Rank	Score	Type	ID	Name	Description	CMap Class	Target	MOA
1	100	cc		Serpin peptidase inhibitors LOF	-			
2	100	cc		DNA polymerase inhibitor	-			
3	100	cc		Benzodiazepine receptor agonist	-			
4	100	cp	BRD-K89348303	ramipril	ACE inhibitor		ACE	ACE inhibitor
5	100	cp	BRD-K55591206	epigallocatechin	Nitric oxide synthase inhibitor		FASN, APP, BACE1, CYP19A1, DYRK1A, ELANE, ENOX2, EP300, IDO1, KAT2B, KDR, MMP14, MMP2, PPARA, PREP, SLC5A1	Nitric oxide synthase inhibitor, Bacterial DNA gyrase inhibitor
6	100	cp	BRD-K61217870	n-(3-acetamidophenyl)-3-chlorobenzamide	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
7	100	cp	BRD-K01779529	fluoropyruvate	Pyruvate dehydrogenase kinase inhibitor			Pyruvate dehydrogenase kinase inhibitor
8	100	cp	BRD-A48430263	pioglitazone	Insulin sensitizer		PPARG, INS, TRPM3	Insulin sensitizer, PPAR receptor agonist
9	100	kd	CGS001-25925	ZNF521	Zinc fingers, C2H2-type			
10	100	kd	CGS001-162655	ZNF519	Zinc fingers, C2H2-type			
11	100	kd	CGS001-9925	ZBTB5	BTB/POZ domain containing			
12	100	kd	CGS001-9097	USP14	Ubiquitin-specific peptidases			
13	100	kd	CGS001-7381	UQCRB	Mitochondrial respiratory chain complex / Complex III			
14	100	kd	CGS001-7334	UBE2N	Ubiquitin-conjugating enzymes E2			
15	100	kd	CGS001-5987	TRIM27	-			
16	100	kd	CGS001-55504	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
17	100	kd	CGS001-333929	SNAI3	Snail homologs			
18	100	kd	CGS001-6584	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
19	100	kd	CGS001-51804	SIX4	Homeoboxes / SINE class			
20	100	kd	CGS001-5268	SERPINB5	Serine (or cysteine) peptidase inhibitors			
21	100	kd	CGS001-8766	RAB11A	RAB, member RAS oncogene			
22	100	kd	CGS001-5688	PSMA7	Proteasome subunits			
23	100	kd	CGS001-5534	PPP3R1	EF-hand domain containing			
24	100	kd	CGS001-5194	PEX13	-			
25	100	kd	CGS001-54681	P4HTM	-			
26	100	kd	CGS001-347736	NME9	-			
27	100	kd	CGS001-10608	MXD4	Basic helix-loop-helix proteins			
28	100	kd	CGS001-4548	MTR	-			
29	100	kd	CGS001-4212	MEIS2	Homeoboxes / TALE class			
30	100	kd	CGS001-4067	LYN	Src family			
31	100	kd	CGS001-59352	LGR6	GPCR / Class A : Orphans			
32	100	kd	CGS001-3856	KRT8	Intermediate filaments type II, keratins (basic)			
33	100	kd	CGS001-1316	KLF6	Kruppel-like transcription factors			
34	100	kd	CGS001-3664	IRF6	-			
35	100	kd	CGS001-3297	HSF1	-			
36	100	kd	CGS001-3217	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
37	100	kd	CGS001-2882	GPX7	-			
38	100	kd	CGS001-51292	GMPR2	-			
39	100	kd	CGS001-8322	FZD4	GPCR / Class F : Frizzled receptors			
40	100	kd	CGS001-1112	FOXN3	Forkhead boxes			
41	100	kd	CGS001-2280	FKBP1A	Cis-trans-isomerases			
42	100	kd	CGS001-2172	FABP6	Fatty acid binding protein family			
43	100	kd	CGS001-54821	ERCC6L	-			
44	100	kd	CGS001-55723	ASF1B	-			
45	100	kd	CGS001-2	A2M	-			
46	100	cp	BRD-K15502390	nevirapine	Reverse transcriptase inhibitor		CYP2B6, CYP2C19, CYP3A4	Reverse transcriptase inhibitor
47	99.98	kd	CGS001-55148	UBR7	Ubiquitin protein ligase E3 component n-recognins			
48	99.98	kd	CGS001-9319	TRIP13	ATPases / AAA-type			
49	99.98	kd	CGS001-55234	SMU1	WD repeat domain containing			
50	99.98	kd	CGS001-8503	PIK3R3	Phosphatidylinositol kinases			
51	99.98	kd	CGS001-4836	NMT1	-			
52	99.98	kd	CGS001-308	ANXA5	Annexins			
53	99.98	kd	CGS001-81611	ANP32E	ANP32 acidic nuclear phosphoproteins			
54	99.96	oe	ccsbBroad304_01425	RPL22	L ribosomal proteins			
55	99.96	oe	ccsbBroad304_02002	RNMT	-			
56	99.96	oe	ccsbBroad304_02115	PTTG1	-			
57	99.96	oe	ccsbBroad304_02336	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
58	99.96	oe	ccsbBroad304_00903	KCNQ1	Voltage-gated potassium channels			
59	99.96	oe	ccsbBroad304_00841	IKBKB	IKK family			
60	99.96	oe	ccsbBroad304_06420	ICAM3	CD molecules			
61	99.96	oe	ccsbBroad304_06057	CSNK1G3	Casein kinase 1 (CK1) family			
62	99.96	oe	ccsbBroad304_05000	ZNF524	Zinc fingers, C2H2-type			
63	99.96	oe	ccsbBroad304_01831	TUBA1A	Tubulins			
64	99.96	oe	ccsbBroad304_01699	TPD52L2	-			
65	99.96	oe	ccsbBroad304_11186	TGFBR2	Type II receptor serine/threonine kinases			
66	99.96	oe	ccsbBroad304_07053	TFPI	-			
67	99.96	oe	ccsbBroad304_01578	SOS2	Rho guanine nucleotide exchange factors			
68	99.96	oe	ccsbBroad304_02340	SORBS3	-			
69	99.96	oe	ccsbBroad304_03451	SLC35F2	SLC35 family of nucleotide sugar transporters			
70	99.96	oe	ccsbBroad304_06675	SLC22A18	Orphan or poorly characterized SLC22 family members			
71	99.96	oe	ccsbBroad304_02705	SIRT2	Histone deacetylases			
72	99.96	oe	ccsbBroad304_11109	RPS6KB1	p70 subfamily			
73	99.96	oe	ccsbBroad304_01457	RPS19	S ribosomal proteins			
74	99.96	oe	ccsbBroad304_02209	RNF14	RING-type (C3HC4) zinc fingers			
75	99.96	oe	ccsbBroad304_01310	PSMB2	Proteasome subunits			
76	99.96	oe	ccsbBroad304_01266	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
77	99.96	oe	ccsbBroad304_06742	PML	RING-type (C3HC4) zinc fingers			
78	99.96	oe	ccsbBroad304_02058	PLOD3	-			
79	99.96	oe	ccsbBroad304_01208	PITPNA	-			
80	99.96	oe	ccsbBroad304_01202	PIK3CB	Phosphatidylinositol kinases			
81	99.96	oe	ccsbBroad304_02295	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
82	99.96	oe	ccsbBroad304_07920	NUP62	-			
83	99.96	oe	ccsbBroad304_07582	NET1	Rho guanine nucleotide exchange factors			
84	99.96	oe	ccsbBroad304_02276	MVP	-			
85	99.96	oe	ccsbBroad304_08203	LAP3	Leucyl aminopeptidase			
86	99.96	oe	ccsbBroad304_00783	HPRT1	-			
87	99.96	oe	ccsbBroad304_06324	GPX7	-			
88	99.96	oe	ccsbBroad304_14158	GPR87	GPCR / Class A : Orphans			
89	99.96	oe	ccsbBroad304_03182	GLOD4	-			
90	99.96	oe	ccsbBroad304_06209	FGF9	Endogenous ligands			
91	99.96	oe	ccsbBroad304_06087	DDB2	WD repeat domain containing			
92	99.96	oe	ccsbBroad304_08093	DCPS	-			
93	99.96	oe	ccsbBroad304_01949	CAMK1	CAMK1 family			
94	99.96	oe	ccsbBroad304_00080	APOA2	Apolipoproteins			
95	99.96	cp	BRD-K61192372	capecitabine	DNA synthesis inhibitor		TYMS, DPYD	DNA synthesis inhibitor, Thymidylate synthase inhibitor
96	99.96	cp	BRD-K29905972	axitinib	PDGFR receptor inhibitor		KDR, FLT1, FLT4, CSF1, CYP2C19, CYP3A5, KIT, PDGFRB, PLK4	PDGFR receptor inhibitor, VEGFR inhibitor
97	99.96	cp	BRD-K00184207	GR-206	Aryl hydrocarbon receptor ligand			Aryl hydrocarbon receptor ligand
98	99.96	cp	BRD-K47943470	tyrphostin-51	EGFR inhibitor			EGFR inhibitor
99	99.96	cp	BRD-K46435977	valaciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
100	99.96	cp	BRD-K60160658	tiagabine	GABA uptake inhibitor		SLC6A1, CYP2C19	GABA uptake inhibitor
101	99.96	cp	BRD-K32311154	nifekalant	Potassium channel blocker			Potassium channel blocker
102	99.96	cp	BRD-K00532621	midazolam	Benzodiazepine receptor agonist		CYP3A5, CYP3A7, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3	Benzodiazepine receptor agonist
103	99.96	cp	BRD-K84141129	VU-0400193-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
104	99.96	cp	BRD-M07438658	lapatinib	EGFR inhibitor		EGFR, ERBB2, CYP3A5	EGFR inhibitor, ErbB2 inhibitor
105	99.96	cp	BRD-K15402119	huperzine-a	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
106	99.96	cp	BRD-A74771556	nikkomycin	Chitin inhibitor			Chitin inhibitor
107	99.96	cp	BRD-A73680854	PT-630	Dipeptidyl peptidase inhibitor		DPP4, FAP	Dipeptidyl peptidase inhibitor
108	99.96	cp	BRD-A67373739	AICA-ribonucleotide	AMPK activator		ATIC, PRKAA1	AMPK activator
109	99.96	cp	BRD-A43974575	tranylcypromine	Monoamine oxidase inhibitor		MAOA, MAOB, KDM1A, CYP2A6	Monoamine oxidase inhibitor
110	99.96	cp	BRD-K74765201	tomelukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
111	99.96	cp	BRD-A33084410	5'-guanidinonaltrindole	Opioid receptor antagonist			Opioid receptor antagonist
112	99.96	cp	BRD-K56509348	BMS-182874	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
113	99.96	cp	BRD-A84493640	atovaquone	Mitochondrial electron transport inhibitor		DHODH	Mitochondrial electron transport inhibitor
114	99.96	cp	BRD-K68246049	TTNPB	Retinoid receptor agonist		RARB, RARA, RARG	Retinoid receptor agonist
115	99.96	cp	BRD-K60511616	pravastatin	HMGCR inhibitor		HMGCR, SLCO1B1	HMGCR inhibitor
116	99.96	cp	BRD-A41451487	PK-11195	Benzodiazepine receptor antagonist		TSPO, NR1I2, NR1I3	Benzodiazepine receptor antagonist
117	99.96	cp	BRD-A79981887	midodrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
118	99.96	cp	BRD-K92138166	mammea-a	other antibiotic			other antibiotic
119	99.96	cp	BRD-K64670467	JNJ-16259685	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
120	99.96	cp	BRD-A38898897	GW-311616	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
121	99.96	cp	BRD-K02275692	cefotiam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
122	99.96	cp	BRD-K04976539	aminogenistein	SRC inhibitor		LCK	SRC inhibitor
123	99.96	cp	BRD-K78280988	anandamide	Cannabinoid receptor agonist		CNR1, CNR2, TRPV1, CACNA1G, CACNA1H, CACNA1I, GLRA1, GPR119, GPR18, GPR55, KCNA2, KCND3, KCNK3, KCNK9, TRPM8	Cannabinoid receptor agonist
124	99.96	kd	CGS001-118738	ZNF488	Zinc fingers, C2H2-type			
125	99.96	kd	CGS001-285676	ZNF454	Zinc fingers, C2H2-type			
126	99.96	kd	CGS001-10991	SLC38A3	System N-like transporters			
127	99.96	kd	CGS001-120103	SLC36A4	SLC36 family of proton-coupled amino acid transporters			
128	99.96	kd	CGS001-8879	SGPL1	Sphingosine 1-phosphate lyase			
129	99.96	kd	CGS001-6253	RTN2	-			
130	99.96	kd	CGS001-79960	PHF17	-			
131	99.96	kd	CGS001-4856	NOV	-			
132	99.96	kd	CGS001-22889	KIAA0907	-			
133	99.96	kd	CGS001-3628	INPP1	Inositol polyphosphate phosphatases			
134	99.96	kd	CGS001-3294	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
135	99.96	kd	CGS001-2550	GABBR1	GABA receptors			
136	99.96	kd	CGS001-2348	FOLR1	-			
137	99.96	kd	CGS001-2077	ERF	ETS Transcription Factors			
138	99.96	kd	CGS001-54566	EPB41L4B	-			
139	99.96	kd	CGS001-805	CALM2	EF-hand domain containing			
140	99.96	cp	BRD-K41143549	BRD-K41143549	Glutamate receptor antagonist			Glutamate receptor antagonist
141	99.93	oe	ccsbBroad304_05121	ZNF296	Zinc fingers, C2H2-type			
142	99.93	oe	ccsbBroad304_07590	WARS2	Aminoacyl tRNA synthetases / Class I			
143	99.93	oe	ccsbBroad304_00370	CS	-			
144	99.93	cp	BRD-K91696562	orantinib	FGFR inhibitor		PDGFRB, AURKA, AURKB, KDR, EGFR, FGFR1, FGFR2, PDGFRA, TBK1	FGFR inhibitor, VEGFR inhibitor, PDGFR receptor inhibitor
145	99.93	cp	BRD-A61858259	CAY-10415	Insulin sensitizer		INS	Insulin sensitizer
146	99.93	cp	BRD-K72264770	QW-BI-011	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
147	99.93	cp	BRD-K82846253	repaglinide	Insulin secretagogue		ABCC8, CYP2C8, CYP3A5, INS, KCNJ11, PPARG	Insulin secretagogue
148	99.93	cp	BRD-K21565985	xylazine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
149	99.93	cp	BRD-A61793559	metolazone	Carbonic anhydrase inhibitor		SLC12A3, CA2, CA7	Carbonic anhydrase inhibitor
150	99.93	kd	CGS001-7153	TOP2A	DNA Topoisomerases			
151	99.93	kd	CGS001-257397	TAB3	-			
152	99.93	kd	CGS001-6774	STAT3	SH2 domain containing			
153	99.93	kd	CGS001-6591	SNAI2	Snail homologs			
154	99.93	kd	CGS001-5315	PKM2	-			
155	99.93	kd	CGS001-79581	GPR172A	-			
156	99.93	kd	CGS001-54584	GNB1L	WD repeat domain containing			
157	99.93	kd	CGS001-3169	FOXA1	Forkhead boxes			
158	99.93	kd	CGS001-717	C2	Complement system			
159	99.93	kd	CGS001-8874	ARHGEF7	Rho guanine nucleotide exchange factors			
160	99.93	oe	ccsbBroad304_01380	RBBP7	WD repeat domain containing			
161	99.93	oe	ccsbBroad304_04309	HDAC10	Histone deacetylases			
162	99.91	oe	ccsbBroad304_09745	ZNF519	Zinc fingers, C2H2-type			
163	99.91	oe	ccsbBroad304_01953	PIAS1	Zinc fingers, MIZ-type			
164	99.91	oe	ccsbBroad304_14439	OPN5	GPCR / Class A : Opsin receptors			
165	99.91	oe	ccsbBroad304_02443	HAX1	-			
166	99.91	oe	ccsbBroad304_03533	CDCA8	-			
167	99.91	oe	ccsbBroad304_00239	CCNG1	-			
168	99.91	cp	BRD-K08273968	griseofulvin	Tubulin inhibitor		KRT12	Tubulin inhibitor
169	99.91	cp	BRD-K08806317	timolol	Adrenergic receptor antagonist		ADRB2, ADRB1	Adrenergic receptor antagonist
170	99.91	cp	BRD-K06024458	n-arachidonyl-GABA	cannabinoid receptor agonist			cannabinoid receptor agonist
171	99.91	kd	CGS001-7421	VDR	Vitamin D receptors			
172	99.91	kd	CGS001-9898	UBAP2L	-			
173	99.91	kd	CGS001-8784	TNFRSF18	Tumour necrosis factor (TNF) receptor family			
174	99.91	kd	CGS001-6832	SUPV3L1	-			
175	99.91	kd	CGS001-4316	MMP7	Matrix metallopeptidase			
176	99.91	kd	CGS001-91133	L3MBTL4	Sterile alpha motif (SAM) domain containing			
177	99.91	kd	CGS001-26086	GPSM1	Tetratricopeptide (TTC) repeat domain containing			
178	99.91	kd	CGS001-10093	ARPC4	Actin related protein 2/3 complex subunits			
179	99.9	kd	CGS001-3482	IGF2R	CD molecules			
180	99.9	kd	CGS001-23274	CLEC16A	C-type lectin domain containing			
181	99.89	oe	ccsbBroad304_07798	EXOC3	-			
182	99.89	oe	ccsbBroad304_03874	UBL5	-			
183	99.89	oe	ccsbBroad304_06102	DLX3	Homeoboxes / ANTP class : NKL subclass			
184	99.89	cp	BRD-K57926513	tyrphostin-AG-1295	PDGFR receptor inhibitor		FLT3, KDR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
185	99.89	cp	BRD-K23369905	oxiconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
186	99.89	cp	BRD-A26711594	nicardipine	Calcium channel blocker		CACNA1C, ADORA3, ADRA1A, ADRA1B, ADRA1D, CACNA1D, CACNA2D1, CACNB2, CALM1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, PDE1A, PDE1B	Calcium channel blocker
187	99.89	cp	BRD-A48809242	IB-MECA	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
188	99.89	cp	BRD-A30655177	LFM-A13	BTK inhibitor		BTK	BTK inhibitor
189	99.89	kd	CGS001-7311	UBA52	L ribosomal proteins			
190	99.89	kd	CGS001-8859	STK19	G11 family			
191	99.89	kd	CGS001-1827	RCAN1	-			
192	99.89	kd	CGS001-3206	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
193	99.89	kd	CGS001-10841	FTCD	-			
194	99.89	kd	CGS001-1984	EIF5A	-			
195	99.89	kd	CGS001-1644	DDC	Catecholamine turnover			
196	99.89	kd	CGS001-1488	CTBP2	-			
197	99.89	oe	ccsbBroad304_00225	CAT	-			
198	99.87	oe	ccsbBroad304_02109	XPR1	-			
199	99.87	oe	ccsbBroad304_06450	ILK	Ankyrin repeat domain containing			
200	99.87	oe	ccsbBroad304_00771	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
201	99.87	cp	BRD-K22631935	neurodazine	Neurogenesis of non-pluripotent C2C12 myoblast inducer			Neurogenesis of non-pluripotent C2C12 myoblast inducer
202	99.87	cp	BRD-K34441861	moexipril	ACE inhibitor		ACE, ACE2	ACE inhibitor
203	99.87	cp	BRD-K18816859	L-694247	Serotonin receptor agonist		HTR1D, HTR1A, HTR1B	Serotonin receptor agonist
204	99.87	kd	CGS001-55311	ZNF444	Zinc fingers, C2H2-type			
205	99.87	kd	CGS001-7337	UBE3A	-			
206	99.87	kd	CGS001-63948	DMRTB1	-			
207	99.87	kd	CGS001-1152	CKB	-			
208	99.85	oe	ccsbBroad304_00873	INPP1	Inositol polyphosphate phosphatases			
209	99.85	cp	BRD-K82109576	vincristine	Tubulin inhibitor		TUBB, TUBA4A	Tubulin inhibitor
210	99.85	cp	BRD-K57930253	nitrazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, SCN1A	Benzodiazepine receptor agonist
211	99.85	cp	BRD-A01145011	zebularine	DNA methyltransferase inhibitor		CDA, DNMT1	DNA methyltransferase inhibitor
212	99.85	cp	BRD-A18043272	phensuximide	Succinimide antiepileptic			Succinimide antiepileptic
213	99.85	cp	BRD-K92760278	riboflavin	Vitamin B			Vitamin B
214	99.85	cp	BRD-K95676198	JAK3-inhibitor-V	JAK inhibitor		JAK3	JAK inhibitor
215	99.85	kd	CGS001-6510	SLC1A5	Alanine/serine/cysteine transporter subfamily			
216	99.85	kd	CGS001-2114	ETS2	ETS Transcription Factors			
217	99.82	cp	BRD-K62012036	acitretin	Retinoid receptor agonist		RARA, RARB, RARG, RBP1, RXRA, RXRB, RXRG, STAT3	Retinoid receptor agonist
218	99.82	cp	BRD-K43764301	dexketoprofen	Cyclooxygenase inhibitor		CXCR1, PTGS1, PTGS2, SLC5A8	Cyclooxygenase inhibitor
219	99.82	cp	BRD-A48261811	argatroban	Thrombin inhibitor		F2, CYP3A5	Thrombin inhibitor
220	99.82	cp	BRD-K32755366	reserpic-acid	Norepinephrine transporter inhibitor			Norepinephrine transporter inhibitor
221	99.82	cp	BRD-K60060639	methyllidocaine	antiarrhythmic medication			antiarrhythmic medication
222	99.82	cp	BRD-A96485169	EBPC	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
223	99.82	cp	BRD-A42571354	cetirizine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
224	99.82	kd	CGS001-146050	ZSCAN29	Zinc fingers, C2H2-type			
225	99.82	kd	CGS001-5320	PLA2G2A	Hydrolases			
226	99.82	kd	CGS001-4282	MIF	-			
227	99.82	kd	CGS001-57459	GATAD2B	GATA zinc finger domain containing			
228	99.81	kd	CGS001-1356	CP	-			
229	99.8	cc		Reverse transcriptase inhibitor	-			
230	99.8	cp	BRD-K24656285	farnesol	FXR agonist		MAOB, MVK, NR1H4	FXR agonist, Monoamine oxidase inhibitor, NFkB pathway activator, PPAR receptor agonist
231	99.8	cp	BRD-K18618618	cimetidine	Histamine receptor antagonist		HRH2, SLC29A4, SLC47A1, SLC47A2	Histamine receptor antagonist
232	99.8	kd	CGS001-56848	SPHK2	Sphingosine kinase			
233	99.78	oe	ccsbBroad304_01114	NUP88	-			
234	99.78	cp	BRD-K63195589	tipifarnib	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
235	99.78	cp	BRD-K26373640	IKK-2-inhibitor	IKK inhibitor		IKBKB	IKK inhibitor, SYK inhibitor
236	99.78	cp	BRD-A04668240	CGP-52432	GABA receptor antagonist		GABBR1, GABBR2	GABA receptor antagonist
237	99.78	cp	BRD-K95609758	BMS-191011	Potassium channel activator		KCNMA1	Potassium channel activator
238	99.78	cp	BRD-K28075147	biochanin-a	Estrogen receptor agonist			Estrogen receptor agonist
239	99.78	cp	BRD-K21450440	benzthiazide	Carbonic anhydrase inhibitor		CA2, CA1, CA12, CA4, CA9, SLC12A3	Carbonic anhydrase inhibitor
240	99.78	kd	CGS001-5930	RBBP6	-			
241	99.78	kd	CGS001-2966	GTF2H2	General transcription factors			
242	99.76	cp	BRD-K99749624	linifanib	PDGFR receptor inhibitor		CSF1R, KDR, PDGFRB, FLT1, FLT3, FLT4, CSF1, KIT, PDGFRA, RET, TEK	PDGFR receptor inhibitor, VEGFR inhibitor
243	99.76	cp	BRD-K94887716	TFMPP	Serotonin receptor agonist			Serotonin receptor agonist, Serotonin receptor antagonist
244	99.76	cp	BRD-K59633790	VU-0420363-1	SARS coronavirus 3C-like protease inhibitor			SARS coronavirus 3C-like protease inhibitor
245	99.76	cp	BRD-K65285700	BRD-K65285700	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
246	99.76	cp	BRD-K45033733	famciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
247	99.76	cp	BRD-K23913458	coumarin	Vitamin K antagonist		CA1, CA12, CA14, CA2, CA4, CA6, CA9, CYP2A6	Vitamin K antagonist
248	99.76	kd	CGS001-7483	WNT9A	Wingless-type MMTV integration sites			
249	99.76	kd	CGS001-871	SERPINH1	Serine (or cysteine) peptidase inhibitors			
250	99.76	kd	CGS001-2131	EXT1	Exostosin glycosyltransferase family			
251	99.74	cp	BRD-K55034111	pefloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
252	99.74	cp	BRD-K52075715	oxibendazole	Tubulin inhibitor		TUBB, TUBB4B	Tubulin inhibitor
253	99.74	cp	BRD-K53570330	carbofuran	Cholinesterase inhibitor			Cholinesterase inhibitor
254	99.74	cp	BRD-K56558538	ambroxol	Sodium channel blocker		GBA	Sodium channel blocker
255	99.74	kd	CGS001-1457	CSNK2A1	Casein kinase 2 (CK2) family			
256	99.74	kd	CGS001-7465	WEE1	WEE family			
257	99.74	kd	CGS001-3146	HMGB1	High-mobility group / Canonical			
258	99.74	kd	CGS001-2878	GPX3	-			
259	99.74	kd	CGS001-7852	CXCR4	Chemokine receptors			
260	99.74	cp	BRD-K93461745	buspirone	Serotonin receptor agonist		HTR1A, DRD2	Serotonin receptor agonist
261	99.73	kd	CGS001-8527	DGKD	Pleckstrin homology (PH) domain containing			
262	99.72	cp	BRD-K59570838	homoveratrylamine	Dopamine analog			Dopamine analog
263	99.72	cp	BRD-K19309090	SR-95639A	Acetylcholine receptor agonist		CHRM1	Acetylcholine receptor agonist
264	99.72	cp	BRD-K12244279	MEK1-2-inhibitor	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
265	99.72	kd	CGS001-7003	TEAD1	-			
266	99.72	kd	CGS001-6757	SSX2	-			
267	99.72	kd	CGS001-10513	APPBP2	-			
268	99.71	oe	ccsbBroad304_03640	CEP72	-			
269	99.71	cp	BRD-A47706533	L-BSO	Glutathione transferase inhibitor		GCLM	Glutathione transferase inhibitor
270	99.69	oe	ccsbBroad304_08531	ZNF331	Zinc fingers, C2H2-type			
271	99.69	oe	ccsbBroad304_03394	GPR84	GPCR / Class A : Fatty acid receptors			
272	99.69	cp	BRD-A92670106	tocainide	Sodium channel blocker		SCN5A	Sodium channel blocker
273	99.69	kd	CGS001-7504	XK	Blood group antigens			
274	99.69	kd	CGS001-6658	SOX3	SRY (sex determining region Y)-boxes			
275	99.69	kd	CGS001-55509	BATF3	basic leucine zipper proteins			
276	99.69	kd	CGS001-301	ANXA1	Annexins			
277	99.69	kd	CGS001-340273	ABCB5	ATP binding cassette transporters / subfamily B			
278	99.68	kd	CGS001-5223	PGAM1	-			
279	99.67	oe	ccsbBroad304_00551	FECH	-			
280	99.67	cp	BRD-K91900765	VX-745	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
281	99.67	kd	CGS001-55163	PNPO	-			
282	99.67	kd	CGS001-4860	PNP	-			
283	99.67	kd	CGS001-51451	LCMT1	-			
284	99.67	kd	CGS001-3225	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
285	99.67	kd	CGS001-51704	GPRC5B	GPCR / Class C : Orphans			
286	99.67	kd	CGS001-2730	GCLM	-			
287	99.67	kd	CGS001-375318	AQP12A	Ion channels / Aquaporins			
288	99.65	oe	ccsbBroad304_06982	SNRNP70	RNA binding motif (RRM) containing			
289	99.65	oe	ccsbBroad304_03028	RBMX	RNA binding motif (RRM) containing			
290	99.65	oe	ccsbBroad304_01844	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
291	99.65	kd	CGS001-7546	ZIC2	Zinc fingers, C2H2-type			
292	99.64	kd	CGS001-84109	QRFPR	GPCR / Class A : RF amide peptide receptors			
293	99.63	oe	ccsbBroad304_07981	SENP6	Ulp1 endopeptidase			
294	99.63	oe	ccsbBroad304_02533	NOXA1	-			
295	99.63	oe	ccsbBroad304_00793	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
296	99.63	cp	BRD-K89708791	rifaximin	RNA synthesis inhibitor		NR1I2, CYP3A4	RNA synthesis inhibitor
297	99.63	cp	BRD-K52662033	lidocaine	Histamine receptor agonist		SCN5A, EGFR, SCN10A, SCN9A	Histamine receptor agonist
298	99.63	kd	CGS001-199704	ZNF585A	Zinc fingers, C2H2-type			
299	99.63	kd	CGS001-6548	SLC9A1	SLC9 family of sodium/hydrogen exchangers			
300	99.63	kd	CGS001-29998	GLTSCR1	-			
301	99.63	kd	CGS001-10755	GIPC1	-			
302	99.61	oe	ccsbBroad304_08453	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
303	99.61	cp	BRD-K02992638	lamivudine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
304	99.61	cp	BRD-A44090213	indoprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2, CXCR1, CXCR2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
305	99.61	cp	BRD-A09472452	flecainide	Sodium channel blocker		SCN5A, KCNA5, KCNA7, SCN4A	Sodium channel blocker
306	99.61	cp	BRD-K89274813	DMP-543	Acetylcholine release stimulant			Acetylcholine release stimulant
307	99.61	cp	BRD-K08287586	butylparaben	DNA synthesis inhibitor			DNA synthesis inhibitor
308	99.61	kd	CGS001-51005	AMDHD2	-			
309	99.61	cp	BRD-K07881437	danusertib	Aurora kinase inhibitor		AURKA, AURKB, AURKC, FGFR1, NTRK1, RET, BCR, SLK	Aurora kinase inhibitor, Growth factor receptor inhibitor
310	99.58	cc		Cannabinoid receptor agonist	-			
311	99.58	cp	BRD-A34806832	proscillaridin	ATPase inhibitor		ATP1A1	ATPase inhibitor
312	99.56	oe	ccsbBroad304_14047	TACC3	-			
313	99.56	oe	ccsbBroad304_01371	RALA	-			
314	99.56	cp	BRD-K11634954	GBR-13069	Dopamine uptake inhibitor		SLC6A3	Dopamine uptake inhibitor
315	99.56	kd	CGS001-51222	ZNF219	Zinc fingers, C2H2-type			
316	99.56	kd	CGS001-3455	IFNAR2	Interferon receptor family			
317	99.56	kd	CGS001-9474	ATG5	-			
318	99.54	oe	ccsbBroad304_03147	IL20	Interleukins and interleukin receptors			
319	99.54	oe	ccsbBroad304_01252	PPIA	Cis-trans-isomerases			
320	99.54	cp	BRD-K81916719	triclabendazole	Microtubule inhibitor		DNMT1	Microtubule inhibitor
321	99.54	cp	BRD-A07000685	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
322	99.54	kd	CGS001-84288	EFCAB2	EF-hand domain containing			
323	99.53	kd	CGS001-6364	CCL20	Chemokine ligands			
324	99.52	oe	ccsbBroad304_02688	MTF2	Zinc fingers, PHD-type			
325	99.52	oe	ccsbBroad304_04675	ATG4A	-			
326	99.52	cp	BRD-K68507560	dicycloverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3	Acetylcholine receptor antagonist
327	99.52	kd	CGS001-22938	SNW1	-			
328	99.52	kd	CGS001-50846	DHH	-			
329	99.51	cp	BRD-K02404261	caffeine	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ATM, ITPR1, RYR1, ADORA3, ATR, ITPR2, ITPR3, PDE10A, PDE11A, PDE1A, PDE1B, PDE1C, PDE2A, PDE3A, PDE3B, PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PDE6A, PDE6B, PDE6C, PDE7A, PDE7B, PDE8A, PDE8B, PDE9A, PIK3CA, PIK3CB, PIK3CD, PRKDC, RYR2, RYR3	Adenosine receptor antagonist, Diuretic, Phosphodiesterase inhibitor
330	99.5	cc		Retinoid receptor agonist	-			
331	99.5	oe	ccsbBroad304_03391	PRKAG3	AMPK subfamily			
332	99.5	cp	BRD-K40892394	AR-C133057XX	Nitric oxide synthase inhibitor		NOS2, NOS1	Nitric oxide synthase inhibitor
333	99.5	cp	BRD-K71731651	PNU-120596	Acetylcholine receptor agonist		CHRNA7	Acetylcholine receptor agonist
334	99.5	cp	BRD-A87719232	naproxen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
335	99.5	kd	CGS001-6741	SSB	La ribonucleoprotein domain containing			
336	99.5	kd	CGS001-25898	RCHY1	RING-type (C3HC4) zinc fingers			
337	99.47	cp	BRD-K54314721	zolmitriptan	Serotonin receptor agonist		HTR1B, HTR1D, HTR1A, HTR1F, HTR1E	Serotonin receptor agonist
338	99.47	kd	CGS001-5624	PROC	Endogenous ligands			
339	99.46	kd	CGS001-152687	ZNF595	Zinc fingers, C2H2-type			
340	99.45	cp	BRD-A22256192	terazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
341	99.45	kd	CGS001-5018	OXA1L	-			
342	99.45	kd	CGS001-283078	MKX	Homeoboxes / TALE class			
343	99.45	kd	CGS001-163688	CALML6	EF-hand domain containing			
344	99.45	cp	BRD-K55991774	BAS-09104376	HIV integrase inhibitor			HIV integrase inhibitor
345	99.43	oe	ccsbBroad304_01651	TCF7L2	-			
346	99.43	oe	ccsbBroad304_01781	WNT7B	Endogenous ligands			
347	99.43	oe	ccsbBroad304_02826	SLC7A11	Solute carriers			
348	99.43	oe	ccsbBroad304_01832	PAX8	Paired boxes			
349	99.43	kd	CGS001-29984	RHOD	-			
350	99.43	kd	CGS001-5450	POU2AF1	-			
351	99.43	kd	CGS001-57504	MTA3	GATA zinc finger domain containing			
352	99.43	kd	CGS001-55120	FANCL	Fanconi anemia, complementation groups			
353	99.42	kd	CGS001-344	APOC2	Apolipoproteins			
354	99.41	oe	ccsbBroad304_03155	DHH	-			
355	99.41	oe	ccsbBroad304_05038	HORMAD2	-			
356	99.41	cp	BRD-A71459254	cymarin	ATPase inhibitor		ATP1A1	ATPase inhibitor
357	99.41	kd	CGS001-29982	NRBF2	-			
358	99.39	oe	ccsbBroad304_01992	B4GALT3	Beta 4-glycosyltransferases			
359	99.39	cp	BRD-M40783228	mesna	Antioxidant			Antioxidant
360	99.39	cp	BRD-K36529613	PU-H71	HSP inhibitor		HSP90AA1	HSP inhibitor
361	99.39	kd	CGS001-51715	RAB23	RAB, member RAS oncogene			
362	99.39	kd	CGS001-25793	FBXO7	F-boxes / other			
363	99.37	oe	ccsbBroad304_01617	STX4	-			
364	99.37	oe	ccsbBroad304_03121	NRBF2	-			
365	99.37	cp	BRD-K55420858	mirin	MRE11A exonuclease inhibitor		MRE11A	MRE11A exonuclease inhibitor
366	99.37	kd	CGS001-54815	GATAD2A	GATA zinc finger domain containing			
367	99.35	cp	BRD-K98769987	flumazenil	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor antagonist
368	99.34	cp	BRD-K55703048	latrepirdine	Glutamate receptor antagonist		HTR6, GRIN2B, HRH1	Glutamate receptor antagonist
369	99.34	kd	CGS001-5868	RAB5A	RAB, member RAS oncogene			
370	99.34	kd	CGS001-57396	CLK4	CDC-like kinases			
371	99.33	oe	ccsbBroad304_00001	NAT1	-			
372	99.32	oe	ccsbBroad304_08292	IP6K2	-			
373	99.32	cp	BRD-K25741894	skimmianine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Furoquinoline alkaloid
374	99.32	cp	BRD-K49519092	immethridine	Histamine receptor agonist		HRH3	Histamine receptor agonist
375	99.31	kd	CGS001-472	ATM	Other PIKK family kinases			
376	99.28	oe	ccsbBroad304_02446	TADA3	-			
377	99.28	oe	ccsbBroad304_06332	GSTM2	Glutathione S-transferases / Soluble			
378	99.28	kd	CGS001-143471	PSMA8	Proteasome (prosome, macropain) subunits			
379	99.27	oe	ccsbBroad304_07663	IGF2BP3	RNA binding motif (RRM) containing			
380	99.27	kd	CGS001-10476	ATP5H	ATPases / F-type			
381	99.26	cp	BRD-K57033106	tripelennamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
382	99.26	kd	CGS001-6709	SPTAN1	EF-hand domain containing			
383	99.25	oe	ccsbBroad304_00041	NR0B1	DAX-like receptors			
384	99.24	cp	BRD-K04833372	GSK-1904529A	IGF-1 inhibitor		IGF1R, INSR	IGF-1 inhibitor, IGF-1R inhibitor, Insulin receptor ligand
385	99.24	kd	CGS001-7453	WARS	Aminoacyl tRNA synthetases / Class I			
386	99.24	kd	CGS001-10553	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
387	99.23	kd	CGS001-51170	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
388	99.23	kd	CGS001-360023	ZBTB41	BTB/POZ domain containing			
389	99.21	cp	BRD-K00317371	RITA	MDM inhibitor		MDM2, TXNRD1, TXNRD2	MDM inhibitor
390	99.21	cp	BRD-K75478907	GS-39783	GABA receptor modulator		GABBR1	GABA receptor modulator
391	99.21	kd	CGS001-6097	RORC	Retinoic acid-related orphans			
392	99.2	cc		Phospholipases LOF	-			
393	99.2	cp	BRD-A14985772	ascorbyl-palmitate	antioxidant			antioxidant
394	99.2	kd	CGS001-10465	PPIH	-			
395	99.19	oe	ccsbBroad304_00880	IRF2	-			
396	99.19	cp	BRD-K16277217	piperacetazine	Dopamine receptor antagonist			Dopamine receptor antagonist
397	99.19	kd	CGS001-6611	SMS	-			
398	99.19	kd	CGS001-5535	PPP3R2	EF-hand domain containing			
399	99.19	kd	CGS001-4905	NSF	ATPases / AAA-type			
400	99.19	kd	CGS001-4795	NFKBIL1	-			
401	99.17	oe	ccsbBroad304_06301	GOT2	-			
402	99.17	kd	CGS001-10892	MALT1	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
403	99.15	cp	BRD-K89125793	tinidazole	Antiprotozoal			Antiprotozoal
404	99.15	cp	BRD-K92301463	16,16-dimethylprostaglandin-e2	Prostanoid receptor agonist		HPGD	Prostanoid receptor agonist
405	99.14	kd	CGS001-5091	PC	Carboxylases			
406	99.12	oe	ccsbBroad304_01710	TRAF2	RING-type (C3HC4) zinc fingers			
407	99.12	cp	BRD-K69600043	thiethylperazine	Dopamine receptor antagonist		DRD1, DRD2, DRD4	Dopamine receptor antagonist
408	99.12	kd	CGS001-7727	ZNF174	Zinc fingers, C2H2-type			
409	99.12	kd	CGS001-10276	NET1	Rho guanine nucleotide exchange factors			
410	99.12	kd	CGS001-2783	GNB2	WD repeat domain containing			
411	99.12	kd	CGS001-892	CCNC	-			
412	99.1	cp	BRD-K37130656	rivaroxaban	Coagulation inhibitor		F10, CYP2J2, CYP3A5	Coagulation inhibitor
413	99.1	kd	CGS001-9123	SLC16A3	SLC16 family of monocarboxylate transporters			
414	99.1	cp	BRD-K48427617	U-0124	MEK inhibitor			MEK inhibitor
415	99.08	cp	BRD-A49906757	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
416	99.08	kd	CGS001-10477	UBE2E3	Ubiquitin-conjugating enzymes E2			
417	99.08	kd	CGS001-5269	SERPINB6	Serine (or cysteine) peptidase inhibitors			
418	99.08	oe	ccsbBroad304_01974	RNASET2	-			
419	99.07	kd	CGS001-2963	GTF2F2	General transcription factors			
420	99.06	kd	CGS001-147694	ZNF548	Zinc fingers, C2H2-type			
421	99.06	cp	BRD-K29733039	deforolimus	MTOR inhibitor		MTOR	MTOR inhibitor
422	99.04	cp	BRD-K61177364	NBI-27914	CRF receptor antagonist		CRHR1	CRF receptor antagonist
423	99.03	kd	CGS001-9061	PAPSS1	-			
424	99.02	kd	CGS001-3054	HCFC1	-			
425	99.02	kd	CGS001-10059	DNM1L	-			
426	98.99	oe	ccsbBroad304_04472	HIST1H2BK	Histones / Replication-dependent			
427	98.99	cp	BRD-K90885812	propantheline	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
428	98.99	cp	BRD-A73859745	glycodeoxycholic-acid	Apoptosis stimulant			Apoptosis stimulant
429	98.98	cp	BRD-A59808129	guggulsterone	Cholesterol inhibitor		NR1H4, PGR, AR, ESR1, IKBKB, NR1I2, NR3C1, NR3C2	Cholesterol inhibitor, Estrogen receptor agonist, FXR antagonist, IKK inhibitor, Pregnane X receptor agonist, Progesterone receptor agonist
430	98.98	kd	CGS001-3572	IL6ST	IL-6 receptor family			
431	98.97	kd	CGS001-5699	PSMB10	Proteasome (prosome, macropain) subunits			
432	98.97	kd	CGS001-84759	PCGF1	Polycomb group ring fingers			
433	98.97	kd	CGS001-10018	BCL2L11	-			
434	98.97	kd	CGS001-19	ABCA1	ATP binding cassette transporters / subfamily A			
435	98.96	kd	CGS001-10923	SUB1	-			
436	98.96	kd	CGS001-3459	IFNGR1	Interferon receptor family			
437	98.93	cp	BRD-K51476772	ST-638	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
438	98.93	kd	CGS001-292	SLC25A5	Mitochondrial nucleotide transporter subfamily			
439	98.91	oe	ccsbBroad304_10047	GPR148	GPCR / Class A : Orphans			
440	98.88	cp	BRD-K06080977	eicosatetraynoic-acid	Cyclooxygenase inhibitor		ALOX12, PPARA, PPARG, PTGS1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor
441	98.88	cp	BRD-A67862938	naftidrofuryl	Adrenergic receptor antagonist			Adrenergic receptor antagonist
442	98.88	kd	CGS001-3920	LAMP2	CD molecules			
443	98.88	kd	CGS001-3611	ILK	Ankyrin repeat domain containing			
444	98.86	cp	BRD-A87387433	cefpodoxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
445	98.84	cp	BRD-K20714604	RS-56812	Serotonin receptor partial agonist		HTR3A	Serotonin receptor partial agonist
446	98.84	kd	CGS001-7733	ZNF180	Zinc fingers, C2H2-type			
447	98.84	kd	CGS001-6046	BRD2	Bromodomain kinase (BRDK) family			
448	98.82	cp	BRD-K07265709	razoxane	Chelating agent		TOP2A, TOP2B	Chelating agent, Topoisomerase inhibitor
449	98.82	cp	BRD-K08890269	CO-102862	Sodium channel blocker		SCN2A, SCN4A, SCN9A	Sodium channel blocker
450	98.82	kd	CGS001-6934	TCF7L2	-			
451	98.82	kd	CGS001-2168	FABP1	Fatty acid-binding proteins			
452	98.8	kd	CGS001-9344	TAOK2	TAO subfamily			
453	98.8	kd	CGS001-629	CFB	Complement system			
454	98.77	oe	ccsbBroad304_00936	LGALS1	Endogenous ligands			
455	98.77	cp	BRD-K87048468	RS-102221	Serotonin receptor antagonist		HTR2C, HTR2A, HTR2B	Serotonin receptor antagonist
456	98.77	cp	BRD-K08547377	irinotecan	Topoisomerase inhibitor		TOP1, CYP3A5, TOP1MT	Topoisomerase inhibitor
457	98.77	kd	CGS001-374291	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
458	98.75	cc		General transcription factors group 2 LOF	-			
459	98.75	kd	CGS001-147948	ZNF582	Zinc fingers, C2H2-type			
460	98.75	kd	CGS001-2243	FGA	Endogenous ligands			
461	98.74	kd	CGS001-8453	CUL2	-			
462	98.73	oe	ccsbBroad304_05148	SLC30A8	SLC30 zinc transporter family			
463	98.73	kd	CGS001-6799	SULT1A2	Sulfotransferases, cytosolic			
464	98.73	kd	CGS001-2747	GLUD2	-			
465	98.72	cp	BRD-K09907482	PRL-3-inhibitor-I	Tyrosine phosphatase inhibitor		PTP4A3	Tyrosine phosphatase inhibitor
466	98.72	kd	CGS001-11073	TOPBP1	-			
467	98.71	oe	ccsbBroad304_05801	ALDH3A1	Aldehyde dehydrogenases			
468	98.71	kd	CGS001-83463	MXD3	Basic helix-loop-helix proteins			
469	98.69	cp	BRD-K06335600	tizanidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP1A2, NISCH	Adrenergic receptor agonist
470	98.68	cp	BRD-A70083328	secnidazole	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor, Microtubule inhibitor, Antiprotozoal
471	98.68	kd	CGS001-10214	SSX3	-			
472	98.67	cp	BRD-K73109821	diazoxide	Potassium channel activator		ATP1A1, CA1, CA2, KCNJ11, KCNMA1, SLC12A3	Potassium channel activator
473	98.66	cp	BRD-A45664787	iloprost	Platelet aggregation inhibitor		PTGIR, PTGER1, PTGER2, PDE4A, PDE4B, PDE4C, PDE4D, PLAT, PTGDR, PTGER3, PTGER4, PTGFR, TBXA2R	Platelet aggregation inhibitor, Prostanoid receptor agonist
474	98.65	cc		MDM inhibitor	-			
475	98.64	cp	BRD-K87049188	fusaric-acid	Dopamine beta hydroxylase inhibitor		DBH	Dopamine beta hydroxylase inhibitor
476	98.62	kd	CGS001-55634	ZNF673	-			
477	98.61	cp	BRD-K63504947	semaxanib	VEGFR inhibitor		KDR, FLT1, KIT, PDGFRB, FGFR1, FLT3, MET, PDGFRA, RET	VEGFR inhibitor
478	98.6	oe	ccsbBroad304_00883	ISG20	-			
479	98.6	cp	BRD-K97799481	theophylline	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3, CHIA, CYP2E1, CYP3A4, HDAC2, PDE3A, PDE4A, PDE4B, PDE5A	Adenosine receptor antagonist
480	98.58	oe	ccsbBroad304_08532	SIRPG	Immunoglobulin superfamily / C1-set domain containing			
481	98.58	cp	BRD-A03216249	mepivacaine	Potassium channel blocker		SCN10A, SCN9A	Potassium channel blocker, Sodium channel blocker
482	98.58	cp	BRD-K10961822	latanoprost	Prostanoid receptor agonist		PTGFR	Prostanoid receptor agonist
483	98.58	cp	BRD-K53857191	risperidone	Dopamine receptor antagonist		DRD2, HTR2A, ADRA1A, ADRA1B, DRD3, HRH1, HTR1A, HTR1D, HTR2C, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CYP3A5, DRD1, DRD4, HTR1B, HTR1E, HTR1F, HTR6, HTR7	Dopamine receptor antagonist, Serotonin receptor antagonist
484	98.58	cp	BRD-A24429032	HEAT	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
485	98.58	kd	CGS001-7443	VRK1	Vaccina related kinase (VRK) family			
486	98.58	kd	CGS001-28511	NKIRAS2	-			
487	98.58	kd	CGS001-22859	LPHN1	Adhesion Class GPCRs			
488	98.57	kd	CGS001-9988	DMTF1	-			
489	98.56	oe	ccsbBroad304_00183	C1S	Complement system			
490	98.56	cp	BRD-K39983086	loteprednol	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Phospholipase inhibitor
491	98.55	oe	ccsbBroad304_06592	MMP14	Matrix metallopeptidase			
492	98.55	kd	CGS001-4791	NFKB2	NFkappaB transcription factor family			
493	98.54	cp	BRD-K74763371	bosentan	Endothelin receptor antagonist		EDNRB, EDNRA, ABCB1, CYP2C19, CYP3A4	Endothelin receptor antagonist
494	98.54	kd	CGS001-3799	KIF5B	Kinesins			
495	98.54	kd	CGS001-1198	CLK3	CDC-like kinases			
496	98.53	kd	CGS001-8777	MPDZ	-			
497	98.52	cp	BRD-K76908866	CP-724714	EGFR inhibitor		ERBB2	EGFR inhibitor, Receptor tyrosine protein kinase inhibitor, Tyrosine kinase inhibitor
498	98.52	cp	BRD-A80775386	hyperforin	Cyclooxygenase inhibitor		NR1I2, ALOX5, PTGS1, TRPC6	Cyclooxygenase inhibitor, Dopamine uptake inhibitor, Interleukin receptor antagonist, Lipoxygenase inhibitor, Serotonin reuptake inhibitor
499	98.52	kd	CGS001-10437	IFI30	-			
500	98.51	kd	CGS001-10253	SPRY2	-			
501	98.51	kd	CGS001-56923	NMUR2	GPCR / Class A : Neuromedin U receptors			
502	98.51	kd	CGS001-8692	HYAL2	-			
503	98.51	cp	BRD-A32161980	carbetocin	Oxytocin receptor agonist		OXTR	Oxytocin receptor agonist
504	98.48	kd	CGS001-10781	ZNF266	Zinc fingers, C2H2-type			
505	98.47	kd	CGS001-9263	STK17A	Death-associated kinase (DAPK) family			
506	98.47	cp	BRD-A30590053	MR-16728	Acetylcholine release enhancer			Acetylcholine release enhancer, Acetylcholine release stimulant
507	98.47	kd	CGS001-54490	UGT2B28	UDP glucuronosyltransferases			
508	98.47	kd	CGS001-2876	GPX1	-			
509	98.47	kd	CGS001-1952	CELSR2	Cadherins / Major cadherins			
510	98.46	kd	CGS001-883	CCBL1	Hydrogen sulphide synthesis			
511	98.43	kd	CGS001-662	BNIP1	-			
512	98.41	kd	CGS001-11105	PRDM7	Zinc fingers, C2H2-type			
513	98.38	oe	ccsbBroad304_06318	GPER	-			
514	98.38	cp	BRD-A41304429	practolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
515	98.37	kd	CGS001-57657	HCN3	Cyclic nucleotide-regulated channels			
516	98.35	kd	CGS001-26298	EHF	-			
517	98.35	kd	CGS001-10902	BRD8	Bromodomain kinase (BRDK) family			
518	98.35	cp	BRD-K26979635	NS-3694	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
519	98.34	oe	ccsbBroad304_05006	ZNF583	Zinc fingers, C2H2-type			
520	98.34	oe	ccsbBroad304_13934	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
521	98.34	oe	ccsbBroad304_00722	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
522	98.33	kd	CGS001-94233	OPN4	GPCR / Class A : Opsin receptors			
523	98.33	kd	CGS001-3032	HADHB	-			
524	98.33	kd	CGS001-652	BMP4	Bone morphogenetic proteins			
525	98.32	kd	CGS001-51734	SEPX1	-			
526	98.32	kd	CGS001-5338	PLD2	Hydrolases			
527	98.32	kd	CGS001-701	BUB1B	Bub family			
528	98.31	kd	CGS001-3593	IL12B	Interleukins and interleukin receptors			
529	98.3	oe	ccsbBroad304_06290	GNA15	-			
530	98.3	kd	CGS001-1036	CDO1	-			
531	98.29	cp	BRD-K12539581	nocodazole	Tubulin inhibitor		HPGDS	Tubulin inhibitor
532	98.29	cp	BRD-K95202259	ML-3163	p38 MAPK inhibitor		CYP2D6, CYP3A4, MAPK11, MAPK12, MAPK14	p38 MAPK inhibitor
533	98.29	kd	CGS001-5442	POLRMT	-			
534	98.29	kd	CGS001-165140	OXER1	GPCR / Class A : Leukotriene receptors			
535	98.27	kd	CGS001-84838	ZNF496	Zinc fingers, C2H2-type			
536	98.25	cp	BRD-K50311478	tosyl-phenylalanyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
537	98.23	cp	BRD-A29289453	PCA-4248	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
538	98.23	cp	BRD-K59256312	gabexate	Serine protease inhibitor		PRSS1, TPSAB1	Serine protease inhibitor
539	98.23	kd	CGS001-3400	ID4	Basic helix-loop-helix proteins			
540	98.22	cp	BRD-K24994810	androstenol	GABA receptor modulator		NR1I3	GABA receptor modulator
541	98.22	cp	BRD-K82746043	navitoclax	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
542	98.22	kd	CGS001-2535	FZD2	GPCR / Class F : Frizzled receptors			
543	98.21	kd	CGS001-1374	CPT1A	-			
544	98.2	oe	ccsbBroad304_06753	POU5F1	Homeoboxes / POU class			
545	98.2	kd	CGS001-11319	ECD	-			
546	98.19	cp	BRD-K88429204	pyrimethamine	Dihydrofolate reductase inhibitor		DHFR, DHFRP1, HEXA, SLC47A1, STAT3	Dihydrofolate reductase inhibitor
547	98.18	oe	ccsbBroad304_01540	SLC2A1	Solute carriers			
548	98.16	oe	ccsbBroad304_13633	PI4KAP2	-			
549	98.16	cp	BRD-A22380646	pantoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
550	98.16	kd	CGS001-10092	ARPC5	Actin related protein 2/3 complex subunits			
551	98.16	kd	CGS001-164668	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
552	98.14	cp	BRD-K61314889	IWR-1-ENDO	PARP inhibitor		TNKS, TNKS2	PARP inhibitor
553	98.12	oe	ccsbBroad304_02855	SPDEF	ETS Transcription Factors			
554	98.12	oe	ccsbBroad304_01187	SLC25A3	Mitochondrial phosphate transporters			
555	98.12	cp	BRD-A71765365	mepireserpate	Catecholamine depleting sympatholytic		SLC18A2, SLC18A1	Catecholamine depleting sympatholytic
556	98.11	kd	CGS001-2597	GAPDH	-			
557	98.1	cc		Cyclooxygenase inhibitor	-			
558	98.1	oe	ccsbBroad304_00016	ACTN4	EF-hand domain containing			
559	98.1	cp	BRD-K93176058	AC-55649	Retinoid receptor agonist		RARB, RARA	Retinoid receptor agonist
560	98.08	cp	BRD-K14993104	bemegride	Chemoreceptor agonist		GABRA1	Chemoreceptor agonist
561	98.07	kd	CGS001-6732	SRPK1	SRPK family			
562	98.06	cp	BRD-K35377380	I-OMe-AG-538	IGF-1 inhibitor			IGF-1 inhibitor
563	98.05	cp	BRD-A65615053	zacopride	Serotonin receptor antagonist		HTR3A, HTR4, HTR3B, HTR5A	Serotonin receptor antagonist
564	98.05	kd	CGS001-657	BMPR1A	Type I receptor serine/threonine kinases			
565	98.04	oe	ccsbBroad304_07077	TSPAN8	Tetraspanins			
566	98.03	oe	ccsbBroad304_06911	MAPK12	MAPK:p38 subfamily			
567	98.02	cp	BRD-A83695761	chromanol	Potassium channel blocker			Potassium channel blocker
568	97.98	oe	ccsbBroad304_03186	GMNN	-			
569	97.97	cp	BRD-K02867583	minaprine	Serotonin reuptake inhibitor		HTR2B, SLC6A4, ACHE, CHRM1, DRD1, DRD2, HTR2A, HTR2C, MAOA	Serotonin reuptake inhibitor
570	97.94	kd	CGS001-7398	USP1	Ubiquitin-specific peptidases			
571	97.94	kd	CGS001-9447	AIM2	-			
572	97.93	kd	CGS001-22850	ADNP2	Zinc fingers, C2H2-type			
573	97.92	kd	CGS001-57594	HOMEZ	Homeoboxes / ZF class			
574	97.92	kd	CGS001-355	FAS	Tumour necrosis factor (TNF) receptor family			
575	97.91	oe	ccsbBroad304_02310	ARPC4	Actin related protein 2/3 complex subunits			
576	97.91	kd	CGS001-10587	TXNRD2	-			
577	97.91	kd	CGS001-10626	TRIM16	Tripartite motif containing			
578	97.91	kd	CGS001-10969	EBNA1BP2	-			
579	97.89	oe	ccsbBroad304_03591	ETNK1	-			
580	97.88	kd	CGS001-11182	SLC2A6	Solute carriers			
581	97.84	oe	ccsbBroad304_01281	PRKCA	Delta subfamily			
582	97.82	kd	CGS001-11072	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
583	97.8	cp	BRD-A29731977	17-hydroxyprogesterone-caproate	progesterone receptor agonist		CYP1A2, CYP2B6, CYP3A5, PGR	progesterone receptor agonist
584	97.79	cp	BRD-K70358946	aripiprazole	Serotonin receptor agonist		DRD2, HTR1A, HTR2A, HRH1, HTR1B, HTR1D, HTR2C, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR1E, HTR3A, HTR6, HTR7	Serotonin receptor agonist, Serotonin receptor antagonist
585	97.79	kd	CGS001-1244	ABCC2	ATP binding cassette transporters / subfamily C			
