Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
2	100	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
3	100	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
4	99.99	cc		Mitogen activated protein kinases LOF	-			
5	99.99	oe	ccsbBroad304_00219	CARS	Aminoacyl tRNA synthetases / Class I			
6	99.97	cp	BRD-K75295174	alisertib	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
7	99.97	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
8	99.97	oe	ccsbBroad304_01880	LAGE3	-			
9	99.97	oe	ccsbBroad304_01054	GADD45B	-			
10	99.97	oe	ccsbBroad304_02843	FTSJ1	-			
11	99.97	oe	ccsbBroad304_03604	ENOSF1	-			
12	99.97	oe	ccsbBroad304_00464	DTNA	-			
13	99.97	oe	ccsbBroad304_03372	CAB39	-			
14	99.97	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
15	99.97	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
16	99.97	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
17	99.97	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
18	99.97	oe	ccsbBroad304_12106	PXK	Slob family			
19	99.97	oe	ccsbBroad304_01271	PPT1	-			
20	99.97	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
21	99.97	oe	ccsbBroad304_01074	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
22	99.97	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
23	99.97	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
24	99.97	oe	ccsbBroad304_00809	HUS1	-			
25	99.97	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
26	99.97	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
27	99.97	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
28	99.97	oe	ccsbBroad304_00644	GCLC	-			
29	99.97	oe	ccsbBroad304_00570	FIGF	-			
30	99.97	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
31	99.97	oe	ccsbBroad304_05833	APEH	Prolyl oligopeptidase			
32	99.97	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
33	99.97	oe	ccsbBroad304_00036	AFP	-			
34	99.97	oe	ccsbBroad304_00033	ADSS	-			
35	99.97	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
36	99.97	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
37	99.97	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
38	99.97	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
39	99.97	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
40	99.97	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
41	99.97	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
42	99.97	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
43	99.97	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
44	99.97	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
45	99.97	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
46	99.97	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
47	99.97	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
48	99.97	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
49	99.97	kd	CGS001-10221	TRIB1	Trbl family			
50	99.97	kd	CGS001-10474	TADA3	-			
51	99.97	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
52	99.97	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
53	99.97	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
54	99.97	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
55	99.97	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
56	99.97	kd	CGS001-2770	GNAI1	-			
57	99.97	kd	CGS001-1786	DNMT1	Methyltransferases			
58	99.97	kd	CGS001-79947	DHDDS	-			
59	99.97	kd	CGS001-1606	DGKA	EF-hand domain containing			
60	99.97	kd	CGS001-11129	CLASRP	-			
61	99.97	kd	CGS001-84433	CARD11	-			
62	99.96	oe	ccsbBroad304_01651	TCF7L2	-			
63	99.96	oe	ccsbBroad304_04619	GNG8	-			
64	99.96	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
65	99.96	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
66	99.96	oe	ccsbBroad304_03853	LSM2	-			
67	99.96	oe	ccsbBroad304_03268	GMPR2	-			
68	99.96	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
69	99.96	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
70	99.96	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
71	99.96	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
72	99.96	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
73	99.96	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
74	99.96	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
75	99.96	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
76	99.96	kd	CGS001-4171	MCM2	-			
77	99.96	kd	CGS001-3098	HK1	-			
78	99.96	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
79	99.96	kd	CGS001-2771	GNAI2	-			
80	99.96	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
81	99.96	kd	CGS001-717	C2	Complement system			
82	99.95	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
83	99.94	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
84	99.94	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
85	99.94	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
86	99.94	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
87	99.94	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
88	99.94	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
89	99.94	oe	ccsbBroad304_00170	BNIP1	-			
90	99.94	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
91	99.94	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
92	99.94	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
93	99.94	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
94	99.94	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
95	99.94	kd	CGS001-51002	TPRKB	-			
96	99.94	kd	CGS001-29110	TBK1	IKK family			
97	99.94	kd	CGS001-4781	NFIB	-			
98	99.94	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
99	99.94	kd	CGS001-9787	DLGAP5	-			
100	99.94	kd	CGS001-1374	CPT1A	-			
101	99.94	oe	ccsbBroad304_00745	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
102	99.94	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
103	99.93	oe	ccsbBroad304_07704	SUB1	-			
104	99.93	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
105	99.93	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
106	99.93	oe	ccsbBroad304_00615	GAPDH	-			
107	99.93	oe	ccsbBroad304_01930	CUL2	-			
108	99.93	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
109	99.93	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
110	99.93	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
111	99.93	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
112	99.93	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
113	99.93	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
114	99.93	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
115	99.93	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
116	99.91	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
117	99.91	oe	ccsbBroad304_01163	PDHA1	-			
118	99.91	oe	ccsbBroad304_13850	EIF4A2	DEAD-boxes			
119	99.91	oe	ccsbBroad304_00221	CASP3	Caspases			
120	99.91	oe	ccsbBroad304_00116	ASS1	-			
121	99.91	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
122	99.91	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
123	99.91	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
124	99.91	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
125	99.91	kd	CGS001-89882	TPD52L3	-			
126	99.91	kd	CGS001-10465	PPIH	-			
127	99.91	kd	CGS001-391013	PLA2G2C	-			
128	99.91	kd	CGS001-80018	NAA25	N(alpha)-acetyltransferase subunits			
129	99.91	kd	CGS001-10289	EIF1B	-			
130	99.91	kd	CGS001-1329	COX5B	Mitochondrial respiratory chain complex			
131	99.91	kd	CGS001-328	APEX1	-			
132	99.9	cp	BRD-K67174588	toremifene	Estrogen receptor antagonist		ESR1, CYP3A5	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
133	99.9	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
134	99.9	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
135	99.9	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
136	99.9	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
137	99.9	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
138	99.9	kd	CGS001-8884	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
139	99.9	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
140	99.9	kd	CGS001-55179	FAIM	-			
141	99.9	kd	CGS001-10423	CDIPT	-			
142	99.89	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
143	99.88	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
144	99.88	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
145	99.88	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
146	99.88	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
147	99.88	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
148	99.88	kd	CGS001-2538	G6PC	-			
149	99.87	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
150	99.87	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
151	99.87	oe	ccsbBroad304_01247	POU2AF1	-			
152	99.87	oe	ccsbBroad304_06539	LSS	Lanosterol biosynthesis pathway			
153	99.87	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
154	99.87	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
155	99.87	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
156	99.87	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
157	99.87	kd	CGS001-389421	LIN28B	-			
158	99.86	oe	ccsbBroad304_03309	RNF138	RING-type (C3HC4) zinc fingers			
159	99.86	oe	ccsbBroad304_00370	CS	-			
160	99.85	oe	ccsbBroad304_02231	USP6NL	-			
161	99.85	oe	ccsbBroad304_10231	SETDB1	Histone methyltransferases (HMTs)			
162	99.85	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
163	99.85	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
164	99.85	kd	CGS001-9404	LPXN	-			
165	99.85	kd	CGS001-7919	DDX39B	DEAD-boxes			
166	99.84	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
167	99.84	oe	ccsbBroad304_02443	HAX1	-			
168	99.84	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
169	99.84	kd	CGS001-6732	SRPK1	SRPK family			
170	99.84	kd	CGS001-3169	FOXA1	Forkhead boxes			
171	99.83	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
172	99.82	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
173	99.82	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
174	99.82	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
175	99.82	kd	CGS001-1195	CLK1	CDC-like kinases			
176	99.81	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
177	99.81	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
178	99.81	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
179	99.81	kd	CGS001-10670	RRAGA	-			
180	99.79	oe	ccsbBroad304_08346	COQ3	-			
181	99.79	oe	ccsbBroad304_00277	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
182	99.79	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
183	99.79	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
184	99.78	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
185	99.78	kd	CGS001-5992	RFX4	-			
186	99.78	kd	CGS001-3980	LIG3	-			
187	99.78	kd	CGS001-79581	GPR172A	-			
188	99.76	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
189	99.76	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
190	99.76	kd	CGS001-4016	LOXL1	-			
191	99.76	kd	CGS001-64077	LHPP	-			
192	99.76	kd	CGS001-27241	BBS9	-			
193	99.75	kd	CGS001-8720	MBTPS1	Subtilisin			
194	99.74	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
195	99.73	cp	BRD-K39569857	avrainvillamide-analog-3	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
196	99.73	oe	ccsbBroad304_01872	DGCR14	-			
197	99.73	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
198	99.73	kd	CGS001-8089	YEATS4	-			
199	99.73	kd	CGS001-116443	GRIN3A	Glutamate receptors			
200	99.73	oe	ccsbBroad304_02030	CFLAR	Endogenous ligands			
201	99.72	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
202	99.72	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
203	99.72	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
204	99.72	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
205	99.72	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
206	99.72	kd	CGS001-1949	EFNB3	Ephrins			
207	99.72	kd	CGS001-367	AR	Nuclear hormone receptors			
208	99.71	oe	ccsbBroad304_06282	GLDC	-			
209	99.71	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
210	99.71	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
211	99.71	kd	CGS001-4522	MTHFD1	-			
212	99.7	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
213	99.69	cp	BRD-K24576554	AT-9283	JAK inhibitor		AURKA, AURKB, ABL1, BCR, FLT3, JAK2, JAK3, RPS6KA6, STK17A	JAK inhibitor, Aurora kinase inhibitor, ABL inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, Mitotic inhibitor, Protein kinase inhibitor
214	99.69	oe	ccsbBroad304_01395	RFX5	-			
215	99.69	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
216	99.69	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
217	99.69	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
218	99.69	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
219	99.67	cp	BRD-K52313696	tacedinaline	HDAC inhibitor		HDAC1	HDAC inhibitor
220	99.66	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
221	99.66	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
222	99.66	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
223	99.66	kd	CGS001-9833	MELK	MELK subfamily			
224	99.66	kd	CGS001-5927	KDM5A	Histone demethylases			
225	99.65	oe	ccsbBroad304_00709	GUK1	-			
226	99.65	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
227	99.65	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
228	99.65	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
229	99.65	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
230	99.65	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
231	99.65	kd	CGS001-4605	MYBL2	-			
232	99.63	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
233	99.63	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
234	99.63	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
235	99.63	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
236	99.63	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
237	99.63	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
238	99.63	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
239	99.63	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
240	99.63	kd	CGS001-8895	CPNE3	-			
241	99.62	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
242	99.62	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
243	99.62	oe	ccsbBroad304_06382	HMGCL	-			
244	99.62	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
245	99.62	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
246	99.6	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
247	99.6	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
248	99.6	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
249	99.6	kd	CGS001-701	BUB1B	Bub family			
250	99.59	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
251	99.59	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
252	99.57	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
253	99.57	oe	ccsbBroad304_04153	PHF17	-			
254	99.57	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
255	99.57	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
256	99.57	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
257	99.57	kd	CGS001-7097	TLR2	Toll-like receptor family			
258	99.57	kd	CGS001-9709	HERPUD1	-			
259	99.56	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
260	99.55	oe	ccsbBroad304_00650	GNA11	-			
261	99.54	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
262	99.54	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
263	99.53	oe	ccsbBroad304_02058	PLOD3	-			
264	99.53	oe	ccsbBroad304_01208	PITPNA	-			
265	99.5	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
266	99.49	kd	CGS001-22954	TRIM32	-			
267	99.48	oe	ccsbBroad304_01143	PAFAH1B3	-			
268	99.48	oe	ccsbBroad304_14242	MCCC2	-			
269	99.48	kd	CGS001-10146	G3BP1	RNA binding motif (RRM) containing			
270	99.47	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
271	99.47	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
272	99.47	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
273	99.45	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
274	99.44	oe	ccsbBroad304_03097	CNOT7	-			
275	99.43	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
276	99.43	oe	ccsbBroad304_00423	DAXX	-			
277	99.43	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
278	99.42	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
279	99.42	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
280	99.4	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
281	99.4	oe	ccsbBroad304_06654	NPM1	-			
282	99.4	kd	CGS001-8805	TRIM24	TIF1 family			
283	99.39	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
284	99.38	oe	ccsbBroad304_06665	OAT	-			
285	99.38	oe	ccsbBroad304_01073	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
286	99.38	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
287	99.38	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
288	99.37	kd	CGS001-51599	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
289	99.37	kd	CGS001-2247	FGF2	Endogenous ligands			
290	99.36	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
291	99.35	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
292	99.35	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
293	99.35	kd	CGS001-2731	GLDC	-			
294	99.34	oe	ccsbBroad304_00515	ERH	-			
295	99.34	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
296	99.34	kd	CGS001-3326	HSP90AB1	Heat shock proteins / HSPC			
297	99.33	oe	ccsbBroad304_06458	IRF3	-			
298	99.32	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
299	99.32	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
300	99.32	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
301	99.32	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
302	99.32	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
303	99.31	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
304	99.31	kd	CGS001-3032	HADHB	-			
305	99.3	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
306	99.29	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
307	99.29	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
308	99.29	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
309	99.28	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
310	99.28	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
311	99.27	kd	CGS001-5428	POLG	DNA polymerases			
312	99.25	oe	ccsbBroad304_00164	BLMH	-			
313	99.22	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
314	99.22	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
315	99.22	kd	CGS001-523	ATP6V1A	ATPases / V-type			
316	99.21	oe	ccsbBroad304_01066	NDUFA4	-			
317	99.21	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
318	99.21	kd	CGS001-5164	PDK2	PDHK family			
319	99.18	kd	CGS001-4077	NBR1	-			
320	99.17	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
321	99.15	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
322	99.15	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
323	99.15	oe	ccsbBroad304_02551	CPSF4	-			
324	99.15	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
325	99.15	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
326	99.15	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
327	99.13	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
328	99.13	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
329	99.13	oe	ccsbBroad304_13903	MTAP	-			
330	99.12	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
331	99.1	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
332	99.1	kd	CGS001-2882	GPX7	-			
333	99.09	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
334	99.08	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
335	99.07	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
336	99.05	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
337	99.02	oe	ccsbBroad304_12008	NLK	nmo subfamily			
338	99.02	kd	CGS001-2752	GLUL	-			
339	99.01	kd	CGS001-8349	HIST2H2BE	Histones / Replication-dependent			
340	99	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
341	99	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
342	98.99	oe	ccsbBroad304_00359	CPT1A	-			
343	98.98	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
344	98.98	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
345	98.97	kd	CGS001-2353	FOS	basic leucine zipper proteins			
346	98.95	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
347	98.93	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
348	98.92	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
349	98.91	kd	CGS001-1509	CTSD	Cathepsins			
350	98.88	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
351	98.87	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
352	98.86	oe	ccsbBroad304_03555	PANK4	-			
353	98.86	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
354	98.86	kd	CGS001-7423	VEGFB	-			
355	98.85	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
356	98.85	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
357	98.85	kd	CGS001-5163	PDK1	-			
358	98.85	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
359	98.84	cc		Thymidylate synthase inhibitor	-			
360	98.84	kd	CGS001-89910	UBE3B	-			
361	98.84	kd	CGS001-4086	SMAD1	SMADs			
362	98.84	kd	CGS001-9638	FEZ1	-			
363	98.82	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
364	98.82	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
365	98.82	kd	CGS001-4193	MDM2	-			
366	98.81	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
367	98.81	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
368	98.79	oe	ccsbBroad304_02287	GNPDA1	-			
369	98.78	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
370	98.78	kd	CGS001-8864	PER2	-			
371	98.76	oe	ccsbBroad304_01618	STXBP1	-			
372	98.75	oe	ccsbBroad304_00818	IDH3A	-			
373	98.73	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
374	98.73	kd	CGS001-10111	RAD50	-			
375	98.72	oe	ccsbBroad304_14047	TACC3	-			
376	98.72	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
377	98.7	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
378	98.7	oe	ccsbBroad304_06150	EIF4E	Translation Initiation Factor 4E			
379	98.7	oe	ccsbBroad304_02297	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
380	98.7	kd	CGS001-54442	KCTD5	-			
381	98.7	kd	CGS001-2242	FES	Fer family			
382	98.69	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
383	98.68	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
384	98.67	oe	ccsbBroad304_00746	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
385	98.66	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
386	98.66	oe	ccsbBroad304_07890	CBX7	-			
387	98.63	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
388	98.63	kd	CGS001-587	BCAT2	-			
389	98.62	oe	ccsbBroad304_06294	GNAZ	-			
390	98.62	oe	ccsbBroad304_01835	CXCR4	Chemokine receptors			
391	98.62	oe	ccsbBroad304_00020	ACY1	-			
392	98.58	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
393	98.58	kd	CGS001-150094	SIK1	QIK subfamily			
394	98.56	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
395	98.56	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
396	98.54	kd	CGS001-665	BNIP3L	-			
397	98.53	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
398	98.52	kd	CGS001-60528	ELAC2	-			
399	98.51	cc		LIM class homeoboxes GOF	-			
400	98.5	oe	ccsbBroad304_01408	RNF5	RING-type (C3HC4) zinc fingers			
401	98.48	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
402	98.48	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
403	98.48	kd	CGS001-3690	ITGB3	Integrins			
404	98.47	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
405	98.46	oe	ccsbBroad304_00658	GNG5	-			
406	98.46	kd	CGS001-79006	METRN	-			
407	98.45	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
408	98.45	kd	CGS001-6204	RPS10	S ribosomal proteins			
409	98.44	kd	CGS001-4282	MIF	-			
410	98.42	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
411	98.42	kd	CGS001-1376	CPT2	-			
412	98.41	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
413	98.41	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
414	98.41	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
415	98.41	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
416	98.36	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
417	98.36	kd	CGS001-481	ATP1B1	ATPases / P-type			
418	98.34	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
419	98.33	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
420	98.32	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
421	98.31	kd	CGS001-9474	ATG5	-			
422	98.29	kd	CGS001-340371	NRBP2	NRBP family			
423	98.27	kd	CGS001-25942	SIN3A	-			
424	98.25	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
425	98.23	kd	CGS001-1746	DLX2	Homeoboxes / ANTP class : NKL subclass			
426	98.23	kd	CGS001-80347	COASY	-			
427	98.22	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
428	98.22	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
429	98.2	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
430	98.2	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
431	98.18	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
432	98.17	oe	ccsbBroad304_06894	RPS6	S ribosomal proteins			
433	98.17	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
434	98.17	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
435	98.17	kd	CGS001-4610	MYCL1	-			
436	98.16	kd	CGS001-2212	FCGR2A	CD molecules			
437	98.15	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
438	98.15	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
439	98.14	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
440	98.14	kd	CGS001-2159	F10	Chymotrypsin			
441	98.1	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
442	98.1	kd	CGS001-5966	REL	NFkappaB transcription factor family			
443	98.09	kd	CGS001-10325	RRAGB	-			
444	98.08	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
445	98.07	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
446	98.06	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
447	98.04	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
448	98.02	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
449	98.02	kd	CGS001-8576	STK16	NAK family			
450	98.02	kd	CGS001-399664	MEX3D	Mex-3 homologs			
451	98.02	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
452	98.01	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
453	98	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
454	97.99	kd	CGS001-9231	DLG5	-			
455	97.98	oe	ccsbBroad304_07875	SPECC1L	-			
456	97.98	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
457	97.98	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
458	97.98	kd	CGS001-253430	IPMK	-			
459	97.98	kd	CGS001-10672	GNA13	-			
460	97.95	kd	CGS001-5446	PON3	Paraoxonases			
461	97.93	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
462	97.92	oe	ccsbBroad304_01787	YES1	Src family			
463	97.92	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
464	97.91	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
465	97.91	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
466	97.91	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
467	97.9	kd	CGS001-2057	EPOR	Prolactin receptor family			
468	97.89	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
469	97.89	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
470	97.88	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
471	97.83	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
472	97.82	kd	CGS001-10973	ASCC3	-			
473	97.8	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
474	97.8	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
475	97.79	oe	ccsbBroad304_00424	DBI	-			
476	97.78	kd	CGS001-1659	DHX8	DEAH-boxes			
477	97.77	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
478	97.76	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
479	97.75	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
480	97.74	oe	ccsbBroad304_05985	CFL1	-			
481	97.74	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
482	97.74	kd	CGS001-54899	PXK	Slob family			
483	97.73	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
484	97.72	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
485	97.72	kd	CGS001-36	ACADSB	-			
486	97.7	oe	ccsbBroad304_00060	AMBP	Lipocalins			
487	97.69	kd	CGS001-25793	FBXO7	F-boxes / other			
488	97.68	oe	ccsbBroad304_03357	RASD1	-			
489	97.66	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
490	97.66	kd	CGS001-1951	CELSR3	Cadherins / Major cadherins			
491	97.62	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
492	97.61	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
493	97.61	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
494	97.6	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
495	97.58	oe	ccsbBroad304_08104	MED4	-			
496	97.56	oe	ccsbBroad304_03405	CHRAC1	-			
497	97.56	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
498	97.56	kd	CGS001-2639	GCDH	-			
499	97.56	kd	CGS001-1763	DNA2	-			
500	97.55	oe	ccsbBroad304_08386	SMOX	-			
501	97.55	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
502	97.51	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
503	97.5	oe	ccsbBroad304_06424	IFI16	-			
504	97.49	cc		BMP Signaling LOF	-			
505	97.48	kd	CGS001-9801	MRPL19	Mitochondrial ribosomal proteins / large subunits			
506	97.45	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
507	97.44	oe	ccsbBroad304_01203	PIM1	PIM family			
508	97.43	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
509	97.42	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
510	97.41	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
511	97.41	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
512	97.37	oe	ccsbBroad304_02045	BUD31	-			
513	97.37	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
514	97.36	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
515	97.34	oe	ccsbBroad304_05547	TMEM110	-			
516	97.34	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
517	97.33	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
518	97.3	oe	ccsbBroad304_02869	ASF1A	-			
519	97.28	oe	ccsbBroad304_02875	BRP44	-			
520	97.26	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
521	97.23	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
522	97.21	oe	ccsbBroad304_07569	TRIB1	Trbl family			
523	97.2	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
524	97.19	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
525	97.19	kd	CGS001-5653	KLK6	Chymotrypsin			
526	97.18	kd	CGS001-10928	RALBP1	-			
527	97.18	kd	CGS001-4700	NDUFA6	LYR motif containing			
528	97.17	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
529	97.16	kd	CGS001-900	CCNG1	-			
530	97.13	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
531	97.13	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
532	97.12	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
533	97.11	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
534	97.09	oe	ccsbBroad304_03080	C16ORF80	-			
535	97.08	kd	CGS001-6727	SRP14	-			
536	97.07	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
537	97.07	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
538	97.05	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
539	96.95	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
540	96.95	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
541	96.94	oe	ccsbBroad304_00964	SMAD7	SMADs			
542	96.91	oe	ccsbBroad304_06155	ELF1	ETS Transcription Factors			
543	96.9	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
544	96.89	oe	ccsbBroad304_02133	CD83	CD molecules			
545	96.88	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
546	96.86	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
547	96.85	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
548	96.83	kd	CGS001-597	BCL2A1	-			
549	96.81	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
550	96.81	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
551	96.8	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
552	96.79	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
553	96.76	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
554	96.74	kd	CGS001-2475	MTOR	FRAP subfamily			
555	96.71	oe	ccsbBroad304_02578	EBNA1BP2	-			
556	96.69	oe	ccsbBroad304_00079	APOA1	Apolipoproteins			
557	96.66	kd	CGS001-230	ALDOC	-			
558	96.64	oe	ccsbBroad304_00969	MAGEA10	-			
559	96.63	oe	ccsbBroad304_06235	G6PD	-			
560	96.62	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
561	96.61	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
562	96.61	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
563	96.57	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
564	96.57	kd	CGS001-1495	CTNNA1	Catenins			
565	96.55	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
566	96.54	kd	CGS001-1314	COPA	Endogenous ligands			
567	96.53	oe	ccsbBroad304_00865	ILF2	-			
568	96.51	cc		HIV protease inhibitor	-			
569	96.49	kd	CGS001-50813	COPS7A	-			
570	96.48	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
571	96.48	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
572	96.48	kd	CGS001-2037	EPB41L2	-			
573	96.45	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
574	96.44	oe	ccsbBroad304_07140	XPC	-			
575	96.43	kd	CGS001-6513	SLC2A1	Solute carriers			
576	96.42	oe	ccsbBroad304_08553	STAP2	-			
577	96.41	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
578	96.39	oe	ccsbBroad304_03652	EXOC2	-			
579	96.36	oe	ccsbBroad304_07851	FAM120A	-			
580	96.36	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
581	96.36	oe	ccsbBroad304_08045	NOX1	-			
582	96.35	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
583	96.34	oe	ccsbBroad304_06975	SMARCC2	-			
584	96.33	oe	ccsbBroad304_00120	ATOX1	-			
585	96.31	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
586	96.29	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
587	96.28	kd	CGS001-9943	OXSR1	FRAY subfamily			
588	96.26	kd	CGS001-4299	AFF1	-			
589	96.22	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
590	96.22	kd	CGS001-3927	LASP1	-			
591	96.22	kd	CGS001-1512	CTSH	Cathepsins			
592	96.21	kd	CGS001-1962	EHHADH	-			
593	96.2	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
594	96.2	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
595	96.13	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
596	96.1	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
597	96.06	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
598	96.05	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
599	96.03	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
600	96.02	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
601	96.01	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
602	96.01	kd	CGS001-57804	POLD4	DNA polymerases			
603	96.01	kd	CGS001-10096	ACTR3	-			
604	95.98	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
605	95.98	kd	CGS001-2550	GABBR1	GABA receptors			
606	95.95	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
607	95.9	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
608	95.9	kd	CGS001-32	ACACB	Carboxylases			
609	95.85	kd	CGS001-29105	C16ORF80	-			
610	95.83	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
611	95.83	kd	CGS001-2079	ERH	-			
612	95.82	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
613	95.79	kd	CGS001-6714	SRC	Src family			
614	95.78	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
615	95.77	kd	CGS001-10434	LYPLA1	-			
616	95.75	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
617	95.72	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
618	95.7	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
619	95.7	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
620	95.69	kd	CGS001-9817	KEAP1	Kelch-like proteins			
621	95.63	kd	CGS001-3925	STMN1	-			
622	95.63	kd	CGS001-5105	PCK1	-			
623	95.62	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
624	95.62	kd	CGS001-10447	FAM3C	-			
625	95.61	kd	CGS001-7525	YES1	Src family			
626	95.57	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
627	95.57	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
628	95.57	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
629	95.56	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
630	95.54	kd	CGS001-57787	MARK4	MARK subfamily			
631	95.53	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
632	95.51	kd	CGS001-25913	POT1	-			
633	95.5	oe	ccsbBroad304_03113	DSE	-			
634	95.5	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
635	95.49	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
636	95.48	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
637	95.46	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
638	95.44	oe	ccsbBroad304_00231	CBFB	-			
639	95.42	oe	ccsbBroad304_04387	MKI67IP	-			
640	95.4	kd	CGS001-200734	SPRED2	-			
641	95.4	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
642	95.39	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
643	95.36	oe	ccsbBroad304_06755	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
644	95.36	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
645	95.32	oe	ccsbBroad304_07267	PDLIM4	-			
646	95.31	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
647	95.3	kd	CGS001-25819	CCRN4L	-			
648	95.29	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
649	95.27	oe	ccsbBroad304_01613	STK11	LKB subfamily			
650	95.26	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
651	95.21	kd	CGS001-56654	NPDC1	-			
652	95.2	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
653	95.2	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
654	95.2	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
655	95.17	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
656	95.17	kd	CGS001-694	BTG1	-			
657	95.14	oe	ccsbBroad304_00759	HMOX2	Haem oxygenase			
658	95.11	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
659	95.11	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
660	95.1	oe	ccsbBroad304_02220	MTFR1	-			
661	95.08	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
662	95.07	kd	CGS001-29984	RHOD	-			
663	95.01	kd	CGS001-5906	RAP1A	-			
664	94.94	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
665	94.92	cc		Sigma receptor antagonist	-			
666	94.92	oe	ccsbBroad304_07557	NAMPT	-			
667	94.92	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
668	94.9	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
669	94.86	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
670	94.86	kd	CGS001-55802	DCP1A	-			
671	94.85	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
672	94.82	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
673	94.81	kd	CGS001-5091	PC	Carboxylases			
674	94.79	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
675	94.79	kd	CGS001-10390	CEPT1	-			
676	94.78	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
677	94.76	kd	CGS001-1211	CLTA	-			
678	94.74	kd	CGS001-169841	ZNF169	Zinc fingers, C2H2-type			
679	94.7	kd	CGS001-2152	F3	CD molecules			
680	94.68	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
681	94.62	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
682	94.61	cp	BRD-A70731303	avrainvillamide-analog-5	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
683	94.58	kd	CGS001-26277	TINF2	-			
684	94.58	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
685	94.57	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
686	94.57	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
687	94.54	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
688	94.51	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
689	94.5	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
690	94.5	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
691	94.47	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
692	94.38	oe	ccsbBroad304_03237	LEF1	-			
693	94.37	kd	CGS001-5682	PSMA1	Proteasome subunits			
694	94.36	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
695	94.34	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
696	94.32	oe	ccsbBroad304_00150	BAX	-			
697	94.32	oe	ccsbBroad304_00097	ARF6	ADP-ribosylation factors			
698	94.32	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
699	94.25	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
700	94.24	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
701	94.23	kd	CGS001-51292	GMPR2	-			
702	94.23	kd	CGS001-1465	CSRP1	-			
703	94.21	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
704	94.2	kd	CGS001-6050	RNH1	-			
705	94.19	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
706	94.19	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
707	94.12	cc		Leucine rich repeat kinase inhibitor	-			
708	94.09	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
709	94.07	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
710	94.02	oe	ccsbBroad304_02845	PRPF6	-			
711	93.95	cc		Na-K-Cl transporter inhibitor	-			
712	93.86	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
713	93.84	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
714	93.82	kd	CGS001-3251	HPRT1	-			
715	93.81	kd	CGS001-7353	UFD1L	-			
716	93.81	kd	CGS001-8050	PDHX	-			
717	93.8	kd	CGS001-5018	OXA1L	-			
718	93.79	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
719	93.75	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
720	93.72	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
721	93.71	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
722	93.71	kd	CGS001-255738	PCSK9	Subtilisin			
723	93.7	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
724	93.7	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
725	93.69	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
726	93.69	kd	CGS001-5144	PDE4D	Phosphodiesterases			
727	93.69	kd	CGS001-9807	IP6K1	-			
728	93.64	kd	CGS001-4255	MGMT	-			
729	93.61	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
730	93.6	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
731	93.57	kd	CGS001-51268	PIPOX	-			
732	93.54	oe	ccsbBroad304_14174	CDKAL1	-			
733	93.51	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
734	93.51	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
735	93.5	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
736	93.47	kd	CGS001-10057	ABCC5	ATP binding cassette transporters / subfamily C			
737	93.46	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
738	93.43	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
739	93.37	kd	CGS001-84617	TUBB6	Tubulins			
740	93.3	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
741	93.3	kd	CGS001-23212	RRS1	-			
742	93.23	oe	ccsbBroad304_09195	MCM8	-			
743	93.23	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
744	93.21	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
745	93.19	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
746	93.13	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
747	93.09	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
748	93.07	kd	CGS001-11156	PTP4A3	Protein tyrosine phosphatases			
749	93.03	kd	CGS001-23161	SNX13	Sorting nexins			
750	93	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
751	92.88	kd	CGS001-2523	FUT1	Fucosyltransferases			
752	92.86	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
753	92.85	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
754	92.85	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
755	92.83	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
756	92.82	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
757	92.75	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
758	92.75	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
759	92.7	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
760	92.7	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
761	92.67	cc		Homeobox Gene GOF	-			
762	92.61	kd	CGS001-1198	CLK3	CDC-like kinases			
763	92.59	oe	ccsbBroad304_04522	ZNF625	Zinc fingers, C2H2-type			
764	92.57	oe	ccsbBroad304_00459	DPYD	-			
765	92.56	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
766	92.56	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
767	92.55	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
768	92.54	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
769	92.53	oe	ccsbBroad304_01445	RPS3	S ribosomal proteins			
770	92.53	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
771	92.5	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
772	92.48	oe	ccsbBroad304_00833	IFNG	Interferons			
773	92.47	kd	CGS001-5743	PTGS2	Cyclooxygenase			
774	92.47	kd	CGS001-308	ANXA5	Annexins			
775	92.45	kd	CGS001-10190	TXNDC9	-			
776	92.41	oe	ccsbBroad304_08536	PARL	-			
777	92.4	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
778	92.39	kd	CGS001-629	CFB	Complement system			
779	92.38	kd	CGS001-53340	SPA17	-			
780	92.36	kd	CGS001-8220	DGCR14	-			
781	92.33	oe	ccsbBroad304_01101	NME1	-			
782	92.32	oe	ccsbBroad304_03506	AURKAIP1	-			
783	92.28	kd	CGS001-10084	PQBP1	-			
784	92.26	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
785	92.24	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
786	92.23	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
787	92.22	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
788	92.15	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
789	92.14	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
790	92.1	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
791	92.08	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
792	92.01	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
793	92	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
794	92	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
795	91.92	kd	CGS001-51564	HDAC7	Histone deacetylases			
796	91.88	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
797	91.86	oe	ccsbBroad304_12226	NAGK	-			
798	91.86	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
799	91.84	oe	ccsbBroad304_06420	ICAM3	CD molecules			
800	91.79	oe	ccsbBroad304_08266	PIPOX	-			
801	91.76	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
802	91.73	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
803	91.73	kd	CGS001-9374	PPT2	-			
804	91.7	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
805	91.7	kd	CGS001-5092	PCBD1	-			
806	91.68	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
807	91.67	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
808	91.66	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
809	91.64	oe	ccsbBroad304_02922	TES	-			
810	91.62	kd	CGS001-29937	NENF	-			
811	91.57	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
812	91.56	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
813	91.54	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
814	91.53	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
815	91.51	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
816	91.51	kd	CGS001-4801	NFYB	-			
817	91.46	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
818	91.44	kd	CGS001-2078	ERG	ETS Transcription Factors			
819	91.43	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
820	91.41	oe	ccsbBroad304_01186	PHB	-			
821	91.4	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
822	91.3	kd	CGS001-9967	THRAP3	-			
823	91.28	kd	CGS001-2768	GNA12	-			
824	91.28	kd	CGS001-23142	DCUN1D4	-			
825	91.25	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
826	91.22	oe	ccsbBroad304_07029	TADA2A	-			
827	91.22	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
828	91.22	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
829	91.21	kd	CGS001-30	ACAA1	-			
830	91.15	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
831	91.13	oe	ccsbBroad304_02633	LSM6	-			
832	91.12	kd	CGS001-5579	PRKCB	Alpha subfamily			
833	91.1	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
834	91.06	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
835	91.02	kd	CGS001-813	CALU	EF-hand domain containing			
836	90.9	oe	ccsbBroad304_01282	PRKCB	Alpha subfamily			
837	90.9	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
838	90.85	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
839	90.82	cc		Adenosine receptor agonist	-			
840	90.82	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
841	90.78	oe	ccsbBroad304_13939	MOK	RCK family			
842	90.75	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
843	90.73	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
844	90.71	kd	CGS001-6509	SLC1A4	Alanine/serine/cysteine transporter subfamily			
845	90.68	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
846	90.65	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
847	90.59	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
848	90.56	oe	ccsbBroad304_06291	GNAI1	-			
849	90.56	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
850	90.55	kd	CGS001-7405	UVRAG	-			
851	90.54	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
852	90.53	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
853	90.52	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
854	90.51	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
855	90.46	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
856	90.45	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
857	90.44	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
858	90.42	kd	CGS001-55837	EAPP	-			
859	90.41	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
860	90.33	oe	ccsbBroad304_01371	RALA	-			
861	90.32	oe	ccsbBroad304_00549	FDX1	-			
862	90.29	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
863	90.26	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
864	90.23	oe	ccsbBroad304_10427	DHX8	DEAH-boxes			
865	90.19	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
866	90.17	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
867	90.15	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
868	90.09	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
869	90.08	kd	CGS001-64943	NT5DC2	-			
870	90.08	kd	CGS001-2244	FGB	Endogenous ligands			
871	89.97	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
872	89.92	kd	CGS001-8771	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
873	89.88	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
874	89.86	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
875	89.8	oe	ccsbBroad304_08605	PBK	TOPK family			
876	89.75	kd	CGS001-8848	TSC22D1	-			
877	89.73	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
878	89.72	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
879	89.7	kd	CGS001-7849	PAX8	Paired boxes			
880	89.69	oe	ccsbBroad304_06287	GM2A	-			
881	89.66	kd	CGS001-2098	ESD	-			
882	89.65	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
883	89.61	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
884	89.55	oe	ccsbBroad304_06089	DDIT3	-			
885	89.54	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
886	89.47	oe	ccsbBroad304_03072	GTPBP8	-			
887	89.44	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
888	89.43	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
889	89.41	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
890	89.41	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
891	89.34	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
892	89.28	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
893	89.27	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
894	89.21	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
895	89.18	oe	ccsbBroad304_05821	ANXA1	Annexins			
896	89.13	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
897	89.1	oe	ccsbBroad304_00496	ELF4	ETS Transcription Factors			
898	89.06	oe	ccsbBroad304_01008	KITLG	-			
899	89.03	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
900	88.99	kd	CGS001-3630	INS	-			
