8536	-99.92	kd	CGS001-54555	DDX49	DEAD-boxes			
8537	-99.92	kd	CGS001-8702	B4GALT4	Beta 4-glycosyltransferases			
8538	-99.92	kd	CGS001-178	AGL	-			
8539	-99.93	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
8540	-99.93	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
8541	-99.93	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
8542	-99.93	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
8543	-99.93	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
8544	-99.93	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
8545	-99.95	kd	CGS001-9406	ZRANB2	Zinc fingers, RAN-binding domain containing			
8546	-99.95	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
8547	-99.95	kd	CGS001-27347	STK39	FRAY subfamily			
8548	-99.95	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
8549	-99.95	kd	CGS001-284119	PTRF	-			
8550	-99.95	kd	CGS001-10113	PREB	WD repeat domain containing			
8551	-99.95	kd	CGS001-5480	PPIC	-			
8552	-99.95	kd	CGS001-4916	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
8553	-99.95	kd	CGS001-1728	NQO1	-			
8554	-99.95	kd	CGS001-10797	MTHFD2	-			
8555	-99.95	kd	CGS001-55876	GSDMB	-			
8556	-99.95	kd	CGS001-7832	BTG2	-			
8557	-99.95	kd	CGS001-95	ACY1	-			
8558	-99.97	cc		Thromboxane receptor antagonist	-			
8559	-99.99	cc		Ubiquitin-specific peptidases LOF	-			