586	97.75	cp	BRD-K74212935	ergocryptine	Dopamine agonist			Dopamine agonist
587	97.74	kd	CGS001-5601	MAPK9	MAPK:JNK subfamily			
588	97.74	kd	CGS001-8522	GAS7	-			
589	97.72	kd	CGS001-5734	PTGER4	GPCR / Class A : Prostanoid receptors			
590	97.71	oe	ccsbBroad304_07763	NUDT6	Nudix motif containing			
591	97.7	kd	CGS001-4946	OAZ1	-			
592	97.69	cp	BRD-A22844106	tenoxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
593	97.69	kd	CGS001-4967	OGDH	-			
594	97.68	cp	BRD-K05926469	lenalidomide	Antineoplastic		CRBN, TNF, CDH5, PTGS2, TNFSF11	Antineoplastic
595	97.68	cp	BRD-K27499107	carbacyclin	IP receptor activator		PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	IP receptor activator, PPAR receptor agonist
596	97.68	kd	CGS001-64087	MCCC2	-			
597	97.67	oe	ccsbBroad304_09429	FOXP4	Forkhead boxes			
598	97.64	oe	ccsbBroad304_04775	NTAN1	-			
599	97.64	cp	BRD-A74667430	etodolac	Cyclooxygenase inhibitor		PTGS2, PTGS1, RXRA, TRPV1	Cyclooxygenase inhibitor
600	97.64	kd	CGS001-114112	TXNRD3	-			
601	97.63	cp	BRD-K38055836	etamivan	Respiratory stimulant			Respiratory stimulant
602	97.62	kd	CGS001-1978	EIF4EBP1	-			
603	97.62	cp	BRD-A65280694	molindone	Dopamine receptor antagonist		DRD2, HTR2A, CHRM1, DRD5, HRH1, HTR1A	Dopamine receptor antagonist
604	97.61	cp	BRD-K09631521	thiotepa	Cytochrome P450 inhibitor		CYP2B6	Cytochrome P450 inhibitor
605	97.61	kd	CGS001-23077	MYCBP2	-			
606	97.6	oe	ccsbBroad304_08023	EIF2C1	-			
607	97.59	cp	BRD-A04352665	maraviroc	CC chemokine receptor antagonist		CCR5, CYP3A5	CC chemokine receptor antagonist
608	97.59	cp	BRD-A32836748	leu-enkephalin	Opioid receptor agonist		OPRD1, OPRM1	Opioid receptor agonist
609	97.57	cp	BRD-K16664969	GTP-14564	FLT3 inhibitor		FLT3, CSF1R, KIT, PDGFRB	FLT3 inhibitor, Tyrosine kinase inhibitor
610	97.56	cp	BRD-K32710582	EI-247	IGF-1 inhibitor		INSR	IGF-1 inhibitor
611	97.56	cp	BRD-K85503079	perospirone	Dopamine receptor antagonist		DRD2, HTR2A, DRD3, DRD4, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
612	97.56	cp	BRD-K29673530	hypericin	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
613	97.52	kd	CGS001-2185	PTK2B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
614	97.48	oe	ccsbBroad304_03378	ERAP1	Aminopeptidase N			
615	97.45	cp	BRD-K07996107	harpagoside	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
616	97.45	cp	BRD-A18620900	estriol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
617	97.41	cp	BRD-K33396764	alpha-linolenic-acid	Omega 3 fatty acid stimulant		ELOVL4, FADS1, FADS2, FFAR1, FFAR4, PTGS2, SLC8A1, TRPV1	Omega 3 fatty acid stimulant
618	97.37	cp	BRD-K91243525	SR-142948	Neurotensin receptor antagonist		NTSR1	Neurotensin receptor antagonist
619	97.35	kd	CGS001-65264	UBE2Z	Ubiquitin-conjugating enzymes E2			
620	97.33	cp	BRD-K93095519	SJ-172550	MDM inhibitor		MDM4	MDM inhibitor
621	97.33	kd	CGS001-2004	ELK3	ETS Transcription Factors			
622	97.32	oe	ccsbBroad304_00843	IL1B	Interleukins and interleukin receptors			
623	97.31	oe	ccsbBroad304_02394	ZNF267	Zinc fingers, C2H2-type			
624	97.3	oe	ccsbBroad304_01411	RORC	Retinoic acid-related orphans			
625	97.29	cp	BRD-K22385716	LY-303511	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B, MTOR	Casein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
626	97.23	kd	CGS001-3170	FOXA2	Forkhead boxes			
627	97.22	kd	CGS001-84811	BUD13	-			
628	97.22	oe	ccsbBroad304_01249	PPARG	Peroxisome proliferator-activated receptors			
629	97.21	oe	ccsbBroad304_08971	ZNF669	Zinc fingers, C2H2-type			
630	97.19	cp	BRD-K89014967	AS-703026	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
631	97.17	kd	CGS001-440387	CTRB2	-			
632	97.16	cp	BRD-K91601245	mercaptopurine	Immunosuppressant		HPRT1, IMPDH1, IMPDH2, PPAT	Immunosuppressant, Protein synthesis inhibitor, Purine antagonist
633	97.15	oe	ccsbBroad304_02890	SYF2	-			
634	97.14	oe	ccsbBroad304_01447	RPS6KA3	RSK subfamily			
635	97.13	kd	CGS001-9784	SNX17	Sorting nexins			
636	97.11	kd	CGS001-6257	RXRB	Retinoid X receptors			
637	97.11	kd	CGS001-4677	NARS	Aminoacyl tRNA synthetases / Class II			
638	97.07	oe	ccsbBroad304_02579	YWHAQ	-			
639	97.07	kd	CGS001-8767	RIPK2	Receptor interacting protein kinase (RIPK) family			
640	97.02	kd	CGS001-10929	SRSF8	Serine/arginine-rich splicing factors			
641	97.02	kd	CGS001-6446	SGK1	SGK family			
642	97.01	kd	CGS001-7520	XRCC5	XRCC DNA Repair			
643	97	cp	BRD-K33211335	dextromethorphan	Glutamate receptor antagonist		SIGMAR1, CHRNA2, CHRNA3, CHRNA4, CHRNA7, CHRNB2, CHRNB4, CYBA, CYBB, CYP3A5, GRIN1, GRIN3A, NCF1, NCF2, NCF4, OPRD1, OPRK1, OPRM1, PGRMC1, RAC1, RAC2, SLC6A2, SLC6A4	Glutamate receptor antagonist, Sigma receptor agonist
644	96.98	cp	BRD-K61097567	SB-218795	Tachykinin antagonist		TACR3	Tachykinin antagonist
645	96.96	oe	ccsbBroad304_06079	CYP51A1	Cytochrome P450s			
646	96.96	oe	ccsbBroad304_05907	BUB1B	Bub family			
647	96.93	kd	CGS001-9943	OXSR1	FRAY subfamily			
648	96.89	kd	CGS001-8204	NRIP1	-			
649	96.87	cp	BRD-A08877921	cephalotaxine	Protein synthesis inhibitor			Protein synthesis inhibitor
650	96.87	kd	CGS001-336	APOA2	Apolipoproteins			
651	96.84	cc		FGFR inhibitor	-			
652	96.83	kd	CGS001-5962	RDX	-			
653	96.8	oe	ccsbBroad304_02590	SLC27A3	SLC27 family of fatty acid transporters			
654	96.77	cp	BRD-K73982490	BI-78D3	JNK inhibitor		MAPK8	JNK inhibitor
655	96.75	cp	BRD-A75552914	isoxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
656	96.74	cp	BRD-A24381660	zeranol	Estrogen receptor agonist			Estrogen receptor agonist
657	96.72	oe	ccsbBroad304_00047	AKT2	Akt (Protein kinase B)			
658	96.72	kd	CGS001-4811	NID1	-			
659	96.72	kd	CGS001-836	CASP3	Caspases			
660	96.71	cp	BRD-K62310379	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
661	96.7	kd	CGS001-7536	SF1	Zinc fingers, CCHC domain containing			
662	96.69	cp	BRD-K80778372	RO-19-4605	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA benzodiazepine site receptor inverse agonist
663	96.69	kd	CGS001-112885	PHF21B	Zinc fingers, PHD-type			
664	96.68	oe	ccsbBroad304_02270	FAM20B	-			
665	96.68	kd	CGS001-1525	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
666	96.67	cp	BRD-K65146499	nabumetone	Cyclooxygenase inhibitor		PTGS2, AKR1C3, CYP2B6, CYP2C19, CYP2E1, PTGS1	Cyclooxygenase inhibitor
667	96.67	cp	BRD-A49160188	donepezil	Acetylcholinesterase inhibitor		ACHE, HTR2A	Acetylcholinesterase inhibitor
668	96.67	kd	CGS001-2588	GALNS	Arylsulfatase family			
669	96.66	kd	CGS001-8549	LGR5	GPCR / Class A : Orphans			
670	96.65	kd	CGS001-345	APOC3	Apolipoproteins			
671	96.64	cp	BRD-K81209512	AG-494	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
672	96.64	kd	CGS001-117196	MRGPRX4	GPCR / Class A : Orphans			
673	96.63	oe	ccsbBroad304_02402	TMEM5	-			
674	96.63	kd	CGS001-9767	PHF16	-			
675	96.63	kd	CGS001-2260	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
676	96.62	oe	ccsbBroad304_00144	B2M	Immunoglobulin superfamily / C1-set domain containing			
677	96.61	cp	BRD-K97330509	SRC-kinase-inhibitor-II	SRC inhibitor			SRC inhibitor
678	96.59	oe	ccsbBroad304_09992	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
679	96.57	kd	CGS001-5163	PDK1	-			
680	96.55	cp	BRD-K50018155	RS-67506	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
681	96.54	cp	BRD-A30815329	felodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1H, CACNA1S, CACNA2D1, CACNA2D2, CACNB2, CALM1, CFTR, NR3C2, PDE1A, PDE1B, TNNC1, TNNC2	Calcium channel blocker
682	96.54	kd	CGS001-84878	ZBTB45	BTB/POZ domain containing			
683	96.46	kd	CGS001-80237	ELL3	-			
684	96.43	oe	ccsbBroad304_07374	PTPLA	-			
685	96.37	kd	CGS001-6652	SORD	-			
686	96.35	oe	ccsbBroad304_07153	ZNF24	Zinc fingers, C2H2-type			
687	96.3	cp	BRD-K75699339	rizatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1F, HTR1A, HTR1E	Serotonin receptor agonist
688	96.29	cp	BRD-K49945136	GR-113808	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
689	96.29	kd	CGS001-84875	PARP10	Poly (ADP-ribose) polymerases			
690	96.28	kd	CGS001-8807	IL18RAP	CD molecules			
691	96.26	oe	ccsbBroad304_13929	PRKACA	Protein kinase A			
692	96.26	oe	ccsbBroad304_07411	LPXN	-			
693	96.26	kd	CGS001-1147	CHUK	IKK family			
694	96.25	kd	CGS001-219	ALDH1B1	Aldehyde dehydrogenases			
695	96.22	oe	ccsbBroad304_00412	CYP3A5	Cytochrome P450s			
696	96.22	kd	CGS001-462	SERPINC1	Serine (or cysteine) peptidase inhibitors			
697	96.21	oe	ccsbBroad304_12518	STK33	CAMK-unique family			
698	96.2	cp	BRD-K32610195	androstenedione	Cytochrome P450 inhibitor		AKR1C3, HSD17B1, HSD3B1	Cytochrome P450 inhibitor
699	96.19	oe	ccsbBroad304_05818	SLC25A5	Mitochondrial nucleotide transporter subfamily			
700	96.18	kd	CGS001-7089	TLE2	WD repeat domain containing			
701	96.18	kd	CGS001-2203	FBP1	-			
702	96.17	cc		Dihydrofolate reductase inhibitor	-			
703	96.16	cc		Ubiquitin-specific peptidases LOF	-			
704	96.16	kd	CGS001-23200	ATP11B	Phospholipid-transporting ATPases			
705	96.14	cp	BRD-U01690642	acetyl-geranyl-cysteine	Isoprenylated protein methylation inhibitor			Isoprenylated protein methylation inhibitor
706	96.13	oe	ccsbBroad304_06745	PNN	-			
707	96.12	oe	ccsbBroad304_06174	ERCC1	-			
708	96.12	oe	ccsbBroad304_07761	CORO1A	Coronins			
709	96.11	kd	CGS001-26292	MYCBP	-			
710	96.11	kd	CGS001-3784	KCNQ1	Voltage-gated potassium channels			
711	96.11	kd	CGS001-3397	ID1	Basic helix-loop-helix proteins			
712	96.08	kd	CGS001-58528	RRAGD	-			
713	96.07	kd	CGS001-4286	MITF	Basic helix-loop-helix proteins			
714	96.06	oe	ccsbBroad304_00854	IL8	-			
715	96.06	cp	BRD-K34995470	SU-1498	VEGFR inhibitor		ERBB2, KDR	VEGFR inhibitor
716	96.03	cp	BRD-A18763547	BAX-channel-blocker	Cytochrome C release inhibitor		BAX	Cytochrome C release inhibitor
717	95.99	cp	BRD-K47693913	evoxine	Furoquinoline alkaloid			Furoquinoline alkaloid
718	95.98	kd	CGS001-259249	MRGPRX1	GPCR / Class A : Orphans			
719	95.98	kd	CGS001-3456	IFNB1	Interferons			
720	95.97	oe	ccsbBroad304_00356	CPD	Carboxypeptidase A			
721	95.95	oe	ccsbBroad304_02278	THRAP3	-			
722	95.95	cp	BRD-K40782193	QX-222	Sodium channel blocker			Sodium channel blocker
723	95.95	cp	BRD-K46441700	GR-55562	Serotonin receptor antagonist		HTR1B, HTR1D	Serotonin receptor antagonist
724	95.95	kd	CGS001-8650	NUMB	-			
725	95.94	oe	ccsbBroad304_00282	CDKN1A	-			
726	95.94	cp	BRD-K62200014	anagrelide	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
727	95.93	cc		Sigma receptor antagonist	-			
728	95.93	cp	BRD-K08589866	linsitinib	IGF-1 inhibitor		IGF1R, INSR, INSRR	IGF-1 inhibitor
729	95.91	kd	CGS001-6804	STX1A	-			
730	95.9	cp	BRD-A03359064	ICI-89406	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
731	95.89	kd	CGS001-116519	APOA5	Apolipoproteins			
732	95.88	kd	CGS001-10180	RBM6	G patch domain containing			
733	95.86	cp	BRD-K56064827	EI-273	PKC inhibitor		PRKCA, PRKCG	PKC inhibitor
734	95.85	kd	CGS001-8495	PPFIBP2	Sterile alpha motif (SAM) domain containing			
735	95.84	kd	CGS001-23387	SIK3	QIK subfamily			
736	95.84	kd	CGS001-1737	DLAT	-			
737	95.82	kd	CGS001-6812	STXBP1	-			
738	95.81	cp	BRD-K54210043	NS-1619	Calcium channel activator		KCNMA1, KCNT1, KCNT2, KCNU1	Calcium channel activator
739	95.81	kd	CGS001-5286	PIK3C2A	Phosphatidylinositol-4-phosphate 3-kinase family			
740	95.79	oe	ccsbBroad304_07923	LSM5	-			
741	95.78	kd	CGS001-55165	CEP55	-			
742	95.77	cp	BRD-K85603128	resorcinol	Phosphodiesterase inhibitor		CA12, CA14, CA2, PTGS1	Phosphodiesterase inhibitor
743	95.76	cp	BRD-A31204924	mitotane	Antineoplastic		CYP11B1, CYP11A1, CYP3A4, ESR1, FDX1	Antineoplastic
744	95.76	cp	BRD-K39746403	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
745	95.76	kd	CGS001-79751	SLC25A22	Mitochondrial amino acid transporter subfamily			
746	95.75	cp	BRD-A84702196	penicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
747	95.75	kd	CGS001-2735	GLI1	Zinc fingers, C2H2-type			
748	95.74	cp	BRD-A57457122	VU-0400071-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
749	95.72	oe	ccsbBroad304_01084	NEU1	-			
750	95.72	kd	CGS001-6672	SP100	Zinc fingers, PHD-type			
751	95.71	oe	ccsbBroad304_00179	BTG1	-			
752	95.69	cp	BRD-K74195153	irsogladine	Phosphodiesterase inhibitor		PDE4A	Phosphodiesterase inhibitor
753	95.68	cp	BRD-K22096725	ALW-II-49-7	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHA7, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
754	95.66	oe	ccsbBroad304_02825	POLA2	DNA polymerases			
755	95.66	cp	BRD-K50859149	sulfafurazole	Bacterial antifolate			Bacterial antifolate
756	95.65	cp	BRD-K97365803	PI-828	PI3K inhibitor			PI3K inhibitor
757	95.59	cp	BRD-K21971034	OM-137	Aurora kinase inhibitor			Aurora kinase inhibitor
758	95.59	kd	CGS001-6601	SMARCC2	-			
759	95.58	cp	BRD-K61993165	niacin	NAD precursor with lipid lowering effects		HCAR2, HCAR3, ACHE, DGAT2, HCAR1, NNMT, PTGDR, QPRT	NAD precursor with lipid lowering effects, Vitamin B
760	95.56	cp	BRD-K87226815	cycloserine	Bacterial cell wall synthesis inhibitor		GRIN1	Bacterial cell wall synthesis inhibitor
761	95.54	kd	CGS001-27125	AFF4	-			
762	95.53	oe	ccsbBroad304_01555	SNAI2	Snail homologs			
763	95.53	cp	BRD-K63979671	etifenin	Compound used in hepatobiliary scans of the liver			Compound used in hepatobiliary scans of the liver
764	95.5	cp	BRD-A89434049	sarmentogenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
765	95.49	kd	CGS001-58508	MLL3	-			
766	95.48	cp	BRD-K53545112	CNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist
767	95.48	kd	CGS001-23314	SATB2	Homeoboxes / CUT class			
768	95.48	kd	CGS001-26020	LRP10	Low density lipoprotein receptors			
769	95.45	cp	BRD-K19605405	ZM-241385	Adenosine receptor antagonist		ADORA2A, ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
770	95.4	kd	CGS001-148156	ZNF558	Zinc fingers, C2H2-type			
771	95.4	kd	CGS001-8853	ASAP2	Ankyrin repeat domain containing			
772	95.35	kd	CGS001-4176	MCM7	-			
773	95.34	kd	CGS001-3558	IL2	Interleukins and interleukin receptors			
774	95.34	kd	CGS001-90861	HN1L	-			
775	95.32	cp	BRD-A29426959	carbinoxamine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist, L-type calcium channel blocker
776	95.31	cp	BRD-A85472596	L-670596	Prostanoid receptor antagonist			Prostanoid receptor antagonist
777	95.24	cp	BRD-K46212057	voriconazole	Cytochrome P450 inhibitor		CYP2C19, CYP51A1	Cytochrome P450 inhibitor
778	95.24	kd	CGS001-124583	CANT1	-			
779	95.19	cp	BRD-A72066420	mifobate	PPAR receptor antagonist		PPARG, REN	PPAR receptor antagonist
780	95.17	kd	CGS001-7204	TRIO	Rho guanine nucleotide exchange factors			
781	95.15	cp	BRD-K04046242	equilin	Estrogen receptor agonist		HSD17B1	Estrogen receptor agonist
782	95.15	cp	BRD-K18799075	BAY-59-3074	Cannabinoid receptor partial agonist		CNR1, CNR2	Cannabinoid receptor partial agonist
783	95.14	cp	BRD-A65013509	oxybutynin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4	Acetylcholine receptor antagonist
784	95.14	kd	CGS001-57474	ZNF490	Zinc fingers, C2H2-type			
785	95.11	oe	ccsbBroad304_02484	PAICS	-			
786	95.08	cp	BRD-K44876623	zolpidem	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3	Benzodiazepine receptor agonist
787	95.08	cp	BRD-A92826379	lupanine	Sodium channel blocker		INS	Sodium channel blocker
788	95.07	cp	BRD-K79437791	acetyl-farnesyl-cysteine	Inhibitor of methylation of endogenous isoprenylated proteins		PPARG	Inhibitor of methylation of endogenous isoprenylated proteins
789	95.06	kd	CGS001-9355	LHX2	Homeoboxes / LIM class			
790	95.03	oe	ccsbBroad304_06329	GRPR	GPCR / Class A : Bombesin receptors			
791	95.03	cp	BRD-K61480498	epoxycholesterol	LXR agonist		NR1H2, NR1H3	LXR agonist
792	95	oe	ccsbBroad304_00164	BLMH	-			
793	94.99	kd	CGS001-7424	VEGFC	-			
794	94.96	oe	ccsbBroad304_06720	PHYH	-			
795	94.96	kd	CGS001-3431	SP110	Non-enzymatic BRD containing proteins			
796	94.94	kd	CGS001-10538	BATF	basic leucine zipper proteins			
797	94.92	oe	ccsbBroad304_00421	DAPK1	Death-associated kinase (DAPK) family			
798	94.92	kd	CGS001-6850	SYK	Syk family			
799	94.92	kd	CGS001-170591	S100Z	EF-hand domain containing			
800	94.9	oe	ccsbBroad304_00763	HNF4A	Hepatocyte nuclear factor-4 receptors			
801	94.9	cp	BRD-A42346008	metanephrine	Epinephrine metabolite			Epinephrine metabolite
802	94.9	kd	CGS001-5546	PRCC	-			
803	94.87	oe	ccsbBroad304_07135	WNT10B	Wingless-type MMTV integration sites			
804	94.87	kd	CGS001-27102	EIF2AK1	Other PEK family kinases			
805	94.86	cp	BRD-A65550283	ginsenoside	Steroid hormone receptor agonist			Steroid hormone receptor agonist
806	94.85	cp	BRD-K70301876	escitalopram	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ADRA1A, CHRM1, CYP2C19, HRH1, SLC6A2, SLC6A3	Selective serotonin reuptake inhibitor (SSRI)
807	94.85	kd	CGS001-6827	SUPT4H1	-			
808	94.82	kd	CGS001-91392	ZNF502	Zinc fingers, C2H2-type			
809	94.79	cp	BRD-K57222227	indometacin	Cyclooxygenase inhibitor		PTGS1, PTGS2, PPARG, PTGDR2, GLO1, PLA2G2A, PPARA, PTGR2, SLC46A1	Cyclooxygenase inhibitor
810	94.78	cp	BRD-K68264559	brimonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, AOX1	Adrenergic receptor agonist
811	94.77	kd	CGS001-6304	SATB1	Homeoboxes / CUT class			
812	94.75	kd	CGS001-57661	PHRF1	Zinc fingers, PHD-type			
813	94.72	cp	BRD-K62982419	cilomilast	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, IL12A, IL12B, IL1B, PDE4C, TNF	Phosphodiesterase inhibitor
814	94.7	kd	CGS001-55872	PBK	TOPK family			
815	94.69	cp	BRD-A42759514	ornidazole	Antiprotozoal			Antiprotozoal
816	94.69	kd	CGS001-23266	LPHN2	Adhesion Class GPCRs			
817	94.68	kd	CGS001-2065	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
818	94.67	kd	CGS001-54732	TMED9	-			
819	94.65	oe	ccsbBroad304_03950	ATG3	-			
820	94.64	oe	ccsbBroad304_04655	TRIM9	-			
821	94.64	cp	BRD-K08109516	L-701324	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
822	94.64	kd	CGS001-7248	TSC1	-			
823	94.63	oe	ccsbBroad304_03713	RNF20	RING-type (C3HC4) zinc fingers			
824	94.54	oe	ccsbBroad304_06523	LIG1	-			
825	94.53	cp	BRD-A61470182	n-formylmethionylalanine	macrophage activator			macrophage activator
826	94.53	kd	CGS001-114609	TIRAP	-			
827	94.53	kd	CGS001-5641	LGMN	Legumain			
828	94.5	cp	BRD-K18250272	propoxycaine	Local anesthetic			Local anesthetic
829	94.47	cp	BRD-K13725475	rhodomyrtoxin	Cytotoxic agent			Cytotoxic agent, DNA intercalator
830	94.45	cp	BRD-A51714012	venlafaxine	Adrenergic inhibitor		SLC6A2, SLC6A4, CYP2C19, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
831	94.43	cp	BRD-K84639753	safinamide	Dopamine uptake inhibitor		MAOB, SLC6A3	Dopamine uptake inhibitor, Glutamate inhibitor, Monoamine oxidase inhibitor
832	94.43	kd	CGS001-10325	RRAGB	-			
833	94.42	oe	ccsbBroad304_00513	ERCC3	General transcription factors			
834	94.4	oe	ccsbBroad304_04038	ELOVL6	-			
835	94.39	cp	BRD-K15262564	mupirocin	Isoleucyl-tRNA synthetase inhibitor			Isoleucyl-tRNA synthetase inhibitor
836	94.37	kd	CGS001-7292	TNFSF4	CD molecules			
837	94.34	oe	ccsbBroad304_07459	SOCS5	SH2 domain containing			
838	94.34	kd	CGS001-3735	KARS	Aminoacyl tRNA synthetases / Class II			
839	94.29	kd	CGS001-55892	MYNN	BTB/POZ domain containing			
840	94.29	kd	CGS001-4072	EPCAM	CD molecules			
841	94.26	kd	CGS001-54901	CDKAL1	-			
842	94.23	cp	BRD-K72420232	WZ-4002	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor
843	94.23	kd	CGS001-204	AK2	Adenylate kinases			
844	94.2	kd	CGS001-26301	GBGT1	Glycosyltransferase family 6 domain containing			
845	94.18	cp	BRD-A43930669	L-368899	Oxytocin receptor antagonist		OXTR, AVPR1A, AVPR2, OXT	Oxytocin receptor antagonist
846	94.17	kd	CGS001-515	ATP5F1	ATPases / F-type			
847	94.15	kd	CGS001-6271	S100A1	EF-hand domain containing			
848	94.11	oe	ccsbBroad304_02466	ARPC1A	Actin related protein 2/3 complex subunits			
849	94.1	cp	BRD-A15435692	BMY-14802	Sigma receptor antagonist		HTR1A, SIGMAR1	Sigma receptor antagonist
850	94.1	kd	CGS001-23119	HIC2	BTB/POZ domain containing			
851	94.08	oe	ccsbBroad304_06704	PDE4D	Phosphodiesterases			
852	94.06	cp	BRD-K86873305	piperacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
853	94.02	cp	BRD-A34706053	CGP-12177	Adrenergic receptor agonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
854	93.98	oe	ccsbBroad304_01292	EIF2AK2	Other PEK family kinases			
855	93.97	cp	BRD-K14550461	doxercalciferol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
856	93.96	kd	CGS001-1788	DNMT3A	Methyltransferases			
857	93.95	kd	CGS001-57007	CXCR7	-			
858	93.91	cp	BRD-K47192521	icosapent	Platelet aggregation inhibitor		PTGS1, PTGS2, ACSL3, ACSL4, FADS1, FFAR1, PPARD, PPARG, SLC8A1, TRPV1	Platelet aggregation inhibitor
859	93.91	kd	CGS001-9831	ZNF623	Zinc fingers, C2H2-type			
860	93.89	cp	BRD-K68997413	PF-3845	FAAH inhibitor		FAAH	FAAH inhibitor
861	93.87	kd	CGS001-55832	CAND1	-			
862	93.86	cp	BRD-K52930707	rescinnamine	ACE inhibitor		ACE	ACE inhibitor
863	93.8	oe	ccsbBroad304_08596	EAPP	-			
864	93.78	oe	ccsbBroad304_07805	SCAF8	RNA binding motif (RRM) containing			
865	93.78	cp	BRD-K20285085	fostamatinib	SYK inhibitor		SYK, FLT3, RET	SYK inhibitor
866	93.78	kd	CGS001-10793	ZNF273	Zinc fingers, C2H2-type			
867	93.75	cp	BRD-K45252063	clofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
868	93.74	kd	CGS001-5618	PRLR	Prolactin receptor family			
869	93.71	kd	CGS001-5613	PRKX	Protein kinase A			
870	93.67	cp	BRD-A65145453	ATPA	Glutamate receptor agonist		GRIK1, GRIA2	Glutamate receptor agonist
871	93.63	kd	CGS001-10765	KDM5B	Histone demethylases			
872	93.61	cp	BRD-K17349619	HLI-373	MDM inhibitor		MDM2	MDM inhibitor
873	93.57	cp	BRD-A90515964	guaifenesin	Expectorant			Expectorant
874	93.57	kd	CGS001-10725	NFAT5	Nuclear factor of activated T-cells			
875	93.52	kd	CGS001-5498	PPOX	-			
876	93.5	cp	BRD-K66944906	fraxidin	Carbonic anhydrase inhibitor		CA1	Carbonic anhydrase inhibitor
877	93.48	cp	BRD-A26097136	bulleyaconitine-a	Non-opiod analgesic			Non-opiod analgesic
878	93.44	kd	CGS001-6625	SNRNP70	RNA binding motif (RRM) containing			
879	93.44	kd	CGS001-57326	PBXIP1	-			
880	93.44	kd	CGS001-4707	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
881	93.43	kd	CGS001-1515	CTSL2	-			
882	93.4	oe	ccsbBroad304_00032	ADSL	-			
883	93.39	kd	CGS001-27347	STK39	FRAY subfamily			
884	93.37	oe	ccsbBroad304_06660	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
885	93.37	oe	ccsbBroad304_08663	NMUR2	GPCR / Class A : Neuromedin U receptors			
886	93.36	oe	ccsbBroad304_01383	RBMS1	RNA binding motif (RRM) containing			
887	93.36	oe	ccsbBroad304_01287	MAPK8	MAPK:JNK subfamily			
888	93.36	cp	BRD-K96134740	kitasamycin	Protein synthesis inhibitor			Protein synthesis inhibitor
889	93.35	cp	BRD-K05804044	AZ-628	RAF inhibitor		BRAF, RAF1	RAF inhibitor
890	93.35	cp	BRD-K94920105	DR-2313	PARP inhibitor		PARP1, PARP3	PARP inhibitor
891	93.33	kd	CGS001-10613	ERLIN1	-			
892	93.32	cp	BRD-K67566344	KU-0063794	MTOR inhibitor		MTOR	MTOR inhibitor
893	93.32	kd	CGS001-4798	NFRKB	INO80 complex subunits			
894	93.27	cp	BRD-K19360254	ergocornine	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
895	93.26	kd	CGS001-11035	RIPK3	Receptor interacting protein kinase (RIPK) family			
896	93.25	oe	ccsbBroad304_06518	LDHA	-			
897	93.22	kd	CGS001-64094	SMOC2	EF-hand domain containing			
898	93.21	oe	ccsbBroad304_06837	RAF1	RAF family			
899	93.16	kd	CGS001-10643	IGF2BP3	RNA binding motif (RRM) containing			
900	93.13	kd	CGS001-6335	SCN9A	Voltage-gated sodium channels			
901	93.1	cp	BRD-K14200658	syrosingopine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
902	93.05	cp	BRD-K78633253	EXO-1	ARF inhibitor			ARF inhibitor
903	93.04	kd	CGS001-6778	STAT6	SH2 domain containing			
904	93.04	kd	CGS001-1841	DTYMK	-			
905	93.03	cp	BRD-A09467419	mebeverine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
906	93	cp	BRD-K64402243	ivachtin	Caspase inhibitor		CASP3	Caspase inhibitor
907	93	kd	CGS001-5446	PON3	Paraoxonases			
908	92.95	cp	BRD-A78391468	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
909	92.91	cp	BRD-K85871428	SC-68376	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
910	92.88	cp	BRD-K66876909	linezolid	Bacterial 50S ribosomal subunit inhibitor		MAOA	Bacterial 50S ribosomal subunit inhibitor
911	92.87	oe	ccsbBroad304_05759	ACAT2	Lanosterol biosynthesis pathway			
912	92.84	oe	ccsbBroad304_01820	ZNF217	Zinc fingers, C2H2-type			
913	92.84	kd	CGS001-150094	SIK1	QIK subfamily			
914	92.83	kd	CGS001-7554	ZNF8	Zinc fingers, C2H2-type			
915	92.81	kd	CGS001-6883	TAF12	-			
916	92.8	kd	CGS001-11112	HIBADH	-			
917	92.77	oe	ccsbBroad304_01186	PHB	-			
918	92.77	cp	BRD-K10843433	phenylbutazone	Cyclooxygenase inhibitor		PTGS2, PTGS1, PTGIS	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
919	92.75	oe	ccsbBroad304_04817	GABPB2	Ankyrin repeat domain containing			
920	92.74	oe	ccsbBroad304_00429	AKR1C2	Aldo-keto reductases			
921	92.72	oe	ccsbBroad304_01809	ZNF136	Zinc fingers, C2H2-type			
922	92.7	cp	BRD-K43405658	tyrphostin-AG-527	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
923	92.68	kd	CGS001-1044	CDX1	Homeoboxes / ANTP class : HOXL subclass			
924	92.56	cp	BRD-K86727142	embelin	HCV inhibitor		XIAP	HCV inhibitor, XIAP inhibitor
925	92.55	oe	ccsbBroad304_07245	PPFIBP2	Sterile alpha motif (SAM) domain containing			
926	92.55	kd	CGS001-26147	PHF19	Zinc fingers, PHD-type			
927	92.54	oe	ccsbBroad304_07204	TAF15	RNA binding motif (RRM) containing			
928	92.53	oe	ccsbBroad304_06590	MMP7	Matrix metallopeptidase			
929	92.53	kd	CGS001-3127	HLA-DRB5	Immunoglobulin superfamily / C1-set domain containing			
930	92.51	oe	ccsbBroad304_04496	LHX4	Homeoboxes / LIM class			
931	92.51	cp	BRD-K02715688	hydrastine	Tyrosine hydroxylase inhibitor			Tyrosine hydroxylase inhibitor
932	92.47	kd	CGS001-898	CCNE1	-			
933	92.46	cp	BRD-K89687904	PKCbeta-inhibitor	PKC inhibitor		PRKCB	PKC inhibitor
934	92.46	cp	BRD-K05464208	JX-401	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
935	92.44	cc		MEK inhibitor	-			
936	92.42	kd	CGS001-57521	RPTOR	WD repeat domain containing			
937	92.41	kd	CGS001-1209	CLPTM1	-			
938	92.38	oe	ccsbBroad304_00696	CXCL2	Endogenous ligands			
939	92.38	cp	BRD-K78278890	NM-PP1	Mutant kinase inhibitor		CAMK2A, LCK, MAPK8, PRKACA, RIPK2, SRC	Mutant kinase inhibitor
940	92.33	kd	CGS001-5645	PRSS2	Serine peptidases			
941	92.32	oe	ccsbBroad304_01819	ZNF213	Zinc fingers, C2H2-type			
942	92.29	cc		GABA receptor antagonist	-			
943	92.28	oe	ccsbBroad304_06558	MAOB	Catecholamine turnover			
944	92.27	oe	ccsbBroad304_00397	CTSK	Cathepsins			
945	92.27	kd	CGS001-8148	TAF15	RNA binding motif (RRM) containing			
946	92.25	oe	ccsbBroad304_01138	P4HB	Protein disulfide isomerases			
947	92.24	kd	CGS001-5432	POLR2C	RNA polymerase subunits			
948	92.22	cp	BRD-K68341547	W-9	Calmodulin antagonist		CALM2	Calmodulin antagonist
949	92.22	kd	CGS001-6583	SLC22A4	Organic zwitterions/cation transporters (OCTN)			
950	92.2	cp	BRD-K35128472	2-aminopurine	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
951	92.18	cp	BRD-K72024482	MRS-1754	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA2A, ADORA3	Adenosine receptor antagonist
952	92.12	kd	CGS001-158	ADSL	-			
953	92.1	kd	CGS001-50865	HEBP1	Endogenous ligands			
954	92.09	oe	ccsbBroad304_06066	CTSL1	-			
955	92.09	cp	BRD-K57080016	selumetinib	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor
956	92.09	cp	BRD-A20968261	WAY-213613	Glutamate inhibitor		SLC1A2	Glutamate inhibitor
957	92.09	kd	CGS001-3093	UBE2K	Ubiquitin-conjugating enzymes E2			
958	92.09	kd	CGS001-29946	SERTAD3	-			
959	92.08	kd	CGS001-26277	TINF2	-			
960	92.07	cp	BRD-K02953697	naringin	Cytochrome P450 inhibitor		SLCO1A2	Cytochrome P450 inhibitor
961	92.07	kd	CGS001-6050	RNH1	-			
962	92.06	cp	BRD-K19525698	ozagrel	Thromboxane synthase inhibitor		TBXAS1	Thromboxane synthase inhibitor
963	92.04	oe	ccsbBroad304_11251	BRD3	Bromodomain kinase (BRDK) family			
964	92.03	oe	ccsbBroad304_03806	MCOLN1	Voltage-gated ion channels / Transient receptor potential cation channels			
965	92.02	kd	CGS001-11154	AP4S1	-			
966	92.01	cp	BRD-K68191783	ALW-II-38-3	Ephrin inhibitor		DDR1, EPHA2, EPHA4, EPHB2, EPHB4, EPHB6	Ephrin inhibitor
967	92.01	cp	BRD-A02180903	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Anti-inflammatory
968	92	kd	CGS001-3995	FADS3	Fatty acid desaturases			
969	91.97	kd	CGS001-23066	CAND2	-			
970	91.96	cp	BRD-K48692744	NU-1025	PARP inhibitor		PARP1	PARP inhibitor, DNA dependent protein kinase inhibitor
971	91.94	kd	CGS001-5716	PSMD10	Ankyrin repeat domain containing			
972	91.89	cp	BRD-K62374253	rufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
973	91.88	oe	ccsbBroad304_08709	SCYL3	-			
974	91.86	kd	CGS001-3565	IL4	Interleukins and interleukin receptors			
975	91.85	cp	BRD-A06784547	MRS-1334	Adenosine receptor antagonist			Adenosine receptor antagonist
976	91.84	cc		Wnt family LOF	-			
977	91.84	cp	BRD-K53123955	niridazole	Phosphofructokinase inhibitor			Phosphofructokinase inhibitor
978	91.82	cp	BRD-K42095107	daidzein	Estrogen receptor agonist		ESRRA, ESRRB, ESRRG, TRPC5	Estrogen receptor agonist
979	91.79	kd	CGS001-7919	DDX39B	DEAD-boxes			
980	91.78	kd	CGS001-7345	UCHL1	Ubiquitin C-terminal hydrolase			
981	91.77	kd	CGS001-3710	ITPR3	Ion channels / Inositol triphosphate receptors			
982	91.76	kd	CGS001-81533	ITFG1	-			
983	91.74	kd	CGS001-11142	PKIG	-			
984	91.71	kd	CGS001-7484	WNT9B	Wingless-type MMTV integration sites			
985	91.65	cp	BRD-K03384561	roquinimex	Angiogenesis inhibitor			Angiogenesis inhibitor, TNF production inhibitor
986	91.64	kd	CGS001-902	CCNH	General transcription factor IIH complex subunits			
987	91.63	cp	BRD-A37837077	cyclazosin	Adrenergic receptor antagonist		ADRA1B, ADRA1A, ADRA1D	Adrenergic receptor antagonist
988	91.61	cp	BRD-K05396879	15-delta-prostaglandin-j2	PPAR receptor agonist		PPARG, NR1H4	PPAR receptor agonist
989	91.57	oe	ccsbBroad304_04654	ZIM3	Zinc fingers, C2H2-type			
990	91.57	cp	BRD-K84895041	BMY-45778	IP1 prostacyclin receptor agonist		PTGIR	IP1 prostacyclin receptor agonist
991	91.53	oe	ccsbBroad304_03615	ZNF673	-			
992	91.53	cp	BRD-A39522003	OMDM-2	FAAH inhibitor		GPR119	FAAH inhibitor
993	91.52	cp	BRD-K51302260	KU-C103871	GSP agonist		SMAD3	GSP agonist
994	91.51	oe	ccsbBroad304_02143	CNOT8	-			
995	91.42	oe	ccsbBroad304_07880	SIRT5	Histone deacetylases			
996	91.29	oe	ccsbBroad304_07759	PWP1	WD repeat domain containing			
997	91.27	kd	CGS001-79177	ZNF576	Zinc fingers, C2H2-type			
998	91.24	kd	CGS001-10112	KIF20A	Kinesins			
999	91.22	kd	CGS001-7088	TLE1	WD repeat domain containing			
1000	91.21	oe	ccsbBroad304_03357	RASD1	-			
1001	91.2	oe	ccsbBroad304_06173	NR2F6	COUP-TF-like receptors			
1002	91.2	kd	CGS001-10621	POLR3F	RNA polymerase subunits			
1003	91.16	oe	ccsbBroad304_09508	HMGB4	High-mobility group / Canonical			
1004	91.16	cp	BRD-K23335153	AMN-082	Glutamate receptor modulator		GRM7	Glutamate receptor modulator, Glutamate receptor positive allosteric modulator
1005	91.14	cp	BRD-A45140972	meclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor, Bacterial 50S ribosomal subunit inhibitor
1006	91.13	cp	BRD-K88304388	dextrorphan	Glutamate receptor antagonist		OPRM1, OPRK1, OPRD1, GRIN1, HTR1A, SLC6A2	Glutamate receptor antagonist
1007	91.13	kd	CGS001-5104	SERPINA5	Serine (or cysteine) peptidase inhibitors			
1008	91.11	oe	ccsbBroad304_07311	HDAC3	Histone deacetylases			
1009	91.1	oe	ccsbBroad304_10441	PEPD	Methionyl aminopeptidase			
1010	91.1	cp	BRD-K09635134	l-erythro-MAPP	negative control for D-erythro-MAPP			negative control for D-erythro-MAPP
1011	91.09	kd	CGS001-284312	ZSCAN1	Zinc fingers, C2H2-type			
1012	91.07	oe	ccsbBroad304_06928	SDHB	Mitochondrial respiratory chain complex / Complex II			
1013	91	cp	BRD-K02965346	SU-11274	Hepatocyte growth factor receptor inhibitor		MET	Hepatocyte growth factor receptor inhibitor, Tyrosine kinase inhibitor
1014	90.97	oe	ccsbBroad304_02845	PRPF6	-			
1015	90.97	kd	CGS001-5025	P2RX4	Ligand-gated ion channels / Purinergic receptors, ionotropic			
1016	90.92	cp	BRD-A55815733	phylloquinone	Vitamin K		BGLAP, GGCX	Vitamin K, Gamma carboxylase enzyme
1017	90.9	cp	BRD-K71289571	zafirlukast	Leukotriene receptor antagonist		CYSLTR1, CYSLTR2	Leukotriene receptor antagonist
1018	90.89	oe	ccsbBroad304_01767	VDR	Vitamin D receptors			
1019	90.87	kd	CGS001-3693	ITGB5	Integrins			
1020	90.87	kd	CGS001-113878	DTX2	RING-type (C3HC4) zinc fingers			
1021	90.86	cp	BRD-K09668667	benzo(a)pyrene	Carcinogen			Carcinogen
1022	90.83	cp	BRD-A44008656	doxylamine	Histamine receptor antagonist		HRH1, CHRM1	Histamine receptor antagonist
1023	90.81	oe	ccsbBroad304_02879	ZNF473	Zinc fingers, C2H2-type			
1024	90.75	cp	BRD-K83023055	GR-135531	Melatonin receptor agonist			Melatonin receptor agonist
1025	90.74	kd	CGS001-6188	RPS3	S ribosomal proteins			
1026	90.71	kd	CGS001-6009	RHEB	-			
1027	90.67	kd	CGS001-9531	BAG3	-			
1028	90.63	cp	BRD-A48237631	mitomycin-c	DNA alkylating agent			DNA alkylating agent, DNA inhibitor, DNA synthesis inhibitor
1029	90.59	kd	CGS001-23395	LARS2	Aminoacyl tRNA synthetases / Class I			
1030	90.58	kd	CGS001-5723	PSPH	-			
1031	90.57	oe	ccsbBroad304_02553	BLCAP	-			
1032	90.57	kd	CGS001-7105	TSPAN6	Tetraspanins			
1033	90.52	oe	ccsbBroad304_00402	CYB561	Cytochrome b genes			
1034	90.52	cp	BRD-K09255212	clioquinol	Chelating agent		OPRK1	Chelating agent
1035	90.48	kd	CGS001-164091	PAQR7	-			
1036	90.43	kd	CGS001-2831	NPBWR1	GPCR / Class A : Neuropeptide receptors : W/B			
1037	90.39	kd	CGS001-2197	FAU	S ribosomal proteins			
1038	90.37	cp	BRD-A10523515	GSK-429286A	Rho associated kinase inhibitor		ROCK1	Rho associated kinase inhibitor
1039	90.37	cp	BRD-K83010055	VU-0415374-1	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1040	90.34	oe	ccsbBroad304_06287	GM2A	-			
1041	90.3	kd	CGS001-85480	TSLP	-			
1042	90.29	cp	BRD-A98378129	talniflumate	Cyclooxygenase inhibitor		CLCA1	Cyclooxygenase inhibitor
1043	90.29	cp	BRD-A37776212	ICI-204448	Opioid receptor agonist		OPRK1	Opioid receptor agonist
1044	90.27	cp	BRD-K99291625	SB-203580	p38 MAPK inhibitor		MAPK14, MAPK1, MAPK11, AKT1, ALOX5, CHEK1, CYP2D6, CYP3A4, GAK, GSK3B, LCK, MAPK10, MAPK12, MAPK8, MAPK9, PRKCA, RAF1, RIPK2, ROCK1, RPS6KB1, SGK1, SRC, TNF	p38 MAPK inhibitor
1045	90.27	kd	CGS001-2837	UTS2R	Urotensin receptor			
1046	90.26	oe	ccsbBroad304_02455	CREB3	basic leucine zipper proteins			
1047	90.24	oe	ccsbBroad304_01067	NDUFA7	Mitochondrial respiratory chain complex / Complex I			
1048	90.24	oe	ccsbBroad304_08839	IFIH1	-			
1049	90.24	kd	CGS001-51128	SAR1B	-			
1050	90.24	kd	CGS001-80347	COASY	-			
1051	90.15	kd	CGS001-64429	ZDHHC6	Zinc fingers, DHHC-type			
1052	90.14	oe	ccsbBroad304_00127	ATP5B	ATPases / F-type			
1053	90.13	cp	BRD-K97181089	amiloride	Sodium channel blocker		SCNN1A, ASIC1, ASIC2, SCNN1B, SCNN1G, AOC1, ASIC3, PKD2, PKD2L1, PLAU, SCNN1D, SLC9A1, TRPC7, TRPV2	Sodium channel blocker
1054	90.13	kd	CGS001-51116	MRPS2	Mitochondrial ribosomal proteins / small subunits			
1055	90.1	kd	CGS001-51375	SNX7	Sorting nexins			
1056	90.04	oe	ccsbBroad304_00964	SMAD7	SMADs			
1057	90.03	cp	BRD-A55369275	CGP-54626	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
1058	90.03	kd	CGS001-3488	IGFBP5	insulin-like growth factor (IGF) binding proteins			
1059	90.02	kd	CGS001-2099	ESR1	Estrogen receptors			
1060	90.01	oe	ccsbBroad304_01709	NR2C1	Testicular receptors			
1061	89.9	cp	BRD-K09416995	lovastatin	HMGCR inhibitor		HMGCR, CYP3A5, HDAC2, ITGAL, NR1I2	HMGCR inhibitor
1062	89.9	kd	CGS001-6884	TAF13	-			
1063	89.86	kd	CGS001-4208	MEF2C	Myocyte enhancer factors			
1064	89.84	cp	BRD-K08973992	linoleic-acid	Oxidative stress inducer		FABP4, FFAR1, FFAR4, HNF4A, KCNB1, PPARG, TRPM8	Oxidative stress inducer
1065	89.83	cp	BRD-K75615183	talipexole	Adrenergic receptor agonist		DRD2, HTR3A	Adrenergic receptor agonist, Dopamine receptor agonist
1066	89.82	cp	BRD-A37817666	picrotoxin	GABA receptor antagonist		GABRA1, GLRA2, GLRA3, GABRR1, GLRA1, GLRB, HTR3A, HTR3B	GABA receptor antagonist
1067	89.81	kd	CGS001-6597	SMARCA4	Non-enzymatic BRD containing proteins			
1068	89.8	kd	CGS001-9815	GIT2	Ankyrin repeat domain containing			
1069	89.78	cp	BRD-K03981224	ethisterone	Progestogen hormone		TYR	Progestogen hormone
1070	89.78	cp	BRD-A31800922	procyclidine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1071	89.7	oe	ccsbBroad304_02448	UBE2E3	Ubiquitin-conjugating enzymes E2			
1072	89.68	cp	BRD-K64785675	TG100-115	-666		PIK3CG, PIK3CA, PIK3CB, PIK3CD	-666
1073	89.67	kd	CGS001-415116	PIM3	PIM family			
1074	89.64	cp	BRD-K30677119	PP-30	RAF inhibitor		RAF1	RAF inhibitor
1075	89.64	kd	CGS001-811	CALR	-			
1076	89.63	oe	ccsbBroad304_02217	FEZ1	-			
1077	89.63	kd	CGS001-51547	SIRT7	Histone deacetylases (HDACs)			
1078	89.63	cp	BRD-A02333338	cyclopamine	Smoothened receptor antagonist		SMO, DHH, IHH, PTCH1	Smoothened receptor antagonist
1079	89.6	kd	CGS001-57211	GPR126	Adhesion Class GPCRs			
1080	89.59	kd	CGS001-89765	RSPH1	-			
1081	89.58	kd	CGS001-64121	RRAGC	-			
1082	89.57	kd	CGS001-8565	YARS	Aminoacyl tRNA synthetases / Class I			
1083	89.57	cp	BRD-K93880783	stavudine	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor, Reverse transcriptase inhibitor
1084	89.56	kd	CGS001-9448	MAP4K4	MAPKKKK:MSN subfamily			
1085	89.54	oe	ccsbBroad304_02287	GNPDA1	-			
1086	89.52	kd	CGS001-10891	PPARGC1A	RNA binding motif (RRM) containing			
1087	89.51	kd	CGS001-9455	HOMER2	-			
1088	89.5	kd	CGS001-25932	CLIC4	Ion channels / Chloride channels : Intracellular			
1089	89.49	cp	BRD-K92726801	hydrastinine	Haemostatic agent			Haemostatic agent
1090	89.49	kd	CGS001-7159	TP53BP2	Ankyrin repeat domain containing			
1091	89.42	oe	ccsbBroad304_04046	ZNF426	Zinc fingers, C2H2-type			
1092	89.4	kd	CGS001-29116	MYLIP	-			
1093	89.29	oe	ccsbBroad304_07217	AXIN2	-			
1094	89.26	cp	BRD-K25224017	pirenperone	Serotonin receptor antagonist		HTR2A, HTR7	Serotonin receptor antagonist
1095	89.26	cp	BRD-A84174393	meloxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1096	89.25	oe	ccsbBroad304_02526	POP4	-			
1097	89.25	cp	BRD-K02607075	tubocurarine	Acetylcholine receptor antagonist		CHRNA2, HTR3A, ACHE, HTR3B, KCNN1, KCNN2, KCNN3, ZACN	Acetylcholine receptor antagonist
1098	89.21	oe	ccsbBroad304_06055	CSNK1A1	Casein kinase 1 (CK1) family			
1099	89.21	kd	CGS001-64123	ELTD1	Adhesion Class GPCRs			
1100	89.2	oe	ccsbBroad304_00313	TBCB	-			
1101	89.18	kd	CGS001-6391	SDHC	Mitochondrial respiratory chain complex / Complex II			
1102	89.16	kd	CGS001-4245	MGAT1	-			
1103	89.13	oe	ccsbBroad304_02626	PKIG	-			
1104	89.13	cp	BRD-K63089472	farnesylthioacetic-acid	Inhibitor of methyl esterification of farnesylated proteins			Inhibitor of methyl esterification of farnesylated proteins
1105	89.12	oe	ccsbBroad304_05152	SSBP4	-			
1106	89.09	cp	BRD-K79131256	albendazole	Anthelmintic		CYP1A2, CYP2J2, TUBA1A, TUBB, TUBB4B	Anthelmintic, Tubulin inhibitor
1107	89.08	kd	CGS001-9703	KIAA0100	-			
1108	89.07	cp	BRD-K28667793	pyrazinamide	Fatty acid synthase inhibitor		FASN	Fatty acid synthase inhibitor
1109	89.05	kd	CGS001-5985	RFC5	ATPases / AAA-type			
1110	89.02	oe	ccsbBroad304_06739	PLOD1	-			
1111	88.98	oe	ccsbBroad304_07036	TCF4	Basic helix-loop-helix proteins			
1112	88.92	cp	BRD-K62206109	VUF-5681	Histamine receptor antagonist		HRH3	Histamine receptor antagonist
1113	88.92	kd	CGS001-10308	ZNF267	Zinc fingers, C2H2-type			
1114	88.9	cp	BRD-K46018455	bezafibrate	PPAR receptor agonist		PPARA, PPARD, PPARG, HSD11B1, LPL	PPAR receptor agonist
1115	88.89	oe	ccsbBroad304_06226	FTL	-			
1116	88.88	cp	BRD-K12120659	GR-144053	Integrin antagonist		ITGB3, ITGA2B	Integrin antagonist
1117	88.88	kd	CGS001-57491	AHRR	Basic helix-loop-helix proteins			
1118	88.77	cp	BRD-K94070024	depomedrol	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
1119	88.77	kd	CGS001-466	ATF1	basic leucine zipper proteins			
1120	88.73	oe	ccsbBroad304_08183	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1121	88.71	oe	ccsbBroad304_07557	NAMPT	-			
1122	88.71	cp	BRD-K06878038	deferiprone	Chelating agent		CYP4F2	Chelating agent
1123	88.69	cp	BRD-K19554809	MK-212	Serotonin receptor agonist		HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
1124	88.62	cp	BRD-K51941867	LM-1685	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
1125	88.6	oe	ccsbBroad304_06926	SDHA	Mitochondrial respiratory chain complex			
1126	88.51	cp	BRD-A99177642	deltaline	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
1127	88.51	kd	CGS001-286380	FOXD4L3	-			
1128	88.45	kd	CGS001-2987	GUK1	-			
1129	88.44	cp	BRD-K41895714	AS-605240	PI3K inhibitor		MAOB, PIK3CA, PIK3CB, PIK3CD, PIK3CG	PI3K inhibitor
1130	88.4	kd	CGS001-80218	NAA50	N(alpha)-acetyltransferase subunits			
1131	88.38	oe	ccsbBroad304_00520	ETV1	ETS Transcription Factors			
1132	88.34	oe	ccsbBroad304_00775	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
1133	88.31	cp	BRD-K39915878	loxapine	Dopamine receptor antagonist		DRD2, DRD3, DRD4, DRD1, HRH1, HTR2A, HTR2C, HTR6, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD5, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR3A, HTR5A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor antagonist, Dopamine receptor ligand, Serotonin receptor antagonist
1134	88.31	kd	CGS001-25799	ZNF324	Zinc fingers, C2H2-type			
1135	88.25	oe	ccsbBroad304_00962	SMAD4	SMADs			
1136	88.24	kd	CGS001-163059	ZNF433	Zinc fingers, C2H2-type			
1137	88.11	kd	CGS001-10007	GNPDA1	-			
1138	88.1	oe	ccsbBroad304_09768	ZNF366	Zinc fingers, C2H2-type			
1139	88.09	oe	ccsbBroad304_02203	MAD2L1BP	-			
1140	88.08	cc		FXR antagonist	-			
1141	88.08	cp	BRD-K48722833	iloperidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR6, HTR7, ADRA1A, ADRA2C, DRD1, DRD3, DRD4, HRH1	Dopamine receptor antagonist, Serotonin receptor antagonist
1142	87.92	oe	ccsbBroad304_01268	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1143	87.8	kd	CGS001-1948	EFNB2	Ephrins			
1144	87.78	kd	CGS001-2776	GNAQ	-			
1145	87.71	cp	BRD-K69688083	mestinon	Cholinesterase inhibitor		ACHE, BCHE	Cholinesterase inhibitor
1146	87.69	cp	BRD-K95851186	CGP-13501	GABA receptor modulator		GABBR1	GABA receptor modulator
1147	87.61	oe	ccsbBroad304_04626	EGLN3	-			
1148	87.6	oe	ccsbBroad304_06309	UTS2R	Urotensin receptor			
1149	87.57	cp	BRD-K20152659	gamma-homolinolenic-acid	Cholesterol inhibitor		PTGS1, PTGS2	Cholesterol inhibitor, Platelet aggregation inhibitor, Prostanoid receptor agonist, Prostanoid receptor stimulant
1150	87.55	kd	CGS001-23576	DDAH1	Dimethylarginine dimethylaminohydrolases			
1151	87.55	oe	ccsbBroad304_11714	ATMIN	Zinc fingers, C2H2-type			
1152	87.54	kd	CGS001-2872	MKNK2	MKN subfamily			
1153	87.52	kd	CGS001-4189	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
1154	87.51	oe	ccsbBroad304_01648	SERPINA7	Serine (or cysteine) peptidase inhibitors			
1155	87.46	oe	ccsbBroad304_01327	PSPH	-			
1156	87.44	kd	CGS001-4779	NFE2L1	basic leucine zipper proteins			
1157	87.39	kd	CGS001-5573	PRKAR1A	Protein kinase A			
1158	87.39	kd	CGS001-1128	CHRM1	Cholinergic receptors			
1159	87.36	kd	CGS001-6626	SNRPA	RNA binding motif (RRM) containing			
1160	87.34	kd	CGS001-6251	RSU1	-			
1161	87.33	oe	ccsbBroad304_06777	PRNP	CD molecules			
1162	87.33	oe	ccsbBroad304_04947	DYNLL2	Cytoplasmic dyneins			
1163	87.3	cc		Tumor necrosis factor superfamily LOF	-			
1164	87.29	cp	BRD-A51820102	econazole	Bacterial cell wall synthesis inhibitor		CYP51A1, NPY1R, NPY2R, TRPM2, TRPV5	Bacterial cell wall synthesis inhibitor, Lanosterol demethylase inhibitor, Sterol demethylase inhibitor
1165	87.26	cp	BRD-K07888196	tyrphostin-AG-538	IGF-1 inhibitor		EGFR	IGF-1 inhibitor