901	88.96	kd	CGS001-57680	CHD8	-			
902	88.92	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
903	88.88	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
904	88.87	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
905	88.86	oe	ccsbBroad304_03148	IL21R	IL-2 receptor family			
906	88.85	kd	CGS001-9966	TNFSF15	Tumor necrosis factor (ligand) superfamily			
907	88.85	kd	CGS001-8829	NRP1	CD molecules			
908	88.83	kd	CGS001-7248	TSC1	-			
909	88.78	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
910	88.78	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
911	88.74	oe	ccsbBroad304_01812	ZNF175	Zinc fingers, C2H2-type			
912	88.66	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
913	88.64	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
914	88.47	kd	CGS001-23536	ADAT1	-			
915	88.44	oe	ccsbBroad304_07920	NUP62	-			
916	88.43	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
917	88.41	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
918	88.4	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
919	88.36	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
920	88.34	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
921	88.33	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
922	88.33	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
923	88.31	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
924	88.28	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
925	88.28	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
926	88.23	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
927	88.23	kd	CGS001-1727	CYB5R3	-			
928	88.22	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
929	88.22	kd	CGS001-51070	NOSIP	-			
930	88.18	cc		Beta-adrenergic receptor agonist	-			
931	88.17	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
932	88.15	oe	ccsbBroad304_06569	MCM5	-			
933	88.15	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
934	88.04	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
935	88.04	oe	ccsbBroad304_07798	EXOC3	-			
936	88.03	kd	CGS001-63948	DMRTB1	-			
937	88.02	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
938	87.96	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
939	87.96	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
940	87.91	cc		C2 domain containing LOF	-			
941	87.91	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
942	87.89	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
943	87.89	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
944	87.83	kd	CGS001-182	JAG1	CD molecules			
945	87.8	oe	ccsbBroad304_02115	PTTG1	-			
946	87.8	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
947	87.77	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
948	87.75	oe	ccsbBroad304_10024	ZNF680	Zinc fingers, C2H2-type			
949	87.75	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
950	87.74	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
951	87.66	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
952	87.64	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
953	87.61	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
954	87.59	oe	ccsbBroad304_06645	NQO2	-			
955	87.58	oe	ccsbBroad304_07280	LAMTOR3	-			
956	87.47	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
957	87.46	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
958	87.43	oe	ccsbBroad304_00210	CALR	-			
959	87.38	cc		ATP synthase inhibitor	-			
960	87.35	oe	ccsbBroad304_06855	RDX	-			
961	87.35	oe	ccsbBroad304_00524	EXT2	Exostosin glycosyltransferase family			
962	87.34	oe	ccsbBroad304_02496	MTX2	-			
963	87.34	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
964	87.32	oe	ccsbBroad304_01699	TPD52L2	-			
965	87.28	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
966	87.26	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
967	87.25	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
968	87.25	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
969	87.24	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
970	87.23	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
971	87.2	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
972	87.19	oe	ccsbBroad304_00738	HINT1	-			
973	87.15	kd	CGS001-10476	ATP5H	ATPases / F-type			
974	87.11	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
975	87.09	kd	CGS001-965	CD58	CD molecules			
976	87.07	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
977	87.07	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
978	87.06	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
979	87.06	kd	CGS001-9120	SLC16A6	SLC16 family of monocarboxylate transporters			
980	87.01	oe	ccsbBroad304_06720	PHYH	-			
981	86.97	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
982	86.93	kd	CGS001-9170	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
983	86.91	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
984	86.91	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
985	86.87	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
986	86.85	kd	CGS001-2931	GSK3A	GSK subfamily			
987	86.8	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
988	86.78	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
989	86.76	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
990	86.73	oe	ccsbBroad304_05756	ACAA1	-			
991	86.72	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
992	86.69	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
993	86.67	oe	ccsbBroad304_01841	BAG6	-			
994	86.63	oe	ccsbBroad304_00933	LDHB	-			
995	86.62	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
996	86.59	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
997	86.58	oe	ccsbBroad304_02741	PDS5A	-			
998	86.58	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
999	86.57	kd	CGS001-2113	ETS1	ETS Transcription Factors			
1000	86.52	kd	CGS001-23585	TMEM50A	-			
1001	86.46	oe	ccsbBroad304_07018	SUPT5H	-			
1002	86.45	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1003	86.43	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
1004	86.42	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
1005	86.4	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1006	86.34	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
1007	86.34	oe	ccsbBroad304_02683	COG2	Components of oligomeric golgi complex			
1008	86.29	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
1009	86.29	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
1010	86.26	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
1011	86.24	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
1012	86.23	kd	CGS001-5037	PEBP1	-			
1013	86.22	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
1014	86.21	kd	CGS001-111	ADCY5	Adenylate cyclases			
1015	86.17	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
1016	86.17	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
1017	86.16	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
1018	86.12	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
1019	86.11	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
1020	86.1	oe	ccsbBroad304_03934	LEPRE1	-			
1021	86.08	oe	ccsbBroad304_01279	PRKAG1	AMPK subfamily			
1022	86.08	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
1023	86.04	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1024	85.99	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
1025	85.94	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
1026	85.94	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
1027	85.93	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
1028	85.9	oe	ccsbBroad304_09225	BUD13	-			
1029	85.81	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
1030	85.78	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
1031	85.74	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
1032	85.73	oe	ccsbBroad304_00049	ALDH2	Aldehyde dehydrogenases			
1033	85.71	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
1034	85.7	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
1035	85.65	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1036	85.64	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1037	85.62	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
1038	85.62	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
1039	85.62	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
1040	85.61	kd	CGS001-23223	RRP12	-			
1041	85.52	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1042	85.46	kd	CGS001-5236	PGM1	-			
1043	85.41	oe	ccsbBroad304_00471	E2F6	-			
1044	85.4	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
1045	85.4	kd	CGS001-1892	ECHS1	-			
1046	85.38	kd	CGS001-58472	SQRDL	-			
1047	85.34	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1048	85.3	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
1049	85.27	kd	CGS001-53343	NUDT9	Nudix motif containing			
1050	85.2	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
1051	85.16	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
1052	85.14	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
1053	85.02	kd	CGS001-6884	TAF13	-			
1054	84.99	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
1055	84.99	kd	CGS001-55810	FOXJ2	Forkhead boxes			
1056	84.97	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
1057	84.94	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
1058	84.86	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
1059	84.8	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
1060	84.72	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
1061	84.7	kd	CGS001-10452	TOMM40	-			
1062	84.68	kd	CGS001-3034	HAL	-			
1063	84.66	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
1064	84.63	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
1065	84.6	oe	ccsbBroad304_00276	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
1066	84.59	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
1067	84.58	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
1068	84.51	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
1069	84.48	oe	ccsbBroad304_01114	NUP88	-			
1070	84.45	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
1071	84.43	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
1072	84.38	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
1073	84.35	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
1074	84.32	oe	ccsbBroad304_08325	LIPT1	-			
1075	84.31	kd	CGS001-4312	MMP1	Matrix metallopeptidase			
1076	84.3	oe	ccsbBroad304_09358	MAPK1IP1L	-			
1077	84.28	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
1078	84.21	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
1079	84.18	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1080	84.13	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
1081	84.09	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
1082	84.06	cc		Tumor necrosis factor superfamily LOF	-			
1083	84.05	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
1084	84.01	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
1085	83.95	oe	ccsbBroad304_01131	OXCT1	-			
1086	83.95	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
1087	83.94	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
1088	83.92	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
1089	83.86	kd	CGS001-6647	SOD1	-			
1090	83.8	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
1091	83.8	oe	ccsbBroad304_06998	SRPK1	SRPK family			
1092	83.77	kd	CGS001-10493	VAT1	-			
1093	83.76	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
1094	83.72	kd	CGS001-51001	MTERFD1	-			
1095	83.71	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1096	83.7	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
1097	83.64	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
1098	83.63	kd	CGS001-3978	LIG1	-			
1099	83.63	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
1100	83.61	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
1101	83.6	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
1102	83.57	oe	ccsbBroad304_02306	PQBP1	-			
1103	83.52	kd	CGS001-11325	DDX42	DEAD-boxes			
1104	83.31	oe	ccsbBroad304_00052	ALDH3A2	Aldehyde dehydrogenases			
1105	83.28	oe	ccsbBroad304_07515	GFPT2	-			
1106	83.2	oe	ccsbBroad304_00795	HSF2	-			
1107	83.15	oe	ccsbBroad304_06255	LRRC32	-			
1108	83.11	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
1109	83.09	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
1110	83.09	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
1111	83.08	oe	ccsbBroad304_02396	TCIRG1	ATPases / V-type			
1112	83.06	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
1113	83.05	kd	CGS001-91433	RCCD1	-			
1114	83	kd	CGS001-64863	METTL4	-			
1115	82.96	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
1116	82.9	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
1117	82.85	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
1118	82.84	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1119	82.82	kd	CGS001-51271	UBAP1	-			
1120	82.78	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
1121	82.74	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
1122	82.72	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
1123	82.68	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1124	82.59	kd	CGS001-4190	MDH1	-			
1125	82.54	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
1126	82.52	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
1127	82.51	kd	CGS001-10691	GMEB1	-			
1128	82.44	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
1129	82.44	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1130	82.43	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
1131	82.43	kd	CGS001-11151	CORO1A	Coronins			
1132	82.42	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
1133	82.33	oe	ccsbBroad304_02052	KYNU	-			
1134	82.33	kd	CGS001-4734	NEDD4	-			
1135	82.3	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
1136	82.27	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
1137	82.25	oe	ccsbBroad304_06191	FABP6	Fatty acid binding protein family			
1138	82.25	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
1139	82.23	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
1140	82.19	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
1141	82.18	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
1142	82.18	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
1143	82.15	cc		Protein phosphatase catalytic subunits LOF	-			
1144	82.15	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
1145	82.14	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
1146	82.06	kd	CGS001-55604	LRRC16A	-			
1147	82	cc		PI3K Signaling LOF	-			
1148	81.93	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
1149	81.91	kd	CGS001-5590	PRKCZ	Iota subfamily			
1150	81.86	kd	CGS001-8639	AOC3	Oxidoreductases			
1151	81.83	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
1152	81.76	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
1153	81.76	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
1154	81.74	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
1155	81.74	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
1156	81.74	kd	CGS001-306	ANXA3	Annexins			
1157	81.67	kd	CGS001-79109	MAPKAP1	-			
1158	81.65	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
1159	81.49	kd	CGS001-54915	YTHDF1	-			
1160	81.47	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
1161	81.45	oe	ccsbBroad304_03266	ERGIC2	-			
1162	81.32	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
1163	81.27	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
1164	81.27	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
1165	81.27	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
1166	81.24	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
1167	81.24	kd	CGS001-2896	GRN	-			
1168	81.23	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1169	81.22	oe	ccsbBroad304_02011	TNFRSF6B	Tumour necrosis factor (TNF) receptor family			
1170	81.22	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
1171	81.21	cc		VEGFR inhibitor	-			
1172	81.2	oe	ccsbBroad304_00986	MCM2	-			
1173	81.19	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
1174	81.16	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
1175	81.15	oe	ccsbBroad304_01845	RDBP	-			
1176	81.06	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
1177	81.03	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
1178	81.02	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1179	81.01	oe	ccsbBroad304_07768	NISCH	-			
1180	81.01	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
1181	80.96	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
1182	80.93	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
1183	80.88	oe	ccsbBroad304_02566	MORF4L1	-			
1184	80.87	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
1185	80.81	oe	ccsbBroad304_07548	TSSC4	-			
1186	80.79	oe	ccsbBroad304_04064	PRR15L	-			
1187	80.76	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
1188	80.76	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
1189	80.73	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1190	80.72	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
1191	80.7	kd	CGS001-3689	ITGB2	Integrins			
1192	80.68	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
1193	80.65	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
1194	80.65	oe	ccsbBroad304_05948	CCND2	-			
1195	80.6	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
1196	80.6	kd	CGS001-51071	DERA	-			
1197	80.54	kd	CGS001-3995	FADS3	Fatty acid desaturases			
1198	80.53	oe	ccsbBroad304_08775	SQRDL	-			
1199	80.53	kd	CGS001-116511	MAS1L	GPCR / Class A : Orphans			
1200	80.5	oe	ccsbBroad304_13891	LCK	Src family			
1201	80.49	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
1202	80.47	kd	CGS001-8535	CBX4	-			
1203	80.44	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
1204	80.37	oe	ccsbBroad304_07097	TRAF1	-			
1205	80.35	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
1206	80.35	kd	CGS001-3035	HARS	Aminoacyl tRNA synthetases / Class II			
1207	80.34	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
1208	80.29	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
1209	80.26	kd	CGS001-8835	SOCS2	SH2 domain containing			
1210	80.22	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
1211	80.22	kd	CGS001-6757	SSX2	-			
1212	80.2	oe	ccsbBroad304_00514	ERF	ETS Transcription Factors			
1213	80.19	kd	CGS001-4668	NAGA	-			
1214	80.12	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
1215	80.02	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
1216	80.02	oe	ccsbBroad304_03591	ETNK1	-			
1217	79.98	kd	CGS001-7311	UBA52	L ribosomal proteins			
1218	79.9	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
1219	79.86	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
1220	79.79	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
1221	79.75	cc		Serine proteases GOF	-			
1222	79.71	kd	CGS001-9415	FADS2	Fatty acid desaturases			
1223	79.7	kd	CGS001-56521	DNAJC12	Heat shock proteins / DNAJ (HSP40)			
1224	79.67	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
1225	79.62	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
1226	79.56	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
1227	79.55	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
1228	79.51	kd	CGS001-10671	DCTN6	-			
1229	79.48	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
1230	79.42	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
1231	79.4	kd	CGS001-7078	TIMP3	-			
1232	79.4	kd	CGS001-10400	PEMT	-			
1233	79.36	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
1234	79.3	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1235	79.27	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
1236	79.22	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
1237	79.19	oe	ccsbBroad304_01485	SC5DL	-			
1238	79.19	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
1239	79.15	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
1240	79.06	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
1241	79.05	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
1242	78.89	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
1243	78.83	kd	CGS001-1196	CLK2	CDC-like kinases			
1244	78.82	kd	CGS001-5373	PMM2	-			
1245	78.81	kd	CGS001-253260	RICTOR	-			
1246	78.8	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
1247	78.62	oe	ccsbBroad304_06021	KLF6	Kruppel-like transcription factors			
1248	78.57	oe	ccsbBroad304_01661	TFCP2	-			
1249	78.57	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
1250	78.56	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
1251	78.56	kd	CGS001-9128	PRPF4	WD repeat domain containing			
1252	78.55	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1253	78.54	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
1254	78.5	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
1255	78.42	kd	CGS001-661	POLR3D	RNA polymerase subunits			
1256	78.39	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
1257	78.39	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
1258	78.38	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
1259	78.38	kd	CGS001-9870	KIAA0317	-			
1260	78.37	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
1261	78.33	oe	ccsbBroad304_01152	PCNA	-			
1262	78.26	oe	ccsbBroad304_04752	IKBIP	-			
1263	78.14	oe	ccsbBroad304_00003	ABAT	GABA turnover			
1264	78.13	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
1265	78.13	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
1266	78.11	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
1267	78.09	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
1268	78.05	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
1269	78.03	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
1270	78.01	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
1271	77.99	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
1272	77.99	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
1273	77.96	kd	CGS001-2115	ETV1	ETS Transcription Factors			
1274	77.96	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
1275	77.94	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
1276	77.89	kd	CGS001-55893	ZNF395	Zinc fingers, C2H2-type			
1277	77.88	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
1278	77.8	kd	CGS001-5518	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
1279	77.78	oe	ccsbBroad304_05758	ACADSB	-			
1280	77.76	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
1281	77.74	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
1282	77.74	oe	ccsbBroad304_00001	NAT1	-			
1283	77.74	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
1284	77.73	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
1285	77.56	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
1286	77.52	oe	ccsbBroad304_00130	ATP5F1	ATPases / F-type			
1287	77.44	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
1288	77.39	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
1289	77.35	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
1290	77.34	oe	ccsbBroad304_13598	NRBP2	NRBP family			
1291	77.33	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
1292	77.25	oe	ccsbBroad304_08116	TBK1	IKK family			
1293	77.22	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
1294	77.21	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
1295	77.16	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
1296	77.15	oe	ccsbBroad304_06090	DDOST	-			
1297	77.08	oe	ccsbBroad304_06670	OGG1	-			
1298	77.06	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
1299	77.04	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
1300	77.04	kd	CGS001-5223	PGAM1	-			
1301	77.03	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
1302	77.03	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
1303	77.01	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
1304	76.99	kd	CGS001-150280	HORMAD2	-			
1305	76.96	cc		Zinc fingers RanBP2 type LOF	-			
1306	76.92	oe	ccsbBroad304_00490	EIF4EBP1	-			
1307	76.92	oe	ccsbBroad304_00469	DUT	-			
1308	76.88	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
1309	76.84	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
1310	76.83	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
1311	76.79	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
1312	76.67	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
1313	76.66	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
1314	76.66	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
1315	76.64	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
1316	76.61	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
1317	76.61	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
1318	76.61	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
1319	76.61	kd	CGS001-64223	MLST8	WD repeat domain containing			
1320	76.58	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
1321	76.58	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
1322	76.52	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
1323	76.51	cc		C2 domain containing protein kinases LOF	-			
1324	76.46	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1325	76.45	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
1326	76.44	kd	CGS001-801	CALM1	EF-hand domain containing			
1327	76.4	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
1328	76.3	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
1329	76.22	cc		Ubiquitin-specific peptidases LOF	-			
1330	76.21	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
1331	76.14	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
1332	76.12	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
1333	76.02	oe	ccsbBroad304_07017	SUOX	-			
1334	76	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
1335	75.99	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
1336	75.93	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
1337	75.92	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
1338	75.89	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
1339	75.86	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
1340	75.85	kd	CGS001-151306	GPBAR1	Bile acid receptor			
1341	75.73	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
1342	75.69	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
1343	75.68	kd	CGS001-7029	TFDP2	-			
1344	75.67	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
1345	75.67	kd	CGS001-8896	BUD31	-			
1346	75.67	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
1347	75.63	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
1348	75.58	kd	CGS001-5645	PRSS2	Serine peptidases			
1349	75.56	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
1350	75.5	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
1351	75.49	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
1352	75.45	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
1353	75.45	oe	ccsbBroad304_04675	ATG4A	-			
1354	75.32	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
1355	75.31	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
1356	75.3	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
1357	75.23	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
1358	75.21	oe	ccsbBroad304_00268	CD81	CD molecules			
1359	75.17	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1360	75.16	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
1361	75.16	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
1362	75.14	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
1363	75.08	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
1364	75.06	kd	CGS001-1605	DAG1	-			
1365	75	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1366	74.97	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
1367	74.91	kd	CGS001-7001	PRDX2	-			
1368	74.9	kd	CGS001-6520	SLC3A2	SLC3 family			
1369	74.86	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
1370	74.72	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
1371	74.69	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
1372	74.62	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
1373	74.52	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
1374	74.52	kd	CGS001-55437	STRADB	STLK subfamily			
1375	74.51	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
1376	74.43	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
1377	74.4	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1378	74.37	oe	ccsbBroad304_02485	STAMBP	-			
1379	74.36	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
1380	74.2	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
1381	74.19	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
1382	74.18	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
1383	74.16	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
1384	74.05	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
1385	74.03	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
1386	73.94	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
1387	73.87	oe	ccsbBroad304_00006	ACADM	-			
1388	73.81	oe	ccsbBroad304_01735	UBE2D1	Ubiquitin-conjugating enzymes E2			
1389	73.79	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
1390	73.78	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
1391	73.73	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
1392	73.71	oe	ccsbBroad304_00155	CCND1	-			
1393	73.68	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
1394	73.54	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
1395	73.54	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
1396	73.53	oe	ccsbBroad304_04891	TMEM174	-			
1397	73.52	oe	ccsbBroad304_06518	LDHA	-			
1398	73.49	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
1399	73.49	kd	CGS001-818	CAMK2G	CAMK2 family			
1400	73.38	oe	ccsbBroad304_02500	RRAGA	-			
1401	73.38	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
1402	73.38	kd	CGS001-7728	ZNF175	Zinc fingers, C2H2-type			
1403	73.38	kd	CGS001-5982	RFC2	ATPases / AAA-type			
1404	73.26	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
1405	73.25	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1406	73.25	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
1407	73.23	oe	ccsbBroad304_10116	SHC4	SH2 domain containing			
1408	73.11	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
1409	73.09	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
1410	73.06	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
1411	73.04	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
1412	72.97	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
1413	72.91	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
1414	72.91	kd	CGS001-7771	ZFP112	-			
1415	72.83	kd	CGS001-8431	NR0B2	DAX-like receptors			
1416	72.78	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
1417	72.75	kd	CGS001-10475	TRIM38	-			
1418	72.65	kd	CGS001-51128	SAR1B	-			
1419	72.63	oe	ccsbBroad304_02438	FAM3C	-			
1420	72.61	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
1421	72.58	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
1422	72.48	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
1423	72.45	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
1424	72.37	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1425	72.35	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
1426	72.34	cc		BCL inhibitor	-			
1427	72.32	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
1428	72.2	cc		IL4 Pathway LOF	-			
1429	72.16	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
1430	72.09	oe	ccsbBroad304_00491	EIF4EBP2	-			
1431	72.07	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1432	72.03	oe	ccsbBroad304_02501	DCTN6	-			
1433	72.02	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
1434	72.01	oe	ccsbBroad304_06852	RBP4	Lipocalins			
1435	71.98	kd	CGS001-7360	UGP2	-			
1436	71.93	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
1437	71.93	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
1438	71.89	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
1439	71.88	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
1440	71.85	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
1441	71.71	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
1442	71.66	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
1443	71.66	oe	ccsbBroad304_02026	NRP1	CD molecules			
1444	71.66	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
1445	71.61	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
1446	71.61	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
1447	71.6	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
1448	71.58	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
1449	71.54	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
1450	71.53	kd	CGS001-185	AGTR1	Angiotensin receptors			
1451	71.48	kd	CGS001-133690	CAPSL	EF-hand domain containing			
1452	71.45	kd	CGS001-11284	PNKP	-			
1453	71.44	cc		Interleukin receptors LOF	-			
1454	71.44	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
1455	71.43	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
1456	71.42	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
1457	71.31	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
1458	71.3	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
1459	71.25	oe	ccsbBroad304_02432	IFI30	-			
1460	71.23	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
1461	71.2	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
1462	71.17	oe	ccsbBroad304_00957	M6PR	-			
1463	71.16	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
1464	71.15	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
1465	71.13	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1466	71.08	kd	CGS001-3590	IL11RA	IL-6 receptor family			
1467	71.06	oe	ccsbBroad304_06745	PNN	-			
1468	71.05	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
1469	71.04	oe	ccsbBroad304_00072	ANXA7	Annexins			
1470	70.98	kd	CGS001-835	CASP2	Caspases			
1471	70.97	kd	CGS001-4947	OAZ2	-			
1472	70.94	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
1473	70.89	oe	ccsbBroad304_01164	PDHB	-			
1474	70.87	oe	ccsbBroad304_00836	IGF2	-			
1475	70.76	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
1476	70.7	oe	ccsbBroad304_03173	TMED7	-			
1477	70.66	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
1478	70.62	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1479	70.6	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
1480	70.59	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
1481	70.51	kd	CGS001-7292	TNFSF4	CD molecules			
1482	70.47	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
1483	70.45	cc		Akt Signaling GOF	-			
1484	70.45	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
1485	70.42	oe	ccsbBroad304_07766	RASSF1	-			
1486	70.37	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
1487	70.36	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
1488	70.26	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
1489	70.25	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
1490	70.23	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
1491	70.21	kd	CGS001-896	CCND3	-			
1492	70.2	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
1493	70.19	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
1494	70.19	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
1495	70.16	oe	ccsbBroad304_03767	TOMM22	-			
1496	70.12	kd	CGS001-56647	BCCIP	-			
1497	70.1	oe	ccsbBroad304_01139	PA2G4	-			
1498	70.09	kd	CGS001-5898	RALA	-			
1499	69.92	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
1500	69.79	kd	CGS001-1488	CTBP2	-			
1501	69.78	kd	CGS001-51097	SCCPDH	-			
1502	69.7	oe	ccsbBroad304_02560	RNPS1	RNA binding motif (RRM) containing			
1503	69.64	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
1504	69.63	oe	ccsbBroad304_05098	MAGEB6	-			
1505	69.6	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
1506	69.59	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
1507	69.56	oe	ccsbBroad304_00122	ATP1B1	ATPases / P-type			
1508	69.56	kd	CGS001-23463	ICMT	-			
1509	69.54	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
1510	69.51	oe	ccsbBroad304_01013	MIF	-			
1511	69.48	cc		Estrogen receptor agonist	-			
1512	69.48	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
1513	69.35	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
1514	69.34	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
1515	69.31	oe	ccsbBroad304_02572	SERINC3	-			
1516	69.31	kd	CGS001-2184	FAH	-			
1517	69.24	kd	CGS001-901	CCNG2	-			
1518	69.18	oe	ccsbBroad304_06718	PFN2	-			
1519	69.15	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
1520	69.14	kd	CGS001-4696	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
1521	69.12	kd	CGS001-7416	VDAC1	Voltage-dependent anion channels			
1522	69.09	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
1523	69.07	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
1524	69.05	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1525	68.94	kd	CGS001-10007	GNPDA1	-			
1526	68.93	kd	CGS001-6285	S100B	EF-hand domain containing			
1527	68.8	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
1528	68.77	oe	ccsbBroad304_00392	CTLA4	CD molecules			
1529	68.73	kd	CGS001-79600	TCTN1	Tectonic proteins			
1530	68.72	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
1531	68.71	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
1532	68.69	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
1533	68.62	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
1534	68.6	oe	ccsbBroad304_04976	SERPINA12	Serine (or cysteine) peptidase inhibitors			
1535	68.51	kd	CGS001-435	ASL	-			
1536	68.5	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
1537	68.33	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
1538	68.32	oe	ccsbBroad304_05194	LIPH	-			
1539	68.27	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
1540	68.26	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
1541	68.26	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
1542	68.26	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
1543	68.01	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1544	67.96	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
1545	67.95	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
1546	67.93	cc		X linked mental retardation group 2 LOF	-			
1547	67.75	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
1548	67.7	kd	CGS001-29103	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
1549	67.68	oe	ccsbBroad304_03129	ERO1L	-			
1550	67.64	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
1551	67.53	kd	CGS001-9670	IPO13	Importins			
1552	67.52	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
1553	67.5	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
1554	67.47	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
1555	67.46	kd	CGS001-9531	BAG3	-			
1556	67.28	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
1557	67.23	oe	ccsbBroad304_07616	ZNF238	-			
1558	67.23	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
1559	67.18	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
1560	67.16	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
1561	67.15	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
1562	67.14	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
1563	67.12	oe	ccsbBroad304_08093	DCPS	-			
1564	67.03	oe	ccsbBroad304_08925	ZNF576	Zinc fingers, C2H2-type			
1565	66.98	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
1566	66.98	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
1567	66.96	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1568	66.94	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
1569	66.92	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
1570	66.91	oe	ccsbBroad304_01374	RAP1A	-			
1571	66.9	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1572	66.9	kd	CGS001-161725	OTUD7A	OTU domain containing			
1573	66.89	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
1574	66.87	kd	CGS001-23678	SGK3	SGK family			
1575	66.81	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
1576	66.73	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
1577	66.68	kd	CGS001-64240	ABCG5	ATP binding cassette transporters / subfamily G			
1578	66.62	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
1579	66.6	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
1580	66.6	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
1581	66.56	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
1582	66.54	oe	ccsbBroad304_02834	GABARAPL1	-			
1583	66.54	kd	CGS001-348	APOE	Apolipoproteins			
1584	66.53	oe	ccsbBroad304_06159	CTTN	-			
1585	66.53	oe	ccsbBroad304_00418	CD55	CD molecules			
1586	66.52	kd	CGS001-6603	SMARCD2	-			
1587	66.46	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
1588	66.38	oe	ccsbBroad304_04396	ZNF559	Zinc fingers, C2H2-type			
1589	66.35	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
1590	66.27	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
1591	66.27	kd	CGS001-29940	DSE	-			
1592	66.19	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
1593	66.18	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
1594	66.15	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
1595	66.15	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
1596	66.14	oe	ccsbBroad304_00995	MECP2	-			
1597	65.94	oe	ccsbBroad304_02357	SSX3	-			
1598	65.87	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
1599	65.85	oe	ccsbBroad304_08481	CEP55	-			
1600	65.76	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1601	65.76	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
1602	65.75	kd	CGS001-1382	CRABP2	Fatty acid-binding proteins			
1603	65.69	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
1604	65.66	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
1605	65.66	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
1606	65.62	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
1607	65.62	kd	CGS001-10398	MYL9	EF-hand domain containing			
1608	65.6	oe	ccsbBroad304_01413	RPA2	-			
1609	65.49	kd	CGS001-64422	ATG3	-			
1610	65.46	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
1611	65.45	oe	ccsbBroad304_10230	STK19	G11 family			
1612	65.42	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
1613	65.41	kd	CGS001-3566	IL4R	IL-2 receptor family			
1614	65.35	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
1615	65.32	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
1616	65.3	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
1617	65.26	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
1618	65.24	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
1619	65.24	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1620	65.23	kd	CGS001-1120	CHKB	-			
1621	65.19	oe	ccsbBroad304_00819	IDH3B	-			
1622	65.14	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
1623	65.05	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
1624	65.05	kd	CGS001-9500	MAGED1	-			
1625	64.99	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
1626	64.99	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
1627	64.94	kd	CGS001-10329	TMEM5	-			
1628	64.81	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
1629	64.8	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
1630	64.77	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
1631	64.72	oe	ccsbBroad304_02956	EHF	-			
1632	64.71	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
1633	64.66	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
1634	64.65	kd	CGS001-873	CBR1	Prostaglandin synthases			
1635	64.63	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1636	64.61	cc		Retinoid receptor agonist	-			
1637	64.61	kd	CGS001-7157	TP53	-			
1638	64.58	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
1639	64.44	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
1640	64.39	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
1641	64.33	kd	CGS001-9847	KIAA0528	-			
1642	64.29	kd	CGS001-6282	S100A11	EF-hand domain containing			
1643	64.28	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
1644	64.28	oe	ccsbBroad304_04399	PGBD1	-			
1645	64.27	oe	ccsbBroad304_07094	TPMT	-			
1646	64.27	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
1647	64.24	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
1648	64.19	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
1649	64.19	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
1650	64.18	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1651	64.16	oe	ccsbBroad304_01002	METTL1	-			
1652	64.14	cc		FXR antagonist	-			
1653	64.14	cp	BRD-K66766661	17-beta-estradiol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1654	64.1	kd	CGS001-56675	NRIP3	-			
1655	64.1	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
1656	64.04	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
1657	64.02	oe	ccsbBroad304_00349	COX4I1	Mitochondrial respiratory chain complex			
1658	64.01	oe	ccsbBroad304_00783	HPRT1	-			
1659	63.98	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
1660	63.97	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
1661	63.97	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
1662	63.85	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
1663	63.84	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
1664	63.8	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
1665	63.73	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
1666	63.58	kd	CGS001-9697	TRAM2	-			
1667	63.5	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
1668	63.5	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
1669	63.46	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
1670	63.43	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
1671	63.41	cc		Bacterial DNA gyrase inhibitor	-			
1672	63.41	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
1673	63.41	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1674	63.4	oe	ccsbBroad304_07834	GGA2	-			
1675	63.39	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
1676	63.24	oe	ccsbBroad304_00661	GNGT2	-			
1677	63.23	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
1678	63.2	cc		HRH1 antagonist	-			
1679	63.18	oe	ccsbBroad304_08662	MCCC1	-			
1680	63.16	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
1681	63.14	kd	CGS001-3682	ITGAE	Integrins			
1682	63.13	kd	CGS001-6511	SLC1A6	Glutamate transporter subfamily			
1683	63.06	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
1684	63.03	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
1685	62.98	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
1686	62.93	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
1687	62.9	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
1688	62.87	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
1689	62.78	kd	CGS001-3664	IRF6	-			
1690	62.75	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
1691	62.74	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
1692	62.73	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
1693	62.72	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
1694	62.7	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
1695	62.66	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
1696	62.64	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
1697	62.6	oe	ccsbBroad304_07808	RAB11FIP2	-			
1698	62.6	kd	CGS001-4088	SMAD3	SMADs			
1699	62.58	kd	CGS001-3418	IDH2	-			
1700	62.56	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
1701	62.42	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
1702	62.41	oe	ccsbBroad304_00739	ZBTB48	BTB/POZ domain containing			
1703	62.32	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
1704	62.25	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
1705	62.24	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
1706	62.22	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
1707	62.16	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
1708	62.11	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
1709	62.03	kd	CGS001-54108	CHRAC1	-			
1710	61.98	oe	ccsbBroad304_07561	YAF2	-			
1711	61.98	kd	CGS001-4303	FOXO4	Forkhead boxes			
1712	61.98	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
1713	61.96	oe	ccsbBroad304_02270	FAM20B	-			
1714	61.95	oe	ccsbBroad304_00941	LIG3	-			
1715	61.94	kd	CGS001-29763	PACSIN3	-			
1716	61.91	kd	CGS001-6598	SMARCB1	-			
1717	61.91	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
1718	61.89	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
1719	61.86	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
1720	61.78	kd	CGS001-57147	SCYL3	-			
1721	61.74	kd	CGS001-57222	ERGIC1	-			
1722	61.72	kd	CGS001-9124	PDLIM1	-			
1723	61.71	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
1724	61.68	kd	CGS001-23530	NNT	-			
1725	61.65	kd	CGS001-10018	BCL2L11	-			
1726	61.52	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
1727	61.51	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
1728	61.48	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
1729	61.47	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
1730	61.43	kd	CGS001-11007	CCDC85B	-			
1731	61.37	kd	CGS001-58478	ENOPH1	-			
1732	61.31	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1733	61.29	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
1734	61.26	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
1735	61.24	oe	ccsbBroad304_02686	COPZ1	-			
1736	61.22	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
1737	61.14	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
1738	61.13	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
1739	61.05	oe	ccsbBroad304_06870	RNH1	-			
1740	61.01	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
1741	60.93	cc		Cyclooxygenase inhibitor	-			
1742	60.9	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
1743	60.89	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
1744	60.86	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
1745	60.79	kd	CGS001-55612	FERMT1	Fermitins			
1746	60.72	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
1747	60.71	oe	ccsbBroad304_06237	GAA	Glycosidases			
1748	60.65	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
1749	60.59	oe	ccsbBroad304_05135	PARP15	-			
1750	60.57	oe	ccsbBroad304_04465	RERG	-			
1751	60.55	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
1752	60.55	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
1753	60.53	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
1754	60.53	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
1755	60.28	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
1756	60.27	kd	CGS001-9926	LPGAT1	-			
1757	60.22	kd	CGS001-3659	IRF1	-			
1758	60.22	kd	CGS001-8692	HYAL2	-			
1759	60.21	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
1760	60.16	oe	ccsbBroad304_07362	NMI	-			
1761	60.04	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
1762	60.04	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
1763	60	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
1764	59.97	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
1765	59.91	kd	CGS001-2023	ENO1	-			
1766	59.91	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
1767	59.9	cc		Bile acid	-			
1768	59.89	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
1769	59.86	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
1770	59.86	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
1771	59.73	oe	ccsbBroad304_07102	TSG101	-			
1772	59.73	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