1166	87.24	oe	ccsbBroad304_01890	FZD7	GPCR / Class F : Frizzled receptors			
1167	87.21	oe	ccsbBroad304_01350	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
1168	87.19	kd	CGS001-3676	ITGA4	Integrins			
1169	87.17	cp	BRD-K01567962	pyrazolanthrone	JNK inhibitor		MAPK10, MAPK8, MAPK9, TTK, LRRK2, MAPK8IP1	JNK inhibitor
1170	87.04	kd	CGS001-2731	GLDC	-			
1171	86.97	kd	CGS001-6887	TAL2	Basic helix-loop-helix proteins			
1172	86.88	cp	BRD-K30570479	VU-0400195-3	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
1173	86.82	cp	BRD-K19416115	sitagliptin	Dipeptidyl peptidase inhibitor		DPP4, CYP2C8, FASLG, HMGCR, SLC22A8	Dipeptidyl peptidase inhibitor
1174	86.81	kd	CGS001-3598	IL13RA2	IL-2 receptor family			
1175	86.8	cp	BRD-A80574334	oxalomalic-acid	Isocitrate dehydrogenase inhibitor		ACO1, IDH1	Isocitrate dehydrogenase inhibitor
1176	86.8	cp	BRD-K04146668	GW-441756	Growth factor receptor inhibitor		LRRK2, NTRK1	Growth factor receptor inhibitor
1177	86.78	kd	CGS001-7001	PRDX2	-			
1178	86.74	oe	ccsbBroad304_00423	DAXX	-			
1179	86.7	cp	BRD-K05673000	dicloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1180	86.7	kd	CGS001-598	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1181	86.69	cp	BRD-K35531059	molsidomine	Guanylyl cyclase activator		GUCY1A3	Guanylyl cyclase activator
1182	86.69	cp	BRD-K37848908	ceforanide	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
1183	86.67	oe	ccsbBroad304_00406	CYP1A1	Cytochrome P450s			
1184	86.6	cp	BRD-K09778810	FGIN-1-27	Inositol monophosphatase inhibitor		TSPO	Inositol monophosphatase inhibitor
1185	86.59	kd	CGS001-1537	CYC1	Mitochondrial respiratory chain complex / Complex III			
1186	86.58	cp	BRD-A29260609	acebutolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
1187	86.56	kd	CGS001-6491	STIL	-			
1188	86.53	cp	BRD-K93258693	GW-9662	PPAR receptor antagonist		PPARG, NCOA2, RXRA	PPAR receptor antagonist
1189	86.51	cp	BRD-K67100011	pivmecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1190	86.46	cp	BRD-K92817986	BJM-CSC-19	MEK inhibitor			MEK inhibitor
1191	86.42	cp	BRD-K27871032	lysergol	Ergoline alkaloid		HTR1B, HTR1D, HTR1E	Ergoline alkaloid
1192	86.41	cp	BRD-A23683907	NAS-181	Serotonin receptor antagonist		HTR1B	Serotonin receptor antagonist
1193	86.38	oe	ccsbBroad304_02838	SDF2L1	-			
1194	86.37	kd	CGS001-7071	KLF10	Kruppel-like transcription factors			
1195	86.35	kd	CGS001-10795	ZNF268	Zinc fingers, C2H2-type			
1196	86.27	cp	BRD-K49456190	prima-1-met	thioredoxin inhibitor		TP53	thioredoxin inhibitor
1197	86.26	oe	ccsbBroad304_06845	RARRES3	-			
1198	86.21	oe	ccsbBroad304_07097	TRAF1	-			
1199	86.17	oe	ccsbBroad304_07074	TLR2	Toll-like receptor family			
1200	86.17	cp	BRD-K27450477	EHNA	Adenosine deaminase inhibitor		ADA, PDE2A, ADORA2A	Adenosine deaminase inhibitor
1201	86.17	cp	BRD-K17008822	BD-1008	Sigma receptor antagonist			Sigma receptor antagonist
1202	86.17	cp	BRD-K98426715	tubacin	HDAC inhibitor		HDAC6	HDAC inhibitor
1203	86.12	kd	CGS001-6603	SMARCD2	-			
1204	86.11	oe	ccsbBroad304_06974	SLC22A5	Organic zwitterions/cation transporters (OCTN)			
1205	86.07	cp	BRD-A17448384	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist
1206	86.06	oe	ccsbBroad304_07657	ATP5L	ATPases / F-type			
1207	86.05	cp	BRD-K28667196	fillalbin	Increases arterial blood pressure			Increases arterial blood pressure
1208	86.02	kd	CGS001-10392	NOD1	Nucleotide-binding domain and leucine rich repeat containing			
1209	86.01	kd	CGS001-11157	LSM6	-			
1210	85.98	oe	ccsbBroad304_00491	EIF4EBP2	-			
1211	85.97	kd	CGS001-4016	LOXL1	-			
1212	85.93	kd	CGS001-9788	MTSS1	-			
1213	85.92	kd	CGS001-7342	UBP1	-			
1214	85.89	cp	BRD-K33226500	indinavir	HIV protease inhibitor		CYP3A5	HIV protease inhibitor
1215	85.78	kd	CGS001-7263	TST	-			
1216	85.75	kd	CGS001-10252	SPRY1	-			
1217	85.73	oe	ccsbBroad304_06778	PROC	Endogenous ligands			
1218	85.66	cp	BRD-K86191271	cytosporone-b	NUR77 receptor agonist		NR4A1	NUR77 receptor agonist
1219	85.65	cp	BRD-A09161221	nomilin	HSP inhibitor			HSP inhibitor
1220	85.62	kd	CGS001-2787	GNG5	-			
1221	85.6	cp	BRD-A01826957	xanthinol	Vasodilator			Vasodilator
1222	85.59	oe	ccsbBroad304_09413	ZNF554	Zinc fingers, C2H2-type			
1223	85.57	oe	ccsbBroad304_00954	LYN	Src family			
1224	85.57	kd	CGS001-1845	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1225	85.57	oe	ccsbBroad304_02566	MORF4L1	-			
1226	85.5	kd	CGS001-1632	ECI1	-			
1227	85.5	cp	BRD-K34098590	tienilic-acid	Sodium/potassium/chloride transporter inhibitor		CYP2C9, SLC12A1, SLC22A12	Sodium/potassium/chloride transporter inhibitor
1228	85.49	oe	ccsbBroad304_10431	HADHB	-			
1229	85.49	oe	ccsbBroad304_00028	ADH5	Alcohol dehydrogenases			
1230	85.49	cp	BRD-K63923597	barasertib	Aurora kinase inhibitor		AURKB, AURKC	Aurora kinase inhibitor
1231	85.47	oe	ccsbBroad304_02501	DCTN6	-			
1232	85.47	kd	CGS001-2976	GTF3C2	General transcription factors			
1233	85.47	kd	CGS001-10987	COPS5	-			
1234	85.35	cp	BRD-K57179821	crotamiton	Antipruritic			Antipruritic
1235	85.32	kd	CGS001-10049	DNAJB6	Heat shock proteins / DNAJ (HSP40)			
1236	85.24	cc		P38 MAPK inhibitor	-			
1237	85.19	kd	CGS001-29102	DROSHA	-			
1238	85.06	kd	CGS001-3992	FADS1	Fatty acid desaturases			
1239	85.03	oe	ccsbBroad304_06789	PSEN2	Presenilin			
1240	85.01	oe	ccsbBroad304_01748	UFD1L	-			
1241	85	kd	CGS001-238	ALK	Leukocyte tyrosine kinase (LTK) receptor family			
1242	84.99	kd	CGS001-3416	IDE	Pitrilysin			
1243	84.96	kd	CGS001-7016	TESK1	TESK subfamily			
1244	84.95	oe	ccsbBroad304_02633	LSM6	-			
1245	84.95	kd	CGS001-55206	SBNO1	-			
1246	84.92	oe	ccsbBroad304_04406	PLA2G12B	-			
1247	84.89	oe	ccsbBroad304_03215	MRPS2	Mitochondrial ribosomal proteins / small subunits			
1248	84.85	cp	BRD-K50720187	flupirtine	Glutamate receptor antagonist		KCNQ2, ADRA2A, KCNQ1, KCNQ3	Glutamate receptor antagonist
1249	84.85	cp	BRD-A11813248	AM-92016	Potassium channel blocker		GRIN1, GRIN2B	Potassium channel blocker
1250	84.84	kd	CGS001-51174	TUBD1	Tubulins			
1251	84.83	cp	BRD-A97701745	pindolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A, HTR1B, HTR2A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist
1252	84.79	kd	CGS001-10845	CLPX	ATPases / AAA-type			
1253	84.77	cc		Calmodulin antagonist	-			
1254	84.75	cp	BRD-K92731339	perindopril	ACE inhibitor		ACE	ACE inhibitor
1255	84.73	cp	BRD-A09062839	amylocaine	Local anesthetic			Local anesthetic
1256	84.63	kd	CGS001-3242	HPD	Oxidoreductases			
1257	84.62	kd	CGS001-23753	SDF2L1	-			
1258	84.61	cp	BRD-K32584078	BML-257	AKT inhibitor		AKT1	AKT inhibitor, HCV inhibitor
1259	84.52	kd	CGS001-56139	PCDHA10	Cadherins / Protocadherins : Clustered			
1260	84.49	oe	ccsbBroad304_02401	AKR1A1	Aldo-keto reductases			
1261	84.48	kd	CGS001-11168	PSIP1	-			
1262	84.37	kd	CGS001-624	BDKRB2	Bradykinin receptors			
1263	84.34	oe	ccsbBroad304_00135	ATP6V0C	ATPases / V-type			
1264	84.34	cp	BRD-K43887077	dopamine	Dopamine receptor agonist		DRD2, DRD1, DRD3, DRD4, DRD5, DBH, HTR1A, HTR7, SLC6A2, SLC6A3, SLC6A4	Dopamine receptor agonist
1265	84.24	kd	CGS001-995	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1266	84.23	oe	ccsbBroad304_02057	P4HA2	-			
1267	84.2	kd	CGS001-5031	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
1268	84.18	kd	CGS001-596	BCL2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
1269	84.12	kd	CGS001-134864	TAAR1	GPCR / Class A : Trace amine associated receptors			
1270	84.09	cp	BRD-K74430258	1,2-dichlorobenzene	Hepatotoxicant			Hepatotoxicant, Organic compound
1271	84.07	cp	BRD-A52193669	withaferin-a	IKK inhibitor		ACHE, BCHE, IKBKB	IKK inhibitor
1272	84.05	oe	ccsbBroad304_01323	PSMD9	Proteasome (prosome, macropain) subunits			
1273	84.02	oe	ccsbBroad304_02137	TRIP13	ATPases / AAA-type			
1274	84.02	cp	BRD-K30197592	5-methoxytryptamine	Serotonin receptor agonist		HTR2A, HTR6, HTR1B, HTR1D, HTR1E, HTR1F, HTR2C, HTR4, HTR7, TRPM8	Serotonin receptor agonist
1275	84.02	kd	CGS001-79071	ELOVL6	-			
1276	83.98	cp	BRD-K37846922	3,3'-diindolylmethane	CHK inhibitor		AHR, AR, CYP1A2, GUSB, IDO1	CHK inhibitor, Cytochrome P450 activator, Indoleamine 2,3-dioxygenase inhibitor
1277	83.97	oe	ccsbBroad304_01304	PSEN1	Presenilin			
1278	83.93	kd	CGS001-10128	LRPPRC	-			
1279	83.9	oe	ccsbBroad304_04431	PHF5A	Zinc fingers, PHD-type			
1280	83.9	kd	CGS001-10014	HDAC5	Histone deacetylases			
1281	83.89	cp	BRD-K44094599	tacrolimus	Calcineurin inhibitor		FKBP1A, CYP3A5, CYP3A7	Calcineurin inhibitor
1282	83.88	cp	BRD-K86509404	iso-olomoucine	CDK inhibitor			CDK inhibitor
1283	83.86	cp	BRD-A24122750	saclofen	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
1284	83.84	cp	BRD-K82091397	SB-239063	p38 MAPK inhibitor		MAPK11, MAPK14, PTGS2, TNF	p38 MAPK inhibitor
1285	83.84	kd	CGS001-54620	FBXL19	F-boxes / Leucine-rich repeats			
1286	83.82	oe	ccsbBroad304_00222	CASP6	Caspases			
1287	83.78	kd	CGS001-6595	SMARCA2	Non-enzymatic BRD containing proteins			
1288	83.78	kd	CGS001-1545	CYP1B1	Cytochrome P450s			
1289	83.71	cp	BRD-K53959060	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor, Glycogen synthase kinase inhibitor, Leucine rich repeat kinase inhibitor, SRC inhibitor, Serum/glucocorticoid regulated kinase inhibitor
1290	83.67	oe	ccsbBroad304_07197	PDHX	-			
1291	83.66	cp	BRD-K72222507	quinapril	ACE inhibitor		ACE	ACE inhibitor
1292	83.59	kd	CGS001-115196	ZNF554	Zinc fingers, C2H2-type			
1293	83.58	cp	BRD-K04185004	oxybuprocaine	Local anesthetic		SCN10A	Local anesthetic
1294	83.55	cp	BRD-K03440695	boldine	Acetylcholine receptor antagonist		CHRNA4, CHRNB2, DRD1, DRD2	Acetylcholine receptor antagonist, Dopamine receptor antagonist
1295	83.52	kd	CGS001-65123	INTS3	-			
1296	83.5	cp	BRD-K60770992	pergolide	Dopamine receptor agonist		DRD1, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, KCNA5	Dopamine receptor agonist
1297	83.34	cp	BRD-K28168037	fenretinide	Apoptosis stimulant		CYP2C8, CYP3A5, RARA, RARG	Apoptosis stimulant, Retinoid receptor agonist
1298	83.29	cp	BRD-A56020723	CA-074-Me	Cathepsin inhibitor		CTSB	Cathepsin inhibitor
1299	83.25	oe	ccsbBroad304_13991	NCOA3	Histone acetyltransferases			
1300	83.24	kd	CGS001-199777	ZNF626	Zinc fingers, C2H2-type			
1301	83.22	cp	BRD-K29173907	isoflupredone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
1302	83.19	kd	CGS001-58478	ENOPH1	-			
1303	83.15	cp	BRD-A54845972	dihydroergotamine	Serotonin receptor agonist		HTR1D, HTR1B, ADRA2A, DRD2, HTR1E, HTR1F, HTR2B, HTR7	Serotonin receptor agonist
1304	83.14	kd	CGS001-375	ARF1	ADP-ribosylation factors			
1305	83.01	oe	ccsbBroad304_01066	NDUFA4	-			
1306	83	kd	CGS001-11140	CDC37	-			
1307	82.89	cp	BRD-A99571536	dubinidine	Anti-epileptic			Anti-epileptic
1308	82.87	cp	BRD-K92000912	AM-251	Cannabinoid receptor antagonist		CNR1, GPR18, GPR55	Cannabinoid receptor antagonist
1309	82.86	oe	ccsbBroad304_06840	RAP1GDS1	Armadillo repeat containing			
1310	82.84	cp	BRD-K34533029	tyrphostin-AG-494	EGFR inhibitor		EGFR	EGFR inhibitor
1311	82.79	kd	CGS001-8517	IKBKG	Zinc fingers, C2HC-type containing			
1312	82.77	kd	CGS001-9797	TATDN2	-			
1313	82.7	kd	CGS001-523	ATP6V1A	ATPases / V-type			
1314	82.68	oe	ccsbBroad304_05803	ALDH3B2	Aldehyde dehydrogenases			
1315	82.66	oe	ccsbBroad304_02578	EBNA1BP2	-			
1316	82.66	cp	BRD-A67438293	treprostinil	Prostacyclin analog		PTGIR, CYP2C8, P2RY12, PPARD, PTGDR, PTGER1, PTGER2, PTGER3, PTGER4	Prostacyclin analog
1317	82.66	cp	BRD-K52620403	STO-609	Calmodulin antagonist		CAMKK1, CAMKK2	Calmodulin antagonist
1318	82.65	kd	CGS001-2244	FGB	Endogenous ligands			
1319	82.62	kd	CGS001-9093	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
1320	82.57	oe	ccsbBroad304_01576	SOAT1	-			
1321	82.51	oe	ccsbBroad304_04998	ZNF418	Zinc fingers, C2H2-type			
1322	82.51	cp	BRD-K49657628	tyrphostin-AG-18	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
1323	82.49	cp	BRD-A00100033	nifurtimox	DNA inhibitor			DNA inhibitor
1324	82.46	kd	CGS001-8702	B4GALT4	Beta 4-glycosyltransferases			
1325	82.43	kd	CGS001-10401	PIAS3	Zinc fingers, MIZ-type			
1326	82.42	kd	CGS001-5515	PPP2CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
1327	82.38	kd	CGS001-2254	FGF9	Endogenous ligands			
1328	82.32	kd	CGS001-6347	CCL2	Chemokine ligands			
1329	82.31	cp	BRD-K41713976	E-4031	Potassium channel blocker		KCNH2, KCNH1	Potassium channel blocker
1330	82.28	cc		Aurora kinase inhibitor	-			
1331	82.26	cc		General transcription factors group 1 LOF	-			
1332	82.26	cp	BRD-K53561341	KIN001-220	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
1333	82.25	kd	CGS001-140612	ZFP28	Zinc fingers, C2H2-type			
1334	82.22	cp	BRD-K69556541	ryanodine	Calcium channel blocker		RYR1, RYR2, RYR3	Calcium channel blocker
1335	82.21	kd	CGS001-55214	LEPREL1	-			
1336	82.2	kd	CGS001-109	ADCY3	Adenylyl cyclases			
1337	82.14	kd	CGS001-286075	ZNF707	Zinc fingers, C2H2-type			
1338	82.14	kd	CGS001-8525	DGKZ	-			
1339	82.1	cp	BRD-K15868788	SDZ-205-557	Serotonin receptor antagonist		HTR3A, HTR3B, HTR4	Serotonin receptor antagonist
1340	82.09	kd	CGS001-2957	GTF2A1	General transcription factors			
1341	82.06	oe	ccsbBroad304_06179	ERG	ETS Transcription Factors			
1342	82.05	cp	BRD-A71009679	KUC103420N	-666			-666
1343	81.95	kd	CGS001-8446	DUSP11	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
1344	81.94	kd	CGS001-117194	MRGPRX2	GPCR / Class A : Orphans			
1345	81.89	kd	CGS001-55632	G2E3	Zinc fingers, PHD-type			
1346	81.83	oe	ccsbBroad304_00679	GPR39	GPCR / Class A : Orphans			
1347	81.78	oe	ccsbBroad304_00573	FKBP4	Tetratricopeptide (TTC) repeat domain containing			
1348	81.78	kd	CGS001-6520	SLC3A2	SLC3 family			
1349	81.75	kd	CGS001-7428	VHL	-			
1350	81.74	cp	BRD-K79930101	GW-583340	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, ErbB2 inhibitor, Receptor tyrosine protein kinase inhibitor
1351	81.66	kd	CGS001-6286	S100P	EF-hand domain containing			
1352	81.59	cp	BRD-K09859624	methantheline	Acetylcholine receptor antagonist		CHRM1, HRH2	Acetylcholine receptor antagonist
1353	81.58	cc		Cell Cycle Inhibition GOF	-			
1354	81.53	oe	ccsbBroad304_00612	GALNS	Arylsulfatase family			
1355	81.52	cp	BRD-K39520573	GW-5074	Leucine rich repeat kinase inhibitor		LRRK1, LRRK2, NTRK1, RAF1	Leucine rich repeat kinase inhibitor, RAF inhibitor
1356	81.51	oe	ccsbBroad304_07314	ASAP2	Ankyrin repeat domain containing			
1357	81.5	cp	BRD-K36864847	BD-1047	Adrenergic receptor antagonist		SIGMAR1	Adrenergic receptor antagonist
1358	81.43	cp	BRD-A49172652	lansoprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4, CYP3A5	ATPase inhibitor
1359	81.37	kd	CGS001-7481	WNT11	Wingless-type MMTV integration sites			
1360	81.33	kd	CGS001-467	ATF3	basic leucine zipper proteins			
1361	81.32	kd	CGS001-338557	O3FAR1	-			
1362	81.23	kd	CGS001-5004	ORM1	Lipocalins			
1363	81.19	kd	CGS001-23369	PUM2	-			
1364	81.18	kd	CGS001-221	ALDH3B1	Aldehyde dehydrogenases			
1365	81.16	cp	BRD-A28318179	aminomethyltransferase	Nitric oxide synthase inhibitor		NOS2	Nitric oxide synthase inhibitor
1366	81.16	kd	CGS001-54386	TERF2IP	-			
1367	81.04	cp	BRD-U82589721	HG-5-113-01	Protein kinase inhibitor		ABL1, LTK, STK10	Protein kinase inhibitor
1368	81.02	oe	ccsbBroad304_01589	SQLE	Lanosterol biosynthesis pathway			
1369	80.96	cp	BRD-A96255180	ribavirin	Antiviral		IMPDH1, ADK, ENPP1, IMPDH2, NT5C2	Antiviral
1370	80.95	cp	BRD-K43797669	genistein	Tyrosine kinase inhibitor		CFTR, ESR2, EGFR, ESR1, ESRRA, ESRRB, ESRRG, NCOA1, NCOA2, PPARG, PTK2B, TOP2A, TRPC5	Tyrosine kinase inhibitor
1371	80.89	kd	CGS001-7692	ZNF133	Zinc fingers, C2H2-type			
1372	80.88	kd	CGS001-5684	PSMA3	Proteasome subunits			
1373	80.79	cp	BRD-K92428232	GSK-461364	PLK inhibitor		PLK1	PLK inhibitor
1374	80.77	kd	CGS001-54578	UGT1A6	UDP glucuronosyltransferases			
1375	80.74	kd	CGS001-1287	COL4A5	Collagens			
1376	80.73	oe	ccsbBroad304_02862	CCRN4L	-			
1377	80.57	cp	BRD-K10176267	L-701252	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
1378	80.57	kd	CGS001-4664	NAB1	-			
1379	80.57	kd	CGS001-139378	GPR112	Adhesion Class GPCRs			
1380	80.49	oe	ccsbBroad304_00163	PRDM1	Zinc fingers, C2H2-type			
1381	80.49	cp	BRD-A34751532	homosalate	HSP inducer			HSP inducer
1382	80.41	cp	BRD-A83855350	naltrexone	Opioid receptor antagonist		OPRK1, OPRM1, OPRD1, SIGMAR1	Opioid receptor antagonist
1383	80.41	kd	CGS001-10287	RGS19	Regulators of G-protein signaling			
1384	80.4	cp	BRD-K71499074	diclofenamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA12, CA7	Carbonic anhydrase inhibitor
1385	80.39	cc		S100 calcium binding proteins LOF	-			
1386	80.33	cp	BRD-K12762134	XAV-939	Tankyrase inhibitor		TNKS, TNKS2	Tankyrase inhibitor
1387	80.32	kd	CGS001-708	C1QBP	-			
1388	80.28	cc		Non Homologous End Joining LOF	-			
1389	80.28	kd	CGS001-10933	MORF4L1	-			
1390	80.26	cp	BRD-K31054881	BMY-7378	Adrenergic receptor antagonist		HTR1A, ADRA1D, ADRA1A, ADRA1B	Adrenergic receptor antagonist, Serotonin receptor antagonist
1391	80.2	cp	BRD-K03600606	catechin	Beta secretase inhibitor		BACE1, CA1, CA12, CA14, CA2, CA4, CA6, CA9, FASN, PTGS1, SCN5A	Beta secretase inhibitor, Fatty acid synthase inhibitor, LDL antioxidant
1392	80.16	kd	CGS001-117581	TWIST2	Basic helix-loop-helix proteins			
1393	80.13	kd	CGS001-50808	AK3	-			
1394	80.09	kd	CGS001-5584	PRKCI	Iota subfamily			
1395	80.03	cp	BRD-K81876028	CP-93129	Serotonin receptor agonist		HTR1A, HTR1B	Serotonin receptor agonist
1396	80.03	cp	BRD-K49865102	PD-0325901	MEK inhibitor		MAP2K1, MAP2K2	MEK inhibitor, MAP kinase inhibitor, Protein kinase inhibitor
1397	80	kd	CGS001-80714	PBX4	Homeoboxes / TALE class			
1398	79.93	kd	CGS001-146540	ZNF785	Zinc fingers, C2H2-type			
1399	79.91	oe	ccsbBroad304_03433	DDIT4	-			
1400	79.91	kd	CGS001-25801	GCA	EF-hand domain containing			
1401	79.89	cp	BRD-K09764130	mead-ethanolamide	Cannabinoid receptor agonist			Cannabinoid receptor agonist
1402	79.88	kd	CGS001-5433	POLR2D	RNA polymerase subunits			
1403	79.86	oe	ccsbBroad304_00578	FLI1	ETS Transcription Factors			
1404	79.84	kd	CGS001-10628	TXNIP	-			
1405	79.83	cp	BRD-K13571841	pepstatin	Aspartic protease inhibitor		CTSB, CTSD, CTSL, REN	Aspartic protease inhibitor
1406	79.8	oe	ccsbBroad304_05901	POLR3D	RNA polymerase subunits			
1407	79.76	cp	BRD-K17306061	aprepitant	Tachykinin antagonist		TACR1, CYP2C19	Tachykinin antagonist
1408	79.74	oe	ccsbBroad304_00995	MECP2	-			
1409	79.7	cp	BRD-K25906698	immepip	Histamine receptor agonist		HRH3, HRH4	Histamine receptor agonist
1410	79.67	cp	BRD-K59184148	SB-216763	Glycogen synthase kinase inhibitor		GSK3B, CCNA2, CDK2, GSK3A	Glycogen synthase kinase inhibitor
1411	79.61	cp	BRD-K33818169	GW-3965	LXR agonist		NR1H2, NR1H3, ABCA1	LXR agonist, ABC transporter expression enhancer
1412	79.54	cp	BRD-K50135270	GBR-12935	Dopamine uptake inhibitor		AGTR1, SLC6A3	Dopamine uptake inhibitor
1413	79.52	kd	CGS001-6655	SOS2	Rho guanine nucleotide exchange factors			
1414	79.5	oe	ccsbBroad304_08230	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
1415	79.46	kd	CGS001-8869	ST3GAL5	Sialyltransferases			
1416	79.43	oe	ccsbBroad304_00515	ERH	-			
1417	79.4	kd	CGS001-147686	ZNF418	Zinc fingers, C2H2-type			
1418	79.35	kd	CGS001-3105	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
1419	79.34	cp	BRD-K62965247	tipifarnib-P2	farnesyltransferase inhibitor		FNTA, FNTB	farnesyltransferase inhibitor
1420	79.33	cp	BRD-K32107296	temozolomide	DNA alkylating agent		TOP2A	DNA alkylating agent
1421	79.33	cp	BRD-A91699651	chloroquine	Antimalarial		CYP2C8, GSTA2, MRGPRX1, TLR9, TNF	Antimalarial
1422	79.27	kd	CGS001-90678	LRSAM1	Sterile alpha motif (SAM) domain containing			
1423	79.19	cp	BRD-A54927599	KF-38789	P-selectin inhibitor		SELP	P-selectin inhibitor
1424	79.18	cp	BRD-A47633927	NPC-15199	ICAM1 antagonist		ICAM1, PPARG	ICAM1 antagonist
1425	79.17	oe	ccsbBroad304_07326	EIF2B2	-			
1426	79.17	cp	BRD-A00520476	otenzepad	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
1427	79.17	kd	CGS001-5575	PRKAR1B	Protein kinase A			
1428	79.16	oe	ccsbBroad304_02834	GABARAPL1	-			
1429	79.16	cp	BRD-K70281171	U-99194	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
1430	79.13	kd	CGS001-27109	ATP5S	-			
1431	79.06	oe	ccsbBroad304_06785	PRSS2	Serine peptidases			
1432	79.05	cp	BRD-K97061094	azacyclonol	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
1433	79.05	kd	CGS001-8569	MKNK1	MKN subfamily			
1434	79.04	oe	ccsbBroad304_00433	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1435	79.03	kd	CGS001-7157	TP53	-			
1436	79	cc		Homeobox Gene GOF	-			
1437	79	cp	BRD-K33459542	ditolylguanidine	Sigma receptor agonist		GRIN1, GRIN2A, GRIN2B, SIGMAR1	Sigma receptor agonist
1438	78.97	cp	BRD-K28428262	brivanib	FGFR inhibitor		FGFR1, KDR, FLT1, CYP3A4, FGFR2, FGFR3, FLT4, KCNH2	FGFR inhibitor, VEGFR inhibitor
1439	78.87	oe	ccsbBroad304_07918	CBLC	RING-type (C3HC4) zinc fingers			
1440	78.84	cp	BRD-K95402279	geranylgeraniol	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
1441	78.82	cp	BRD-A80641450	FR-139317	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
1442	78.8	kd	CGS001-9453	GGPS1	Lanosterol biosynthesis pathway			
1443	78.77	kd	CGS001-3659	IRF1	-			
1444	78.6	oe	ccsbBroad304_01453	RPS14	S ribosomal proteins			
1445	78.54	kd	CGS001-22921	MSRB2	-			
1446	78.52	oe	ccsbBroad304_05564	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
1447	78.5	oe	ccsbBroad304_04243	PLA2G12A	Phospholipase A2			
1448	78.49	kd	CGS001-6720	SREBF1	Basic helix-loop-helix proteins			
1449	78.48	kd	CGS001-7534	YWHAZ	-			
1450	78.45	oe	ccsbBroad304_03415	GFOD1	-			
1451	78.36	cp	BRD-A35108200	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist
1452	78.34	cp	BRD-K58772419	AZD-6482	PI3K inhibitor		PIK3CD, PIK3CG, PIK3CA, PIK3CB	PI3K inhibitor
1453	78.34	kd	CGS001-6935	ZEB1	Zinc fingers, C2H2-type			
1454	78.3	cp	BRD-K25310650	ormetoprim	Bacterial antifolate			Bacterial antifolate
1455	78.29	oe	ccsbBroad304_03006	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
1456	78.21	oe	ccsbBroad304_07600	NSA2	-			
1457	78.17	kd	CGS001-5711	PSMD5	Proteasome (prosome, macropain) subunits			
1458	78.16	cp	BRD-K31542390	mycophenolic-acid	Dehydrogenase inhibitor		IMPDH1, IMPDH2	Dehydrogenase inhibitor, Inositol monophosphatase inhibitor
1459	78.15	oe	ccsbBroad304_00624	GCK	Hexokinases			
1460	78.13	cp	BRD-K18316707	O-1918	Cannabinoid receptor antagonist			Cannabinoid receptor antagonist
1461	78.1	cp	BRD-K28120222	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor
1462	78.07	cp	BRD-K35687265	ON-01910	PLK inhibitor		CDK1, FLT1, FYN, MCL1, PDGFRA, PLK1, PLK2, SRC	PLK inhibitor
1463	78.04	cp	BRD-K50938287	sumatriptan	Serotonin receptor agonist		HTR1D, HTR1B, HTR1A, HTR1F, HTR1E, HTR5A, HTR6, HTR7	Serotonin receptor agonist
1464	78.01	oe	ccsbBroad304_01903	HIST2H2BE	Histones / Replication-dependent			
1465	77.99	cp	BRD-K08703257	3-amino-benzamide	PARP inhibitor		PARP1	PARP inhibitor
1466	77.98	oe	ccsbBroad304_10846	GGT1	CD molecules			
1467	77.96	cp	BRD-K09635314	M-3M3FBS	phospholipase activator		PLCB2, PLCB3, PLCD1, PLCG1, PLCG2	phospholipase activator
1468	77.95	oe	ccsbBroad304_03118	NRBP1	NRBP family			
1469	77.93	kd	CGS001-11164	NUDT5	Nudix motif containing			
1470	77.88	kd	CGS001-2565	GABRG1	GABA receptors			
1471	77.86	cp	BRD-K76205745	losartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
1472	77.85	cp	BRD-A75478957	PD-166793	Metalloproteinase inhibitor		MMP13, MMP2, MMP3	Metalloproteinase inhibitor, Collagenase inhibitor
1473	77.77	kd	CGS001-58492	ZNF77	Zinc fingers, C2H2-type			
1474	77.65	kd	CGS001-9697	TRAM2	-			
1475	77.63	oe	ccsbBroad304_10026	ZNF517	Zinc fingers, C2H2-type			
1476	77.61	kd	CGS001-55781	RIOK2	RIO2 subfamily			
1477	77.58	kd	CGS001-2664	GDI1	-			
1478	77.5	kd	CGS001-7319	UBE2A	Ubiquitin-conjugating enzymes E2			
1479	77.47	kd	CGS001-3300	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
1480	77.44	kd	CGS001-6608	SMO	GPCR / Class F : Frizzled receptors			
1481	77.43	kd	CGS001-3709	ITPR2	Ion channels / Inositol triphosphate receptors			
1482	77.4	kd	CGS001-9122	SLC16A4	SLC16 family of monocarboxylate transporters			
1483	77.35	oe	ccsbBroad304_09761	GPR156	GPCR / Class C : Orphans			
1484	77.31	cp	BRD-K71103788	duloxetine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, HTR2A, HTR2C, HTR6	Serotonin reuptake inhibitor, Norepinephrine reuptake inhibitor
1485	77.28	kd	CGS001-57684	ZBTB26	BTB/POZ domain containing			
1486	77.27	cc		Zinc fingers RanBP2 type LOF	-			
1487	77.14	kd	CGS001-63874	ABHD4	Abhydrolase domain containing			
1488	77.08	kd	CGS001-51014	TMED7	-			
1489	77.01	cp	BRD-A39390670	rabeprazole	ATPase inhibitor		ATP4A, CYP2C19	ATPase inhibitor, Gastrin inhibitor
1490	76.99	oe	ccsbBroad304_00652	GNAS	-			
1491	76.97	cp	BRD-K40887525	ritanserin	Serotonin receptor antagonist		HTR2A, HTR2C, HTR2B, ADRA1A, ADRA1B, ADRA1D, HTR1A, HTR1B, HTR1D, HTR5A, HTR6, HTR7	Serotonin receptor antagonist
1492	76.94	cc		BMP Signaling LOF	-			
1493	76.93	oe	ccsbBroad304_06185	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
1494	76.91	cp	BRD-A23290232	westcort	Glucocorticoid receptor agonist			Glucocorticoid receptor agonist
1495	76.9	oe	ccsbBroad304_07542	ABCF2	ATP binding cassette transporters / subfamily F			
1496	76.9	kd	CGS001-788	SLC25A20	Mitochondrial amino acid transporter subfamily			
1497	76.81	cp	BRD-K46862739	metyrapone	Cytochrome P450 inhibitor		CYP11B1, HSD11B1, NR3C2	Cytochrome P450 inhibitor
1498	76.79	oe	ccsbBroad304_07709	AFG3L2	ATPases / AAA-type			
1499	76.78	kd	CGS001-873	CBR1	Prostaglandin synthases			
1500	76.76	cp	BRD-K77625572	etomoxir	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT1B	Carnitine palmitoyltransferase inhibitor
1501	76.76	cp	BRD-K37516142	idebenone	Calcium channel modulator			Calcium channel modulator
1502	76.76	cp	BRD-K48735772	PD-158780	EGFR inhibitor		EGFR	EGFR inhibitor
1503	76.75	oe	ccsbBroad304_03980	DCLRE1B	-			
1504	76.68	oe	ccsbBroad304_06255	LRRC32	-			
1505	76.66	cp	BRD-K08252256	diclofenac	Cyclooxygenase inhibitor		PTGS1, PTGS2, AKR1C3, ALOX5, ASIC1, ASIC3, CYP2C8, KCNQ2, KCNQ3, PLA2G2A, PPARG, SCN4A	Cyclooxygenase inhibitor
1506	76.64	oe	ccsbBroad304_06830	RAB5A	RAB, member RAS oncogene			
1507	76.59	cp	BRD-A56675431	altizide	Thiazide diuretic			Thiazide diuretic
1508	76.58	kd	CGS001-822	CAPG	-			
1509	76.57	kd	CGS001-5927	KDM5A	Histone demethylases			
1510	76.55	kd	CGS001-9915	ARNT2	Basic helix-loop-helix proteins			
1511	76.52	oe	ccsbBroad304_07123	UQCRFS1	Mitochondrial respiratory chain complex / Complex III			
1512	76.48	cp	BRD-K90574421	ipsapirone	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1513	76.45	cp	BRD-A75517195	thiazolopyrimidine	CDC inhibitor			CDC inhibitor
1514	76.45	kd	CGS001-317701	VN1R2	GPCR / Unclassified : Vomeronasal receptors, type 1			
1515	76.43	kd	CGS001-115950	ZNF653	Zinc fingers, C2H2-type			
1516	76.38	oe	ccsbBroad304_06770	PRKAA1	AMPK subfamily			
1517	76.32	kd	CGS001-51466	EVL	-			
1518	76.31	kd	CGS001-1666	DECR1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1519	76.29	cp	BRD-K41859756	NVP-AUY922	HSP inhibitor		HSP90AA1, HSP90AA2, HSP90AB1	HSP inhibitor
1520	76.28	kd	CGS001-27148	STK36	Unc-51-like kinase (ULK) family			
1521	76.24	kd	CGS001-2583	B4GALNT1	Beta 4-glycosyltransferases			
1522	76.22	cp	BRD-A72596465	GW-6471	PPAR receptor antagonist		PPARA	PPAR receptor antagonist
1523	76.21	oe	ccsbBroad304_10230	STK19	G11 family			
1524	76.2	kd	CGS001-3202	HOXA5	Homeoboxes / ANTP class : HOXL subclass			
1525	76.18	cp	BRD-K74913225	brinzolamide	Carbonic anhydrase inhibitor		CA2, CA1, CA7, CA12, CA14, CA4, CA5A, CYP2B6, CYP2C8	Carbonic anhydrase inhibitor
1526	76.18	kd	CGS001-7057	THBS1	-			
1527	76.17	kd	CGS001-3665	IRF7	-			
1528	76.15	cp	BRD-K06467078	corynanthine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
1529	76.11	kd	CGS001-125919	ZNF543	Zinc fingers, C2H2-type			
1530	76.08	cp	BRD-K33453211	levocabastine	Histamine receptor antagonist		HRH1, NTSR2	Histamine receptor antagonist
1531	76.02	cp	BRD-K60038276	irbesartan	Angiotensin receptor antagonist		AGTR1, JUN, SLC10A1	Angiotensin receptor antagonist
1532	75.93	cp	BRD-K05181084	NGB-2904	Dopamine receptor antagonist		DRD3	Dopamine receptor antagonist
1533	75.9	cp	BRD-A43882281	pinacidil	ATP channel activator		ABCC9, KCNJ8	ATP channel activator, Potassium channel activator
1534	75.9	kd	CGS001-10943	MSL3	-			
1535	75.85	oe	ccsbBroad304_00737	UBE2K	Ubiquitin-conjugating enzymes E2			
1536	75.85	cp	BRD-K09186807	KIN001-244	Phosphoinositide dependent kinase inhibitor		PDPK1	Phosphoinositide dependent kinase inhibitor
1537	75.84	kd	CGS001-1759	DNM1	Pleckstrin homology (PH) domain containing			
1538	75.8	oe	ccsbBroad304_03266	ERGIC2	-			
1539	75.79	kd	CGS001-9958	USP15	Ubiquitin-specific peptidases			
1540	75.77	kd	CGS001-3776	KCNK2	Two-P potassium channels			
1541	75.7	cp	BRD-K36324071	NF-449	Purinergic receptor antagonist		P2RX1	Purinergic receptor antagonist
1542	75.69	kd	CGS001-613	BCR	Rho guanine nucleotide exchange factors			
1543	75.64	oe	ccsbBroad304_05838	APOC2	Apolipoproteins			
1544	75.63	kd	CGS001-8431	NR0B2	DAX-like receptors			
1545	75.62	cp	BRD-K73391359	quinisocaine	Local anesthetic			Local anesthetic
1546	75.61	cp	BRD-K32828673	chelidonine	Tubulin inhibitor			Tubulin inhibitor
1547	75.58	oe	ccsbBroad304_06183	EWSR1	RNA binding motif (RRM) containing			
1548	75.58	cp	BRD-K45479396	BP-554	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1549	75.49	cp	BRD-K06712146	YM-90709	IL5 inhibitor		CSF2RB, IL5RA	IL5 inhibitor
1550	75.48	kd	CGS001-7486	WRN	-			
1551	75.46	cp	BRD-K61737877	VEGF-receptor-2-kinase-inhibitor-IV	VEGFR inhibitor		KDR	VEGFR inhibitor
1552	75.3	kd	CGS001-4090	SMAD5	SMADs			
1553	75.29	oe	ccsbBroad304_07678	ZNF266	Zinc fingers, C2H2-type			
1554	75.25	kd	CGS001-6387	CXCL12	Endogenous ligands			
1555	75.24	cp	BRD-K74761218	WT-171	HDAC inhibitor		HDAC6	HDAC inhibitor
1556	75.17	kd	CGS001-10623	POLR3C	RNA polymerase subunits			
1557	75.12	oe	ccsbBroad304_03437	DDX49	DEAD-boxes			
1558	75.11	oe	ccsbBroad304_00447	DLD	-			
1559	74.99	oe	ccsbBroad304_08862	SMYD3	Chromatin-modifying enzymes / K-methyltransferases			
1560	74.89	cp	BRD-K73838513	cinacalcet	Calcium channel activator		CASR	Calcium channel activator
1561	74.84	cp	BRD-K61269089	daphnetin	Protein kinase inhibitor			Protein kinase inhibitor
1562	74.81	oe	ccsbBroad304_12106	PXK	Slob family			
1563	74.8	cp	BRD-K88611939	aniracetam	Glutamate receptor agonist		DRD2, GRIA1, GRIA2, GRIA3, HTR2A, GRIA4	Glutamate receptor agonist
1564	74.76	cp	BRD-A60197193	amisulpride	Dopamine receptor antagonist		DRD2, DRD3, HTR2A, HTR7	Dopamine receptor antagonist
1565	74.48	kd	CGS001-4170	MCL1	-			
1566	74.48	kd	CGS001-55107	ANO1	Calcium activated chloride channel			
1567	74.41	cp	BRD-M64432851	sunitinib	FLT3 inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RET tyrosine kinase inhibitor, VEGFR inhibitor
1568	74.4	oe	ccsbBroad304_02786	ZNF281	Zinc fingers, C2H2-type			
1569	74.39	cp	BRD-K20995441	U-54494A	Opioid receptor agonist			Opioid receptor agonist
1570	74.35	cp	BRD-A54236247	racephedrine	Adrenergic receptor agonist			Adrenergic receptor agonist
1571	74.34	cp	BRD-K40742111	baeomycesic-acid	Lipoxygenase inhibitor			Lipoxygenase inhibitor
1572	74.32	kd	CGS001-6775	STAT4	SH2 domain containing			
1573	74.3	kd	CGS001-5754	PTK7	Type VI RTKs: PTK7/CCK4			
1574	74.29	cp	BRD-K14693417	cinchonine	P-glycoprotein inhibitor		CYP2D6	P-glycoprotein inhibitor
1575	74.28	kd	CGS001-2828	GPR4	GPCR / Class A : Orphans			
1576	74.22	kd	CGS001-9761	MLEC	-			
1577	74.17	kd	CGS001-5134	PDCD2	Zinc fingers, MYND-type			
1578	74.04	cp	BRD-K06926592	tretinoin	Retinoid receptor agonist		RARG, RORB, ALDH1A1, ALDH1A2, GPRC5A, NR0B1, NR2C2, PPARD, RARA, RARB, RARRES1, RORC, RXRB, RXRG	Retinoid receptor agonist, Retinoid receptor ligand
1579	74.02	oe	ccsbBroad304_03072	GTPBP8	-			
1580	73.98	kd	CGS001-976	CD97	Adhesion Class GPCRs			
1581	73.97	cp	BRD-A98299281	velnacrine	cholinesterase inhibitor		ACHE	cholinesterase inhibitor
1582	73.91	kd	CGS001-23710	GABARAPL1	-			
1583	73.85	cp	BRD-K02590140	O-2050	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
1584	73.7	kd	CGS001-4704	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1585	73.66	kd	CGS001-813	CALU	EF-hand domain containing			
1586	73.64	kd	CGS001-639	PRDM1	Zinc fingers, C2H2-type			
1587	73.61	kd	CGS001-389114	ZNF662	Zinc fingers, C2H2-type			
1588	73.6	oe	ccsbBroad304_06235	G6PD	-			
1589	73.58	cp	BRD-A97104540	fenoterol	Adrenergic receptor agonist		ADRB2, ADRB1, ADRB3	Adrenergic receptor agonist
1590	73.57	oe	ccsbBroad304_01650	TCEA1	General transcription factors			
1591	73.57	cp	BRD-K68095457	palmitoylethanolamide	Cannabinoid receptor agonist		CNR2, GPR119, GPR55	Cannabinoid receptor agonist
1592	73.56	kd	CGS001-10644	IGF2BP2	RNA binding motif (RRM) containing			
1593	73.54	oe	ccsbBroad304_00757	HMGA1	High-mobility group / Canonical			
1594	73.53	oe	ccsbBroad304_05590	NOTCH2NL	-			
1595	73.42	cp	BRD-K53523901	arctigenin	MEK inhibitor		ADIPOR1, AHR, CHUK, MAP2K1	MEK inhibitor
1596	73.29	kd	CGS001-9131	AIFM1	-			
1597	73.21	kd	CGS001-11343	MGLL	Endocannabinoid turnover			
1598	73.14	cp	BRD-K70976396	cefoxitin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1599	73.04	oe	ccsbBroad304_02391	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
1600	73.03	oe	ccsbBroad304_06642	NIT1	-			
1601	73.01	oe	ccsbBroad304_00704	GSTZ1	Glutathione S-transferases / Soluble			
1602	72.98	kd	CGS001-10651	MTX2	-			
1603	72.9	kd	CGS001-8573	CASK	CASK family			
1604	72.88	cp	BRD-K67017579	cilostazol	Phosphodiesterase inhibitor		PDE3A, CYP2C19, CYP3A5, PDE3B	Phosphodiesterase inhibitor
1605	72.85	oe	ccsbBroad304_06711	PFAS	-			
1606	72.79	oe	ccsbBroad304_03405	CHRAC1	-			
1607	72.76	kd	CGS001-51109	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
1608	72.75	kd	CGS001-80762	NDFIP1	-			
1609	72.72	kd	CGS001-5468	PPARG	Peroxisome proliferator-activated receptors			
1610	72.64	cp	BRD-K87991767	umbelliferone	Cyclooxygenase inhibitor		CA9, CA12, PTGS2	Cyclooxygenase inhibitor
1611	72.59	oe	ccsbBroad304_05817	ANPEP	Aminopeptidase N			
1612	72.57	cp	BRD-K46317332	proadifen	Nitric oxide synthase inhibitor		NOS1	Nitric oxide synthase inhibitor
1613	72.54	oe	ccsbBroad304_05054	DTX3L	RING-type (C3HC4) zinc fingers			
1614	72.54	cp	BRD-K12513978	fenbufen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
1615	72.5	cp	BRD-A64228451	terreic-acid	BTK inhibitor		BTK	BTK inhibitor
1616	72.48	oe	ccsbBroad304_08289	PRKAG2	AMPK subfamily			
1617	72.45	cp	BRD-A13084692	troglitazone	Insulin sensitizer		PPARG, ACSL4, AKR1B1, CCL2, CYP3A4, ESRRA, ESRRG, INS, SERPINE1, SLC29A1, TRPM3	Insulin sensitizer, PPAR receptor agonist
1618	72.43	cp	BRD-K03670461	tyrphostin-AG-82	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
1619	72.41	kd	CGS001-222894	FERD3L	Basic helix-loop-helix proteins			
1620	72.4	kd	CGS001-7086	TKT	-			
1621	72.29	oe	ccsbBroad304_03923	LRRC4	Immunoglobulin superfamily / I-set domain containing			
1622	72.28	cp	BRD-K47983010	BX-795	IKK inhibitor		PDPK1, CDK2, CHEK1, GSK3B, IKBKE, KDR, PDK1, TBK1	IKK inhibitor
1623	72.28	cp	BRD-A17411484	carprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
1624	72.18	cp	BRD-K17294426	clebopride	Dopamine receptor antagonist		DRD2, ACHE	Dopamine receptor antagonist
1625	72.17	kd	CGS001-151636	DTX3L	RING-type (C3HC4) zinc fingers			
1626	72.09	kd	CGS001-4331	MNAT1	RING-type (C3HC4) zinc fingers			
1627	72.08	kd	CGS001-5243	ABCB1	ATP binding cassette transporters / subfamily B			
1628	71.95	kd	CGS001-22827	PUF60	RNA binding motif (RRM) containing			
1629	71.9	kd	CGS001-3660	IRF2	-			
1630	71.9	kd	CGS001-117154	DACH2	-			
1631	71.88	kd	CGS001-27430	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
1632	71.88	cp	BRD-K38436528	imipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM3, CHRM4, CHRM5, CYP2C19, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, KCND2, KCND3, KCNH1, KCNH2, SLC6A3	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
1633	71.68	oe	ccsbBroad304_00517	ESR1	Estrogen receptors			
1634	71.67	kd	CGS001-210	ALAD	-			
1635	71.66	kd	CGS001-121549	ASCL4	Basic helix-loop-helix proteins			
1636	71.57	kd	CGS001-10312	TCIRG1	ATPases / V-type			
1637	71.56	oe	ccsbBroad304_06687	SERPINB2	Serine (or cysteine) peptidase inhibitors			
1638	71.54	kd	CGS001-5578	PRKCA	Delta subfamily			
1639	71.45	cc		Aminoacyl tRNA synthetases class II LOF	-			
1640	71.44	cp	BRD-K38197229	bumetanide	Solute carrier family member inhibitor		SLC12A1, SLC12A2, CFTR, GPR35, SLC12A4, SLC12A5	Solute carrier family member inhibitor
1641	71.36	kd	CGS001-91433	RCCD1	-			
1642	71.18	oe	ccsbBroad304_07037	TCF12	Basic helix-loop-helix proteins			
1643	71.1	cp	BRD-K32744045	disulfiram	Aldehyde dehydrogenase inhibitor		ALDH2, ALDH1A2, ALDH5A1, ALDH7A1, CYP2E1, DBH, DNMT1, TRPA1	Aldehyde dehydrogenase inhibitor, TRPV agonist, DNA methyltransferase inhibitor
1644	70.99	kd	CGS001-7572	ZNF24	Zinc fingers, C2H2-type			
1645	70.93	cp	BRD-K70401845	erlotinib	EGFR inhibitor		EGFR, NR1I2	EGFR inhibitor
1646	70.9	kd	CGS001-875	CBS	Hydrogen sulphide synthesis			
1647	70.86	kd	CGS001-10109	ARPC2	Actin related protein 2/3 complex subunits			
1648	70.84	kd	CGS001-51021	MRPS16	Mitochondrial ribosomal proteins / small subunits			
1649	70.8	cp	BRD-K07888107	depudecin	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
1650	70.75	kd	CGS001-8780	RIOK3	RIO3 subfamily			
1651	70.7	cp	BRD-K34170797	fexaramine	FXR agonist		NR1H4	FXR agonist
1652	70.7	kd	CGS001-2153	F5	Blood coagulation components			
1653	70.69	kd	CGS001-27336	HTATSF1	RNA binding motif (RRM) containing			
1654	70.69	kd	CGS001-2264	FGFR4	Type V RTKs: FGF (fibroblast growth factor) receptor family			
1655	70.66	kd	CGS001-4734	NEDD4	-			
1656	70.6	oe	ccsbBroad304_02653	PRAF2	-			
1657	70.57	oe	ccsbBroad304_07260	LGR5	GPCR / Class A : Orphans			
1658	70.48	kd	CGS001-81848	SPRY4	-			
1659	70.4	cp	BRD-K53263234	CITCO	CAR agonist		NR1I3	CAR agonist
1660	70.4	kd	CGS001-4487	MSX1	Homeoboxes / ANTP class : NKL subclass			
1661	70.38	kd	CGS001-10013	HDAC6	Histone deacetylases			
1662	70.37	cp	BRD-K16444452	ibudilast	Leukotriene receptor antagonist		PDE4A, PDE4B, PDE4C, MIF, PDE10A, PDE3A, PDE4D, TLR4, CYSLTR1, IL1B, IL6, PDE11A, PDE5A	Leukotriene receptor antagonist, Phosphodiesterase inhibitor
1663	70.37	kd	CGS001-27095	TRAPPC3	Trafficking protein particle complex			
1664	70.29	cp	BRD-K35723520	darinaparsin	Apoptosis stimulant			Apoptosis stimulant
1665	70.29	kd	CGS001-27243	CHMP2A	Charged multivesicular body proteins			
1666	70.12	kd	CGS001-23242	COBL	-			
1667	70.08	oe	ccsbBroad304_06695	PCK2	-			
1668	70.01	cp	BRD-K35498378	alrestatin	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
1669	69.98	kd	CGS001-85366	MYLK2	Myosin Light Chain Kinase (MLCK) family			
1670	69.98	oe	ccsbBroad304_01779	WNT5A	Endogenous ligands			
1671	69.94	cc		Apolipoproteins LOF	-			
1672	69.89	cp	BRD-K01815685	indole	aryl hydrocarbon receptor agonist		AHR, IDO1	aryl hydrocarbon receptor agonist
1673	69.88	kd	CGS001-1120	CHKB	-			
1674	69.84	oe	ccsbBroad304_00861	IL13RA1	IL-2 receptor family			
1675	69.84	cp	BRD-A36066264	estradiol-benzoate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
1676	69.82	cp	BRD-A74500471	ethambutol	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1677	69.8	oe	ccsbBroad304_01257	PPOX	-			
1678	69.8	oe	ccsbBroad304_02243	DLGAP5	-			
1679	69.77	kd	CGS001-3376	IARS	Aminoacyl tRNA synthetases / Class I			
1680	69.74	cp	BRD-K84996949	sinensetin	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
1681	69.74	kd	CGS001-403	ARL3	ADP-ribosylation factors			
1682	69.67	cc		Sirtuins GOF	-			
1683	69.65	cp	BRD-K07325606	hispidin	PKC inhibitor		PREP, PRKCB, PTGS2, XDH	PKC inhibitor
1684	69.64	oe	ccsbBroad304_01137	P2RY6	GPCR / Class A : Purinergic receptors, P2Y			
1685	69.61	kd	CGS001-10447	FAM3C	-			
1686	69.58	oe	ccsbBroad304_06278	GK	Glycerol kinases			
1687	69.55	kd	CGS001-1030	CDKN2B	-			
1688	69.55	kd	CGS001-1009	CDH11	Cadherins / Major cadherins			
1689	69.48	cp	BRD-K42679050	Y-27152	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
1690	69.44	kd	CGS001-9200	PTPLA	-			
1691	69.39	cp	BRD-K51730347	diphencyprone	Immunostimulant			Immunostimulant
1692	69.33	kd	CGS001-10887	PROKR1	GPCR / Class A : Prokineticin receptors			
1693	69.27	cp	BRD-K64835161	BRD-K64835161	-666		CLK1, CLK4, DYRK1B	-666
1694	69.22	kd	CGS001-9961	MVP	-			
1695	69.16	cp	BRD-K26134695	calpeptin	Calpain inhibitor			Calpain inhibitor
1696	69.15	kd	CGS001-116931	MED12L	-			
1697	69.1	oe	ccsbBroad304_07945	GCA	EF-hand domain containing			
1698	69.1	kd	CGS001-139135	PASD1	-			
1699	69.09	oe	ccsbBroad304_06274	GJA1	Ion channels / Gap junction proteins (connexins)			
1700	69.08	oe	ccsbBroad304_04055	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
1701	69.08	oe	ccsbBroad304_05980	CDKN1B	-			
1702	68.96	kd	CGS001-79891	ZNF671	Zinc fingers, C2H2-type			
1703	68.92	cp	BRD-A44133049	azasetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
1704	68.89	oe	ccsbBroad304_09345	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
1705	68.89	oe	ccsbBroad304_00048	ALDH1A1	Aldehyde dehydrogenases			
1706	68.82	kd	CGS001-695	BTK	Pleckstrin homology (PH) domain containing			
1707	68.8	kd	CGS001-10783	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
1708	68.75	oe	ccsbBroad304_05098	MAGEB6	-			
1709	68.75	cp	BRD-K59273480	propentofylline	Adenosine reuptake inhibitor		ACHE	Adenosine reuptake inhibitor, Phosphodiesterase inhibitor
1710	68.74	kd	CGS001-23300	ATMIN	Zinc fingers, C2H2-type			
1711	68.65	oe	ccsbBroad304_13810	AHCY	Adenosine turnover			
1712	68.32	cp	BRD-K59419204	AM-281	Cannabinoid receptor antagonist		CNR1, CNR2, GPR55	Cannabinoid receptor antagonist
1713	68.27	cp	BRD-A96897502	U-74389F	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
1714	68.26	oe	ccsbBroad304_02604	B3GNT1	-			
1715	68.24	cp	BRD-K43880410	pregnenolone	glutamate receptor modulator		CYP17A1, PGR, SULT2B1	glutamate receptor modulator
1716	68.23	oe	ccsbBroad304_07827	STK38L	NDR family			
1717	68.2	cp	BRD-K12994359	valdecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CYP2C19	Cyclooxygenase inhibitor
1718	68.17	oe	ccsbBroad304_14011	PAPSS1	-			
1719	68.14	cp	BRD-K65910366	KUC103904N	-666			-666
1720	68.12	cp	BRD-K04010869	prostaglandin-a1	HSP inducer			HSP inducer, NFkB pathway inhibitor
1721	68.12	kd	CGS001-4193	MDM2	-			
1722	68.09	oe	ccsbBroad304_06521	LGALS3	Endogenous ligands			
1723	68.03	cp	BRD-K69840642	ISOX	HDAC inhibitor		HDAC6	HDAC inhibitor
1724	68.01	oe	ccsbBroad304_01471	S100A1	EF-hand domain containing			
1725	67.96	kd	CGS001-2861	GPR37	GPCR / Class A : Orphans			
1726	67.93	cp	BRD-A24228527	ofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
1727	67.86	cp	BRD-K15164005	apoptosis-activator-II	Carboxylesterase inhibitor		BCHE, CES1	Carboxylesterase inhibitor
1728	67.79	kd	CGS001-5430	POLR2A	RNA polymerase subunits			
1729	67.77	oe	ccsbBroad304_08585	RIOK2	RIO2 subfamily			
1730	67.77	kd	CGS001-5495	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
1731	67.72	oe	ccsbBroad304_03113	DSE	-			
1732	67.72	kd	CGS001-2184	FAH	-			
1733	67.68	cp	BRD-A77299732	salubrinal	Eukaryotic translation initiation factor inhibitor		EIF2S1, SLC6A9	Eukaryotic translation initiation factor inhibitor
1734	67.68	cp	BRD-K67847053	guanabenz	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C	Adrenergic receptor agonist
1735	67.67	kd	CGS001-5331	PLCB3	Phosphoinositide-specific phospholipase C			
1736	67.62	kd	CGS001-7407	VARS	Aminoacyl tRNA synthetases / Class I			