1773	59.72	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
1774	59.66	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
1775	59.64	kd	CGS001-663	BNIP2	-			
1776	59.61	cp	BRD-K34508425	KUC103898N	-666			-666
1777	59.61	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
1778	59.59	oe	ccsbBroad304_02221	HS2ST1	Sulfotransferases, membrane-bound			
1779	59.54	oe	ccsbBroad304_02057	P4HA2	-			
1780	59.54	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
1781	59.54	kd	CGS001-9841	ZBTB24	BTB/POZ domain containing			
1782	59.3	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
1783	59.28	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
1784	59.28	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
1785	59.26	kd	CGS001-1950	EGF	-			
1786	59.24	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
1787	59.2	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
1788	59.18	kd	CGS001-51380	CSAD	-			
1789	59.16	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
1790	59.14	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
1791	59.13	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
1792	59.03	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
1793	59.02	oe	ccsbBroad304_03415	GFOD1	-			
1794	59.01	kd	CGS001-4695	NDUFA2	Mitochondrial respiratory chain complex / Complex I			
1795	58.99	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
1796	58.98	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
1797	58.94	kd	CGS001-9180	OSMR	IL-6 receptor family			
1798	58.92	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
1799	58.83	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
1800	58.82	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
1801	58.8	kd	CGS001-23344	ESYT1	Synaptotagmins			
1802	58.73	oe	ccsbBroad304_01974	RNASET2	-			
1803	58.62	cc		Progesterone receptor antagonist	-			
1804	58.57	kd	CGS001-79094	CHAC1	-			
1805	58.55	kd	CGS001-2017	CTTN	-			
1806	58.5	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
1807	58.44	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
1808	58.44	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
1809	58.42	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
1810	58.42	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
1811	58.41	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
1812	58.41	oe	ccsbBroad304_06172	EPS8	-			
1813	58.37	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1814	58.36	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
1815	58.29	cc		Vesicular Transport LOF	-			
1816	58.29	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
1817	58.25	oe	ccsbBroad304_13998	PDXK	-			
1818	58.25	oe	ccsbBroad304_07662	NPRL2	-			
1819	58.25	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1820	58.2	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
1821	58.18	kd	CGS001-5883	RAD9A	-			
1822	58.17	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
1823	58.15	kd	CGS001-9318	COPS2	-			
1824	58.12	oe	ccsbBroad304_06318	GPER	-			
1825	58.09	oe	ccsbBroad304_07923	LSM5	-			
1826	58.09	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
1827	58.02	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
1828	57.91	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
1829	57.89	kd	CGS001-3131	HLF	-			
1830	57.88	kd	CGS001-64750	SMURF2	-			
1831	57.87	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
1832	57.86	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
1833	57.85	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
1834	57.82	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
1835	57.82	kd	CGS001-23710	GABARAPL1	-			
1836	57.67	oe	ccsbBroad304_01576	SOAT1	-			
1837	57.66	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
1838	57.66	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1839	57.63	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
1840	57.61	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
1841	57.56	kd	CGS001-11340	EXOSC8	-			
1842	57.45	kd	CGS001-6347	CCL2	Chemokine ligands			
1843	57.41	kd	CGS001-7852	CXCR4	Chemokine receptors			
1844	57.37	kd	CGS001-1676	DFFA	-			
1845	57.35	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
1846	57.3	oe	ccsbBroad304_03103	SNX11	Sorting nexins			
1847	57.26	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
1848	57.18	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
1849	57.17	oe	ccsbBroad304_01234	POLB	DNA polymerases			
1850	57.1	oe	ccsbBroad304_06098	DHCR24	-			
1851	57.07	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1852	57.01	cc		Vitamin D receptor agonist	-			
1853	57.01	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
1854	57.01	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
1855	57.01	kd	CGS001-345	APOC3	Apolipoproteins			
1856	57	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
1857	56.99	kd	CGS001-283450	C12ORF51	-			
1858	56.97	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
1859	56.97	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
1860	56.91	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
1861	56.87	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
1862	56.87	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
1863	56.87	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
1864	56.83	oe	ccsbBroad304_10431	HADHB	-			
1865	56.83	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
1866	56.77	kd	CGS001-1026	CDKN1A	-			
1867	56.76	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
1868	56.73	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
1869	56.69	oe	ccsbBroad304_01855	NCOA4	-			
1870	56.64	oe	ccsbBroad304_07372	ZBED1	Pseudoautosomal regions / PAR1			
1871	56.63	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
1872	56.63	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
1873	56.56	oe	ccsbBroad304_00876	INSIG1	-			
1874	56.55	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
1875	56.52	oe	ccsbBroad304_01466	RRM2	Ribonucleoside-diphosphate reductases			
1876	56.49	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
1877	56.46	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
1878	56.46	kd	CGS001-64080	RBKS	-			
1879	56.43	oe	ccsbBroad304_08684	CXCR7	-			
1880	56.34	oe	ccsbBroad304_07252	DGKZ	-			
1881	56.32	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
1882	56.32	kd	CGS001-80135	RPF1	-			
1883	56.31	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
1884	56.25	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
1885	56.18	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
1886	56.12	oe	ccsbBroad304_03640	CEP72	-			
1887	56.11	oe	ccsbBroad304_00249	CD14	CD molecules			
1888	56.11	kd	CGS001-58477	SRPRB	-			
1889	56.1	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
1890	56.03	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
1891	56.02	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
1892	56.01	kd	CGS001-6652	SORD	-			
1893	55.95	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
1894	55.93	cc		Serotonin receptor agonist	-			
1895	55.92	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
1896	55.92	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
1897	55.92	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
1898	55.87	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
1899	55.87	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
1900	55.84	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
1901	55.84	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
1902	55.8	kd	CGS001-11262	SP140	Zinc fingers, PHD-type			
1903	55.79	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
1904	55.74	kd	CGS001-24140	FTSJ1	-			
1905	55.73	oe	ccsbBroad304_07238	STK24	YSK subfamily			
1906	55.72	kd	CGS001-5575	PRKAR1B	Protein kinase A			
1907	55.67	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
1908	55.64	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
1909	55.6	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
1910	55.56	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
1911	55.55	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
1912	55.51	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
1913	55.49	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
1914	55.41	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
1915	55.38	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1916	55.34	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
1917	55.3	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
1918	55.26	kd	CGS001-94234	FOXQ1	Forkhead boxes			
1919	55.25	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
1920	55.23	oe	ccsbBroad304_04170	PANK2	-			
1921	55.23	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
1922	55.21	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
1923	55.21	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
1924	55.14	oe	ccsbBroad304_05887	CFB	Complement system			
1925	55.11	kd	CGS001-6223	RPS19	S ribosomal proteins			
1926	55.1	kd	CGS001-5962	RDX	-			
1927	55.07	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
1928	55.02	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1929	55.01	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
1930	54.94	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
1931	54.93	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
1932	54.87	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
1933	54.87	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
1934	54.86	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
1935	54.84	oe	ccsbBroad304_02123	RPS6KA5	MSK subfamily			
1936	54.84	oe	ccsbBroad304_08339	CMPK1	-			
1937	54.83	oe	ccsbBroad304_00652	GNAS	-			
1938	54.82	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
1939	54.79	kd	CGS001-64135	IFIH1	-			
1940	54.64	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
1941	54.63	kd	CGS001-3676	ITGA4	Integrins			
1942	54.57	kd	CGS001-3077	HFE	Immunoglobulin superfamily / C1-set domain containing			
1943	54.47	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
1944	54.46	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
1945	54.3	kd	CGS001-28511	NKIRAS2	-			
1946	54.29	cc		PKC inhibitor	-			
1947	54.22	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
1948	54.13	oe	ccsbBroad304_02716	NMNAT2	-			
1949	54.12	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
1950	54.12	kd	CGS001-6477	SIAH1	-			
1951	54.1	kd	CGS001-55715	DOK4	Pleckstrin homology (PH) domain containing			
1952	53.94	oe	ccsbBroad304_03040	NKIRAS2	-			
1953	53.93	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
1954	53.91	oe	ccsbBroad304_03874	UBL5	-			
1955	53.91	kd	CGS001-6857	SYT1	Synaptotagmins			
1956	53.91	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
1957	53.87	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
1958	53.87	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
1959	53.69	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
1960	53.65	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
1961	53.65	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1962	53.65	kd	CGS001-27297	CRCP	-			
1963	53.63	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
1964	53.62	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
1965	53.59	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
1966	53.59	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
1967	53.59	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
1968	53.57	oe	ccsbBroad304_00568	FHL2	-			
1969	53.55	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
1970	53.54	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
1971	53.5	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1972	53.5	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
1973	53.46	oe	ccsbBroad304_06324	GPX7	-			
1974	53.37	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1975	53.3	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
1976	53.28	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
1977	53.27	oe	ccsbBroad304_00214	CAPN1	EF-hand domain containing			
1978	53.24	kd	CGS001-8453	CUL2	-			
1979	53.18	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
1980	53.09	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
1981	53.08	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
1982	53.04	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
1983	53.01	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
1984	52.97	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
1985	52.94	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
1986	52.93	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
1987	52.91	kd	CGS001-7295	TXN	-			
1988	52.9	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
1989	52.85	oe	ccsbBroad304_03308	YTHDF2	-			
1990	52.81	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
1991	52.78	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
1992	52.78	oe	ccsbBroad304_06739	PLOD1	-			
1993	52.74	kd	CGS001-5831	PYCR1	-			
1994	52.73	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
1995	52.7	kd	CGS001-10904	BLCAP	-			
1996	52.65	kd	CGS001-3248	HPGD	Prostaglandin synthases			
1997	52.64	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
1998	52.58	kd	CGS001-23139	MAST2	MAST family			
1999	52.54	kd	CGS001-65243	ZNF643	-			
2000	52.47	kd	CGS001-8624	PSMG1	-			
2001	52.46	cc		Wnt family LOF	-			
2002	52.44	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
2003	52.42	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
2004	52.26	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
2005	52.24	oe	ccsbBroad304_02653	PRAF2	-			
2006	52.12	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
2007	52.06	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
2008	52.05	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
2009	52.02	oe	ccsbBroad304_02502	GNA13	-			
2010	52.02	kd	CGS001-54821	ERCC6L	-			
2011	52.01	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
2012	51.98	oe	ccsbBroad304_02384	SMNDC1	Tudor domain containing			
2013	51.97	kd	CGS001-8480	RAE1	WD repeat domain containing			
2014	51.91	kd	CGS001-8802	SUCLG1	-			
2015	51.85	kd	CGS001-6832	SUPV3L1	-			
2016	51.83	kd	CGS001-337867	UBAC2	-			
2017	51.81	kd	CGS001-26298	EHF	-			
2018	51.8	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
2019	51.76	kd	CGS001-4173	MCM4	-			
2020	51.75	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2021	51.69	oe	ccsbBroad304_06777	PRNP	CD molecules			
2022	51.69	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
2023	51.69	kd	CGS001-5934	RBL2	-			
2024	51.68	oe	ccsbBroad304_07287	HYAL2	-			
2025	51.65	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
2026	51.59	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
2027	51.53	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
2028	51.41	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
2029	51.4	oe	ccsbBroad304_06695	PCK2	-			
2030	51.35	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2031	51.28	kd	CGS001-6256	RXRA	Retinoid X receptors			
2032	51.27	oe	ccsbBroad304_01623	SUPT4H1	-			
2033	51.27	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
2034	51.25	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
2035	51.25	cp	BRD-K99545815	PF-562271	Focal adhesion kinase inhibitor		PTK2, PTK2B	Focal adhesion kinase inhibitor
2036	51.17	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
2037	51.13	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
2038	51.06	kd	CGS001-1119	CHKA	-			
2039	51.05	kd	CGS001-1362	CPD	Carboxypeptidase A			
2040	51.03	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
2041	50.92	kd	CGS001-3033	HADH	-			
2042	50.87	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
2043	50.83	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2044	50.8	kd	CGS001-9447	AIM2	-			
2045	50.78	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
2046	50.69	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
2047	50.67	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
2048	50.61	oe	ccsbBroad304_00614	GAMT	-			
2049	50.61	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
2050	50.59	oe	ccsbBroad304_03565	ADI1	-			
2051	50.58	oe	ccsbBroad304_00397	CTSK	Cathepsins			
2052	50.56	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
2053	50.55	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
2054	50.53	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
2055	50.49	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
2056	50.45	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
2057	50.42	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
2058	50.4	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
2059	50.39	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
2060	50.38	oe	ccsbBroad304_02804	KLHDC2	-			
2061	50.36	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
2062	50.34	kd	CGS001-11124	FAF1	UBX domain containing			
2063	50.3	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
2064	50.25	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
2065	50.23	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
2066	50.23	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
2067	50.23	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
2068	50.2	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
2069	50.2	kd	CGS001-81848	SPRY4	-			
2070	50.18	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
2071	50.14	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
2072	50.07	kd	CGS001-29978	UBQLN2	Ubiquilin family			
2073	50.02	kd	CGS001-1356	CP	-			
2074	50.02	kd	CGS001-64781	CERK	Ceramide kinase			
2075	50.01	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
2076	49.98	cc		Lipocalins GOF	-			
2077	49.95	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
2078	49.93	oe	ccsbBroad304_04194	ELL3	-			
2079	49.93	oe	ccsbBroad304_04626	EGLN3	-			
2080	49.93	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
2081	49.9	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
2082	49.84	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
2083	49.84	kd	CGS001-5366	PMAIP1	-			
2084	49.81	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
2085	49.78	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
2086	49.77	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
2087	49.76	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
2088	49.62	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
2089	49.61	kd	CGS001-4194	MDM4	-			
2090	49.58	oe	ccsbBroad304_14020	SH3BP5	-			
2091	49.56	oe	ccsbBroad304_00532	F11	Chymotrypsin			
2092	49.54	oe	ccsbBroad304_02674	STK38	NDR family			
2093	49.5	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
2094	49.49	oe	ccsbBroad304_00648	GLRX	-			
2095	49.48	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
2096	49.48	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2097	49.42	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
2098	49.38	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
2099	49.36	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
2100	49.35	oe	ccsbBroad304_02708	TRIM32	-			
2101	49.35	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
2102	49.33	cc		GATA Zinc finger domain containing LOF	-			
2103	49.3	kd	CGS001-1611	DAP	-			
2104	49.29	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
2105	49.25	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
2106	49.24	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
2107	49.23	kd	CGS001-23014	FBXO21	F-boxes / other			
2108	49.22	oe	ccsbBroad304_00098	ARG1	Arginase			
2109	49.15	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
2110	49.12	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
2111	49.11	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
2112	49.04	oe	ccsbBroad304_06048	CRYZ	-			
2113	49.04	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
2114	49	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
2115	49	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
2116	48.99	kd	CGS001-10468	FST	-			
2117	48.94	cc		FOS transcription factor family GOF	-			
2118	48.89	cc		Non Homologous End Joining LOF	-			
2119	48.87	kd	CGS001-9443	MED7	-			
2120	48.86	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
2121	48.83	kd	CGS001-22921	MSRB2	-			
2122	48.77	oe	ccsbBroad304_05902	BNIP3	-			
2123	48.75	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
2124	48.74	kd	CGS001-8435	SOAT2	-			
2125	48.67	oe	ccsbBroad304_03269	CD320	CD molecules			
2126	48.65	kd	CGS001-8914	TIMELESS	-			
2127	48.64	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
2128	48.61	kd	CGS001-8974	P4HA2	-			
2129	48.6	oe	ccsbBroad304_00053	ALDOA	-			
2130	48.6	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
2131	48.49	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
2132	48.46	oe	ccsbBroad304_03910	CCDC90A	-			
2133	48.46	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
2134	48.46	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
2135	48.43	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
2136	48.38	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
2137	48.3	kd	CGS001-3066	HDAC2	Histone deacetylases			
2138	48.29	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
2139	48.21	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
2140	48.19	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
2141	48.19	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
2142	48.18	oe	ccsbBroad304_02837	BHMT2	-			
2143	48.14	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
2144	48.13	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
2145	48.13	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
2146	48.11	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
2147	48.09	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
2148	47.98	kd	CGS001-378	ARF4	ADP-ribosylation factors			
2149	47.92	oe	ccsbBroad304_02086	PDLIM1	-			
2150	47.89	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
2151	47.79	oe	ccsbBroad304_08452	PIH1D1	-			
2152	47.73	oe	ccsbBroad304_06642	NIT1	-			
2153	47.73	kd	CGS001-4151	MB	-			
2154	47.72	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
2155	47.67	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
2156	47.61	kd	CGS001-4701	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
2157	47.59	oe	ccsbBroad304_08292	IP6K2	-			
2158	47.59	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2159	47.56	oe	ccsbBroad304_01677	TLE2	WD repeat domain containing			
2160	47.55	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
2161	47.54	oe	ccsbBroad304_02361	MFSD10	-			
2162	47.52	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
2163	47.5	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
2164	47.5	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
2165	47.49	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
2166	47.47	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
2167	47.45	oe	ccsbBroad304_02386	EIF1B	-			
2168	47.43	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
2169	47.41	kd	CGS001-6461	SHB	SH2 domain containing			
2170	47.4	kd	CGS001-572	BAD	-			
2171	47.39	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
2172	47.36	kd	CGS001-4830	NME1	-			
2173	47.33	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
2174	47.29	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
2175	47.29	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
2176	47.29	kd	CGS001-5188	PET112	-			
2177	47.28	oe	ccsbBroad304_07827	STK38L	NDR family			
2178	47.27	kd	CGS001-116519	APOA5	Apolipoproteins			
2179	47.26	kd	CGS001-1647	GADD45A	-			
2180	47.24	kd	CGS001-6601	SMARCC2	-			
2181	47.21	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
2182	47.21	oe	ccsbBroad304_02668	PNKP	-			
2183	47.21	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
2184	47.19	oe	ccsbBroad304_01723	TTK	TTK family			
2185	47.19	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
2186	47.07	kd	CGS001-8841	HDAC3	Histone deacetylases			
2187	47.03	kd	CGS001-944	TNFSF8	CD molecules			
2188	47	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
2189	47	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
2190	47	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
2191	46.95	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
2192	46.93	oe	ccsbBroad304_06004	CKB	-			
2193	46.9	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
2194	46.89	oe	ccsbBroad304_01105	PNP	-			
2195	46.85	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
2196	46.83	oe	ccsbBroad304_00102	RND3	-			
2197	46.83	oe	ccsbBroad304_02203	MAD2L1BP	-			
2198	46.83	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
2199	46.82	kd	CGS001-26292	MYCBP	-			
2200	46.79	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
2201	46.78	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2202	46.76	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
2203	46.74	kd	CGS001-64094	SMOC2	EF-hand domain containing			
2204	46.71	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
2205	46.71	kd	CGS001-4287	ATXN3	Ataxins			
2206	46.69	oe	ccsbBroad304_08167	DNTTIP2	-			
2207	46.61	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
2208	46.58	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
2209	46.53	oe	ccsbBroad304_10232	PDIA5	Protein disulfide isomerases			
2210	46.52	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
2211	46.48	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
2212	46.45	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
2213	46.44	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
2214	46.38	kd	CGS001-8531	CSDA	-			
2215	46.36	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
2216	46.35	oe	ccsbBroad304_00099	ARG2	Arginase			
2217	46.35	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
2218	46.29	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
2219	46.28	kd	CGS001-9412	MED21	-			
2220	46.24	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
2221	46.17	kd	CGS001-54505	DHX29	DEAH-boxes			
2222	46.16	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
2223	46.15	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
2224	46.11	oe	ccsbBroad304_01205	PIN1	-			
2225	46.11	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
2226	46.1	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
2227	46.1	kd	CGS001-5529	PPP2R5E	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
2228	46.05	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
2229	45.99	oe	ccsbBroad304_06562	MAT1A	-			
2230	45.96	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
2231	45.94	oe	ccsbBroad304_04404	TUBB6	Tubulins			
2232	45.93	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
2233	45.93	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
2234	45.88	kd	CGS001-5050	PAFAH1B3	-			
2235	45.84	kd	CGS001-55556	ENOSF1	-			
2236	45.78	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
2237	45.74	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
2238	45.72	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
2239	45.62	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
2240	45.58	oe	ccsbBroad304_00390	CTGF	-			
2241	45.57	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
2242	45.56	oe	ccsbBroad304_02759	DICER1	-			
2243	45.54	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
2244	45.52	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
2245	45.52	oe	ccsbBroad304_06765	PRCC	-			
2246	45.51	kd	CGS001-7039	TGFA	-			
2247	45.5	oe	ccsbBroad304_02772	ICMT	-			
2248	45.5	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
2249	45.5	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
2250	45.42	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
2251	45.4	kd	CGS001-2335	FN1	Endogenous ligands			
2252	45.39	kd	CGS001-51441	YTHDF2	-			
2253	45.27	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
2254	45.24	oe	ccsbBroad304_02219	MORF4L2	-			
2255	45.23	oe	ccsbBroad304_06902	RRM1	Ribonucleoside-diphosphate reductases			
2256	45.18	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
2257	45.17	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
2258	45.12	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
2259	45.12	kd	CGS001-10810	WASF3	-			
2260	45.11	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
2261	45.05	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
2262	45.02	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
2263	45.01	cc		Potassium channel blocker	-			
2264	44.99	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
2265	44.99	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
2266	44.92	kd	CGS001-387	RHOA	-			
2267	44.89	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
2268	44.88	oe	ccsbBroad304_03428	EXOSC4	-			
2269	44.86	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
2270	44.84	oe	ccsbBroad304_03951	NARFL	-			
2271	44.82	oe	ccsbBroad304_03191	NOSIP	-			
2272	44.79	kd	CGS001-593	BCKDHA	-			
2273	44.78	oe	ccsbBroad304_02367	CALCOCO2	-			
2274	44.76	kd	CGS001-6722	SRF	-			
2275	44.75	oe	ccsbBroad304_02239	RASSF2	-			
2276	44.69	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
2277	44.67	kd	CGS001-5073	PARN	-			
2278	44.66	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
2279	44.66	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
2280	44.64	kd	CGS001-1837	DTNA	-			
2281	44.63	kd	CGS001-51655	RASD1	-			
2282	44.62	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
2283	44.58	kd	CGS001-23650	TRIM29	-			
2284	44.57	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
2285	44.57	kd	CGS001-25966	C2CD2	-			
2286	44.54	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2287	44.54	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
2288	44.54	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
2289	44.51	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
2290	44.48	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
2291	44.48	oe	ccsbBroad304_02425	CDIPT	-			
2292	44.48	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
2293	44.47	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
2294	44.46	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
2295	44.44	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
2296	44.39	kd	CGS001-1440	CSF3	Endogenous ligands			
2297	44.38	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
2298	44.34	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
2299	44.26	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
2300	44.23	oe	ccsbBroad304_06349	HAGH	-			
2301	44.22	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
2302	44.18	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
2303	44.15	oe	ccsbBroad304_03386	SPA17	-			
2304	44.13	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
2305	44.11	kd	CGS001-949	SCARB1	-			
2306	44.06	oe	ccsbBroad304_04288	RPS6KL1	RSKL family			
2307	44.04	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
2308	43.98	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
2309	43.97	kd	CGS001-2773	GNAI3	-			
2310	43.88	oe	ccsbBroad304_00854	IL8	-			
2311	43.88	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
2312	43.86	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
2313	43.81	kd	CGS001-27034	ACAD8	-			
2314	43.76	oe	ccsbBroad304_02737	JMJD6	-			
2315	43.73	oe	ccsbBroad304_08322	UFM1	-			
2316	43.72	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
2317	43.7	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
2318	43.69	kd	CGS001-6499	SKIV2L	-			
2319	43.67	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
2320	43.65	kd	CGS001-9797	TATDN2	-			
2321	43.62	oe	ccsbBroad304_01933	TEAD2	-			
2322	43.61	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
2323	43.6	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
2324	43.59	kd	CGS001-498	ATP5A1	ATPases / F-type			
2325	43.53	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
2326	43.51	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
2327	43.46	kd	CGS001-22823	MTF2	Zinc fingers, PHD-type			
2328	43.44	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
2329	43.42	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
2330	43.39	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
2331	43.38	kd	CGS001-4691	NCL	RNA binding motif (RRM) containing			
2332	43.37	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2333	43.37	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
2334	43.36	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
2335	43.34	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
2336	43.31	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
2337	43.26	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
2338	43.26	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
2339	43.18	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
2340	43.17	oe	ccsbBroad304_03772	CCNL1	-			
2341	43.16	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
2342	43.12	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
2343	43.1	kd	CGS001-55176	SEC61A2	-			
2344	43.09	kd	CGS001-83440	ADPGK	-			
2345	43.07	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
2346	43.01	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
2347	42.99	kd	CGS001-27113	BBC3	-			
2348	42.97	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
2349	42.95	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
2350	42.95	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2351	42.9	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
2352	42.88	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
2353	42.81	oe	ccsbBroad304_06574	MDH2	-			
2354	42.81	kd	CGS001-3660	IRF2	-			
2355	42.79	kd	CGS001-80349	WDR61	WD repeat domain containing			
2356	42.77	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
2357	42.75	oe	ccsbBroad304_03182	GLOD4	-			
2358	42.7	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
2359	42.69	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
2360	42.63	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
2361	42.63	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
2362	42.6	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
2363	42.59	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
2364	42.57	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
2365	42.55	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
2366	42.55	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
2367	42.51	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
2368	42.48	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
2369	42.48	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
2370	42.44	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
2371	42.44	kd	CGS001-10284	SAP18	-			
2372	42.42	oe	ccsbBroad304_00161	BID	Endogenous ligands			
2373	42.42	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
2374	42.34	oe	ccsbBroad304_07800	EXOSC8	-			
2375	42.32	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
2376	42.25	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
2377	42.25	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
2378	42.25	kd	CGS001-162699	TCEB3C	-			
2379	42.24	kd	CGS001-7057	THBS1	-			
2380	42.16	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2381	42.14	kd	CGS001-578	BAK1	-			
2382	42.11	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
2383	42.08	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
2384	42.04	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
2385	42.02	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
2386	42	kd	CGS001-7917	BAG6	-			
2387	41.98	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2388	41.98	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
2389	41.97	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
2390	41.94	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
2391	41.91	kd	CGS001-3176	HNMT	-			
2392	41.89	oe	ccsbBroad304_10437	STMN1	-			
2393	41.81	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
2394	41.78	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
2395	41.77	kd	CGS001-51593	SRRT	-			
2396	41.74	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
2397	41.72	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
2398	41.7	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
2399	41.69	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
2400	41.69	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
2401	41.68	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
2402	41.65	oe	ccsbBroad304_01257	PPOX	-			
2403	41.58	kd	CGS001-257397	TAB3	-			
2404	41.58	kd	CGS001-9158	FIBP	-			
2405	41.51	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
2406	41.5	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
2407	41.4	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2408	41.38	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
2409	41.24	cc		Kruppel like transcription factors LOF	-			
2410	41.24	kd	CGS001-6871	TADA2A	-			
2411	41.22	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
2412	41.22	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
2413	41.2	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
2414	41.2	kd	CGS001-25874	BRP44	-			
2415	41.14	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2416	41.12	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
2417	41.1	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
2418	41.08	kd	CGS001-30836	DNTTIP2	-			
2419	41.05	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
2420	40.99	cp	BRD-A71009679	KUC103420N	-666			-666
2421	40.96	kd	CGS001-85004	RERG	-			
2422	40.95	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
2423	40.93	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
2424	40.91	oe	ccsbBroad304_06292	GNAI2	-			
2425	40.85	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
2426	40.8	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
2427	40.8	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
2428	40.73	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
2429	40.7	kd	CGS001-3669	ISG20	-			
2430	40.65	oe	ccsbBroad304_02756	RRP8	-			
2431	40.64	kd	CGS001-6118	RPA2	-			
2432	40.57	oe	ccsbBroad304_03023	CRCP	-			
2433	40.56	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2434	40.47	kd	CGS001-4292	MLH1	-			
2435	40.43	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
2436	40.4	kd	CGS001-4121	MAN1A1	-			
2437	40.39	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2438	40.37	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
2439	40.36	oe	ccsbBroad304_01148	PCBD1	-			
2440	40.35	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
2441	40.3	oe	ccsbBroad304_05417	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
2442	40.26	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
2443	40.23	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
2444	40.21	oe	ccsbBroad304_02002	RNMT	-			
2445	40.19	kd	CGS001-55968	NSFL1C	UBX domain containing			
2446	40.15	kd	CGS001-2961	GTF2E2	General transcription factors			
2447	40.15	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
2448	40.13	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
2449	40.12	kd	CGS001-10312	TCIRG1	ATPases / V-type			
2450	40.12	kd	CGS001-6117	RPA1	-			
2451	40.01	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
2452	40	cc		Glycogen synthase kinase inhibitor	-			
2453	39.99	kd	CGS001-8623	ASMTL	Pseudoautosomal regions / PAR1			
2454	39.96	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
2455	39.92	kd	CGS001-8649	LAMTOR3	-			
2456	39.87	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
2457	39.82	kd	CGS001-56940	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
2458	39.77	oe	ccsbBroad304_02862	CCRN4L	-			
2459	39.76	kd	CGS001-6778	STAT6	SH2 domain containing			
2460	39.72	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
2461	39.64	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
2462	39.63	kd	CGS001-5900	RALGDS	-			
2463	39.62	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
2464	39.59	kd	CGS001-7471	WNT1	Endogenous ligands			
2465	39.58	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
2466	39.57	cc		FGFR inhibitor	-			
2467	39.53	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
2468	39.52	oe	ccsbBroad304_06013	CLPTM1	-			
2469	39.49	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
2470	39.49	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
2471	39.47	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
2472	39.46	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
2473	39.44	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
2474	39.43	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
2475	39.4	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
2476	39.39	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
2477	39.36	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
2478	39.35	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
2479	39.33	kd	CGS001-6210	RPS15A	S ribosomal proteins			
2480	39.3	oe	ccsbBroad304_03544	FAIM	-			
2481	39.3	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
2482	39.28	kd	CGS001-397	ARHGDIB	Endogenous ligands			
2483	39.26	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
2484	39.19	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
2485	39.18	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
2486	39.15	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
2487	39.13	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
2488	39.12	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
2489	39.12	kd	CGS001-4710	NDUFB4	Mitochondrial respiratory chain complex / Complex I			
2490	39.1	kd	CGS001-7374	UNG	-			
2491	39.09	cc		DNA synthesis inhibitor	-			
2492	39.09	oe	ccsbBroad304_01215	PLAUR	CD molecules			
2493	39	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
2494	38.98	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
2495	38.96	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
2496	38.95	kd	CGS001-54499	TMCO1	-			
2497	38.93	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
2498	38.91	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
2499	38.91	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
2500	38.88	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
2501	38.86	oe	ccsbBroad304_01962	STK16	NAK family			
2502	38.86	kd	CGS001-624	BDKRB2	Bradykinin receptors			
2503	38.85	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
2504	38.82	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
2505	38.81	oe	ccsbBroad304_00063	AMPD2	-			
2506	38.8	oe	ccsbBroad304_09035	COASY	-			
2507	38.79	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
2508	38.77	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
2509	38.76	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
2510	38.69	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
2511	38.66	oe	ccsbBroad304_06226	FTL	-			
2512	38.65	kd	CGS001-1212	CLTB	-			
2513	38.56	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
2514	38.56	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
2515	38.55	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
2516	38.52	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
2517	38.5	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
2518	38.49	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
2519	38.48	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
2520	38.47	oe	ccsbBroad304_03933	CARD9	-			
2521	38.45	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
2522	38.39	oe	ccsbBroad304_00550	FDXR	-			
2523	38.34	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
2524	38.32	oe	ccsbBroad304_09689	ZNF595	Zinc fingers, C2H2-type			
2525	38.28	oe	ccsbBroad304_03798	PHTF2	-			
2526	38.27	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2527	38.26	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
2528	38.26	kd	CGS001-115	ADCY9	Adenylyl cyclases			
2529	38.25	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
2530	38.24	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
2531	38.2	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
2532	38.18	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
2533	38.14	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
2534	38.06	kd	CGS001-4436	MSH2	-			
2535	38.04	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
2536	38.01	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
2537	38	oe	ccsbBroad304_08786	ZNF350	Zinc fingers, C2H2-type			
2538	37.99	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
2539	37.93	kd	CGS001-4300	MLLT3	-			
2540	37.9	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
2541	37.87	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
2542	37.87	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
2543	37.86	kd	CGS001-1725	DHPS	-			
2544	37.85	oe	ccsbBroad304_06290	GNA15	-			
2545	37.82	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
2546	37.78	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
2547	37.77	oe	ccsbBroad304_01061	NAB2	-			
2548	37.72	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
2549	37.7	kd	CGS001-57819	LSM2	-			
2550	37.69	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
2551	37.69	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
2552	37.6	kd	CGS001-5359	PLSCR1	-			
2553	37.59	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
2554	37.53	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
2555	37.5	kd	CGS001-5891	MOK	RCK family			
2556	37.49	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
2557	37.48	kd	CGS001-4125	MAN2B1	-			
2558	37.45	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
2559	37.42	kd	CGS001-7270	TTF1	-			
2560	37.42	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
2561	37.39	kd	CGS001-3482	IGF2R	CD molecules			
2562	37.36	oe	ccsbBroad304_13499	KSR2	RAF family			
2563	37.33	oe	ccsbBroad304_04053	DERL1	-			
2564	37.31	kd	CGS001-538	ATP7A	ATPases / P-type			
2565	37.31	oe	ccsbBroad304_07564	SLC25A15	Mitochondrial amino acid transporter subfamily			
2566	37.3	oe	ccsbBroad304_06253	GALT	-			
2567	37.28	kd	CGS001-134860	TAAR9	GPCR / Class A : Trace amine associated receptors			
2568	37.27	oe	ccsbBroad304_01852	ZNF212	Zinc fingers, C2H2-type			
2569	37.18	kd	CGS001-161	AP2A2	-			
2570	37.16	kd	CGS001-2000	ELF4	ETS Transcription Factors			
2571	37.14	kd	CGS001-55111	PLEKHJ1	Pleckstrin homology (PH) domain containing			
2572	37.13	oe	ccsbBroad304_00810	HYAL1	-			
2573	37.11	oe	ccsbBroad304_08055	ATP5S	-			
2574	37.08	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2575	37.07	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
2576	37.07	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
2577	37.02	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
2578	36.99	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
2579	36.97	oe	ccsbBroad304_00101	RHOC	-			
2580	36.91	oe	ccsbBroad304_01035	MSH5	-			
2581	36.91	oe	ccsbBroad304_03808	ERGIC1	-			
2582	36.91	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
2583	36.91	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
2584	36.87	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
2585	36.85	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
2586	36.84	kd	CGS001-56616	DIABLO	-			
2587	36.81	oe	ccsbBroad304_02416	TUBB4B	-			
2588	36.78	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
2589	36.73	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2590	36.72	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
2591	36.69	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
2592	36.67	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
2593	36.65	kd	CGS001-4122	MAN2A2	-			
2594	36.64	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
2595	36.61	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
2596	36.6	oe	ccsbBroad304_01607	STAT1	SH2 domain containing			
2597	36.58	oe	ccsbBroad304_09881	RFX6	-			
2598	36.56	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
2599	36.51	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2600	36.5	oe	ccsbBroad304_01392	TRIM27	-			
2601	36.48	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
2602	36.47	kd	CGS001-4482	MSRA	-			
2603	36.46	kd	CGS001-2745	GLRX	-			
2604	36.43	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
2605	36.4	kd	CGS001-6567	SLC16A2	SLC16 family of monocarboxylate transporters			
2606	36.39	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
2607	36.35	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
2608	36.35	kd	CGS001-7158	TP53BP1	-			
2609	36.34	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
2610	36.34	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
2611	36.32	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
2612	36.26	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
2613	36.26	kd	CGS001-149428	BNIPL	-			
2614	36.2	kd	CGS001-124583	CANT1	-			
2615	36.19	kd	CGS001-51015	ISOC1	-			
2616	36.19	kd	CGS001-10969	EBNA1BP2	-			
2617	36.13	oe	ccsbBroad304_04471	C5ORF62	-			
2618	36.06	oe	ccsbBroad304_02157	MED21	-			
2619	36.02	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2620	36	oe	ccsbBroad304_08825	LHPP	-			
2621	35.99	cc		Supressors of cytokine signaling GOF	-			
2622	35.99	kd	CGS001-103	ADAR	-			
2623	35.96	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
2624	35.93	kd	CGS001-5836	PYGL	Glycogen phosphorylases			
2625	35.92	oe	ccsbBroad304_06828	PYCR1	-			
2626	35.87	oe	ccsbBroad304_01609	STAT3	SH2 domain containing			
2627	35.86	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
2628	35.83	oe	ccsbBroad304_00987	MCM3	-			
2629	35.83	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
2630	35.83	oe	ccsbBroad304_08282	ATP6V1D	ATPases / V-type			
2631	35.82	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
2632	35.81	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
2633	35.79	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
2634	35.79	kd	CGS001-4170	MCL1	-			
2635	35.75	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
2636	35.75	kd	CGS001-4846	NOS3	Nitric oxide synthases			
2637	35.74	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
2638	35.72	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2639	35.72	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
2640	35.64	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2641	35.63	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
2642	35.6	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
2643	35.6	kd	CGS001-8464	SUPT3H	-			
2644	35.56	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
2645	35.55	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
2646	35.51	kd	CGS001-3909	LAMA3	Laminins			
2647	35.5	oe	ccsbBroad304_02589	COPS5	-			
2648	35.46	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
2649	35.33	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
2650	35.31	oe	ccsbBroad304_00991	MDH1	-			
2651	35.3	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
2652	35.29	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
2653	35.28	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
2654	35.28	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
2655	35.27	kd	CGS001-9767	PHF16	-			
2656	35.27	kd	CGS001-9270	ITGB1BP1	-			
2657	35.21	kd	CGS001-4267	CD99	CD molecules			
2658	35.2	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
2659	35.19	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
2660	35.16	kd	CGS001-9552	SPAG7	-			