1737	67.53	cp	BRD-A56987319	SQ-22536	Adenylyl cyclase inhibitor		ADCY1, ADCY5	Adenylyl cyclase inhibitor
1738	67.53	kd	CGS001-7748	ZNF195	Zinc fingers, C2H2-type			
1739	67.47	oe	ccsbBroad304_01659	TERF1	-			
1740	67.47	kd	CGS001-672	BRCA1	Fanconi anemia, complementation groups			
1741	67.43	oe	ccsbBroad304_00033	ADSS	-			
1742	67.28	cp	BRD-K02637541	celecoxib	Cyclooxygenase inhibitor		PTGS2, CA12, CASP3, CYP2C19, PDPK1	Cyclooxygenase inhibitor
1743	67.22	kd	CGS001-84823	LMNB2	Intermediate filaments type V, lamins			
1744	67.17	kd	CGS001-128	ADH5	Alcohol dehydrogenases			
1745	67.14	cp	BRD-K35458079	edaravone	Nootropic agent		BCL2	Nootropic agent
1746	67.1	oe	ccsbBroad304_06237	GAA	Glycosidases			
1747	67.08	kd	CGS001-222545	GPRC6A	GPCR / Class C : Calcium-sensing receptors			
1748	67.06	cp	BRD-M45964048	verteporfin	Photosensitizing agent			Photosensitizing agent
1749	67.03	oe	ccsbBroad304_00966	MAFG	-			
1750	67.03	oe	ccsbBroad304_05941	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
1751	66.97	kd	CGS001-11340	EXOSC8	-			
1752	66.94	kd	CGS001-7518	XRCC4	XRCC DNA Repair			
1753	66.89	oe	ccsbBroad304_01010	MGST2	Glutathione S-transferases / Microsomal			
1754	66.87	cp	BRD-K01493881	apigenin	Casein kinase inhibitor		AKR1B1, AR, CDK6, CFTR, CYP19A1, CYP1A2, CYP1B1, HSD17B1, MAOA, ODC1, XDH	Casein kinase inhibitor, Cell proliferation inhibitor, Cytochrome P450 inhibitor
1755	66.83	oe	ccsbBroad304_02041	SLC5A6	Sodium iodide symporter, sodium-dependent multivitamin transporter and sodium-coupled monocarboxylate transporters			
1756	66.8	oe	ccsbBroad304_05942	CBS	Hydrogen sulphide synthesis			
1757	66.71	oe	ccsbBroad304_01531	SHC1	SH2 domain containing			
1758	66.69	cp	BRD-K38449220	seneciphylline	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
1759	66.67	kd	CGS001-10206	TRIM13	RING-type (C3HC4) zinc fingers			
1760	66.66	oe	ccsbBroad304_00677	GPR34	GPCR / Class A : Orphans			
1761	66.64	kd	CGS001-23046	KIF21B	Kinesins			
1762	66.62	kd	CGS001-7879	RAB7A	RAB, member RAS oncogene			
1763	66.55	oe	ccsbBroad304_07641	CCT7	Heat Shock Proteins / Chaperonins			
1764	66.44	cp	BRD-A55393291	testosterone	Androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	Androgen receptor agonist
1765	66.42	cc		Wnt family GOF	-			
1766	66.39	cp	BRD-K93188295	ARC-239	Adrenergic receptor antagonist		ADRA2B, ADRA2A, ADRA2C	Adrenergic receptor antagonist
1767	66.39	kd	CGS001-5891	MOK	RCK family			
1768	66.35	cp	BRD-A93424738	dexamethasone	Glucocorticoid receptor agonist		ANXA1, CYP3A4, CYP3A5, NOS2, NR0B1, NR3C1, NR3C2	Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Glucocorticoid receptor modulator, Corticosteroid agonist
1769	66.29	cp	BRD-A64977602	mirtazapine	Adrenergic receptor antagonist		ADRA2A, HTR2A, HTR2C, ADRA2C, HTR3A, ADRA1A, ADRA1B, ADRA1D, ADRA2B, ADRB1, ADRB2, DRD1, DRD2, DRD3, DRD5, HRH1, HRH3, HTR2B, HTR7, OPRK1, SLC6A2, SLC6A3, SLC6A4	Adrenergic receptor antagonist, Serotonin receptor antagonist
1770	66.24	cp	BRD-K81729199	AQ-RA741	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
1771	66.12	kd	CGS001-53347	UBASH3A	-			
1772	66.12	kd	CGS001-84930	MASTL	MAST family			
1773	66.06	kd	CGS001-11333	PDAP1	-			
1774	65.97	kd	CGS001-4794	NFKBIE	Ankyrin repeat domain containing			
1775	65.92	cp	BRD-K91336023	mesulergine	Dopamine receptor agonist		HTR2A, HTR2C, HTR7, HTR2B, HTR3A, HTR3B, HTR6	Dopamine receptor agonist
1776	65.92	cp	BRD-A19053259	pseudopelletierine	Anthelmintic			Anthelmintic
1777	65.91	kd	CGS001-5707	PSMD1	Proteasome subunits			
1778	65.88	cp	BRD-K89626439	sirolimus	MTOR inhibitor		MTOR, FKBP1A, CCR5, FGF2	MTOR inhibitor
1779	65.84	cp	BRD-K76723084	isotretinoin	Retinoid receptor agonist		CYP2B6, CYP2C19, CYP2C8, CYP3A5, CYP3A7, NR2C2, PPARD, RARA, RARB, RARG, RORB, RORC	Retinoid receptor agonist
1780	65.8	kd	CGS001-5612	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
1781	65.77	oe	ccsbBroad304_03450	TMED9	-			
1782	65.67	oe	ccsbBroad304_00290	CEBPG	basic leucine zipper proteins			
1783	65.66	kd	CGS001-1977	EIF4E	Translation Initiation Factor 4E			
1784	65.63	cp	BRD-K04414442	SB-222200	Tachykinin antagonist		TACR3	Tachykinin antagonist
1785	65.63	kd	CGS001-79109	MAPKAP1	-			
1786	65.63	oe	ccsbBroad304_02036	ARHGEF7	Rho guanine nucleotide exchange factors			
1787	65.62	kd	CGS001-9354	UBE4A	U-box domain containing			
1788	65.52	kd	CGS001-11179	ZNF277	-			
1789	65.51	kd	CGS001-5883	RAD9A	-			
1790	65.5	oe	ccsbBroad304_07080	TM7SF2	-			
1791	65.5	kd	CGS001-174	AFP	-			
1792	65.47	kd	CGS001-153830	RNF145	RING-type (C3HC4) zinc fingers			
1793	65.46	oe	ccsbBroad304_02554	TRAFD1	-			
1794	65.42	cp	BRD-K51751936	alfadolone	GABA receptor agonist			GABA receptor agonist
1795	65.42	kd	CGS001-8821	INPP4B	Inositol polyphosphate phosphatases			
1796	65.29	cp	BRD-A73605923	mocimycin	Protein synthesis inhibitor			Protein synthesis inhibitor
1797	65.27	oe	ccsbBroad304_01998	ABCC3	ATP binding cassette transporters / subfamily C			
1798	65.26	kd	CGS001-3669	ISG20	-			
1799	65.23	kd	CGS001-2073	ERCC5	-			
1800	65.22	kd	CGS001-6722	SRF	-			
1801	65.18	kd	CGS001-7988	ZNF212	Zinc fingers, C2H2-type			
1802	65.16	cp	BRD-A10355991	norketamine	Glutamate receptor antagonist		CYP2B6, CYP2C19, CYP3A5, GRIN1	Glutamate receptor antagonist
1803	65.06	kd	CGS001-23097	CDK19	Cyclin-dependent kinases, CDK8 subfamily			
1804	65.04	cp	BRD-K70511574	sunitinib	PLK inhibitor		FLT3, KDR, KIT, FLT4, FLT1, PDGFRA, PDGFRB, RET, CSF1R, FGFR1	PLK inhibitor
1805	65	cp	BRD-K41731458	triclosan	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor		DNMT1	Enoyl-[acyl-carrier-protein] reductase [NADH] inhibitor
1806	64.98	cp	BRD-K73589491	nizatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
1807	64.93	kd	CGS001-3320	HSP90AA1	Heat shock proteins / HSPC			
1808	64.85	oe	ccsbBroad304_12492	RBM15	RNA binding motif (RRM) containing			
1809	64.7	cp	BRD-K84663978	trequinsin	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, PDE5A, PTGIR	Phosphodiesterase inhibitor
1810	64.64	oe	ccsbBroad304_05936	CASP2	Caspases			
1811	64.59	cp	BRD-K67298865	SB-431542	TGF beta receptor inhibitor		TGFBR1, ACVR1C, ACVR1B	TGF beta receptor inhibitor
1812	64.57	kd	CGS001-3978	LIG1	-			
1813	64.53	oe	ccsbBroad304_02415	TUBB3	Tubulins			
1814	64.52	oe	ccsbBroad304_00462	DR1	-			
1815	64.46	cp	BRD-A51393488	noscapine	Bradykinin receptor antagonist		BDKRB2, SIGMAR1	Bradykinin receptor antagonist, Tubulin inhibitor
1816	64.37	cp	BRD-K32830106	guanfacine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, CYP3A5, HCN1, HCN2, HCN3, HCN4	Adrenergic receptor agonist
1817	64.35	oe	ccsbBroad304_01955	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
1818	64.31	oe	ccsbBroad304_07211	ZRSR2	RNA binding motif (RRM) containing			
1819	64.26	cp	BRD-A25576662	streptozotocin	DNA alkylating agent		SLC2A2	DNA alkylating agent
1820	64.1	oe	ccsbBroad304_01688	TNFRSF1A	Tumour necrosis factor (TNF) receptor family			
1821	64.05	kd	CGS001-51545	ZNF581	Zinc fingers, C2H2-type			
1822	63.98	kd	CGS001-7639	ZNF85	Zinc fingers, C2H2-type			
1823	63.96	cc		Potassium channel blocker	-			
1824	63.94	kd	CGS001-7389	UROD	-			
1825	63.88	cp	BRD-K83302049	protopine	Histamine receptor antagonist		ACHE, SLC6A2, SLC6A4	Histamine receptor antagonist
1826	63.86	oe	ccsbBroad304_04713	MAS1L	GPCR / Class A : Orphans			
1827	63.86	oe	ccsbBroad304_00147	BAG1	-			
1828	63.83	kd	CGS001-389421	LIN28B	-			
1829	63.76	kd	CGS001-5867	RAB4A	RAB, member RAS oncogene			
1830	63.74	cp	BRD-A49225603	alimemazine	Histamine receptor agonist		HRH1	Histamine receptor agonist
1831	63.71	kd	CGS001-54536	EXOC6	-			
1832	63.55	kd	CGS001-3690	ITGB3	Integrins			
1833	63.51	kd	CGS001-81620	CDT1	-			
1834	63.43	cp	BRD-K92446736	zatebradine	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
1835	63.41	oe	ccsbBroad304_01560	SNAPC1	-			
1836	63.38	kd	CGS001-3308	HSPA4	Heat shock proteins / HSP70			
1837	63.34	cp	BRD-K66093087	FGIN-1-43	Benzodiazepine receptor agonist		TSPO	Benzodiazepine receptor agonist
1838	63.19	cp	BRD-K79145749	dibenzepin	Norepinephrine reuptake inhibitor			Norepinephrine reuptake inhibitor
1839	63.14	cp	BRD-K80527266	triacsin-c	Adrenergic receptor antagonist		ACSL1	Adrenergic receptor antagonist
1840	63.08	cp	BRD-K29530284	amlexanox	Histamine receptor modulator		FGF1, IL3, S100A12, S100A13	Histamine receptor modulator
1841	63.07	oe	ccsbBroad304_05133	OXER1	GPCR / Class A : Leukotriene receptors			
1842	63.07	cp	BRD-A15010982	HU-211	Glutamate receptor antagonist		CNR1, CNR2, GLRA1, GLRA2, GLRA3, GPR55, GRIN1, NFKB1	Glutamate receptor antagonist
1843	63.05	cp	BRD-K84085265	CG-930	JNK inhibitor		MAPK8	JNK inhibitor
1844	62.96	oe	ccsbBroad304_06671	OPA1	-			
1845	62.95	oe	ccsbBroad304_06098	DHCR24	-			
1846	62.9	cp	BRD-K39621635	artemether	Antimalarial		ATP1A1, CYP2B6, CYP2C19, CYP3A5	Antimalarial
1847	62.86	oe	ccsbBroad304_00212	CAMLG	-			
1848	62.79	kd	CGS001-5591	PRKDC	Other PIKK family kinases			
1849	62.79	kd	CGS001-1386	ATF2	basic leucine zipper proteins			
1850	62.73	cc		EMSY complex LOF	-			
1851	62.72	kd	CGS001-3295	HSD17B4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
1852	62.55	kd	CGS001-283	ANG	Ribonucleases, RNase A			
1853	62.45	oe	ccsbBroad304_01880	LAGE3	-			
1854	62.37	oe	ccsbBroad304_03940	RFWD2	RING-type (C3HC4) zinc fingers			
1855	62.34	cp	BRD-A87606379	nadolol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRB3	Adrenergic receptor antagonist
1856	62.29	cp	BRD-A62057054	MDL-11939	Serotonin receptor antagonist		HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
1857	62.27	cp	BRD-K26241953	piceatannol	SYK inhibitor		ATP5A1, ATP5B, ATP5C1, IRF3, PTGS2, SIRT1, SYK, TYR	SYK inhibitor
1858	62.24	cp	BRD-K18742343	H-8	PKA inhibitor		PKIA, PRKACA	PKA inhibitor
1859	62.21	cp	BRD-K64881305	ispinesib	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
1860	62.2	kd	CGS001-84108	PCGF6	Polycomb group ring fingers			
1861	62.18	kd	CGS001-539	ATP5O	ATPases / F-type			
1862	62.1	kd	CGS001-23624	CBLC	RING-type (C3HC4) zinc fingers			
1863	62.02	cp	BRD-K01663662	diphenidol	Acetylcholine receptor agonist		CHRM1, CHRM3, CHRM4, CHRM2	Acetylcholine receptor agonist
1864	61.9	cp	BRD-A54596827	solifenacin	Acetylcholine receptor antagonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
1865	61.84	cp	BRD-K53318339	vinpocetine	Phosphodiesterase inhibitor		PDE1A, PDE1C, SCN10A	Phosphodiesterase inhibitor, Sodium channel blocker
1866	61.8	kd	CGS001-6285	S100B	EF-hand domain containing			
1867	61.76	oe	ccsbBroad304_07724	KDELR2	-			
1868	61.7	kd	CGS001-8625	RFXANK	Ankyrin repeat domain containing			
1869	61.65	kd	CGS001-161725	OTUD7A	OTU domain containing			
1870	61.58	kd	CGS001-134391	GPR151	GPCR / Class A : Orphans			
1871	61.55	oe	ccsbBroad304_07655	POLR3C	RNA polymerase subunits			
1872	61.55	kd	CGS001-230	ALDOC	-			
1873	61.52	kd	CGS001-5887	RAD23B	-			
1874	61.46	cp	BRD-K28453807	nitrocaramiphen	Cholinergic receptor antagonist			Cholinergic receptor antagonist
1875	61.43	cp	BRD-K03319035	maprotiline	Norepinephrine reuptake inhibitor		SLC6A2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR2A, HTR2C, HTR7	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
1876	61.42	kd	CGS001-8220	DGCR14	-			
1877	61.41	kd	CGS001-5202	PFDN2	-			
1878	61.38	kd	CGS001-59348	ZNF350	Zinc fingers, C2H2-type			
1879	61.29	cp	BRD-K88358234	xaliproden	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
1880	61.29	cp	BRD-K63945320	dihydrosamidin	Phospholipase inhibitor			Phospholipase inhibitor, Nitric oxide production inhibitor, Platelet activating factor receptor antagonist
1881	61.27	oe	ccsbBroad304_05832	AIRE	Zinc fingers, PHD-type			
1882	61.23	kd	CGS001-79733	E2F8	-			
1883	61.15	kd	CGS001-3161	HMMR	CD molecules			
1884	61.13	oe	ccsbBroad304_06236	XRCC6	XRCC DNA Repair			
1885	61.06	kd	CGS001-140465	MYL6B	EF-hand domain containing			
1886	61.05	cp	BRD-K39965020	doconexent	PPAR receptor agonist		FFAR1, PPARA, PTGS1, PTGS2	PPAR receptor agonist
1887	61.03	kd	CGS001-2961	GTF2E2	General transcription factors			
1888	60.98	cp	BRD-A33168282	sotalol	Adrenergic receptor antagonist		ADRB1, ADRB2, KCNH2	Adrenergic receptor antagonist
1889	60.88	kd	CGS001-353322	ANKRD37	Ankyrin repeat domain containing			
1890	60.84	cp	BRD-A71203467	l-stepholidine	Dopamine receptor antagonist		DRD2, DRD1	Dopamine receptor antagonist
1891	60.81	cp	BRD-K44899736	RO-16-6941	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
1892	60.8	cp	BRD-A16665823	butoconazole	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1893	60.8	cp	BRD-K63068307	ZSTK-474	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
1894	60.79	cp	BRD-K38251852	paxilline	Potassium channel blocker		ABCA1, KCNMA1, NR1H3	Potassium channel blocker
1895	60.78	cp	BRD-K41260949	valproic-acid	HDAC inhibitor		ABAT, HDAC1, SCN1A, SCN3A, ACADSB, ALDH5A1, HDAC2, HDAC9, OGDH, SCN10A, SCN11A, SCN1B, SCN2A, SCN2B, SCN3B, SCN4A, SCN4B, SCN5A, SCN7A, SCN8A, SCN9A	HDAC inhibitor
1896	60.69	kd	CGS001-3108	HLA-DMA	Immunoglobulin superfamily / C1-set domain containing			
1897	60.67	kd	CGS001-332	BIRC5	Inhibitors of apoptosis (IAP) protein family			
1898	60.65	oe	ccsbBroad304_06574	MDH2	-			
1899	60.64	kd	CGS001-5465	PPARA	Peroxisome proliferator-activated receptors			
1900	60.62	kd	CGS001-25913	POT1	-			
1901	60.53	oe	ccsbBroad304_10064	NDUFS7	Mitochondrial respiratory chain complex / Complex I			
1902	60.48	kd	CGS001-6714	SRC	Src family			
1903	60.41	kd	CGS001-57448	BIRC6	Inhibitors of apoptosis (IAP) protein family			
1904	60.32	cp	BRD-K10098805	rhapontin	Apoptosis stimulant			Apoptosis stimulant
1905	60.26	cp	BRD-K12932420	YM-976	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4C, PDE4D, TNF	Phosphodiesterase inhibitor
1906	60.18	oe	ccsbBroad304_00221	CASP3	Caspases			
1907	60.14	cp	BRD-A92630576	trimebutine	Opioid receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Opioid receptor agonist
1908	60.06	cc		RNA Polymerase Enzymes LOF	-			
1909	59.92	cp	BRD-K20338176	cefaclor	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
1910	59.86	oe	ccsbBroad304_07727	LIAS	-			
1911	59.85	cp	BRD-K94353609	fluocinolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist
1912	59.79	cp	BRD-K16554956	PTB1	AMPK activator		PTPN1	AMPK activator
1913	59.75	cp	BRD-K14681867	somatostatin	Somatostatin receptor agonist		SSTR1, SSTR2, SSTR3, SSTR4, SSTR5, GH1, GHR, OPRD1, OPRM1	Somatostatin receptor agonist
1914	59.7	oe	ccsbBroad304_04001	ZNF747	Zinc fingers, C2H2-type			
1915	59.69	kd	CGS001-3065	HDAC1	Histone deacetylases			
1916	59.6	cp	BRD-K18678457	ZD-7288	HCN channel blocker		HCN1, HCN2, HCN3, HCN4	HCN channel blocker
1917	59.57	kd	CGS001-148479	PHF13	Zinc fingers, PHD-type			
1918	59.57	kd	CGS001-53834	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
1919	59.47	kd	CGS001-344387	CDKL4	Cyclin-dependent kinases			
1920	59.43	kd	CGS001-399664	MEX3D	Mex-3 homologs			
1921	59.4	oe	ccsbBroad304_09054	EGFL8	-			
1922	59.4	cp	BRD-K76872913	benzanthrone	Aromatic hydrocarbon derivative			Aromatic hydrocarbon derivative
1923	59.39	cp	BRD-K40578143	GR-79236	Adenosine receptor agonist		ADORA1, ADORA2A	Adenosine receptor agonist
1924	59.38	kd	CGS001-5810	RAD1	-			
1925	59.16	cp	BRD-K69195780	NAN-190	Serotonin receptor agonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, HTR1F	Serotonin receptor agonist
1926	59.13	kd	CGS001-3663	IRF5	-			
1927	59.09	oe	ccsbBroad304_02154	COX5A	Mitochondrial respiratory chain complex			
1928	59.08	kd	CGS001-4942	OAT	-			
1929	59.06	cp	BRD-K20986251	lithocholic-acid	FXR antagonist		NR1I2, VDR, GPBAR1, MDM2, MDM4, NR1H4, PTPN1	FXR antagonist, MDM inhibitor, PXR ligand, Tyrosine phosphatase inhibitor, Vitamin D receptor agonist, Vitamin D receptor ligand
1930	58.84	kd	CGS001-9826	ARHGEF11	Rho guanine nucleotide exchange factors			
1931	58.83	cp	BRD-K30743633	TCPOBOP	CAR agonist		NR1I3	CAR agonist
1932	58.78	cp	BRD-K91290917	amodiaquine	Histamine receptor agonist		HNMT, CYP2C8	Histamine receptor agonist
1933	58.77	cc		NADH ubiquinone oxidoreductase supernumerary subunits LOF	-			
1934	58.67	kd	CGS001-115	ADCY9	Adenylyl cyclases			
1935	58.64	kd	CGS001-9601	PDIA4	Protein disulfide isomerases			
1936	58.56	kd	CGS001-4893	NRAS	RAS subfamily			
1937	58.54	oe	ccsbBroad304_00882	IRS1	Pleckstrin homology (PH) domain containing			
1938	58.53	kd	CGS001-10221	TRIB1	Trbl family			
1939	58.45	kd	CGS001-4775	NFATC3	Nuclear factor of activated T-cells			
1940	58.37	cp	BRD-K36153907	KU-C103885	Cystic fibrosis transmembrane conductance regulator inhibitor			Cystic fibrosis transmembrane conductance regulator inhibitor
1941	58.33	cp	BRD-A51829654	BRL-15572	Serotonin receptor antagonist		HTR1D, HTR1A, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR6	Serotonin receptor antagonist
1942	58.32	oe	ccsbBroad304_02321	ARL4C	ADP-ribosylation factors			
1943	58.31	oe	ccsbBroad304_02719	SWAP70	EF-hand domain containing			
1944	58.31	kd	CGS001-23291	FBXW11	F-boxes / WD-40 domains			
1945	58.28	oe	ccsbBroad304_03080	C16ORF80	-			
1946	58.21	cp	BRD-K22009844	phenprobamate	Muscle relaxant			Muscle relaxant
1947	58.19	oe	ccsbBroad304_07680	NEK6	NIMA (never in mitosis gene a)- related kinase (NEK) family			
1948	58.11	kd	CGS001-1385	CREB1	basic leucine zipper proteins			
1949	58.06	cp	BRD-K50866992	tropisetron	Serotonin receptor antagonist		HTR3A, GLRA1, GLRA2, GLRB, HTR4	Serotonin receptor antagonist
1950	58.06	cp	BRD-K94325918	kinetin-riboside	Apoptosis stimulant			Apoptosis stimulant
1951	58.06	kd	CGS001-5328	PLAU	Chymotrypsin			
1952	58.05	kd	CGS001-80025	PANK2	-			
1953	58.03	kd	CGS001-1950	EGF	-			
1954	58.01	cp	BRD-K88677950	PD-198306	MAP kinase inhibitor		MAP2K1, MAP2K2, MAPK1, MAPK3	MAP kinase inhibitor, MEK inhibitor
1955	57.96	kd	CGS001-571	BACH1	BTB/POZ domain containing			
1956	57.94	cp	BRD-K96144918	mead-acid	KPL-1 tumor suppressor			KPL-1 tumor suppressor
1957	57.93	kd	CGS001-10320	IKZF1	IKAROS zinc fingers			
1958	57.9	oe	ccsbBroad304_06008	AP2M1	-			
1959	57.83	kd	CGS001-4724	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
1960	57.74	kd	CGS001-10975	UQCR11	Mitochondrial respiratory chain complex / Complex III			
1961	57.68	kd	CGS001-10857	PGRMC1	-			
1962	57.63	kd	CGS001-9232	PTTG1	-			
1963	57.6	kd	CGS001-1493	CTLA4	CD molecules			
1964	57.57	oe	ccsbBroad304_03479	YTHDF1	-			
1965	57.49	oe	ccsbBroad304_08724	CYP20A1	Cytochrome P450s			
1966	57.46	oe	ccsbBroad304_00023	ADA	Adenosine turnover			
1967	57.44	cp	BRD-A13122391	triptolide	RNA polymerase inhibitor		CYP2C19, RELA	RNA polymerase inhibitor
1968	57.39	kd	CGS001-808	CALM3	EF-hand domain containing			
1969	57.37	cp	BRD-K26669427	WR-216174	PFMRK inhibitor			PFMRK inhibitor
1970	57.31	oe	ccsbBroad304_00552	FEN1	-			
1971	57.29	cp	BRD-K99946902	hexylresorcinol	Local anesthetic		TYR	Local anesthetic
1972	57.26	kd	CGS001-1997	ELF1	ETS Transcription Factors			
1973	57.24	kd	CGS001-169270	ZNF596	Zinc fingers, C2H2-type			
1974	57.23	cp	BRD-A39290993	cyproterone	Androgen receptor antagonist		AR, ADORA1, ESR1	Androgen receptor antagonist, Progesterone receptor agonist, Testosterone receptor antagonist
1975	57.15	cc		IMPDH inhibitor	-			
1976	57.09	cp	BRD-K40530731	hyoscyamine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
1977	57.08	cp	BRD-K36927236	glibenclamide	Sulfonylurea		KCNJ11, ABCC8, CFTR, KCNJ5, KCNJ8, ABCA1, ABCB11, ABCC9, CPT1A, KCNJ1, SLCO2B1, TRPA1	Sulfonylurea
1978	57.08	kd	CGS001-342357	ZKSCAN2	Zinc fingers, C2H2-type			
1979	57.06	cp	BRD-K43164539	cholic-acid	Bile acid		CES1, FECH, PLA2G1B, ADH1C, COX4I1, COX5A, COX5B, COX6A2, COX6B1, COX6C, COX7A1, COX7B, COX7C, COX8A, ESRRG, FABP6, GPBAR1, MT-CO1, MT-CO2, MT-CO3	Bile acid
1980	57.05	kd	CGS001-4255	MGMT	-			
1981	57.04	cp	BRD-K52512893	SC-19220	Prostanoid receptor antagonist		PTGER1	Prostanoid receptor antagonist
1982	56.93	kd	CGS001-9213	XPR1	-			
1983	56.9	kd	CGS001-2869	GRK5	GRK1/3 subfamily			
1984	56.89	oe	ccsbBroad304_06587	MMP1	Matrix metallopeptidase			
1985	56.87	cp	BRD-K91145395	prostratin	PKC activator		PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCH, PRKCQ	PKC activator
1986	56.84	kd	CGS001-10641	NPRL2	-			
1987	56.6	oe	ccsbBroad304_00986	MCM2	-			
1988	56.6	kd	CGS001-3046	HBE1	-			
1989	56.58	cp	BRD-K45068323	W-13	Calmodulin antagonist		CALM1, MYLK, PDE1A	Calmodulin antagonist
1990	56.5	kd	CGS001-5743	PTGS2	Cyclooxygenase			
1991	56.4	cp	BRD-A62035778	scopolamine	Acetylcholine receptor antagonist		CHRM2, CHRM1, CHRM3, CHRM4, CHRM5, SI	Acetylcholine receptor antagonist
1992	56.4	kd	CGS001-991	CDC20	WD repeat domain containing			
1993	56.3	kd	CGS001-7490	WT1	Zinc fingers, C2H2-type			
1994	56.28	cp	BRD-K92984783	melperone	Serotonin receptor antagonist		DRD2, HTR1A, HTR2A	Serotonin receptor antagonist, Dopamine receptor antagonist
1995	56.24	kd	CGS001-4817	NIT1	-			
1996	56.16	kd	CGS001-664	BNIP3	-			
1997	56.1	cp	BRD-K59574735	ubenimex	Leukotriene inhibitor		LTA4H, ANPEP, RNPEP	Leukotriene inhibitor
1998	56.07	kd	CGS001-51447	IP6K2	-			
1999	56.04	cp	BRD-K14282469	LY-165163	Serotonin receptor antagonist		HTR1A, HTR1D	Serotonin receptor antagonist
2000	56.04	kd	CGS001-10472	ZNF238	-			
2001	55.99	cp	BRD-K34776109	glimepiride	Insulin secretagogue		ABCC8, KCNJ11, KCNJ1	Insulin secretagogue
2002	55.98	oe	ccsbBroad304_00303	CHN1	Rho GTPase activating proteins			
2003	55.98	kd	CGS001-7690	ZNF131	BTB/POZ domain containing			
2004	55.91	oe	ccsbBroad304_00665	GOT1	-			
2005	55.91	cp	BRD-K18619710	digoxigenin	Steroid		ATP1A1	Steroid
2006	55.83	kd	CGS001-8480	RAE1	WD repeat domain containing			
2007	55.74	cp	BRD-A23359898	sibutramine	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, CYP2B6, CYP2C19, CYP3A5	Serotonin reuptake inhibitor
2008	55.73	oe	ccsbBroad304_06007	CISH	SH2 domain containing			
2009	55.7	cp	BRD-K15891719	tenofovir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, Cytochrome P450 inhibitor, DNA polymerase inhibitor, HIV integrase inhibitor
2010	55.68	oe	ccsbBroad304_07136	WNT9A	Wingless-type MMTV integration sites			
2011	55.62	kd	CGS001-5034	P4HB	Protein disulfide isomerases			
2012	55.54	kd	CGS001-64750	SMURF2	-			
2013	55.49	cp	BRD-K80325895	eicosadienoic-acid	-666			-666
2014	55.47	cp	BRD-K55127134	fluphenazine	Dopamine receptor antagonist		DRD2, DRD1, CALM1, CHRNA7, DRD5, HRH1, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
2015	55.45	kd	CGS001-10111	RAD50	-			
2016	55.43	cp	BRD-A82238138	budesonide	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7	Glucocorticoid receptor agonist
2017	55.42	cp	BRD-K50214219	CS-1657	PARP inhibitor		PARP1	PARP inhibitor
2018	55.41	oe	ccsbBroad304_00469	DUT	-			
2019	55.41	cp	BRD-K78959463	FPL-64176	Calcium channel activator		CACNA1C, CACNA1S	Calcium channel activator
2020	55.37	kd	CGS001-5997	RGS2	Endogenous ligands			
2021	55.37	kd	CGS001-8531	CSDA	-			
2022	55.35	cp	BRD-K23875128	RHO-kinase-inhibitor-III[rockout]	Rho associated kinase inhibitor		IMPDH2, ROCK1	Rho associated kinase inhibitor
2023	55.34	cp	BRD-A31227688	kynuramine	Aryl hydrocarbon receptor activator			Aryl hydrocarbon receptor activator
2024	55.26	kd	CGS001-2771	GNAI2	-			
2025	55.17	kd	CGS001-444	ASPH	-			
2026	55.1	cp	BRD-A98702003	carbenoxolone	11-beta-HSD1 inhibitor		HSD11B1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3	11-beta-HSD1 inhibitor
2027	55.08	kd	CGS001-5277	PIGA	Glycosyltransferase group 1 domain containing			
2028	55.04	oe	ccsbBroad304_03161	FOXP3	Forkhead boxes			
2029	55	oe	ccsbBroad304_04633	TP53RK	Bud32 family			
2030	54.97	cp	BRD-K07303502	arachidonyl-trifluoro-methane	Cytosolic phospholipase inhibitor		PLA2G4A	Cytosolic phospholipase inhibitor
2031	54.97	cp	BRD-K67080878	milrinone	Phosphodiesterase inhibitor		PDE3A, PDE2A, PDE3B, PDE5A	Phosphodiesterase inhibitor
2032	54.91	kd	CGS001-5261	PHKG2	Phosphorylase kinase (PHK) family			
2033	54.91	kd	CGS001-8553	BHLHE40	Basic helix-loop-helix proteins			
2034	54.84	oe	ccsbBroad304_08386	SMOX	-			
2035	54.82	cp	BRD-K23623876	decafluorobutane	Contrast agent		GRM5	Contrast agent
2036	54.82	kd	CGS001-5073	PARN	-			
2037	54.8	cp	BRD-A58955223	sulforaphane	Antineoplastic		NFE2L2	Antineoplastic, Aryl hydrocarbon receptor antagonist
2038	54.78	cp	BRD-A52282606	lacidipine	Calcium channel blocker		CACNA1C	Calcium channel blocker
2039	54.78	cp	BRD-K45330754	diethylstilbestrol	Estrogen receptor agonist		ESR1, ESR2, ESRRG, ESRRB	Estrogen receptor agonist
2040	54.74	kd	CGS001-163071	ZNF114	Zinc fingers, C2H2-type			
2041	54.73	oe	ccsbBroad304_01984	EIF3G	RNA binding motif (RRM) containing			
2042	54.73	cp	BRD-K43736954	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2043	54.57	oe	ccsbBroad304_04691	OSR2	Zinc fingers, C2H2-type			
2044	54.57	cp	BRD-K80725632	lavendustin-c	EGFR inhibitor		CAMK2A, EGFR, SRC	EGFR inhibitor
2045	54.47	cp	BRD-K22193694	dioxybenzone	Topical sunscreen agent			Topical sunscreen agent
2046	54.41	cp	BRD-K33864865	LY-225910	CCK receptor antagonist		CCKBR	CCK receptor antagonist
2047	54.37	cp	BRD-K21520694	sulfacetamide	PABA antagonist			PABA antagonist
2048	54.35	cp	BRD-K82357231	desloratadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2049	54.34	oe	ccsbBroad304_02738	RRS1	-			
2050	54.3	cp	BRD-A54487287	cortisone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
2051	54.27	kd	CGS001-3298	HSF2	-			
2052	54.26	oe	ccsbBroad304_03332	SIRT6	Histone deacetylases (HDACs)			
2053	54.25	cp	BRD-A11007541	BCI-hydrochloride	Protein phosphatase inhibitor		DUSP1, DUSP6	Protein phosphatase inhibitor
2054	54.25	kd	CGS001-169436	C9ORF96	-			
2055	54.21	kd	CGS001-8703	B4GALT3	Beta 4-glycosyltransferases			
2056	54.2	oe	ccsbBroad304_00941	LIG3	-			
2057	54.19	cp	BRD-K92015269	GBR-12783	Dopamine uptake inhibitor			Dopamine uptake inhibitor
2058	54.17	kd	CGS001-6513	SLC2A1	Solute carriers			
2059	54.09	kd	CGS001-1432	MAPK14	MAPK:p38 subfamily			
2060	54.06	cp	BRD-K85119730	tolbutamide	ATP channel blocker		ABCC8, CYP2B6, CYP2C19, CYP2C8, KCNJ1, KCNJ11, KCNJ8	ATP channel blocker
2061	53.98	oe	ccsbBroad304_06229	FUS	RNA binding motif (RRM) containing			
2062	53.93	kd	CGS001-644	BLVRA	-			
2063	53.87	oe	ccsbBroad304_03396	FGFRL1	Immunoglobulin superfamily / I-set domain containing			
2064	53.78	oe	ccsbBroad304_01593	SRP14	-			
2065	53.78	kd	CGS001-1906	EDN1	Endogenous ligands			
2066	53.71	cp	BRD-K31699485	DMEOB	glutamate receptor modulator			glutamate receptor modulator
2067	53.71	kd	CGS001-6829	SUPT5H	-			
2068	53.68	cp	BRD-K83144676	olmesartan	Angiotensin antagonist		AGTR1	Angiotensin antagonist
2069	53.64	cp	BRD-A25775766	securinine	GABA receptor antagonist		GABRA1	GABA receptor antagonist, TP53 activator
2070	53.63	cp	BRD-K90333595	phentolamine	Adrenergic receptor antagonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C	Adrenergic receptor antagonist
2071	53.58	kd	CGS001-1763	DNA2	-			
2072	53.54	kd	CGS001-891	CCNB1	-			
2073	53.49	kd	CGS001-650	BMP2	Bone morphogenetic proteins			
2074	53.47	cp	BRD-K04196797	oxcarbazepine	Sodium channel blocker		CYP2C19, CYP3A4, CYP3A5, SCN1A, SCN3A, SCN5A	Sodium channel blocker
2075	53.45	kd	CGS001-3551	IKBKB	IKK family			
2076	53.44	cp	BRD-K06234293	LY-364947	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor, p38 MAPK inhibitor
2077	53.34	oe	ccsbBroad304_07169	ZNF174	Zinc fingers, C2H2-type			
2078	53.32	kd	CGS001-191	AHCY	Adenosine turnover			
2079	53.24	cp	BRD-K54416256	methimazole	Antithyroid		TPO	Antithyroid
2080	53.2	kd	CGS001-8508	NIPSNAP1	-			
2081	53.13	kd	CGS001-4702	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
2082	53.03	cp	BRD-A04308630	genipin	Choleretic agent			Choleretic agent
2083	52.99	oe	ccsbBroad304_07656	TRIM16	Tripartite motif containing			
2084	52.99	kd	CGS001-81876	RAB1B	RAB, member RAS oncogene			
2085	52.97	kd	CGS001-10856	RUVBL2	ATPases / AAA-type			
2086	52.93	cp	BRD-A01295252	trans-7-hydroxy-pipat	Dopamine receptor ligand			Dopamine receptor ligand
2087	52.88	oe	ccsbBroad304_01341	PTPN4	Protein tyrosine phosphatases			
2088	52.76	oe	ccsbBroad304_00844	IL1R1	Interleukins and interleukin receptors			
2089	52.76	cp	BRD-A29644307	nomifensine	Dopamine uptake inhibitor		SLC6A2, SLC6A3, DRD2, MAOA, MAOB, MPO	Dopamine uptake inhibitor, Noradrenaline uptake inhibitor
2090	52.75	cp	BRD-K45861246	azaperone	Dopamine receptor antagonist		DRD2, DRD3	Dopamine receptor antagonist
2091	52.66	kd	CGS001-8463	TEAD2	-			
2092	52.5	kd	CGS001-2159	F10	Chymotrypsin			
2093	52.47	kd	CGS001-54733	SLC35F2	SLC35 family of nucleotide sugar transporters			
2094	52.46	cp	BRD-K77133231	PD-169316	p38 MAPK inhibitor		ALOX5	p38 MAPK inhibitor
2095	52.4	kd	CGS001-3304	HSPA1B	Heat shock proteins / HSP70			
2096	52.34	oe	ccsbBroad304_02136	COPS2	-			
2097	52.29	oe	ccsbBroad304_03848	METTL14	-			
2098	52.29	cp	BRD-A52172093	VU-0413807-2	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I	Calcium channel blocker
2099	52.23	kd	CGS001-51495	PTPLAD1	-			
2100	52.1	kd	CGS001-23142	DCUN1D4	-			
2101	52.07	cp	BRD-K86301799	dipyridamole	Phosphodiesterase inhibitor		ADA, PDE5A, PDE10A, PDE4A, PDE7B, PDE8A, PDE8B, SLC29A1	Phosphodiesterase inhibitor
2102	52.04	cp	BRD-K11905747	spectinomycin	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
2103	52.01	cp	BRD-K47278471	diphenhydramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
2104	51.92	kd	CGS001-7343	UBTF	-			
2105	51.89	kd	CGS001-8797	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
2106	51.84	oe	ccsbBroad304_08452	PIH1D1	-			
2107	51.73	kd	CGS001-6919	TCEA2	-			
2108	51.71	oe	ccsbBroad304_05253	GPR114	Adhesion Class GPCRs			
2109	51.7	cp	BRD-K66175015	afatinib	EGFR inhibitor		EGFR, ERBB2, ERBB4	EGFR inhibitor
2110	51.7	kd	CGS001-7018	TF	-			
2111	51.65	oe	ccsbBroad304_03746	CDC42SE1	-			
2112	51.6	kd	CGS001-5992	RFX4	-			
2113	51.59	oe	ccsbBroad304_01854	MLLT10	Zinc fingers, PHD-type			
2114	51.59	kd	CGS001-5293	PIK3CD	Phosphatidylinositol kinases			
2115	51.59	kd	CGS001-3670	ISL1	Homeoboxes / LIM class			
2116	51.56	kd	CGS001-23368	PPP1R13B	Ankyrin repeat domain containing			
2117	51.5	oe	ccsbBroad304_00593	NR5A2	Fushi tarazu F1-like receptors			
2118	51.41	oe	ccsbBroad304_07993	ZBTB20	BTB/POZ domain containing			
2119	51.41	oe	ccsbBroad304_10438	LGALS8	Lectins, galactoside-binding			
2120	51.41	oe	ccsbBroad304_03773	CIAPIN1	-			
2121	51.41	kd	CGS001-23463	ICMT	-			
2122	51.37	oe	ccsbBroad304_03119	C16ORF5	-			
2123	51.21	kd	CGS001-439	ASNA1	-			
2124	51.19	oe	ccsbBroad304_06451	IMPDH1	Oxidoreductases			
2125	51.18	oe	ccsbBroad304_06494	KLRC1	CD molecules			
2126	51.14	kd	CGS001-4302	MLLT6	Zinc fingers, PHD-type			
2127	51.11	oe	ccsbBroad304_00949	LRPAP1	-			
2128	51.06	oe	ccsbBroad304_06338	GTF2A2	General transcription factors			
2129	51.06	kd	CGS001-4947	OAZ2	-			
2130	50.99	oe	ccsbBroad304_09050	ZNF436	Zinc fingers, C2H2-type			
2131	50.99	kd	CGS001-6713	SQLE	Lanosterol biosynthesis pathway			
2132	50.95	kd	CGS001-3176	HNMT	-			
2133	50.94	oe	ccsbBroad304_02436	ZER1	ZYG11 cell cycle regulator family			
2134	50.85	cp	BRD-K50387473	XMD-892	MAP kinase inhibitor		MAPK7, DCLK2, LRRK2, PLK4, TNK1	MAP kinase inhibitor
2135	50.83	cp	BRD-A05186015	bupropion	Dopamine uptake inhibitor		SLC6A2, SLC6A3, CHRNA3, CYP2B6	Dopamine uptake inhibitor
2136	50.72	cp	BRD-A51410489	yohimbine	Adrenergic receptor antagonist		ADRA2A, ADRA2C, ADRA2B, HTR1A, HTR1B, HTR1D, HTR2B, DRD2, DRD3, HTR1E, HTR1F, HTR2A, HTR2C, HTR5A, HTR7, KCNJ1, KCNJ10, KCNJ11, KCNJ12, KCNJ14, KCNJ15, KCNJ8	Adrenergic receptor antagonist
2137	50.71	oe	ccsbBroad304_06597	MSX2	Homeoboxes / ANTP class : NKL subclass			
2138	50.68	kd	CGS001-26054	SENP6	Ulp1 endopeptidase			
2139	50.68	kd	CGS001-218	ALDH3A1	Aldehyde dehydrogenases			
2140	50.66	oe	ccsbBroad304_00231	CBFB	-			
2141	50.6	kd	CGS001-22926	ATF6	basic leucine zipper proteins			
2142	50.57	oe	ccsbBroad304_02292	BCL2L11	-			
2143	50.57	kd	CGS001-1756	DMD	-			
2144	50.56	kd	CGS001-1718	DHCR24	-			
2145	50.49	oe	ccsbBroad304_01787	YES1	Src family			
2146	50.49	oe	ccsbBroad304_04271	MXD3	Basic helix-loop-helix proteins			
2147	50.47	cp	BRD-A72758037	asiatic-acid	Apoptosis stimulant		PYGM	Apoptosis stimulant
2148	50.39	kd	CGS001-388585	HES5	Basic helix-loop-helix proteins			
2149	50.3	cp	BRD-K50325075	UCL-2077	Slow after hyperpolarization channel blocker			Slow after hyperpolarization channel blocker
2150	50.3	kd	CGS001-80818	ZNF436	Zinc fingers, C2H2-type			
2151	50.24	kd	CGS001-57804	POLD4	DNA polymerases			
2152	50.18	kd	CGS001-9967	THRAP3	-			
2153	50.16	kd	CGS001-2295	FOXF2	Forkhead boxes			
2154	50.14	oe	ccsbBroad304_01240	POLR2F	RNA polymerase subunits			
2155	50.06	kd	CGS001-8493	PPM1D	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
2156	50.05	cc		Cyclins LOF	-			
2157	49.93	cp	BRD-K03557653	sappanone-a	Tyrosinase inhibitor			Tyrosinase inhibitor, Melanin inhibitor
2158	49.91	oe	ccsbBroad304_01139	PA2G4	-			
2159	49.89	kd	CGS001-4683	NBN	-			
2160	49.78	oe	ccsbBroad304_06670	OGG1	-			
2161	49.78	kd	CGS001-10314	LANCL1	-			
2162	49.75	oe	ccsbBroad304_14081	PPP1R13B	Ankyrin repeat domain containing			
2163	49.68	cp	BRD-A04327189	synephrine	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
2164	49.66	kd	CGS001-7332	UBE2L3	Ubiquitin-conjugating enzymes E2			
2165	49.47	cp	BRD-K57546357	prunetin	Breast cancer resistance protein inhibitor		ABCG2, ALDH2	Breast cancer resistance protein inhibitor
2166	49.47	cp	BRD-K10705233	GW-405833	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
2167	49.44	cp	BRD-K94080537	diethyltoluamide	DEET activator of fly antenna ionotropic receptor IR40a			DEET activator of fly antenna ionotropic receptor IR40a
2168	49.44	kd	CGS001-9616	RNF7	RING-type (C3HC4) zinc fingers			
2169	49.44	kd	CGS001-64326	RFWD2	RING-type (C3HC4) zinc fingers			
2170	49.41	oe	ccsbBroad304_01563	SNCA	Parkinson disease			
2171	49.4	kd	CGS001-5682	PSMA1	Proteasome subunits			
2172	49.3	cp	BRD-K84987553	MDM2-inhibitor	MDM inhibitor		MDM2	MDM inhibitor
2173	49.25	cp	BRD-K76810206	nicergoline	Adrenergic receptor antagonist		ADRA1A	Adrenergic receptor antagonist
2174	49.23	kd	CGS001-29899	GPSM2	Tetratricopeptide (TTC) repeat domain containing			
2175	49.18	cp	BRD-K85383046	IAA-94	Chloride channel blocker			Chloride channel blocker
2176	49.17	kd	CGS001-26229	B3GAT3	Beta-1,3-glucuronyltransferases			
2177	49.16	kd	CGS001-1612	DAPK1	Death-associated kinase (DAPK) family			
2178	49.13	oe	ccsbBroad304_06722	SERPINB6	Serine (or cysteine) peptidase inhibitors			
2179	49.08	cp	BRD-A14574269	UB-165	Acetylcholine receptor agonist		CHRNA3, CHRNA4, CHRNB2	Acetylcholine receptor agonist
2180	49.08	kd	CGS001-727	C5	Endogenous ligands			
2181	49.07	cc		Bile acid	-			
2182	49	oe	ccsbBroad304_01546	SLC7A1	SLC7 family			
2183	49	kd	CGS001-23410	SIRT3	Histone deacetylases (HDACs)			
2184	48.99	kd	CGS001-4154	MBNL1	Zinc fingers, CCCH-type domain containing			
2185	48.94	cp	BRD-K83322645	L-693403	Sigma receptor agonist		DRD2, SIGMAR1	Sigma receptor agonist, Sigma receptor antagonist
2186	48.93	cp	BRD-K54704028	BAY-36-7620	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
2187	48.93	cp	BRD-A79672927	tropicamide	Acetylcholine receptor antagonist		CHRM3, CHRM4, CHRM1, CHRM2	Acetylcholine receptor antagonist
2188	48.84	kd	CGS001-27032	ATP2C1	Calcium-ATPases			
2189	48.81	oe	ccsbBroad304_08775	SQRDL	-			
2190	48.78	kd	CGS001-7466	WFS1	-			
2191	48.76	kd	CGS001-94103	ORMDL3	-			
2192	48.75	oe	ccsbBroad304_04991	ZNF785	Zinc fingers, C2H2-type			
2193	48.74	cp	BRD-A06390036	hydroquinidine	Antiarrhythmic			Antiarrhythmic
2194	48.69	oe	ccsbBroad304_03524	PLEKHJ1	Pleckstrin homology (PH) domain containing			
2195	48.66	cp	BRD-K00615600	AG-14361	PARP inhibitor		PARP1	PARP inhibitor
2196	48.64	kd	CGS001-3066	HDAC2	Histone deacetylases			
2197	48.6	kd	CGS001-7189	TRAF6	RING-type (C3HC4) zinc fingers			
2198	48.57	kd	CGS001-9833	MELK	MELK subfamily			
2199	48.46	cc		Norepinephrine reuptake inhibitor	-			
2200	48.36	kd	CGS001-10886	NPFFR2	GPCR / Class A : Neuropeptide receptors : FF/AF			
2201	48.3	oe	ccsbBroad304_02009	RAB11A	RAB, member RAS oncogene			
2202	48.27	oe	ccsbBroad304_03808	ERGIC1	-			
2203	48.25	oe	ccsbBroad304_00081	APOC3	Apolipoproteins			
2204	48.2	oe	ccsbBroad304_11796	ULK3	Unc-51-like kinase (ULK) family			
2205	48.16	kd	CGS001-1543	CYP1A1	Cytochrome P450s			
2206	48.12	oe	ccsbBroad304_08684	CXCR7	-			
2207	48.05	kd	CGS001-607	BCL9	-			
2208	48.02	oe	ccsbBroad304_00548	FDPS	Lanosterol biosynthesis pathway			
2209	47.98	kd	CGS001-10138	YAF2	-			
2210	47.94	cp	BRD-K82941592	rosuvastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
2211	47.92	oe	ccsbBroad304_09198	HOPX	Homeoboxes / PRD class			
2212	47.87	oe	ccsbBroad304_03839	ZBTB26	BTB/POZ domain containing			
2213	47.86	cp	BRD-K71534238	GW-9508	Free fatty acid receptor agonist		FFAR4, FFAR1	Free fatty acid receptor agonist, G protein-coupled receptor agonist
2214	47.83	kd	CGS001-8900	CCNA1	-			
2215	47.79	cp	BRD-K77925998	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
2216	47.79	cp	BRD-K94841585	emodic-acid	Laxative			Laxative
2217	47.78	kd	CGS001-253260	RICTOR	-			
2218	47.76	cc		G2 M Checkpoint LOF	-			
2219	47.67	cp	BRD-K59597909	phenothiazine	Dopamine receptor antagonist			Dopamine receptor antagonist
2220	47.67	cp	BRD-A80502530	cinobufagin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
2221	47.66	kd	CGS001-51465	UBE2J1	Ubiquitin-conjugating enzymes E2			
2222	47.63	kd	CGS001-1399	CRKL	SH2 domain containing			
2223	47.59	oe	ccsbBroad304_02271	LPGAT1	-			
2224	47.59	kd	CGS001-27297	CRCP	-			
2225	47.56	kd	CGS001-83551	TAAR8	GPCR / Class A : Trace amine associated receptors			
2226	47.51	kd	CGS001-5029	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
2227	47.47	cp	BRD-K18135438	chenodeoxycholic-acid	11-beta-HSD1 inhibitor		HSD11B1, NR1H4	11-beta-HSD1 inhibitor, FXR agonist
2228	47.47	kd	CGS001-51002	TPRKB	-			
2229	47.4	oe	ccsbBroad304_02201	CLOCK	Histone acetyltransferases			
2230	47.39	kd	CGS001-7172	TPMT	-			
2231	47.39	kd	CGS001-140735	DYNLL2	Cytoplasmic dyneins			
2232	47.38	cp	BRD-K32247306	primidone	GABA receptor antagonist		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2	GABA receptor antagonist
2233	47.37	cp	BRD-K61341215	vecuronium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
2234	47.33	kd	CGS001-10555	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
2235	47.28	kd	CGS001-2115	ETV1	ETS Transcription Factors			
2236	47.23	cp	BRD-K43236057	piceid	ICAM1 inhibitor		GAA, XDH	ICAM1 inhibitor
2237	47.2	oe	ccsbBroad304_03951	NARFL	-			
2238	47.12	kd	CGS001-9709	HERPUD1	-			
2239	47.08	kd	CGS001-8518	IKBKAP	Elongator acetyltransferase complex subunits			
2240	47.07	kd	CGS001-51001	MTERFD1	-			
2241	47.06	oe	ccsbBroad304_05612	GPR152	GPCR / Class A : Orphans			
2242	47.06	cp	BRD-A25004090	erastin	Ion channel antagonist		VDAC2	Ion channel antagonist
2243	47.06	cp	BRD-K11107424	tiotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
2244	46.96	kd	CGS001-7965	AIMP2	-			
2245	46.93	oe	ccsbBroad304_08239	HSD17B11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
2246	46.88	oe	ccsbBroad304_11738	BRD4	Bromodomain kinase (BRDK) family			
2247	46.82	oe	ccsbBroad304_00534	FABP1	Fatty acid-binding proteins			
2248	46.8	cp	BRD-K36638830	anabasine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2249	46.77	kd	CGS001-147949	ZNF583	Zinc fingers, C2H2-type			
2250	46.72	oe	ccsbBroad304_12008	NLK	nmo subfamily			
2251	46.71	kd	CGS001-7297	TYK2	Janus kinase (JakA) family			
2252	46.54	kd	CGS001-2958	GTF2A2	General transcription factors			
2253	46.51	kd	CGS001-3269	HRH1	Histamine receptors			
2254	46.44	cp	BRD-K27665173	D-64406	PDGFR receptor inhibitor		FLT3, PDGFRA, PDGFRB	PDGFR receptor inhibitor
2255	46.3	kd	CGS001-51720	UIMC1	-			
2256	46.29	oe	ccsbBroad304_07354	ASH2L	Zinc fingers, PHD-type			
2257	46.24	kd	CGS001-5387	PMS2P3	-			
2258	46.17	cp	BRD-K95921201	reserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1	Vesicular monoamine transporter inhibitor
2259	46.16	kd	CGS001-1028	CDKN1C	-			
2260	46.13	kd	CGS001-2138	EYA1	Protein tyrosine phosphatases / Asp-based PTPs			
2261	46.08	kd	CGS001-718	C3	Endogenous ligands			
2262	45.96	oe	ccsbBroad304_05008	ZNF558	Zinc fingers, C2H2-type			
2263	45.92	cp	BRD-A16754160	ampicillin	Bacterial cell wall synthesis inhibitor		SLC15A1	Bacterial cell wall synthesis inhibitor
2264	45.92	kd	CGS001-506	ATP5B	ATPases / F-type			
2265	45.8	kd	CGS001-8829	NRP1	CD molecules			
2266	45.76	oe	ccsbBroad304_07109	TUBB2A	Tubulins			
2267	45.75	cp	BRD-A66199457	asiaticoside	Antineoplastic			Antineoplastic
2268	45.71	cp	BRD-K16551401	PNU-22394	Serotonin receptor agonist		MAOA, MAOB	Serotonin receptor agonist
2269	45.65	kd	CGS001-8834	TMEM11	-			
2270	45.65	kd	CGS001-9404	LPXN	-			
2271	45.61	oe	ccsbBroad304_09592	CTCFL	Zinc fingers, C2H2-type			
2272	45.61	kd	CGS001-58495	OVOL2	Zinc fingers, C2H2-type			
2273	45.6	cp	BRD-A98431941	ephedrine	Adrenergic receptor agonist		ACHE, ADRA1A, ADRB2, SLC18A2, SLC6A2	Adrenergic receptor agonist
2274	45.6	kd	CGS001-353288	KRT26	Intermediate filaments type I, keratins (acidic)			
2275	45.52	kd	CGS001-7444	VRK2	Vaccina related kinase (VRK) family			
2276	45.43	kd	CGS001-4668	NAGA	-			
2277	45.4	oe	ccsbBroad304_07381	MAPKAPK2	MAPKAPK subfamily			
2278	45.4	oe	ccsbBroad304_00226	CAV1	-			
2279	45.39	oe	ccsbBroad304_08605	PBK	TOPK family			
2280	45.29	oe	ccsbBroad304_08307	ZC3HC1	Zinc fingers, C3HC-type			
2281	45.23	kd	CGS001-10939	AFG3L2	ATPases / AAA-type			
2282	45.2	kd	CGS001-2475	MTOR	FRAP subfamily			
2283	45.15	oe	ccsbBroad304_02548	PROKR1	GPCR / Class A : Prokineticin receptors			
2284	45.09	kd	CGS001-2954	GSTZ1	Glutathione S-transferases / Soluble			
2285	45.08	kd	CGS001-151112	ZSWIM2	Zinc fingers, SWIM-type			
2286	45.08	kd	CGS001-8985	PLOD3	-			
2287	45.05	oe	ccsbBroad304_06386	HNMT	-			
2288	44.98	cp	BRD-K64857848	XMD-885	Leucine rich repeat kinase inhibitor		LRRK2, MAPK7	Leucine rich repeat kinase inhibitor, MAP kinase inhibitor
2289	44.94	oe	ccsbBroad304_06748	POLE2	DNA polymerases			
2290	44.92	oe	ccsbBroad304_00211	CALU	EF-hand domain containing			
2291	44.9	oe	ccsbBroad304_08104	MED4	-			
2292	44.8	kd	CGS001-54472	TOLLIP	-			
2293	44.79	cp	BRD-M47937986	cefatrizine	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2294	44.73	kd	CGS001-55765	C1ORF106	-			
2295	44.71	cp	BRD-K48115423	2-(4-methoxybenzylthio)-6-methylpyrimidin-4-ol	Matrix metalloprotease inhibitor		MMP13	Matrix metalloprotease inhibitor
2296	44.68	kd	CGS001-353	APRT	-			
2297	44.57	oe	ccsbBroad304_03637	DOK4	Pleckstrin homology (PH) domain containing			
2298	44.5	kd	CGS001-344561	GPR148	GPCR / Class A : Orphans			
2299	44.4	cp	BRD-K54790157	trioxsalen	DNA synthesis inhibitor			DNA synthesis inhibitor
2300	44.35	kd	CGS001-3174	HNF4G	Hepatocyte nuclear factor-4 receptors			
2301	44.32	cp	BRD-A62182663	YK-4279	Apoptosis stimulant		DHX9, EWSR1, FLI1	Apoptosis stimulant, EWS-FLI1 inhibitor
2302	44.27	oe	ccsbBroad304_01952	MAPKAPK5	MAPKAPK subfamily			
2303	44.15	kd	CGS001-22794	CASC3	-			
2304	44.13	kd	CGS001-7703	PCGF2	Polycomb group ring fingers			
2305	44.09	oe	ccsbBroad304_04457	TOX2	-			
2306	44.04	cp	BRD-A28422058	L-689560	Glutamate receptor antagonist		GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D	Glutamate receptor antagonist
2307	44.04	kd	CGS001-5910	RAP1GDS1	Armadillo repeat containing			
2308	44.03	kd	CGS001-8208	CHAF1B	WD repeat domain containing			
2309	44	kd	CGS001-51422	PRKAG2	AMPK subfamily			
2310	43.87	cp	BRD-K94649603	taxifolin	Opioid receptor antagonist		APOB, APP, HMGCR	Opioid receptor antagonist
2311	43.87	cp	BRD-A01593789	chlormadinone	5-alpha reductase inhibitor		PGR	5-alpha reductase inhibitor, Progesterone receptor agonist
2312	43.81	oe	ccsbBroad304_00688	GRB2	SH2 domain containing			
2313	43.75	kd	CGS001-22949	PTGR1	-			
2314	43.72	cp	BRD-K24240364	GYKI-52466	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4	Glutamate receptor antagonist, Kainate receptor antagonist
2315	43.68	oe	ccsbBroad304_06168	EPHA3	Type XIII RTKs: Ephrin receptor family			
2316	43.67	kd	CGS001-7155	TOP2B	DNA Topoisomerases			
2317	43.6	oe	ccsbBroad304_00098	ARG1	Arginase			
2318	43.6	kd	CGS001-9575	CLOCK	Histone acetyltransferases			
2319	43.57	cp	BRD-K56700933	phenethyl-isothiocyanate	Antineoplastic		CYP2E1	Antineoplastic
2320	43.57	kd	CGS001-944	TNFSF8	CD molecules			
2321	43.5	cp	BRD-A97479839	piperidolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
2322	43.48	kd	CGS001-1513	CTSK	Cathepsins			
2323	43.45	oe	ccsbBroad304_05981	CDO1	-			
2324	43.35	cp	BRD-K02113016	olaparib	PARP inhibitor		PARP1, PARP2, PARP3	PARP inhibitor
2325	43.32	kd	CGS001-7124	TNF	Tumor necrosis factor (ligand) superfamily			
2326	43.28	oe	ccsbBroad304_00816	IDE	Pitrilysin			
2327	43.16	cp	BRD-A78942461	ICI-118551	Adrenergic receptor antagonist			Adrenergic receptor antagonist
2328	43.02	oe	ccsbBroad304_01064	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
2329	43.02	oe	ccsbBroad304_00054	ALDOC	-			
2330	43.02	kd	CGS001-57787	MARK4	MARK subfamily			
2331	42.98	oe	ccsbBroad304_02416	TUBB4B	-			
2332	42.98	kd	CGS001-55300	PI4K2B	Phosphatidylinositol kinases			
2333	42.97	oe	ccsbBroad304_01774	WARS	Aminoacyl tRNA synthetases / Class I			
2334	42.93	kd	CGS001-140690	CTCFL	Zinc fingers, C2H2-type			
2335	42.92	kd	CGS001-2768	GNA12	-			
2336	42.9	cp	BRD-A38913120	BH3I-1	BCL inhibitor		BCL2	BCL inhibitor
2337	42.84	oe	ccsbBroad304_02459	KAT5	Histone acetyltransferases (HATs)			
2338	42.84	kd	CGS001-5291	PIK3CB	Phosphatidylinositol kinases			
2339	42.82	cp	BRD-A24514565	warfarin	Vitamin K antagonist		VKORC1, CYP2C19, CYP2C8, CYP4F2	Vitamin K antagonist
2340	42.82	cp	BRD-K93080877	Ala-Ala-Phe-CMK	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
2341	42.82	cp	BRD-K00656370	6-aminochrysene	Transferase inhibitor			Transferase inhibitor
2342	42.8	kd	CGS001-1606	DGKA	EF-hand domain containing			
2343	42.79	kd	CGS001-4837	NNMT	-			
2344	42.77	kd	CGS001-8896	BUD31	-			
2345	42.68	cp	BRD-K10852020	tolcapone	Catechol O methyltransferase inhibitor		COMT, TTR	Catechol O methyltransferase inhibitor
2346	42.6	oe	ccsbBroad304_04191	NAA50	N(alpha)-acetyltransferase subunits			
2347	42.55	oe	ccsbBroad304_07280	LAMTOR3	-			
2348	42.54	cp	BRD-K47539947	tetradecylthioacetic-acid	Lipid peroxidase inhibitor			Lipid peroxidase inhibitor
2349	42.5	kd	CGS001-51022	GLRX2	-			
2350	42.48	kd	CGS001-3909	LAMA3	Laminins			
2351	42.45	oe	ccsbBroad304_03117	CERS2	Homeoboxes / CERS class			
2352	42.45	kd	CGS001-7052	TGM2	Transglutaminases			
2353	42.36	cp	BRD-A45499626	UBP-302	Glutamate receptor antagonist		GRIK1	Glutamate receptor antagonist
2354	42.33	kd	CGS001-55556	ENOSF1	-			
2355	42.31	oe	ccsbBroad304_05931	CAPG	-			
2356	42.29	kd	CGS001-7371	UCK2	-			
2357	42.24	cp	BRD-K99411983	lumicolchicine	Colchicine isomer, non-binder of microtubules			Colchicine isomer, non-binder of microtubules
2358	42.23	cp	BRD-A67981824	cefotaxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
2359	42.17	cp	BRD-K32821942	azathioprine	Dehydrogenase inhibitor		HPRT1, IMPDH1, PPAT	Dehydrogenase inhibitor
2360	42.14	kd	CGS001-1499	CTNNB1	Catenins			
2361	42.13	oe	ccsbBroad304_08840	KIF9	Kinesins			
2362	42.12	oe	ccsbBroad304_06727	PIK3CG	Phosphatidylinositol kinases			
2363	42.09	oe	ccsbBroad304_01340	PTPN2	Protein tyrosine phosphatases			
2364	42.05	oe	ccsbBroad304_03910	CCDC90A	-			
2365	41.98	kd	CGS001-29937	NENF	-			
2366	41.97	kd	CGS001-10558	SPTLC1	Serine palmitoyltransferase			
2367	41.96	oe	ccsbBroad304_00294	CETN3	EF-hand domain containing			
2368	41.95	kd	CGS001-11284	PNKP	-			
2369	41.94	kd	CGS001-2523	FUT1	Fucosyltransferases			
2370	41.82	oe	ccsbBroad304_01795	ZNF22	Zinc fingers, C2H2-type			
2371	41.82	kd	CGS001-10524	KAT5	Histone acetyltransferases (HATs)			
2372	41.81	oe	ccsbBroad304_09676	ZSWIM2	Zinc fingers, SWIM-type			
2373	41.81	oe	ccsbBroad304_06639	NFYB	-			
2374	41.81	cp	BRD-A62071884	siguazodan	Phosphodiesterase inhibitor		PDE3A	Phosphodiesterase inhibitor
2375	41.76	kd	CGS001-117608	ZNF354B	Zinc fingers, C2H2-type			
2376	41.75	oe	ccsbBroad304_08167	DNTTIP2	-			
2377	41.73	oe	ccsbBroad304_01141	PAFAH1B1	WD repeat domain containing			
2378	41.72	oe	ccsbBroad304_08266	PIPOX	-			
2379	41.68	kd	CGS001-2068	ERCC2	General transcription factor IIH complex subunits			
2380	41.65	oe	ccsbBroad304_06728	PIK3R1	Phosphatidylinositol kinases			
2381	41.65	cp	BRD-K31553034	zibotentan	Endothelin receptor antagonist		EDNRA	Endothelin receptor antagonist
2382	41.64	oe	ccsbBroad304_05123	ZNF791	Zinc fingers, C2H2-type			
2383	41.63	oe	ccsbBroad304_03903	ABHD4	Abhydrolase domain containing			
2384	41.59	oe	ccsbBroad304_05194	LIPH	-			
2385	41.56	kd	CGS001-9541	CIR1	-			
2386	41.54	cp	BRD-K67506692	tyrphostin-AG-126	ERK1 and ERK2 phosphorylation inhibitor			ERK1 and ERK2 phosphorylation inhibitor
2387	41.54	cp	BRD-A26384407	chlortalidone	Carbonic anhydrase inhibitor		CA7, CA1, CA12, CA14, CA4, SLC12A1	Carbonic anhydrase inhibitor
2388	41.48	oe	ccsbBroad304_00526	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
2389	41.46	cc		AHSP Pathway LOF	-			
2390	41.43	cp	BRD-K30867024	SB-216641	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2B, HTR2C	Serotonin receptor antagonist
2391	41.38	oe	ccsbBroad304_03573	BRF2	-			
2392	41.37	oe	ccsbBroad304_13830	FOXN3	Forkhead boxes			
2393	41.28	oe	ccsbBroad304_00705	GTF2A1	General transcription factors			
2394	41.23	oe	ccsbBroad304_01786	XRCC4	XRCC DNA Repair			
2395	41.21	oe	ccsbBroad304_08339	CMPK1	-			
2396	41.21	oe	ccsbBroad304_05756	ACAA1	-			
2397	41.16	oe	ccsbBroad304_06889	RPN2	-			
2398	41.09	cc		V type ATPases LOF	-			
2399	41.04	oe	ccsbBroad304_01611	STAT6	SH2 domain containing			
2400	41	kd	CGS001-57121	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
2401	40.99	kd	CGS001-54442	KCTD5	-			
2402	40.94	cp	BRD-A25143711	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
2403	40.94	kd	CGS001-7165	TPD52L2	-			
2404	40.83	oe	ccsbBroad304_08613	KLHL9	BTB/POZ domain containing			
2405	40.82	cp	BRD-A26845397	isamoltan	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
2406	40.73	cp	BRD-A59215453	lobelanidine	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist, Dopamine receptor modulator, Opioid receptor antagonist, Vesicular monoamine transporter ligand
2407	40.64	kd	CGS001-5058	PAK1	PAKA subfamily			
2408	40.63	oe	ccsbBroad304_12059	ING3	Zinc fingers, PHD-type			
2409	40.63	cp	BRD-K06221026	DUP-697	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
2410	40.58	cp	BRD-K33483813	actarit	Interleukin receptor agonist			Interleukin receptor agonist
2411	40.58	cp	BRD-K04170657	psoromic-acid	Ras GTPase inhibitor			Ras GTPase inhibitor
2412	40.54	cp	BRD-K96119599	leucodin	Melanin inhibitor			Melanin inhibitor
2413	40.49	kd	CGS001-9034	CCRL2	Chemokine receptors			
2414	40.48	cp	BRD-K13800121	parecoxib	Cyclooxygenase inhibitor		LTF, PTGS2	Cyclooxygenase inhibitor
2415	40.45	kd	CGS001-2353	FOS	basic leucine zipper proteins			
2416	40.38	kd	CGS001-3638	INSIG1	-			
2417	40.34	oe	ccsbBroad304_07671	SIX2	Homeoboxes / SINE class			
2418	40.34	kd	CGS001-9891	NUAK1	NuaK subfamily			
2419	40.3	oe	ccsbBroad304_03822	GATAD2B	GATA zinc finger domain containing			
2420	40.23	kd	CGS001-5986	RFNG	Beta 3-glycosyltransferases			
2421	40.2	kd	CGS001-399694	SHC4	SH2 domain containing			
2422	40.2	kd	CGS001-2805	GOT1	-			
2423	40.17	cp	BRD-K29458283	chlorambucil	DNA inhibitor			DNA inhibitor
2424	40.14	cp	BRD-K17796732	JWH-015	Cannabinoid receptor agonist		CNR2, GPR55	Cannabinoid receptor agonist
2425	40.13	cp	BRD-K18574842	nafcillin	Bacterial cell wall synthesis inhibitor		CYP3A4	Bacterial cell wall synthesis inhibitor
2426	40.09	cp	BRD-K46142322	RS-67333	Serotonin receptor partial agonist		HTR4	Serotonin receptor partial agonist
2427	40.05	cp	BRD-K74236984	UNC-0321	Histone lysine methyltransferase inhibitor		EHMT2	Histone lysine methyltransferase inhibitor
2428	40.02	kd	CGS001-975	CD81	CD molecules			
2429	39.98	cp	BRD-K76805682	SB-415286	Glycogen synthase kinase inhibitor		GSK3B, GSK3A, RPS6KB1	Glycogen synthase kinase inhibitor
2430	39.98	kd	CGS001-8317	CDC7	CDC7 family			
2431	39.97	kd	CGS001-4904	YBX1	-			
2432	39.94	oe	ccsbBroad304_02686	COPZ1	-			
2433	39.92	cp	BRD-K08619838	tremorine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
2434	39.91	cp	BRD-K62858456	lomerizine	Calcium channel blocker		ABCB1, CACNA1B, SCN5A	Calcium channel blocker
2435	39.85	kd	CGS001-5434	POLR2E	RNA polymerase subunits			
2436	39.84	oe	ccsbBroad304_06800	PSMB7	Proteasome subunits			
2437	39.81	cp	BRD-K82381502	acetylcholine	Acetylcholine receptor agonist		ACHE, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor agonist
2438	39.74	oe	ccsbBroad304_00328	CLK3	CDC-like kinases			
2439	39.68	oe	ccsbBroad304_02438	FAM3C	-			
2440	39.64	cp	BRD-K46766488	S-14506	Serotonin receptor agonist		HTR1A, DRD2, HTR2C	Serotonin receptor agonist
2441	39.64	cp	BRD-K33193182	methylnorlichexanthone	Aurora kinase inhibitor		AURKB, KDR, PIM1	Aurora kinase inhibitor, PIM inhibitor, VEGFR inhibitor
2442	39.59	kd	CGS001-10642	IGF2BP1	RNA binding motif (RRM) containing			
2443	39.54	oe	ccsbBroad304_04903	ZNF786	Zinc fingers, C2H2-type			
2444	39.54	cp	BRD-A10420615	cyclopiazonic-acid	ATPase inhibitor		ATP2A1	ATPase inhibitor
2445	39.54	kd	CGS001-868	CBLB	RING-type (C3HC4) zinc fingers			
2446	39.53	cp	BRD-K26015241	ODQ	Guanylyl cyclase inhibitor		GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase inhibitor
2447	39.5	oe	ccsbBroad304_02569	BTG3	-			
2448	39.5	cp	BRD-K00610438	altanserin	Serotonin receptor antagonist		HTR2A, HTR2C	Serotonin receptor antagonist
2449	39.42	kd	CGS001-80777	CYB5B	-			
2450	39.4	kd	CGS001-3148	HMGB2	High-mobility group / Canonical			
2451	39.39	kd	CGS001-23464	GCAT	-			
2452	39.39	cp	BRD-A05352148	ipratropium	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
2453	39.37	oe	ccsbBroad304_03129	ERO1L	-			
2454	39.34	kd	CGS001-10617	STAMBP	-			
2455	39.33	kd	CGS001-124535	HSF5	-			
2456	39.32	oe	ccsbBroad304_02349	MPHOSPH9	-			
2457	39.28	kd	CGS001-9221	NOLC1	-			
2458	39.27	oe	ccsbBroad304_03112	NENF	-			
2459	39.23	cp	BRD-K47659338	EMD-386088	Serotonin receptor agonist		HTR6	Serotonin receptor agonist
2460	39.22	cp	BRD-K37865504	LY-2183240	FAAH inhibitor		FAAH	FAAH inhibitor
2461	39.2	kd	CGS001-10058	ABCB6	ATP binding cassette transporters / subfamily B			
2462	39.18	oe	ccsbBroad304_08481	CEP55	-			
2463	39.16	oe	ccsbBroad304_08014	GBGT1	Glycosyltransferase family 6 domain containing			
2464	39.16	oe	ccsbBroad304_06820	PTS	-			
2465	39.14	kd	CGS001-3939	LDHA	-			
2466	39.14	kd	CGS001-32	ACACB	Carboxylases			
2467	39.11	cp	BRD-K41170226	deoxycholic-acid	G protein-coupled receptor agonist		GPBAR1, EFTUD1, FPR1	G protein-coupled receptor agonist, Biliverdin reductase A activator, Unidentified pharmacological activity
2468	39.06	kd	CGS001-79187	FSD1	Fibronectin type III domain containing			
2469	39.01	oe	ccsbBroad304_00422	DARS	Aminoacyl tRNA synthetases / Class II			
2470	39	kd	CGS001-11214	AKAP13	A-kinase anchor proteins			
2471	38.94	kd	CGS001-55082	ARGLU1	-			
2472	38.91	oe	ccsbBroad304_01355	PYGL	Glycogen phosphorylases			
2473	38.9	kd	CGS001-11007	CCDC85B	-			
2474	38.89	oe	ccsbBroad304_03861	ZNF77	Zinc fingers, C2H2-type			
2475	38.87	cp	BRD-A69636825	diltiazem	Calcium channel blocker		CACNA1C, CACNA1S, CACNA2D1, CACNG1, CYP3A5, CYP3A7, HTR3A, KCNA5	Calcium channel blocker
2476	38.86	kd	CGS001-1659	DHX8	DEAH-boxes			
2477	38.85	oe	ccsbBroad304_07851	FAM120A	-			
2478	38.83	cp	BRD-A43974499	reboxetine	Adrenergic receptor antagonist		SLC6A2	Adrenergic receptor antagonist
2479	38.81	kd	CGS001-3177	SLC29A2	SLC29 family			
2480	38.78	kd	CGS001-10135	NAMPT	-			
2481	38.71	oe	ccsbBroad304_09058	SLC25A32	Mitochondrial nucleotide transporter subfamily			
2482	38.65	kd	CGS001-2624	GATA2	GATA zinc finger domain containing			
2483	38.64	oe	ccsbBroad304_06090	DDOST	-			
2484	38.62	kd	CGS001-9917	FAM20B	-			
2485	38.59	cp	BRD-K05395900	nicotine	Acetylcholine receptor agonist		CHRNA10, CHRNA9, AOX1, CHAT, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNB2, CHRNB3, CHRNB4, CYP19A1, CYP2B6, TBXAS1, TRPA1	Acetylcholine receptor agonist
2486	38.57	kd	CGS001-478	ATP1A3	ATPases / P-type			
2487	38.55	oe	ccsbBroad304_04170	PANK2	-			
2488	38.52	oe	ccsbBroad304_00645	GCLM	-			
2489	38.5	oe	ccsbBroad304_01833	IL1R2	Immunoglobulin-like family of IL-1 receptors			
2490	38.44	oe	ccsbBroad304_02964	TIMM9	-			
2491	38.39	cc		Mitogen activated protein kinases LOF	-			
2492	38.38	kd	CGS001-7335	UBE2V1	Ubiquitin-conjugating enzymes E2			
2493	38.37	cc		IKK inhibitor	-			
2494	38.35	kd	CGS001-54957	TXNL4B	-			
2495	38.35	kd	CGS001-3579	CXCR2	Chemokine receptors			
2496	38.3	oe	ccsbBroad304_09821	TMEM154	-			
2497	38.29	kd	CGS001-2908	NR3C1	3-Ketosteroid receptors			
2498	38.29	kd	CGS001-4012	LNPEP	Aminopeptidase N			
2499	38.23	oe	ccsbBroad304_05528	TICAM2	-			
2500	38.23	cp	BRD-K51662849	ilomastat	Matrix metalloprotease inhibitor		ACAN, ADAM28, MMP1, MMP12, MMP13, MMP14, MMP2, MMP3, MMP8, MMP9	Matrix metalloprotease inhibitor
2501	38.22	oe	ccsbBroad304_07875	SPECC1L	-			
2502	38.22	cp	BRD-K13926615	vardenafil	Phosphodiesterase inhibitor		PDE5A, CYP2C19, CYP2C8, CYP3A5, PDE6G, PDE6H	Phosphodiesterase inhibitor
2503	38.2	oe	ccsbBroad304_01088	NFATC3	Nuclear factor of activated T-cells			
2504	38.19	oe	ccsbBroad304_04490	RSPH1	-			
2505	38.14	oe	ccsbBroad304_00597	FUT1	Fucosyltransferases			
2506	38.07	oe	ccsbBroad304_01701	TPI1	-			
2507	37.98	cp	BRD-K78599730	manumycin-a	Farnesyltransferase inhibitor		FNTA, IKBKB	Farnesyltransferase inhibitor, NFkB pathway inhibitor
2508	37.97	oe	ccsbBroad304_02601	RAB31	RAB, member RAS oncogene			
2509	37.95	kd	CGS001-4613	MYCN	Basic helix-loop-helix proteins			
2510	37.9	oe	ccsbBroad304_06708	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
2511	37.87	oe	ccsbBroad304_02392	PAK4	PAKB subfamily			
2512	37.82	cp	BRD-K96354014	nifedipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNA1F, CACNA1H, CACNB2, CALM1, CYP3A5, GLRA1, GLRA3, GLRB, KCNA1, KCNA5, NR1I2, TRPM3	Calcium channel blocker
2513	37.81	kd	CGS001-23509	POFUT1	Fucosyltransferases			
2514	37.79	oe	ccsbBroad304_07128	VHL	-			
2515	37.67	oe	ccsbBroad304_03089	PACSIN3	-			
2516	37.62	cc		Bacterial 30S ribosomal subunit inhibitor	-			
2517	37.62	kd	CGS001-80854	SETD7	Histone methyltransferases (HMTs)			
2518	37.58	kd	CGS001-5576	PRKAR2A	Protein kinase A			
2519	37.58	kd	CGS001-7025	NR2F1	COUP-TF-like receptors			
2520	37.58	cp	BRD-K67102207	phenylbutyrate	HDAC inhibitor		CYP3A5, HDAC1	HDAC inhibitor
2521	37.51	cc		Leucine rich repeat kinase inhibitor	-			
2522	37.48	cp	BRD-K32836707	CAY-10577	Casein kinase inhibitor			Casein kinase inhibitor
2523	37.38	cp	BRD-K92778217	mefenamic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1, KCNQ1, TRPM3	Cyclooxygenase inhibitor
2524	37.34	oe	ccsbBroad304_03623	ZNF692	Zinc fingers, C2H2-type			
2525	37.33	oe	ccsbBroad304_00112	ASNA1	-			
2526	37.31	kd	CGS001-182	JAG1	CD molecules			
2527	37.29	cp	BRD-A26095496	clobetasol	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
2528	37.26	oe	ccsbBroad304_03641	ASF1B	-			
2529	37.21	kd	CGS001-2729	GCLC	-			
2530	37.2	kd	CGS001-2886	GRB7	Pleckstrin homology (PH) domain containing			
2531	37.16	cp	BRD-K38003476	clocortolone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist, Steroid
2532	37.14	kd	CGS001-5050	PAFAH1B3	-			
2533	37.07	cp	BRD-K39944607	ochratoxin-a	Phenylalanyl tRNA synthetase inhibitor		SLC22A6	Phenylalanyl tRNA synthetase inhibitor
2534	36.98	kd	CGS001-3567	IL5	Interleukins and interleukin receptors			
2535	36.93	kd	CGS001-23435	TARDBP	RNA binding motif (RRM) containing			
2536	36.9	oe	ccsbBroad304_06350	HAL	-			
2537	36.88	oe	ccsbBroad304_00661	GNGT2	-			
2538	36.88	cp	BRD-U51951544	ZG-10	JNK inhibitor		MAPK8	JNK inhibitor
2539	36.87	kd	CGS001-843	CASP10	Caspases			
2540	36.86	oe	ccsbBroad304_01566	SNRPA	RNA binding motif (RRM) containing			
2541	36.86	kd	CGS001-55226	NAT10	-			
2542	36.78	kd	CGS001-3964	LGALS8	Lectins, galactoside-binding			
2543	36.76	kd	CGS001-64219	PJA1	RING-type (C3HC4) zinc fingers			
2544	36.74	kd	CGS001-833	CARS	Aminoacyl tRNA synthetases / Class I			
2545	36.72	kd	CGS001-1284	COL4A2	Collagens			
2546	36.7	kd	CGS001-1376	CPT2	-			
2547	36.69	oe	ccsbBroad304_07240	DYRK3	Dyrk2 subfamily			
2548	36.66	kd	CGS001-2956	MSH6	-			
2549	36.64	oe	ccsbBroad304_06068	CXADR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
2550	36.64	kd	CGS001-3775	KCNK1	Two-P potassium channels			
2551	36.61	oe	ccsbBroad304_00857	IL10	Interleukins and interleukin receptors			
2552	36.6	kd	CGS001-3827	KNG1	Endogenous ligands			
2553	36.56	cp	BRD-K53220666	trimetozine	Sedative			Sedative
2554	36.53	oe	ccsbBroad304_08322	UFM1	-			
2555	36.53	kd	CGS001-55038	CDCA4	-			
2556	36.51	oe	ccsbBroad304_02668	PNKP	-			
2557	36.48	kd	CGS001-7247	TSN	-			
2558	36.42	cp	BRD-A36318220	necrostatin-1	RIPK inhibitor		IDO1, KRR1, RIPK1	RIPK inhibitor
2559	36.42	kd	CGS001-677	ZFP36L1	RING-type (C3HC4) zinc fingers			
2560	36.4	oe	ccsbBroad304_08346	COQ3	-			
2561	36.38	oe	ccsbBroad304_01608	STAT2	SH2 domain containing			
2562	36.38	kd	CGS001-7485	WRB	-			
2563	36.34	oe	ccsbBroad304_00106	ARRB1	-			
2564	36.34	kd	CGS001-6621	SNAPC4	-			
2565	36.31	oe	ccsbBroad304_01294	PRKRIR	THAP (C2CH-type zinc finger) domain containing			
2566	36.3	cp	BRD-A19500257	geldanamycin	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
2567	36.29	oe	ccsbBroad304_03532	ANKZF1	Ankyrin repeat domain containing			
2568	36.25	cp	BRD-A41145729	methoprene-acid	Retinoid receptor agonist		NCOA2, NR1H3, RXRA, RXRB	Retinoid receptor agonist
2569	36.22	kd	CGS001-3912	LAMB1	Laminins			
2570	36.18	kd	CGS001-11015	KDELR3	-			
2571	36.15	cp	BRD-A29734509	disopyramide	Sodium channel blocker		SCN5A, CHRM1, CHRM2, CHRM3, KCND2, KCND3, KCNH2	Sodium channel blocker
2572	36.03	kd	CGS001-51172	NAGPA	-			
2573	36.02	kd	CGS001-4953	ODC1	Decarboxylases			
2574	36.01	kd	CGS001-10632	ATP5L	ATPases / F-type			
2575	36	cp	BRD-A47598013	citalopram	Serotonin reuptake inhibitor		SLC6A4, SLC6A2	Serotonin reuptake inhibitor
2576	35.95	cp	BRD-K55454768	TAS-301	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
2577	35.95	oe	ccsbBroad304_01198	PIGA	Glycosyltransferase group 1 domain containing			
2578	35.88	oe	ccsbBroad304_09954	PTRF	-			
2579	35.88	cp	BRD-K91315211	betahistine	Histamine receptor agonist		HRH3, HRH1	Histamine receptor agonist, Histamine receptor antagonist
2580	35.88	kd	CGS001-5371	PML	RING-type (C3HC4) zinc fingers			
2581	35.86	cp	BRD-K49669041	BX-912	Pyruvate dehydrogenase kinase inhibitor		PDPK1, AKT2, CDK2, CHEK1, GSK3B, KDR, PDK1	Pyruvate dehydrogenase kinase inhibitor
2582	35.83	oe	ccsbBroad304_01072	NDUFB6	Mitochondrial respiratory chain complex / Complex I			
2583	35.83	oe	ccsbBroad304_00036	AFP	-			
2584	35.83	cp	BRD-K14965640	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor
2585	35.79	oe	ccsbBroad304_10806	ERBB3	Type I RTKs: ErbB (epidermal growth factor) receptor family			
2586	35.74	oe	ccsbBroad304_02715	WDTC1	DDB1 and CUL4 associated factors			
2587	35.73	oe	ccsbBroad304_14008	MPZL1	Immunoglobulin superfamily / V-set domain containing			
2588	35.72	kd	CGS001-2335	FN1	Endogenous ligands			
2589	35.7	oe	ccsbBroad304_00459	DPYD	-			
2590	35.7	kd	CGS001-9	NAT1	-			
2591	35.69	kd	CGS001-2161	F12	Chymotrypsin			
2592	35.56	oe	ccsbBroad304_00280	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
2593	35.43	oe	ccsbBroad304_05313	NUDT14	Nudix motif containing			
2594	35.37	oe	ccsbBroad304_06992	SRC	Src family			
2595	35.36	oe	ccsbBroad304_05792	AGTR1	Angiotensin receptors			
2596	35.35	oe	ccsbBroad304_09590	ZFP28	Zinc fingers, C2H2-type			
2597	35.33	oe	ccsbBroad304_02266	RHOBTB1	BTB/POZ domain containing			
2598	35.31	kd	CGS001-64407	RGS18	Regulators of G-protein signaling			
2599	35.3	kd	CGS001-839	CASP6	Caspases			
2600	35.29	cp	BRD-U88459701	atorvastatin	HMGCR inhibitor		HMGCR, DPP4, AHR, CYP3A5, FASLG	HMGCR inhibitor
2601	35.26	oe	ccsbBroad304_10484	ZNF707	Zinc fingers, C2H2-type			
2602	35.25	kd	CGS001-10460	TACC3	-			
2603	35.19	oe	ccsbBroad304_01277	PRKAB2	AMPK subfamily			
2604	35.17	kd	CGS001-2717	GLA	-			
2605	35.16	oe	ccsbBroad304_02052	KYNU	-			
2606	35.14	cp	BRD-A16700644	isoxsuprine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
2607	35.11	oe	ccsbBroad304_04146	HDAC11	Histone deacetylases			
2608	35.1	cp	BRD-K70577657	H-9	PKA inhibitor		PRKACA	PKA inhibitor
2609	35.06	cc		Supressors of cytokine signaling GOF	-			
2610	35	kd	CGS001-54811	ZNF562	Zinc fingers, C2H2-type			
2611	34.94	oe	ccsbBroad304_00853	IL7R	IL-2 receptor family			
2612	34.92	kd	CGS001-7181	NR2C1	Testicular receptors			
2613	34.9	cp	BRD-K11163873	phenanthridone	PARP inhibitor		PARP1	PARP inhibitor
2614	34.9	cp	BRD-K47323024	methapyrilene	Histamine receptor antagonist			Histamine receptor antagonist
2615	34.89	cp	BRD-K14329163	BAY-K8644	Calcium channel activator		CACNA1C	Calcium channel activator, L-type calcium channel activator
2616	34.89	cp	BRD-K52459643	prostaglandin-e1	Prostanoid receptor agonist		PTGER1, PTGER2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGER4, PTGIR	Prostanoid receptor agonist
2617	34.87	kd	CGS001-10901	DHRS4	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2618	34.85	kd	CGS001-5889	RAD51C	Fanconi anemia, complementation groups			
2619	34.84	oe	ccsbBroad304_05758	ACADSB	-			
2620	34.76	kd	CGS001-11344	TWF2	Twinfilin subfamily			
2621	34.73	cp	BRD-K01638814	rilmenidine	Adrenergic receptor agonist		NISCH	Adrenergic receptor agonist, Imidazoline receptor agonist
2622	34.68	oe	ccsbBroad304_00702	GSTM1	Glutathione S-transferases / Soluble			
2623	34.63	cp	BRD-K90382497	GW-843682X	PLK inhibitor		PLK1, PLK3	PLK inhibitor
2624	34.59	oe	ccsbBroad304_02589	COPS5	-			
2625	34.58	kd	CGS001-2793	GNGT2	-			
2626	34.57	kd	CGS001-136259	KLF14	Kruppel-like transcription factors			
2627	34.52	kd	CGS001-771	CA12	Carbonic anhydrases			
2628	34.51	cp	BRD-K10670311	sulfasalazine	Antirheumatic		PTGS1, PTGS2, ACAT1, ALOX5, CHUK, IKBKB, PLA2G1B, PPARG, SLC46A1, SLC7A11, TBXAS1	Antirheumatic, NFkB pathway inhibitor
2629	34.51	kd	CGS001-65243	ZNF643	-			
2630	34.51	kd	CGS001-57407	NMRAL1	Short chain dehydrogenase/reductase superfamily / Atypical members			
2631	34.5	oe	ccsbBroad304_06623	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
2632	34.49	oe	ccsbBroad304_02884	POT1	-			
2633	34.49	cp	BRD-K16621777	enobosarm	Androgen receptor modulator		AR	Androgen receptor modulator
2634	34.44	kd	CGS001-6727	SRP14	-			
2635	34.42	kd	CGS001-3592	IL12A	Interleukins and interleukin receptors			
2636	34.39	kd	CGS001-2589	GALNT1	Glycosyltransferase family 2 domain containing			
2637	34.35	cp	BRD-K71926323	marbofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
2638	34.33	kd	CGS001-10810	WASF3	-			
2639	34.32	oe	ccsbBroad304_04294	ATG10	-			
2640	34.29	kd	CGS001-4758	NEU1	-			
2641	34.25	cc		Bacterial cell wall synthesis inhibitor	-			
2642	34.23	kd	CGS001-2762	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
2643	34.22	oe	ccsbBroad304_02145	VAMP3	Vesicle-associated membrane proteins			
2644	34.19	cp	BRD-K19111024	clofibric-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
2645	34.11	kd	CGS001-22955	SCMH1	Sterile alpha motif (SAM) domain containing			
2646	34.09	kd	CGS001-4615	MYD88	-			
2647	34.08	oe	ccsbBroad304_05213	ZNF449	Zinc fingers, C2H2-type			
2648	34.06	oe	ccsbBroad304_06797	PSMA5	Proteasome subunits			
2649	34.04	oe	ccsbBroad304_00937	LGALS2	Lectins, galactoside-binding			
2650	34.03	cp	BRD-A54880345	etomidate	GABA receptor modulator		GABRA1, ADRA2B, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	GABA receptor modulator
2651	34.03	kd	CGS001-129685	TAF8	-			
2652	33.98	kd	CGS001-8027	STAM	-			
2653	33.92	kd	CGS001-4927	NUP88	-			
2654	33.89	kd	CGS001-9670	IPO13	Importins			
2655	33.83	kd	CGS001-1738	DLD	-			
2656	33.8	oe	ccsbBroad304_07294	TNFSF10	CD molecules			
2657	33.8	kd	CGS001-9908	G3BP2	RNA binding motif (RRM) containing			
2658	33.74	kd	CGS001-8467	SMARCA5	-			
2659	33.7	oe	ccsbBroad304_06204	FDFT1	Lanosterol biosynthesis pathway			
2660	33.67	cp	BRD-K91623615	ABT-751	Tubulin inhibitor		TUBB	Tubulin inhibitor
2661	33.63	kd	CGS001-984	CDK11B	Cyclin-dependent kinases, PITSLRE subfamily			
2662	33.61	kd	CGS001-3221	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
2663	33.6	kd	CGS001-84890	ADO	-			
2664	33.56	kd	CGS001-328	APEX1	-			
2665	33.53	kd	CGS001-5932	RBBP8	-			
2666	33.51	cp	BRD-A36707673	hydroxycholesterol	LXR agonist		ABCA1, NR1H2, NR1H3	LXR agonist
2667	33.51	kd	CGS001-5033	P4HA1	-			
2668	33.49	oe	ccsbBroad304_04728	TWIST2	Basic helix-loop-helix proteins			
2669	33.49	kd	CGS001-1452	CSNK1A1	Casein kinase 1 (CK1) family			
2670	33.46	oe	ccsbBroad304_07252	DGKZ	-			
2671	33.45	cp	BRD-K64614248	salicin	Anti-inflammatory			Anti-inflammatory
2672	33.43	oe	ccsbBroad304_03512	ATG16L1	WD repeat domain containing			
2673	33.39	kd	CGS001-2568	GABRP	GABA receptors			
2674	33.38	oe	ccsbBroad304_00067	SLC25A4	Mitochondrial nucleotide transporter subfamily			
2675	33.38	kd	CGS001-10494	STK25	YSK subfamily			
2676	33.3	oe	ccsbBroad304_06535	LPL	-			
2677	33.29	kd	CGS001-8935	SKAP2	Pleckstrin homology (PH) domain containing			
2678	33.25	kd	CGS001-4700	NDUFA6	LYR motif containing			
2679	33.23	oe	ccsbBroad304_11055	PRKCH	Eta subfamily			
2680	33.23	oe	ccsbBroad304_07358	DNAJA3	Heat shock proteins / DNAJ (HSP40)			
2681	33.18	kd	CGS001-538	ATP7A	ATPases / P-type			
2682	33.17	oe	ccsbBroad304_06384	HMOX1	Haem oxygenase			
2683	33.15	cc		HSP inhibitor	-			
2684	33.14	kd	CGS001-9632	SEC24C	-			
2685	33.14	kd	CGS001-1453	CSNK1D	Casein kinase 1 (CK1) family			
2686	33.12	oe	ccsbBroad304_07088	TP53	-			
2687	33.11	oe	ccsbBroad304_01463	RPS27A	S ribosomal proteins			
2688	33.1	kd	CGS001-26520	TIMM9	-			
2689	33.06	kd	CGS001-23011	RAB21	RAB, member RAS oncogene			
2690	33	kd	CGS001-3490	IGFBP7	insulin-like growth factor (IGF) binding proteins			
2691	32.99	kd	CGS001-348	APOE	Apolipoproteins			
2692	32.98	cc		Sterol demethylase inhibitor	-			
2693	32.98	cp	BRD-K73978287	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist, Immunosuppressant, Corticosteroid agonist
2694	32.92	oe	ccsbBroad304_01105	PNP	-			
2695	32.9	oe	ccsbBroad304_06588	MMP2	Matrix metallopeptidase			
2696	32.8	kd	CGS001-26959	HBP1	-			
2697	32.79	oe	ccsbBroad304_07238	STK24	YSK subfamily			
2698	32.74	kd	CGS001-306	ANXA3	Annexins			
2699	32.73	oe	ccsbBroad304_10857	MKNK2	MKN subfamily			
2700	32.73	kd	CGS001-5036	PA2G4	-			
2701	32.72	kd	CGS001-115201	ATG4A	-			
2702	32.69	kd	CGS001-29105	C16ORF80	-			
2703	32.68	kd	CGS001-11098	PRSS23	Serine peptidases / Serine peptidases			
2704	32.66	kd	CGS001-23492	CBX7	-			
2705	32.64	oe	ccsbBroad304_00797	HSPA2	Heat shock proteins / HSP70			
2706	32.64	kd	CGS001-2521	FUS	RNA binding motif (RRM) containing			
2707	32.62	oe	ccsbBroad304_01391	RFC5	ATPases / AAA-type			
2708	32.6	kd	CGS001-4914	NTRK1	Type VII RTKs: Neurotrophin receptor/Trk family			
2709	32.6	kd	CGS001-211	ALAS1	-			
2710	32.57	oe	ccsbBroad304_00707	GTF2E2	General transcription factors			
2711	32.57	oe	ccsbBroad304_02012	FADD	-			
2712	32.55	kd	CGS001-126626	GABPB2	Ankyrin repeat domain containing			
2713	32.52	cp	BRD-U73238814	QL-XI-92	DDR1 inhibitor		DDR1	DDR1 inhibitor
2714	32.49	kd	CGS001-9637	FEZ2	-			
2715	32.46	oe	ccsbBroad304_03037	TMEM97	-			
2716	32.45	oe	ccsbBroad304_00165	BMI1	Polycomb group ring fingers			
2717	32.44	oe	ccsbBroad304_00125	FXYD2	Ion transport regulator			
2718	32.42	cp	BRD-K93918653	quizartinib	FLT3 inhibitor		FLT3, CSF1R, KIT, RET, PDGFRA, PDGFRB	FLT3 inhibitor
2719	32.4	kd	CGS001-6502	SKP2	F-boxes / Leucine-rich repeats			
2720	32.38	kd	CGS001-9443	MED7	-			
2721	32.36	kd	CGS001-23013	SPEN	RNA binding motif (RRM) containing			
2722	32.33	oe	ccsbBroad304_03461	ZNF562	Zinc fingers, C2H2-type			
2723	32.33	kd	CGS001-259	AMBP	Lipocalins			
2724	32.31	cp	BRD-K96862998	pirfenidone	TGF beta receptor inhibitor		TNF, FURIN, MAPK14, TNFRSF1A	TGF beta receptor inhibitor
2725	32.31	kd	CGS001-5906	RAP1A	-			
2726	32.29	kd	CGS001-1676	DFFA	-			
2727	32.24	kd	CGS001-340385	ZNF517	Zinc fingers, C2H2-type			
2728	32.21	oe	ccsbBroad304_06367	HK1	-			
2729	32.21	kd	CGS001-123803	NTAN1	-			
2730	32.2	kd	CGS001-2710	GK	Glycerol kinases			
2731	32.2	kd	CGS001-5603	MAPK13	MAPK:p38 subfamily			
2732	32.16	oe	ccsbBroad304_03847	GPR107	GPCR / Unclassified : 7TM orphan receptors			
2733	32.13	kd	CGS001-8870	IER3	-			
2734	32.04	oe	ccsbBroad304_07478	CCP110	-			
2735	32.03	oe	ccsbBroad304_07428	PSMF1	Proteasome (prosome, macropain) subunits			
2736	31.92	cp	BRD-K82143716	flucytosine	Antifungal		DNMT1	Antifungal
2737	31.9	oe	ccsbBroad304_07617	HMGN4	High-mobility group / Canonical			
2738	31.87	kd	CGS001-3113	HLA-DPA1	Immunoglobulin superfamily / C1-set domain containing			
2739	31.84	oe	ccsbBroad304_03850	TRIB3	Trbl family			
2740	31.83	oe	ccsbBroad304_03269	CD320	CD molecules			
2741	31.81	oe	ccsbBroad304_02354	TRIM13	RING-type (C3HC4) zinc fingers			
2742	31.8	oe	ccsbBroad304_09358	MAPK1IP1L	-			
2743	31.79	oe	ccsbBroad304_02772	ICMT	-			
2744	31.77	kd	CGS001-150280	HORMAD2	-			
2745	31.76	kd	CGS001-142	PARP1	Poly (ADP-ribose) polymerases			
2746	31.76	kd	CGS001-27197	GPR82	GPCR / Class A : Orphans			
2747	31.75	cp	BRD-K04111260	raclopride	Dopamine receptor antagonist		DRD2, DRD3, HTR1A	Dopamine receptor antagonist
2748	31.74	kd	CGS001-8438	RAD54L	-			
2749	31.69	oe	ccsbBroad304_07061	TGM2	Transglutaminases			
2750	31.68	kd	CGS001-51444	RNF138	RING-type (C3HC4) zinc fingers			
2751	31.66	oe	ccsbBroad304_07345	CCRL2	Chemokine receptors			
2752	31.64	kd	CGS001-4200	ME2	-			
2753	31.61	oe	ccsbBroad304_06186	F2R	Protease activated receptors			
2754	31.5	kd	CGS001-1840	DTX1	-			
2755	31.48	oe	ccsbBroad304_06392	HOXB7	Homeoboxes / ANTP class : HOXL subclass			
2756	31.44	cp	BRD-K35483542	alitretinoin	Retinoid receptor agonist		RARG, RARA, RARB, RXRA, RXRG, ABCA1, CYP2C8, CYP3A7, RXRB, VKORC1	Retinoid receptor agonist
2757	31.43	oe	ccsbBroad304_01318	PSMD2	Proteasome subunits			
2758	31.41	kd	CGS001-5898	RALA	-			
2759	31.37	kd	CGS001-92609	TIMM50	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
2760	31.37	kd	CGS001-9813	KIAA0494	-			
2761	31.32	oe	ccsbBroad304_08553	STAP2	-			
2762	31.31	kd	CGS001-23210	JMJD6	-			
2763	31.3	kd	CGS001-5253	PHF2	Histone demethylases			
2764	31.28	oe	ccsbBroad304_03565	ADI1	-			
2765	31.28	kd	CGS001-6117	RPA1	-			
2766	31.26	kd	CGS001-5532	PPP3CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
2767	31.23	cp	BRD-K39339537	epirizole	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
2768	31.16	kd	CGS001-54101	RIPK4	Receptor interacting protein kinase (RIPK) family			
2769	31.15	oe	ccsbBroad304_00150	BAX	-			
2770	31.13	oe	ccsbBroad304_02922	TES	-			
2771	31.12	oe	ccsbBroad304_05786	ADRB2	GPCR / Class A : Adrenoceptors : beta			
2772	31.12	cp	BRD-K52219182	BRD-K52219182	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
2773	31.12	kd	CGS001-213	ALB	-			
2774	31.09	oe	ccsbBroad304_07699	GPR83	GPCR / Class A : Orphans			
2775	31.09	oe	ccsbBroad304_02576	MLLT11	-			
2776	31.07	oe	ccsbBroad304_02618	DIDO1	Zinc fingers, PHD-type			
2777	30.99	kd	CGS001-6822	SULT2A1	Sulfotransferases, cytosolic			
2778	30.96	kd	CGS001-4258	MGST2	Glutathione S-transferases / Microsomal			
2779	30.94	cp	BRD-K00337317	NU-7441	DNA dependent protein kinase inhibitor		PRKDC, ABCB1	DNA dependent protein kinase inhibitor, P-glycoprotein inhibitor
2780	30.87	kd	CGS001-5695	PSMB7	Proteasome subunits			
2781	30.85	cp	BRD-K55301415	abiraterone	17,20 lyase inhibitor		CYP17A1, CYP11B1	17,20 lyase inhibitor, Androgen biosynthesis inhibitor, Cytochrome P450 inhibitor, Steroid sulfatase inhibitor
2782	30.83	cp	BRD-K88759641	EMD-66684	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
2783	30.83	kd	CGS001-8878	SQSTM1	-			
2784	30.83	kd	CGS001-11336	EXOC3	-			
2785	30.78	kd	CGS001-7004	TEAD4	-			
2786	30.7	kd	CGS001-6309	SC5DL	-			
2787	30.69	oe	ccsbBroad304_06870	RNH1	-			
2788	30.69	kd	CGS001-8239	USP9X	Ubiquitin-specific peptidases			
2789	30.69	kd	CGS001-6519	SLC3A1	SLC3 family			
2790	30.68	cp	BRD-U08759356	EI-346-erlotinib-analog	EGFR inhibitor		EGFR	EGFR inhibitor
2791	30.66	oe	ccsbBroad304_06528	FADS3	Fatty acid desaturases			
2792	30.65	cp	BRD-K66707493	lawsone	Coloring agent			Coloring agent
2793	30.64	kd	CGS001-11041	B3GNT1	-			
2794	30.64	cp	BRD-A75769826	SDM25N	Opioid receptor antagonist		OPRD1	Opioid receptor antagonist
2795	30.61	oe	ccsbBroad304_06211	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
2796	30.61	kd	CGS001-8165	AKAP1	A-kinase anchor proteins			
2797	30.6	kd	CGS001-9759	HDAC4	Histone deacetylases			
2798	30.59	kd	CGS001-7982	ST7	-			
2799	30.53	kd	CGS001-6390	SDHB	Mitochondrial respiratory chain complex / Complex II			
2800	30.51	cp	BRD-K62736196	guanabenz	-666		ADRA2A, ADRA2B, ADRA2C	-666
2801	30.49	oe	ccsbBroad304_00839	IGFBP6	insulin-like growth factor (IGF) binding proteins			
2802	30.45	kd	CGS001-498	ATP5A1	ATPases / F-type			
2803	30.44	kd	CGS001-64080	RBKS	-			
2804	30.44	kd	CGS001-5792	PTPRF	Receptor tyrosine phosphatases (RTP)			
2805	30.42	oe	ccsbBroad304_03372	CAB39	-			
2806	30.42	kd	CGS001-5901	RAN	-			
2807	30.33	oe	ccsbBroad304_01945	IKBKG	Zinc fingers, C2HC-type containing			
2808	30.3	oe	ccsbBroad304_04153	PHF17	-			
2809	30.2	cp	BRD-K76587808	fraxetin	Antioxidant			Antioxidant
2810	30.19	oe	ccsbBroad304_00281	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
2811	30.13	kd	CGS001-171017	ZNF384	Zinc fingers, C2H2-type			
2812	30.08	kd	CGS001-2287	FKBP3	-			
2813	30.06	cp	BRD-K47717570	NBQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIA3, GRIA4, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
2814	30.06	kd	CGS001-1119	CHKA	-			
2815	30.02	kd	CGS001-10898	CPSF4	-			
2816	30	cp	BRD-A64227845	SKF-77434	Dopamine receptor agonist		DRD1	Dopamine receptor agonist
2817	30	cp	BRD-A08187463	racecadotril	Enkephalinase inhibitor		MME	Enkephalinase inhibitor
2818	29.99	cp	BRD-K36965586	m-chlorophenylbiguanide	Serotonin receptor agonist		HTR3A, HTR3B	Serotonin receptor agonist
2819	29.99	kd	CGS001-26271	FBXO5	F-boxes / other			
2820	29.95	kd	CGS001-2145	EZH1	Chromatin-modifying enzymes / K-methyltransferases			
2821	29.94	kd	CGS001-4891	SLC11A2	SLC11 family of proton-coupled metal ion transporters			
2822	29.88	kd	CGS001-23635	SSBP2	-			
2823	29.86	kd	CGS001-22809	ATF5	basic leucine zipper proteins			
2824	29.85	kd	CGS001-2990	GUSB	-			
2825	29.83	cp	BRD-K47328134	lysylphenylalanyl-tyrosine	Heparin activation inhibitor			Heparin activation inhibitor
2826	29.82	oe	ccsbBroad304_09284	UBE3B	-			
2827	29.81	kd	CGS001-2770	GNAI1	-			
2828	29.8	kd	CGS001-79073	TMEM109	-			
2829	29.79	oe	ccsbBroad304_02298	DNM1L	-			
2830	29.78	kd	CGS001-5590	PRKCZ	Iota subfamily			
2831	29.76	cp	BRD-K98684188	GSK-0660	PPAR receptor antagonist		PPARD	PPAR receptor antagonist
2832	29.73	kd	CGS001-3215	HOXB5	Homeoboxes / ANTP class : HOXL subclass			
2833	29.68	oe	ccsbBroad304_02752	TRIM2	RING-type (C3HC4) zinc fingers			
2834	29.67	kd	CGS001-2277	FIGF	-			
2835	29.63	oe	ccsbBroad304_00087	FAS	Tumour necrosis factor (TNF) receptor family			
2836	29.62	oe	ccsbBroad304_03122	RHOD	-			
2837	29.62	oe	ccsbBroad304_00259	CD40	Tumour necrosis factor (TNF) receptor family			
2838	29.61	kd	CGS001-776	CACNA1D	Calcium channel subunits			
2839	29.6	oe	ccsbBroad304_00615	GAPDH	-			
2840	29.6	cp	BRD-K63606607	bufalin	ATPase inhibitor		ATP1A1	ATPase inhibitor
2841	29.59	kd	CGS001-90655	TGIF2LY	Homeoboxes / TALE class			
2842	29.59	kd	CGS001-23536	ADAT1	-			
2843	29.57	oe	ccsbBroad304_00350	COX5B	Mitochondrial respiratory chain complex			
2844	29.57	cp	BRD-A50675702	fipronil	GABA gated chloride channel blocker			GABA gated chloride channel blocker, Chloride channel blocker
2845	29.57	kd	CGS001-9231	DLG5	-			
2846	29.53	oe	ccsbBroad304_09910	BCL6B	BTB/POZ domain containing			
2847	29.53	kd	CGS001-83593	RASSF5	-			
2848	29.53	kd	CGS001-8883	NAE1	Ubiquitin-like modifier activating enzymes			
2849	29.53	kd	CGS001-1856	DVL2	Dishevelled homologs			
2850	29.52	oe	ccsbBroad304_09765	ZBTB49	BTB/POZ domain containing			
2851	29.51	kd	CGS001-7023	TFAP4	Basic helix-loop-helix proteins			
2852	29.48	kd	CGS001-5055	SERPINB2	Serine (or cysteine) peptidase inhibitors			
2853	29.47	oe	ccsbBroad304_04933	GPR119	GPCR / Class A : Orphans			
2854	29.45	kd	CGS001-5981	RFC1	ATPases / AAA-type			
2855	29.45	kd	CGS001-894	CCND2	-			
2856	29.45	kd	CGS001-10554	AGPAT1	1-acylglycerol-3-phosphate O-acyltransferases			
2857	29.43	cp	BRD-K02950022	BMS-299897	Gamma secretase inhibitor			Gamma secretase inhibitor
2858	29.42	kd	CGS001-64805	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
2859	29.42	kd	CGS001-2108	ETFA	-			
2860	29.41	kd	CGS001-11011	TLK2	Tousled-like kinase (TLK) family			
2861	29.36	kd	CGS001-3033	HADH	-			
2862	29.29	oe	ccsbBroad304_00044	AK2	Adenylate kinases			
2863	29.29	kd	CGS001-51564	HDAC7	Histone deacetylases			
2864	29.23	cc		TGF beta receptor inhibitor	-			
2865	29.18	oe	ccsbBroad304_07683	ZNF268	Zinc fingers, C2H2-type			
2866	29.16	kd	CGS001-255725	OR52B2	GPCR / Class A : Olfactory receptors			
2867	29.13	oe	ccsbBroad304_02257	ZBTB24	BTB/POZ domain containing			
2868	29.1	kd	CGS001-2629	GBA	-			
2869	29.07	oe	ccsbBroad304_06198	FCGR2A	CD molecules			
2870	29.07	kd	CGS001-5728	PTEN	Protein tyrosine phosphatases / Class I Cys-based PTPs : PTENs			
2871	29.03	kd	CGS001-8227	AKAP17A	A-kinase anchor proteins			
2872	29.02	kd	CGS001-4665	NAB2	-			
2873	29.01	oe	ccsbBroad304_07075	TLR5	Toll-like receptor family			
2874	29.01	kd	CGS001-64858	DCLRE1B	-			
2875	28.98	kd	CGS001-4780	NFE2L2	basic leucine zipper proteins			
2876	28.97	cp	BRD-K18757346	U-46619	Thromboxane receptor agonist		PTGDR, PTGDR2, PTGER1, PTGER2, PTGER3, PTGER4, PTGFR, PTGIR, TBXA2R	Thromboxane receptor agonist
2877	28.94	cp	BRD-K45446451	JZL-184	Monoacylglucerol lipase inhibitor		MGLL	Monoacylglucerol lipase inhibitor
2878	28.92	oe	ccsbBroad304_08054	EIF2AK1	Other PEK family kinases			
2879	28.88	cp	BRD-K09471561	levofloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
2880	28.88	kd	CGS001-5345	SERPINF2	Serine (or cysteine) peptidase inhibitors			
2881	28.83	kd	CGS001-58497	PRUNE	-			
2882	28.82	kd	CGS001-405	ARNT	Basic helix-loop-helix proteins			
2883	28.81	kd	CGS001-149233	IL23R	IL-12 receptor family			
2884	28.79	kd	CGS001-90649	ZNF486	Zinc fingers, C2H2-type			
2885	28.78	kd	CGS001-6908	TBP	General transcription factors			
2886	28.76	cp	BRD-K96740444	itopride	Dopamine receptor antagonist		DRD2, ACHE, CHRM3	Dopamine receptor antagonist
2887	28.75	oe	ccsbBroad304_04715	MRGPRF	GPCR / Class A : Orphans			
2888	28.74	kd	CGS001-22934	RPIA	-			
2889	28.73	kd	CGS001-6643	SNX2	Sorting nexins			
2890	28.7	oe	ccsbBroad304_13936	PTPRF	Receptor tyrosine phosphatases (RTP)			
2891	28.7	kd	CGS001-6434	TRA2B	RNA binding motif (RRM) containing			
2892	28.69	kd	CGS001-4708	NDUFB2	Mitochondrial respiratory chain complex / Complex I			
2893	28.68	cc		PARP inhibitor	-			
2894	28.6	kd	CGS001-136051	ZNF786	Zinc fingers, C2H2-type			
2895	28.59	kd	CGS001-6605	SMARCE1	-			
2896	28.57	oe	ccsbBroad304_00418	CD55	CD molecules			
2897	28.57	kd	CGS001-4783	NFIL3	basic leucine zipper proteins			
2898	28.57	kd	CGS001-2053	EPHX2	-			
2899	28.56	kd	CGS001-3622	ING2	Zinc fingers, PHD-type			
2900	28.51	kd	CGS001-23549	DNPEP	Aminopeptidase I			
2901	28.5	kd	CGS001-3115	HLA-DPB1	Immunoglobulin superfamily / C1-set domain containing			
2902	28.46	cp	BRD-A68930007	ouabain	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
2903	28.45	oe	ccsbBroad304_01741	UBE2V1	Ubiquitin-conjugating enzymes E2			
2904	28.45	kd	CGS001-3028	HSD17B10	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
2905	28.42	kd	CGS001-84647	PLA2G12B	-			
2906	28.42	kd	CGS001-1495	CTNNA1	Catenins			
2907	28.42	kd	CGS001-993	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
2908	28.41	kd	CGS001-4194	MDM4	-			
2909	28.4	kd	CGS001-2495	FTH1	-			
2910	28.4	kd	CGS001-56033	BARX1	Homeoboxes / ANTP class : NKL subclass			
2911	28.38	kd	CGS001-6461	SHB	SH2 domain containing			
2912	28.37	oe	ccsbBroad304_02361	MFSD10	-			
2913	28.36	cp	BRD-K46678324	RHO-kinase-inhibitor-II	Rho associated kinase inhibitor			Rho associated kinase inhibitor
2914	28.36	kd	CGS001-58533	SNX6	Sorting nexins			
2915	28.36	kd	CGS001-4720	NDUFS2	Mitochondrial respiratory chain complex / Complex I			
2916	28.3	oe	ccsbBroad304_04257	SPRY4	-			
2917	28.29	oe	ccsbBroad304_10035	ZKSCAN2	Zinc fingers, C2H2-type			
2918	28.22	kd	CGS001-11257	TP53TG1	-			
2919	28.21	cp	BRD-K08619574	thioproperazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, DRD1, DRD2, HTR1A, HTR2A	Dopamine receptor antagonist
2920	28.2	kd	CGS001-4801	NFYB	-			
2921	28.18	kd	CGS001-23534	TNPO3	Importins			
2922	28.18	kd	CGS001-5445	PON2	Paraoxonases			
2923	28.16	oe	ccsbBroad304_04465	RERG	-			
2924	28.12	cp	BRD-A78322124	dobutamine	Adrenergic receptor agonist		ADRB1, ADRB2, ADRA1A	Adrenergic receptor agonist
2925	28.12	kd	CGS001-8607	RUVBL1	ATPases / AAA-type			
2926	28.08	cp	BRD-K81473089	tacrine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Acetylcholine release stimulant, Butyrylcholinesterase inhibitor, Potassium channel antagonist
2927	28.07	cp	BRD-A96456596	FPL-55712	Leukotriene receptor antagonist			Leukotriene receptor antagonist
2928	28.07	kd	CGS001-63892	THADA	-			
2929	28.07	kd	CGS001-2098	ESD	-			
2930	28.06	oe	ccsbBroad304_06292	GNAI2	-			
2931	28.05	kd	CGS001-23636	NUP62	-			
2932	28.05	kd	CGS001-1594	CYP27B1	Cytochrome P450s			
2933	27.98	kd	CGS001-3486	IGFBP3	insulin-like growth factor (IGF) binding proteins			
2934	27.98	kd	CGS001-1070	CETN3	EF-hand domain containing			
2935	27.96	kd	CGS001-130497	OSR1	Zinc fingers, C2H2-type			
2936	27.9	cp	BRD-K24538644	KUC104502N	-666		OPRK1	-666
2937	27.88	kd	CGS001-11000	SLC27A3	SLC27 family of fatty acid transporters			
2938	27.87	oe	ccsbBroad304_09281	TPD52L3	-			
2939	27.87	oe	ccsbBroad304_09615	LACC1	-			
2940	27.87	kd	CGS001-5310	PKD1	Voltage-gated ion channels / Transient receptor potential cation channels			
2941	27.87	kd	CGS001-3692	EIF6	-			
2942	27.83	cp	BRD-A19195498	trimipramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, SLC6A3, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5, HRH1, HTR1A, HTR1D, HTR2A, HTR2C, HTR3A	Norepinephrine reuptake inhibitor, Tricyclic antidepressant
2943	27.83	kd	CGS001-821	CANX	-			
2944	27.82	cp	BRD-K60762818	desipramine	Tricyclic antidepressant		SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD2, HRH1, HTR1A, HTR2A, HTR2C, SMPD1	Tricyclic antidepressant
2945	27.81	kd	CGS001-6599	SMARCC1	-			
2946	27.78	kd	CGS001-2355	FOSL2	basic leucine zipper proteins			
2947	27.76	oe	ccsbBroad304_06348	HIST1H2BD	Histones / Replication-dependent			
2948	27.76	kd	CGS001-5881	RAC3	Endogenous ligands			