2661	35.16	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
2662	35.14	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
2663	35.12	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
2664	35.12	oe	ccsbBroad304_03556	SMU1	WD repeat domain containing			
2665	35.12	kd	CGS001-3800	KIF5C	Kinesins			
2666	35.1	kd	CGS001-83448	PUS7L	-			
2667	35.09	kd	CGS001-2524	FUT2	Fucosyltransferases			
2668	35.08	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
2669	35.06	oe	ccsbBroad304_02337	SLC25A13	Mitochondrial amino acid transporter subfamily			
2670	35.06	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
2671	35.05	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
2672	35.03	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
2673	35.01	oe	ccsbBroad304_09020	RUFY1	Zinc fingers, FYVE domain containing			
2674	34.99	kd	CGS001-56889	TM9SF3	-			
2675	34.97	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
2676	34.97	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
2677	34.93	oe	ccsbBroad304_01640	TAF12	-			
2678	34.91	kd	CGS001-11179	ZNF277	-			
2679	34.88	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
2680	34.85	kd	CGS001-1534	CYB561	Cytochrome b genes			
2681	34.83	oe	ccsbBroad304_07326	EIF2B2	-			
2682	34.81	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
2683	34.8	cc		Bacterial 30S ribosomal subunit inhibitor	-			
2684	34.8	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
2685	34.8	kd	CGS001-7105	TSPAN6	Tetraspanins			
2686	34.8	kd	CGS001-22908	SACM1L	-			
2687	34.77	oe	ccsbBroad304_00183	C1S	Complement system			
2688	34.76	kd	CGS001-4946	OAZ1	-			
2689	34.75	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
2690	34.7	kd	CGS001-5624	PROC	Endogenous ligands			
2691	34.67	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
2692	34.67	oe	ccsbBroad304_02838	SDF2L1	-			
2693	34.64	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2694	34.64	kd	CGS001-1788	DNMT3A	Methyltransferases			
2695	34.59	oe	ccsbBroad304_01150	PCCB	Carboxylases			
2696	34.5	oe	ccsbBroad304_02576	MLLT11	-			
2697	34.48	oe	ccsbBroad304_00225	CAT	-			
2698	34.46	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
2699	34.4	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
2700	34.4	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
2701	34.38	oe	ccsbBroad304_02446	TADA3	-			
2702	34.38	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
2703	34.37	kd	CGS001-54623	PAF1	-			
2704	34.34	kd	CGS001-8985	PLOD3	-			
2705	34.3	oe	ccsbBroad304_02955	MYCBP	-			
2706	34.25	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
2707	34.25	kd	CGS001-4232	MEST	-			
2708	34.21	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
2709	34.2	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
2710	34.19	oe	ccsbBroad304_02815	SSBP2	-			
2711	34.19	oe	ccsbBroad304_06449	ILF3	-			
2712	34.16	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
2713	34.15	oe	ccsbBroad304_03305	ANAPC5	Anaphase promoting complex subunits			
2714	34.11	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
2715	34.1	kd	CGS001-5538	PPT1	-			
2716	34.1	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
2717	34.09	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
2718	34.09	oe	ccsbBroad304_05763	ACTB	-			
2719	34.08	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
2720	34.04	oe	ccsbBroad304_00874	INS	-			
2721	34.02	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
2722	34.02	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
2723	33.96	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
2724	33.96	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
2725	33.96	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
2726	33.93	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
2727	33.91	kd	CGS001-170463	SSBP4	-			
2728	33.83	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
2729	33.78	oe	ccsbBroad304_07349	MAP7	-			
2730	33.78	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
2731	33.75	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
2732	33.73	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
2733	33.71	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
2734	33.7	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
2735	33.68	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
2736	33.67	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
2737	33.67	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
2738	33.66	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
2739	33.63	kd	CGS001-2309	FOXO3	Forkhead boxes			
2740	33.61	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2741	33.59	kd	CGS001-7386	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
2742	33.58	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2743	33.49	kd	CGS001-51290	ERGIC2	-			
2744	33.44	oe	ccsbBroad304_00665	GOT1	-			
2745	33.43	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
2746	33.43	oe	ccsbBroad304_05802	ALDH1B1	Aldehyde dehydrogenases			
2747	33.41	kd	CGS001-7298	TYMS	Methyltransferases			
2748	33.39	kd	CGS001-4048	LTA4H	Hydrolases			
2749	33.36	oe	ccsbBroad304_01184	PGK1	-			
2750	33.31	kd	CGS001-10247	HRSP12	-			
2751	33.26	kd	CGS001-5045	FURIN	Subtilisin			
2752	33.23	kd	CGS001-4616	GADD45B	-			
2753	33.21	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
2754	33.16	oe	ccsbBroad304_00100	RHOA	-			
2755	33.16	kd	CGS001-11182	SLC2A6	Solute carriers			
2756	33.14	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2757	33.13	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
2758	33.08	kd	CGS001-56731	SLC2A4RG	-			
2759	33.08	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
2760	33.08	oe	ccsbBroad304_00112	ASNA1	-			
2761	33.04	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
2762	32.97	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
2763	32.95	kd	CGS001-506	ATP5B	ATPases / F-type			
2764	32.91	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
2765	32.9	oe	ccsbBroad304_01190	PHKG2	Phosphorylase kinase (PHK) family			
2766	32.88	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
2767	32.86	kd	CGS001-93594	WDR67	-			
2768	32.85	kd	CGS001-10046	MAMLD1	-			
2769	32.83	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
2770	32.83	kd	CGS001-3161	HMMR	CD molecules			
2771	32.81	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
2772	32.81	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
2773	32.81	kd	CGS001-23636	NUP62	-			
2774	32.77	kd	CGS001-1869	E2F1	-			
2775	32.76	kd	CGS001-5062	PAK2	PAKA subfamily			
2776	32.75	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2777	32.72	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
2778	32.68	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
2779	32.67	oe	ccsbBroad304_06136	ECHS1	-			
2780	32.65	oe	ccsbBroad304_01421	RPL11	L ribosomal proteins			
2781	32.65	kd	CGS001-23658	LSM5	-			
2782	32.64	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
2783	32.62	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
2784	32.6	oe	ccsbBroad304_00383	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
2785	32.58	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
2786	32.54	kd	CGS001-93185	IGSF8	CD molecules			
2787	32.54	kd	CGS001-1528	CYB5A	Cytochrome b genes			
2788	32.53	oe	ccsbBroad304_03980	DCLRE1B	-			
2789	32.52	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
2790	32.5	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
2791	32.49	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
2792	32.47	kd	CGS001-22903	BTBD3	BTB/POZ domain containing			
2793	32.41	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
2794	32.41	kd	CGS001-25836	NIPBL	-			
2795	32.32	oe	ccsbBroad304_00993	MDM4	-			
2796	32.32	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2797	32.29	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
2798	32.28	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
2799	32.25	oe	ccsbBroad304_06711	PFAS	-			
2800	32.23	kd	CGS001-3551	IKBKB	IKK family			
2801	32.16	oe	ccsbBroad304_01754	UCK2	-			
2802	32.16	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
2803	32.15	kd	CGS001-55082	ARGLU1	-			
2804	32.14	kd	CGS001-54512	EXOSC4	-			
2805	32.12	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
2806	32.12	kd	CGS001-1384	CRAT	-			
2807	32.08	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
2808	32.08	oe	ccsbBroad304_01659	TERF1	-			
2809	32.08	oe	ccsbBroad304_02506	EBP	-			
2810	32.07	kd	CGS001-2877	GPX2	-			
2811	32.03	kd	CGS001-23077	MYCBP2	-			
2812	32.03	kd	CGS001-11004	KIF2C	Kinesins			
2813	31.97	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
2814	31.96	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
2815	31.92	oe	ccsbBroad304_07478	CCP110	-			
2816	31.91	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
2817	31.85	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
2818	31.85	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
2819	31.83	kd	CGS001-7090	TLE3	WD repeat domain containing			
2820	31.81	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
2821	31.78	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
2822	31.74	oe	ccsbBroad304_06180	ESD	-			
2823	31.74	kd	CGS001-2956	MSH6	-			
2824	31.73	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
2825	31.71	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
2826	31.7	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
2827	31.68	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
2828	31.67	kd	CGS001-22938	SNW1	-			
2829	31.66	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
2830	31.62	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
2831	31.58	oe	ccsbBroad304_01760	USP1	Ubiquitin-specific peptidases			
2832	31.58	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
2833	31.5	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
2834	31.48	oe	ccsbBroad304_01165	PDK1	-			
2835	31.43	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
2836	31.43	kd	CGS001-22978	NT5C2	Adenosine turnover			
2837	31.38	kd	CGS001-23378	RRP8	-			
2838	31.35	oe	ccsbBroad304_04655	TRIM9	-			
2839	31.34	kd	CGS001-59286	UBL5	-			
2840	31.34	kd	CGS001-5004	ORM1	Lipocalins			
2841	31.32	kd	CGS001-53632	PRKAG3	AMPK subfamily			
2842	31.3	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
2843	31.25	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
2844	31.25	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
2845	31.24	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
2846	31.23	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
2847	31.21	kd	CGS001-664	BNIP3	-			
2848	31.19	kd	CGS001-3456	IFNB1	Interferons			
2849	31.12	oe	ccsbBroad304_00725	HADHA	-			
2850	31.09	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
2851	31.06	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
2852	31	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
2853	31	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
2854	30.99	kd	CGS001-11157	LSM6	-			
2855	30.97	oe	ccsbBroad304_06523	LIG1	-			
2856	30.91	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
2857	30.9	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
2858	30.88	oe	ccsbBroad304_05937	CASP7	Caspases			
2859	30.83	kd	CGS001-10736	SIX2	Homeoboxes / SINE class			
2860	30.81	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
2861	30.79	kd	CGS001-5053	PAH	Amino acid hydroxylases			
2862	30.75	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
2863	30.75	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
2864	30.75	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
2865	30.73	kd	CGS001-6856	SYPL1	-			
2866	30.6	kd	CGS001-84722	PSRC1	-			
2867	30.58	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
2868	30.47	kd	CGS001-4836	NMT1	-			
2869	30.46	cc		Tachykinin antagonist	-			
2870	30.45	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
2871	30.43	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
2872	30.4	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
2873	30.38	kd	CGS001-147179	WIPF2	-			
2874	30.37	kd	CGS001-708	C1QBP	-			
2875	30.32	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
2876	30.32	kd	CGS001-6469	SHH	-			
2877	30.29	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
2878	30.29	kd	CGS001-23492	CBX7	-			
2879	30.2	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
2880	30.2	kd	CGS001-29883	CNOT7	-			
2881	30.19	kd	CGS001-54205	CYCS	-			
2882	30.18	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
2883	30.17	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
2884	30.15	oe	ccsbBroad304_06174	ERCC1	-			
2885	30.04	kd	CGS001-6723	SRM	-			
2886	30.04	kd	CGS001-861	RUNX1	-			
2887	30.02	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
2888	30	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
2889	30	kd	CGS001-11164	NUDT5	Nudix motif containing			
2890	29.99	kd	CGS001-2295	FOXF2	Forkhead boxes			
2891	29.97	oe	ccsbBroad304_09281	TPD52L3	-			
2892	29.95	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
2893	29.93	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
2894	29.92	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
2895	29.92	kd	CGS001-4804	NGFR	Tumour necrosis factor (TNF) receptor family			
2896	29.87	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
2897	29.87	kd	CGS001-1840	DTX1	-			
2898	29.86	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
2899	29.86	oe	ccsbBroad304_07219	CDC7	CDC7 family			
2900	29.81	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
2901	29.78	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
2902	29.76	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
2903	29.76	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
2904	29.75	kd	CGS001-55703	POLR3B	RNA polymerase subunits			
2905	29.66	oe	ccsbBroad304_01333	PTGFR	GPCR / Class A : Prostanoid receptors			
2906	29.63	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
2907	29.51	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
2908	29.5	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
2909	29.5	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
2910	29.47	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2911	29.45	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
2912	29.44	kd	CGS001-1105	CHD1	-			
2913	29.38	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
2914	29.38	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
2915	29.37	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
2916	29.35	oe	ccsbBroad304_02565	RALBP1	-			
2917	29.32	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
2918	29.32	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
2919	29.29	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
2920	29.25	kd	CGS001-4811	NID1	-			
2921	29.23	kd	CGS001-2697	GJA1	Ion channels / Gap junction proteins (connexins)			
2922	29.22	oe	ccsbBroad304_07922	TRIM29	-			
2923	29.2	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
2924	29.18	kd	CGS001-10827	FAM114A2	-			
2925	29.17	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
2926	29.15	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2927	29.12	cp	BRD-A74907996	equol	Estrogen receptor agonist		ESR2, ESR1	Estrogen receptor agonist
2928	29.1	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
2929	29.04	kd	CGS001-1154	CISH	SH2 domain containing			
2930	29.02	oe	ccsbBroad304_02100	BUB3	WD repeat domain containing			
2931	29.01	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
2932	28.98	kd	CGS001-51734	SEPX1	-			
2933	28.93	oe	ccsbBroad304_06462	ITGAE	Integrins			
2934	28.92	kd	CGS001-545	ATR	ATR subfamily			
2935	28.91	oe	ccsbBroad304_03047	BZW2	-			
2936	28.9	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
2937	28.89	cc		Lysine acetyltransferases LOF	-			
2938	28.89	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
2939	28.83	oe	ccsbBroad304_08426	TEX10	-			
2940	28.83	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2941	28.78	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
2942	28.72	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
2943	28.71	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
2944	28.69	cc		GPCR Subset GOF	-			
2945	28.69	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
2946	28.67	kd	CGS001-55620	STAP2	-			
2947	28.63	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
2948	28.62	oe	ccsbBroad304_03239	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2949	28.59	kd	CGS001-1128	CHRM1	Cholinergic receptors			
2950	28.55	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
2951	28.55	kd	CGS001-57018	CCNL1	-			
2952	28.49	kd	CGS001-8525	DGKZ	-			
2953	28.45	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
2954	28.43	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
2955	28.4	kd	CGS001-10497	UNC13B	-			
2956	28.33	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
2957	28.32	oe	ccsbBroad304_03112	NENF	-			
2958	28.32	kd	CGS001-5106	PCK2	-			
2959	28.32	kd	CGS001-11116	FGFR1OP	-			
2960	28.32	kd	CGS001-8872	CDC123	-			
2961	28.32	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
2962	28.3	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
2963	28.29	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
2964	28.27	kd	CGS001-55191	NADSYN1	-			
2965	28.22	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
2966	28.2	oe	ccsbBroad304_02378	STUB1	Tetratricopeptide (TTC) repeat domain containing			
2967	28.19	kd	CGS001-54407	SLC38A2	System A-like transporters			
2968	28.18	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
2969	28.18	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
2970	28.18	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
2971	28.13	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
2972	28.12	kd	CGS001-8295	TRRAP	TRRAP subfamily			
2973	28.1	kd	CGS001-7466	WFS1	-			
2974	28.09	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
2975	28.09	kd	CGS001-4795	NFKBIL1	-			
2976	28.01	kd	CGS001-22794	CASC3	-			
2977	27.97	oe	ccsbBroad304_00949	LRPAP1	-			
2978	27.95	cc		Dihydrofolate reductase inhibitor	-			
2979	27.93	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
2980	27.9	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
2981	27.84	oe	ccsbBroad304_01960	CASK	CASK family			
2982	27.8	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
2983	27.79	kd	CGS001-6009	RHEB	-			
2984	27.75	oe	ccsbBroad304_02467	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
2985	27.75	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
2986	27.72	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
2987	27.68	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
2988	27.61	cc		MDM inhibitor	-			
2989	27.55	oe	ccsbBroad304_04490	RSPH1	-			
2990	27.55	kd	CGS001-790	CAD	-			
2991	27.54	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
2992	27.5	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
2993	27.49	kd	CGS001-350	APOH	Apolipoproteins			
2994	27.47	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
2995	27.46	oe	ccsbBroad304_00447	DLD	-			
2996	27.46	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
2997	27.45	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
2998	27.4	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
2999	27.38	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
3000	27.3	cc		Bacterial cell wall synthesis inhibitor	-			
3001	27.23	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
3002	27.18	oe	ccsbBroad304_03311	EVL	-			
3003	27.18	kd	CGS001-283	ANG	Ribonucleases, RNase A			
3004	27.12	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
3005	27.07	kd	CGS001-54861	SNRK	SNRK subfamily			
3006	27.02	oe	ccsbBroad304_00817	IDH2	-			
3007	27.02	kd	CGS001-8634	RTCD1	-			
3008	26.99	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3009	26.95	kd	CGS001-5708	PSMD2	Proteasome subunits			
3010	26.94	kd	CGS001-8801	SUCLG2	-			
3011	26.93	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
3012	26.92	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
3013	26.9	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3014	26.89	oe	ccsbBroad304_00510	EPHX2	-			
3015	26.89	kd	CGS001-57026	PDXP	-			
3016	26.87	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
3017	26.87	kd	CGS001-57157	PHTF2	-			
3018	26.8	kd	CGS001-5306	PITPNA	-			
3019	26.79	oe	ccsbBroad304_07320	SQSTM1	-			
3020	26.77	oe	ccsbBroad304_00262	CD59	CD molecules			
3021	26.69	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
3022	26.65	kd	CGS001-6827	SUPT4H1	-			
3023	26.58	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
3024	26.56	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
3025	26.56	oe	ccsbBroad304_07292	TNFSF13	CD molecules			
3026	26.53	oe	ccsbBroad304_01538	SKP2	F-boxes / Leucine-rich repeats			
3027	26.52	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
3028	26.41	oe	ccsbBroad304_04616	ORMDL3	-			
3029	26.35	oe	ccsbBroad304_01724	TTR	-			
3030	26.24	oe	ccsbBroad304_10758	CTBP2	-			
3031	26.23	kd	CGS001-4817	NIT1	-			
3032	26.21	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
3033	26.21	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
3034	26.14	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
3035	26.11	kd	CGS001-3988	LIPA	-			
3036	26.1	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
3037	26.02	oe	ccsbBroad304_04257	SPRY4	-			
3038	25.99	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
3039	25.97	kd	CGS001-7477	WNT7B	Endogenous ligands			
3040	25.96	oe	ccsbBroad304_01087	NF2	A-kinase anchor proteins			
3041	25.83	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
3042	25.8	oe	ccsbBroad304_02831	SGK3	SGK family			
3043	25.8	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
3044	25.71	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
3045	25.67	kd	CGS001-58528	RRAGD	-			
3046	25.53	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
3047	25.51	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
3048	25.47	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
3049	25.46	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
3050	25.46	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
3051	25.44	oe	ccsbBroad304_03235	TUBD1	Tubulins			
3052	25.44	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
3053	25.37	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
3054	25.34	kd	CGS001-29888	STRN4	WD repeat domain containing			
3055	25.29	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
3056	25.29	kd	CGS001-3949	LDLR	Low density lipoprotein receptors			
3057	25.21	kd	CGS001-3421	IDH3G	-			
3058	25.21	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
3059	25.17	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
3060	25.15	oe	ccsbBroad304_01394	RFX4	-			
3061	25.1	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
3062	25.09	oe	ccsbBroad304_05981	CDO1	-			
3063	25.06	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
3064	25.03	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
3065	24.96	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
3066	24.93	kd	CGS001-54498	SMOX	-			
3067	24.91	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
3068	24.89	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
3069	24.87	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
3070	24.84	oe	ccsbBroad304_06663	OAS1	-			
3071	24.82	oe	ccsbBroad304_08511	RFK	-			
3072	24.8	kd	CGS001-255877	BCL6B	BTB/POZ domain containing			
3073	24.78	oe	ccsbBroad304_06648	CNOT3	-			
3074	24.78	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
3075	24.68	kd	CGS001-89766	UMODL1	-			
3076	24.53	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
3077	24.51	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
3078	24.27	oe	ccsbBroad304_06264	GBP2	-			
3079	24.23	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
3080	24.23	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
3081	24.19	kd	CGS001-3636	INPPL1	Inositol polyphosphate phosphatases			
3082	24.19	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
3083	24.13	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
3084	24.02	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
3085	24	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
3086	23.98	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
3087	23.98	kd	CGS001-571	BACH1	BTB/POZ domain containing			
3088	23.91	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
3089	23.91	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
3090	23.88	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
3091	23.86	kd	CGS001-4069	LYZ	-			
3092	23.85	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
3093	23.81	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
3094	23.79	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
3095	23.73	oe	ccsbBroad304_01977	AOC3	Oxidoreductases			
3096	23.71	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
3097	23.55	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
3098	23.41	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
3099	23.4	oe	ccsbBroad304_03119	C16ORF5	-			
3100	23.38	oe	ccsbBroad304_04379	LZIC	-			
3101	23.36	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
3102	23.36	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
3103	23.33	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
3104	23.28	kd	CGS001-5110	PCMT1	-			
3105	23.27	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
3106	23.24	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
3107	23.19	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
3108	23.16	kd	CGS001-55379	LRRC59	-			
3109	23.11	oe	ccsbBroad304_06365	HIF1A	Basic helix-loop-helix proteins			
3110	23.1	kd	CGS001-6829	SUPT5H	-			
3111	23.08	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
3112	23.08	kd	CGS001-317705	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
3113	23.06	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
3114	23.05	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
3115	23.04	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
3116	22.97	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
3117	22.97	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3118	22.95	oe	ccsbBroad304_02460	ATG7	Ubiquitin-like modifier activating enzymes			
3119	22.89	kd	CGS001-205	AK4	Adenylate kinases			
3120	22.86	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
3121	22.74	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
3122	22.7	kd	CGS001-8313	AXIN2	-			
3123	22.68	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
3124	22.61	cc		Androgen receptor modulator	-			
3125	22.47	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
3126	22.38	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
3127	22.17	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
3128	22.12	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
3129	22.1	kd	CGS001-3242	HPD	Oxidoreductases			
3130	22.09	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
3131	22.07	kd	CGS001-80204	FBXO11	Protein arginine N-methyltransferases			
3132	21.93	kd	CGS001-8826	IQGAP1	-			
3133	21.92	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3134	21.9	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
3135	21.81	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
3136	21.73	kd	CGS001-2592	GALT	-			
3137	21.67	cc		PDGFR/KIT inhibitor	-			
3138	21.62	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
3139	21.6	kd	CGS001-154197	PNLDC1	-			
3140	21.47	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
3141	21.43	cc		Rho associated kinase inhibitor	-			
3142	21.37	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
3143	21.36	kd	CGS001-38	ACAT1	Lanosterol biosynthesis pathway			
3144	21.32	kd	CGS001-3725	JUN	basic leucine zipper proteins			
3145	21.27	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
3146	21.25	kd	CGS001-6776	STAT5A	SH2 domain containing			
3147	21.21	kd	CGS001-9232	PTTG1	-			
3148	21.21	kd	CGS001-23464	GCAT	-			
3149	21.08	cc		Akt Signaling LOF	-			
3150	21.01	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
3151	20.99	kd	CGS001-1643	DDB2	WD repeat domain containing			
3152	20.95	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
3153	20.95	kd	CGS001-144811	LACC1	-			
3154	20.82	kd	CGS001-100	ADA	Adenosine turnover			
3155	20.73	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
3156	20.62	kd	CGS001-2002	ELK1	ETS Transcription Factors			
3157	20.56	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3158	20.49	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
3159	20.24	kd	CGS001-388677	NOTCH2NL	-			
3160	20.18	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
3161	20.06	oe	ccsbBroad304_00606	GABPB1	Ankyrin repeat domain containing			
3162	19.97	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
3163	19.94	oe	ccsbBroad304_00966	MAFG	-			
3164	19.9	kd	CGS001-29775	CARD10	-			
3165	19.78	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
3166	19.61	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
3167	19.55	oe	ccsbBroad304_09774	ZNF92	Zinc fingers, C2H2-type			
3168	19.53	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
3169	19.53	kd	CGS001-5498	PPOX	-			
3170	19.51	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
3171	19.49	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
3172	19.44	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
3173	19.23	oe	ccsbBroad304_01091	NFIB	-			
3174	19.2	cc		PKA inhibitor	-			
3175	19.2	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
3176	19.19	oe	ccsbBroad304_04775	NTAN1	-			
3177	19.01	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
3178	18.92	kd	CGS001-10198	MPHOSPH9	-			
3179	18.89	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
3180	18.87	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
3181	18.84	oe	ccsbBroad304_05745	CD24	CD molecules			
3182	18.84	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
3183	18.62	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
3184	18.59	kd	CGS001-1981	EIF4G1	Parkinson disease			
3185	18.56	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
3186	18.51	kd	CGS001-3685	ITGAV	Integrins			
3187	18.4	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
3188	18.11	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
3189	17.94	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
3190	17.92	kd	CGS001-7187	TRAF3	-			
3191	17.84	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
3192	17.83	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
3193	17.82	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
3194	17.66	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
3195	17.59	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
3196	17.48	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
3197	17.47	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
3198	17.38	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
3199	17.29	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
3200	17.23	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
3201	17.13	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
3202	16.96	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
3203	16.96	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
3204	16.96	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
3205	16.91	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
3206	16.77	kd	CGS001-54957	TXNL4B	-			
3207	16.57	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
3208	16.47	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
3209	16.37	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
3210	16.26	kd	CGS001-9156	EXO1	-			
3211	16.09	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
3212	16.02	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
3213	15.71	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
3214	15.71	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
3215	15.71	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
3216	15.7	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
3217	15.67	kd	CGS001-8743	TNFSF10	CD molecules			
3218	15.59	cc		Wnt family GOF	-			
3219	15.57	kd	CGS001-2957	GTF2A1	General transcription factors			
3220	15.51	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
3221	15.45	oe	ccsbBroad304_04534	HN1L	-			
3222	15.42	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
3223	15.38	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
3224	15.37	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
3225	15.36	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
3226	15.26	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
3227	14.92	cc		PPAR receptor agonist	-			
3228	14.79	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
3229	14.73	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
3230	14.62	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
3231	14.42	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
3232	14.3	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
3233	14.3	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
3234	14.21	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
3235	13.93	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
3236	13.42	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
3237	13.33	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
3238	13.19	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
3239	13.08	cc		RNA Polymerase Enzymes LOF	-			
3240	13.02	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
3241	12.82	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
3242	12.65	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
3243	12.63	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
3244	12.35	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
3245	12.2	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
3246	12.2	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
3247	12.19	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
3248	11.81	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
3249	11.41	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
3250	11.13	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
3251	11.03	cc		Imidazoline ligand	-			
3252	10.79	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
3253	10.75	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
3254	10.51	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3255	10.49	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
3256	10	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
3257	9.24	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
3258	9.18	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
3259	8.72	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
3260	8.3	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
3261	6.6	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
3262	6	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
3263	5.76	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
3264	-6.8	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
3265	-7.07	cc		JAK inhibitor	-			
3266	-7.28	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
3267	-7.79	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
3268	-8.35	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
3269	-8.62	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
3270	-8.87	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
3271	-8.96	kd	CGS001-3479	IGF1	Endogenous ligands			
3272	-9.69	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
3273	-9.69	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
3274	-11.11	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
3275	-11.19	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
3276	-11.49	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
3277	-11.61	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
3278	-11.61	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3279	-11.63	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
3280	-11.7	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
3281	-11.8	cc		DNA Replication LOF	-			
3282	-11.96	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
3283	-12.28	kd	CGS001-5979	RET	Type XIV RTKs: RET			
3284	-12.46	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
3285	-12.55	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
3286	-12.65	cc		Mediator complex LOF	-			
3287	-12.7	cc		P38 MAPK inhibitor	-			
3288	-12.77	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
3289	-12.8	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
3290	-13.08	kd	CGS001-50808	AK3	-			
3291	-13.1	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3292	-13.25	kd	CGS001-23462	HEY1	Basic helix-loop-helix proteins			
3293	-13.29	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
3294	-13.38	cc		SRY LOF	-			
3295	-13.5	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
3296	-13.54	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
3297	-13.61	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
3298	-13.86	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
3299	-13.93	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
3300	-14.28	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
3301	-14.41	oe	ccsbBroad304_00799	HSP90AB1	Heat shock proteins / HSPC			
3302	-14.7	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
3303	-14.78	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
3304	-14.86	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
3305	-14.89	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
3306	-14.91	cc		Cannabinoid receptor agonist	-			
3307	-14.94	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
3308	-14.98	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
3309	-15.1	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3310	-15.24	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
3311	-15.34	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
3312	-15.38	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
3313	-15.45	cp	BRD-K15842202	eudesmic-acid	-666			-666
3314	-15.5	kd	CGS001-2588	GALNS	Arylsulfatase family			
3315	-15.52	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
3316	-15.74	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
3317	-15.74	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
3318	-15.77	kd	CGS001-9541	CIR1	-			
3319	-15.81	kd	CGS001-5202	PFDN2	-			
3320	-15.84	cc		MEK inhibitor	-			
3321	-15.85	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
3322	-15.89	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
3323	-16.09	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
3324	-16.1	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
3325	-16.13	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
3326	-16.25	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
3327	-16.32	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
3328	-16.39	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
3329	-16.5	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
3330	-16.55	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
3331	-16.57	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
3332	-16.76	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
3333	-16.82	kd	CGS001-4976	OPA1	-			
3334	-16.98	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
3335	-17.19	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
3336	-17.24	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3337	-17.38	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
3338	-17.38	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3339	-17.53	kd	CGS001-3065	HDAC1	Histone deacetylases			
3340	-17.62	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
3341	-17.66	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
3342	-17.92	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
3343	-17.99	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
3344	-18	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
3345	-18.07	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
3346	-18.09	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
3347	-18.12	oe	ccsbBroad304_06557	MAOA	Catecholamine turnover			
3348	-18.14	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
3349	-18.21	cc		NFkB pathway inhibitor	-			
3350	-18.24	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
3351	-18.31	kd	CGS001-2919	CXCL1	Endogenous ligands			
3352	-18.52	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
3353	-18.53	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
3354	-18.63	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
3355	-18.63	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
3356	-18.7	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
3357	-18.71	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
3358	-18.74	kd	CGS001-60493	FASTKD5	-			
3359	-18.78	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
3360	-18.84	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
3361	-18.88	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
3362	-18.88	kd	CGS001-1633	DCK	-			
3363	-18.97	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
3364	-19	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
3365	-19.04	kd	CGS001-7965	AIMP2	-			
3366	-19.16	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
3367	-19.17	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3368	-19.23	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
3369	-19.35	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
3370	-19.38	oe	ccsbBroad304_02452	NXF1	-			
3371	-19.49	kd	CGS001-513	ATP5D	ATPases / F-type			
3372	-19.49	oe	ccsbBroad304_00162	BIK	-			
3373	-19.58	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
3374	-19.62	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
3375	-19.79	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3376	-19.81	oe	ccsbBroad304_06370	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
3377	-19.83	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
3378	-19.84	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
3379	-19.9	kd	CGS001-1111	CHEK1	CHK1 subfamily			
3380	-19.9	oe	ccsbBroad304_06140	EEF1D	-			
3381	-19.93	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
3382	-19.97	oe	ccsbBroad304_00054	ALDOC	-			
3383	-20	kd	CGS001-10314	LANCL1	-			
3384	-20.04	cc		Progesterone receptor agonist	-			
3385	-20.06	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
3386	-20.13	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
3387	-20.15	kd	CGS001-7504	XK	Blood group antigens			
3388	-20.16	kd	CGS001-10544	PROCR	CD molecules			
3389	-20.19	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
3390	-20.22	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
3391	-20.24	cc		IGF-1 inhibitor	-			
3392	-20.48	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
3393	-20.5	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
3394	-20.51	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3395	-20.58	kd	CGS001-10078	TSSC4	-			
3396	-20.6	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
3397	-20.68	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
3398	-20.71	kd	CGS001-166647	GPR125	Adhesion Class GPCRs			
3399	-20.84	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
3400	-20.93	kd	CGS001-27125	AFF4	-			
3401	-20.94	kd	CGS001-6201	RPS7	S ribosomal proteins			
3402	-20.97	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
3403	-20.98	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
3404	-21.01	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
3405	-21.02	oe	ccsbBroad304_06040	CRY1	-			
3406	-21.04	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
3407	-21.05	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3408	-21.09	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
3409	-21.11	kd	CGS001-3171	FOXA3	Forkhead boxes			
3410	-21.18	oe	ccsbBroad304_09833	SENP5	-			
3411	-21.22	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3412	-21.26	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
3413	-21.31	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
3414	-21.35	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
3415	-21.41	oe	ccsbBroad304_06035	CRABP1	Fatty acid-binding proteins			
3416	-21.42	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
3417	-21.45	kd	CGS001-5688	PSMA7	Proteasome subunits			
3418	-21.51	oe	ccsbBroad304_00856	CXCR2	Chemokine receptors			
3419	-21.52	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
3420	-21.52	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
3421	-21.54	oe	ccsbBroad304_02497	YKT6	-			
3422	-21.55	oe	ccsbBroad304_01327	PSPH	-			
3423	-21.59	kd	CGS001-4931	NVL	ATPases / AAA-type			
3424	-21.6	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
3425	-21.64	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
3426	-21.64	kd	CGS001-23647	ARFIP2	-			
3427	-21.65	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
3428	-21.73	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
3429	-21.74	cc		FLT3 inhibitor	-			
3430	-21.77	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
3431	-21.8	oe	ccsbBroad304_01401	RIT1	-			
3432	-21.83	kd	CGS001-1036	CDO1	-			
3433	-21.85	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
3434	-21.89	kd	CGS001-122402	TDRD9	Tudor domain containing			
3435	-21.9	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
3436	-21.93	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
3437	-21.93	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
3438	-21.96	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
3439	-22	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
3440	-22.04	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
3441	-22.09	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
3442	-22.13	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
3443	-22.13	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3444	-22.13	kd	CGS001-11232	POLG2	DNA polymerases			
3445	-22.15	oe	ccsbBroad304_01527	SGK1	SGK family			
3446	-22.15	kd	CGS001-662	BNIP1	-			
3447	-22.16	oe	ccsbBroad304_06178	ERCC5	-			
3448	-22.19	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
3449	-22.35	oe	ccsbBroad304_07754	FGFR1OP	-			
3450	-22.36	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
3451	-22.41	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
3452	-22.41	kd	CGS001-54584	GNB1L	WD repeat domain containing			
3453	-22.42	kd	CGS001-51727	CMPK1	-			
3454	-22.42	kd	CGS001-966	CD59	CD molecules			
3455	-22.43	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
3456	-22.44	kd	CGS001-10923	SUB1	-			
3457	-22.48	kd	CGS001-2072	ERCC4	-			
3458	-22.55	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
3459	-22.59	oe	ccsbBroad304_03186	GMNN	-			
3460	-22.61	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
3461	-22.63	oe	ccsbBroad304_07012	STK3	MST subfamily			
3462	-22.7	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
3463	-22.73	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
3464	-22.84	cc		Aminoacyl tRNA synthetases class II LOF	-			
3465	-22.85	kd	CGS001-10214	SSX3	-			
3466	-22.86	kd	CGS001-2878	GPX3	-			
3467	-22.89	kd	CGS001-5894	RAF1	RAF family			
3468	-22.97	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3469	-22.97	kd	CGS001-55644	OSGEP	-			
3470	-22.99	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
3471	-23.02	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
3472	-23.04	oe	ccsbBroad304_07843	FCHO1	-			
3473	-23.04	kd	CGS001-271	AMPD2	-			
3474	-23.07	cc		Angiotensin receptor antagonist	-			
3475	-23.11	kd	CGS001-5245	PHB	-			
3476	-23.12	kd	CGS001-4221	MEN1	-			
3477	-23.2	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
3478	-23.2	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
3479	-23.21	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
3480	-23.23	oe	ccsbBroad304_08461	CDCA4	-			
3481	-23.23	oe	ccsbBroad304_06836	RAD23B	-			
3482	-23.23	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
3483	-23.24	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
3484	-23.25	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
3485	-23.28	kd	CGS001-4907	NT5E	Adenosine turnover			
3486	-23.29	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
3487	-23.32	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
3488	-23.33	kd	CGS001-5562	PRKAA1	AMPK subfamily			
3489	-23.36	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
3490	-23.44	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
3491	-23.47	kd	CGS001-23509	POFUT1	Fucosyltransferases			
3492	-23.47	kd	CGS001-375449	MAST4	MAST family			
3493	-23.54	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3494	-23.6	kd	CGS001-169436	C9ORF96	-			
3495	-23.61	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
3496	-23.62	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
3497	-23.64	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
3498	-23.65	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
3499	-23.69	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
3500	-23.71	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
3501	-23.73	kd	CGS001-6611	SMS	-			
3502	-23.75	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
3503	-23.78	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
3504	-23.89	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
3505	-23.92	kd	CGS001-10105	PPIF	-			
3506	-23.94	kd	CGS001-2197	FAU	S ribosomal proteins			
3507	-23.94	kd	CGS001-335	APOA1	Apolipoproteins			
3508	-23.97	oe	ccsbBroad304_00837	IGFBP4	insulin-like growth factor (IGF) binding proteins			
3509	-24.04	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
3510	-24.05	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
3511	-24.07	oe	ccsbBroad304_04649	ADC	-			
3512	-24.08	kd	CGS001-7832	BTG2	-			
3513	-24.15	kd	CGS001-9131	AIFM1	-			
3514	-24.17	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
3515	-24.17	kd	CGS001-8804	CREG1	-			
3516	-24.18	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
3517	-24.22	oe	ccsbBroad304_05757	ACADS	-			
3518	-24.22	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
3519	-24.22	kd	CGS001-64858	DCLRE1B	-			
3520	-24.25	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
3521	-24.27	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
3522	-24.31	oe	ccsbBroad304_00430	GADD45A	-			
3523	-24.31	kd	CGS001-7020	TFAP2A	-			
3524	-24.34	oe	ccsbBroad304_03264	UBAP1	-			
3525	-24.45	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
3526	-24.48	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
3527	-24.49	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
3528	-24.49	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
3529	-24.54	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
3530	-24.54	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
3531	-24.55	kd	CGS001-1312	COMT	Catecholamine turnover			
3532	-24.57	kd	CGS001-29116	MYLIP	-			
3533	-24.62	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
3534	-24.63	oe	ccsbBroad304_01372	RALB	-			
3535	-24.63	kd	CGS001-11198	SUPT16H	-			
3536	-24.64	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
3537	-24.69	oe	ccsbBroad304_07491	IP6K1	-			
3538	-24.69	oe	ccsbBroad304_04786	CANT1	-			
3539	-24.71	kd	CGS001-5002	SLC22A18	Orphan or poorly characterized SLC22 family members			
3540	-24.75	kd	CGS001-23030	KDM4B	Histone demethylases			
3541	-24.76	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
3542	-24.79	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
3543	-24.87	kd	CGS001-4245	MGAT1	-			
3544	-24.9	oe	ccsbBroad304_02109	XPR1	-			
3545	-24.91	kd	CGS001-6774	STAT3	SH2 domain containing			
3546	-24.93	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
3547	-24.99	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
3548	-25	kd	CGS001-91304	C19ORF6	-			
3549	-25.04	oe	ccsbBroad304_02012	FADD	-			
3550	-25.09	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
3551	-25.09	oe	ccsbBroad304_00811	ICAM1	CD molecules			
3552	-25.11	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
3553	-25.12	oe	ccsbBroad304_04541	ZNF502	Zinc fingers, C2H2-type			
3554	-25.12	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3555	-25.12	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
3556	-25.15	kd	CGS001-23131	GPATCH8	G patch domain containing			
3557	-25.2	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
3558	-25.21	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
3559	-25.21	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
3560	-25.23	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
3561	-25.26	kd	CGS001-8669	EIF3J	-			
3562	-25.27	kd	CGS001-3159	HMGA1	High-mobility group / Canonical			
3563	-25.27	oe	ccsbBroad304_01326	PSME1	Proteasome (prosome, macropain) subunits			
3564	-25.28	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
3565	-25.29	kd	CGS001-5690	PSMB2	Proteasome subunits			
3566	-25.31	kd	CGS001-8467	SMARCA5	-			
3567	-25.33	oe	ccsbBroad304_06916	SCP2	-			
3568	-25.35	oe	ccsbBroad304_04054	PHF23	Zinc fingers, PHD-type			
3569	-25.35	kd	CGS001-10482	NXF1	-			
3570	-25.36	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
3571	-25.38	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
3572	-25.47	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
3573	-25.47	kd	CGS001-1028	CDKN1C	-			
3574	-25.49	kd	CGS001-5427	POLE2	DNA polymerases			
3575	-25.55	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
3576	-25.55	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
3577	-25.57	oe	ccsbBroad304_09503	KLHDC9	-			
3578	-25.57	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
3579	-25.58	kd	CGS001-5338	PLD2	Hydrolases			
3580	-25.6	kd	CGS001-3569	IL6	Interferons			
3581	-25.63	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
3582	-25.67	kd	CGS001-122618	PLD4	-			
3583	-25.68	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
3584	-25.68	kd	CGS001-4144	MAT2A	-			
3585	-25.71	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
3586	-25.72	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
3587	-25.72	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
3588	-25.75	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
3589	-25.77	kd	CGS001-9140	ATG12	-			
3590	-25.79	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
3591	-25.81	oe	ccsbBroad304_06367	HK1	-			
3592	-25.88	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
3593	-25.9	oe	ccsbBroad304_03696	C19ORF10	-			
3594	-25.9	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
3595	-25.91	oe	ccsbBroad304_13880	IDH3G	-			
3596	-25.92	kd	CGS001-57057	TBX20	T-boxes			
3597	-25.94	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
3598	-25.94	oe	ccsbBroad304_01641	TAF13	-			
3599	-25.97	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
3600	-25.99	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
3601	-26.02	kd	CGS001-4683	NBN	-			
3602	-26.05	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
3603	-26.05	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
3604	-26.08	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
3605	-26.11	kd	CGS001-351	APP	Endogenous ligands			
3606	-26.11	oe	ccsbBroad304_06683	FURIN	Subtilisin			
3607	-26.14	kd	CGS001-29982	NRBF2	-			
3608	-26.18	oe	ccsbBroad304_07173	ZNF202	Zinc fingers, C2H2-type			
3609	-26.2	oe	ccsbBroad304_06535	LPL	-			
3610	-26.23	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
3611	-26.3	oe	ccsbBroad304_03614	G2E3	Zinc fingers, PHD-type			
3612	-26.31	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
3613	-26.33	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
3614	-26.34	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
3615	-26.34	kd	CGS001-64428	NARFL	-			
3616	-26.37	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
3617	-26.43	cp	BRD-K65910366	KUC103904N	-666			-666
3618	-26.44	kd	CGS001-2203	FBP1	-			
3619	-26.45	oe	ccsbBroad304_01379	RBBP6	-			
3620	-26.48	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
3621	-26.52	oe	ccsbBroad304_02671	ECD	-			
3622	-26.55	oe	ccsbBroad304_06565	MB	-			
3623	-26.59	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3624	-26.62	oe	ccsbBroad304_06354	SERPIND1	Serine (or cysteine) peptidase inhibitors			
3625	-26.64	oe	ccsbBroad304_01605	SSX2	-			
3626	-26.64	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
3627	-26.65	kd	CGS001-10253	SPRY2	-			
3628	-26.66	kd	CGS001-51805	COQ3	-			
3629	-26.68	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3630	-26.72	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
3631	-26.8	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
3632	-26.8	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
3633	-26.82	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
3634	-26.84	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
3635	-26.91	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3636	-26.93	kd	CGS001-2274	FHL2	-			
3637	-26.95	oe	ccsbBroad304_00222	CASP6	Caspases			
3638	-26.95	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
3639	-26.98	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
3640	-26.99	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
3641	-27	oe	ccsbBroad304_02373	SPRY2	-			
3642	-27	oe	ccsbBroad304_00888	ITPK1	-			
3643	-27	kd	CGS001-388	RHOB	-			
3644	-27	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
3645	-27.02	kd	CGS001-3163	HMOX2	Haem oxygenase			
3646	-27.03	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
3647	-27.05	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
3648	-27.06	kd	CGS001-930	CD19	CD molecules			
3649	-27.1	oe	ccsbBroad304_06996	SRM	-			
3650	-27.14	oe	ccsbBroad304_07088	TP53	-			
3651	-27.15	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
3652	-27.25	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
3653	-27.27	kd	CGS001-4594	MUT	-			
3654	-27.28	kd	CGS001-1736	DKC1	-			
3655	-27.28	oe	ccsbBroad304_02853	QPCT	Aminopeptidase Y			
3656	-27.3	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
3657	-27.31	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
3658	-27.32	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
3659	-27.34	kd	CGS001-23028	KDM1A	Histone demethylase			
3660	-27.34	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
3661	-27.37	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3662	-27.41	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
3663	-27.41	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
3664	-27.48	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
3665	-27.49	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3666	-27.52	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
3667	-27.53	oe	ccsbBroad304_07024	SYK	Syk family			
3668	-27.54	oe	ccsbBroad304_03864	OVOL2	Zinc fingers, C2H2-type			
3669	-27.54	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
3670	-27.58	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
3671	-27.61	oe	ccsbBroad304_07528	DMTF1	-			
3672	-27.61	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
3673	-27.63	kd	CGS001-50943	FOXP3	Forkhead boxes			
3674	-27.65	kd	CGS001-10614	HEXIM1	-			
3675	-27.67	kd	CGS001-10657	KHDRBS1	-			
3676	-27.68	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
3677	-27.68	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
3678	-27.7	kd	CGS001-11136	SLC7A9	SLC7 family			
3679	-27.7	kd	CGS001-4651	MYO10	Pleckstrin homology (PH) domain containing			
3680	-27.76	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
3681	-27.79	kd	CGS001-9354	UBE4A	U-box domain containing			
3682	-27.86	kd	CGS001-23369	PUM2	-			
3683	-27.86	kd	CGS001-26227	PHGDH	-			
3684	-27.88	kd	CGS001-6788	STK3	MST subfamily			
3685	-27.92	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
3686	-27.93	oe	ccsbBroad304_07401	TXNL1	-			
3687	-27.95	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
3688	-27.95	kd	CGS001-2717	GLA	-			
3689	-27.97	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
3690	-27.98	kd	CGS001-3560	IL2RB	IL-2 receptor family			
3691	-28.02	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
3692	-28.05	oe	ccsbBroad304_00085	APRT	-			
3693	-28.06	oe	ccsbBroad304_02097	LPAR2	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
3694	-28.08	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
3695	-28.1	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
3696	-28.11	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
3697	-28.12	kd	CGS001-353	APRT	-			
3698	-28.13	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
3699	-28.14	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
3700	-28.16	oe	ccsbBroad304_08217	SCCPDH	-			
3701	-28.16	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
3702	-28.17	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
3703	-28.17	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
3704	-28.2	oe	ccsbBroad304_01398	RHEB	-			
3705	-28.21	oe	ccsbBroad304_03497	TXNL4B	-			
3706	-28.24	kd	CGS001-6632	SNRPD1	-			
3707	-28.27	oe	ccsbBroad304_01675	TK1	-			
3708	-28.29	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
3709	-28.33	kd	CGS001-65123	INTS3	-			
3710	-28.38	oe	ccsbBroad304_01483	SAT1	-			
3711	-28.41	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3712	-28.43	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
3713	-28.46	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
3714	-28.46	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
3715	-28.52	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
3716	-28.53	oe	ccsbBroad304_00070	ANXA5	Annexins			
3717	-28.54	kd	CGS001-4837	NNMT	-			
3718	-28.55	oe	ccsbBroad304_02510	CNPY3	Trinucleotide (CAG) repeat containing			
3719	-28.56	kd	CGS001-5167	ENPP1	-			
3720	-28.57	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
3721	-28.59	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
3722	-28.59	kd	CGS001-345611	IRGM	-			
3723	-28.59	oe	ccsbBroad304_03812	PBXIP1	-			
3724	-28.62	kd	CGS001-58533	SNX6	Sorting nexins			
3725	-28.65	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
3726	-28.69	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
3727	-28.7	kd	CGS001-427	ASAH1	Acid ceramidase			
3728	-28.71	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
3729	-28.73	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
3730	-28.75	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
3731	-28.79	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
3732	-28.82	kd	CGS001-63892	THADA	-			
3733	-28.85	kd	CGS001-8678	BECN1	-			
3734	-28.87	kd	CGS001-5300	PIN1	-			
3735	-28.9	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
3736	-28.93	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
3737	-28.94	oe	ccsbBroad304_08802	ELAC2	-			
3738	-28.94	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
3739	-28.97	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
3740	-29.02	oe	ccsbBroad304_00728	HBE1	-			
3741	-29.02	kd	CGS001-5198	PFAS	-			
3742	-29.03	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
3743	-29.07	kd	CGS001-7040	TGFB1	Endogenous ligands			
3744	-29.08	kd	CGS001-4439	MSH5	-			
3745	-29.09	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
3746	-29.12	oe	ccsbBroad304_07780	POLG2	DNA polymerases			
3747	-29.12	kd	CGS001-55206	SBNO1	-			
3748	-29.13	kd	CGS001-79073	TMEM109	-			
3749	-29.16	oe	ccsbBroad304_02738	RRS1	-			
3750	-29.18	oe	ccsbBroad304_00327	CLK2	CDC-like kinases			
3751	-29.19	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
3752	-29.23	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
3753	-29.25	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
3754	-29.28	kd	CGS001-5933	RBL1	-			
3755	-29.31	cc		Cyclin dependent kinases LOF	-			
3756	-29.33	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
3757	-29.36	kd	CGS001-8681	JMJD7-PLA2G4B	-			
3758	-29.36	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3759	-29.43	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
3760	-29.47	oe	ccsbBroad304_03089	PACSIN3	-			
3761	-29.48	kd	CGS001-2747	GLUD2	-			
3762	-29.51	kd	CGS001-56916	SMARCAD1	-			
3763	-29.52	oe	ccsbBroad304_07679	ZNF274	Zinc fingers, C2H2-type			
3764	-29.52	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
3765	-29.54	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
3766	-29.54	kd	CGS001-57048	PLSCR3	-			
3767	-29.55	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
3768	-29.56	oe	ccsbBroad304_03773	CIAPIN1	-			
3769	-29.61	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
3770	-29.64	kd	CGS001-9788	MTSS1	-			
3771	-29.66	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
3772	-29.71	kd	CGS001-51466	EVL	-			
3773	-29.75	kd	CGS001-80212	CCDC92	-			
3774	-29.76	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
3775	-29.76	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
3776	-29.76	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
3777	-29.79	kd	CGS001-5015	OTX2	Homeoboxes / PRD class			
3778	-29.8	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
3779	-29.84	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
3780	-29.86	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
3781	-29.87	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
3782	-29.88	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3783	-29.89	kd	CGS001-3821	KLRC1	CD molecules			
3784	-30.03	oe	ccsbBroad304_08602	HDAC8	Histone deacetylases			
3785	-30.04	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
3786	-30.05	kd	CGS001-149233	IL23R	IL-12 receptor family			
3787	-30.07	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
3788	-30.08	oe	ccsbBroad304_07045	TEAD4	-			
3789	-30.1	oe	ccsbBroad304_03118	NRBP1	NRBP family			
3790	-30.13	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
3791	-30.18	oe	ccsbBroad304_01351	PEX19	-			
3792	-30.21	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
3793	-30.23	kd	CGS001-634	CEACAM1	CD molecules			
3794	-30.24	oe	ccsbBroad304_10212	GRHL3	-			
3795	-30.24	oe	ccsbBroad304_03641	ASF1B	-			
3796	-30.25	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
3797	-30.28	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
3798	-30.33	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
3799	-30.33	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
3800	-30.35	kd	CGS001-9988	DMTF1	-			
3801	-30.36	kd	CGS001-23621	BACE1	Pepsin			
3802	-30.37	oe	ccsbBroad304_02857	BAMBI	-			
3803	-30.38	kd	CGS001-80314	EPC1	-			
3804	-30.42	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
3805	-30.46	oe	ccsbBroad304_06144	EFNB3	Ephrins			
3806	-30.57	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
3807	-30.58	oe	ccsbBroad304_06954	SLC1A1	Glutamate transporter subfamily			
3808	-30.58	kd	CGS001-8192	CLPP	ATPases / AAA-type			
3809	-30.62	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
3810	-30.63	kd	CGS001-6258	RXRG	Retinoid X receptors			
3811	-30.64	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
3812	-30.65	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
3813	-30.65	kd	CGS001-170302	ARX	Homeoboxes / PRD class			
3814	-30.66	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
3815	-30.68	kd	CGS001-8807	IL18RAP	CD molecules			
3816	-30.68	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
3817	-30.69	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
3818	-30.69	oe	ccsbBroad304_07531	TANK	-			
3819	-30.71	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
3820	-30.79	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
3821	-30.83	kd	CGS001-3579	CXCR2	Chemokine receptors			
3822	-30.84	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
3823	-30.86	kd	CGS001-7018	TF	-			
3824	-30.89	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
3825	-30.9	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
3826	-30.93	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
3827	-30.94	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
3828	-30.96	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
3829	-30.98	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
3830	-30.98	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
3831	-31.01	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
3832	-31.02	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
3833	-31.04	oe	ccsbBroad304_03232	VPS28	-			
3834	-31.04	kd	CGS001-2673	GFPT1	-			
3835	-31.04	kd	CGS001-55793	FAM63A	-			
3836	-31.04	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
3837	-31.06	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
3838	-31.07	kd	CGS001-7263	TST	-			
3839	-31.07	kd	CGS001-10174	SORBS3	-			
3840	-31.09	oe	ccsbBroad304_01832	PAX8	Paired boxes			
3841	-31.09	kd	CGS001-1604	CD55	CD molecules			
3842	-31.11	kd	CGS001-10681	GNB5	WD repeat domain containing			
3843	-31.12	kd	CGS001-11168	PSIP1	-			
3844	-31.14	kd	CGS001-10513	APPBP2	-			
3845	-31.16	oe	ccsbBroad304_03164	MTERFD1	-			
3846	-31.18	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
3847	-31.19	oe	ccsbBroad304_08023	EIF2C1	-			
3848	-31.19	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3849	-31.19	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
3850	-31.2	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
3851	-31.2	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
3852	-31.21	kd	CGS001-5479	PPIB	-			
3853	-31.22	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
3854	-31.22	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
3855	-31.26	oe	ccsbBroad304_08898	TRAK2	-			
3856	-31.27	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
3857	-31.28	kd	CGS001-55214	LEPREL1	-			
3858	-31.29	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
3859	-31.3	oe	ccsbBroad304_01523	SRSF4	RNA binding motif (RRM) containing			
3860	-31.33	oe	ccsbBroad304_05936	CASP2	Caspases			
3861	-31.34	oe	ccsbBroad304_02596	KDELR3	-			
3862	-31.36	cc		HSP inhibitor	-			
3863	-31.36	kd	CGS001-7251	TSG101	-			
3864	-31.37	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
3865	-31.39	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
3866	-31.4	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
3867	-31.43	oe	ccsbBroad304_08660	SMARCAD1	-			
3868	-31.43	oe	ccsbBroad304_08645	BCCIP	-			
3869	-31.44	kd	CGS001-5362	PLXNA2	Plexins			
3870	-31.46	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
3871	-31.47	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
3872	-31.52	oe	ccsbBroad304_10846	GGT1	CD molecules			
3873	-31.53	kd	CGS001-9612	NCOR2	-			
3874	-31.55	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
3875	-31.57	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
3876	-31.57	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
3877	-31.6	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
3878	-31.62	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
3879	-31.65	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
3880	-31.67	kd	CGS001-84669	USP32	EF-hand domain containing			
3881	-31.67	kd	CGS001-2004	ELK3	ETS Transcription Factors			
3882	-31.68	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
3883	-31.69	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
3884	-31.71	oe	ccsbBroad304_00961	SMAD2	SMADs			
3885	-31.76	oe	ccsbBroad304_06278	GK	Glycerol kinases			
3886	-31.76	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
3887	-31.77	oe	ccsbBroad304_00523	EXT1	Exostosin glycosyltransferase family			
3888	-31.79	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
3889	-31.82	kd	CGS001-151126	ZNF385B	-			
3890	-31.85	oe	ccsbBroad304_01577	SOD1	-			
3891	-31.85	kd	CGS001-5727	PTCH1	-			
3892	-31.85	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
3893	-31.86	oe	ccsbBroad304_13975	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3894	-31.86	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3895	-31.87	cc		Sterol demethylase inhibitor	-			
3896	-31.89	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
3897	-31.91	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
3898	-31.91	kd	CGS001-11142	PKIG	-			
3899	-31.92	oe	ccsbBroad304_01976	EIF4EBP3	-			
3900	-31.92	kd	CGS001-83729	INHBE	-			
3901	-31.99	oe	ccsbBroad304_08596	EAPP	-			
3902	-32	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
3903	-32.05	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
3904	-32.09	oe	ccsbBroad304_00371	MAPK14	MAPK:p38 subfamily			
3905	-32.12	cc		Interleukins GOF	-			
3906	-32.12	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
3907	-32.13	oe	ccsbBroad304_02217	FEZ1	-			
3908	-32.15	kd	CGS001-1445	CSK	Csk family			
3909	-32.18	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
3910	-32.21	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
3911	-32.23	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
3912	-32.25	oe	ccsbBroad304_07277	RTCD1	-			
3913	-32.27	oe	ccsbBroad304_03728	DIABLO	-			
3914	-32.27	oe	ccsbBroad304_03732	NPDC1	-			
3915	-32.28	cc		NADH ubiquinone oxidoreductase core subunits GOF	-			
3916	-32.28	oe	ccsbBroad304_06094	DFFA	-			
3917	-32.28	oe	ccsbBroad304_01870	CHAF1B	WD repeat domain containing			
3918	-32.29	kd	CGS001-10617	STAMBP	-			
3919	-32.31	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
3920	-32.32	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
3921	-32.35	kd	CGS001-727	C5	Endogenous ligands			
3922	-32.36	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3923	-32.37	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
3924	-32.38	oe	ccsbBroad304_07137	WT1	Zinc fingers, C2H2-type			
3925	-32.4	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
3926	-32.41	oe	ccsbBroad304_07941	FBXO7	F-boxes / other			
3927	-32.43	kd	CGS001-6850	SYK	Syk family			
3928	-32.46	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
3929	-32.49	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
3930	-32.52	oe	ccsbBroad304_04544	RCCD1	-			
3931	-32.52	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
3932	-32.52	kd	CGS001-4853	NOTCH2	Ankyrin repeat domain containing			
3933	-32.53	kd	CGS001-4665	NAB2	-			
3934	-32.54	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
3935	-32.61	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
3936	-32.62	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
3937	-32.65	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
3938	-32.65	kd	CGS001-2114	ETS2	ETS Transcription Factors			
3939	-32.72	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
3940	-32.72	kd	CGS001-384	ARG2	Arginase			
3941	-32.73	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
3942	-32.75	oe	ccsbBroad304_07080	TM7SF2	-			
3943	-32.76	kd	CGS001-4905	NSF	ATPases / AAA-type			
3944	-32.76	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
3945	-32.77	oe	ccsbBroad304_00552	FEN1	-			
3946	-32.78	kd	CGS001-50846	DHH	-			
3947	-32.79	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
3948	-32.84	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
3949	-32.89	oe	ccsbBroad304_04683	ZNF689	Zinc fingers, C2H2-type			
3950	-32.89	oe	ccsbBroad304_05823	ANXA2	Annexins			
3951	-32.93	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
3952	-32.93	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
3953	-32.96	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
3954	-33.06	kd	CGS001-56922	MCCC1	-			
3955	-33.07	kd	CGS001-7185	TRAF1	-			
3956	-33.12	oe	ccsbBroad304_02553	BLCAP	-			
3957	-33.17	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
3958	-33.19	kd	CGS001-5887	RAD23B	-			
3959	-33.2	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
3960	-33.21	kd	CGS001-29911	HOOK2	-			
3961	-33.24	oe	ccsbBroad304_07888	CBX6	-			
3962	-33.27	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
3963	-33.31	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
3964	-33.33	kd	CGS001-535	ATP6V0A1	ATPases / V-type			
3965	-33.37	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
3966	-33.38	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
3967	-33.39	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
3968	-33.4	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
3969	-33.43	kd	CGS001-823	CAPN1	EF-hand domain containing			
3970	-33.46	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
3971	-33.46	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
3972	-33.47	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
3973	-33.48	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
3974	-33.49	oe	ccsbBroad304_01923	UXT	-			
3975	-33.54	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
3976	-33.6	oe	ccsbBroad304_01166	PDK2	PDHK family			
3977	-33.62	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
3978	-33.62	kd	CGS001-4864	NPC1	-			
3979	-33.63	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
3980	-33.63	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
3981	-33.65	cc		Glucocorticoid receptor agonist	-			
3982	-33.66	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
3983	-33.66	kd	CGS001-5909	RAP1GAP	-			
3984	-33.68	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
3985	-33.69	kd	CGS001-2356	FPGS	-			
3986	-33.74	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
3987	-33.79	oe	ccsbBroad304_03444	PAF1	-			
3988	-33.8	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
3989	-33.81	oe	ccsbBroad304_03859	ENOPH1	-			
3990	-33.82	kd	CGS001-5824	PEX19	-			
3991	-33.82	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
3992	-33.83	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
3993	-33.84	kd	CGS001-955	ENTPD6	-			
3994	-33.87	kd	CGS001-5170	PDPK1	PDK1 family			
3995	-33.87	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
3996	-33.89	oe	ccsbBroad304_00226	CAV1	-			
3997	-33.93	oe	ccsbBroad304_02110	VAPB	-			
3998	-33.93	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
3999	-33.94	kd	CGS001-6643	SNX2	Sorting nexins			
4000	-33.97	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4001	-34	kd	CGS001-10914	PAPOLA	-			
4002	-34.02	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
4003	-34.02	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
4004	-34.02	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
4005	-34.03	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
4006	-34.05	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
4007	-34.08	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
4008	-34.1	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
4009	-34.12	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
4010	-34.15	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
4011	-34.2	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
4012	-34.25	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
4013	-34.29	oe	ccsbBroad304_00710	GUSB	-			
4014	-34.31	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
4015	-34.32	oe	ccsbBroad304_06435	RBPJ	-			
4016	-34.33	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
4017	-34.36	kd	CGS001-6195	RPS6KA1	RSK subfamily			
4018	-34.37	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
4019	-34.39	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
4020	-34.4	kd	CGS001-10250	SRRM1	-			
4021	-34.41	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
4022	-34.42	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
4023	-34.43	kd	CGS001-10298	PAK4	PAKB subfamily			
4024	-34.45	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
4025	-34.45	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
4026	-34.48	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
4027	-34.49	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
4028	-34.49	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
4029	-34.53	kd	CGS001-5925	RB1	Endogenous ligands			
4030	-34.55	oe	ccsbBroad304_08102	MRPL18	Mitochondrial ribosomal proteins / large subunits			
4031	-34.55	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
4032	-34.56	kd	CGS001-5621	PRNP	CD molecules			
4033	-34.59	oe	ccsbBroad304_10882	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
4034	-34.64	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4035	-34.64	kd	CGS001-84515	MCM8	-			
4036	-34.65	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
4037	-34.65	kd	CGS001-9380	GRHPR	-			
4038	-34.67	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
4039	-34.67	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
4040	-34.69	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
4041	-34.72	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
4042	-34.75	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
4043	-34.79	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
4044	-34.8	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
4045	-34.86	oe	ccsbBroad304_09615	LACC1	-			
4046	-34.89	oe	ccsbBroad304_06845	RARRES3	-			
4047	-34.89	oe	ccsbBroad304_02349	MPHOSPH9	-			
4048	-34.91	oe	ccsbBroad304_01078	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
4049	-34.94	oe	ccsbBroad304_08694	TBX20	T-boxes			
4050	-34.94	kd	CGS001-29946	SERTAD3	-			
4051	-34.95	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
4052	-34.98	kd	CGS001-2621	GAS6	-			
4053	-35.06	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
4054	-35.09	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
4055	-35.1	kd	CGS001-84923	FAM104A	-			
4056	-35.11	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
4057	-35.12	kd	CGS001-6196	RPS6KA2	RSK subfamily			
4058	-35.12	kd	CGS001-10013	HDAC6	Histone deacetylases			
4059	-35.13	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4060	-35.16	oe	ccsbBroad304_01644	TAP1	ATP binding cassette transporters / subfamily B			
4061	-35.33	kd	CGS001-10682	EBP	-			
4062	-35.35	oe	ccsbBroad304_00152	BCAT2	-			
4063	-35.35	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
4064	-35.38	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
4065	-35.4	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
4066	-35.42	kd	CGS001-7088	TLE1	WD repeat domain containing			
4067	-35.44	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
4068	-35.44	kd	CGS001-18	ABAT	GABA turnover			
4069	-35.45	kd	CGS001-6514	SLC2A2	Solute carriers			
4070	-35.46	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
4071	-35.47	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
4072	-35.47	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4073	-35.47	kd	CGS001-57521	RPTOR	WD repeat domain containing			
4074	-35.49	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
4075	-35.5	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
4076	-35.5	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
4077	-35.51	oe	ccsbBroad304_02778	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4078	-35.51	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
4079	-35.52	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
4080	-35.54	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
4081	-35.54	oe	ccsbBroad304_00542	FBP1	-			
4082	-35.54	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
4083	-35.55	oe	ccsbBroad304_03950	ATG3	-			
4084	-35.56	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
4085	-35.6	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
4086	-35.6	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
4087	-35.6	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
4088	-35.6	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
4089	-35.61	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
4090	-35.63	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
4091	-35.64	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
4092	-35.69	kd	CGS001-329	BIRC2	Inhibitors of apoptosis (IAP) protein family			
4093	-35.7	cc		Gamma secretase inhibitor	-			
4094	-35.7	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
4095	-35.7	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
4096	-35.71	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
4097	-35.72	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
4098	-35.73	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
4099	-35.75	oe	ccsbBroad304_01701	TPI1	-			
4100	-35.8	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
4101	-35.8	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
4102	-35.84	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
4103	-35.86	oe	ccsbBroad304_06761	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4104	-35.86	kd	CGS001-670	BPHL	-			
4105	-35.87	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
4106	-35.87	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
4107	-35.89	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
4108	-35.91	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4109	-35.96	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
4110	-35.96	kd	CGS001-1737	DLAT	-			
4111	-35.99	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
4112	-36.06	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
4113	-36.06	kd	CGS001-2932	GSK3B	GSK subfamily			
4114	-36.07	kd	CGS001-2230	FDX1	-			
4115	-36.08	oe	ccsbBroad304_09095	PUS7L	-			
4116	-36.08	kd	CGS001-7276	TTR	-			
4117	-36.08	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
4118	-36.13	kd	CGS001-6646	SOAT1	-			
4119	-36.14	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4120	-36.15	kd	CGS001-2161	F12	Chymotrypsin			
4121	-36.17	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
4122	-36.17	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
4123	-36.23	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
4124	-36.24	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
4125	-36.26	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
4126	-36.27	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
4127	-36.29	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
4128	-36.3	oe	ccsbBroad304_01624	SUPV3L1	-			
4129	-36.3	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
4130	-36.3	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
4131	-36.32	oe	ccsbBroad304_02205	WTAP	-			
4132	-36.33	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
4133	-36.34	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
4134	-36.35	oe	ccsbBroad304_02580	TMED10	-			
4135	-36.37	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
4136	-36.42	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
4137	-36.42	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
4138	-36.43	kd	CGS001-80274	SCUBE1	-			
4139	-36.47	oe	ccsbBroad304_06976	SMARCE1	-			
4140	-36.49	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
4141	-36.5	oe	ccsbBroad304_00394	CTSD	Cathepsins			
4142	-36.5	kd	CGS001-4172	MCM3	-			
4143	-36.57	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
4144	-36.64	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
4145	-36.66	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
4146	-36.66	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
4147	-36.67	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
4148	-36.76	kd	CGS001-533	ATP6V0B	ATPases / V-type			
4149	-36.78	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
4150	-36.78	kd	CGS001-55038	CDCA4	-			
4151	-36.8	oe	ccsbBroad304_01263	PPP2R1A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4152	-36.82	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
4153	-36.86	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
4154	-36.87	kd	CGS001-2963	GTF2F2	General transcription factors			
4155	-36.87	kd	CGS001-11336	EXOC3	-			
4156	-36.88	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4157	-36.91	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
4158	-36.92	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
4159	-36.93	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
4160	-36.93	kd	CGS001-7079	TIMP4	-			
4161	-36.97	oe	ccsbBroad304_09284	UBE3B	-			
4162	-37.03	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
4163	-37.08	kd	CGS001-4547	MTTP	-			
4164	-37.16	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
4165	-37.23	kd	CGS001-5660	PSAP	Endogenous ligands			
4166	-37.26	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
4167	-37.29	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
4168	-37.3	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
4169	-37.3	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
4170	-37.35	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
4171	-37.36	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
4172	-37.38	oe	ccsbBroad304_02047	AP1S2	-			
4173	-37.44	kd	CGS001-890	CCNA2	-			
4174	-37.45	kd	CGS001-2053	EPHX2	-			
4175	-37.48	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
4176	-37.48	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
4177	-37.52	oe	ccsbBroad304_06837	RAF1	RAF family			
4178	-37.52	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
4179	-37.57	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
4180	-37.58	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
4181	-37.58	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
4182	-37.58	oe	ccsbBroad304_03580	ABCF3	ATP binding cassette transporters / subfamily F			
4183	-37.6	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
4184	-37.6	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
4185	-37.6	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
4186	-37.63	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
4187	-37.63	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
4188	-37.65	kd	CGS001-3638	INSIG1	-			
4189	-37.66	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
4190	-37.67	kd	CGS001-2155	F7	Chymotrypsin			
4191	-37.68	oe	ccsbBroad304_03121	NRBF2	-			
4192	-37.69	kd	CGS001-9267	CYTH1	Pleckstrin homology (PH) domain containing			
4193	-37.71	oe	ccsbBroad304_04202	MED28	-			
4194	-37.81	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
4195	-37.82	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
4196	-37.82	kd	CGS001-9276	COPB2	WD repeat domain containing			
4197	-37.83	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
4198	-37.85	oe	ccsbBroad304_02919	KIAA1279	-			
4199	-37.85	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
4200	-37.85	kd	CGS001-3416	IDE	Pitrilysin			
4201	-37.86	kd	CGS001-7099	TLR4	Toll-like receptor family			
4202	-37.87	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
4203	-37.88	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
4204	-37.89	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
4205	-37.95	oe	ccsbBroad304_03848	METTL14	-			
4206	-37.98	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
4207	-37.99	oe	ccsbBroad304_00382	CSNK2A2	Casein kinase 2 (CK2) family			
4208	-37.99	kd	CGS001-2108	ETFA	-			
4209	-37.99	kd	CGS001-55748	CNDP2	Carnosine dipeptidase			
4210	-38.04	oe	ccsbBroad304_00963	SMAD5	SMADs			
4211	-38.07	kd	CGS001-475	ATOX1	-			
4212	-38.09	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
4213	-38.09	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
4214	-38.1	oe	ccsbBroad304_01174	PEX13	-			
4215	-38.12	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4216	-38.16	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
4217	-38.16	kd	CGS001-29083	GTPBP8	-			
4218	-38.18	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
4219	-38.18	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
4220	-38.19	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4221	-38.21	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
4222	-38.3	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
4223	-38.3	kd	CGS001-4067	LYN	Src family			
4224	-38.31	kd	CGS001-23102	TBC1D2B	-			
4225	-38.37	kd	CGS001-6364	CCL20	Chemokine ligands			
4226	-38.38	kd	CGS001-399694	SHC4	SH2 domain containing			
4227	-38.45	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
4228	-38.47	oe	ccsbBroad304_07605	LYPLA1	-			
4229	-38.51	oe	ccsbBroad304_06234	G6PC	-			
4230	-38.51	oe	ccsbBroad304_00032	ADSL	-			
4231	-38.52	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
4232	-38.56	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
4233	-38.59	cp	BRD-K59773493	benzohydroxamic-acid	Antifungal			Antifungal
4234	-38.74	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
4235	-38.75	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
4236	-38.77	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
4237	-38.79	oe	ccsbBroad304_04072	HMGN5	High-mobility group / Canonical			
4238	-38.79	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
4239	-38.83	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
4240	-38.84	oe	ccsbBroad304_02080	USP14	Ubiquitin-specific peptidases			
4241	-38.84	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
4242	-38.86	kd	CGS001-11140	CDC37	-			
4243	-38.88	oe	ccsbBroad304_02368	TIMM17B	-			
4244	-38.88	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
4245	-38.91	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
4246	-38.93	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
4247	-38.95	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
4248	-38.97	oe	ccsbBroad304_02569	BTG3	-			
4249	-38.98	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
4250	-38.99	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
4251	-39	kd	CGS001-5613	PRKX	Protein kinase A			
4252	-39.01	oe	ccsbBroad304_02092	SYNGR3	-			
4253	-39.02	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4254	-39.04	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
4255	-39.04	kd	CGS001-6500	SKP1	-			
4256	-39.05	oe	ccsbBroad304_02554	TRAFD1	-			
4257	-39.06	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
4258	-39.13	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
4259	-39.14	oe	ccsbBroad304_02399	TNIP1	-			
4260	-39.14	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
4261	-39.15	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
4262	-39.15	kd	CGS001-3572	IL6ST	IL-6 receptor family			
4263	-39.16	oe	ccsbBroad304_09954	PTRF	-			
4264	-39.17	cc		PKC activator	-			
4265	-39.2	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
4266	-39.23	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
4267	-39.25	kd	CGS001-1493	CTLA4	CD molecules			
4268	-39.26	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
4269	-39.37	oe	ccsbBroad304_03625	HIF1AN	-			
4270	-39.38	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
4271	-39.4	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
4272	-39.4	kd	CGS001-8428	STK24	YSK subfamily			
4273	-39.44	oe	ccsbBroad304_07511	KIF14	Kinesins			
4274	-39.46	kd	CGS001-8800	PEX11A	-			
4275	-39.54	kd	CGS001-7431	VIM	Intermediate filaments type III			
4276	-39.56	kd	CGS001-5686	PSMA5	Proteasome subunits			
4277	-39.57	kd	CGS001-26128	KIAA1279	-			
4278	-39.61	kd	CGS001-116832	RPL39L	L ribosomal proteins			
4279	-39.62	kd	CGS001-9759	HDAC4	Histone deacetylases			
4280	-39.63	oe	ccsbBroad304_02322	ZNF263	Zinc fingers, C2H2-type			
4281	-39.65	oe	ccsbBroad304_01360	RAB4A	RAB, member RAS oncogene			
4282	-39.65	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
4283	-39.65	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
4284	-39.66	oe	ccsbBroad304_00960	SMAD1	SMADs			
4285	-39.66	kd	CGS001-4176	MCM7	-			
4286	-39.7	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
4287	-39.7	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
4288	-39.71	kd	CGS001-9200	PTPLA	-			
4289	-39.75	kd	CGS001-64333	ARHGAP9	Rho GTPase activating proteins			
4290	-39.76	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
4291	-39.76	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
4292	-39.76	kd	CGS001-3157	HMGCS1	Lanosterol biosynthesis pathway			
4293	-39.77	oe	ccsbBroad304_04398	MRPL43	Mitochondrial ribosomal proteins / large subunits			
4294	-39.79	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
4295	-39.8	kd	CGS001-23047	PDS5B	-			
4296	-39.84	cc		Topoisomerase inhibitor	-			
4297	-39.84	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
4298	-39.85	oe	ccsbBroad304_00389	CTBP1	-			
4299	-39.85	oe	ccsbBroad304_03554	NAT10	-			
4300	-39.88	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
4301	-39.89	cc		HMGCR inhibitor	-			
4302	-39.89	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
4303	-39.91	cc		CDK inhibitor	-			
4304	-39.91	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
4305	-39.92	oe	ccsbBroad304_00883	ISG20	-			
4306	-39.92	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4307	-39.95	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
4308	-39.97	oe	ccsbBroad304_00689	GRB7	Pleckstrin homology (PH) domain containing			
4309	-39.97	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
4310	-39.98	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
4311	-39.98	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
4312	-39.99	cc		S100 calcium binding proteins LOF	-			
4313	-40	kd	CGS001-1841	DTYMK	-			
4314	-40.03	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
4315	-40.04	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
4316	-40.07	cc		Reverse transcriptase inhibitor	-			
4317	-40.14	oe	ccsbBroad304_00250	CD19	CD molecules			
4318	-40.16	oe	ccsbBroad304_02487	TXNIP	-			
4319	-40.16	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4320	-40.17	oe	ccsbBroad304_06734	PLAT	Chymotrypsin			
4321	-40.17	kd	CGS001-6275	S100A4	EF-hand domain containing			
4322	-40.18	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
4323	-40.23	oe	ccsbBroad304_04128	ALG9	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
4324	-40.26	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
4325	-40.26	kd	CGS001-8731	RNMT	-			
4326	-40.26	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
4327	-40.29	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
4328	-40.3	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
4329	-40.32	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
4330	-40.32	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
4331	-40.34	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
4332	-40.36	oe	ccsbBroad304_09396	TIRAP	-			
4333	-40.37	oe	ccsbBroad304_00492	EIF5A	-			
4334	-40.37	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
4335	-40.38	oe	ccsbBroad304_00034	AES	-			
4336	-40.4	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
4337	-40.43	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
4338	-40.45	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
4339	-40.47	oe	ccsbBroad304_03371	RAB23	RAB, member RAS oncogene			
4340	-40.54	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
4341	-40.54	kd	CGS001-11200	CHEK2	CHK1 subfamily			
4342	-40.57	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
4343	-40.58	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
4344	-40.6	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
4345	-40.63	oe	ccsbBroad304_03917	RBKS	-			
4346	-40.66	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
4347	-40.69	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
4348	-40.74	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
4349	-40.82	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
4350	-40.82	kd	CGS001-6443	SGCB	-			
4351	-40.83	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
4352	-40.88	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
4353	-40.89	kd	CGS001-2288	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
4354	-40.89	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
4355	-40.93	kd	CGS001-51720	UIMC1	-			
4356	-40.93	kd	CGS001-7913	DEK	-			
4357	-40.94	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
4358	-40.96	oe	ccsbBroad304_00572	FKBP3	-			
4359	-40.96	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
4360	-40.98	oe	ccsbBroad304_02094	FIBP	-			
4361	-40.98	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
4362	-41.04	oe	ccsbBroad304_08993	DHDDS	-			
4363	-41.09	cc		KCNJ11 modulator	-			
4364	-41.12	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
4365	-41.15	kd	CGS001-819	CAMLG	-			
4366	-41.18	kd	CGS001-2067	ERCC1	-			
4367	-41.2	oe	ccsbBroad304_02746	FBXW11	F-boxes / WD-40 domains			
4368	-41.22	kd	CGS001-6491	STIL	-			
4369	-41.25	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
4370	-41.29	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
4371	-41.3	oe	ccsbBroad304_00962	SMAD4	SMADs			
4372	-41.3	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
4373	-41.3	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
4374	-41.33	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
4375	-41.34	cp	BRD-K10065684	dantron	Laxative			Laxative
4376	-41.35	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
4377	-41.35	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
4378	-41.39	oe	ccsbBroad304_00626	GDI1	-			
4379	-41.39	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
4380	-41.39	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
4381	-41.4	oe	ccsbBroad304_00115	ASPH	-			
4382	-41.44	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
4383	-41.45	oe	ccsbBroad304_06993	SRD5A1	-			
4384	-41.46	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
4385	-41.47	kd	CGS001-776	CACNA1D	Calcium channel subunits			
4386	-41.5	cc		Targets of VEGFR inhibitors GOF	-			
4387	-41.51	kd	CGS001-2597	GAPDH	-			
4388	-41.53	oe	ccsbBroad304_13633	PI4KAP2	-			
4389	-41.55	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
4390	-41.59	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
4391	-41.6	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4392	-41.61	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
4393	-41.62	kd	CGS001-4087	SMAD2	SMADs			
4394	-41.65	oe	ccsbBroad304_00620	GCDH	-			
4395	-41.75	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
4396	-41.75	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
4397	-41.77	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
4398	-41.78	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
4399	-41.81	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
4400	-41.83	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4401	-41.85	oe	ccsbBroad304_03032	HTATSF1	RNA binding motif (RRM) containing			
4402	-41.86	kd	CGS001-382	ARF6	ADP-ribosylation factors			
4403	-41.87	kd	CGS001-84647	PLA2G12B	-			
4404	-41.9	oe	ccsbBroad304_06549	SMAD3	SMADs			
4405	-41.91	cc		Calmodulin antagonist	-			
4406	-41.94	oe	ccsbBroad304_07411	LPXN	-			
4407	-41.95	cc		Tubulin inhibitor	-			
4408	-41.95	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
4409	-41.95	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
4410	-41.98	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
4411	-42.01	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
4412	-42.1	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
4413	-42.16	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
4414	-42.19	oe	ccsbBroad304_04788	OVCA2	-			
4415	-42.22	kd	CGS001-10613	ERLIN1	-			