2949	27.76	kd	CGS001-8974	P4HA2	-			
2950	27.72	oe	ccsbBroad304_09225	BUD13	-			
2951	27.68	cp	BRD-K89152108	liothyronine	Thyroid hormone stimulant		THRA, THRB	Thyroid hormone stimulant
2952	27.65	oe	ccsbBroad304_03164	MTERFD1	-			
2953	27.64	cc		Kinase anchoring proteins LOF	-			
2954	27.62	kd	CGS001-222546	RFX6	-			
2955	27.61	oe	ccsbBroad304_00279	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
2956	27.59	oe	ccsbBroad304_03418	ZFAND6	Zinc fingers, AN1-type domain containing			
2957	27.59	kd	CGS001-5479	PPIB	-			
2958	27.59	kd	CGS001-26128	KIAA1279	-			
2959	27.56	oe	ccsbBroad304_01951	BLZF1	-			
2960	27.54	kd	CGS001-163081	ZNF567	Zinc fingers, C2H2-type			
2961	27.54	kd	CGS001-57798	GATAD1	GATA zinc finger domain containing			
2962	27.52	kd	CGS001-7074	TIAM1	Rho guanine nucleotide exchange factors			
2963	27.5	kd	CGS001-5265	SERPINA1	Serine (or cysteine) peptidase inhibitors			
2964	27.46	oe	ccsbBroad304_06976	SMARCE1	-			
2965	27.44	kd	CGS001-3560	IL2RB	IL-2 receptor family			
2966	27.43	kd	CGS001-2937	GSS	-			
2967	27.41	kd	CGS001-9945	GFPT2	-			
2968	27.4	oe	ccsbBroad304_04086	TCTN1	Tectonic proteins			
2969	27.39	oe	ccsbBroad304_03934	LEPRE1	-			
2970	27.32	oe	ccsbBroad304_06449	ILF3	-			
2971	27.3	cp	BRD-A62434282	goserelin	Gonadotropin releasing factor hormone receptor agonist		GNRHR, GNRH1, LHCGR	Gonadotropin releasing factor hormone receptor agonist, Luteinizing hormone releasing hormone agonist
2972	27.24	oe	ccsbBroad304_01388	RELB	NFkappaB transcription factor family			
2973	27.24	kd	CGS001-9564	BCAR1	Cas scaffolding proteins			
2974	27.23	kd	CGS001-10468	FST	-			
2975	27.22	kd	CGS001-2017	CTTN	-			
2976	27.2	cp	BRD-K14767410	SC-560	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
2977	27.17	kd	CGS001-7753	ZNF202	Zinc fingers, C2H2-type			
2978	27.15	oe	ccsbBroad304_00269	CD97	Adhesion Class GPCRs			
2979	27.15	oe	ccsbBroad304_00550	FDXR	-			
2980	27.13	kd	CGS001-342926	ZNF677	Zinc fingers, C2H2-type			
2981	27.13	kd	CGS001-3203	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
2982	27.11	oe	ccsbBroad304_00085	APRT	-			
2983	27.1	cp	BRD-K54316499	tolterodine	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRM1, CHRM4, CHRM5	Acetylcholine receptor antagonist
2984	27.1	kd	CGS001-1879	EBF1	-			
2985	27.08	oe	ccsbBroad304_06435	RBPJ	-			
2986	27.06	oe	ccsbBroad304_08394	UGT1A6	UDP glucuronosyltransferases			
2987	27	cp	BRD-A07440155	labetalol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1D, ADRA1B	Adrenergic receptor antagonist
2988	26.97	oe	ccsbBroad304_08228	PHF11	Zinc fingers, PHD-type			
2989	26.95	kd	CGS001-5950	RBP4	Lipocalins			
2990	26.93	kd	CGS001-6505	SLC1A1	Glutamate transporter subfamily			
2991	26.91	kd	CGS001-5920	RARRES3	-			
2992	26.9	kd	CGS001-5914	RARA	Retinoic acid receptors			
2993	26.89	cp	BRD-K27305650	LY-294002	MTOR inhibitor		MTOR, PIK3CD, PIK3CG, PIK3CA, PIK3CB, PLK1, PRKDC, AKT1, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PDE2A, PRKCA, ROCK1, RPS6KB1, SGK1	MTOR inhibitor, PI3K inhibitor, DNA dependent protein kinase inhibitor, Phosphodiesterase inhibitor, PLK inhibitor
2994	26.88	kd	CGS001-89766	UMODL1	-			
2995	26.79	kd	CGS001-10149	GPR64	Adhesion Class GPCRs			
2996	26.71	cp	BRD-K48923948	BMS-641988	Androgen receptor antagonist		AR	Androgen receptor antagonist
2997	26.69	cp	BRD-K82164249	andarine	Androgen receptor modulator		AR	Androgen receptor modulator
2998	26.69	kd	CGS001-79366	HMGN5	High-mobility group / Canonical			
2999	26.65	kd	CGS001-4174	MCM5	-			
3000	26.65	kd	CGS001-115330	GPR146	GPCR / Class A : Orphans			
3001	26.64	kd	CGS001-6038	RNASE4	Ribonucleases, RNase A			
3002	26.64	kd	CGS001-3276	PRMT1	Protein arginine N-methyltransferases			
3003	26.63	cp	BRD-A88774919	doxycycline	Bacterial 30S ribosomal subunit inhibitor		MMP8, MMP1	Bacterial 30S ribosomal subunit inhibitor, Metalloproteinase inhibitor
3004	26.62	oe	ccsbBroad304_07890	CBX7	-			
3005	26.62	cp	BRD-A94756469	digoxin	ATPase inhibitor		ATP1A1, ABCB1, RORC, SLCO1B3	ATPase inhibitor
3006	26.58	oe	ccsbBroad304_04767	SOCS4	SH2 domain containing			
3007	26.58	kd	CGS001-2149	F2R	Protease activated receptors			
3008	26.57	cp	BRD-K38305202	domperidone	Dopamine receptor antagonist		DRD2, DRD3, ABCG2, CYP3A5	Dopamine receptor antagonist
3009	26.56	kd	CGS001-6944	VPS72	-			
3010	26.56	kd	CGS001-23075	SWAP70	EF-hand domain containing			
3011	26.54	kd	CGS001-3481	IGF2	-			
3012	26.54	kd	CGS001-3087	HHEX	Homeoboxes / ANTP class : NKL subclass			
3013	26.52	cp	BRD-A52660433	tetrindole	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
3014	26.51	kd	CGS001-400	ARL1	ADP-ribosylation factors			
3015	26.47	kd	CGS001-5689	PSMB1	Proteasome subunits			
3016	26.43	oe	ccsbBroad304_01655	DYNLT3	Cytoplasmic dyneins			
3017	26.43	kd	CGS001-4711	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
3018	26.39	oe	ccsbBroad304_00836	IGF2	-			
3019	26.39	kd	CGS001-4886	NPY1R	GPCR / Class A : Neuropeptide receptors : Y			
3020	26.38	oe	ccsbBroad304_09368	OPN4	GPCR / Class A : Opsin receptors			
3021	26.38	cp	BRD-K14880289	GW-501516	PPAR receptor agonist		PPARD, INS, PPARA	PPAR receptor agonist, Insulin sensitizer
3022	26.37	kd	CGS001-1534	CYB561	Cytochrome b genes			
3023	26.36	oe	ccsbBroad304_08170	PIK3R4	Phosphatidylinositol kinases			
3024	26.36	oe	ccsbBroad304_02581	ASCC3	-			
3025	26.3	oe	ccsbBroad304_01239	POLR2E	RNA polymerase subunits			
3026	26.25	kd	CGS001-64764	CREB3L2	basic leucine zipper proteins			
3027	26.22	oe	ccsbBroad304_00361	ATF2	basic leucine zipper proteins			
3028	26.22	cp	BRD-A42628519	iopanoic-acid	Radiopaque medium			Radiopaque medium
3029	26.21	oe	ccsbBroad304_02414	IRF9	-			
3030	26.21	kd	CGS001-8491	MAP4K3	MAPKKKK:KHS subfamily			
3031	26.19	kd	CGS001-2180	ACSL1	Acyl-CoA synthetase family			
3032	26.16	oe	ccsbBroad304_06735	PLAU	Chymotrypsin			
3033	26.16	oe	ccsbBroad304_00471	E2F6	-			
3034	26.14	cp	BRD-K79254416	decitabine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
3035	26.13	cp	BRD-A91008255	bepridil	Calcium channel blocker		ATP1A1, CACNA1A, CACNA1C, CACNA1H, CACNA2D2, CALM1, KCNQ1, KCNQ4, PDE1A, PDE1B, SCN5A, TNNC1	Calcium channel blocker, L-type calcium channel blocker
3036	26.06	kd	CGS001-3667	IRS1	Pleckstrin homology (PH) domain containing			
3037	26.03	oe	ccsbBroad304_00084	APOH	Apolipoproteins			
3038	26.03	kd	CGS001-51593	SRRT	-			
3039	26.03	kd	CGS001-6697	SPR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3040	26.03	kd	CGS001-112398	EGLN2	2-oxoglutarate oxygenases			
3041	26.03	kd	CGS001-130	ADH6	Alcohol dehydrogenases			
3042	25.97	cp	BRD-K54472332	elvitegravir	HIV integrase inhibitor			HIV integrase inhibitor
3043	25.97	kd	CGS001-6514	SLC2A2	Solute carriers			
3044	25.92	kd	CGS001-533	ATP6V0B	ATPases / V-type			
3045	25.91	cp	BRD-K78373679	RO-3306	CDK inhibitor		CDK1	CDK inhibitor
3046	25.9	oe	ccsbBroad304_01929	DYRK2	Dyrk2 subfamily			
3047	25.9	kd	CGS001-2773	GNAI3	-			
3048	25.88	kd	CGS001-5092	PCBD1	-			
3049	25.86	kd	CGS001-203523	ZNF449	Zinc fingers, C2H2-type			
3050	25.82	kd	CGS001-9184	BUB3	WD repeat domain containing			
3051	25.81	kd	CGS001-2232	FDXR	-			
3052	25.79	kd	CGS001-5715	PSMD9	Proteasome (prosome, macropain) subunits			
3053	25.77	kd	CGS001-6663	SOX10	SRY (sex determining region Y)-boxes			
3054	25.73	cp	BRD-M16762496	PIK-75	DNA protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA protein kinase inhibitor, PI3K inhibitor
3055	25.72	cp	BRD-K37456065	VU-0365114-2	M5 modulator		CHRM5	M5 modulator
3056	25.68	oe	ccsbBroad304_06339	GTF2F2	General transcription factors			
3057	25.68	kd	CGS001-4190	MDH1	-			
3058	25.64	cp	BRD-A52326238	isogedunin	HSP inhibitor			HSP inhibitor
3059	25.62	oe	ccsbBroad304_02979	RNF11	RING-type (C3HC4) zinc fingers			
3060	25.62	kd	CGS001-4221	MEN1	-			
3061	25.62	kd	CGS001-2147	F2	Endogenous ligands			
3062	25.6	oe	ccsbBroad304_01960	CASK	CASK family			
3063	25.56	kd	CGS001-54807	ZNF586	Zinc fingers, C2H2-type			
3064	25.54	cc		Proteasome Pathway LOF	-			
3065	25.54	oe	ccsbBroad304_07808	RAB11FIP2	-			
3066	25.53	kd	CGS001-5264	PHYH	-			
3067	25.51	oe	ccsbBroad304_06458	IRF3	-			
3068	25.51	oe	ccsbBroad304_00572	FKBP3	-			
3069	25.49	cp	BRD-K70505054	ranitidine	Histamine receptor antagonist		HRH2, SLC22A2	Histamine receptor antagonist
3070	25.48	oe	ccsbBroad304_01580	SOX10	SRY (sex determining region Y)-boxes			
3071	25.47	oe	ccsbBroad304_08045	NOX1	-			
3072	25.47	cp	BRD-K15025317	BAY-11-7821	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
3073	25.47	kd	CGS001-9441	MED26	-			
3074	25.46	cp	BRD-K18518344	digitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
3075	25.46	kd	CGS001-5019	OXCT1	-			
3076	25.44	kd	CGS001-9290	GPR55	GPCR / Class A : Orphans			
3077	25.42	oe	ccsbBroad304_01215	PLAUR	CD molecules			
3078	25.4	oe	ccsbBroad304_00105	ARNTL	Basic helix-loop-helix proteins			
3079	25.4	kd	CGS001-6813	STXBP2	-			
3080	25.38	kd	CGS001-10046	MAMLD1	-			
3081	25.37	kd	CGS001-3212	HOXB2	Homeoboxes / ANTP class : HOXL subclass			
3082	25.33	oe	ccsbBroad304_01347	RAD1	-			
3083	25.33	kd	CGS001-5860	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
3084	25.33	kd	CGS001-367	AR	Nuclear hormone receptors			
3085	25.32	oe	ccsbBroad304_02887	CLIC4	Ion channels / Chloride channels : Intracellular			
3086	25.31	cp	BRD-K52721684	PCO-400	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
3087	25.29	cp	BRD-K95237249	probenecid	Uricosuric blocker		SLC22A6, ABCC1, PANX1, SLC22A11, SLC22A8, SLCO1C1, TRPV2	Uricosuric blocker
3088	25.29	kd	CGS001-65263	PYCRL	-			
3089	25.29	kd	CGS001-960	CD44	CD molecules			
3090	25.28	kd	CGS001-128368	OR10Z1	GPCR / Class A : Olfactory receptors			
3091	25.22	kd	CGS001-2674	GFRA1	GDNF receptor family			
3092	25.19	kd	CGS001-10664	CTCF	Zinc fingers, C2H2-type			
3093	25.18	kd	CGS001-7533	YWHAH	-			
3094	25.17	kd	CGS001-79135	APOO	Apolipoproteins			
3095	25.14	kd	CGS001-23335	WDR7	WD repeat domain containing			
3096	25.14	kd	CGS001-10250	SRRM1	-			
3097	25.13	kd	CGS001-58477	SRPRB	-			
3098	25.13	kd	CGS001-204219	CERS3	Homeoboxes / CERS class			
3099	25.03	cp	BRD-K45542189	diethylcarbamazine	Lipoxygenase inhibitor		ALOX5, PTGS1	Lipoxygenase inhibitor
3100	25	cp	BRD-A35519318	benidipine	Calcium channel blocker		CACNA1C, CACNA1G, CYP3A5	Calcium channel blocker
3101	24.93	oe	ccsbBroad304_00532	F11	Chymotrypsin			
3102	24.92	kd	CGS001-6932	TCF7	-			
3103	24.86	kd	CGS001-83729	INHBE	-			
3104	24.85	kd	CGS001-23321	TRIM2	RING-type (C3HC4) zinc fingers			
3105	24.84	oe	ccsbBroad304_04235	TDRD3	Tudor domain containing			
3106	24.81	cp	BRD-K68620903	dydrogesterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3107	24.81	kd	CGS001-4214	MAP3K1	MAPKKK:STE11 family			
3108	24.81	kd	CGS001-386724	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
3109	24.8	cp	BRD-K59962020	CHEMBL-374350	NFkB pathway inhibitor			NFkB pathway inhibitor
3110	24.79	kd	CGS001-9459	ARHGEF6	Rho guanine nucleotide exchange factors			
3111	24.78	oe	ccsbBroad304_00110	ASGR2	C-type lectin domain containing			
3112	24.78	kd	CGS001-79143	MBOAT7	-			
3113	24.76	kd	CGS001-3559	IL2RA	IL-2 receptor family			
3114	24.73	kd	CGS001-7984	ARHGEF5	Rho guanine nucleotide exchange factors			
3115	24.7	kd	CGS001-54600	UGT1A9	UDP glucuronosyltransferases			
3116	24.68	kd	CGS001-9360	PPIG	-			
3117	24.66	oe	ccsbBroad304_08221	RDH11	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
3118	24.59	kd	CGS001-5859	QARS	Aminoacyl tRNA synthetases / Class I			
3119	24.58	kd	CGS001-9218	VAPA	-			
3120	24.55	kd	CGS001-10434	LYPLA1	-			
3121	24.55	kd	CGS001-151306	GPBAR1	Bile acid receptor			
3122	24.55	kd	CGS001-30	ACAA1	-			
3123	24.53	kd	CGS001-57721	METTL14	-			
3124	24.53	kd	CGS001-10142	AKAP9	A-kinase anchor proteins			
3125	24.49	kd	CGS001-25942	SIN3A	-			
3126	24.49	kd	CGS001-283450	C12ORF51	-			
3127	24.47	kd	CGS001-122402	TDRD9	Tudor domain containing			
3128	24.46	oe	ccsbBroad304_06760	PPP2R3A	EF-hand domain containing			
3129	24.41	kd	CGS001-10607	TBL3	WD repeat domain containing			
3130	24.41	kd	CGS001-80274	SCUBE1	-			
3131	24.39	kd	CGS001-10026	PIGK	Phosphatidylinositol glycan anchor biosynthesis			
3132	24.38	kd	CGS001-1650	DDOST	-			
3133	24.36	oe	ccsbBroad304_01180	PFKFB3	-			
3134	24.24	kd	CGS001-7039	TGFA	-			
3135	24.22	kd	CGS001-59286	UBL5	-			
3136	24.22	kd	CGS001-2063	NR2F6	COUP-TF-like receptors			
3137	24.2	oe	ccsbBroad304_11549	ZNF273	Zinc fingers, C2H2-type			
3138	24.14	kd	CGS001-661	POLR3D	RNA polymerase subunits			
3139	24.13	kd	CGS001-4976	OPA1	-			
3140	24.12	cp	BRD-K16233984	eriochrome-black-t	Azo dye			Azo dye
3141	24.09	oe	ccsbBroad304_08978	ZNF672	Zinc fingers, C2H2-type			
3142	24.08	cp	BRD-K89046952	ciclacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3143	24.07	cp	BRD-K56334280	amonafide	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
3144	24.06	kd	CGS001-5526	PPP2R5B	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
3145	24.02	kd	CGS001-2678	GGT1	CD molecules			
3146	24	oe	ccsbBroad304_06431	IFNAR2	Interferon receptor family			
3147	23.98	kd	CGS001-3172	HNF4A	Hepatocyte nuclear factor-4 receptors			
3148	23.98	kd	CGS001-91949	COG7	Components of oligomeric golgi complex			
3149	23.96	kd	CGS001-2821	GPI	-			
3150	23.94	oe	ccsbBroad304_00250	CD19	CD molecules			
3151	23.89	kd	CGS001-10153	CEBPZ	-			
3152	23.88	cp	BRD-A32949107	MRS-1845	Calcium channel blocker		ORAI1	Calcium channel blocker
3153	23.87	kd	CGS001-8050	PDHX	-			
3154	23.85	kd	CGS001-54555	DDX49	DEAD-boxes			
3155	23.8	kd	CGS001-2132	EXT2	Exostosin glycosyltransferase family			
3156	23.78	kd	CGS001-3717	JAK2	Janus kinase (JakA) family			
3157	23.76	oe	ccsbBroad304_08389	DHX29	DEAH-boxes			
3158	23.76	kd	CGS001-51382	ATP6V1D	ATPases / V-type			
3159	23.74	oe	ccsbBroad304_05836	BIRC5	Inhibitors of apoptosis (IAP) protein family			
3160	23.73	kd	CGS001-6664	SOX11	SRY (sex determining region Y)-boxes			
3161	23.66	cp	BRD-A11135865	nor-binaltorphimine	Opioid receptor antagonist			Opioid receptor antagonist
3162	23.65	kd	CGS001-51335	NGRN	-			
3163	23.63	kd	CGS001-23244	PDS5A	-			
3164	23.61	cp	BRD-K77771411	moxonidine	Imidazoline receptor agonist		NISCH, ADRA2A, ADRA2B, ADRA2C	Imidazoline receptor agonist
3165	23.6	kd	CGS001-5654	HTRA1	Serine peptidases / Serine peptidases			
3166	23.59	cp	BRD-K08219523	5-nonyloxytryptamine	Serotonin receptor agonist		HTR1B, HTR1D	Serotonin receptor agonist
3167	23.58	oe	ccsbBroad304_07275	PSMG1	-			
3168	23.58	kd	CGS001-64781	CERK	Ceramide kinase			
3169	23.56	oe	ccsbBroad304_02372	SPRY1	-			
3170	23.55	oe	ccsbBroad304_01313	PSMB9	Proteasome (prosome, macropain) subunits			
3171	23.54	kd	CGS001-3927	LASP1	-			
3172	23.53	cc		IGF-1 inhibitor	-			
3173	23.5	cp	BRD-A92537424	danazol	Estrogen receptor antagonist		ESR1, GNRHR, AR, CCL2, CYP2C8, GNRHR2, PGR, TNF	Estrogen receptor antagonist, Progesterone receptor agonist
3174	23.47	oe	ccsbBroad304_00929	LBR	Tudor domain containing			
3175	23.47	cp	BRD-K51575138	TPCA-1	IKK inhibitor		IKBKB	IKK inhibitor
3176	23.47	kd	CGS001-8609	KLF7	Kruppel-like transcription factors			
3177	23.44	kd	CGS001-54805	CNNM2	-			
3178	23.42	cp	BRD-K72816382	cinalukast	Leukotriene receptor antagonist		CYSLTR1	Leukotriene receptor antagonist
3179	23.36	kd	CGS001-1459	CSNK2A2	Casein kinase 2 (CK2) family			
3180	23.32	kd	CGS001-23029	RBM34	RNA binding motif (RRM) containing			
3181	23.29	kd	CGS001-5966	REL	NFkappaB transcription factor family			
3182	23.27	kd	CGS001-1577	CYP3A5	Cytochrome P450s			
3183	23.26	kd	CGS001-3673	ITGA2	Integrins			
3184	23.23	cp	BRD-K82216340	medroxyprogesterone	progesterone receptor agonist		PGR, ESR1	progesterone receptor agonist
3185	23.22	cp	BRD-K56115039	BU-226	Imidazoline receptor ligand			Imidazoline receptor ligand
3186	23.17	oe	ccsbBroad304_05002	ZNF563	Zinc fingers, C2H2-type			
3187	23.17	kd	CGS001-6768	ST14	Serine peptidases / Transmembrane			
3188	23.13	cp	BRD-K81418486	vorinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, HDAC10, HDAC11, HDAC5, HDAC9	HDAC inhibitor
3189	23.1	cp	BRD-K40901640	cinanserin	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
3190	23.09	cp	BRD-K14696368	9-methyl-5H-6-thia-4,5-diaza-chrysene-6,6-dioxide	NFkB pathway inhibitor		RELA	NFkB pathway inhibitor
3191	23.08	kd	CGS001-10084	PQBP1	-			
3192	23.07	oe	ccsbBroad304_05948	CCND2	-			
3193	23.06	kd	CGS001-79145	CHCHD7	Coiled-coil-helix-coiled-coil-helix domain containing			
3194	23.06	kd	CGS001-392	ARHGAP1	Rho GTPase activating proteins			
3195	23.05	cp	BRD-A84389091	L-655708	GABA receptor inverse agonist		GABRA5, GABRA1, GABRA2, GABRA3, GABRG2	GABA receptor inverse agonist
3196	23.03	cp	BRD-K74141488	naftifine	Fungal squalene epoxidase inhibitor		SQLE	Fungal squalene epoxidase inhibitor
3197	23.01	kd	CGS001-10873	ME3	-			
3198	23	oe	ccsbBroad304_03928	RRAGC	-			
3199	22.94	kd	CGS001-39	ACAT2	Lanosterol biosynthesis pathway			
3200	22.93	kd	CGS001-29956	CERS2	Homeoboxes / CERS class			
3201	22.93	kd	CGS001-567	B2M	Immunoglobulin superfamily / C1-set domain containing			
3202	22.84	kd	CGS001-7923	HSD17B8	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
3203	22.82	kd	CGS001-5337	PLD1	Phosphatidylcholine-specific phospholipase D			
3204	22.75	kd	CGS001-5933	RBL1	-			
3205	22.74	kd	CGS001-57026	PDXP	-			
3206	22.73	cp	BRD-K72093121	vidarabine	Antiviral		ADCY5	Antiviral
3207	22.72	kd	CGS001-93185	IGSF8	CD molecules			
3208	22.71	cp	BRD-K37618799	MRS-1220	Adenosine receptor antagonist		ADORA2B, ADORA3	Adenosine receptor antagonist
3209	22.6	kd	CGS001-10456	HAX1	-			
3210	22.58	kd	CGS001-10150	MBNL2	Zinc fingers, CCCH-type domain containing			
3211	22.56	kd	CGS001-6198	RPS6KB1	p70 subfamily			
3212	22.46	kd	CGS001-3554	IL1R1	Interleukins and interleukin receptors			
3213	22.45	kd	CGS001-10336	PCGF3	Polycomb group ring fingers			
3214	22.42	oe	ccsbBroad304_01771	VIM	Intermediate filaments type III			
3215	22.4	cp	BRD-K21350491	phenamil	TRPV antagonist		PKD2L1	TRPV antagonist
3216	22.33	kd	CGS001-6845	VAMP7	Pseudoautosomal regions / PAR2			
3217	22.32	kd	CGS001-8324	FZD7	GPCR / Class F : Frizzled receptors			
3218	22.27	oe	ccsbBroad304_02324	TRAP1	Heat shock proteins / HSPC			
3219	22.27	oe	ccsbBroad304_01613	STK11	LKB subfamily			
3220	22.21	cp	BRD-K26657438	imiquimod	TLR agonist		TLR7, TLR8	TLR agonist, Interferon inducer
3221	22.15	cp	BRD-K20141153	atomoxetine	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Norepinephrine transporter inhibitor
3222	22.08	kd	CGS001-9928	KIF14	Kinesins			
3223	22.06	cp	BRD-K22031190	diflunisal	Prostanoid receptor antagonist		PTGS2, PTGS1	Prostanoid receptor antagonist
3224	22.02	kd	CGS001-9412	MED21	-			
3225	21.96	cp	BRD-K47639036	flavoxate	Acetylcholine receptor antagonist		CHRM1, CHRM2	Acetylcholine receptor antagonist
3226	21.85	kd	CGS001-115992	RNF166	RING-type (C3HC4) zinc fingers			
3227	21.83	kd	CGS001-4830	NME1	-			
3228	21.83	kd	CGS001-79947	DHDDS	-			
3229	21.81	cp	BRD-A95939040	sertaconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
3230	21.77	kd	CGS001-51176	LEF1	-			
3231	21.77	kd	CGS001-34	ACADM	-			
3232	21.76	cp	BRD-K32795028	1-benzylimidazole	Thromboxane synthase inhibitor		CYP11B1, QPCT	Thromboxane synthase inhibitor
3233	21.72	oe	ccsbBroad304_02756	RRP8	-			
3234	21.69	kd	CGS001-9133	CCNB2	-			
3235	21.64	cp	BRD-K63874012	thioperamide	Histamine receptor antagonist		HRH3, HRH4	Histamine receptor antagonist
3236	21.64	kd	CGS001-890	CCNA2	-			
3237	21.64	cp	BRD-K92723993	imatinib	BCR-ABL kinase inhibitor		ABL1, KIT, PDGFRA, BCR, CSF1R, PDGFRB, ABCG2, CYP2C19, CYP2C8, CYP3A5, DDR1, NTRK1, RET	BCR-ABL kinase inhibitor, KIT inhibitor, PDGFR receptor inhibitor
3238	21.63	kd	CGS001-11186	RASSF1	-			
3239	21.55	kd	CGS001-2030	SLC29A1	SLC29 family			
3240	21.48	kd	CGS001-160	AP2A1	-			
3241	21.45	cp	BRD-K29582115	ziprasidone	Dopamine receptor antagonist		DRD2, HTR2A, HTR1A, HTR1D, HRH1, HTR1B, HTR1E, HTR2C, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, DRD4, DRD5, HTR3A, HTR6, SLC6A4	Dopamine receptor antagonist, Serotonin receptor antagonist
3242	21.45	kd	CGS001-1173	AP2M1	-			
3243	21.44	kd	CGS001-55239	OGFOD1	-			
3244	21.42	cp	BRD-K19894101	MST-312	Telomerase inhibitor		TERT	Telomerase inhibitor
3245	21.42	kd	CGS001-994	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
3246	21.37	kd	CGS001-9314	KLF4	Kruppel-like transcription factors			
3247	21.37	cp	BRD-K67043667	altretamine	DNA synthesis inhibitor			DNA synthesis inhibitor
3248	21.22	kd	CGS001-6443	SGCB	-			
3249	21.14	cp	BRD-K90733503	cefalexin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3250	21.11	kd	CGS001-11129	CLASRP	-			
3251	21.07	oe	ccsbBroad304_11503	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
3252	20.99	cp	BRD-K46068882	eugenitol	Bacterial quorum sensing inhibitor		AR, MAOA	Bacterial quorum sensing inhibitor, Chromone, Monoamine oxidase inhibitor, Androgen receptor antagonist
3253	20.83	cp	BRD-K14643723	4-(2-Amino-ethyl)-benzenesulfonamide	carbonic anhydrase inhibitor		CA2, CA1, CA9, CA12, CA14, CA4	carbonic anhydrase inhibitor
3254	20.81	cp	BRD-A56359832	zileuton	Leukotriene inhibitor		ALOX5	Leukotriene inhibitor, Lipoxygenase inhibitor
3255	20.77	kd	CGS001-205	AK4	Adenylate kinases			
3256	20.76	cp	BRD-K77008974	WYE-354	MTOR inhibitor		MTOR	MTOR inhibitor
3257	20.75	kd	CGS001-23597	ACOT9	Acyl CoA thioesterases			
3258	20.7	kd	CGS001-3104	ZBTB48	BTB/POZ domain containing			
3259	20.59	kd	CGS001-3708	ITPR1	Ion channels / Inositol triphosphate receptors			
3260	20.45	cp	BRD-K63516691	T-0156	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
3261	20.37	cp	BRD-A53077924	tianeptine	Selective serotonin reuptake enhancer (SSRE)		SLC6A4	Selective serotonin reuptake enhancer (SSRE)
3262	20.32	kd	CGS001-149428	BNIPL	-			
3263	20.28	oe	ccsbBroad304_13869	HLA-A	Immunoglobulin superfamily / C1-set domain containing			
3264	20.25	cp	BRD-A68039575	liquiritigenin	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3265	20.2	kd	CGS001-5306	PITPNA	-			
3266	20.15	kd	CGS001-8604	SLC25A12	Mitochondrial amino acid transporter subfamily			
3267	20.08	kd	CGS001-7030	TFE3	Basic helix-loop-helix proteins			
3268	20.08	kd	CGS001-2997	GYS1	Glycosyltransferase group 1 domain containing			
3269	20.04	kd	CGS001-5351	PLOD1	-			
3270	20.02	kd	CGS001-5565	PRKAB2	AMPK subfamily			
3271	19.9	cp	BRD-A01320529	salmeterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3272	19.73	cp	BRD-K35559145	levomepromazine	Dopamine receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, DRD5, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
3273	19.51	cp	BRD-A41301928	bongkrek-acid	Mitochondrial ADP, ATP translocase inhibitor		SLC25A4	Mitochondrial ADP, ATP translocase inhibitor
3274	19.43	cp	BRD-K09397065	SR-57227A	Serotonin receptor agonist		HTR3A	Serotonin receptor agonist
3275	19.27	cp	BRD-K24132293	piperlongumine	Glutathione transferase inhibitor			Glutathione transferase inhibitor
3276	19.21	kd	CGS001-10421	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
3277	19.14	cp	BRD-K75089421	procainamide	Sodium channel blocker		SCN5A, DNMT1	Sodium channel blocker
3278	19.14	kd	CGS001-85027	C5ORF62	-			
3279	19.06	kd	CGS001-5770	PTPN1	Protein tyrosine phosphatases			
3280	19.03	kd	CGS001-124274	GPR139	GPCR / Class A : Orphans			
3281	18.94	kd	CGS001-1994	ELAVL1	RNA binding motif (RRM) containing			
3282	18.82	cp	BRD-K32164935	tolazamide	ATP channel blocker		KCNJ1, KCNJ10	ATP channel blocker
3283	18.81	cp	BRD-A82656074	naltrindole	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3284	18.78	kd	CGS001-64746	ACBD3	A-kinase anchor proteins			
3285	18.71	cp	BRD-A94543220	bifonazole	Sterol demethylase inhibitor		CYP2B6	Sterol demethylase inhibitor
3286	18.66	kd	CGS001-84971	ATG4D	-			
3287	18.61	cp	BRD-K12184916	dactolisib	MTOR inhibitor		MTOR, PIK3CA, PIK3CG, PIK3CD, ATR, PIK3CB	MTOR inhibitor, PI3K inhibitor, Protein kinase inhibitor
3288	18.61	kd	CGS001-1810	DR1	-			
3289	18.48	cp	BRD-K82255054	propofol	GABA receptor agonist		CYP2B6, FAAH, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, SCN2A, SCN4A, TRPV1	GABA receptor agonist
3290	18.42	cp	BRD-K20287671	SU-4312	PDGFR receptor inhibitor		KDR, PDGFRB	PDGFR receptor inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
3291	18.31	kd	CGS001-51027	BOLA1	-			
3292	18.23	cp	BRD-K56614220	clofazimine	GK0582 inhibitor			GK0582 inhibitor
3293	18.21	cp	BRD-K88849294	lobaric-acid	Tyrosine phosphatase inhibitor		PTPN1	Tyrosine phosphatase inhibitor
3294	18.2	kd	CGS001-7076	TIMP1	-			
3295	18.18	cp	BRD-K18909381	CGS-12066B	Serotonin receptor agonist		HTR1B, HTR1A, HTR1D, HTR2A, HTR2B, HTR2C	Serotonin receptor agonist
3296	18.1	kd	CGS001-1154	CISH	SH2 domain containing			
3297	18.05	kd	CGS001-7251	TSG101	-			
3298	17.96	cp	BRD-A15034104	bergenin	Interleukin inhibitor		PTPN1	Interleukin inhibitor
3299	17.96	cp	BRD-K28307902	flutamide	Androgen receptor antagonist		AR, AHR, CYP2C19	Androgen receptor antagonist
3300	17.96	kd	CGS001-10533	ATG7	Ubiquitin-like modifier activating enzymes			
3301	17.91	cp	BRD-K99174507	cardiogenol-c	Cardiomyogenesis inducer			Cardiomyogenesis inducer
3302	17.85	kd	CGS001-133690	CAPSL	EF-hand domain containing			
3303	17.82	kd	CGS001-81579	PLA2G12A	Phospholipase A2			
3304	17.75	cp	BRD-K65786282	CGP-7930	GABA receptor modulator		GABBR1	GABA receptor modulator, GABA receptor positive allosteric modulator
3305	17.74	cp	BRD-K02265150	amoxapine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, HTR2A, HTR6, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD3, DRD4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH1, HRH4, HTR1A, HTR1B, HTR2B, HTR2C, HTR3A, HTR7, SLC6A3	Norepinephrine reuptake inhibitor
3306	17.7	cp	BRD-K68143200	SA-792541	CDC inhibitor		CASP3, CDC25A, CDC25B	CDC inhibitor
3307	17.66	kd	CGS001-8464	SUPT3H	-			
3308	17.61	cp	BRD-K57011718	UK-356618	Metalloproteinase inhibitor		MMP3, MMP13, MMP14, MMP2, MMP9	Metalloproteinase inhibitor
3309	17.5	kd	CGS001-54851	ANKRD49	Ankyrin repeat domain containing			
3310	17.46	kd	CGS001-83881	MIXL1	Homeoboxes / PRD class			
3311	17.43	kd	CGS001-80212	CCDC92	-			
3312	17.42	cp	BRD-A94793051	gestrinone	Progesterone receptor antagonist		PGR, AR, ESR1	Progesterone receptor antagonist
3313	17.38	cp	BRD-K32501161	vanoxerine	Dopamine uptake inhibitor		SLC6A3, MAOA, MAOB	Dopamine uptake inhibitor
3314	17.27	kd	CGS001-8558	CDK10	Cyclin-dependent kinases, CDK10 subfamily			
3315	17.18	cp	BRD-A17428743	BW-723C86	Serotonin receptor agonist		HTR2B, HTR2A, HTR2C	Serotonin receptor agonist
3316	17.13	kd	CGS001-2542	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
3317	17.09	cp	BRD-K44084986	Y-27632	Rho associated kinase inhibitor		ROCK1, ROCK2, LRRK2, PKIA, PKN2, PRKACA, PRKCE	Rho associated kinase inhibitor
3318	17.09	cp	BRD-K09638361	SA-63133	-666		CSNK1E, CSNK1A1, CSNK1D, CSNK1G2	-666
3319	16.93	cp	BRD-K85402309	dovitinib	EGFR inhibitor		EGFR, FGFR3, PDGFRB, CSF1R, FGFR1, FGFR2, FLT1, FLT3, FLT4, INSR, KDR, KIT, PDGFRA	EGFR inhibitor, FLT3 inhibitor, FGFR inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
3320	16.86	cp	BRD-U44700465	HG-5-88-01	Protein kinase inhibitor		ADCK4, EGFR	Protein kinase inhibitor
3321	16.74	cp	BRD-K09549677	mibefradil	T-type calcium channel blocker		CACNA1G, CACNA1H, CACNA1C, CACNA1I, ANO1, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP3A5, CYP3A7, SCN2A, SCN4A, SCN5A, SCN9A	T-type calcium channel blocker
3322	16.73	cp	BRD-K35240538	methylprednisolone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3323	16.63	cp	BRD-K97509413	coumestrol	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
3324	16.63	cp	BRD-K78294846	osthol	Calcium channel blocker			Calcium channel blocker
3325	16.62	kd	CGS001-57167	SALL4	Zinc fingers, C2H2-type			
3326	16.53	cp	BRD-K95309561	dienestrol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
3327	16.53	kd	CGS001-54205	CYCS	-			
3328	16.41	kd	CGS001-1503	CTPS	-			
3329	16.33	cp	BRD-K67844266	MLN-4924	Nedd activating enzyme inhibitor		NAE1, UBA3	Nedd activating enzyme inhibitor
3330	16.15	cp	BRD-A45543382	metrizamide	Radiopaque medium			Radiopaque medium
3331	16.06	cp	BRD-K43978949	PIT	Purinergic receptor antagonist		P2RY1	Purinergic receptor antagonist
3332	16.01	cp	BRD-K32977963	eugenol	Androgen receptor antagonist		AR, MAOA	Androgen receptor antagonist
3333	15.9	cp	BRD-A36630025	SN-38	Topoisomerase inhibitor		TOP1	Topoisomerase inhibitor
3334	15.87	cp	BRD-K72029282	probucol	Atherogenesis inhibitor		ABCA1, ABCB11, CES1	Atherogenesis inhibitor
3335	15.87	cp	BRD-K12079898	PD-160170	Neuropeptide receptor antagonist		NPY1R	Neuropeptide receptor antagonist
3336	15.86	cp	BRD-A78360835	cercosporin	Photoactivated toxin			Photoactivated toxin
3337	15.83	cp	BRD-K23566484	nilutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
3338	15.62	cp	BRD-K01902415	pirinixic-acid	PPAR receptor agonist		PPARA	PPAR receptor agonist
3339	15.58	cp	BRD-K23922020	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
3340	15.52	cp	BRD-K73290745	ICI-199441	Opioid receptor agonist		OPRK1, CYP2D6, OPRD1, OPRM1, UTS2R	Opioid receptor agonist
3341	15.46	cp	BRD-K97863768	prothionamide	Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor			Mycobacterium tuberculosis enoyl-[acyl-carrier-protein] reductase [NADH] (inhA) inhibitor
3342	15.41	cp	BRD-A43331270	niguldipine	Calcium channel blocker		ADRA1A, CACNA1C, ADRA1B, ADRA1D	Calcium channel blocker, Adrenergic receptor antagonist
3343	15.4	kd	CGS001-10733	PLK4	Polo-like kinase (PLK) family			
3344	15.39	kd	CGS001-317703	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
3345	15.27	cc		SRY LOF	-			
3346	15.18	cp	BRD-K86600316	RS-79948	Adrenergic receptor antagonist			Adrenergic receptor antagonist
3347	15.15	cp	BRD-K50140147	NVP-TAE684	ALK inhibitor		ALK, INSR	ALK inhibitor
3348	15.13	cp	BRD-A85860691	chaetocin	Histone lysine methyltransferase inhibitor		EHMT2, SUV39H1	Histone lysine methyltransferase inhibitor
3349	14.9	kd	CGS001-5928	RBBP4	WD repeat domain containing			
3350	14.89	cp	BRD-A72703248	SKF-96365	Calcium channel blocker		CYP3A4, TRPC1, PKD2, TRPC3, TRPC4, TRPC5, TRPV2	Calcium channel blocker
3351	14.89	kd	CGS001-7477	WNT7B	Endogenous ligands			
3352	14.83	cp	BRD-K16977723	PP-3	EGFR inhibitor			EGFR inhibitor
3353	14.64	cp	BRD-A14395271	mesoridazine	Dopamine receptor antagonist		DRD2, HTR2A	Dopamine receptor antagonist
3354	14.5	cc		PKA inhibitor	-			
3355	14.47	cp	BRD-K94919853	10H-phenothiazin-10-yl)(p-tolyl)methanone	Butyrylcholinesterase inhibitor		BCHE	Butyrylcholinesterase inhibitor
3356	14.44	cp	BRD-K04412738	tramadol	Norepinephrine reuptake inhibitor		OPRM1, SLC6A2, SLC6A4, CHRFAM7A, CHRM3, CYP2B6, GRIN3A, HTR2C, OPRD1, OPRK1	Norepinephrine reuptake inhibitor, Opioid receptor agonist, Serotonin reuptake inhibitor
3357	14.28	cp	BRD-K88679075	methandriol	Androgenic steroid			Androgenic steroid
3358	14.28	cp	BRD-K07762753	aminopurvalanol-a	Tyrosine kinase inhibitor		CDK1, CDK2, CDK5, CDK6	Tyrosine kinase inhibitor, CDK inhibitor
3359	14.27	kd	CGS001-9817	KEAP1	Kelch-like proteins			
3360	14.26	cp	BRD-A26334849	propafenone	Antiarrhythmic		KCNH2, SCN5A, ADRB1, ADRB2, KCNA5, KCNK2, KCNK3	Antiarrhythmic
3361	14.23	cp	BRD-K28470988	L-690330	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
3362	14.14	kd	CGS001-126208	ZNF787	Zinc fingers, C2H2-type			
3363	14.03	cp	BRD-K55930204	phenytoin	Hydantoin antiepileptic		ABCB1, CYP2B6, CYP2C19, CYP3A4, SCN1A, SCN2A, SCN5A	Hydantoin antiepileptic
3364	14.01	cp	BRD-K83508485	FK-888	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
3365	13.99	cp	BRD-A88282067	delcorine	Antiarrhythmic			Antiarrhythmic, Ganglionic blocker
3366	13.85	cp	BRD-A11990600	lorazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, TSPO	Benzodiazepine receptor agonist
3367	13.74	cp	BRD-K81376179	TCS-359	FLT3 inhibitor		FLT3	FLT3 inhibitor
3368	13.72	cp	BRD-K82135108	elesclomol	Oxidative stress inducer		TOP2A	Oxidative stress inducer
3369	13.66	cp	BRD-K77171813	proxyfan	Histamine receptor modulator		HRH3	Histamine receptor modulator
3370	13.59	cp	BRD-A28746609	paclitaxel	Tubulin inhibitor		TUBB, NR1I2, ABCB1, BCL2, CYP2C8, MAP2, MAP4, MAPT, TLR4, TUBB1	Tubulin inhibitor
3371	13.55	cp	BRD-A89175223	bisoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3372	13.54	cp	BRD-A40639672	ketorolac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3373	13.41	cp	BRD-K68867920	quetiapine	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, DRD1, HRH1, HTR1D, HTR1E, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD3, DRD4, DRD5, HTR1B, HTR1F, HTR2C, HTR3A, HTR6, HTR7, SLC6A2	Dopamine receptor antagonist, Serotonin receptor antagonist
3374	13.36	cp	BRD-K11717138	benzbromarone	Chloride channel blocker		ABCC1, SLC22A12	Chloride channel blocker
3375	13.28	cp	BRD-K63165456	norcyclobenzaprine	Adrenergic receptor agonist		HTR2A	Adrenergic receptor agonist, Serotonin receptor antagonist
3376	13.24	cp	BRD-K97118047	4,5,6,7-tetrabromobenzotriazole	Casein kinase inhibitor		CSNK2A1, AKT1, CHEK1, CSNK2A2, CSNK2B, GSK3B, LCK, MAP2K1, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	Casein kinase inhibitor
3377	13.24	kd	CGS001-673	BRAF	RAF family			
3378	13.18	cp	BRD-K65503129	HSP90-inhibitor	HSP inhibitor		HSP90AA1, HSP90AB1	HSP inhibitor
3379	13.07	cp	BRD-K46742498	alosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
3380	13.04	cp	BRD-A31521121	methocarbamol	Muscle relaxant		CA1	Muscle relaxant
3381	13.02	cp	BRD-A17819071	gedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
3382	12.91	kd	CGS001-11329	STK38	NDR family			
3383	12.83	cp	BRD-K40645748	mefloquine	Adenosine receptor antagonist		ADORA2A, HBA1, PANX1	Adenosine receptor antagonist, Hemoglobin antagonist
3384	12.65	cp	BRD-K06388322	pramipexole	Dopamine receptor agonist		DRD3, DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3385	12.64	cp	BRD-K09991945	GSK-3-inhibitor-II	PKC inhibitor		GSK3B	PKC inhibitor
3386	12.51	cp	BRD-K15916496	clotrimazole	Cytochrome P450 inhibitor		KCNN4, CYP3A4, CYP51A1, NR1I2, NR1I3, TRPM2, TRPM4, TRPM8	Cytochrome P450 inhibitor, Imidazoline receptor ligand
3387	12.48	cp	BRD-K77793136	hydroxyfasudil	Rho associated kinase inhibitor		ROCK1, PKIA, PRKACA, ROCK2	Rho associated kinase inhibitor
3388	12.47	cp	BRD-K85242180	beta-CCP	Indoleamine 2,3-dioxygenase inhibitor		GABRA1, GABRG2, IDO1	Indoleamine 2,3-dioxygenase inhibitor
3389	12.34	cp	BRD-K40227168	vinburnine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
3390	12.16	cp	BRD-K15601958	SEW-2871	Lysophospholipid receptor agonist		S1PR1	Lysophospholipid receptor agonist
3391	12	cp	BRD-A41995253	brucine	Glycine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Glycine receptor antagonist
3392	11.97	cp	BRD-K13544237	r(-)-propylnorapomorphine	Dopamine receptor agonist		DRD2, DRD1, DRD3	Dopamine receptor agonist, TRPA1 modulator
3393	11.91	cp	BRD-K18905250	ST-91	Adrenergic receptor agonist			Adrenergic receptor agonist
3394	11.88	cc		X linked mental retardation group 2 LOF	-			
3395	11.84	cp	BRD-K67013324	luzindole	Melatonin receptor antagonist		MTNR1B, MTNR1A	Melatonin receptor antagonist
3396	11.83	cp	BRD-K48300629	zonisamide	Sodium channel blocker		CA1, CA12, CA7, SCN1A, CA10, CA11, CA13, CA14, CA2, CA3, CA4, CA5A, CA5B, CA6, CA8, CA9, CACNA1G, CACNA1H, CACNA1I, MAOA, MAOB, SCN11A, SCN1B, SCN2A, SCN2B, SCN3A, SCN3B, SCN4A, SCN4B, SCN5A, SCN9A	Sodium channel blocker, T-type calcium channel blocker
3397	11.83	cp	BRD-K28578425	cilostamide	Phosphodiesterase inhibitor		PDE3A, PDE3B	Phosphodiesterase inhibitor
3398	11.55	cp	BRD-K00959089	thenoyltrifluoroacetone	Chelating agent		CES1, PPARA, SDHA	Chelating agent
3399	11.45	cp	BRD-A49046702	SKF-89976A	GABA uptake inhibitor		SLC6A1	GABA uptake inhibitor
3400	11.44	cp	BRD-K92428153	mycophenolate-mofetil	Dehydrogenase inhibitor		IMPDH1, IMPDH2, HCAR2	Dehydrogenase inhibitor, Hydroxycarboxylic acid receptor agonist, Immunosuppressant, Inosine monophosphate dehydrogenase inhibitor, Inositol monophosphatase inhibitor
3401	11.39	cp	BRD-K70490179	rimcazole	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
3402	11.38	cp	BRD-K48935217	epothilone	Microtubule inhibitor		TUBA1A, TUBA1B, TUBA1C, TUBA3C, TUBA4A, TUBA8, TUBB, TUBB1, TUBB3, TUBB4A, TUBB4B	Microtubule inhibitor
3403	11.33	cp	BRD-K90524085	MY-5445	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor, Platelet aggregation inhibitor
3404	11.16	cp	BRD-K64935403	ebelactone-b	Lipase inhibitor		PNLIP	Lipase inhibitor
3405	11.15	cp	BRD-K80315159	DPPE	Histamine receptor antagonist		ABCB1, HRH1	Histamine receptor antagonist
3406	11.13	cp	BRD-K56047318	RHC-80267	Triacylglycerol lipase inhibitor		DAGLA, DAGLB, LIPC, LIPE, LIPG	Triacylglycerol lipase inhibitor
3407	11.07	kd	CGS001-51231	VRK3	Vaccina related kinase (VRK) family			
3408	10.79	cp	BRD-K75181824	acetyl-geranygeranyl-cysteine	Inhibitor of methyl esterification of geranylgeranylated proteins			Inhibitor of methyl esterification of geranylgeranylated proteins
3409	10.76	cp	BRD-K61401890	deguelin	NADH-ubiquinone oxidoreductase (Complex I) inhibitor		AKT1, PTGS2	NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3410	10.67	cp	BRD-K59522102	piperine	Monoamine oxidase inhibitor		MAOA, MAOB, TRPV1	Monoamine oxidase inhibitor
3411	10.61	cp	BRD-K69932463	AZD-8055	MTOR inhibitor		MTOR	MTOR inhibitor
3412	10.46	cp	BRD-K74733595	APHA-compound-8	HDAC inhibitor		HDAC8	HDAC inhibitor
3413	10.39	cp	BRD-A55756846	H-7	PKA inhibitor		PKIA, PRKACA, PRKAR1A	PKA inhibitor
3414	10.29	cp	BRD-K97764662	PD-173074	FGFR inhibitor		FGFR1, FGFR3, FGFR2, FGFR4, FLT1, FLT4, KDR, PDGFRA, PDGFRB	FGFR inhibitor, VEGFR inhibitor
3415	10	cp	BRD-A50764878	MDL-73005EF	Serotonin receptor antagonist		HTR1A	Serotonin receptor antagonist
3416	9.89	cp	BRD-K53790871	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist, Corticosteroid agonist, Immunosuppressant
3417	9.85	cp	BRD-K28346421	rifapentine	RNA polymerase inhibitor		CYP2C8, CYP3A4	RNA polymerase inhibitor
3418	9.8	cc		Androgen receptor modulator	-			
3419	9.76	cp	BRD-K08115555	tyrphostin-AG-1288	TNF production inhibitor		COMT	TNF production inhibitor
3420	9.58	cp	BRD-A74904029	EI-231	Casein kinase inhibitor		CSNK2A1, CSNK2A2, CSNK2B	Casein kinase inhibitor
3421	9.58	cp	BRD-A10903566	imiloxan	Adrenergic receptor antagonist		ADRA2B	Adrenergic receptor antagonist
3422	9.53	cp	BRD-K14221570	benzopurpurin-4b	HIV entry inhibitor			HIV entry inhibitor
3423	9.51	cp	BRD-A07395371	esmolol	Adrenergic receptor antagonist		ADRB1	Adrenergic receptor antagonist
3424	9.51	cp	BRD-A20239487	atenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3425	9.32	cp	BRD-K86204871	terconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
3426	9.31	cp	BRD-K05977823	tenovins	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor, TP53 activator
3427	9	cp	BRD-K93280214	gabazine	GABA receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRG2	GABA receptor antagonist
3428	8.53	cp	BRD-K15791587	L-733060	Tachykinin antagonist		TACR1	Tachykinin antagonist
3429	8.23	cp	BRD-A63043573	cabergoline	Dopamine receptor agonist		DRD2, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1B, ADRA1D, ADRB1, ADRB2, HTR7, PRL	Dopamine receptor agonist
3430	7.88	cp	BRD-A75935363	atracurium	Acetylcholine receptor antagonist		CHRNA2	Acetylcholine receptor antagonist
3431	7.57	cp	BRD-K88741031	methyl-2,5-dihydroxycinnamate	EGFR inhibitor		EGFR	EGFR inhibitor, Tyrosine kinase inhibitor
3432	7.5	cp	BRD-K79092138	nitrofural	Bacterial DNA inhibitor			Bacterial DNA inhibitor
3433	7.44	cp	BRD-K09132007	D-4476	TGF beta receptor inhibitor		CSNK1A1, CSNK1D, TGFB1	TGF beta receptor inhibitor
3434	7.17	cp	BRD-A55594068	vinblastine	Microtubule inhibitor		TUBB, JUN, TUBA1A, TUBD1, TUBE1, TUBG1	Microtubule inhibitor, Tubulin inhibitor
3435	6.95	cp	BRD-K63915849	AS-604850	PI3K inhibitor		PIK3CG, PIK3CA	PI3K inhibitor
3436	6.8	cp	BRD-K55191674	benzylpenicillin	Penicillin binding protein inhibitor			Penicillin binding protein inhibitor
3437	6.77	cp	BRD-K68332390	ponalrestat	Aldose reductase inhibitor		AKR1B1	Aldose reductase inhibitor
3438	6.28	cp	BRD-K73991644	isoquercetin	Aldose reductase inhibitor		AKR1B1, ACE	Aldose reductase inhibitor
3439	6.22	cp	BRD-A91866971	SQ-29548	Thromboxane receptor antagonist			Thromboxane receptor antagonist
3440	5.62	cp	BRD-A33711280	metixene	Acetylcholine receptor antagonist		CHRM5, CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor antagonist
3441	5.62	cp	BRD-K48367671	febuxostat	Xanthine oxidase inhibitor		XDH	Xanthine oxidase inhibitor
3442	5.62	cp	BRD-K82484965	carmoxirole	Dopamine receptor agonist		DRD2	Dopamine receptor agonist
3443	5.21	cp	BRD-A16694057	bisphenol-a	PPAR receptor antagonist		AR, ESR2, ESRRG, PPARG	PPAR receptor antagonist
3444	5.19	cp	BRD-K34581968	BMS-536924	IGF-1 inhibitor		IGF1R, AKT1, CCNE1, CDK2, CYP3A4, ERBB2, INSR, KDR, LCK, MAPK1, MET, PDGFRA, PDGFRB	IGF-1 inhibitor
3445	5.08	cp	BRD-K41051431	mecillinam	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3446	5	cp	BRD-K26674531	GR-235	Estrogen receptor agonist		ESR1, IKBKB, NR1H4, NR1I2, PGR	Estrogen receptor agonist, FXR antagonist, Progesterone receptor agonist
3447	4.81	cp	BRD-K03642198	AY-9944	Hedgehog pathway modulator			Hedgehog pathway modulator
3448	4.79	cc		Imidazoline ligand	-			
3449	4.03	cp	BRD-K27351809	nomegestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3450	3.95	cc		Rho associated kinase inhibitor	-			
3451	3.24	cp	BRD-A70268693	PG-9	Acetylcholine receptor agonist			Acetylcholine receptor agonist
3452	-2.41	cp	BRD-K38323065	phenacetin	Cyclooxygenase inhibitor		PTGS1	Cyclooxygenase inhibitor
3453	-4.46	cp	BRD-K87158025	benzamil	Sodium channel blocker		PKD2L1, SCNN1A, SCNN1B, SCNN1G, ASIC1, SCNN1D, SLC8A1	Sodium channel blocker
3454	-4.57	cp	BRD-K64245000	GW-4064	FXR agonist		NR1H4	FXR agonist
3455	-4.97	cp	BRD-K34508425	KUC103898N	-666			-666
3456	-5.04	cp	BRD-A10303790	talampicillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3457	-5.06	kd	CGS001-65975	STK33	CAMK-unique family			
3458	-5.57	cp	BRD-K55044200	amoxicillin	Penicillin binding protein inhibitor		SLC15A1	Penicillin binding protein inhibitor
3459	-5.67	cp	BRD-K11696279	BU-239	Imidazoline receptor agonist			Imidazoline receptor agonist, Imidazoline receptor ligand
3460	-5.7	cp	BRD-K96778649	tyrphostin-47	EGFR inhibitor		EGFR	EGFR inhibitor
3461	-5.77	cp	BRD-K63150726	JTE-907	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
3462	-6.05	cp	BRD-K71860425	CDK2-5-inhibitor	CDK inhibitor		CDK2, CDK5	CDK inhibitor
3463	-6.32	cp	BRD-K80431395	triciribine	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
3464	-6.39	cp	BRD-A41692738	TGX-221	PI3K inhibitor		PIK3CB, PIK3CD	PI3K inhibitor
3465	-6.54	cp	BRD-A38747044	KU-14R	Imidazoline receptor ligand			Imidazoline receptor ligand, Putative I3 antagonist
3466	-6.61	cp	BRD-K95739795	tetrabenazine	Vesicular monoamine transporter inhibitor		SLC18A2, DRD2, SLC18A1	Vesicular monoamine transporter inhibitor
3467	-6.68	cp	BRD-A62525898	prednisone	Glucocorticoid receptor agonist		NR3C1, HSD11B1	Glucocorticoid receptor agonist
3468	-6.96	cp	BRD-A31007383	SDZ-WAG-994	Adenosine receptor agonist		ADORA1	Adenosine receptor agonist
3469	-7.04	cp	BRD-K11801786	trimidox	Ribonucleotide reductase inhibitor		RRM1	Ribonucleotide reductase inhibitor
3470	-7.07	cc		NKL subclass homeoboxes and pseudogenes LOF	-			
3471	-7.22	cp	BRD-K44779798	miglitol	Glucosidase inhibitor		GAA, MGAM, GANAB, GANC, SLC5A4	Glucosidase inhibitor