4416	-42.25	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
4417	-42.26	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
4418	-42.31	oe	ccsbBroad304_01336	PTGS2	Cyclooxygenase			
4419	-42.35	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
4420	-42.36	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
4421	-42.37	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
4422	-42.4	cp	BRD-A02189320	met-leu-phe	-666			-666
4423	-42.41	kd	CGS001-5565	PRKAB2	AMPK subfamily			
4424	-42.46	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
4425	-42.49	cc		G2 M Checkpoint LOF	-			
4426	-42.5	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
4427	-42.51	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
4428	-42.53	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
4429	-42.54	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
4430	-42.57	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
4431	-42.66	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
4432	-42.71	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
4433	-42.71	kd	CGS001-23475	QPRT	-			
4434	-42.76	oe	ccsbBroad304_07053	TFPI	-			
4435	-42.78	kd	CGS001-439	ASNA1	-			
4436	-42.79	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
4437	-42.84	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
4438	-42.85	kd	CGS001-84547	PGBD1	-			
4439	-42.85	kd	CGS001-1284	COL4A2	Collagens			
4440	-42.86	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
4441	-42.86	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
4442	-42.87	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
4443	-42.91	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
4444	-42.91	kd	CGS001-6696	SPP1	Endogenous ligands			
4445	-42.91	kd	CGS001-23743	BHMT2	-			
4446	-42.93	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
4447	-42.94	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
4448	-42.98	oe	ccsbBroad304_02419	NDRG1	-			
4449	-42.99	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
4450	-42.99	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
4451	-42.99	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
4452	-43.09	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
4453	-43.09	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
4454	-43.11	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
4455	-43.11	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
4456	-43.13	oe	ccsbBroad304_00237	CCND3	-			
4457	-43.15	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
4458	-43.17	kd	CGS001-3155	HMGCL	-			
4459	-43.22	oe	ccsbBroad304_02175	MAGED1	-			
4460	-43.23	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
4461	-43.26	oe	ccsbBroad304_01985	EIF3H	-			
4462	-43.31	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
4463	-43.31	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
4464	-43.34	kd	CGS001-9805	SCRN1	-			
4465	-43.35	kd	CGS001-4758	NEU1	-			
4466	-43.36	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
4467	-43.38	kd	CGS001-1827	RCAN1	-			
4468	-43.4	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
4469	-43.43	kd	CGS001-90861	HN1L	-			
4470	-43.46	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
4471	-43.47	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
4472	-43.49	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
4473	-43.55	kd	CGS001-822	CAPG	-			
4474	-43.55	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
4475	-43.56	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
4476	-43.56	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
4477	-43.59	kd	CGS001-10953	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
4478	-43.6	cp	BRD-K10466330	AVA	Nucleophosmin inhibitor			Nucleophosmin inhibitor
4479	-43.64	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
4480	-43.64	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
4481	-43.65	kd	CGS001-10285	SMNDC1	Tudor domain containing			
4482	-43.69	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
4483	-43.73	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
4484	-43.78	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
4485	-43.79	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
4486	-43.79	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
4487	-43.8	kd	CGS001-3481	IGF2	-			
4488	-43.88	kd	CGS001-2852	GPER	-			
4489	-43.89	kd	CGS001-1831	TSC22D3	-			
4490	-43.92	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
4491	-43.93	oe	ccsbBroad304_03155	DHH	-			
4492	-43.94	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
4493	-43.94	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
4494	-43.97	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
4495	-43.97	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
4496	-44.03	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
4497	-44.04	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
4498	-44.06	oe	ccsbBroad304_00931	LCN2	Lipocalins			
4499	-44.07	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
4500	-44.07	kd	CGS001-65263	PYCRL	-			
4501	-44.19	kd	CGS001-5588	PRKCQ	Delta subfamily			
4502	-44.2	oe	ccsbBroad304_01280	PRKAR1A	Protein kinase A			
4503	-44.23	kd	CGS001-22887	FOXJ3	Forkhead boxes			
4504	-44.29	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
4505	-44.32	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
4506	-44.33	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
4507	-44.36	kd	CGS001-644	BLVRA	-			
4508	-44.39	kd	CGS001-84971	ATG4D	-			
4509	-44.4	oe	ccsbBroad304_02018	SUCLA2	-			
4510	-44.48	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
4511	-44.49	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
4512	-44.59	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
4513	-44.6	oe	ccsbBroad304_00239	CCNG1	-			
4514	-44.6	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
4515	-44.6	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4516	-44.6	oe	ccsbBroad304_13952	SHMT2	-			
4517	-44.61	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
4518	-44.69	oe	ccsbBroad304_02484	PAICS	-			
4519	-44.69	kd	CGS001-6185	RPN2	-			
4520	-44.71	oe	ccsbBroad304_06575	MEF2A	Myocyte enhancer factors			
4521	-44.75	oe	ccsbBroad304_08480	PNPO	-			
4522	-44.8	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4523	-44.8	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
4524	-44.84	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
4525	-44.85	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4526	-44.87	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
4527	-44.87	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
4528	-44.88	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
4529	-44.88	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4530	-44.9	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
4531	-44.93	oe	ccsbBroad304_06066	CTSL1	-			
4532	-44.95	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
4533	-44.99	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4534	-45	oe	ccsbBroad304_02579	YWHAQ	-			
4535	-45	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
4536	-45.07	oe	ccsbBroad304_01142	PAFAH1B2	-			
4537	-45.07	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
4538	-45.15	kd	CGS001-9218	VAPA	-			
4539	-45.18	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
4540	-45.21	cc		ATPase inhibitor	-			
4541	-45.24	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
4542	-45.26	kd	CGS001-10988	METAP2	Methionyl aminopeptidase			
4543	-45.31	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
4544	-45.33	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
4545	-45.34	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4546	-45.36	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
4547	-45.39	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
4548	-45.4	kd	CGS001-5355	PLP2	-			
4549	-45.42	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
4550	-45.43	oe	ccsbBroad304_02884	POT1	-			
4551	-45.47	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4552	-45.53	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4553	-45.54	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
4554	-45.55	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
4555	-45.57	kd	CGS001-79733	E2F8	-			
4556	-45.58	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4557	-45.61	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
4558	-45.65	oe	ccsbBroad304_01674	TIMP4	-			
4559	-45.65	kd	CGS001-642	BLMH	-			
4560	-45.71	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
4561	-45.8	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
4562	-45.81	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
4563	-45.83	kd	CGS001-10841	FTCD	-			
4564	-45.85	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
4565	-45.86	oe	ccsbBroad304_02458	STK25	YSK subfamily			
4566	-45.86	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
4567	-45.87	oe	ccsbBroad304_01593	SRP14	-			
4568	-45.88	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
4569	-45.9	kd	CGS001-122809	SOCS4	SH2 domain containing			
4570	-45.9	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
4571	-45.91	oe	ccsbBroad304_01744	UCHL1	Ubiquitin C-terminal hydrolase			
4572	-45.91	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
4573	-45.91	kd	CGS001-57721	METTL14	-			
4574	-45.92	oe	ccsbBroad304_03739	NRIP3	-			
4575	-45.92	kd	CGS001-3046	HBE1	-			
4576	-45.93	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
4577	-45.93	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
4578	-45.95	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
4579	-45.96	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
4580	-45.97	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
4581	-45.98	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
4582	-45.99	oe	ccsbBroad304_03573	BRF2	-			
4583	-46.01	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
4584	-46.02	cc		Aromatase inhibitor	-			
4585	-46.06	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
4586	-46.06	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
4587	-46.07	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
4588	-46.12	oe	ccsbBroad304_02278	THRAP3	-			
4589	-46.2	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
4590	-46.21	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
4591	-46.27	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
4592	-46.29	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
4593	-46.3	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
4594	-46.31	oe	ccsbBroad304_00985	MCL1	-			
4595	-46.34	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
4596	-46.35	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
4597	-46.4	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
4598	-46.49	oe	ccsbBroad304_00617	GBA	-			
4599	-46.49	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
4600	-46.51	oe	ccsbBroad304_06038	CRK	SH2 domain containing			
4601	-46.52	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
4602	-46.57	kd	CGS001-2615	LRRC32	-			
4603	-46.63	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
4604	-46.63	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
4605	-46.69	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
4606	-46.69	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
4607	-46.8	kd	CGS001-54805	CNNM2	-			
4608	-46.81	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
4609	-46.82	kd	CGS001-283150	FOXR1	Forkhead boxes			
4610	-46.83	kd	CGS001-2010	EMD	-			
4611	-46.83	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
4612	-46.87	kd	CGS001-2645	GCK	Hexokinases			
4613	-46.92	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
4614	-46.93	oe	ccsbBroad304_01183	PGD	-			
4615	-47.02	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
4616	-47.03	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
4617	-47.09	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
4618	-47.12	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
4619	-47.16	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
4620	-47.17	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
4621	-47.24	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
4622	-47.3	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
4623	-47.32	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
4624	-47.36	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
4625	-47.36	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
4626	-47.37	kd	CGS001-11344	TWF2	Twinfilin subfamily			
4627	-47.43	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
4628	-47.43	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
4629	-47.44	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
4630	-47.46	oe	ccsbBroad304_06134	ECH1	-			
4631	-47.49	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
4632	-47.51	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
4633	-47.6	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
4634	-47.63	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4635	-47.63	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
4636	-47.63	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
4637	-47.69	oe	ccsbBroad304_00501	EMD	-			
4638	-47.7	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
4639	-47.73	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
4640	-47.77	oe	ccsbBroad304_01658	PRDX2	-			
4641	-47.8	kd	CGS001-6387	CXCL12	Endogenous ligands			
4642	-47.83	kd	CGS001-2099	ESR1	Estrogen receptors			
4643	-47.84	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
4644	-47.91	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4645	-47.92	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
4646	-47.94	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4647	-47.95	oe	ccsbBroad304_05528	TICAM2	-			
4648	-47.96	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
4649	-47.99	kd	CGS001-9159	PCSK7	Subtilisin			
4650	-48	kd	CGS001-5019	OXCT1	-			
4651	-48.03	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
4652	-48.04	oe	ccsbBroad304_02276	MVP	-			
4653	-48.04	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
4654	-48.07	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
4655	-48.08	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
4656	-48.13	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
4657	-48.13	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
4658	-48.17	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
4659	-48.21	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
4660	-48.21	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
4661	-48.24	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
4662	-48.28	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
4663	-48.29	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
4664	-48.32	kd	CGS001-5663	PSEN1	Presenilin			
4665	-48.33	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4666	-48.35	kd	CGS001-25824	PRDX5	-			
4667	-48.36	kd	CGS001-7035	TFPI	-			
4668	-48.37	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
4669	-48.37	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
4670	-48.38	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
4671	-48.45	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
4672	-48.46	oe	ccsbBroad304_09354	IGSF8	CD molecules			
4673	-48.52	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
4674	-48.52	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
4675	-48.53	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
4676	-48.55	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
4677	-48.55	kd	CGS001-116931	MED12L	-			
4678	-48.58	oe	ccsbBroad304_01001	MEST	-			
4679	-48.6	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
4680	-48.61	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
4681	-48.65	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
4682	-48.71	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
4683	-48.75	oe	ccsbBroad304_08840	KIF9	Kinesins			
4684	-48.76	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
4685	-48.8	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
4686	-48.83	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
4687	-48.84	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
4688	-48.86	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4689	-48.87	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
4690	-48.88	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
4691	-48.91	kd	CGS001-1662	DDX10	DEAD-boxes			
4692	-48.94	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
4693	-48.97	kd	CGS001-87	ACTN1	EF-hand domain containing			
4694	-49.01	oe	ccsbBroad304_01673	TIMP3	-			
4695	-49.02	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
4696	-49.04	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
4697	-49.05	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
4698	-49.06	kd	CGS001-5618	PRLR	Prolactin receptor family			
4699	-49.11	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
4700	-49.12	kd	CGS001-23451	SF3B1	-			
4701	-49.23	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4702	-49.26	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
4703	-49.28	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
4704	-49.38	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
4705	-49.4	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
4706	-49.44	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
4707	-49.49	oe	ccsbBroad304_07832	XPO7	Exportins			
4708	-49.5	kd	CGS001-400	ARL1	ADP-ribosylation factors			
4709	-49.51	oe	ccsbBroad304_08365	CYCS	-			
4710	-49.61	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
4711	-49.61	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
4712	-49.62	kd	CGS001-26993	AKAP8L	-			
4713	-49.67	kd	CGS001-55577	NAGK	-			
4714	-49.7	oe	ccsbBroad304_00866	IMPA1	Inositol monophosphatase			
4715	-49.7	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
4716	-49.74	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
4717	-49.77	oe	ccsbBroad304_07379	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4718	-49.79	kd	CGS001-10972	TMED10	-			
4719	-49.85	oe	ccsbBroad304_06671	OPA1	-			
4720	-49.88	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
4721	-49.96	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
4722	-49.97	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
4723	-49.99	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
4724	-50	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
4725	-50.04	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4726	-50.06	oe	ccsbBroad304_07490	SCRN1	-			
4727	-50.07	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
4728	-50.14	kd	CGS001-3420	IDH3B	-			
4729	-50.16	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
4730	-50.22	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
4731	-50.25	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
4732	-50.26	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
4733	-50.33	oe	ccsbBroad304_05038	HORMAD2	-			
4734	-50.35	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
4735	-50.36	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
4736	-50.37	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
4737	-50.39	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
4738	-50.39	kd	CGS001-4860	PNP	-			
4739	-50.4	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
4740	-50.43	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
4741	-50.43	kd	CGS001-4637	MYL6	EF-hand domain containing			
4742	-50.45	oe	ccsbBroad304_00525	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
4743	-50.52	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
4744	-50.62	oe	ccsbBroad304_06095	DFFB	-			
4745	-50.62	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
4746	-50.67	kd	CGS001-9221	NOLC1	-			
4747	-50.67	oe	ccsbBroad304_07906	DDAH2	Dimethylarginine dimethylaminohydrolases			
4748	-50.68	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
4749	-50.77	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
4750	-50.77	kd	CGS001-3827	KNG1	Endogenous ligands			
4751	-50.81	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
4752	-50.83	oe	ccsbBroad304_02053	BTRC	F-boxes / WD-40 domains			
4753	-50.85	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
4754	-50.86	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
4755	-50.89	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
4756	-50.89	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
4757	-50.89	kd	CGS001-9871	SEC24D	-			
4758	-50.93	oe	ccsbBroad304_00509	EPHX1	-			
4759	-50.94	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
4760	-51.02	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
4761	-51.02	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
4762	-51.02	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
4763	-51.03	kd	CGS001-9687	GREB1	-			
4764	-51.06	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
4765	-51.08	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
4766	-51.09	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
4767	-51.1	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
4768	-51.1	kd	CGS001-1429	CRYZ	-			
4769	-51.12	kd	CGS001-8323	FZD6	GPCR / Class F : Frizzled receptors			
4770	-51.13	kd	CGS001-1514	CTSL1	-			
4771	-51.15	oe	ccsbBroad304_07651	HEXIM1	-			
4772	-51.16	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
4773	-51.16	oe	ccsbBroad304_00975	MAT2A	-			
4774	-51.2	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4775	-51.23	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
4776	-51.24	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
4777	-51.25	kd	CGS001-3895	KTN1	-			
4778	-51.3	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4779	-51.31	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
4780	-51.32	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
4781	-51.33	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
4782	-51.41	kd	CGS001-178	AGL	-			
4783	-51.42	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
4784	-51.47	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
4785	-51.5	oe	ccsbBroad304_04406	PLA2G12B	-			
4786	-51.5	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
4787	-51.56	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
4788	-51.56	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
4789	-51.58	kd	CGS001-1948	EFNB2	Ephrins			
4790	-51.61	oe	ccsbBroad304_05192	SPRED2	-			
4791	-51.63	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
4792	-51.68	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
4793	-51.68	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
4794	-51.71	oe	ccsbBroad304_14066	CHEK2	CHK1 subfamily			
4795	-51.73	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
4796	-51.81	kd	CGS001-1655	DDX5	DEAD-boxes			
4797	-51.82	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
4798	-51.83	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
4799	-51.85	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
4800	-51.85	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
4801	-51.92	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
4802	-51.93	oe	ccsbBroad304_01146	PARN	-			
4803	-51.93	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
4804	-52.02	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
4805	-52.03	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
4806	-52.06	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
4807	-52.06	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
4808	-52.11	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
4809	-52.17	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
4810	-52.18	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
4811	-52.23	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
4812	-52.28	oe	ccsbBroad304_00489	EHHADH	-			
4813	-52.29	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
4814	-52.33	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
4815	-52.36	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
4816	-52.42	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
4817	-52.51	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
4818	-52.52	cp	BRD-K17953061	staurosporine	PKC inhibitor		CDK2, GSK3B, CAMK2B, CDK1, CDK5, CHEK1, CHRM1, CHRM2, CHRM4, CSK, DAPK1, GPR35, IKBKB, ITK, LCK, LRRK2, MAP2K4, MAP2K6, MAPKAPK2, PAK2, PDPK1, PHKG2, PIK3CG, PIM1, PKN1, PRKACB, PRKCI, PRKCQ, RPS6KA1, STK3, SYK, TNIK, ZAP70	PKC inhibitor
4819	-52.54	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
4820	-52.57	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
4821	-52.61	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
4822	-52.61	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
4823	-52.62	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
4824	-52.69	kd	CGS001-23075	SWAP70	EF-hand domain containing			
4825	-52.69	kd	CGS001-216	ALDH1A1	Aldehyde dehydrogenases			
4826	-52.7	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
4827	-52.71	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
4828	-52.75	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
4829	-52.81	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
4830	-52.85	kd	CGS001-64121	RRAGC	-			
4831	-52.85	kd	CGS001-1029	CDKN2A	-			
4832	-52.89	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
4833	-52.98	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
4834	-53	oe	ccsbBroad304_03533	CDCA8	-			
4835	-53.04	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
4836	-53.06	oe	ccsbBroad304_01373	RAN	-			
4837	-53.06	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
4838	-53.13	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
4839	-53.15	oe	ccsbBroad304_06862	RGS3	-			
4840	-53.17	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
4841	-53.17	kd	CGS001-23196	FAM120A	-			
4842	-53.25	oe	ccsbBroad304_02509	GMEB1	-			
4843	-53.36	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
4844	-53.37	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
4845	-53.38	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
4846	-53.4	cc		IKK inhibitor	-			
4847	-53.42	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
4848	-53.42	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
4849	-53.44	kd	CGS001-2987	GUK1	-			
4850	-53.51	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
4851	-53.55	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
4852	-53.57	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
4853	-53.59	kd	CGS001-22828	SCAF8	RNA binding motif (RRM) containing			
4854	-53.61	oe	ccsbBroad304_05907	BUB1B	Bub family			
4855	-53.63	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
4856	-53.64	oe	ccsbBroad304_07632	PROCR	CD molecules			
4857	-53.65	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
4858	-53.66	kd	CGS001-1287	COL4A5	Collagens			
4859	-53.67	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
4860	-53.67	kd	CGS001-6342	SCP2	-			
4861	-53.69	kd	CGS001-10252	SPRY1	-			
4862	-53.72	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
4863	-53.72	kd	CGS001-1997	ELF1	ETS Transcription Factors			
4864	-53.75	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
4865	-53.81	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
4866	-53.88	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
4867	-53.89	cc		HOXL subclass homeoboxes LOF	-			
4868	-53.91	kd	CGS001-2109	ETFB	-			
4869	-53.96	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
4870	-54.07	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
4871	-54.14	cc		Protein synthesis inhibitor	-			
4872	-54.16	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
4873	-54.26	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
4874	-54.27	kd	CGS001-7016	TESK1	TESK subfamily			
4875	-54.28	oe	ccsbBroad304_06383	HMMR	CD molecules			
4876	-54.29	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
4877	-54.3	oe	ccsbBroad304_01560	SNAPC1	-			
4878	-54.32	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
4879	-54.35	oe	ccsbBroad304_00816	IDE	Pitrilysin			
4880	-54.35	oe	ccsbBroad304_02604	B3GNT1	-			
4881	-54.35	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
4882	-54.35	kd	CGS001-2073	ERCC5	-			
4883	-54.43	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
4884	-54.44	oe	ccsbBroad304_06008	AP2M1	-			
4885	-54.44	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
4886	-54.48	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
4887	-54.53	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
4888	-54.64	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
4889	-54.68	oe	ccsbBroad304_04292	INHBE	-			
4890	-54.68	kd	CGS001-9655	SOCS5	SH2 domain containing			
4891	-54.68	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
4892	-54.72	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4893	-54.76	kd	CGS001-24148	PRPF6	-			
4894	-54.76	kd	CGS001-11108	PRDM4	Zinc fingers, C2H2-type			
4895	-54.85	cc		Histone deacetylases LOF	-			
4896	-54.86	oe	ccsbBroad304_00881	IRF5	-			
4897	-54.89	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
4898	-54.91	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
4899	-54.91	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
4900	-54.91	oe	ccsbBroad304_04240	CLPB	Ankyrin repeat domain containing			
4901	-54.92	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
4902	-54.93	kd	CGS001-4925	NUCB2	EF-hand domain containing			
4903	-54.93	kd	CGS001-4507	MTAP	-			
4904	-55	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
4905	-55	kd	CGS001-6944	VPS72	-			
4906	-55.03	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
4907	-55.08	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
4908	-55.1	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
4909	-55.11	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
4910	-55.13	kd	CGS001-6895	TARBP2	-			
4911	-55.18	cc		Phospholipases GOF	-			
4912	-55.37	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
4913	-55.42	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
4914	-55.43	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
4915	-55.45	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
4916	-55.48	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
4917	-55.48	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
4918	-55.51	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
4919	-55.53	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
4920	-55.57	oe	ccsbBroad304_06538	LSP1	-			
4921	-55.58	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
4922	-55.61	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
4923	-55.7	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
4924	-55.72	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
4925	-55.72	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
4926	-55.77	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
4927	-55.78	cc		Tricyclic antidepressant	-			
4928	-55.82	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
4929	-55.86	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
4930	-55.86	kd	CGS001-9695	EDEM1	-			
4931	-55.88	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
4932	-55.89	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
4933	-55.9	oe	ccsbBroad304_04565	COG7	Components of oligomeric golgi complex			
4934	-55.94	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
4935	-55.96	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
4936	-56	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
4937	-56	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4938	-56.01	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
4939	-56.03	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
4940	-56.06	oe	ccsbBroad304_07178	ZFP112	-			
4941	-56.14	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
4942	-56.18	oe	ccsbBroad304_00693	NR3C1	3-Ketosteroid receptors			
4943	-56.29	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
4944	-56.32	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
4945	-56.34	oe	ccsbBroad304_06754	PPARD	Nuclear hormone receptors			
4946	-56.46	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
4947	-56.47	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
4948	-56.5	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
4949	-56.52	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
4950	-56.54	kd	CGS001-1054	CEBPG	basic leucine zipper proteins			
4951	-56.58	oe	ccsbBroad304_00954	LYN	Src family			
4952	-56.63	oe	ccsbBroad304_05890	BHMT	-			
4953	-56.67	cc		Apolipoproteins LOF	-			
4954	-56.68	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
4955	-56.69	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
4956	-56.8	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
4957	-56.86	oe	ccsbBroad304_02218	IKBKE	IKK family			
4958	-56.87	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
4959	-56.87	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
4960	-56.89	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
4961	-56.97	cc		Bromodomain Inhibitor	-			
4962	-56.98	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
4963	-57	kd	CGS001-22889	KIAA0907	-			
4964	-57.05	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
4965	-57.17	kd	CGS001-201516	ZSCAN4	Zinc fingers, C2H2-type			
4966	-57.19	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
4967	-57.27	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
4968	-57.34	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
4969	-57.34	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
4970	-57.35	oe	ccsbBroad304_14291	GDPD5	-			
4971	-57.35	oe	ccsbBroad304_05931	CAPG	-			
4972	-57.38	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4973	-57.38	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
4974	-57.39	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
4975	-57.54	oe	ccsbBroad304_03037	TMEM97	-			
4976	-57.54	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
4977	-57.57	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
4978	-57.59	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
4979	-57.66	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
4980	-57.66	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
4981	-57.67	kd	CGS001-29916	SNX11	Sorting nexins			
4982	-57.68	kd	CGS001-9375	TM9SF2	-			
4983	-57.7	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
4984	-57.75	oe	ccsbBroad304_00171	BNIP3L	-			
4985	-57.81	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
4986	-57.85	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
4987	-58.04	kd	CGS001-79716	NPEPL1	Leucyl aminopeptidase			
4988	-58.04	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
4989	-58.07	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
4990	-58.11	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
4991	-58.13	kd	CGS001-63933	CCDC90A	-			
4992	-58.2	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
4993	-58.23	kd	CGS001-83593	RASSF5	-			
4994	-58.25	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
4995	-58.3	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
4996	-58.31	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
4997	-58.38	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
4998	-58.4	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
4999	-58.42	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
5000	-58.46	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
5001	-58.5	kd	CGS001-3956	LGALS1	Endogenous ligands			
5002	-58.67	oe	ccsbBroad304_03433	DDIT4	-			
5003	-58.68	oe	ccsbBroad304_00009	ACLY	-			
5004	-58.73	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
5005	-58.73	oe	ccsbBroad304_01948	GAS7	-			
5006	-58.75	oe	ccsbBroad304_14143	NUSAP1	-			
5007	-58.77	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
5008	-58.83	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
5009	-58.84	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
5010	-58.84	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
5011	-58.87	kd	CGS001-10001	MED6	-			
5012	-59.01	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
5013	-59.03	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
5014	-59.08	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
5015	-59.12	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
5016	-59.16	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
5017	-59.2	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
5018	-59.26	kd	CGS001-54884	RETSAT	-			
5019	-59.29	kd	CGS001-117289	TAGAP	Rho GTPase activating proteins			
5020	-59.35	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
5021	-59.39	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
5022	-59.4	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
5023	-59.44	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
5024	-59.54	oe	ccsbBroad304_02526	POP4	-			
5025	-59.56	kd	CGS001-3030	HADHA	-			
5026	-59.61	kd	CGS001-9111	NMI	-			
5027	-59.61	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
5028	-59.65	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
5029	-59.67	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
5030	-59.7	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
5031	-59.72	oe	ccsbBroad304_02822	ARFIP2	-			
5032	-59.72	kd	CGS001-3516	RBPJ	-			
5033	-59.74	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
5034	-59.78	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5035	-59.81	oe	ccsbBroad304_04294	ATG10	-			
5036	-59.82	oe	ccsbBroad304_06583	MITF	Basic helix-loop-helix proteins			
5037	-59.82	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
5038	-59.82	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
5039	-59.85	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
5040	-59.86	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
5041	-59.92	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
5042	-59.96	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
5043	-60.02	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
5044	-60.02	kd	CGS001-7086	TKT	-			
5045	-60.04	oe	ccsbBroad304_01748	UFD1L	-			
5046	-60.06	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
5047	-60.12	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
5048	-60.13	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
5049	-60.13	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
5050	-60.14	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
5051	-60.2	kd	CGS001-27161	EIF2C2	-			
5052	-60.22	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5053	-60.25	cc		Sodium channel blocker	-			
5054	-60.25	oe	ccsbBroad304_03310	LCMT1	-			
5055	-60.26	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
5056	-60.43	oe	ccsbBroad304_05749	A2M	-			
5057	-60.44	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
5058	-60.45	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
5059	-60.47	cc		Sirtuins GOF	-			
5060	-60.5	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5061	-60.51	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
5062	-60.53	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
5063	-60.55	oe	ccsbBroad304_07078	TSPAN6	Tetraspanins			
5064	-60.56	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
5065	-60.57	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
5066	-60.59	kd	CGS001-595	CCND1	-			
5067	-60.61	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
5068	-60.63	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
5069	-60.63	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
5070	-60.66	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
5071	-60.67	kd	CGS001-9275	BCL7B	-			
5072	-60.69	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
5073	-60.69	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
5074	-60.72	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
5075	-60.74	kd	CGS001-3992	FADS1	Fatty acid desaturases			
5076	-60.75	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
5077	-60.76	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5078	-60.77	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
5079	-60.79	kd	CGS001-9322	TRIP10	-			
5080	-60.82	oe	ccsbBroad304_01019	MLH1	-			
5081	-60.82	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
5082	-60.86	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
5083	-60.9	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
5084	-60.9	kd	CGS001-839	CASP6	Caspases			
5085	-60.91	oe	ccsbBroad304_01862	YEATS4	-			
5086	-60.93	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
5087	-60.96	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
5088	-61	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
5089	-61	kd	CGS001-2582	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5090	-61.09	kd	CGS001-183	AGT	Endogenous ligands			
5091	-61.11	oe	ccsbBroad304_02890	SYF2	-			
5092	-61.12	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
5093	-61.15	kd	CGS001-7013	TERF1	-			
5094	-61.19	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5095	-61.23	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5096	-61.25	cc		Serotonin receptor antagonist	-			
5097	-61.25	oe	ccsbBroad304_01519	SET	-			
5098	-61.3	oe	ccsbBroad304_07861	COBL	-			
5099	-61.3	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
5100	-61.35	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
5101	-61.38	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
5102	-61.41	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
5103	-61.43	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
5104	-61.43	kd	CGS001-857	CAV1	-			
5105	-61.44	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
5106	-61.45	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
5107	-61.45	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
5108	-61.48	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
5109	-61.49	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
5110	-61.5	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5111	-61.5	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
5112	-61.51	cc		SRC inhibitor	-			
5113	-61.52	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
5114	-61.57	oe	ccsbBroad304_08879	CASD1	-			
5115	-61.59	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
5116	-61.62	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
5117	-61.62	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
5118	-61.63	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
5119	-61.65	kd	CGS001-3998	LMAN1	-			
5120	-61.66	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
5121	-61.71	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
5122	-61.74	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
5123	-61.75	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
5124	-61.79	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
5125	-61.83	kd	CGS001-2175	FANCA	Fanconi anemia, complementation groups			
5126	-61.85	oe	ccsbBroad304_02990	LYPD3	-			
5127	-61.85	kd	CGS001-8833	GMPS	-			
5128	-62.03	cc		Proteasome Pathway LOF	-			
5129	-62.08	kd	CGS001-5881	RAC3	Endogenous ligands			
5130	-62.11	kd	CGS001-5257	PHKB	-			
5131	-62.2	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
5132	-62.2	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
5133	-62.21	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
5134	-62.22	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
5135	-62.27	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
5136	-62.28	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
5137	-62.29	kd	CGS001-433	ASGR2	C-type lectin domain containing			
5138	-62.34	oe	ccsbBroad304_06188	F10	Chymotrypsin			
5139	-62.35	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
5140	-62.36	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
5141	-62.44	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
5142	-62.46	kd	CGS001-5209	PFKFB3	-			
5143	-62.47	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
5144	-62.52	kd	CGS001-6284	S100A13	S100 calcium binding proteins			
5145	-62.55	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
5146	-62.55	kd	CGS001-8569	MKNK1	MKN subfamily			
5147	-62.56	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
5148	-62.61	oe	ccsbBroad304_00657	GNG4	-			
5149	-62.67	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
5150	-62.67	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
5151	-62.69	kd	CGS001-1756	DMD	-			
5152	-62.71	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
5153	-62.73	oe	ccsbBroad304_03878	SENP2	-			
5154	-62.73	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
5155	-62.77	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
5156	-62.81	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
5157	-62.85	kd	CGS001-6519	SLC3A1	SLC3 family			
5158	-62.85	kd	CGS001-3663	IRF5	-			
5159	-62.88	oe	ccsbBroad304_01147	PC	Carboxylases			
5160	-62.89	oe	ccsbBroad304_02414	IRF9	-			
5161	-62.91	kd	CGS001-84890	ADO	-			
5162	-62.92	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
5163	-62.98	cp	BRD-K25079130	avrainvillamide-analog-4	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
5164	-62.99	oe	ccsbBroad304_06350	HAL	-			
5165	-63	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
5166	-63.04	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
5167	-63.07	kd	CGS001-5581	PRKCE	Eta subfamily			
5168	-63.1	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
5169	-63.21	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
5170	-63.28	kd	CGS001-7083	TK1	-			
5171	-63.29	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
5172	-63.39	cp	BRD-K76674262	homoharringtonine	Protein synthesis inhibitor		RPL3	Protein synthesis inhibitor
5173	-63.4	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
5174	-63.44	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
5175	-63.45	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
5176	-63.52	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
5177	-63.53	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5178	-63.54	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
5179	-63.54	kd	CGS001-388650	FAM69A	-			
5180	-63.54	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
5181	-63.61	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
5182	-63.71	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
5183	-63.81	oe	ccsbBroad304_02451	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
5184	-63.81	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
5185	-63.84	kd	CGS001-10523	CHERP	G patch domain containing			
5186	-63.89	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5187	-63.9	kd	CGS001-2678	GGT1	CD molecules			
5188	-63.93	kd	CGS001-472	ATM	Other PIKK family kinases			
5189	-63.94	kd	CGS001-2760	GM2A	-			
5190	-64	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
5191	-64	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
5192	-64.02	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
5193	-64.07	oe	ccsbBroad304_00212	CAMLG	-			
5194	-64.08	oe	ccsbBroad304_02136	COPS2	-			
5195	-64.12	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
5196	-64.13	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
5197	-64.14	oe	ccsbBroad304_13813	ARAF	RAF family			
5198	-64.22	kd	CGS001-5253	PHF2	Histone demethylases			
5199	-64.23	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5200	-64.24	kd	CGS001-174	AFP	-			
5201	-64.26	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
5202	-64.27	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
5203	-64.39	kd	CGS001-10943	MSL3	-			
5204	-64.49	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
5205	-64.51	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
5206	-64.51	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
5207	-64.52	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
5208	-64.53	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
5209	-64.57	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
5210	-64.59	oe	ccsbBroad304_06952	SKP1	-			
5211	-64.6	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
5212	-64.64	oe	ccsbBroad304_14011	PAPSS1	-			
5213	-64.66	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
5214	-64.69	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
5215	-64.73	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
5216	-64.76	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
5217	-64.78	kd	CGS001-8837	CFLAR	Endogenous ligands			
5218	-64.79	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
5219	-64.79	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5220	-64.79	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
5221	-64.85	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
5222	-64.86	kd	CGS001-4833	NME4	-			
5223	-64.88	kd	CGS001-9791	PTDSS1	-			
5224	-64.91	kd	CGS001-23588	KLHDC2	-			
5225	-64.99	oe	ccsbBroad304_10207	ERLIN1	-			
5226	-65.06	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
5227	-65.09	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
5228	-65.17	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
5229	-65.19	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
5230	-65.27	kd	CGS001-5387	PMS2P3	-			
5231	-65.33	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
5232	-65.35	kd	CGS001-9451	EIF2AK3	PEK subfamily			
5233	-65.38	oe	ccsbBroad304_02964	TIMM9	-			
5234	-65.39	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
5235	-65.41	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
5236	-65.45	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
5237	-65.48	kd	CGS001-3608	ILF2	-			
5238	-65.48	kd	CGS001-1497	CTNS	-			
5239	-65.49	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
5240	-65.52	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
5241	-65.54	kd	CGS001-10868	USP20	Ubiquitin-specific peptidases			
5242	-65.54	kd	CGS001-27097	TAF5L	WD repeat domain containing			
5243	-65.56	kd	CGS001-8667	EIF3H	-			
5244	-65.56	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5245	-65.61	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
5246	-65.66	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
5247	-65.71	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
5248	-65.74	kd	CGS001-826	CAPNS1	EF-hand domain containing			
5249	-65.76	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
5250	-65.76	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
5251	-65.9	kd	CGS001-28960	DCPS	-			
5252	-65.91	kd	CGS001-139135	PASD1	-			
5253	-65.93	oe	ccsbBroad304_01769	VEGFB	-			
5254	-65.98	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
5255	-65.98	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
5256	-66.02	kd	CGS001-2287	FKBP3	-			
5257	-66.04	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
5258	-66.13	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
5259	-66.16	oe	ccsbBroad304_03450	TMED9	-			
5260	-66.18	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
5261	-66.24	oe	ccsbBroad304_01716	TSN	-			
5262	-66.24	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
5263	-66.31	cc		Proteasome inhibitor	-			
5264	-66.32	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
5265	-66.37	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5266	-66.41	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