3472	-7.37	cp	BRD-A15297126	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
3473	-7.5	cp	BRD-A75455249	kavain	Calcium channel modulator		MTOR	Calcium channel modulator, Sodium channel blocker
3474	-7.55	cp	BRD-K85925969	zalcitabine	Nucleoside reverse transcriptase inhibitor			Nucleoside reverse transcriptase inhibitor
3475	-7.56	cp	BRD-A48257147	PHCCC	Glutamate receptor agonist		GRM1, GRM4	Glutamate receptor agonist
3476	-7.72	cp	BRD-K70883034	nimetazepam	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	GABA receptor agonist
3477	-7.75	cp	BRD-K63641886	cefuroxime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3478	-8.16	cp	BRD-K23204545	busulfan	DNA inhibitor			DNA inhibitor
3479	-8.29	cp	BRD-K24859147	KIN001-242	Protein kinase inhibitor		RPS6KA3	Protein kinase inhibitor
3480	-8.36	cp	BRD-K93433262	alfacalcidol	Vitamin D receptor agonist		VDR, CYP27B1, CYP3A5	Vitamin D receptor agonist
3481	-8.74	cp	BRD-K27710560	splitomycin	SIRT inhibitor		SIRT1, SIRT2	SIRT inhibitor
3482	-8.86	kd	CGS001-5052	PRDX1	-			
3483	-9.04	cp	BRD-A35989968	megestrol	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3484	-9.09	cp	BRD-K59332007	linopirdine	Potassium channel blocker		KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
3485	-9.23	cp	BRD-K37720887	SB-525334	TGF beta receptor inhibitor		TGFBR1	TGF beta receptor inhibitor
3486	-9.3	cp	BRD-K17378184	prestwick-559	Dopamine receptor agonist		DRD3, ADRA1A, ADRA1D, ADRA2A, DRD1, DRD2, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
3487	-9.47	cp	BRD-A77722753	hydralazine	Vasodilator		AOC3, P4HA1	Vasodilator
3488	-9.47	cp	BRD-A02367930	ethinyl-estradiol	DNA directed DNA polymerase stimulant		CYP2C8, ESR1, ESR2, NR1I2	DNA directed DNA polymerase stimulant, Estrogenic component in oral contraceptives, Estrogen receptor agonist
3489	-9.57	cp	BRD-K26429091	J-104129	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
3490	-9.58	cp	BRD-A76093993	cromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
3491	-9.6	cp	BRD-K70778732	trazodone	Adrenergic receptor antagonist		HTR2A, HTR2C, SLC6A4, ADRA1A, ADRA2A, HRH1, HTR1A, HTR2B	Adrenergic receptor antagonist, Serotonin receptor antagonist, Serotonin reuptake inhibitor
3492	-9.68	cp	BRD-K74514084	pazopanib	KIT inhibitor		KDR, KIT, FLT1, FLT4, PDGFRB, PDGFRA, BRAF, CSF1R, CYP2B6, CYP2C8, CYP2E1, DDR2, FGF1, FGFR1, FGFR3, ITK, SH2B3	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
3493	-9.82	kd	CGS001-25	ABL1	Abl family			
3494	-9.89	cp	BRD-K28115081	apafant	Platelet activating factor receptor antagonist		PTAFR	Platelet activating factor receptor antagonist
3495	-10.06	cp	BRD-K95655893	MAZ-51	VEGFR inhibitor		FLT4	VEGFR inhibitor
3496	-10.11	cp	BRD-A73741725	exemestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
3497	-10.16	cp	BRD-A46179541	doxapram	Potassium channel blocker		KCNK3, KCNK9	Potassium channel blocker
3498	-10.24	cp	BRD-A62184259	cycloheximide	Protein synthesis inhibitor		GSK3B, RPL3	Protein synthesis inhibitor
3499	-10.26	kd	CGS001-10000	AKT3	Akt (Protein kinase B)			
3500	-10.52	cp	BRD-K16336526	capsaicin	TRPV agonist		TRPV1, CFTR, ENOX2	TRPV agonist
3501	-10.61	cp	BRD-K99818283	PIK-90	PI3K inhibitor			PI3K inhibitor
3502	-10.72	cp	BRD-A63836183	PD-123319	Angiotensin receptor antagonist		AGTR2	Angiotensin receptor antagonist
3503	-10.74	cp	BRD-K05434375	HA-1004	Calcium channel blocker			Calcium channel blocker
3504	-10.85	cp	BRD-K43796186	benzyl-quinazolin-4-yl-amine	EGFR inhibitor		EGFR	EGFR inhibitor
3505	-10.98	cp	BRD-K31238592	devazepide	CCK receptor antagonist		CCKAR, CCKBR, GAST	CCK receptor antagonist
3506	-11.14	cp	BRD-K32906660	bis-tyrphostin	EGFR inhibitor		DNM1, EGFR	EGFR inhibitor
3507	-11.52	cp	BRD-K67977190	eprosartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3508	-11.52	cp	BRD-K95901403	XL-147	PI3K inhibitor		PIK3CA, PIK3CD, PIK3CG	PI3K inhibitor
3509	-11.56	cp	BRD-K40213712	SAL-1	Adenosine receptor antagonist		ADORA2B, ADORA2A	Adenosine receptor antagonist
3510	-11.6	cp	BRD-K99696746	fatostatin	SREBP inhibitor		SREBF1, SREBF2	SREBP inhibitor
3511	-11.62	cp	BRD-K93332168	isocarboxazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
3512	-11.67	kd	CGS001-10589	DRAP1	-			
3513	-11.72	cp	BRD-A50737080	CGK-733	ATR kinase inhibitor		ATM, ATR	ATR kinase inhibitor
3514	-11.87	kd	CGS001-1021	CDK6	Cyclin-dependent kinases, CDK4 subfamily			
3515	-12	cp	BRD-K95763993	trapidil	PDGFR receptor inhibitor		PDGFRA	PDGFR receptor inhibitor
3516	-12.03	cp	BRD-K49890030	gavestinel	Glutamate receptor antagonist		GLRB	Glutamate receptor antagonist
3517	-12.05	cc		Cyclin dependent kinases LOF	-			
3518	-12.11	cp	BRD-A47144777	dihydro-7-desacetyldeoxygedunin	HSP inhibitor		HSP90AA1	HSP inhibitor
3519	-12.29	cc		Nucleoside reverse transcriptase inhibitor	-			
3520	-12.32	kd	CGS001-29968	PSAT1	-			
3521	-12.34	kd	CGS001-51268	PIPOX	-			
3522	-12.61	cp	BRD-K82823804	SA-792987	PKC inhibitor		WEE1	PKC inhibitor
3523	-12.64	cc		PI3K Signaling LOF	-			
3524	-12.64	cp	BRD-A11605036	thiocolchicoside	GABA receptor antagonist		GABRA1, GABRB2, GABRG2, GLRA1, GLRB	GABA receptor antagonist
3525	-12.72	cp	BRD-K00675675	CL-82198	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
3526	-12.81	cp	BRD-A20126139	medrysone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3527	-12.88	cp	BRD-K29113274	ketoconazole	Sterol demethylase inhibitor		AR, CYP19A1, CYP21A2, CYP2C19, CYP3A5, CYP3A7, KCNA10	Sterol demethylase inhibitor
3528	-12.91	cp	BRD-A85587465	bemesetron	Serotonin receptor antagonist		HTR3A, HTR3B	Serotonin receptor antagonist
3529	-13.01	cp	BRD-K15834839	lobendazole	Anthelmintic			Anthelmintic
3530	-13.03	kd	CGS001-6199	RPS6KB2	p70 subfamily			
3531	-13.06	cp	BRD-K88625236	nonoxynol-9	Membrane integrity inhibitor			Membrane integrity inhibitor
3532	-13.07	cp	BRD-A81795050	U-18666A	Oxidosqualene cyclase inhibitor			Oxidosqualene cyclase inhibitor
3533	-13.11	cp	BRD-A92439610	triamcinolone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, SERPINA6	Glucocorticoid receptor agonist
3534	-13.19	cp	BRD-A61856038	tremulacin	Lipoxygenase inhibitor			Lipoxygenase inhibitor
3535	-13.2	cp	BRD-K35573744	erbstatin-analog	EGFR inhibitor		EGFR	EGFR inhibitor
3536	-13.26	cp	BRD-A99833829	bethanechol	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist
3537	-13.26	cp	BRD-K82731415	olomoucine	CDK inhibitor		CDK1, CDK2, CDK5, MAPK1	CDK inhibitor
3538	-13.31	cp	BRD-A22684332	procaterol	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
3539	-13.32	cp	BRD-A15530910	carpindolol	Adrenergic receptor antagonist			Adrenergic receptor antagonist, Serotonin receptor antagonist
3540	-13.5	kd	CGS001-6427	SRSF2	RNA binding motif (RRM) containing			
3541	-13.52	kd	CGS001-8743	TNFSF10	CD molecules			
3542	-13.55	cp	BRD-K43290182	Ro-04-6790	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
3543	-13.57	cp	BRD-A34208323	VU-0404997-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
3544	-13.6	cp	BRD-K93658967	aloisine	CDK inhibitor		CDK2, CDK5, CDK1, CDK5R1, CFTR, PTK2B, ZAP70	CDK inhibitor, CFTR channel agonist, Glycogen synthase kinase inhibitor
3545	-13.61	kd	CGS001-79894	ZNF672	Zinc fingers, C2H2-type			
3546	-13.67	cp	BRD-A65671304	candesartan	Angiotensin receptor antagonist		AGTR1, AGTR2	Angiotensin receptor antagonist
3547	-13.68	cp	BRD-K32318651	acyclovir	DNA polymerase inhibitor		PNP	DNA polymerase inhibitor
3548	-13.78	cp	BRD-A69917777	aminopentamide	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
3549	-13.9	cp	BRD-A76279427	myriocin	Serine palmitoyltransferase inhibitor		AKT1, SPTLC1, SPTLC2, SPTLC3	Serine palmitoyltransferase inhibitor
3550	-13.97	cp	BRD-K68873215	phosphodiesterase-V-inhibitor-II	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
3551	-14.02	cp	BRD-K33312228	halometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3552	-14.08	cp	BRD-A65282128	cefazolin	Bacterial cell wall synthesis inhibitor		PON1, SLC22A8	Bacterial cell wall synthesis inhibitor
3553	-14.09	cp	BRD-K81847782	scandenin	Plant compound with antimicrobial activity			Plant compound with antimicrobial activity
3554	-14.16	cp	BRD-K12867552	THM-I-94	HDAC inhibitor		HDAC1, HDAC10, HDAC2, HDAC3, HDAC6, HDAC8	HDAC inhibitor
3555	-14.28	cp	BRD-A41722204	sulmazole	Adenosine receptor antagonist			Adenosine receptor antagonist
3556	-14.3	kd	CGS001-26523	EIF2C1	-			
3557	-14.32	cp	BRD-K17896185	FIT	Opioid receptor agonist		OPRD1	Opioid receptor agonist
3558	-14.44	kd	CGS001-5478	PPIA	Cis-trans-isomerases			
3559	-14.61	cp	BRD-A52650764	ingenol	PKC activator		PRKCD, PRKCE	PKC activator
3560	-14.64	cp	BRD-K23192422	lestaurtinib	FLT3 inhibitor		FLT3, NTRK1, JAK2, NTRK2, NTRK3	FLT3 inhibitor, Growth factor receptor inhibitor, JAK inhibitor
3561	-14.72	cp	BRD-K45435259	SCH-23390	Dopamine receptor antagonist		DRD1, DRD5, HTR2C, KCNJ4, KCNJ6	Dopamine receptor antagonist
3562	-14.76	cp	BRD-A37492983	iocetamic-acid	Radiopaque medium			Radiopaque medium
3563	-14.78	cp	BRD-K46937689	phenazone	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
3564	-14.85	cp	BRD-K09963420	saquinavir	HIV protease inhibitor		CYP3A4, CYP3A5	HIV protease inhibitor
3565	-14.92	cp	BRD-K83837640	JNJ-26854165	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, MDM2	HDAC inhibitor
3566	-14.96	cp	BRD-K79684402	RO-10-5824	Dopamine receptor agonist		DRD4	Dopamine receptor agonist
3567	-15.03	cp	BRD-K78659596	MLN-2238	Proteasome inhibitor		PSMB1	Proteasome inhibitor
3568	-15.08	cp	BRD-K02526760	QS-11	ARFGAP inhibitor		ARFGAP1	ARFGAP inhibitor
3569	-15.18	cp	BRD-A67799922	phenoxybenzamine	Adrenergic receptor antagonist		ADRA2B, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2C, ADRB2, CALM1	Adrenergic receptor antagonist
3570	-15.18	kd	CGS001-1445	CSK	Csk family			
3571	-15.2	cc		Akt Signaling LOF	-			
3572	-15.2	cc		Serotonin receptor antagonist	-			
3573	-15.2	kd	CGS001-80230	RUFY1	Zinc fingers, FYVE domain containing			
3574	-15.23	kd	CGS001-9016	SLC25A14	Mitochondrial uncoupling proteins			
3575	-15.28	cp	BRD-A42167015	carteolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
3576	-15.29	cp	BRD-K79366068	PSB-069	NTPDase inhibitor		ENTPD1, ENTPD2, ENTPD3	NTPDase inhibitor
3577	-15.34	oe	ccsbBroad304_08255	ZNF219	Zinc fingers, C2H2-type			
3578	-15.35	kd	CGS001-291	SLC25A4	Mitochondrial nucleotide transporter subfamily			
3579	-15.38	kd	CGS001-6016	RIT1	-			
3580	-15.4	cp	BRD-U94846492	quinine	Hemozoin biocrystallization inhibitor		KCNN4, ABCB1, CYP2D6, GP9, KCNB2, SLC29A4	Hemozoin biocrystallization inhibitor
3581	-15.64	cp	BRD-A34817987	itraconazole	Cytochrome P450 inhibitor		CYP3A5, CYP3A7, CYP51A1, KDR	Cytochrome P450 inhibitor
3582	-15.74	cp	BRD-A33447119	oxfendazole	Anthelmintic			Anthelmintic
3583	-15.75	kd	CGS001-9019	MPZL1	Immunoglobulin superfamily / V-set domain containing			
3584	-15.75	oe	ccsbBroad304_00658	GNG5	-			
3585	-15.84	kd	CGS001-9451	EIF2AK3	PEK subfamily			
3586	-15.86	cc		Integrin subunits alpha LOF	-			
3587	-15.99	kd	CGS001-7471	WNT1	Endogenous ligands			
3588	-16	cp	BRD-K94441233	mevastatin	HMGCR inhibitor		HMGCR	HMGCR inhibitor
3589	-16.04	cp	BRD-K73999723	telmisartan	Angiotensin receptor antagonist		AGTR1, PPARG, CYP2C19, CYP2J2, PPARA	Angiotensin receptor antagonist
3590	-16.04	cp	BRD-A50311610	meclozine	CAR agonist		NR1I3, HRH1	CAR agonist
3591	-16.05	cp	BRD-A39415247	norethisterone	Progesterone receptor agonist		PGR	Progesterone receptor agonist
3592	-16.16	cp	BRD-K06159959	CCMQ	Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites			Inhibitor of the binding of homoquinolinic acid to non-NMDA sensitive sites
3593	-16.19	cp	BRD-K77695569	tiabendazole	Angiogenesis inhibitor			Angiogenesis inhibitor
3594	-16.3	kd	CGS001-7525	YES1	Src family			
3595	-16.37	cp	BRD-K05906022	limonin	HIV protease inhibitor			HIV protease inhibitor
3596	-16.39	cp	BRD-K22227508	targinine	Nitric oxide synthase inhibitor		NOS2, NOS3	Nitric oxide synthase inhibitor
3597	-16.39	cp	BRD-K67831364	ZM-323881	VEGFR inhibitor		KDR	VEGFR inhibitor
3598	-16.41	kd	CGS001-5531	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3599	-16.48	cp	BRD-A31312900	montelukast	Leukotriene receptor antagonist		CYSLTR1, ALOX5, CYP2C8	Leukotriene receptor antagonist
3600	-16.56	kd	CGS001-545	ATR	ATR subfamily			
3601	-16.63	kd	CGS001-1212	CLTB	-			
3602	-16.64	cp	BRD-K81783531	VX-222	HCV inhibitor			HCV inhibitor
3603	-16.67	kd	CGS001-6189	RPS3A	S ribosomal proteins			
3604	-16.67	kd	CGS001-1305	COL13A1	Collagens			
3605	-16.69	kd	CGS001-1326	MAP3K8	MAPKKK:STE-unique family			
3606	-16.76	kd	CGS001-8792	TNFRSF11A	Tumour necrosis factor (TNF) receptor family			
3607	-16.77	cp	BRD-A20131130	2',5'-dideoxyadenosine	Adenylyl cyclase inhibitor			Adenylyl cyclase inhibitor
3608	-16.78	cp	BRD-K68407802	KIN001-055	EGFR inhibitor		EGFR, JAK3	EGFR inhibitor, JAK inhibitor, Leukotriene inhibitor, Mediator release inhibitor
3609	-16.83	kd	CGS001-5423	POLB	DNA polymerases			
3610	-16.91	kd	CGS001-5289	PIK3C3	Phosphatidylinositol 3-kinase family			
3611	-16.93	cp	BRD-K51066026	aminoindazole	Ionophore			Ionophore
3612	-17.06	cp	BRD-K49404994	levetiracetam	Calcium channel blocker		SV2A, CACNA1B, SCN1A	Calcium channel blocker
3613	-17.06	kd	CGS001-8535	CBX4	-			
3614	-17.17	kd	CGS001-27242	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
3615	-17.19	cp	BRD-K08132273	tyrphostin	EGFR inhibitor		ERBB2	EGFR inhibitor
3616	-17.21	kd	CGS001-4048	LTA4H	Hydrolases			
3617	-17.22	cp	BRD-K81169441	cerivastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A5	HMGCR inhibitor
3618	-17.27	kd	CGS001-4637	MYL6	EF-hand domain containing			
3619	-17.27	kd	CGS001-160851	DGKH	Pleckstrin homology (PH) domain containing			
3620	-17.31	oe	ccsbBroad304_13811	ALDH3B1	Aldehyde dehydrogenases			
3621	-17.41	kd	CGS001-310	ANXA7	Annexins			
3622	-17.46	kd	CGS001-10782	ZNF274	Zinc fingers, C2H2-type			
3623	-17.56	kd	CGS001-103	ADAR	-			
3624	-17.59	kd	CGS001-8772	FADD	-			
3625	-17.61	cp	BRD-K18523449	mestanolone	Androgenic steroid			Androgenic steroid
3626	-17.63	kd	CGS001-2512	FTL	-			
3627	-17.68	kd	CGS001-965	CD58	CD molecules			
3628	-17.72	cc		Tubulin inhibitor	-			
3629	-17.74	kd	CGS001-84775	ZNF607	Zinc fingers, C2H2-type			
3630	-17.74	kd	CGS001-10038	PARP2	Poly (ADP-ribose) polymerases			
3631	-17.77	kd	CGS001-11267	SNF8	-			
3632	-17.81	cp	BRD-K97158071	droperidol	Dopamine receptor antagonist		DRD2, ADRA1A	Dopamine receptor antagonist
3633	-17.81	cp	BRD-K57631554	aminolevulinic-acid	Oxidizing agent		ALAD	Oxidizing agent
3634	-17.84	kd	CGS001-23476	BRD4	Bromodomain kinase (BRDK) family			
3635	-17.89	cp	BRD-K96471533	nitazoxanide	Pyruvate ferredoxin oxidoreductase inhibitor			Pyruvate ferredoxin oxidoreductase inhibitor
3636	-17.89	kd	CGS001-7080	NKX2-1	Homeoboxes / ANTP class : NKL subclass			
3637	-17.99	kd	CGS001-23429	RYBP	-			
3638	-18	kd	CGS001-286530	P2RY8	GPCR / Class A : Purinergic receptors, P2Y			
3639	-18.07	kd	CGS001-8899	PRPF4B	PRP4 subfamily			
3640	-18.12	kd	CGS001-7543	ZFX	Zinc fingers, C2H2-type			
3641	-18.16	cp	BRD-K40965114	cyanopindolol	Adrenergic receptor antagonist		HTR1D	Adrenergic receptor antagonist
3642	-18.17	cp	BRD-K98763141	niflumic-acid	Cyclooxygenase inhibitor		CLCNKA, PTGS2, ANO1, CLCN1, CLCNKB, KCNQ1, PLA2G1B, PLA2G4A, PTGS1, UGT1A9	Cyclooxygenase inhibitor
3643	-18.26	cp	BRD-K59456551	methotrexate	Dihydrofolate reductase inhibitor		DHFR, AOX1, FOLR1, TYMS	Dihydrofolate reductase inhibitor
3644	-18.3	oe	ccsbBroad304_00738	HINT1	-			
3645	-18.31	cp	BRD-K28137194	loreclezole	GABA receptor agonist		GABRB2, GABRB3	GABA receptor agonist
3646	-18.31	kd	CGS001-9519	TBPL1	-			
3647	-18.31	kd	CGS001-6622	SNCA	Parkinson disease			
3648	-18.31	kd	CGS001-22796	COG2	Components of oligomeric golgi complex			
3649	-18.4	cp	BRD-K56957086	dacinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
3650	-18.4	cp	BRD-K67680372	CI-966	GAT inhibitor		SLC6A1	GAT inhibitor
3651	-18.46	kd	CGS001-4482	MSRA	-			
3652	-18.48	oe	ccsbBroad304_00778	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
3653	-18.51	kd	CGS001-262	AMD1	Decarboxylases			
3654	-18.52	cp	BRD-A55484088	BNTX	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
3655	-18.54	cp	BRD-K63151507	MNITMT	Lymphocyte inhibitor			Lymphocyte inhibitor
3656	-18.54	cp	BRD-K13819402	desoxypeganine	Acetylcholinesterase inhibitor		ACHE, MAOA	Acetylcholinesterase inhibitor, Monoamine oxidase inhibitor
3657	-18.54	cp	BRD-K37289225	clozapine	Dopamine receptor antagonist		DRD2, DRD4, ADRA1A, ADRA1B, CHRM1, DRD1, DRD3, HRH1, HRH4, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2C, HTR6, HTR7, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CALY, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD5, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
3658	-18.6	kd	CGS001-8826	IQGAP1	-			
3659	-18.65	cp	BRD-K60219430	serdemetan	MDM inhibitor		MDM2	MDM inhibitor
3660	-18.65	cp	BRD-K33860217	CP-94253	Serotonin receptor agonist		HTR1B	Serotonin receptor agonist
3661	-18.68	kd	CGS001-1646	AKR1C2	Aldo-keto reductases			
3662	-18.75	cp	BRD-A44551378	LFM-A12	EGFR inhibitor		EGFR	EGFR inhibitor
3663	-18.75	kd	CGS001-1066	CES1	Carboxylesterases			
3664	-18.79	kd	CGS001-5300	PIN1	-			
3665	-18.86	kd	CGS001-2322	FLT3	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
3666	-18.88	cp	BRD-K64994968	progesterone	Progesterone receptor agonist		PGR, CYP17A1, NR3C2, CATSPER1, CATSPER2, CATSPER3, CATSPER4, CYP2C19, ESR1, OPRK1, TRPC5	Progesterone receptor agonist
3667	-18.89	cp	BRD-A19633847	perhexiline	Carnitine palmitoyltransferase inhibitor		CPT1A, CPT2	Carnitine palmitoyltransferase inhibitor
3668	-18.95	oe	ccsbBroad304_02605	PAPD7	-			
3669	-18.98	kd	CGS001-162963	ZNF610	Zinc fingers, C2H2-type			
3670	-19.08	cp	BRD-K06198550	isorotenone	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
3671	-19.12	kd	CGS001-1025	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
3672	-19.15	cp	BRD-K70327191	benzoxiquine	Anti-infective			Anti-infective
3673	-19.19	cp	BRD-A02713983	dihydrodeoxygedunin	Growth factor receptor activator		NTRK2	Growth factor receptor activator
3674	-19.19	kd	CGS001-6915	TBXA2R	GPCR / Class A : Prostanoid receptors			
3675	-19.3	kd	CGS001-7046	TGFBR1	Type I receptor serine/threonine kinases			
3676	-19.32	cp	BRD-K99595596	salsolinol	Monoamine oxidase inhibitor		DRD2	Monoamine oxidase inhibitor, Tyrosine hydroxylase inhibitor
3677	-19.34	kd	CGS001-81034	SLC25A32	Mitochondrial nucleotide transporter subfamily			
3678	-19.4	kd	CGS001-2309	FOXO3	Forkhead boxes			
3679	-19.5	cp	BRD-K28360340	TW-37	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
3680	-19.58	oe	ccsbBroad304_00174	BRAF	RAF family			
3681	-19.66	cp	BRD-K01612348	meropenem	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
3682	-19.67	cp	BRD-K74112339	acetohydroxamic-acid	Urease inhibitor			Urease inhibitor
3683	-19.71	cp	BRD-K12219985	glipizide	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, PPARG	Sulfonylurea
3684	-19.75	kd	CGS001-3643	INSR	Type II RTKs: Insulin receptor family			
3685	-19.77	cp	BRD-A13946108	sulindac	Cyclooxygenase inhibitor		AKR1B1, PTGS1, PTGS2, MAPK3, PPARD, PTGDR2	Cyclooxygenase inhibitor
3686	-19.78	kd	CGS001-4719	NDUFS1	Mitochondrial respiratory chain complex / Complex I			
3687	-19.78	oe	ccsbBroad304_01686	TNFAIP3	OTU domain containing			
3688	-19.8	kd	CGS001-3383	ICAM1	CD molecules			
3689	-19.81	oe	ccsbBroad304_02804	KLHDC2	-			
3690	-19.86	kd	CGS001-1955	MEGF9	-			
3691	-19.9	kd	CGS001-3600	IL15	Interleukins and interleukin receptors			
3692	-19.91	kd	CGS001-55536	CDCA7L	-			
3693	-19.93	oe	ccsbBroad304_04227	SETD7	Histone methyltransferases (HMTs)			
3694	-19.96	kd	CGS001-50	ACO2	-			
3695	-20.01	oe	ccsbBroad304_01204	PIK3CD	Phosphatidylinositol kinases			
3696	-20.02	oe	ccsbBroad304_00626	GDI1	-			
3697	-20.03	oe	ccsbBroad304_02452	NXF1	-			
3698	-20.04	kd	CGS001-383	ARG1	Arginase			
3699	-20.13	cp	BRD-A57382968	piroxicam	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
3700	-20.13	kd	CGS001-3614	IMPDH1	Oxidoreductases			
3701	-20.17	cp	BRD-K13049116	BMS-754807	IGF-1 inhibitor		IGF1R, AKT1	IGF-1 inhibitor
3702	-20.2	kd	CGS001-1903	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
3703	-20.22	cp	BRD-K16478699	PLX-4720	RAF inhibitor		BRAF, KDR	RAF inhibitor
3704	-20.23	cp	BRD-A41112154	oleanolic-acid	G protein-coupled receptor agonist			G protein-coupled receptor agonist
3705	-20.29	kd	CGS001-9869	SETDB1	Histone methyltransferases (HMTs)			
3706	-20.35	kd	CGS001-4792	NFKBIA	Ankyrin repeat domain containing			
3707	-20.37	cp	BRD-A35588707	teniposide	Topoisomerase inhibitor		TOP2A, CYP3A5	Topoisomerase inhibitor
3708	-20.37	kd	CGS001-26227	PHGDH	-			
3709	-20.37	kd	CGS001-8574	AKR7A2	Aldo-keto reductases			
3710	-20.41	cp	BRD-K11558771	droxinostat	HDAC inhibitor		HDAC6, HDAC8	HDAC inhibitor
3711	-20.45	kd	CGS001-2623	GATA1	GATA zinc finger domain containing			
3712	-20.5	kd	CGS001-2356	FPGS	-			
3713	-20.5	kd	CGS001-1509	CTSD	Cathepsins			
3714	-20.51	kd	CGS001-4299	AFF1	-			
3715	-20.56	oe	ccsbBroad304_01361	RAB27A	RAB, member RAS oncogene			
3716	-20.59	kd	CGS001-7468	WHSC1	Zinc fingers, PHD-type			
3717	-20.59	kd	CGS001-51070	NOSIP	-			
3718	-20.59	kd	CGS001-84525	HOPX	Homeoboxes / PRD class			
3719	-20.61	kd	CGS001-1195	CLK1	CDC-like kinases			
3720	-20.66	kd	CGS001-284	ANGPT1	Fibrinogen C domain containing			
3721	-20.7	cp	BRD-K63828191	raloxifene	Estrogen receptor antagonist		ESR1, ESR2, ACVRL1, ENG	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
3722	-20.7	cp	BRD-K73395020	SA-1478088	-666		MMP12, MMP14, MMP2, MMP8, MMP9	-666
3723	-20.73	kd	CGS001-93349	SP140L	Zinc fingers, PHD-type			
3724	-20.74	kd	CGS001-54108	CHRAC1	-			
3725	-20.76	oe	ccsbBroad304_02425	CDIPT	-			
3726	-20.76	kd	CGS001-6098	ROS1	Type XVII RTKs: ROS receptors			
3727	-20.8	kd	CGS001-55644	OSGEP	-			
3728	-20.83	kd	CGS001-55312	RFK	-			
3729	-20.89	cp	BRD-K45158365	valsartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
3730	-20.94	oe	ccsbBroad304_05124	ZNF114	Zinc fingers, C2H2-type			
3731	-20.97	oe	ccsbBroad304_06264	GBP2	-			
3732	-20.98	kd	CGS001-8655	DYNLL1	Cytoplasmic dyneins			
3733	-21	kd	CGS001-8634	RTCD1	-			
3734	-21.01	cp	BRD-A69512159	carbidopa	Aromatic L-amino acid decarboxylase inhibitor		DDC	Aromatic L-amino acid decarboxylase inhibitor
3735	-21.03	kd	CGS001-8325	FZD8	GPCR / Class F : Frizzled receptors			
3736	-21.05	oe	ccsbBroad304_00376	CSK	Csk family			
3737	-21.11	kd	CGS001-675	BRCA2	Fanconi anemia, complementation groups			
3738	-21.15	kd	CGS001-285267	ZNF619	Zinc fingers, C2H2-type			
3739	-21.18	cp	BRD-K11663430	pyroxamide	HDAC inhibitor		HDAC1	HDAC inhibitor
3740	-21.23	kd	CGS001-2146	EZH2	Chromatin-modifying enzymes / K-methyltransferases			
3741	-21.23	kd	CGS001-2593	GAMT	-			
3742	-21.24	oe	ccsbBroad304_00129	ATP5D	ATPases / F-type			
3743	-21.28	cp	BRD-K61323504	SB-225002	CC chemokine receptor antagonist		CXCR2	CC chemokine receptor antagonist
3744	-21.31	kd	CGS001-5362	PLXNA2	Plexins			
3745	-21.39	oe	ccsbBroad304_03264	UBAP1	-			
3746	-21.39	oe	ccsbBroad304_00751	HMGB2	High-mobility group / Canonical			
3747	-21.41	kd	CGS001-9308	CD83	CD molecules			
3748	-21.46	cp	BRD-K49519144	LY-2140023	Glutamate receptor agonist		GRM3, GRM2	Glutamate receptor agonist
3749	-21.5	kd	CGS001-387509	GPR153	GPCR / Class A : Orphans			
3750	-21.54	kd	CGS001-84969	TOX2	-			
3751	-21.57	oe	ccsbBroad304_03444	PAF1	-			
3752	-21.61	kd	CGS001-3420	IDH3B	-			
3753	-21.62	oe	ccsbBroad304_07288	B4GALT4	Beta 4-glycosyltransferases			
3754	-21.68	cp	BRD-K30189597	SYK-inhibitor	SYK inhibitor		SYK	SYK inhibitor
3755	-21.73	cp	BRD-K50464341	berbamine	Calmodulin antagonist		CALM1	Calmodulin antagonist
3756	-21.75	kd	CGS001-3925	STMN1	-			
3757	-21.75	kd	CGS001-79603	CERS4	Homeoboxes / CERS class			
3758	-21.76	cp	BRD-K56745457	azauridine	Antiviral			Antiviral
3759	-21.77	kd	CGS001-89884	LHX4	Homeoboxes / LIM class			
3760	-21.77	kd	CGS001-30836	DNTTIP2	-			
3761	-21.78	oe	ccsbBroad304_00568	FHL2	-			
3762	-21.79	kd	CGS001-6617	SNAPC1	-			
3763	-21.79	kd	CGS001-1080	CFTR	ATP binding cassette transporters / subfamily C			
3764	-21.83	kd	CGS001-79006	METRN	-			
3765	-21.86	cp	BRD-K06014311	DH-97	Melatonin receptor antagonist		MTNR1B	Melatonin receptor antagonist
3766	-21.87	kd	CGS001-3489	IGFBP6	insulin-like growth factor (IGF) binding proteins			
3767	-21.89	kd	CGS001-55617	TASP1	Glycosylasparaginase precursor			
3768	-21.93	cp	BRD-K99107520	felbamate	Glutamate receptor antagonist		GRIN2A, GRIN2B, GRIN3A	Glutamate receptor antagonist
3769	-21.94	cp	BRD-K97309399	thiothixene	Dopamine receptor antagonist		HTR2A, DRD1, DRD2, HRH1	Dopamine receptor antagonist
3770	-21.99	cp	BRD-K15563106	phloretin	Sodium/glucose cotransporter inhibitor		AQP9, CLCN3, SLC23A1	Sodium/glucose cotransporter inhibitor
3771	-21.99	kd	CGS001-10673	TNFSF13B	CD molecules			
3772	-21.99	kd	CGS001-5925	RB1	Endogenous ligands			
3773	-22.01	oe	ccsbBroad304_06206	FGA	Endogenous ligands			
3774	-22.02	kd	CGS001-1843	DUSP1	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3775	-22.03	kd	CGS001-4698	NDUFA5	Mitochondrial respiratory chain complex / Complex I			
3776	-22.04	cp	BRD-A93255169	thalidomide	TNF production inhibitor		TNF, CRBN, CYP1A2, CYP2B6, CYP2C19, CYP3A5, FGFR2, NFKB1, ORM1, ORM2, PTGS2	TNF production inhibitor
3777	-22.06	cp	BRD-K51541829	RO-25-6981	Ionotropic glutamate receptor antagonist		GRIN2B, SLC18A2	Ionotropic glutamate receptor antagonist, Monamine transporter modulator
3778	-22.07	cp	BRD-K63533170	AM-630	Cannabinoid receptor antagonist		CNR2, CNR1	Cannabinoid receptor antagonist
3779	-22.09	kd	CGS001-26001	RNF167	RING-type (C3HC4) zinc fingers			
3780	-22.1	oe	ccsbBroad304_00879	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
3781	-22.13	kd	CGS001-58499	ZNF462	Zinc fingers, C2H2-type			
3782	-22.14	kd	CGS001-6810	STX4	-			
3783	-22.2	oe	ccsbBroad304_02681	MGLL	Endocannabinoid turnover			
3784	-22.2	kd	CGS001-54106	TLR9	Toll-like receptor family			
3785	-22.21	kd	CGS001-55890	GPRC5C	GPCR / Class C : Orphans			
3786	-22.22	kd	CGS001-10671	DCTN6	-			
3787	-22.23	kd	CGS001-5411	PNN	-			
3788	-22.25	kd	CGS001-11198	SUPT16H	-			
3789	-22.25	kd	CGS001-9886	RHOBTB1	BTB/POZ domain containing			
3790	-22.28	oe	ccsbBroad304_00020	ACY1	-			
3791	-22.29	cp	BRD-K52751261	TAK-715	p38 MAPK inhibitor		MAPK14, TNF	p38 MAPK inhibitor
3792	-22.29	kd	CGS001-112812	FDX1L	-			
3793	-22.31	kd	CGS001-23743	BHMT2	-			
3794	-22.32	oe	ccsbBroad304_06058	CSNK2B	Casein kinase 2 (CK2) family			
3795	-22.32	cp	BRD-A38749782	fludrocortisone	Glucocorticoid receptor agonist		NR3C2, AR, NR3C1	Glucocorticoid receptor agonist, Mineralocorticoid receptor agonist
3796	-22.32	cp	BRD-A09533288	verapamil	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1G, CACNA1S, CACNA1A, CACNA1B, CACNA1F, CACNA1I, CACNB1, CACNB2, CACNB3, CACNB4, CYP2C8, CYP2E1, CYP3A4, CYP3A5, CYP3A7, DRD2, KCNA10, KCNA7, KCNH2, KCNJ11, NALCN, SCN5A, SLC29A4, SLC6A4	Calcium channel blocker
3797	-22.34	oe	ccsbBroad304_01936	RAE1	WD repeat domain containing			
3798	-22.36	kd	CGS001-5604	MAP2K1	MAPKK:STE7 family			
3799	-22.36	kd	CGS001-23658	LSM5	-			
3800	-22.39	oe	ccsbBroad304_02538	RUVBL2	ATPases / AAA-type			
3801	-22.4	cp	BRD-K81128206	edrophonium	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
3802	-22.4	kd	CGS001-4763	NF1	-			
3803	-22.41	kd	CGS001-51026	GOLT1B	-			
3804	-22.42	cp	BRD-A41941932	vitexin	Antioxidant			Antioxidant
3805	-22.45	oe	ccsbBroad304_01146	PARN	-			
3806	-22.45	kd	CGS001-25948	KBTBD2	BTB/POZ domain containing			
3807	-22.47	kd	CGS001-163049	ZNF791	Zinc fingers, C2H2-type			
3808	-22.49	oe	ccsbBroad304_07500	PJA2	RING-type (C3HC4) zinc fingers			
3809	-22.49	kd	CGS001-55500	ETNK1	-			
3810	-22.53	cp	BRD-K01648091	LE-300	Dopamine receptor antagonist		DRD5, DRD1, HTR2A	Dopamine receptor antagonist
3811	-22.54	oe	ccsbBroad304_09881	RFX6	-			
3812	-22.56	oe	ccsbBroad304_01026	MNAT1	RING-type (C3HC4) zinc fingers			
3813	-22.56	cp	BRD-K93331255	lypressin	Vasopressin receptor agonist		AVPR1A, AVPR1B, AVPR2	Vasopressin receptor agonist
3814	-22.57	cp	BRD-A92177080	betamethasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
3815	-22.58	oe	ccsbBroad304_10487	BPHL	-			
3816	-22.59	kd	CGS001-116985	ARAP1	Ankyrin repeat domain containing			
3817	-22.6	oe	ccsbBroad304_01685	TNFAIP1	BTB/POZ domain containing			
3818	-22.63	kd	CGS001-4216	MAP3K4	MAPKKK:STE11 family			
3819	-22.69	cp	BRD-K07117950	imperatorin	CDK inhibitor		ACHE, HTR7	CDK inhibitor
3820	-22.69	kd	CGS001-8836	GGH	Gamma-glutamyl hydrolase			
3821	-22.71	cp	BRD-K57569181	pentoxifylline	Phosphodiesterase inhibitor		TNF, ACHE, ADORA1, ADORA2A, ADRA2B, CHIA, NT5E, PDE4A, PDE4B, PDE5A	Phosphodiesterase inhibitor
3822	-22.73	kd	CGS001-89849	ATG16L2	WD repeat domain containing			
3823	-22.74	kd	CGS001-4217	MAP3K5	MAPKKK:STE11 family			
3824	-22.81	cp	BRD-K15196155	IBC-293	Hydroxycarboxylic acid receptor agonist		HCAR3	Hydroxycarboxylic acid receptor agonist
3825	-22.82	kd	CGS001-384	ARG2	Arginase			
3826	-22.84	cp	BRD-K62363391	dapsone	Bacterial antifolate		DHFR	Bacterial antifolate
3827	-22.86	oe	ccsbBroad304_05923	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
3828	-22.88	kd	CGS001-4092	SMAD7	SMADs			
3829	-22.88	kd	CGS001-9520	NPEPPS	Aminopeptidase N			
3830	-22.9	kd	CGS001-475	ATOX1	-			
3831	-22.92	cp	BRD-A80793822	pemoline	Dopamine receptor agonist			Dopamine receptor agonist
3832	-22.94	oe	ccsbBroad304_07768	NISCH	-			
3833	-22.95	kd	CGS001-25989	ULK3	Unc-51-like kinase (ULK) family			
3834	-22.98	kd	CGS001-64175	LEPRE1	-			
3835	-22.99	kd	CGS001-5971	RELB	NFkappaB transcription factor family			
3836	-23.01	kd	CGS001-206358	SLC36A1	SLC36 family of proton-coupled amino acid transporters			
3837	-23.03	kd	CGS001-25937	WWTR1	Hippo Signaling			
3838	-23.04	oe	ccsbBroad304_00498	ELK1	ETS Transcription Factors			
3839	-23.04	kd	CGS001-3248	HPGD	Prostaglandin synthases			
3840	-23.04	kd	CGS001-150	ADRA2A	GPCR / Class A : Adrenoceptors : alpha			
3841	-23.06	kd	CGS001-3608	ILF2	-			
3842	-23.11	kd	CGS001-50813	COPS7A	-			
3843	-23.17	kd	CGS001-5595	MAPK3	MAPK:ERK subfamily			
3844	-23.18	oe	ccsbBroad304_06349	HAGH	-			
3845	-23.21	kd	CGS001-7855	FZD5	GPCR / Class F : Frizzled receptors			
3846	-23.22	cp	BRD-K78692225	leflunomide	Dihydroorotate dehydrogenase inhibitor		DHODH, AHR, CYP2C19, JAK3, PTK2B, STAT6	Dihydroorotate dehydrogenase inhibitor, PDGFR receptor inhibitor
3847	-23.25	kd	CGS001-5530	PPP3CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
3848	-23.26	kd	CGS001-6715	SRD5A1	-			
3849	-23.26	kd	CGS001-8837	CFLAR	Endogenous ligands			
3850	-23.28	kd	CGS001-5744	PTHLH	Endogenous ligands			
3851	-23.28	kd	CGS001-4234	METTL1	-			
3852	-23.32	kd	CGS001-857	CAV1	-			
3853	-23.35	cp	BRD-A42423104	benproperine	Antitussive			Antitussive
3854	-23.36	cp	BRD-K89375097	pirenzepine	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Acetylcholine receptor antagonist
3855	-23.36	kd	CGS001-983	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
3856	-23.4	kd	CGS001-10381	TUBB3	Tubulins			
3857	-23.41	oe	ccsbBroad304_06993	SRD5A1	-			
3858	-23.43	kd	CGS001-83694	RPS6KL1	RSKL family			
3859	-23.43	kd	CGS001-9374	PPT2	-			
3860	-23.45	kd	CGS001-5048	PAFAH1B1	WD repeat domain containing			
3861	-23.45	kd	CGS001-56675	NRIP3	-			
3862	-23.51	cp	BRD-K52522949	NCH-51	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
3863	-23.54	kd	CGS001-4694	NDUFA1	Mitochondrial respiratory chain complex / Complex I			
3864	-23.56	cp	BRD-K50398167	meclofenamic-acid	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, CNR1, KCNQ2, KCNQ3	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
3865	-23.6	oe	ccsbBroad304_13998	PDXK	-			
3866	-23.61	kd	CGS001-2950	GSTP1	Glutathione S-transferases			
3867	-23.63	kd	CGS001-641	BLM	-			
3868	-23.64	kd	CGS001-387129	NPSR1	GPCR / Class A : Neuropeptide receptors : S			
3869	-23.64	kd	CGS001-55699	IARS2	Aminoacyl tRNA synthetases / Class I			
3870	-23.67	kd	CGS001-9791	PTDSS1	-			
3871	-23.69	kd	CGS001-5829	PXN	-			
3872	-23.69	kd	CGS001-23365	ARHGEF12	Rho guanine nucleotide exchange factors			
3873	-23.69	kd	CGS001-152	ADRA2C	GPCR / Class A : Adrenoceptors : alpha			
3874	-23.71	kd	CGS001-1949	EFNB3	Ephrins			
3875	-23.71	oe	ccsbBroad304_05930	CAMK2D	CAMK2 family			
3876	-23.72	cp	BRD-K26548821	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
3877	-23.72	kd	CGS001-10398	MYL9	EF-hand domain containing			
3878	-23.74	cp	BRD-K88871508	lisuride	Dopamine receptor agonist		DRD2, HTR2B, HTR2C, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, ADRA1A, HRH1, HTR6	Dopamine receptor agonist
3879	-23.74	cp	BRD-K57304726	PRE-084	Sigma receptor agonist		SIGMAR1	Sigma receptor agonist
3880	-23.77	kd	CGS001-1861	TOR1A	-			
3881	-23.8	kd	CGS001-6929	TCF3	Basic helix-loop-helix proteins			
3882	-23.82	cp	BRD-A81233518	glycopyrrolate	Acetylcholine receptor antagonist		CHRM1, CHRM3, CHRM2, CHRM4, CHRM5	Acetylcholine receptor antagonist
3883	-23.85	kd	CGS001-10488	CREB3	basic leucine zipper proteins			
3884	-23.87	cp	BRD-K69763916	LY-341495	Glutamate receptor antagonist		GRM2, GRM3	Glutamate receptor antagonist
3885	-23.95	cp	BRD-K82036761	sertraline	Serotonin receptor antagonist		SLC6A4, CYP2C19, SLC6A3	Serotonin receptor antagonist
3886	-23.98	kd	CGS001-231	AKR1B1	Aldo-keto reductases			
3887	-24.02	kd	CGS001-6258	RXRG	Retinoid X receptors			
3888	-24.03	kd	CGS001-3479	IGF1	Endogenous ligands			
3889	-24.04	cp	BRD-A84189516	baccatin-III	Paclitaxel precursor			Paclitaxel precursor
3890	-24.06	kd	CGS001-23030	KDM4B	Histone demethylases			
3891	-24.07	cp	BRD-K37194137	III606050	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
3892	-24.07	kd	CGS001-578	BAK1	-			
3893	-24.08	oe	ccsbBroad304_04405	KISS1R	GPCR / Class A : RF amide peptide receptors			
3894	-24.09	kd	CGS001-246778	IL27	Interleukins and interleukin receptors			
3895	-24.09	kd	CGS001-8449	DHX16	DEAH-boxes			
3896	-24.09	kd	CGS001-597	BCL2A1	-			
3897	-24.13	kd	CGS001-84873	GPR128	Adhesion Class GPCRs			
3898	-24.15	oe	ccsbBroad304_01948	GAS7	-			
3899	-24.16	kd	CGS001-6990	DYNLT3	Cytoplasmic dyneins			
3900	-24.17	kd	CGS001-7032	TFF2	-			
3901	-24.17	kd	CGS001-6648	SOD2	-			
3902	-24.18	oe	ccsbBroad304_08325	LIPT1	-			
3903	-24.19	oe	ccsbBroad304_09420	RASGRP4	EF-hand domain containing			
3904	-24.19	kd	CGS001-1362	CPD	Carboxypeptidase A			
3905	-24.22	kd	CGS001-55937	APOM	Apolipoproteins			
3906	-24.23	cc		Nucleoporin LOF	-			
3907	-24.24	cp	BRD-K08996725	zolantidine	Histamine receptor antagonist			Histamine receptor antagonist
3908	-24.28	cp	BRD-K17497770	butein	EGFR inhibitor		ACE, CXCL8, IL6, SIRT1, SRD5A1, SRD5A2, TNF	EGFR inhibitor, SRC inhibitor
3909	-24.29	oe	ccsbBroad304_02534	UTP14A	-			
3910	-24.29	cp	BRD-K49671696	ketanserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, DRD1, DRD5, HTR1A, HTR1B, HTR1D, HTR2B, HTR5A, HTR7, SLC18A1, SLC18A2	Serotonin receptor antagonist
3911	-24.31	oe	ccsbBroad304_00670	GPR4	GPCR / Class A : Orphans			
3912	-24.31	oe	ccsbBroad304_03386	SPA17	-			
3913	-24.31	kd	CGS001-4793	NFKBIB	Ankyrin repeat domain containing			
3914	-24.33	cp	BRD-A34255068	rolipram	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D, PDE4C, PDE5A	Phosphodiesterase inhibitor, Interleukin receptor antagonist
3915	-24.33	kd	CGS001-6389	SDHA	Mitochondrial respiratory chain complex			
3916	-24.37	cp	BRD-K96670504	lonidamine	Glucokinase inhibitor		GCK	Glucokinase inhibitor
3917	-24.37	cp	BRD-A27554692	altrenogest	Progestogen hormone		PGR	Progestogen hormone
3918	-24.39	oe	ccsbBroad304_03937	MLST8	WD repeat domain containing			
3919	-24.39	kd	CGS001-7780	SLC30A2	SLC30 zinc transporter family			
3920	-24.39	kd	CGS001-5062	PAK2	PAKA subfamily			
3921	-24.44	kd	CGS001-5451	POU2F1	Homeoboxes / POU class			
3922	-24.49	kd	CGS001-9134	CCNE2	-			
3923	-24.5	kd	CGS001-1958	EGR1	Zinc fingers, C2H2-type			
3924	-24.52	oe	ccsbBroad304_01822	ZNF227	Zinc fingers, C2H2-type			
3925	-24.57	oe	ccsbBroad304_13813	ARAF	RAF family			
3926	-24.57	cp	BRD-K68132782	terbinafine	Fungal squalene epoxidase inhibitor		CYP2C19, CYP2C8, SQLE	Fungal squalene epoxidase inhibitor
3927	-24.57	kd	CGS001-10493	VAT1	-			
3928	-24.58	kd	CGS001-10131	TRAP1	Heat shock proteins / HSPC			
3929	-24.59	oe	ccsbBroad304_00472	EBF1	-			
3930	-24.6	kd	CGS001-9276	COPB2	WD repeat domain containing			
3931	-24.61	kd	CGS001-8800	PEX11A	-			
3932	-24.62	kd	CGS001-162	AP1B1	-			
3933	-24.65	cp	BRD-A70514680	articaine	Local anesthetic			Local anesthetic
3934	-24.65	kd	CGS001-345611	IRGM	-			
3935	-24.66	kd	CGS001-7695	ZNF136	Zinc fingers, C2H2-type			
3936	-24.67	cp	BRD-K80672993	M2-PK-activator	-666		PKM	-666
3937	-24.69	oe	ccsbBroad304_06149	EIF4B	RNA binding motif (RRM) containing			
3938	-24.69	kd	CGS001-222611	GPR111	Adhesion Class GPCRs			
3939	-24.7	oe	ccsbBroad304_06238	GABBR1	GABA receptors			
3940	-24.7	oe	ccsbBroad304_03497	TXNL4B	-			
3941	-24.7	kd	CGS001-10406	WFDC2	WAP four-disulfide core domain containing			
3942	-24.7	kd	CGS001-6210	RPS15A	S ribosomal proteins			
3943	-24.7	kd	CGS001-221391	OPN5	GPCR / Class A : Opsin receptors			
3944	-24.71	kd	CGS001-54788	DNAJB12	Heat shock proteins / DNAJ (HSP40)			
3945	-24.72	oe	ccsbBroad304_00993	MDM4	-			
3946	-24.75	kd	CGS001-9475	ROCK2	Pleckstrin homology (PH) domain containing			
3947	-24.75	kd	CGS001-4077	NBR1	-			
3948	-24.76	kd	CGS001-2925	GRPR	GPCR / Class A : Bombesin receptors			
3949	-24.78	cp	BRD-K13169950	NSC-3852	HDAC inhibitor		HDAC1	HDAC inhibitor
3950	-24.78	kd	CGS001-51079	NDUFA13	Mitochondrial respiratory chain complex / Complex I			
3951	-24.79	kd	CGS001-7374	UNG	-			
3952	-24.79	kd	CGS001-5737	PTGFR	GPCR / Class A : Prostanoid receptors			
3953	-24.81	kd	CGS001-5566	PRKACA	Protein kinase A			
3954	-24.82	oe	ccsbBroad304_05787	ADRBK1	BARK/GRK2 subfamily			
3955	-24.83	oe	ccsbBroad304_01378	RASA1	Pleckstrin homology (PH) domain containing			
3956	-24.84	cp	BRD-A80017228	bendroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A3, CA1, CA2, CA4, KCNMA1, SLC12A1	Sodium/potassium/chloride transporter inhibitor
3957	-24.88	oe	ccsbBroad304_06130	DUSP4	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3958	-24.9	kd	CGS001-10474	TADA3	-			
3959	-24.9	kd	CGS001-27198	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
3960	-24.92	oe	ccsbBroad304_07569	TRIB1	Trbl family			
3961	-24.94	oe	ccsbBroad304_09993	VN1R4	GPCR / Unclassified : Vomeronasal receptors, type 1			
3962	-24.94	oe	ccsbBroad304_05485	ZNF677	Zinc fingers, C2H2-type			
3963	-24.94	kd	CGS001-4851	NOTCH1	Ankyrin repeat domain containing			
3964	-24.94	kd	CGS001-1844	DUSP2	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
3965	-24.95	kd	CGS001-23386	NUDCD3	-			
3966	-24.96	kd	CGS001-7187	TRAF3	-			
3967	-24.97	cp	BRD-K25875056	SC-9	Protein tyrosine kinase activator			Protein tyrosine kinase activator
3968	-24.98	cp	BRD-K13514097	everolimus	MTOR inhibitor		MTOR, CYP3A5, FKBP1A	MTOR inhibitor
3969	-25.01	kd	CGS001-3373	HYAL1	-			
3970	-25.01	kd	CGS001-116113	FOXP4	Forkhead boxes			
3971	-25.02	kd	CGS001-3675	ITGA3	Integrins			
3972	-25.08	kd	CGS001-11014	KDELR2	-			
3973	-25.09	kd	CGS001-90233	ZNF551	Zinc fingers, C2H2-type			
3974	-25.14	kd	CGS001-5438	POLR2I	RNA polymerase subunits			
3975	-25.14	kd	CGS001-51290	ERGIC2	-			
3976	-25.15	oe	ccsbBroad304_08802	ELAC2	-			
3977	-25.15	kd	CGS001-29082	CHMP4A	Charged multivesicular body proteins			
3978	-25.15	cp	BRD-K05977355	fluconazole	Sterol demethylase inhibitor		CYP3A5, CYP3A7	Sterol demethylase inhibitor
3979	-25.18	cp	BRD-K30480208	torasemide	Electrolyte reabsorption inhibitor		SLC12A1, CYP2C8, SLC12A2	Electrolyte reabsorption inhibitor, Thromboxane receptor antagonist
3980	-25.18	kd	CGS001-8444	DYRK3	Dyrk2 subfamily			
3981	-25.18	kd	CGS001-25819	CCRN4L	-			
3982	-25.18	kd	CGS001-23786	BCL2L13	-			
3983	-25.2	kd	CGS001-8576	STK16	NAK family			
3984	-25.2	kd	CGS001-4121	MAN1A1	-			
3985	-25.22	kd	CGS001-1604	CD55	CD molecules			
3986	-25.28	kd	CGS001-1407	CRY1	-			
3987	-25.29	oe	ccsbBroad304_01320	PSMD4	Proteasome (prosome, macropain) subunits			
3988	-25.31	kd	CGS001-4172	MCM3	-			
3989	-25.31	kd	CGS001-8520	HAT1	Histone acetyltransferases (HATs)			
3990	-25.32	oe	ccsbBroad304_07466	VGLL4	-			
3991	-25.32	kd	CGS001-10365	KLF2	Kruppel-like transcription factors			
3992	-25.33	kd	CGS001-6928	HNF1B	Homeoboxes / HNF class			
3993	-25.33	kd	CGS001-223	ALDH9A1	Aldehyde dehydrogenases			
3994	-25.34	oe	ccsbBroad304_04189	FBXO11	Protein arginine N-methyltransferases			
3995	-25.35	oe	ccsbBroad304_01676	TLE1	WD repeat domain containing			
3996	-25.36	kd	CGS001-9868	TOMM70A	Tetratricopeptide (TTC) repeat domain containing			
3997	-25.39	kd	CGS001-5435	POLR2F	RNA polymerase subunits			
3998	-25.39	kd	CGS001-79837	PIP4K2C	1-phosphatidylinositol-5-phosphate 4-kinase family			
3999	-25.42	kd	CGS001-874	CBR3	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4000	-25.47	cp	BRD-K01292756	pimozide	Dopamine receptor antagonist		DRD2, DRD3, CACNA1I, CALM1, HRH1, HTR1A, HTR2A, KCNA10, KCNH2	Dopamine receptor antagonist
4001	-25.5	cp	BRD-K83637872	SANT-1	Smoothened receptor antagonist		DHH, IHH, PTCH1, SMO	Smoothened receptor antagonist
4002	-25.51	cc		Protein phosphatase catalytic subunits LOF	-			
4003	-25.53	oe	ccsbBroad304_06828	PYCR1	-			
4004	-25.55	oe	ccsbBroad304_01363	RABGGTA	Prenyltransferase alpha subunit repeat containing			
4005	-25.55	oe	ccsbBroad304_01101	NME1	-			
4006	-25.55	kd	CGS001-4850	CNOT4	RNA binding motif (RRM) containing			
4007	-25.56	cp	BRD-K14807180	SB-221284	Serotonin receptor antagonist		HTR2B, HTR2C, HTR2A	Serotonin receptor antagonist
4008	-25.57	oe	ccsbBroad304_01309	PSMB1	Proteasome subunits			
4009	-25.57	kd	CGS001-2852	GPER	-			
4010	-25.63	kd	CGS001-64077	LHPP	-			
4011	-25.64	kd	CGS001-7569	ZNF182	Zinc fingers, C2H2-type			
4012	-25.64	kd	CGS001-256281	NUDT14	Nudix motif containing			
4013	-25.64	oe	ccsbBroad304_02408	HMG20B	High mobility group / Non-canonical			
4014	-25.65	cp	BRD-K18787491	U-0126	MEK inhibitor		AKT1, CHEK1, GSK3B, JAK2, LCK, MAP2K1, MAP2K2, MAP2K7, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor
4015	-25.66	oe	ccsbBroad304_04732	ZNF488	Zinc fingers, C2H2-type			
4016	-25.66	kd	CGS001-7358	UGDH	-			
4017	-25.69	oe	ccsbBroad304_06253	GALT	-			
4018	-25.71	cp	BRD-M30523314	vinorelbine	Tubulin inhibitor		TUBB	Tubulin inhibitor
4019	-25.71	kd	CGS001-55031	USP47	Ubiquitin-specific peptidases			
4020	-25.71	kd	CGS001-51655	RASD1	-			
4021	-25.71	kd	CGS001-3726	JUNB	basic leucine zipper proteins			
4022	-25.73	kd	CGS001-7423	VEGFB	-			
4023	-25.74	cp	BRD-K86465814	HO-013	PPAR receptor agonist		PPARG	PPAR receptor agonist
4024	-25.74	kd	CGS001-58472	SQRDL	-			
4025	-25.77	kd	CGS001-59350	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
4026	-25.77	kd	CGS001-3589	IL11	Endogenous ligands			
4027	-25.78	kd	CGS001-2033	EP300	Chromatin-modifying enzymes / K-acetyltransferases			
4028	-25.78	kd	CGS001-831	CAST	-			
4029	-25.79	kd	CGS001-23530	NNT	-			
4030	-25.81	oe	ccsbBroad304_01255	PPM1B	Serine/threonine phosphatases / Protein phosphatases, Mg2+/Mn2+ dependent			
4031	-25.82	kd	CGS001-9181	ARHGEF2	Rho guanine nucleotide exchange factors			
4032	-25.89	oe	ccsbBroad304_02582	UQCR11	Mitochondrial respiratory chain complex / Complex III			
4033	-25.89	kd	CGS001-6118	RPA2	-			
4034	-25.9	oe	ccsbBroad304_08010	FBXO5	F-boxes / other			