5267	-66.55	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
5268	-66.65	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
5269	-66.68	oe	ccsbBroad304_08839	IFIH1	-			
5270	-66.69	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
5271	-66.7	oe	ccsbBroad304_09821	TMEM154	-			
5272	-66.73	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
5273	-66.8	oe	ccsbBroad304_00398	CTSL2	-			
5274	-66.81	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
5275	-66.82	kd	CGS001-1955	MEGF9	-			
5276	-66.86	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
5277	-66.86	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
5278	-66.89	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
5279	-66.89	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
5280	-66.9	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
5281	-66.91	kd	CGS001-5566	PRKACA	Protein kinase A			
5282	-66.95	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
5283	-66.96	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
5284	-66.99	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
5285	-67.01	kd	CGS001-2548	GAA	Glycosidases			
5286	-67.03	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
5287	-67.04	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
5288	-67.05	kd	CGS001-23192	ATG4B	Aut2 peptidase			
5289	-67.07	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
5290	-67.15	oe	ccsbBroad304_02534	UTP14A	-			
5291	-67.16	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
5292	-67.17	oe	ccsbBroad304_03850	TRIB3	Trbl family			
5293	-67.19	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
5294	-67.27	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
5295	-67.29	oe	ccsbBroad304_06820	PTS	-			
5296	-67.31	kd	CGS001-6233	RPS27A	S ribosomal proteins			
5297	-67.37	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
5298	-67.4	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
5299	-67.42	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
5300	-67.44	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
5301	-67.44	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
5302	-67.44	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
5303	-67.45	kd	CGS001-23149	FCHO1	-			
5304	-67.49	oe	ccsbBroad304_02195	SPAG7	-			
5305	-67.57	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
5306	-67.67	oe	ccsbBroad304_00529	F3	CD molecules			
5307	-67.68	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
5308	-67.76	oe	ccsbBroad304_02285	MED6	-			
5309	-67.78	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
5310	-67.8	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
5311	-67.8	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
5312	-67.8	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
5313	-67.84	kd	CGS001-1201	CLN3	-			
5314	-67.92	oe	ccsbBroad304_09708	PNLDC1	-			
5315	-67.93	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
5316	-67.95	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
5317	-67.95	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
5318	-68.03	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
5319	-68.07	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
5320	-68.13	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
5321	-68.21	oe	ccsbBroad304_05927	CALM1	EF-hand domain containing			
5322	-68.28	kd	CGS001-64116	SLC39A8	SLC39 family of metal ion transporters			
5323	-68.3	oe	ccsbBroad304_02533	NOXA1	-			
5324	-68.33	kd	CGS001-226	ALDOA	-			
5325	-68.37	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
5326	-68.4	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5327	-68.41	kd	CGS001-23210	JMJD6	-			
5328	-68.43	oe	ccsbBroad304_00841	IKBKB	IKK family			
5329	-68.46	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
5330	-68.47	oe	ccsbBroad304_02138	TRIP10	-			
5331	-68.47	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
5332	-68.48	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
5333	-68.49	kd	CGS001-10412	NSA2	-			
5334	-68.49	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
5335	-68.52	kd	CGS001-6446	SGK1	SGK family			
5336	-68.62	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
5337	-68.65	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
5338	-68.71	kd	CGS001-125965	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
5339	-68.73	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5340	-68.75	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
5341	-68.82	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
5342	-68.83	cc		Cyclins LOF	-			
5343	-68.84	kd	CGS001-6622	SNCA	Parkinson disease			
5344	-68.91	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
5345	-68.96	oe	ccsbBroad304_03928	RRAGC	-			
5346	-69.01	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
5347	-69.07	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
5348	-69.12	oe	ccsbBroad304_02197	VPS26A	-			
5349	-69.16	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5350	-69.2	oe	ccsbBroad304_00179	BTG1	-			
5351	-69.21	oe	ccsbBroad304_03570	QRSL1	-			
5352	-69.21	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
5353	-69.24	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
5354	-69.25	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
5355	-69.33	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
5356	-69.33	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
5357	-69.38	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
5358	-69.51	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
5359	-69.55	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
5360	-69.61	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
5361	-69.62	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
5362	-69.65	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
5363	-69.72	oe	ccsbBroad304_02229	TRAM2	-			
5364	-69.78	oe	ccsbBroad304_06225	FTH1	-			
5365	-69.79	kd	CGS001-6119	RPA3	-			
5366	-69.79	kd	CGS001-3269	HRH1	Histamine receptors			
5367	-69.84	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
5368	-69.92	kd	CGS001-4200	ME2	-			
5369	-70	kd	CGS001-5827	PXMP2	-			
5370	-70.01	kd	CGS001-51022	GLRX2	-			
5371	-70.02	kd	CGS001-9249	DHRS3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
5372	-70.19	oe	ccsbBroad304_04190	CCDC92	-			
5373	-70.23	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
5374	-70.23	kd	CGS001-9641	IKBKE	IKK family			
5375	-70.24	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
5376	-70.27	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
5377	-70.28	kd	CGS001-9738	CCP110	-			
5378	-70.32	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5379	-70.32	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
5380	-70.37	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
5381	-70.44	kd	CGS001-4090	SMAD5	SMADs			
5382	-70.45	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
5383	-70.51	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
5384	-70.52	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
5385	-70.53	cc		Phospholipases LOF	-			
5386	-70.53	kd	CGS001-1066	CES1	Carboxylesterases			
5387	-70.6	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
5388	-70.66	oe	ccsbBroad304_02048	BCL10	-			
5389	-70.67	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
5390	-70.7	kd	CGS001-11180	WDR6	WD repeat domain containing			
5391	-70.72	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
5392	-70.78	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
5393	-70.79	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
5394	-70.86	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
5395	-70.88	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5396	-70.88	kd	CGS001-23386	NUDCD3	-			
5397	-70.89	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
5398	-70.94	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5399	-70.98	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
5400	-70.99	kd	CGS001-31	ACACA	Carboxylases			
5401	-71	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
5402	-71.02	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
5403	-71.04	oe	ccsbBroad304_02163	MED7	-			
5404	-71.05	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
5405	-71.06	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
5406	-71.09	kd	CGS001-5920	RARRES3	-			
5407	-71.12	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
5408	-71.12	kd	CGS001-840	CASP7	Caspases			
5409	-71.13	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
5410	-71.15	kd	CGS001-5664	PSEN2	Presenilin			
5411	-71.19	kd	CGS001-22930	RAB3GAP1	-			
5412	-71.21	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
5413	-71.25	oe	ccsbBroad304_00278	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
5414	-71.26	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5415	-71.27	oe	ccsbBroad304_00747	HLF	-			
5416	-71.3	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
5417	-71.34	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
5418	-71.34	kd	CGS001-6793	STK10	SLK subfamily			
5419	-71.34	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
5420	-71.35	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
5421	-71.38	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
5422	-71.38	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
5423	-71.39	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
5424	-71.4	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
5425	-71.41	kd	CGS001-8575	PRKRA	-			
5426	-71.44	oe	ccsbBroad304_01025	ALDH6A1	Aldehyde dehydrogenases			
5427	-71.46	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
5428	-71.5	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
5429	-71.59	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5430	-71.62	cc		IMPDH inhibitor	-			
5431	-71.7	oe	ccsbBroad304_02801	CASP14	Caspases			
5432	-71.7	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
5433	-71.71	oe	ccsbBroad304_08888	ACD	-			
5434	-71.72	oe	ccsbBroad304_09006	RPF1	-			
5435	-71.72	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
5436	-71.89	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
5437	-71.89	kd	CGS001-57019	CIAPIN1	-			
5438	-71.91	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5439	-71.93	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5440	-71.94	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
5441	-72	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5442	-72.07	oe	ccsbBroad304_06386	HNMT	-			
5443	-72.07	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
5444	-72.09	oe	ccsbBroad304_08709	SCYL3	-			
5445	-72.18	kd	CGS001-1504	CTRB1	-			
5446	-72.2	oe	ccsbBroad304_09303	LRSAM1	Sterile alpha motif (SAM) domain containing			
5447	-72.21	oe	ccsbBroad304_06018	COMT	Catecholamine turnover			
5448	-72.21	kd	CGS001-1069	CETN2	EF-hand domain containing			
5449	-72.22	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
5450	-72.24	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
5451	-72.29	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
5452	-72.34	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
5453	-72.38	kd	CGS001-6938	TCF12	Basic helix-loop-helix proteins			
5454	-72.39	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
5455	-72.39	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
5456	-72.44	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
5457	-72.46	cc		GABA receptor antagonist	-			
5458	-72.47	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
5459	-72.51	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
5460	-72.57	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
5461	-72.58	kd	CGS001-25797	QPCT	Aminopeptidase Y			
5462	-72.6	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
5463	-72.6	kd	CGS001-286380	FOXD4L3	-			
5464	-72.6	kd	CGS001-9784	SNX17	Sorting nexins			
5465	-72.62	kd	CGS001-843	CASP10	Caspases			
5466	-72.68	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
5467	-72.72	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
5468	-72.82	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
5469	-72.89	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
5470	-72.94	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
5471	-72.98	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
5472	-73	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
5473	-73	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
5474	-73.02	oe	ccsbBroad304_03858	SRPRB	-			
5475	-73.06	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
5476	-73.08	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
5477	-73.09	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
5478	-73.09	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
5479	-73.1	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
5480	-73.13	kd	CGS001-5411	PNN	-			
5481	-73.14	kd	CGS001-64343	AZI2	-			
5482	-73.18	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
5483	-73.19	kd	CGS001-80746	TSEN2	tRNA splicing endonuclease subunits			
5484	-73.2	oe	ccsbBroad304_01084	NEU1	-			
5485	-73.23	kd	CGS001-5264	PHYH	-			
5486	-73.24	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
5487	-73.26	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
5488	-73.29	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
5489	-73.33	kd	CGS001-7316	UBC	-			
5490	-73.34	oe	ccsbBroad304_02345	TXNDC9	-			
5491	-73.39	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
5492	-73.41	oe	ccsbBroad304_02017	PEX11A	-			
5493	-73.42	kd	CGS001-5361	PLXNA1	Plexins			
5494	-73.43	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
5495	-73.46	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
5496	-73.48	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
5497	-73.49	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
5498	-73.5	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
5499	-73.57	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
5500	-73.6	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
5501	-73.61	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
5502	-73.61	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
5503	-73.71	kd	CGS001-5378	PMS1	-			
5504	-73.72	oe	ccsbBroad304_02318	KIF20A	Kinesins			
5505	-73.73	cc		RAF inhibitor	-			
5506	-73.74	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
5507	-73.76	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
5508	-73.76	kd	CGS001-10494	STK25	YSK subfamily			
5509	-73.8	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
5510	-73.83	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
5511	-73.84	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
5512	-73.84	kd	CGS001-8536	CAMK1	CAMK1 family			
5513	-73.87	cc		EGFR inhibitor	-			
5514	-73.93	oe	ccsbBroad304_06889	RPN2	-			
5515	-73.93	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
5516	-73.99	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5517	-74	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
5518	-74.07	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
5519	-74.07	kd	CGS001-2783	GNB2	WD repeat domain containing			
5520	-74.12	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
5521	-74.13	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
5522	-74.14	kd	CGS001-4602	MYB	-			
5523	-74.19	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5524	-74.31	oe	ccsbBroad304_07820	SNW1	-			
5525	-74.31	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
5526	-74.41	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5527	-74.42	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
5528	-74.42	kd	CGS001-114785	MBD6	-			
5529	-74.49	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
5530	-74.49	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
5531	-74.51	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
5532	-74.53	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
5533	-74.58	oe	ccsbBroad304_00113	ASNS	-			
5534	-74.61	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
5535	-74.67	kd	CGS001-1155	TBCB	-			
5536	-74.67	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
5537	-74.68	kd	CGS001-51160	VPS28	-			
5538	-74.69	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
5539	-74.73	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
5540	-74.74	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
5541	-74.74	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
5542	-74.76	oe	ccsbBroad304_01617	STX4	-			
5543	-74.78	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
5544	-74.87	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
5545	-74.89	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
5546	-74.89	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
5547	-74.91	kd	CGS001-3460	IFNGR2	Interferon receptor family			
5548	-74.92	kd	CGS001-718	C3	Endogenous ligands			
5549	-74.96	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
5550	-74.96	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
5551	-74.96	kd	CGS001-3845	KRAS	RAS subfamily			
5552	-74.97	kd	CGS001-10606	PAICS	-			
5553	-75.03	kd	CGS001-2782	GNB1	WD repeat domain containing			
5554	-75.04	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
5555	-75.09	oe	ccsbBroad304_06133	TOR1A	-			
5556	-75.13	kd	CGS001-2781	GNAZ	-			
5557	-75.14	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
5558	-75.18	oe	ccsbBroad304_00880	IRF2	-			
5559	-75.21	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
5560	-75.25	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
5561	-75.25	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
5562	-75.28	oe	ccsbBroad304_07208	NRIP1	-			
5563	-75.29	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
5564	-75.33	kd	CGS001-55165	CEP55	-			
5565	-75.39	oe	ccsbBroad304_00462	DR1	-			
5566	-75.41	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
5567	-75.42	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
5568	-75.53	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
5569	-75.54	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
5570	-75.6	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
5571	-75.6	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5572	-75.62	oe	ccsbBroad304_11024	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5573	-75.69	cc		HDAC inhibitor	-			
5574	-75.8	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
5575	-75.83	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
5576	-75.84	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
5577	-75.91	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
5578	-75.94	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
5579	-75.96	kd	CGS001-5480	PPIC	-			
5580	-75.97	kd	CGS001-7296	TXNRD1	-			
5581	-75.99	kd	CGS001-1854	DUT	-			
5582	-76.04	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
5583	-76.07	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
5584	-76.23	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
5585	-76.33	kd	CGS001-51447	IP6K2	-			
5586	-76.33	oe	ccsbBroad304_10491	PFKL	-			
5587	-76.35	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
5588	-76.57	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
5589	-76.61	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
5590	-76.61	kd	CGS001-64324	NSD1	Histone methyltransferases (HMTs)			
5591	-76.62	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
5592	-76.64	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
5593	-76.73	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
5594	-76.84	oe	ccsbBroad304_03615	ZNF673	-			
5595	-76.85	oe	ccsbBroad304_10487	BPHL	-			
5596	-76.88	kd	CGS001-383	ARG1	Arginase			
5597	-76.89	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
5598	-76.9	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
5599	-76.93	oe	ccsbBroad304_00600	FYN	Src family			
5600	-76.93	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
5601	-76.94	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
5602	-76.94	kd	CGS001-7486	WRN	-			
5603	-76.99	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
5604	-77.05	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
5605	-77.1	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
5606	-77.12	kd	CGS001-10607	TBL3	WD repeat domain containing			
5607	-77.16	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
5608	-77.18	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
5609	-77.18	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5610	-77.2	kd	CGS001-5997	RGS2	Endogenous ligands			
5611	-77.21	kd	CGS001-5230	PGK1	-			
5612	-77.26	kd	CGS001-10652	YKT6	-			
5613	-77.26	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
5614	-77.27	kd	CGS001-11230	PRAF2	-			
5615	-77.28	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
5616	-77.37	oe	ccsbBroad304_01556	SMARCB1	-			
5617	-77.41	oe	ccsbBroad304_07889	QPRT	-			
5618	-77.43	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
5619	-77.47	kd	CGS001-11040	PIM2	PIM family			
5620	-77.5	oe	ccsbBroad304_02499	CTCF	Zinc fingers, C2H2-type			
5621	-77.53	cc		PI3K inhibitor	-			
5622	-77.6	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
5623	-77.61	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
5624	-77.61	kd	CGS001-54881	TEX10	-			
5625	-77.65	cp	BRD-K29313308	HDAC3-selective	HDAC inhibitor		HDAC3	HDAC inhibitor
5626	-77.65	kd	CGS001-836	CASP3	Caspases			
5627	-77.66	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
5628	-77.67	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
5629	-77.72	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
5630	-77.76	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
5631	-77.81	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
5632	-77.81	kd	CGS001-57149	LYRM1	LYR motif containing			
5633	-77.82	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
5634	-77.83	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
5635	-77.83	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
5636	-77.84	oe	ccsbBroad304_06126	TSC22D3	-			
5637	-77.84	kd	CGS001-4664	NAB1	-			
5638	-77.85	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
5639	-77.87	kd	CGS001-2030	SLC29A1	SLC29 family			
5640	-77.91	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5641	-77.96	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
5642	-77.97	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
5643	-78.01	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
5644	-78.02	kd	CGS001-51014	TMED7	-			
5645	-78.05	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
5646	-78.13	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
5647	-78.17	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
5648	-78.2	oe	ccsbBroad304_05439	O3FAR1	-			
5649	-78.21	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
5650	-78.36	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
5651	-78.37	kd	CGS001-114609	TIRAP	-			
5652	-78.38	kd	CGS001-638	BIK	-			
5653	-78.39	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
5654	-78.48	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
5655	-78.51	kd	CGS001-1398	CRK	SH2 domain containing			
5656	-78.53	oe	ccsbBroad304_07220	CDC45	-			
5657	-78.58	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
5658	-78.61	kd	CGS001-7389	UROD	-			
5659	-78.63	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
5660	-78.65	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5661	-78.65	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5662	-78.65	kd	CGS001-7358	UGDH	-			
5663	-78.66	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
5664	-78.72	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
5665	-78.73	oe	ccsbBroad304_06651	NOV	-			
5666	-78.73	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
5667	-78.75	oe	ccsbBroad304_02626	PKIG	-			
5668	-78.75	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
5669	-78.77	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
5670	-78.87	oe	ccsbBroad304_03479	YTHDF1	-			
5671	-78.97	cp	BRD-K80348542	cephaeline	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
5672	-78.99	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
5673	-78.99	kd	CGS001-11041	B3GNT1	-			
5674	-79.03	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
5675	-79.03	kd	CGS001-1490	CTGF	-			
5676	-79.04	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
5677	-79.06	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
5678	-79.07	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
5679	-79.08	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
5680	-79.09	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
5681	-79.11	oe	ccsbBroad304_08340	POLR3K	RNA polymerase subunits			
5682	-79.19	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
5683	-79.2	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
5684	-79.2	oe	ccsbBroad304_07688	FAM114A2	-			
5685	-79.33	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
5686	-79.34	oe	ccsbBroad304_10240	CROT	-			
5687	-79.42	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
5688	-79.42	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
5689	-79.42	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
5690	-79.43	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
5691	-79.48	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
5692	-79.51	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
5693	-79.52	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
5694	-79.53	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
5695	-79.53	kd	CGS001-64786	TBC1D15	-			
5696	-79.54	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
5697	-79.68	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
5698	-79.69	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
5699	-79.69	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
5700	-79.7	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5701	-79.7	kd	CGS001-1879	EBF1	-			
5702	-79.72	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
5703	-79.73	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
5704	-79.74	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
5705	-79.79	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
5706	-79.85	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
5707	-79.88	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
5708	-79.88	kd	CGS001-5194	PEX13	-			
5709	-79.9	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
5710	-79.91	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
5711	-79.93	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
5712	-80.08	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
5713	-80.1	kd	CGS001-6277	S100A6	EF-hand domain containing			
5714	-80.11	oe	ccsbBroad304_14389	PSMA8	Proteasome (prosome, macropain) subunits			
5715	-80.15	kd	CGS001-11212	PROSC	-			
5716	-80.18	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
5717	-80.24	oe	ccsbBroad304_02702	MSRB2	-			
5718	-80.24	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
5719	-80.28	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5720	-80.33	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
5721	-80.34	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
5722	-80.35	oe	ccsbBroad304_01180	PFKFB3	-			
5723	-80.4	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
5724	-80.44	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
5725	-80.48	oe	ccsbBroad304_05899	BMP4	Bone morphogenetic proteins			
5726	-80.49	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
5727	-80.52	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
5728	-80.53	oe	ccsbBroad304_06783	LGMN	Legumain			
5729	-80.58	cc		General transcription factors group 2 LOF	-			
5730	-80.58	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
5731	-80.59	oe	ccsbBroad304_02032	TSC22D1	-			
5732	-80.59	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
5733	-80.6	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
5734	-80.66	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
5735	-80.66	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
5736	-80.76	kd	CGS001-10645	CAMKK2	Meta subfamily			
5737	-80.77	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
5738	-80.78	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
5739	-80.81	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
5740	-80.81	kd	CGS001-47	ACLY	-			
5741	-80.84	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
5742	-80.86	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5743	-80.86	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
5744	-80.86	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
5745	-80.89	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
5746	-80.89	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
5747	-80.9	oe	ccsbBroad304_04154	DENND2D	DENN/MADD domain containing			
5748	-80.9	kd	CGS001-1738	DLD	-			
5749	-80.95	oe	ccsbBroad304_05152	SSBP4	-			
5750	-80.95	oe	ccsbBroad304_06525	LIPA	-			
5751	-80.97	oe	ccsbBroad304_06372	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
5752	-80.99	oe	ccsbBroad304_09254	PAQR8	-			
5753	-81	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
5754	-81.09	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
5755	-81.09	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
5756	-81.18	oe	ccsbBroad304_01664	TGFA	-			
5757	-81.26	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
5758	-81.27	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
5759	-81.29	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
5760	-81.41	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
5761	-81.42	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
5762	-81.42	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
5763	-81.43	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
5764	-81.44	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
5765	-81.5	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
5766	-81.51	oe	ccsbBroad304_07128	VHL	-			
5767	-81.52	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
5768	-81.54	kd	CGS001-3932	LCK	Src family			
5769	-81.55	oe	ccsbBroad304_06985	SORD	-			
5770	-81.58	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
5771	-81.62	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
5772	-81.62	kd	CGS001-27244	SESN1	-			
5773	-81.63	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
5774	-81.64	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
5775	-81.77	kd	CGS001-29102	DROSHA	-			
5776	-81.78	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
5777	-81.8	kd	CGS001-2821	GPI	-			
5778	-81.85	kd	CGS001-11044	PAPD7	-			
5779	-81.86	kd	CGS001-9455	HOMER2	-			
5780	-81.88	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
5781	-81.88	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
5782	-81.92	cp	BRD-K53665955	MK-5108	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
5783	-81.96	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
5784	-81.97	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5785	-81.99	kd	CGS001-403	ARL3	ADP-ribosylation factors			
5786	-82	oe	ccsbBroad304_02788	PRAME	-			
5787	-82	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
5788	-82.01	kd	CGS001-117154	DACH2	-			
5789	-82.04	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
5790	-82.05	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
5791	-82.09	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
5792	-82.13	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
5793	-82.19	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
5794	-82.2	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
5795	-82.21	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
5796	-82.25	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
5797	-82.31	kd	CGS001-3606	IL18	Interleukins and interleukin receptors			
5798	-82.34	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
5799	-82.36	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5800	-82.36	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5801	-82.36	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
5802	-82.39	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
5803	-82.41	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
5804	-82.42	kd	CGS001-2664	GDI1	-			
5805	-82.46	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
5806	-82.53	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
5807	-82.54	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
5808	-82.55	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
5809	-82.56	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5810	-82.59	oe	ccsbBroad304_00815	ID2	Basic helix-loop-helix proteins			
5811	-82.6	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
5812	-82.63	kd	CGS001-9467	SH3BP5	-			
5813	-82.69	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
5814	-82.69	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
5815	-82.7	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
5816	-82.73	oe	ccsbBroad304_06085	DCK	-			
5817	-82.75	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
5818	-82.79	oe	ccsbBroad304_02622	PRDM4	Zinc fingers, C2H2-type			
5819	-82.79	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
5820	-82.82	kd	CGS001-11243	PMF1	-			
5821	-82.92	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
5822	-82.96	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5823	-82.98	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
5824	-82.98	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
5825	-82.98	kd	CGS001-23499	MACF1	EF-hand domain containing			
5826	-83.05	kd	CGS001-771	CA12	Carbonic anhydrases			
5827	-83.07	cc		Toll like receptors LOF	-			
5828	-83.13	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
5829	-83.16	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
5830	-83.18	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
5831	-83.24	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
5832	-83.26	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
5833	-83.29	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
5834	-83.29	kd	CGS001-10641	NPRL2	-			
5835	-83.38	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5836	-83.41	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
5837	-83.45	kd	CGS001-10318	TNIP1	-			
5838	-83.51	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
5839	-83.53	kd	CGS001-51053	GMNN	-			
5840	-83.55	oe	ccsbBroad304_01654	TCTA	-			
5841	-83.55	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
5842	-83.59	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
5843	-83.61	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
5844	-83.64	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
5845	-83.64	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
5846	-83.64	kd	CGS001-59343	SENP2	-			
5847	-83.72	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
5848	-83.72	kd	CGS001-2034	EPAS1	Basic helix-loop-helix proteins			
5849	-83.78	oe	ccsbBroad304_13933	PSME2	Proteasome (prosome, macropain) subunits			
5850	-83.78	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5851	-83.8	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
5852	-83.83	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
5853	-83.84	kd	CGS001-6217	RPS16	S ribosomal proteins			
5854	-83.85	oe	ccsbBroad304_06680	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
5855	-83.86	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
5856	-83.87	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
5857	-83.88	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
5858	-83.88	kd	CGS001-5162	PDHB	-			
5859	-84.02	kd	CGS001-169026	SLC30A8	SLC30 zinc transporter family			
5860	-84.04	oe	ccsbBroad304_02789	ADAT1	-			
5861	-84.07	kd	CGS001-4175	MCM6	-			
5862	-84.09	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
5863	-84.12	oe	ccsbBroad304_00956	LYZ	-			
5864	-84.17	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
5865	-84.27	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
5866	-84.29	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
5867	-84.33	kd	CGS001-2277	FIGF	-			
5868	-84.39	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
5869	-84.39	kd	CGS001-2077	ERF	ETS Transcription Factors			
5870	-84.43	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
5871	-84.49	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
5872	-84.49	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
5873	-84.5	oe	ccsbBroad304_00690	GRN	-			
5874	-84.51	kd	CGS001-4179	CD46	CD molecules			
5875	-84.54	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
5876	-84.56	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
5877	-84.57	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
5878	-84.64	kd	CGS001-6189	RPS3A	S ribosomal proteins			
5879	-84.65	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
5880	-84.68	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
5881	-84.7	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
5882	-84.73	oe	ccsbBroad304_08797	FASTKD5	-			
5883	-84.77	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
5884	-84.84	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
5885	-84.85	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
5886	-84.85	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
5887	-84.86	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
5888	-84.88	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
5889	-84.88	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
5890	-84.89	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
5891	-84.95	cc		SMAD family LOF	-			
5892	-84.96	oe	ccsbBroad304_05980	CDKN1B	-			
5893	-85.02	oe	ccsbBroad304_11405	UBE3C	-			
5894	-85.02	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
5895	-85.02	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
5896	-85.04	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
5897	-85.04	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
5898	-85.05	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
5899	-85.06	kd	CGS001-10755	GIPC1	-			
5900	-85.09	kd	CGS001-85442	KNDC1	-			
5901	-85.12	kd	CGS001-1072	CFL1	-			
5902	-85.17	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
5903	-85.19	oe	ccsbBroad304_00118	ATIC	-			
5904	-85.19	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
5905	-85.23	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
5906	-85.23	kd	CGS001-51293	CD320	CD molecules			
5907	-85.25	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
5908	-85.26	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
5909	-85.27	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
5910	-85.34	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
5911	-85.35	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
5912	-85.41	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
5913	-85.44	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
5914	-85.44	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
5915	-85.45	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
5916	-85.54	oe	ccsbBroad304_00651	GNAI3	-			
5917	-85.59	cc		NFKB Activation GOF	-			
5918	-85.59	oe	ccsbBroad304_02313	ACTR3	-			
5919	-85.66	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
5920	-85.72	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
5921	-85.81	oe	ccsbBroad304_02398	LANCL1	-			
5922	-85.84	oe	ccsbBroad304_11910	RBM15B	RNA binding motif (RRM) containing			
5923	-85.85	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
5924	-85.85	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
5925	-85.88	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
5926	-85.9	oe	ccsbBroad304_07884	RYBP	-			
5927	-85.9	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
5928	-85.92	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
5929	-85.93	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5930	-85.95	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
5931	-85.97	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
5932	-85.99	oe	ccsbBroad304_07197	PDHX	-			
5933	-85.99	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
5934	-86.02	kd	CGS001-112858	TP53RK	Bud32 family			
5935	-86.05	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
5936	-86.08	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
5937	-86.11	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
5938	-86.16	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
5939	-86.2	kd	CGS001-5160	PDHA1	-			
5940	-86.22	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
5941	-86.24	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
5942	-86.3	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
5943	-86.3	kd	CGS001-4046	LSP1	-			
5944	-86.34	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
5945	-86.4	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
5946	-86.4	cp	BRD-K91370081	anisomycin	DNA synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	DNA synthesis inhibitor
5947	-86.44	kd	CGS001-1070	CETN3	EF-hand domain containing			
5948	-86.47	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
5949	-86.49	oe	ccsbBroad304_08935	CERS4	Homeoboxes / CERS class			
5950	-86.5	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
5951	-86.51	oe	ccsbBroad304_07050	TFAP2A	-			
5952	-86.53	kd	CGS001-10472	ZNF238	-			
5953	-86.63	kd	CGS001-83933	HDAC10	Histone deacetylases			
5954	-86.69	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
5955	-86.71	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
5956	-86.74	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
5957	-86.77	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
5958	-86.78	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
5959	-86.81	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
5960	-86.82	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
5961	-86.83	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
5962	-86.84	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
5963	-86.88	oe	ccsbBroad304_03618	OSGEP	-			
5964	-86.96	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
5965	-86.98	oe	ccsbBroad304_07760	KAT7	Histone acetyltransferases (HATs)			
5966	-86.99	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
5967	-87.01	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
5968	-87.03	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
5969	-87.05	oe	ccsbBroad304_01038	MSRA	-			
5970	-87.07	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
5971	-87.08	kd	CGS001-7165	TPD52L2	-			
5972	-87.1	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
5973	-87.12	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
5974	-87.12	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
5975	-87.13	oe	ccsbBroad304_02268	G3BP2	RNA binding motif (RRM) containing			
5976	-87.22	kd	CGS001-7077	TIMP2	-			
5977	-87.26	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
5978	-87.27	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
5979	-87.27	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
5980	-87.3	oe	ccsbBroad304_07761	CORO1A	Coronins			
5981	-87.34	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
5982	-87.34	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
5983	-87.35	kd	CGS001-4998	ORC1	ATPases / AAA-type			
5984	-87.4	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
5985	-87.4	kd	CGS001-8870	IER3	-			
5986	-87.41	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
5987	-87.44	kd	CGS001-9688	NUP93	-			
5988	-87.45	kd	CGS001-54541	DDIT4	-			
5989	-87.47	oe	ccsbBroad304_07071	TKT	-			
5990	-87.51	kd	CGS001-3029	HAGH	-			
5991	-87.52	kd	CGS001-23242	COBL	-			
5992	-87.54	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
5993	-87.54	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
5994	-87.55	oe	ccsbBroad304_02505	GNB5	WD repeat domain containing			
5995	-87.62	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
5996	-87.65	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
5997	-87.66	kd	CGS001-7982	ST7	-			
5998	-87.68	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
5999	-87.73	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
6000	-87.83	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
6001	-87.87	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
6002	-87.9	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
6003	-87.9	kd	CGS001-23670	TMEM2	-			
6004	-87.94	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
6005	-87.97	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
6006	-88.05	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
6007	-88.06	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
6008	-88.08	oe	ccsbBroad304_03647	CNDP2	Carnosine dipeptidase			
6009	-88.11	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
6010	-88.11	kd	CGS001-121599	SPIC	ETS Transcription Factors			
6011	-88.11	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
6012	-88.12	oe	ccsbBroad304_04114	SUV39H2	Histone methyltransferases (HMTs)			
6013	-88.13	oe	ccsbBroad304_07600	NSA2	-			
6014	-88.13	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
6015	-88.17	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
6016	-88.18	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
6017	-88.18	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
6018	-88.21	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
6019	-88.23	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
6020	-88.26	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
6021	-88.27	oe	ccsbBroad304_00486	EFNB2	Ephrins			
6022	-88.27	oe	ccsbBroad304_02340	SORBS3	-			
6023	-88.27	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
6024	-88.3	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
6025	-88.32	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6026	-88.34	kd	CGS001-2885	GRB2	SH2 domain containing			
6027	-88.35	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6028	-88.37	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
6029	-88.37	kd	CGS001-10673	TNFSF13B	CD molecules			
6030	-88.38	cc		Canonical high mobility group proteins LOF	-			
6031	-88.38	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
6032	-88.45	oe	ccsbBroad304_06801	PSMB10	Proteasome (prosome, macropain) subunits			
6033	-88.46	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
6034	-88.47	kd	CGS001-204851	HIPK1	HIPK subfamily			
6035	-88.49	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
6036	-88.5	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
6037	-88.5	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
6038	-88.52	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
6039	-88.57	cp	BRD-K53220666	trimetozine	Sedative			Sedative
6040	-88.61	cc		TGF beta receptor inhibitor	-			
6041	-88.67	kd	CGS001-637	BID	Endogenous ligands			
6042	-88.71	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
6043	-88.74	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
6044	-88.74	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
6045	-88.74	kd	CGS001-10775	POP4	-			
6046	-88.77	cc		PARP inhibitor	-			
6047	-88.86	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
6048	-88.89	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
6049	-88.9	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
6050	-88.93	oe	ccsbBroad304_00472	EBF1	-			
6051	-88.93	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
6052	-88.93	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
6053	-88.94	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
6054	-88.96	kd	CGS001-6184	RPN1	-			
6055	-88.96	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
6056	-88.97	kd	CGS001-327	APEH	Prolyl oligopeptidase			
6057	-88.99	kd	CGS001-2534	FYN	Src family			
6058	-89.04	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
6059	-89.09	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
6060	-89.15	kd	CGS001-2232	FDXR	-			
6061	-89.2	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
6062	-89.21	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
6063	-89.21	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
6064	-89.23	oe	ccsbBroad304_06789	PSEN2	Presenilin			
6065	-89.23	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
6066	-89.27	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
6067	-89.29	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
6068	-89.31	kd	CGS001-1632	ECI1	-			
6069	-89.32	oe	ccsbBroad304_02771	HEY1	Basic helix-loop-helix proteins			
6070	-89.32	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
6071	-89.39	oe	ccsbBroad304_07117	UGCG	Glycosyltransferase family 2 domain containing			
6072	-89.39	oe	ccsbBroad304_02677	PDAP1	-			
6073	-89.41	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
6074	-89.41	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
6075	-89.42	kd	CGS001-11319	ECD	-			
6076	-89.45	oe	ccsbBroad304_06639	NFYB	-			
6077	-89.55	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
6078	-89.56	oe	ccsbBroad304_00174	BRAF	RAF family			
6079	-89.58	oe	ccsbBroad304_01052	MYB	-			
6080	-89.58	oe	ccsbBroad304_00564	FGR	Src family			
6081	-89.61	oe	ccsbBroad304_01481	SARS	Aminoacyl tRNA synthetases / Class II			
6082	-89.66	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
6083	-89.67	oe	ccsbBroad304_07374	PTPLA	-			
6084	-89.67	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
6085	-89.68	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
6086	-89.74	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
6087	-89.78	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
6088	-89.84	oe	ccsbBroad304_07217	AXIN2	-			
6089	-89.86	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
6090	-89.86	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
6091	-89.86	kd	CGS001-7128	TNFAIP3	OTU domain containing			
6092	-89.92	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
6093	-89.93	cp	BRD-A25687296	emetine	Protein synthesis inhibitor		RPS2	Protein synthesis inhibitor
6094	-90.02	oe	ccsbBroad304_06301	GOT2	-			
6095	-90.02	kd	CGS001-9813	KIAA0494	-			
6096	-90.07	kd	CGS001-3939	LDHA	-			
6097	-90.08	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6098	-90.08	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
6099	-90.08	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
6100	-90.1	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
6101	-90.13	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
6102	-90.14	oe	ccsbBroad304_05791	AGT	Endogenous ligands			
6103	-90.18	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
6104	-90.18	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
6105	-90.18	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
6106	-90.2	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
6107	-90.2	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
6108	-90.22	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
6109	-90.23	oe	ccsbBroad304_09578	PASD1	-			
6110	-90.28	kd	CGS001-10587	TXNRD2	-			
6111	-90.29	oe	ccsbBroad304_01090	NFE2L2	basic leucine zipper proteins			
6112	-90.3	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
6113	-90.34	cc		PRD class homeoboxes and psudogenes LOF	-			
6114	-90.35	kd	CGS001-6772	STAT1	SH2 domain containing			
6115	-90.36	oe	ccsbBroad304_01337	PTHLH	Endogenous ligands			
6116	-90.4	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
6117	-90.41	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
6118	-90.54	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
6119	-90.57	cc		Norepinephrine reuptake inhibitor	-			
6120	-90.58	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
6121	-90.62	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
6122	-90.64	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
6123	-90.64	kd	CGS001-2581	GALC	-			
6124	-90.66	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
6125	-90.69	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
6126	-90.71	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
6127	-90.76	kd	CGS001-4697	NDUFA4	-			
6128	-90.78	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
6129	-90.83	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
6130	-90.83	kd	CGS001-51741	WWOX	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6131	-90.89	cp	BRD-K85133207	HDAC1-selective	HDAC inhibitor			HDAC inhibitor
6132	-90.94	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
6133	-90.94	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
6134	-90.95	oe	ccsbBroad304_00624	GCK	Hexokinases			
6135	-91	oe	ccsbBroad304_03179	BOLA1	-			
6136	-91.06	kd	CGS001-2879	GPX4	-			
6137	-91.08	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
6138	-91.12	kd	CGS001-2729	GCLC	-			
6139	-91.22	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
6140	-91.24	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
6141	-91.28	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
6142	-91.28	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
6143	-91.3	kd	CGS001-57404	CYP20A1	Cytochrome P450s			
6144	-91.31	cc		Trace amine receptors LOF	-			
6145	-91.34	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
6146	-91.34	kd	CGS001-54681	P4HTM	-			
6147	-91.36	oe	ccsbBroad304_00329	CLTA	-			
6148	-91.39	oe	ccsbBroad304_05947	CCNC	-			
6149	-91.46	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
6150	-91.48	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
6151	-91.56	oe	ccsbBroad304_07887	GCAT	-			
6152	-91.59	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
6153	-91.6	kd	CGS001-5684	PSMA3	Proteasome subunits			
6154	-91.62	kd	CGS001-55163	PNPO	-			
6155	-91.63	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
6156	-91.64	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
6157	-91.66	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
6158	-91.68	oe	ccsbBroad304_07727	LIAS	-			
6159	-91.73	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
6160	-91.75	oe	ccsbBroad304_07598	PEMT	-			
6161	-91.78	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6162	-91.79	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
6163	-91.8	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
6164	-91.8	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
6165	-91.84	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6166	-91.84	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
6167	-91.86	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
6168	-91.87	oe	ccsbBroad304_07337	TAF1B	-			
6169	-91.87	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
6170	-91.92	kd	CGS001-10020	GNE	-			
6171	-91.95	kd	CGS001-11014	KDELR2	-			
6172	-91.97	kd	CGS001-5914	RARA	Retinoic acid receptors			
6173	-91.98	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
6174	-91.99	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
6175	-92.01	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
6176	-92.02	cp	BRD-K50324045	avrainvillamide-analog-6	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6177	-92.02	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6178	-92.07	cp	BRD-K68488863	ENMD-2076	FLT3 inhibitor		AURKA, FLT3, KDR, PDGFRA, SRC, CSF1R, EPHA1, FGFR1, FGFR2, FGFR3, FLT4, KIT, PTK2	FLT3 inhibitor, VEGFR inhibitor, Aurora kinase inhibitor
6179	-92.11	oe	ccsbBroad304_02010	RIPK2	Receptor interacting protein kinase (RIPK) family			
6180	-92.11	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
6181	-92.13	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
6182	-92.13	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
6183	-92.2	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6184	-92.21	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
6185	-92.25	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
6186	-92.25	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
6187	-92.29	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
6188	-92.3	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
6189	-92.3	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
6190	-92.31	kd	CGS001-9637	FEZ2	-			
6191	-92.34	oe	ccsbBroad304_05894	BLVRA	-			
6192	-92.34	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
6193	-92.39	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
6194	-92.4	oe	ccsbBroad304_01189	PHF1	Zinc fingers, PHD-type			
6195	-92.41	kd	CGS001-375133	PI4KAP2	-			
6196	-92.44	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
6197	-92.45	kd	CGS001-5357	PLS1	EF-hand domain containing			
6198	-92.46	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
6199	-92.48	oe	ccsbBroad304_02087	PRPF4	WD repeat domain containing			
6200	-92.48	kd	CGS001-84365	MKI67IP	-			
6201	-92.48	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
6202	-92.5	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
6203	-92.53	kd	CGS001-8508	NIPSNAP1	-			
6204	-92.55	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
6205	-92.55	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
6206	-92.58	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
6207	-92.58	kd	CGS001-8741	TNFSF13	CD molecules			
6208	-92.59	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
6209	-92.62	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
6210	-92.66	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
6211	-92.69	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
6212	-92.71	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
6213	-92.72	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
6214	-92.73	kd	CGS001-8226	HDHD1	-			
6215	-92.79	kd	CGS001-11329	STK38	NDR family			
6216	-92.82	kd	CGS001-22933	SIRT2	Histone deacetylases			
6217	-92.83	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
6218	-92.84	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
6219	-92.85	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
6220	-92.86	kd	CGS001-56993	TOMM22	-			
6221	-92.86	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
6222	-92.87	oe	ccsbBroad304_02415	TUBB3	Tubulins			
6223	-92.87	kd	CGS001-55486	PARL	-			
6224	-92.88	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
6225	-92.93	oe	ccsbBroad304_07275	PSMG1	-			
6226	-92.94	cc		Serpin peptidase inhibitors LOF	-			
6227	-92.95	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
6228	-92.98	kd	CGS001-3476	IGBP1	-			
6229	-93.03	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
6230	-93.05	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
6231	-93.06	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
6232	-93.06	kd	CGS001-6208	RPS14	S ribosomal proteins			
6233	-93.07	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
6234	-93.11	cc		Potassium channel activator	-			
6235	-93.12	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
6236	-93.16	oe	ccsbBroad304_01584	SPARC	-			
6237	-93.16	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
6238	-93.18	kd	CGS001-6301	SARS	Aminoacyl tRNA synthetases / Class II			
6239	-93.19	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
6240	-93.23	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
6241	-93.25	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
6242	-93.26	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
6243	-93.3	oe	ccsbBroad304_03961	SMURF2	-			
6244	-93.31	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
6245	-93.35	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
6246	-93.36	oe	ccsbBroad304_02372	SPRY1	-			
6247	-93.4	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
6248	-93.4	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
6249	-93.43	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
6250	-93.45	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
6251	-93.52	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
6252	-93.55	kd	CGS001-10180	RBM6	G patch domain containing			
6253	-93.56	oe	ccsbBroad304_02864	PRDX5	-			
6254	-93.6	kd	CGS001-5573	PRKAR1A	Protein kinase A			
6255	-93.61	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
6256	-93.64	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
6257	-93.65	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
6258	-93.66	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
6259	-93.67	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
6260	-93.68	cc		Nucleophosmin inhibitor	-			
6261	-93.73	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
6262	-93.75	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
6263	-93.78	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
6264	-93.88	oe	ccsbBroad304_07124	UROD	-			
6265	-93.89	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
6266	-93.89	kd	CGS001-30001	ERO1L	-			
6267	-93.9	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
6268	-93.93	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
6269	-93.97	oe	ccsbBroad304_00789	HSBP1	-			
6270	-94.02	kd	CGS001-11267	SNF8	-			
6271	-94.06	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
6272	-94.06	kd	CGS001-375	ARF1	ADP-ribosylation factors			
6273	-94.06	kd	CGS001-338	APOB	Apolipoproteins			
6274	-94.09	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
6275	-94.11	kd	CGS001-54106	TLR9	Toll-like receptor family			
6276	-94.12	kd	CGS001-79139	DERL1	-			
6277	-94.13	kd	CGS001-284119	PTRF	-			
6278	-94.16	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
6279	-94.17	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
6280	-94.19	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
6281	-94.19	kd	CGS001-8772	FADD	-			
6282	-94.21	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
6283	-94.25	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
6284	-94.25	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
6285	-94.26	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
6286	-94.27	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
6287	-94.29	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
6288	-94.3	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
6289	-94.32	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
6290	-94.33	cc		Aurora kinase inhibitor	-			
6291	-94.33	kd	CGS001-3575	IL7R	IL-2 receptor family			
6292	-94.36	oe	ccsbBroad304_06888	RPN1	-			
6293	-94.37	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
6294	-94.37	kd	CGS001-527	ATP6V0C	ATPases / V-type			
6295	-94.38	kd	CGS001-10765	KDM5B	Histone demethylases			
6296	-94.39	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6297	-94.39	kd	CGS001-51586	MED15	-			
6298	-94.41	oe	ccsbBroad304_06286	GLUL	-			
6299	-94.42	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
6300	-94.43	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
6301	-94.44	kd	CGS001-26511	CHIC2	-			
6302	-94.45	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
6303	-94.46	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6304	-94.48	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
6305	-94.55	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
6306	-94.55	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
6307	-94.61	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
6308	-94.63	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
6309	-94.65	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
6310	-94.66	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
6311	-94.67	oe	ccsbBroad304_00533	FABP4	Fatty acid binding protein family			
6312	-94.67	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
6313	-94.71	kd	CGS001-6397	SEC14L1	-			
6314	-94.72	kd	CGS001-23581	CASP14	Caspases			
6315	-94.73	kd	CGS001-4074	M6PR	-			
6316	-94.73	kd	CGS001-54555	DDX49	DEAD-boxes			
6317	-94.78	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
6318	-94.78	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
6319	-94.78	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6320	-94.78	kd	CGS001-1062	CENPE	Kinesins			
6321	-94.79	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6322	-94.8	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6323	-94.83	kd	CGS001-190	NR0B1	DAX-like receptors			
6324	-94.86	cc		Estrogen receptor antagonist	-			
6325	-94.89	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
6326	-94.93	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
6327	-94.94	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
6328	-94.94	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
6329	-94.99	kd	CGS001-9710	KIAA0355	-			
6330	-95	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
6331	-95.04	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
6332	-95.05	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
6333	-95.05	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
6334	-95.09	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
6335	-95.09	kd	CGS001-25885	POLR1A	RNA polymerase subunits			
6336	-95.09	kd	CGS001-35	ACADS	-			
6337	-95.1	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
6338	-95.12	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
6339	-95.12	kd	CGS001-56005	C19ORF10	-			
6340	-95.15	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
6341	-95.17	cp	BRD-K42573370	avrainvillamide-analog-2	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6342	-95.22	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
6343	-95.3	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
6344	-95.33	oe	ccsbBroad304_01768	VEGFA	Cytokines and growth factors			
6345	-95.33	kd	CGS001-10491	CRTAP	-			
6346	-95.34	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
6347	-95.36	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
6348	-95.4	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
6349	-95.44	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
6350	-95.44	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
6351	-95.45	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
6352	-95.46	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
6353	-95.47	oe	ccsbBroad304_01662	TFDP2	-			
6354	-95.47	kd	CGS001-8396	PIP4K2B	1-phosphatidylinositol-5-phosphate 4-kinase family			
6355	-95.49	kd	CGS001-4849	CNOT3	-			
6356	-95.51	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
6357	-95.51	oe	ccsbBroad304_00645	GCLM	-			
6358	-95.52	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
6359	-95.52	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
6360	-95.53	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
6361	-95.55	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
6362	-95.56	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
6363	-95.61	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
6364	-95.63	kd	CGS001-9512	PMPCB	-			
6365	-95.67	oe	ccsbBroad304_02402	TMEM5	-			
6366	-95.67	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
6367	-95.69	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
6368	-95.69	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
6369	-95.71	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
6370	-95.72	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6371	-95.72	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
6372	-95.73	kd	CGS001-3832	KIF11	Kinesins			
6373	-95.75	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6374	-95.77	oe	ccsbBroad304_00223	CASP9	Caspases			
6375	-95.78	kd	CGS001-1499	CTNNB1	Catenins			
6376	-95.8	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
6377	-95.8	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
6378	-95.8	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
6379	-95.8	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
6380	-95.8	kd	CGS001-9441	MED26	-			
6381	-95.81	kd	CGS001-9	NAT1	-			
6382	-95.83	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
6383	-95.86	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6384	-95.89	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6385	-95.92	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6386	-95.95	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
6387	-95.96	oe	ccsbBroad304_07118	UGDH	-			
6388	-95.96	kd	CGS001-1999	ELF3	ETS Transcription Factors			
6389	-95.97	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
6390	-96	oe	ccsbBroad304_00980	MBNL1	Zinc fingers, CCCH-type domain containing			
6391	-96.01	oe	ccsbBroad304_00282	CDKN1A	-			
6392	-96.03	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
6393	-96.03	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6394	-96.05	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
6395	-96.07	oe	ccsbBroad304_07119	UGP2	-			
6396	-96.07	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
6397	-96.07	kd	CGS001-3508	IGHMBP2	Zinc fingers, AN1-type domain containing			
6398	-96.08	cc		Ribosomal 40s Subunit LOF	-			
6399	-96.1	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
6400	-96.1	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
6401	-96.13	kd	CGS001-1131	CHRM3	Cholinergic receptors			
6402	-96.14	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
6403	-96.16	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
6404	-96.17	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
6405	-96.18	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
6406	-96.19	kd	CGS001-7126	TNFAIP1	BTB/POZ domain containing			
6407	-96.23	kd	CGS001-8996	NOL3	-			
6408	-96.24	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
6409	-96.24	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
6410	-96.24	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
6411	-96.24	kd	CGS001-2864	FFAR1	Fatty acid receptors			
6412	-96.28	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
6413	-96.29	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6414	-96.3	oe	ccsbBroad304_02143	CNOT8	-			
6415	-96.3	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6416	-96.31	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
6417	-96.33	cp	BRD-A83237092	fulvestrant	Estrogen receptor antagonist		ESR1, EPHX2, ESR2, GPER1	Estrogen receptor antagonist
6418	-96.33	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
6419	-96.34	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
6420	-96.35	oe	ccsbBroad304_07008	STAT5A	SH2 domain containing			
6421	-96.36	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
6422	-96.37	cc		Minor histocompatibility antigens LOF	-			
6423	-96.37	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
6424	-96.38	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
6425	-96.43	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
6426	-96.44	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6427	-96.45	oe	ccsbBroad304_03746	CDC42SE1	-			
6428	-96.48	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
6429	-96.48	oe	ccsbBroad304_02243	DLGAP5	-			
6430	-96.49	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
6431	-96.49	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
6432	-96.52	oe	ccsbBroad304_04038	ELOVL6	-			
6433	-96.52	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
6434	-96.52	kd	CGS001-5108	PCM1	-			
6435	-96.54	oe	ccsbBroad304_01304	PSEN1	Presenilin			
6436	-96.54	kd	CGS001-23076	RRP1B	-			
6437	-96.55	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
6438	-96.55	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
6439	-96.56	oe	ccsbBroad304_02840	PISD	Decarboxylases			
6440	-96.6	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
6441	-96.6	oe	ccsbBroad304_02292	BCL2L11	-			
6442	-96.6	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
6443	-96.61	kd	CGS001-55278	QRSL1	-			
6444	-96.61	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
6445	-96.62	oe	ccsbBroad304_01532	SIAH1	-			
6446	-96.63	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
6447	-96.65	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
6448	-96.67	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
6449	-96.69	oe	ccsbBroad304_07814	SACM1L	-			
6450	-96.72	kd	CGS001-25	ABL1	Abl family			
6451	-96.73	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
6452	-96.73	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
6453	-96.74	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
6454	-96.75	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
6455	-96.75	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
6456	-96.75	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
6457	-96.77	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
6458	-96.79	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
6459	-96.79	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
6460	-96.81	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
6461	-96.81	kd	CGS001-25842	ASF1A	-			
6462	-96.82	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
6463	-96.83	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
6464	-96.83	kd	CGS001-6194	RPS6	S ribosomal proteins			
6465	-96.85	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
6466	-96.88	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
6467	-96.9	cc		T-type calcium channel blocker	-			
6468	-96.91	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
6469	-96.93	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
6470	-96.93	kd	CGS001-10873	ME3	-			
6471	-96.94	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
6472	-96.95	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
6473	-96.96	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
6474	-96.98	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
6475	-96.98	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
6476	-97	kd	CGS001-10898	CPSF4	-			
6477	-97.01	oe	ccsbBroad304_00068	SLC25A6	Mitochondrial nucleotide transporter subfamily			
6478	-97.04	kd	CGS001-5292	PIM1	PIM family			
6479	-97.05	oe	ccsbBroad304_00316	CKS1B	-			
6480	-97.05	kd	CGS001-23753	SDF2L1	-			
6481	-97.06	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
6482	-97.06	kd	CGS001-23118	TAB2	-			
6483	-97.08	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
6484	-97.08	kd	CGS001-11019	LIAS	-			
6485	-97.08	kd	CGS001-10538	BATF	basic leucine zipper proteins			
6486	-97.09	oe	ccsbBroad304_07466	VGLL4	-			
6487	-97.1	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
6488	-97.1	kd	CGS001-29915	HCFC2	-			
6489	-97.12	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
6490	-97.14	oe	ccsbBroad304_07592	CEPT1	-			
6491	-97.15	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
6492	-97.15	kd	CGS001-2966	GTF2H2	General transcription factors			
6493	-97.16	kd	CGS001-3672	ITGA1	Integrins			
6494	-97.18	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
6495	-97.2	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
6496	-97.22	oe	ccsbBroad304_07101	TSC2	-			
6497	-97.22	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
6498	-97.23	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
6499	-97.25	oe	ccsbBroad304_00313	TBCB	-			
6500	-97.26	kd	CGS001-81533	ITFG1	-			
6501	-97.29	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
6502	-97.31	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
6503	-97.31	kd	CGS001-55634	ZNF673	-			
6504	-97.34	cc		Cell Cycle Inhibition GOF	-			
6505	-97.38	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
6506	-97.4	kd	CGS001-11315	PARK7	Parkinson disease			
6507	-97.44	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
6508	-97.45	kd	CGS001-10427	SEC24B	-			
6509	-97.45	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
6510	-97.46	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
6511	-97.47	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
6512	-97.48	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
6513	-97.49	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
6514	-97.5	oe	ccsbBroad304_00147	BAG1	-			
6515	-97.51	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
6516	-97.54	kd	CGS001-9296	ATP6V1F	ATPases / V-type			
6517	-97.56	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
6518	-97.56	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
6519	-97.58	kd	CGS001-6599	SMARCC1	-			
6520	-97.58	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
6521	-97.6	cc		HIF activator	-			
6522	-97.62	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
6523	-97.63	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
6524	-97.64	oe	ccsbBroad304_00518	ETFA	-			
6525	-97.65	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
6526	-97.67	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
6527	-97.7	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
6528	-97.7	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
6529	-97.7	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
6530	-97.72	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6531	-97.73	oe	ccsbBroad304_01347	RAD1	-			
6532	-97.74	kd	CGS001-7840	ALMS1	-			
6533	-97.76	kd	CGS001-6193	RPS5	S ribosomal proteins			
6534	-97.78	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
6535	-97.79	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
6536	-97.8	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
6537	-97.81	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6538	-97.81	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
6539	-97.81	kd	CGS001-5423	POLB	DNA polymerases			
6540	-97.81	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
6541	-97.82	kd	CGS001-1399	CRKL	SH2 domain containing			
6542	-97.84	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
6543	-97.85	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
6544	-97.85	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
6545	-97.86	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
6546	-97.87	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
6547	-97.88	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
6548	-97.9	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
6549	-97.92	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6550	-97.92	kd	CGS001-2266	FGG	Endogenous ligands			
6551	-97.94	oe	ccsbBroad304_03122	RHOD	-			
6552	-97.96	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
6553	-97.97	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
6554	-97.97	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
6555	-98	kd	CGS001-7485	WRB	-			
6556	-98.05	cc		CCK receptor antagonist	-			
6557	-98.06	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
6558	-98.09	oe	ccsbBroad304_01632	SYPL1	-			
6559	-98.09	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
6560	-98.12	kd	CGS001-1152	CKB	-			
6561	-98.14	kd	CGS001-275	AMT	-			
6562	-98.15	kd	CGS001-222546	RFX6	-			
6563	-98.17	cc		Structural maintenance of chromosomes proteins LOF	-			
6564	-98.17	oe	ccsbBroad304_00184	C2	Complement system			
6565	-98.17	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
6566	-98.18	oe	ccsbBroad304_02370	HRSP12	-			
6567	-98.19	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
6568	-98.2	kd	CGS001-9183	ZW10	-			
6569	-98.22	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
6570	-98.24	cc		DNA dependent protein kinase inhibitor	-			
6571	-98.25	kd	CGS001-302	ANXA2	Annexins			
6572	-98.28	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
6573	-98.28	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
6574	-98.28	kd	CGS001-4351	MPI	-			
6575	-98.29	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
6576	-98.3	cc		Thromboxane receptor antagonist	-			
6577	-98.31	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
6578	-98.31	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
6579	-98.32	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
6580	-98.33	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
6581	-98.35	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
6582	-98.35	oe	ccsbBroad304_09756	PAQR7	-			
6583	-98.36	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6584	-98.37	cc		Ribonucleotide reductase inhibitor	-			
6585	-98.37	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
6586	-98.37	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
6587	-98.37	kd	CGS001-124535	HSF5	-			
6588	-98.38	oe	ccsbBroad304_00519	ETFB	-			
6589	-98.38	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
6590	-98.39	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
6591	-98.4	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
6592	-98.41	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
6593	-98.41	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
6594	-98.42	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
6595	-98.42	kd	CGS001-55536	CDCA7L	-			
6596	-98.43	oe	ccsbBroad304_01672	TIMP2	-			
6597	-98.44	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
6598	-98.44	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
6599	-98.44	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
6600	-98.44	oe	ccsbBroad304_02298	DNM1L	-			
6601	-98.46	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
6602	-98.46	oe	ccsbBroad304_06103	DMD	-			
6603	-98.46	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
6604	-98.46	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
6605	-98.47	oe	ccsbBroad304_02581	ASCC3	-			
6606	-98.48	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
6607	-98.48	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
6608	-98.5	oe	ccsbBroad304_02249	KIAA0494	-			
6609	-98.51	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
6610	-98.53	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
6611	-98.54	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
6612	-98.54	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
6613	-98.56	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
6614	-98.56	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
6615	-98.58	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6616	-98.59	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
6617	-98.6	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6618	-98.6	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
6619	-98.6	kd	CGS001-4723	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
6620	-98.61	kd	CGS001-4199	ME1	-			
6621	-98.63	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
6622	-98.64	oe	ccsbBroad304_03197	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
6623	-98.65	cc		Dopamine receptor antagonist	-			
6624	-98.65	cp	BRD-K61691971	avrainvillamide-analog-1	nucleophosmin inhibitor		NPM1	nucleophosmin inhibitor
6625	-98.66	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
6626	-98.66	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
6627	-98.67	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
6628	-98.67	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
6629	-98.68	kd	CGS001-25987	TSKU	-			
6630	-98.68	kd	CGS001-5932	RBBP8	-			
6631	-98.69	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
6632	-98.71	kd	CGS001-6197	RPS6KA3	RSK subfamily			
6633	-98.72	oe	ccsbBroad304_05590	NOTCH2NL	-			
6634	-98.72	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
6635	-98.73	cc		MTOR inhibitor	-			
6636	-98.73	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
6637	-98.74	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
6638	-98.75	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
6639	-98.76	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
6640	-98.76	oe	ccsbBroad304_00401	CYB5A	Cytochrome b genes			
6641	-98.77	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
6642	-98.78	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
6643	-98.78	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
6644	-98.81	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
6645	-98.81	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
6646	-98.82	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
6647	-98.83	kd	CGS001-55746	NUP133	-			
6648	-98.85	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
6649	-98.85	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
6650	-98.87	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
6651	-98.87	kd	CGS001-2100	ESR2	Estrogen receptors			
6652	-98.87	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
6653	-98.88	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
6654	-98.88	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
6655	-98.88	kd	CGS001-347736	NME9	-			
6656	-98.88	kd	CGS001-3281	HSBP1	-			
6657	-98.91	oe	ccsbBroad304_01951	BLZF1	-			
6658	-98.91	kd	CGS001-3383	ICAM1	CD molecules			
6659	-98.92	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
6660	-98.92	kd	CGS001-7082	TJP1	-			
6661	-98.93	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
6662	-98.93	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
6663	-98.93	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
6664	-98.94	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6665	-98.94	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
6666	-98.94	kd	CGS001-1902	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
6667	-98.96	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
6668	-98.97	oe	ccsbBroad304_02605	PAPD7	-			
6669	-98.98	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
6670	-98.98	kd	CGS001-23244	PDS5A	-			
6671	-98.98	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
6672	-99	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
6673	-99.01	cc		V type ATPases LOF	-			
6674	-99.02	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
6675	-99.03	kd	CGS001-7100	TLR5	Toll-like receptor family			
6676	-99.03	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6677	-99.03	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
6678	-99.04	oe	ccsbBroad304_02592	KIF2C	Kinesins			
6679	-99.04	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
6680	-99.07	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6681	-99.07	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
6682	-99.07	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
6683	-99.07	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
6684	-99.07	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
6685	-99.08	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
6686	-99.09	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
6687	-99.09	kd	CGS001-126823	KLHDC9	-			
6688	-99.1	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
6689	-99.11	kd	CGS001-310	ANXA7	Annexins			
6690	-99.12	oe	ccsbBroad304_03817	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
6691	-99.12	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
6692	-99.12	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6693	-99.13	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6694	-99.13	kd	CGS001-54386	TERF2IP	-			
6695	-99.14	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
6696	-99.14	kd	CGS001-56882	CDC42SE1	-			
6697	-99.15	kd	CGS001-54438	GFOD1	-			
6698	-99.16	cc		Purinergic receptors P2Y GOF	-			
6699	-99.16	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
6700	-99.16	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
6701	-99.16	kd	CGS001-4089	SMAD4	SMADs			
6702	-99.16	kd	CGS001-3265	HRAS	RAS subfamily			
6703	-99.17	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6704	-99.18	oe	ccsbBroad304_01663	TFF2	-			
6705	-99.18	oe	ccsbBroad304_00794	HSF1	-			
6706	-99.19	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
6707	-99.19	kd	CGS001-27035	NOX1	-			
6708	-99.21	kd	CGS001-7056	THBD	CD molecules			
6709	-99.21	kd	CGS001-3930	LBR	Tudor domain containing			
6710	-99.22	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
6711	-99.22	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
6712	-99.23	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
6713	-99.23	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
6714	-99.23	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
6715	-99.25	kd	CGS001-7003	TEAD1	-			
6716	-99.25	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
6717	-99.26	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
6718	-99.26	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
6719	-99.26	kd	CGS001-7054	TH	Amino acid hydroxylases			
6720	-99.27	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
6721	-99.27	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
6722	-99.27	kd	CGS001-213	ALB	-			
6723	-99.28	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
6724	-99.28	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
6725	-99.28	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
6726	-99.28	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
6727	-99.31	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
6728	-99.31	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
6729	-99.31	kd	CGS001-2313	FLI1	ETS Transcription Factors			
6730	-99.32	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
6731	-99.33	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
6732	-99.33	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
6733	-99.34	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
6734	-99.34	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
6735	-99.35	cc		Nucleoporin LOF	-			
6736	-99.35	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
6737	-99.35	kd	CGS001-23510	KCTD2	-			
6738	-99.35	oe	ccsbBroad304_05963	CD44	CD molecules			
6739	-99.36	oe	ccsbBroad304_01764	VDAC1	Voltage-dependent anion channels			
6740	-99.36	kd	CGS001-2810	SFN	-			
6741	-99.37	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
6742	-99.37	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
6743	-99.37	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
6744	-99.37	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
6745	-99.37	kd	CGS001-2235	FECH	-			
6746	-99.4	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
6747	-99.4	kd	CGS001-6016	RIT1	-			
6748	-99.4	kd	CGS001-8780	RIOK3	RIO3 subfamily			
6749	-99.41	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
6750	-99.41	kd	CGS001-79902	NUP85	-			
6751	-99.42	kd	CGS001-55526	DHTKD1	-			
6752	-99.43	oe	ccsbBroad304_06992	SRC	Src family			
6753	-99.43	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
6754	-99.44	oe	ccsbBroad304_02230	HERPUD1	-			
6755	-99.44	kd	CGS001-85480	TSLP	-			
6756	-99.45	oe	ccsbBroad304_03420	TOLLIP	-			
6757	-99.45	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
6758	-99.46	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
6759	-99.47	oe	ccsbBroad304_00038	AGL	-			
6760	-99.47	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
6761	-99.47	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
6762	-99.47	kd	CGS001-10797	MTHFD2	-			
6763	-99.48	oe	ccsbBroad304_01102	NMT1	-			
6764	-99.48	oe	ccsbBroad304_07145	ZFP161	-			
6765	-99.5	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
6766	-99.5	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
6767	-99.51	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
6768	-99.51	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
6769	-99.51	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
6770	-99.51	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
6771	-99.53	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
6772	-99.53	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6773	-99.53	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
6774	-99.54	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
6775	-99.56	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
6776	-99.56	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
6777	-99.56	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
6778	-99.56	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
6779	-99.57	oe	ccsbBroad304_07363	AIFM1	-			
6780	-99.57	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6781	-99.57	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
6782	-99.57	kd	CGS001-158	ADSL	-			
6783	-99.58	kd	CGS001-842	CASP9	Caspases			
6784	-99.59	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6785	-99.59	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
6786	-99.59	kd	CGS001-23081	KDM4C	Histone demethylases			
6787	-99.59	oe	ccsbBroad304_00238	CCNE1	-			
6788	-99.6	oe	ccsbBroad304_07412	ZRANB2	Zinc fingers, RAN-binding domain containing			
6789	-99.6	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
6790	-99.6	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
6791	-99.6	kd	CGS001-5033	P4HA1	-			
6792	-99.6	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
6793	-99.6	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
6794	-99.6	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
6795	-99.62	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
6796	-99.62	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
6797	-99.62	kd	CGS001-8727	CTNNAL1	Catenins			
6798	-99.62	oe	ccsbBroad304_00551	FECH	-			
6799	-99.63	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
6800	-99.63	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
6801	-99.63	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
6802	-99.63	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
6803	-99.63	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
6804	-99.64	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
6805	-99.65	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
6806	-99.65	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
6807	-99.65	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6808	-99.65	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
6809	-99.66	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
6810	-99.68	cc		AHSP Pathway LOF	-			
6811	-99.68	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
6812	-99.69	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
6813	-99.69	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
6814	-99.69	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
6815	-99.69	kd	CGS001-5829	PXN	-			
6816	-99.69	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
6817	-99.69	kd	CGS001-256281	NUDT14	Nudix motif containing			
6818	-99.7	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
6819	-99.71	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
6820	-99.71	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
6821	-99.72	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
6822	-99.72	kd	CGS001-51172	NAGPA	-			
6823	-99.73	oe	ccsbBroad304_08878	METTL4	-			
6824	-99.73	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
6825	-99.73	oe	ccsbBroad304_00499	ELK3	ETS Transcription Factors			
6826	-99.73	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
6827	-99.75	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
6828	-99.75	kd	CGS001-83999	KREMEN1	-			
6829	-99.75	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
6830	-99.76	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
6831	-99.78	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
6832	-99.78	kd	CGS001-51750	RTEL1	-			
6833	-99.78	kd	CGS001-673	BRAF	RAF family			
6834	-99.79	oe	ccsbBroad304_02271	LPGAT1	-			
6835	-99.79	oe	ccsbBroad304_09054	EGFL8	-			
6836	-99.79	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
6837	-99.79	kd	CGS001-84619	ZGPAT	G patch domain containing			
6838	-99.79	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
6839	-99.81	oe	ccsbBroad304_00420	DAP	-			
6840	-99.81	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
6841	-99.81	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
6842	-99.81	kd	CGS001-10128	LRPPRC	-			
6843	-99.82	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
6844	-99.82	oe	ccsbBroad304_04457	TOX2	-			
6845	-99.82	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
6846	-99.82	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
6847	-99.84	cp	BRD-A60070924	alpha-estradiol	Estrogen receptor agonist		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Estrogen receptor agonist
6848	-99.84	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
6849	-99.84	oe	ccsbBroad304_03056	MCTS1	-			
6850	-99.84	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
6851	-99.84	kd	CGS001-55662	HIF1AN	-			
6852	-99.84	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
6853	-99.84	kd	CGS001-1503	CTPS	-			
6854	-99.84	kd	CGS001-847	CAT	-			
6855	-99.85	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
6856	-99.85	oe	ccsbBroad304_00832	IFNB1	Interferons			
6857	-99.85	kd	CGS001-6464	SHC1	SH2 domain containing			
6858	-99.85	kd	CGS001-2147	F2	Endogenous ligands			
6859	-99.85	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6860	-99.85	kd	CGS001-113451	ADC	-			
6861	-99.87	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
6862	-99.87	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
6863	-99.87	oe	ccsbBroad304_06494	KLRC1	CD molecules			
6864	-99.87	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
6865	-99.87	oe	ccsbBroad304_08952	E2F8	-			
6866	-99.87	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6867	-99.88	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
6868	-99.88	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
6869	-99.88	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
6870	-99.88	kd	CGS001-4782	NFIC	-			
6871	-99.88	kd	CGS001-2967	GTF2H3	General transcription factors			
6872	-99.9	oe	ccsbBroad304_03658	DCP1A	-			
6873	-99.9	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
6874	-99.9	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
6875	-99.9	kd	CGS001-2767	GNA11	-			
6876	-99.9	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
6877	-99.9	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
6878	-99.91	oe	ccsbBroad304_05183	TXLNA	-			
6879	-99.91	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
6880	-99.91	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
6881	-99.91	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
6882	-99.91	kd	CGS001-6810	STX4	-			
6883	-99.91	kd	CGS001-5255	PHKA1	-			
6884	-99.91	oe	ccsbBroad304_06464	ITGB2	Integrins			
6885	-99.93	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
6886	-99.93	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
6887	-99.93	kd	CGS001-1163	CKS1B	-			
6888	-99.93	kd	CGS001-9133	CCNB2	-			
6889	-99.93	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
6890	-99.94	cc		MCM family LOF	-			
6891	-99.94	cc		DNA polymerase inhibitor	-			
6892	-99.94	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
6893	-99.94	oe	ccsbBroad304_08137	HOOK2	-			
6894	-99.94	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
6895	-99.94	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
6896	-99.94	kd	CGS001-7089	TLE2	WD repeat domain containing			
6897	-99.94	kd	CGS001-81539	SLC38A1	System A-like transporters			
6898	-99.94	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
6899	-99.94	kd	CGS001-5763	PTMS	-			
6900	-99.94	kd	CGS001-5580	PRKCD	Delta subfamily			
6901	-99.94	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
6902	-99.94	kd	CGS001-2160	F11	Chymotrypsin			
6903	-99.94	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
6904	-99.96	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
6905	-99.96	oe	ccsbBroad304_08152	PSAT1	-			
6906	-99.96	oe	ccsbBroad304_02440	PPIE	RNA binding motif (RRM) containing			
6907	-99.96	oe	ccsbBroad304_01211	PKM2	-			
6908	-99.96	oe	ccsbBroad304_00632	GGCX	Carboxylases			
6909	-99.96	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
6910	-99.96	oe	ccsbBroad304_00077	APEX1	-			
6911	-99.96	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6912	-99.96	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
6913	-99.96	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
6914	-99.96	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
6915	-99.96	kd	CGS001-29074	MRPL18	Mitochondrial ribosomal proteins / large subunits			
6916	-99.96	kd	CGS001-3985	LIMK2	LIMK subfamily			
6917	-99.96	kd	CGS001-64170	CARD9	-			
6918	-99.97	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
6919	-99.97	oe	ccsbBroad304_01222	PLP2	-			
6920	-99.97	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
6921	-99.97	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
6922	-99.97	oe	ccsbBroad304_00446	DKC1	-			
6923	-99.97	oe	ccsbBroad304_00376	CSK	Csk family			
6924	-99.97	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
6925	-99.97	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
6926	-99.97	oe	ccsbBroad304_02405	TFG	-			
6927	-99.97	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
6928	-99.97	oe	ccsbBroad304_01469	RSU1	-			
6929	-99.97	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
6930	-99.97	oe	ccsbBroad304_02676	PHB2	-			
6931	-99.97	oe	ccsbBroad304_01034	MSH2	-			
6932	-99.97	oe	ccsbBroad304_07724	KDELR2	-			
6933	-99.97	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
6934	-99.97	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
6935	-99.97	oe	ccsbBroad304_03177	FIS1	-			
6936	-99.97	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
6937	-99.97	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
6938	-99.97	oe	ccsbBroad304_08392	EXOC6	-			
6939	-99.97	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
6940	-99.97	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
6941	-99.97	oe	ccsbBroad304_00146	BAD	-			
6942	-99.97	oe	ccsbBroad304_02173	ATG5	-			
6943	-99.97	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
6944	-99.97	oe	ccsbBroad304_00106	ARRB1	-			
6945	-99.97	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
6946	-99.97	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
6947	-99.97	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
6948	-99.97	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
6949	-99.97	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
6950	-99.97	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6951	-99.97	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
6952	-99.97	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
6953	-99.97	kd	CGS001-6188	RPS3	S ribosomal proteins			
6954	-99.97	kd	CGS001-63891	RNF123	RING-type (C3HC4) zinc fingers			
6955	-99.97	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
6956	-99.97	kd	CGS001-4893	NRAS	RAS subfamily			
6957	-99.97	kd	CGS001-4174	MCM5	-			
6958	-99.97	kd	CGS001-3920	LAMP2	CD molecules			
6959	-99.97	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
6960	-99.97	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
6961	-99.97	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
6962	-99.97	kd	CGS001-79071	ELOVL6	-			
6963	-99.97	kd	CGS001-8900	CCNA1	-			
6964	-99.97	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
6965	-99.97	oe	ccsbBroad304_04726	TAGAP	Rho GTPase activating proteins			
6966	-99.99	oe	ccsbBroad304_07506	UBAP2L	-			
6967	-100	cp	BRD-K79877282	PF-543	Sphingosine kinase inhibitor		SPHK1	Sphingosine kinase inhibitor
6968	-100	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
6969	-100	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
6970	-100	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
6971	-100	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
6972	-100	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