4035	-25.95	oe	ccsbBroad304_02044	EIF2S2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4036	-25.95	kd	CGS001-154197	PNLDC1	-			
4037	-25.98	oe	ccsbBroad304_07172	ZNF195	Zinc fingers, C2H2-type			
4038	-25.98	oe	ccsbBroad304_01375	RARA	Retinoic acid receptors			
4039	-25.98	oe	ccsbBroad304_00030	ADORA2B	GPCR / Class A : Adenosine receptors			
4040	-25.98	cp	BRD-K59037100	oxybenzone	Lipase inhibitor		LIPE	Lipase inhibitor
4041	-25.98	kd	CGS001-56956	LHX9	Homeoboxes / LIM class			
4042	-26.01	kd	CGS001-55657	ZNF692	Zinc fingers, C2H2-type			
4043	-26.03	kd	CGS001-53340	SPA17	-			
4044	-26.04	kd	CGS001-10610	ST6GALNAC2	Sialyltransferases			
4045	-26.06	oe	ccsbBroad304_05821	ANXA1	Annexins			
4046	-26.06	kd	CGS001-8848	TSC22D1	-			
4047	-26.07	kd	CGS001-2010	EMD	-			
4048	-26.07	cp	BRD-K27141178	SB-203186	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
4049	-26.08	oe	ccsbBroad304_01624	SUPV3L1	-			
4050	-26.09	kd	CGS001-9070	ASH2L	Zinc fingers, PHD-type			
4051	-26.11	oe	ccsbBroad304_05876	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
4052	-26.11	kd	CGS001-8243	SMC1A	Structural maintenance of chromosomes proteins			
4053	-26.12	oe	ccsbBroad304_07676	PLK2	Polo-like kinase (PLK) family			
4054	-26.14	oe	ccsbBroad304_04616	ORMDL3	-			
4055	-26.15	oe	ccsbBroad304_02934	B3GAT3	Beta-1,3-glucuronyltransferases			
4056	-26.16	cp	BRD-A71262238	nafadotride	Dopamine receptor antagonist		DRD3, DRD2, HTR1A	Dopamine receptor antagonist
4057	-26.17	kd	CGS001-54850	FBXL12	F-boxes / Leucine-rich repeats			
4058	-26.18	kd	CGS001-5832	ALDH18A1	Aldehyde dehydrogenases			
4059	-26.19	kd	CGS001-3460	IFNGR2	Interferon receptor family			
4060	-26.2	kd	CGS001-25865	PRKD2	Pleckstrin homology (PH) domain containing			
4061	-26.2	kd	CGS001-3613	IMPA2	Inositol monophosphatase			
4062	-26.21	kd	CGS001-3122	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
4063	-26.21	kd	CGS001-760	CA2	Carbonic anhydrases			
4064	-26.23	kd	CGS001-9063	PIAS2	Zinc fingers, MIZ-type			
4065	-26.23	kd	CGS001-84333	PCGF5	Polycomb group ring fingers			
4066	-26.25	oe	ccsbBroad304_00963	SMAD5	SMADs			
4067	-26.25	cp	BRD-K45117373	Y-26763	Potassium channel activator		ABCC9, KCNJ8	Potassium channel activator
4068	-26.25	kd	CGS001-901	CCNG2	-			
4069	-26.26	cc		HOXL subclass homeoboxes LOF	-			
4070	-26.28	cc		Progesterone receptor agonist	-			
4071	-26.32	kd	CGS001-10771	ZMYND11	Zinc fingers, MYND-type			
4072	-26.32	kd	CGS001-6182	MRPL12	Mitochondrial ribosomal proteins / large subunits			
4073	-26.34	oe	ccsbBroad304_06847	RBBP4	WD repeat domain containing			
4074	-26.34	oe	ccsbBroad304_01071	NDUFB5	Mitochondrial respiratory chain complex / Complex I			
4075	-26.34	oe	ccsbBroad304_06294	GNAZ	-			
4076	-26.36	kd	CGS001-4706	NDUFAB1	Mitochondrial respiratory chain complex / Complex I			
4077	-26.4	kd	CGS001-6632	SNRPD1	-			
4078	-26.41	oe	ccsbBroad304_05782	ADORA2A	GPCR / Class A : Adenosine receptors			
4079	-26.43	oe	ccsbBroad304_01242	POLR2I	RNA polymerase subunits			
4080	-26.43	oe	ccsbBroad304_06438	IL2RB	IL-2 receptor family			
4081	-26.46	kd	CGS001-2100	ESR2	Estrogen receptors			
4082	-26.49	kd	CGS001-23650	TRIM29	-			
4083	-26.51	kd	CGS001-2778	GNAS	-			
4084	-26.52	kd	CGS001-2101	ESRRA	Estrogen-related receptors			
4085	-26.55	oe	ccsbBroad304_01396	RGS4	Regulators of G-protein signaling			
4086	-26.56	kd	CGS001-1468	SLC25A10	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
4087	-26.57	kd	CGS001-2247	FGF2	Endogenous ligands			
4088	-26.6	kd	CGS001-81577	GFOD2	-			
4089	-26.62	kd	CGS001-5516	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4090	-26.64	kd	CGS001-2230	FDX1	-			
4091	-26.66	kd	CGS001-92595	ZNF764	Zinc fingers, C2H2-type			
4092	-26.67	kd	CGS001-1962	EHHADH	-			
4093	-26.72	kd	CGS001-59343	SENP2	-			
4094	-26.74	oe	ccsbBroad304_01052	MYB	-			
4095	-26.77	oe	ccsbBroad304_06136	ECHS1	-			
4096	-26.79	kd	CGS001-1960	EGR3	Zinc fingers, C2H2-type			
4097	-26.8	oe	ccsbBroad304_00268	CD81	CD molecules			
4098	-26.82	kd	CGS001-55012	PPP2R3C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4099	-26.83	kd	CGS001-9014	TAF1B	-			
4100	-26.84	kd	CGS001-203	AK1	Adenylate kinases			
4101	-26.87	oe	ccsbBroad304_04018	VKORC1	Oxidoreductases			
4102	-26.89	kd	CGS001-2553	GABPB1	Ankyrin repeat domain containing			
4103	-26.91	kd	CGS001-4173	MCM4	-			
4104	-26.91	kd	CGS001-4023	LPL	-			
4105	-26.93	kd	CGS001-79094	CHAC1	-			
4106	-26.93	oe	ccsbBroad304_01265	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
4107	-26.95	kd	CGS001-9512	PMPCB	-			
4108	-26.95	kd	CGS001-5605	MAP2K2	MAPKK:STE7 family			
4109	-26.96	kd	CGS001-221895	JAZF1	Zinc fingers, C2H2-type			
4110	-26.97	oe	ccsbBroad304_02231	USP6NL	-			
4111	-26.97	kd	CGS001-8435	SOAT2	-			
4112	-26.98	cp	BRD-K47936004	piribedil	Dopamine receptor agonist		DRD2, DRD3, ADRA1A, ADRA2A, ADRA2C, DRD4, HTR1A, HTR2B	Dopamine receptor agonist
4113	-26.98	cp	BRD-K22010301	JLK-6	Gamma secretase inhibitor		PSEN1	Gamma secretase inhibitor, Anti-amyloidogenic
4114	-27	oe	ccsbBroad304_00587	FOSL2	basic leucine zipper proteins			
4115	-27	kd	CGS001-275	AMT	-			
4116	-27.02	cp	BRD-K68190965	GR-46611	Serotonin receptor agonist		HTR1D	Serotonin receptor agonist
4117	-27.02	kd	CGS001-390	RND3	-			
4118	-27.05	kd	CGS001-790	CAD	-			
4119	-27.06	cp	BRD-A45333398	periplocymarin	Apoptosis stimulant			Apoptosis stimulant
4120	-27.06	kd	CGS001-60	ACTB	-			
4121	-27.11	kd	CGS001-4191	MDH2	-			
4122	-27.12	cp	BRD-K44849676	capsazepine	TRPV agonist		TRPV1, TRPV4	TRPV agonist
4123	-27.12	kd	CGS001-8872	CDC123	-			
4124	-27.12	kd	CGS001-4929	NR4A2	Nerve growth factor IB-like receptors			
4125	-27.19	oe	ccsbBroad304_01307	PSMA1	Proteasome subunits			
4126	-27.2	kd	CGS001-7850	IL1R2	Immunoglobulin-like family of IL-1 receptors			
4127	-27.21	oe	ccsbBroad304_07126	VARS	Aminoacyl tRNA synthetases / Class I			
4128	-27.21	kd	CGS001-4287	ATXN3	Ataxins			
4129	-27.23	kd	CGS001-1616	DAXX	-			
4130	-27.24	oe	ccsbBroad304_13939	MOK	RCK family			
4131	-27.26	kd	CGS001-54658	UGT1A1	UDP glucuronosyltransferases			
4132	-27.27	kd	CGS001-5873	RAB27A	RAB, member RAS oncogene			
4133	-27.29	oe	ccsbBroad304_01674	TIMP4	-			
4134	-27.32	oe	ccsbBroad304_01632	SYPL1	-			
4135	-27.36	cp	BRD-A39646320	HC-toxin	HDAC inhibitor		HDAC1	HDAC inhibitor
4136	-27.37	kd	CGS001-10123	ARL4C	ADP-ribosylation factors			
4137	-27.39	oe	ccsbBroad304_01077	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
4138	-27.41	kd	CGS001-84961	FBXL20	F-boxes / Leucine-rich repeats			
4139	-27.43	kd	CGS001-147179	WIPF2	-			
4140	-27.44	kd	CGS001-3934	LCN2	Lipocalins			
4141	-27.45	kd	CGS001-164832	LONRF2	RING-type (C3HC4) zinc fingers			
4142	-27.46	oe	ccsbBroad304_01093	NFKBIA	Ankyrin repeat domain containing			
4143	-27.46	cp	BRD-K16406336	methylene-blue	Guanylyl cyclase inhibitor		ACHE, MAPT	Guanylyl cyclase inhibitor, Monoamine oxidase inhibitor, Nitric oxide production inhibitor, Tau aggregation inhibitor
4144	-27.47	kd	CGS001-622	BDH1	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
4145	-27.5	kd	CGS001-256364	EML3	WD repeat domain containing			
4146	-27.54	cp	BRD-K40619305	larixinic-acid	Compound that interacts with metal centers			Compound that interacts with metal centers
4147	-27.54	kd	CGS001-7752	ZNF200	Zinc fingers, C2H2-type			
4148	-27.55	kd	CGS001-143187	VTI1A	-			
4149	-27.57	kd	CGS001-5982	RFC2	ATPases / AAA-type			
4150	-27.57	kd	CGS001-55718	POLR3E	RNA polymerase subunits			
4151	-27.57	kd	CGS001-1999	ELF3	ETS Transcription Factors			
4152	-27.58	cp	BRD-K20313525	rosmarinic-acid	GABA transaminase inhibitor		MCL1, TYR	GABA transaminase inhibitor
4153	-27.59	kd	CGS001-1072	CFL1	-			
4154	-27.61	kd	CGS001-3214	HOXB4	Homeoboxes / ANTP class : HOXL subclass			
4155	-27.62	cp	BRD-A02759312	betaxolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
4156	-27.66	oe	ccsbBroad304_07056	TGFB1	Endogenous ligands			
4157	-27.69	kd	CGS001-27316	RBMX	RNA binding motif (RRM) containing			
4158	-27.7	cp	BRD-K08554278	bisbenzimide	DNA binding agent		BCL2L1, TOP1	DNA binding agent
4159	-27.76	kd	CGS001-7474	WNT5A	Endogenous ligands			
4160	-27.76	kd	CGS001-4781	NFIB	-			
4161	-27.76	oe	ccsbBroad304_00933	LDHB	-			
4162	-27.77	kd	CGS001-8738	CRADD	-			
4163	-27.78	oe	ccsbBroad304_02981	GPR160	GPCR / Class A : Orphans			
4164	-27.78	oe	ccsbBroad304_06320	FFAR1	Fatty acid receptors			
4165	-27.8	kd	CGS001-23	ABCF1	ATP binding cassette transporters / subfamily F			
4166	-27.81	kd	CGS001-116039	OSR2	Zinc fingers, C2H2-type			
4167	-27.83	kd	CGS001-4223	MEOX2	Homeoboxes / ANTP class : HOXL subclass			
4168	-27.85	oe	ccsbBroad304_01278	PRKACB	Protein kinase A			
4169	-27.87	oe	ccsbBroad304_05527	GPR141	GPCR / Class A : Orphans			
4170	-27.87	oe	ccsbBroad304_02708	TRIM32	-			
4171	-27.87	oe	ccsbBroad304_00477	LPAR1	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
4172	-27.87	kd	CGS001-7538	ZFP36	RING-type (C3HC4) zinc fingers			
4173	-27.87	kd	CGS001-5021	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
4174	-27.87	kd	CGS001-60528	ELAC2	-			
4175	-27.87	kd	CGS001-4179	CD46	CD molecules			
4176	-27.88	oe	ccsbBroad304_00152	BCAT2	-			
4177	-27.88	cp	BRD-K91904471	SD-169	p38 MAPK inhibitor		MAPK14	p38 MAPK inhibitor
4178	-27.88	cp	BRD-K28863208	PNU-282987	Cholinergic receptor agonist		CHRNA7	Cholinergic receptor agonist
4179	-27.88	kd	CGS001-51160	VPS28	-			
4180	-27.89	kd	CGS001-861	RUNX1	-			
4181	-27.89	oe	ccsbBroad304_10212	GRHL3	-			
4182	-27.91	cp	BRD-K10042277	desmethylclozapine	Acetylcholine receptor agonist		CHRM1, DRD2, DRD3, HTR2A	Acetylcholine receptor agonist
4183	-27.92	kd	CGS001-3654	IRAK1	Interleukin-1 receptor-associated kinase (IRAK) family			
4184	-27.92	oe	ccsbBroad304_07738	ABHD2	Abhydrolase domain containing			
4185	-27.94	kd	CGS001-10174	SORBS3	-			
4186	-27.96	kd	CGS001-9807	IP6K1	-			
4187	-27.97	cp	BRD-K53972329	ruxolitinib	JAK inhibitor		JAK1, JAK2, TYK2, JAK3	JAK inhibitor
4188	-27.98	kd	CGS001-3682	ITGAE	Integrins			
4189	-27.99	kd	CGS001-1017	CDK2	Cyclin-dependent kinases, CDK1 subfamily			
4190	-28.02	kd	CGS001-5428	POLG	DNA polymerases			
4191	-28.03	oe	ccsbBroad304_01615	SULT1A2	Sulfotransferases, cytosolic			
4192	-28.05	cp	BRD-K90789829	nefazodone	Adrenergic inhibitor		HTR2A, SLC6A4, HTR2C, SLC6A2, ADRA1A, ADRA1B, ADRA2A, CYP3A4, CYP3A5, CYP3A7, HTR1A, SLC6A3	Adrenergic inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
4193	-28.05	kd	CGS001-11083	DIDO1	Zinc fingers, PHD-type			
4194	-28.07	kd	CGS001-27020	NPTN	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4195	-28.08	cp	BRD-A13133631	fluorometholone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
4196	-28.09	kd	CGS001-4300	MLLT3	-			
4197	-28.1	cc		CCK receptor antagonist	-			
4198	-28.13	oe	ccsbBroad304_02029	GGH	Gamma-glutamyl hydrolase			
4199	-28.13	oe	ccsbBroad304_03047	BZW2	-			
4200	-28.13	kd	CGS001-7010	TEK	Type XII RTKs: TIE family of angiopoietin receptors			
4201	-28.13	kd	CGS001-91754	NEK9	NIMA (never in mitosis gene a)- related kinase (NEK) family			
4202	-28.13	kd	CGS001-8669	EIF3J	-			
4203	-28.13	kd	CGS001-90	ACVR1	Type I receptor serine/threonine kinases			
4204	-28.16	cp	BRD-K92413528	thiazolidinecarboxylic-acid	Reducing agent			Reducing agent
4205	-28.17	oe	ccsbBroad304_00501	EMD	-			
4206	-28.17	cp	BRD-A17453586	MDL-72832	Serotonin receptor agonist		HTR1A	Serotonin receptor agonist
4207	-28.18	oe	ccsbBroad304_10971	MLLT6	Zinc fingers, PHD-type			
4208	-28.19	oe	ccsbBroad304_00006	ACADM	-			
4209	-28.22	kd	CGS001-115509	ZNF689	Zinc fingers, C2H2-type			
4210	-28.22	kd	CGS001-5915	RARB	Retinoic acid receptors			
4211	-28.22	kd	CGS001-283383	GPR133	Adhesion Class GPCRs			
4212	-28.24	kd	CGS001-79088	ZNF426	Zinc fingers, C2H2-type			
4213	-28.24	kd	CGS001-4907	NT5E	Adenosine turnover			
4214	-28.25	oe	ccsbBroad304_01276	PRKAB1	AMPK subfamily			
4215	-28.25	oe	ccsbBroad304_00945	LMNA	Intermediate filaments type V, lamins			
4216	-28.27	kd	CGS001-10557	RPP38	-			
4217	-28.29	kd	CGS001-10397	NDRG1	-			
4218	-28.3	kd	CGS001-83743	GRWD1	WD repeat domain containing			
4219	-28.32	oe	ccsbBroad304_07876	LARS2	Aminoacyl tRNA synthetases / Class I			
4220	-28.33	cc		Interleukins GOF	-			
4221	-28.33	kd	CGS001-54861	SNRK	SNRK subfamily			
4222	-28.33	kd	CGS001-2274	FHL2	-			
4223	-28.33	kd	CGS001-481	ATP1B1	ATPases / P-type			
4224	-28.37	oe	ccsbBroad304_09036	WDR61	WD repeat domain containing			
4225	-28.37	oe	ccsbBroad304_06665	OAT	-			
4226	-28.38	kd	CGS001-7535	ZAP70	Syk family			
4227	-28.38	kd	CGS001-8802	SUCLG1	-			
4228	-28.4	kd	CGS001-6196	RPS6KA2	RSK subfamily			
4229	-28.4	kd	CGS001-9924	PAN2	Ubiquitin-specific peptidases			
4230	-28.41	oe	ccsbBroad304_00736	NRG1	Immunoglobulin superfamily / I-set domain containing			
4231	-28.41	kd	CGS001-5184	PEPD	Methionyl aminopeptidase			
4232	-28.42	kd	CGS001-54881	TEX10	-			
4233	-28.42	kd	CGS001-10020	GNE	-			
4234	-28.45	oe	ccsbBroad304_05902	BNIP3	-			
4235	-28.51	kd	CGS001-10061	ABCF2	ATP binding cassette transporters / subfamily F			
4236	-28.52	oe	ccsbBroad304_07859	PLCB1	Phosphoinositide-specific phospholipase C			
4237	-28.52	oe	ccsbBroad304_06178	ERCC5	-			
4238	-28.52	kd	CGS001-22877	MLXIP	Basic helix-loop-helix proteins			
4239	-28.53	oe	ccsbBroad304_07220	CDC45	-			
4240	-28.56	cp	BRD-K43860855	iobenguane	Antineoplastic			Antineoplastic
4241	-28.58	cp	BRD-A02710418	meptazinol	Opioid receptor agonist		BCHE	Opioid receptor agonist
4242	-28.59	oe	ccsbBroad304_03666	CISD1	CDGSH iron sulfur domain containing			
4243	-28.61	kd	CGS001-2879	GPX4	-			
4244	-28.68	oe	ccsbBroad304_06131	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
4245	-28.71	cp	BRD-K99964838	bosutinib	ABL inhibitor		ABL1, SRC, BCR, CAMK2G, LYN, CAMK1D, CDK2, FRK, FYN, HCK, MAP2K1, MAP2K2, MAP3K2, MAP4K5, STK10, STK24, STK4, TNK2, TXK	ABL inhibitor, BCR-ABL kinase inhibitor, SRC inhibitor
4246	-28.72	oe	ccsbBroad304_07561	YAF2	-			
4247	-28.73	cp	BRD-K11129031	gemfibrozil	Lipoprotein lipase activator		PPARA, CYP2C8, LPL, SLCO1B1, SLCO1B3, SLCO2B1	Lipoprotein lipase activator
4248	-28.75	kd	CGS001-6925	TCF4	Basic helix-loop-helix proteins			
4249	-28.76	kd	CGS001-10682	EBP	-			
4250	-28.77	kd	CGS001-8996	NOL3	-			
4251	-28.78	kd	CGS001-9687	GREB1	-			
4252	-28.8	kd	CGS001-1643	DDB2	WD repeat domain containing			
4253	-28.83	oe	ccsbBroad304_08053	TAF5L	WD repeat domain containing			
4254	-28.83	cp	BRD-A29082194	gitoxigenin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4255	-28.83	cp	BRD-K96527333	dehydroisoandosterone	GABA receptor modulator			GABA receptor modulator
4256	-28.86	kd	CGS001-84328	LZIC	-			
4257	-28.87	cc		Phospholipases GOF	-			
4258	-28.87	oe	ccsbBroad304_07015	SULT1A1	Sulfotransferases, cytosolic			
4259	-28.87	kd	CGS001-2182	ACSL4	Acyl-CoA synthetase family			
4260	-28.94	cp	BRD-K42221274	NNC-711	GAT inhibitor		SLC6A1, SIGMAR1	GAT inhibitor
4261	-28.97	kd	CGS001-8841	HDAC3	Histone deacetylases			
4262	-28.99	oe	ccsbBroad304_06483	KCNK1	Two-P potassium channels			
4263	-29.02	kd	CGS001-4594	MUT	-			
4264	-29.02	kd	CGS001-81570	CLPB	Ankyrin repeat domain containing			
4265	-29.03	oe	ccsbBroad304_06896	RPS6KA1	RSK subfamily			
4266	-29.03	kd	CGS001-3399	ID3	Basic helix-loop-helix proteins			
4267	-29.04	oe	ccsbBroad304_06448	IL18	Interleukins and interleukin receptors			
4268	-29.05	oe	ccsbBroad304_02195	SPAG7	-			
4269	-29.06	kd	CGS001-55437	STRADB	STLK subfamily			
4270	-29.08	cc		GPCR Subset GOF	-			
4271	-29.13	oe	ccsbBroad304_06621	NDUFA8	Mitochondrial respiratory chain complex / Complex I			
4272	-29.16	kd	CGS001-516	ATP5G1	ATPases / F-type			
4273	-29.17	kd	CGS001-6890	TAP1	ATP binding cassette transporters / subfamily B			
4274	-29.17	kd	CGS001-4968	OGG1	-			
4275	-29.18	oe	ccsbBroad304_13822	CALM3	EF-hand domain containing			
4276	-29.19	oe	ccsbBroad304_00744	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
4277	-29.19	kd	CGS001-26472	PPP1R14B	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4278	-29.25	kd	CGS001-57215	THAP11	THAP (C2CH-type zinc finger) domain containing			
4279	-29.28	cc		Glucocorticoid receptor agonist	-			
4280	-29.29	oe	ccsbBroad304_06624	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
4281	-29.29	kd	CGS001-221692	PHACTR1	Phosphatase and actin regulators			
4282	-29.33	kd	CGS001-5934	RBL2	-			
4283	-29.35	kd	CGS001-2931	GSK3A	GSK subfamily			
4284	-29.37	kd	CGS001-23211	ZC3H4	Zinc fingers, CCCH-type domain containing			
4285	-29.38	kd	CGS001-4722	NDUFS3	Mitochondrial respiratory chain complex / Complex I			
4286	-29.4	oe	ccsbBroad304_00066	ANG	Ribonucleases, RNase A			
4287	-29.4	kd	CGS001-100	ADA	Adenosine turnover			
4288	-29.45	kd	CGS001-10652	YKT6	-			
4289	-29.46	kd	CGS001-23118	TAB2	-			
4290	-29.47	cp	BRD-K83794624	pirarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4291	-29.48	kd	CGS001-7167	TPI1	-			
4292	-29.48	kd	CGS001-1528	CYB5A	Cytochrome b genes			
4293	-29.5	cp	BRD-K15933101	ropinirole	Dopamine receptor agonist		DRD2, DRD3, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
4294	-29.5	kd	CGS001-1020	CDK5	Cyclin-dependent kinases, CDK5 subfamily			
4295	-29.51	cc		Sodium channel blocker	-			
4296	-29.51	kd	CGS001-10921	RNPS1	RNA binding motif (RRM) containing			
4297	-29.52	oe	ccsbBroad304_07436	SPTLC2	Serine palmitoyltransferase			
4298	-29.56	cp	BRD-A22769835	homochlorcyclizine	Antihistamine		HRH1	Antihistamine
4299	-29.58	cp	BRD-K11540476	EMF-BCA1-64	Caspase inhibitor		CASP3	Caspase inhibitor
4300	-29.64	oe	ccsbBroad304_00561	FGFR1	Type V RTKs: FGF (fibroblast growth factor) receptor family			
4301	-29.64	kd	CGS001-5159	PDGFRB	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
4302	-29.64	kd	CGS001-7760	ZNF213	Zinc fingers, C2H2-type			
4303	-29.66	cp	BRD-K13664374	dichloroacetic-acid	Pyruvate dehydrogenase kinase inhibitor		PDK1	Pyruvate dehydrogenase kinase inhibitor
4304	-29.67	oe	ccsbBroad304_01034	MSH2	-			
4305	-29.69	kd	CGS001-5621	PRNP	CD molecules			
4306	-29.71	kd	CGS001-9377	COX5A	Mitochondrial respiratory chain complex			
4307	-29.81	cp	BRD-K72034655	peucedanin	Apoptosis stimulant			Apoptosis stimulant
4308	-29.86	oe	ccsbBroad304_01002	METTL1	-			
4309	-29.86	kd	CGS001-2859	GPR35	GPCR / Class A : Orphans			
4310	-29.86	kd	CGS001-23466	CBX6	-			
4311	-29.87	cp	BRD-K60476892	YC-1	Guanylyl cyclase activator		HIF1A, GUCY1A2, GUCY1A3, GUCY1B3	Guanylyl cyclase activator
4312	-29.95	kd	CGS001-1747	DLX3	Homeoboxes / ANTP class : NKL subclass			
4313	-29.97	kd	CGS001-10972	TMED10	-			
4314	-29.97	kd	CGS001-55818	KDM3A	Histone demethylases			
4315	-29.99	oe	ccsbBroad304_01237	POLR2C	RNA polymerase subunits			
4316	-30.02	oe	ccsbBroad304_06957	SLC1A5	Alanine/serine/cysteine transporter subfamily			
4317	-30.02	oe	ccsbBroad304_01452	RPS13	S ribosomal proteins			
4318	-30.06	oe	ccsbBroad304_00800	HSPD1	Heat Shock Proteins / Chaperonins			
4319	-30.06	kd	CGS001-24148	PRPF6	-			
4320	-30.08	oe	ccsbBroad304_09746	ZNF610	Zinc fingers, C2H2-type			
4321	-30.13	kd	CGS001-2109	ETFB	-			
4322	-30.16	cp	BRD-A14798026	mestranol	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
4323	-30.17	oe	ccsbBroad304_01324	PSMD10	Ankyrin repeat domain containing			
4324	-30.17	kd	CGS001-54884	RETSAT	-			
4325	-30.2	oe	ccsbBroad304_08426	TEX10	-			
4326	-30.22	cp	BRD-K25504083	cytochalasin-d	Actin polymerization inhibitor		ACTB	Actin polymerization inhibitor
4327	-30.23	kd	CGS001-84722	PSRC1	-			
4328	-30.25	cp	BRD-A07765530	epinephrine	carbonic anhydrase activator		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, PAH, TNF	carbonic anhydrase activator
4329	-30.25	cp	BRD-K51313569	palbociclib	CDK inhibitor		CDK4, CDK6, CCND3	CDK inhibitor
4330	-30.25	kd	CGS001-5547	PRCP	Lysosomal Pro-Xaa carboxypeptidase			
4331	-30.28	kd	CGS001-23192	ATG4B	Aut2 peptidase			
4332	-30.3	oe	ccsbBroad304_06765	PRCC	-			
4333	-30.3	kd	CGS001-10273	STUB1	Tetratricopeptide (TTC) repeat domain containing			
4334	-30.3	kd	CGS001-1409	CRYAA	Heat shock proteins / HSPB			
4335	-30.31	kd	CGS001-6337	SCNN1A	Epithelial sodium channels (ENaC)			
4336	-30.38	oe	ccsbBroad304_07219	CDC7	CDC7 family			
4337	-30.39	kd	CGS001-3597	IL13RA1	IL-2 receptor family			
4338	-30.43	cc		ATPase inhibitor	-			
4339	-30.43	kd	CGS001-2212	FCGR2A	CD molecules			
4340	-30.46	oe	ccsbBroad304_05180	ZNF626	Zinc fingers, C2H2-type			
4341	-30.46	kd	CGS001-5108	PCM1	-			
4342	-30.46	kd	CGS001-978	CDA	-			
4343	-30.47	cp	BRD-K66615216	moxifloxacin	Bacterial DNA gyrase inhibitor		TOP2A	Bacterial DNA gyrase inhibitor
4344	-30.48	cp	BRD-K40758068	efavirenz	HIV protease inhibitor		CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5	HIV protease inhibitor
4345	-30.5	kd	CGS001-9738	CCP110	-			
4346	-30.53	kd	CGS001-23161	SNX13	Sorting nexins			
4347	-30.55	oe	ccsbBroad304_01258	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4348	-30.57	oe	ccsbBroad304_07832	XPO7	Exportins			
4349	-30.57	kd	CGS001-3123	HLA-DRB1	Immunoglobulin superfamily / C1-set domain containing			
4350	-30.59	oe	ccsbBroad304_02017	PEX11A	-			
4351	-30.59	kd	CGS001-2767	GNA11	-			
4352	-30.6	oe	ccsbBroad304_01184	PGK1	-			
4353	-30.61	oe	ccsbBroad304_11405	UBE3C	-			
4354	-30.64	oe	ccsbBroad304_00772	HOXA6	Homeoboxes / ANTP class : HOXL subclass			
4355	-30.67	cp	BRD-A22713669	BVT-948	Tyrosine phosphatase inhibitor		PTPN1, PTPN11, PTPN2	Tyrosine phosphatase inhibitor
4356	-30.67	kd	CGS001-23761	PISD	Decarboxylases			
4357	-30.7	kd	CGS001-290	ANPEP	Aminopeptidase N			
4358	-30.75	cp	BRD-K57886322	fluocinonide	Glucocorticoid receptor agonist		NR3C1, SERPINA6, SMO	Glucocorticoid receptor agonist
4359	-30.76	kd	CGS001-7078	TIMP3	-			
4360	-30.76	kd	CGS001-65217	PCDH15	Cadherins / Cadherin-related			
4361	-30.76	kd	CGS001-114785	MBD6	-			
4362	-30.79	kd	CGS001-23057	NMNAT2	-			
4363	-30.8	oe	ccsbBroad304_06694	SERPINA5	Serine (or cysteine) peptidase inhibitors			
4364	-30.85	oe	ccsbBroad304_00420	DAP	-			
4365	-30.85	cp	BRD-K61250553	loperamide	Opioid receptor agonist		OPRM1, OPRD1, CACNA1A, CALM1, CYP2B6, CYP2C8, NPR2, OPRK1, POMC	Opioid receptor agonist
4366	-30.89	oe	ccsbBroad304_03570	QRSL1	-			
4367	-30.89	cp	BRD-K96720755	relcovaptan	Vasopressin receptor antagonist		AVPR1A, AVPR1B, AVPR2, OXTR	Vasopressin receptor antagonist
4368	-30.9	oe	ccsbBroad304_07208	NRIP1	-			
4369	-30.9	oe	ccsbBroad304_09035	COASY	-			
4370	-30.91	cp	BRD-K32398298	alprazolam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, CYP3A5, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
4371	-30.91	kd	CGS001-9352	TXNL1	-			
4372	-30.91	kd	CGS001-23196	FAM120A	-			
4373	-30.92	kd	CGS001-8681	JMJD7-PLA2G4B	-			
4374	-30.98	kd	CGS001-285268	ZNF621	Zinc fingers, C2H2-type			
4375	-30.98	kd	CGS001-4204	MECP2	-			
4376	-31	cp	BRD-K90259198	W-7	Calmodulin antagonist		CALM1, CALM2, KCNA5, KCNH2, TNNC1, TNNI3	Calmodulin antagonist, Potassium channel blocker
4377	-31.05	cp	BRD-K37792168	denbufylline	Phosphodiesterase inhibitor		PDE4A, PDE4B, PDE4D	Phosphodiesterase inhibitor
4378	-31.07	kd	CGS001-1829	DSG2	Cadherins / Major cadherins			
4379	-31.11	cp	BRD-K79353516	indolophenanthridine	CALY activator		CALY, DRD1	CALY activator
4380	-31.13	oe	ccsbBroad304_00316	CKS1B	-			
4381	-31.14	cp	BRD-A35338386	NECA	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, HSP90B1	Adenosine receptor agonist
4382	-31.21	kd	CGS001-64425	POLR1E	RNA polymerase subunits			
4383	-31.21	kd	CGS001-10695	CNPY3	Trinucleotide (CAG) repeat containing			
4384	-31.22	oe	ccsbBroad304_03785	INTS12	Zinc fingers, PHD-type			
4385	-31.31	kd	CGS001-2166	FAAH	Endocannabinoid turnover			
4386	-31.33	oe	ccsbBroad304_00961	SMAD2	SMADs			
4387	-31.33	oe	ccsbBroad304_06806	PSMD3	Proteasome (prosome, macropain) subunits			
4388	-31.35	oe	ccsbBroad304_06617	NASP	Tetratricopeptide (TTC) repeat domain containing			
4389	-31.37	kd	CGS001-7625	ZNF74	Zinc fingers, C2H2-type			
4390	-31.39	oe	ccsbBroad304_07887	GCAT	-			
4391	-31.39	kd	CGS001-9690	UBE3C	-			
4392	-31.4	oe	ccsbBroad304_01332	PTGER4	GPCR / Class A : Prostanoid receptors			
4393	-31.41	oe	ccsbBroad304_00863	IL15	Interleukins and interleukin receptors			
4394	-31.41	kd	CGS001-3672	ITGA1	Integrins			
4395	-31.42	oe	ccsbBroad304_00155	CCND1	-			
4396	-31.46	oe	ccsbBroad304_01054	GADD45B	-			
4397	-31.48	oe	ccsbBroad304_02837	BHMT2	-			
4398	-31.48	kd	CGS001-22954	TRIM32	-			
4399	-31.49	oe	ccsbBroad304_01536	SIM2	Basic helix-loop-helix proteins			
4400	-31.51	kd	CGS001-10010	TANK	-			
4401	-31.51	kd	CGS001-5106	PCK2	-			
4402	-31.52	oe	ccsbBroad304_10216	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4403	-31.53	kd	CGS001-53343	NUDT9	Nudix motif containing			
4404	-31.56	kd	CGS001-56916	SMARCAD1	-			
4405	-31.57	oe	ccsbBroad304_08267	KLF3	Kruppel-like transcription factors			
4406	-31.57	kd	CGS001-30849	PIK3R4	Phosphatidylinositol kinases			
4407	-31.57	kd	CGS001-9929	JOSD1	-			
4408	-31.65	oe	ccsbBroad304_07843	FCHO1	-			
4409	-31.66	oe	ccsbBroad304_04780	GPR139	GPCR / Class A : Orphans			
4410	-31.66	oe	ccsbBroad304_02386	EIF1B	-			
4411	-31.66	kd	CGS001-8202	NCOA3	Histone acetyltransferases			
4412	-31.66	kd	CGS001-11057	ABHD2	Abhydrolase domain containing			
4413	-31.68	oe	ccsbBroad304_07528	DMTF1	-			
4414	-31.7	oe	ccsbBroad304_09578	PASD1	-			
4415	-31.7	cp	BRD-K29178788	dictamnine	Furoquinoline alkaloid			Furoquinoline alkaloid
4416	-31.7	kd	CGS001-84619	ZGPAT	G patch domain containing			
4417	-31.74	kd	CGS001-10723	SLC12A7	SLC12 family of cation-coupled chloride transporters			
4418	-31.81	oe	ccsbBroad304_00173	BRCA1	Fanconi anemia, complementation groups			
4419	-31.85	kd	CGS001-80314	EPC1	-			
4420	-31.87	oe	ccsbBroad304_06257	GATA2	GATA zinc finger domain containing			
4421	-31.9	oe	ccsbBroad304_06422	ID3	Basic helix-loop-helix proteins			
4422	-31.9	cp	BRD-A20697603	thiostrepton	FOXM1 inhibitor		FOXM1	FOXM1 inhibitor, Protein synthesis inhibitor
4423	-31.91	oe	ccsbBroad304_07249	PIK3R3	Phosphatidylinositol kinases			
4424	-31.93	oe	ccsbBroad304_01450	RPS10	S ribosomal proteins			
4425	-31.98	kd	CGS001-51181	DCXR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
4426	-32.01	kd	CGS001-8804	CREG1	-			
4427	-32.08	kd	CGS001-79902	NUP85	-			
4428	-32.09	kd	CGS001-79712	GTDC1	Glycosyltransferase group 1 domain containing			
4429	-32.12	oe	ccsbBroad304_00960	SMAD1	SMADs			
4430	-32.14	oe	ccsbBroad304_02496	MTX2	-			
4431	-32.14	oe	ccsbBroad304_01836	MAPKAPK3	MAPKAPK subfamily			
4432	-32.19	kd	CGS001-51548	SIRT6	Histone deacetylases (HDACs)			
4433	-32.21	oe	ccsbBroad304_01577	SOD1	-			
4434	-32.21	oe	ccsbBroad304_02299	NR1H3	Liver X receptor-like receptors			
4435	-32.22	kd	CGS001-4671	NAIP	Inhibitors of apoptosis (IAP) protein family			
4436	-32.23	kd	CGS001-5198	PFAS	-			
4437	-32.25	oe	ccsbBroad304_10227	ZNF85	Zinc fingers, C2H2-type			
4438	-32.25	oe	ccsbBroad304_06089	DDIT3	-			
4439	-32.26	cp	BRD-A30435184	metergoline	Dopamine receptor agonist		DRD2, HTR1A, HTR1B, HTR1D, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C, HTR5A, HTR6, HTR7	Dopamine receptor agonist, Serotonin receptor antagonist
4440	-32.27	cp	BRD-A77291778	cyclopentolate	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
4441	-32.28	cp	BRD-K06208435	YS-035	Calcium channel blocker			Calcium channel blocker
4442	-32.29	oe	ccsbBroad304_00650	GNA11	-			
4443	-32.29	oe	ccsbBroad304_03936	PJA1	RING-type (C3HC4) zinc fingers			
4444	-32.3	oe	ccsbBroad304_00838	IGFBP5	insulin-like growth factor (IGF) binding proteins			
4445	-32.3	cp	BRD-K85985071	ellipticine	Topoisomerase inhibitor		TOP2A, TOP2B	Topoisomerase inhibitor
4446	-32.31	oe	ccsbBroad304_03240	HSPA14	Heat shock proteins / HSP70			
4447	-32.31	kd	CGS001-8193	DPF1	Zinc fingers, PHD-type			
4448	-32.32	kd	CGS001-1211	CLTA	-			
4449	-32.33	kd	CGS001-6793	STK10	SLK subfamily			
4450	-32.36	oe	ccsbBroad304_07515	GFPT2	-			
4451	-32.37	oe	ccsbBroad304_03056	MCTS1	-			
4452	-32.38	oe	ccsbBroad304_06288	GMDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4453	-32.38	oe	ccsbBroad304_00443	DHFR	Oxidoreductases			
4454	-32.38	oe	ccsbBroad304_03599	BATF3	basic leucine zipper proteins			
4455	-32.39	kd	CGS001-8192	CLPP	ATPases / AAA-type			
4456	-32.45	oe	ccsbBroad304_10207	ERLIN1	-			
4457	-32.49	oe	ccsbBroad304_00088	FASLG	Tumour necrosis factor (TNF) receptor family			
4458	-32.5	cp	BRD-K37561857	zardaverine	Phosphodiesterase inhibitor		PDE4D, PDE3A, PDE4A, PDE4B, PDE4C	Phosphodiesterase inhibitor
4459	-32.51	cp	BRD-K11742128	triprolidine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4460	-32.57	cp	BRD-K51967704	BIIB021	HSP inhibitor		AOX1, HSP90AA1	HSP inhibitor
4461	-32.57	cp	BRD-K87024524	phenelzine	Monoamine oxidase inhibitor		MAOB, AOC3, MAOA, ABAT, GAD2, GPT, GPT2, SLC6A2, SLC6A3, SLC6A4	Monoamine oxidase inhibitor
4462	-32.58	oe	ccsbBroad304_06085	DCK	-			
4463	-32.59	oe	ccsbBroad304_08424	SNRK	SNRK subfamily			
4464	-32.61	oe	ccsbBroad304_02923	PHF19	Zinc fingers, PHD-type			
4465	-32.62	kd	CGS001-4488	MSX2	Homeoboxes / ANTP class : NKL subclass			
4466	-32.68	oe	ccsbBroad304_07064	TH	Amino acid hydroxylases			
4467	-32.7	oe	ccsbBroad304_00055	AKR1B1	Aldo-keto reductases			
4468	-32.7	kd	CGS001-3053	SERPIND1	Serine (or cysteine) peptidase inhibitors			
4469	-32.77	kd	CGS001-10125	RASGRP1	EF-hand domain containing			
4470	-32.79	oe	ccsbBroad304_04383	PCGF5	Polycomb group ring fingers			
4471	-32.82	cp	BRD-A79465854	auranofin	NFkB pathway inhibitor		IKBKB, PRDX5, TRPA1, TXNRD1, TXNRD2	NFkB pathway inhibitor
4472	-32.84	oe	ccsbBroad304_14122	TNFRSF21	Tumour necrosis factor (TNF) receptor family			
4473	-32.9	cp	BRD-K91442916	CAM-9-026	Membrane metalloendopeptidase inhibitor			Membrane metalloendopeptidase inhibitor
4474	-32.97	oe	ccsbBroad304_07383	STK17A	Death-associated kinase (DAPK) family			
4475	-32.97	cp	BRD-K92093830	doxorubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
4476	-32.98	cp	BRD-K25905511	buddleoflavonoloside	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
4477	-32.98	kd	CGS001-23443	SLC35A3	SLC35 family of nucleotide sugar transporters			
4478	-33.03	cp	BRD-M72442222	vicriviroc	CC chemokine receptor antagonist		CCR5	CC chemokine receptor antagonist
4479	-33.05	kd	CGS001-2119	ETV5	ETS Transcription Factors			
4480	-33.06	oe	ccsbBroad304_13931	PSMA3	Proteasome subunits			
4481	-33.06	kd	CGS001-79961	DENND2D	DENN/MADD domain containing			
4482	-33.08	oe	ccsbBroad304_11324	RPS6KA4	MSK subfamily			
4483	-33.11	kd	CGS001-10237	SLC35B1	SLC35 family of nucleotide sugar transporters			
4484	-33.17	cp	BRD-K50128260	sildenafil	Phosphodiesterase inhibitor		PDE5A, PDE6G, PDE6H, SLCO1B1, SLCO1B3	Phosphodiesterase inhibitor
4485	-33.17	kd	CGS001-6566	SLC16A1	SLC16 family of monocarboxylate transporters			
4486	-33.18	kd	CGS001-8892	EIF2B2	-			
4487	-33.19	oe	ccsbBroad304_02503	TNFSF13B	CD molecules			
4488	-33.2	kd	CGS001-1859	DYRK1A	Dyrk1 subfamily			
4489	-33.21	oe	ccsbBroad304_00072	ANXA7	Annexins			
4490	-33.22	oe	ccsbBroad304_05005	ZNF582	Zinc fingers, C2H2-type			
4491	-33.22	cp	BRD-K43330982	JTE-013	Lysophospholipid receptor antagonist		S1PR2, P2RY10	Lysophospholipid receptor antagonist
4492	-33.23	kd	CGS001-8233	ZRSR2	RNA binding motif (RRM) containing			
4493	-33.25	kd	CGS001-6208	RPS14	S ribosomal proteins			
4494	-33.26	oe	ccsbBroad304_02783	POFUT1	Fucosyltransferases			
4495	-33.3	oe	ccsbBroad304_02487	TXNIP	-			
4496	-33.3	kd	CGS001-2842	GPR19	GPCR / Class A : Orphans			
4497	-33.37	oe	ccsbBroad304_01811	PCGF2	Polycomb group ring fingers			
4498	-33.43	oe	ccsbBroad304_06433	IGHMBP2	Zinc fingers, AN1-type domain containing			
4499	-33.44	cc		Progesterone receptor antagonist	-			
4500	-33.47	kd	CGS001-1001	CDH3	Cadherins / Major cadherins			
4501	-33.49	cp	BRD-A19736161	ondansetron	Serotonin receptor antagonist		HTR3A, CYP2D6, CYP3A5, HTR1A, HTR1B, HTR3B, HTR4, OPRM1	Serotonin receptor antagonist
4502	-33.51	kd	CGS001-93487	MAPK1IP1L	-			
4503	-33.53	kd	CGS001-2849	GPR26	GPCR / Class A : Orphans			
4504	-33.53	kd	CGS001-90993	CREB3L1	basic leucine zipper proteins			
4505	-33.55	kd	CGS001-5607	MAP2K5	MAPKK:STE7 family			
4506	-33.56	oe	ccsbBroad304_06394	HOXC9	Homeoboxes / ANTP class : HOXL subclass			
4507	-33.56	cp	BRD-K76617868	fasudil	Rho associated kinase inhibitor		ROCK1, ROCK2, PKIA, PRKACA	Rho associated kinase inhibitor
4508	-33.63	kd	CGS001-9126	SMC3	Structural maintenance of chromosomes proteins			
4509	-33.65	cp	BRD-K35430135	SR-59230A	Adrenergic receptor antagonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor antagonist
4510	-33.69	oe	ccsbBroad304_04360	CAPNS2	EF-hand domain containing			
4511	-33.69	oe	ccsbBroad304_07291	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4512	-33.69	kd	CGS001-6048	RNF5	RING-type (C3HC4) zinc fingers			
4513	-33.71	kd	CGS001-10523	CHERP	G patch domain containing			
4514	-33.72	kd	CGS001-2639	GCDH	-			
4515	-33.73	oe	ccsbBroad304_05865	ATP1A3	ATPases / P-type			
4516	-33.73	kd	CGS001-1497	CTNS	-			
4517	-33.8	kd	CGS001-11325	DDX42	DEAD-boxes			
4518	-33.83	oe	ccsbBroad304_00682	GRK6	GRK1/3 subfamily			
4519	-33.83	oe	ccsbBroad304_00305	CHRM3	Cholinergic receptors			
4520	-33.83	kd	CGS001-8942	KYNU	-			
4521	-33.84	oe	ccsbBroad304_03880	RXFP1	GPCR / Class A : Relaxin family peptide receptors			
4522	-33.88	cp	BRD-K67439147	SIB-1893	Glutamate receptor antagonist		GRM5, GRM4	Glutamate receptor antagonist
4523	-33.89	oe	ccsbBroad304_06402	PRMT2	Protein arginine N-methyltransferases			
4524	-33.91	oe	ccsbBroad304_06469	KARS	Aminoacyl tRNA synthetases / Class II			
4525	-33.94	oe	ccsbBroad304_00326	CLK1	CDC-like kinases			
4526	-33.95	oe	ccsbBroad304_03788	LPAR5	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
4527	-33.95	oe	ccsbBroad304_07596	DLC1	Rho GTPase activating proteins			
4528	-33.96	cp	BRD-K54759182	dosulepin	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, HRH1	Norepinephrine reuptake inhibitor, Tricyclic antidepressant, Serotonin reuptake inhibitor
4529	-33.99	oe	ccsbBroad304_01803	ZBTB25	BTB/POZ domain containing			
4530	-33.99	kd	CGS001-139760	GPR119	GPCR / Class A : Orphans			
4531	-34.02	kd	CGS001-6277	S100A6	EF-hand domain containing			
4532	-34.03	cp	BRD-A16332958	modafinil	Adrenergic receptor agonist		ADRA1B, CYP1A2, CYP2B6, CYP2C19, CYP3A4, CYP3A5, SLC6A3	Adrenergic receptor agonist
4533	-34.13	oe	ccsbBroad304_04990	ZNF597	Zinc fingers, C2H2-type			
4534	-34.16	oe	ccsbBroad304_04786	CANT1	-			
4535	-34.18	oe	ccsbBroad304_03933	CARD9	-			
4536	-34.19	cp	BRD-K72541103	JAK3-inhibitor-I	JAK inhibitor		JAK3	JAK inhibitor
4537	-34.21	kd	CGS001-127540	HMGB4	High-mobility group / Canonical			
4538	-34.22	kd	CGS001-10489	LRRC41	-			
4539	-34.25	kd	CGS001-10732	TCFL5	Basic helix-loop-helix proteins			
4540	-34.26	oe	ccsbBroad304_02279	RBX1	RING-type (C3HC4) zinc fingers			
4541	-34.3	kd	CGS001-3126	HLA-DRB4	Immunoglobulin superfamily / C1-set domain containing			
4542	-34.32	oe	ccsbBroad304_07129	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
4543	-34.32	oe	ccsbBroad304_03340	LSR	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4544	-34.34	kd	CGS001-3725	JUN	basic leucine zipper proteins			
4545	-34.37	oe	ccsbBroad304_08418	FBXL12	F-boxes / Leucine-rich repeats			
4546	-34.43	oe	ccsbBroad304_07814	SACM1L	-			
4547	-34.46	oe	ccsbBroad304_03707	PCDHA10	Cadherins / Protocadherins : Clustered			
4548	-34.46	oe	ccsbBroad304_11580	TLK2	Tousled-like kinase (TLK) family			
4549	-34.48	oe	ccsbBroad304_04478	ALG2	Glycosyltransferase group 1 domain containing			
4550	-34.56	oe	ccsbBroad304_01103	NONO	RNA binding motif (RRM) containing			
4551	-34.6	cp	BRD-A90799790	isradipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1F, CACNA1H, CACNA1S, CACNA2D2, CACNB2	Calcium channel blocker
4552	-34.6	kd	CGS001-5588	PRKCQ	Delta subfamily			
4553	-34.64	oe	ccsbBroad304_02330	G3BP1	RNA binding motif (RRM) containing			
4554	-34.64	kd	CGS001-23564	DDAH2	Dimethylarginine dimethylaminohydrolases			
4555	-34.66	kd	CGS001-8408	ULK1	Unc-51-like kinase (ULK) family			
4556	-34.68	oe	ccsbBroad304_01218	PLK1	Polo-like kinase (PLK) family			
4557	-34.69	oe	ccsbBroad304_06411	HSPA9	Heat shock proteins / HSP70			
4558	-34.73	cp	BRD-K27721098	clopidogrel	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19, CYP3A5	Purinergic receptor antagonist
4559	-34.74	kd	CGS001-25803	SPDEF	ETS Transcription Factors			
4560	-34.77	kd	CGS001-801	CALM1	EF-hand domain containing			
4561	-34.8	cp	BRD-K83597974	pargyline	Monoamine oxidase inhibitor		MAOB, MAOA	Monoamine oxidase inhibitor
4562	-34.81	kd	CGS001-221393	GPR115	Adhesion Class GPCRs			
4563	-34.83	kd	CGS001-11151	CORO1A	Coronins			
4564	-34.84	kd	CGS001-23621	BACE1	Pepsin			
4565	-34.86	oe	ccsbBroad304_07304	TNFRSF10B	Tumour necrosis factor (TNF) receptor family			
4566	-34.87	kd	CGS001-4038	LRP4	Low density lipoprotein receptors			
4567	-34.88	kd	CGS001-25976	TIPARP	Poly (ADP-ribose) polymerases			
4568	-34.95	kd	CGS001-207	AKT1	Akt (Protein kinase B)			
4569	-34.96	kd	CGS001-1849	DUSP7	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
4570	-34.96	kd	CGS001-29775	CARD10	-			
4571	-34.97	cp	BRD-A68631409	evodiamine	ATPase inhibitor		TRPV1	ATPase inhibitor, TRPV agonist
4572	-34.97	kd	CGS001-29079	MED4	-			
4573	-35.03	oe	ccsbBroad304_06750	POLR2H	RNA polymerase subunits			
4574	-35.03	kd	CGS001-7422	VEGFA	Cytokines and growth factors			
4575	-35.04	oe	ccsbBroad304_02318	KIF20A	Kinesins			
4576	-35.04	oe	ccsbBroad304_02312	ARPC1B	Actin related protein 2/3 complex subunits			
4577	-35.05	cc		Structural maintenance of chromosomes proteins LOF	-			
4578	-35.05	kd	CGS001-23670	TMEM2	-			
4579	-35.12	cp	BRD-A11678676	wortmannin	PI3K inhibitor		PIK3CA, PIK3CG, PLK1, ATM, ATR, MTOR, PI4KA, PI4KB, PIK3CD, PIK3R1, PLK3, PRKDC	PI3K inhibitor
4580	-35.12	kd	CGS001-9668	ZNF432	Zinc fingers, C2H2-type			
4581	-35.13	cp	BRD-K76133116	benzydamine	Membrane integrity inhibitor		PRSS1, PRSS2	Membrane integrity inhibitor, Prostanoid receptor antagonist, Prostanoid receptor inhibitor
4582	-35.18	kd	CGS001-899	CCNF	F-boxes / other			
4583	-35.2	oe	ccsbBroad304_00782	HPGD	Prostaglandin synthases			
4584	-35.2	kd	CGS001-3569	IL6	Interferons			
4585	-35.22	kd	CGS001-4790	NFKB1	NFkappaB transcription factor family			
4586	-35.23	cp	BRD-K90976994	dehydrocholic-acid	Bile acid			Bile acid
4587	-35.3	kd	CGS001-23239	PHLPP1	Pleckstrin homology (PH) domain containing			
4588	-35.35	cp	BRD-K21548250	moracizine	Sodium channel blocker		SCN5A	Sodium channel blocker
4589	-35.37	kd	CGS001-5693	PSMB5	Proteasome subunits			
4590	-35.39	oe	ccsbBroad304_01448	RPS7	S ribosomal proteins			
4591	-35.43	kd	CGS001-200879	LIPH	-			
4592	-35.44	oe	ccsbBroad304_03506	AURKAIP1	-			
4593	-35.44	cp	BRD-A95445494	maackiain	Sodium/glucose cotransporter inhibitor		SLC5A2	Sodium/glucose cotransporter inhibitor
4594	-35.47	oe	ccsbBroad304_01454	RPS15A	S ribosomal proteins			
4595	-35.47	kd	CGS001-84515	MCM8	-			
4596	-35.5	cc		Targets of VEGFR inhibitors GOF	-			
4597	-35.53	kd	CGS001-23451	SF3B1	-			
4598	-35.53	kd	CGS001-55577	NAGK	-			
4599	-35.55	oe	ccsbBroad304_03769	CTNNBIP1	Catenins			
4600	-35.59	oe	ccsbBroad304_06070	CYC1	Mitochondrial respiratory chain complex / Complex III			
4601	-35.62	kd	CGS001-7846	TUBA1A	Tubulins			
4602	-35.63	kd	CGS001-4680	CEACAM6	CD molecules			
4603	-35.64	kd	CGS001-6576	SLC25A1	Mitochondrial di- and tri-carboxylic acid transporter subfamily			
4604	-35.64	kd	CGS001-9854	C2CD2L	-			
4605	-35.67	oe	ccsbBroad304_12226	NAGK	-			
4606	-35.69	kd	CGS001-23380	SRGAP2	Rho GTPase activating proteins			
4607	-35.75	oe	ccsbBroad304_01446	RPS3A	S ribosomal proteins			
4608	-35.76	kd	CGS001-11065	UBE2C	Ubiquitin-conjugating enzymes E2			
4609	-35.77	oe	ccsbBroad304_00632	GGCX	Carboxylases			
4610	-35.77	kd	CGS001-22944	KIN	-			
4611	-35.81	cp	BRD-A15493168	tetracycline	Bacterial 30S ribosomal subunit inhibitor		PRNP	Bacterial 30S ribosomal subunit inhibitor
4612	-35.84	cp	BRD-K41337261	ZM-306416	ABL inhibitor		FLT1, KDR, EGFR, FLT4	ABL inhibitor, SRC inhibitor, VEGFR inhibitor
4613	-35.86	oe	ccsbBroad304_01321	PSMD5	Proteasome (prosome, macropain) subunits			
4614	-35.89	cp	BRD-K89930444	AG-592	Tyrosine kinase inhibitor			Tyrosine kinase inhibitor
4615	-35.91	cp	BRD-K79116891	proxymetacaine	Sodium channel blocker		SCN10A, SCN5A, SCN9A	Sodium channel blocker
4616	-35.94	cp	BRD-K40990712	hexamethyleneamiloride	Sodium/hydrogen antiport inhibitor		GNRHR, ADRA2A, GNRH1, PLAU, SLC9A1	Sodium/hydrogen antiport inhibitor
4617	-35.94	kd	CGS001-955	ENTPD6	-			
4618	-35.99	cp	BRD-A21723284	naltriben	Opioid receptor antagonist		OPRD1, OPRK1, OPRM1	Opioid receptor antagonist
4619	-35.99	kd	CGS001-115650	TNFRSF13C	Tumour necrosis factor (TNF) receptor family			
4620	-36.01	oe	ccsbBroad304_00620	GCDH	-			
4621	-36.08	cp	BRD-K50938786	ropivacaine	Sodium channel blocker		SCN10A, SCN9A	Sodium channel blocker
4622	-36.11	kd	CGS001-2155	F7	Chymotrypsin			
4623	-36.14	oe	ccsbBroad304_08365	CYCS	-			
4624	-36.16	oe	ccsbBroad304_08694	TBX20	T-boxes			
4625	-36.18	cp	BRD-K74402642	NSC-632839	Ubiquitin specific protease inhibitor		USP2, USP7, SENP2, USP1	Ubiquitin specific protease inhibitor
4626	-36.2	oe	ccsbBroad304_02458	STK25	YSK subfamily			
4627	-36.22	oe	ccsbBroad304_08055	ATP5S	-			
4628	-36.22	cp	BRD-A93236127	digitoxin	ATPase inhibitor		ATP1A1	ATPase inhibitor
4629	-36.24	kd	CGS001-1026	CDKN1A	-			
4630	-36.26	cp	BRD-K67537649	PQ-401	IGF-1 inhibitor		IGF1R	IGF-1 inhibitor, IGF-1R inhibitor
4631	-36.32	cp	BRD-K32330832	VER-155008	HSP inhibitor		HSPA1A	HSP inhibitor
4632	-36.33	kd	CGS001-128674	PROKR2	GPCR / Class A : Prokineticin receptors			
4633	-36.39	oe	ccsbBroad304_02596	KDELR3	-			
4634	-36.41	cp	BRD-A16444946	acarbose	Glucosidase inhibitor		GAA, MGAM, AMY2A, SI	Glucosidase inhibitor
4635	-36.41	cp	BRD-A72483914	spiroxatrine	Serotonin receptor antagonist		HTR1A, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, HTR2B	Serotonin receptor antagonist
4636	-36.45	oe	ccsbBroad304_06538	LSP1	-			
4637	-36.48	kd	CGS001-2853	GPR31	GPCR / Class A : Orphans			
4638	-36.49	oe	ccsbBroad304_05882	BCL6	BTB/POZ domain containing			
4639	-36.49	cp	BRD-K36258877	AZ-10417808	Caspase inhibitor		CASP3	Caspase inhibitor
4640	-36.49	oe	ccsbBroad304_03441	UGT1A9	UDP glucuronosyltransferases			
4641	-36.51	kd	CGS001-5916	RARG	Retinoic acid receptors			
4642	-36.53	cp	BRD-K65331431	retinyl	vitamin analog			vitamin analog
4643	-36.58	oe	ccsbBroad304_05823	ANXA2	Annexins			
4644	-36.6	oe	ccsbBroad304_01985	EIF3H	-			
4645	-36.6	kd	CGS001-7020	TFAP2A	-			
4646	-36.61	kd	CGS001-9146	HGS	Zinc fingers, FYVE domain containing			
4647	-36.62	cp	BRD-K82795137	loratadine	Histamine receptor antagonist		HRH1, CYP2C19, CYP3A5	Histamine receptor antagonist
4648	-36.63	cp	BRD-K79124250	ioxaglic-acid	Radiopaque medium			Radiopaque medium
4649	-36.7	cc		Mediator complex LOF	-			
4650	-36.71	kd	CGS001-6535	SLC6A8	GABA transporter subfamily			
4651	-36.72	oe	ccsbBroad304_01979	AKR1C3	Prostaglandin synthases			
4652	-36.72	kd	CGS001-1727	CYB5R3	-			
4653	-36.77	cp	BRD-A60245366	AS-601245	JNK inhibitor		GSK3B, MAPK10, MAPK8, MAPK9, PIM1	JNK inhibitor
4654	-36.84	oe	ccsbBroad304_02671	ECD	-			
4655	-36.85	cp	BRD-A73368467	fexofenadine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
4656	-36.85	kd	CGS001-10730	YME1L1	ATPases / AAA-type			
4657	-36.86	cp	BRD-K71430621	clobenpropit	Histamine receptor antagonist		HRH3, HRH4, HRH1, HRH2	Histamine receptor antagonist
4658	-36.89	oe	ccsbBroad304_01588	SPP1	Endogenous ligands			
4659	-36.91	kd	CGS001-22933	SIRT2	Histone deacetylases			
4660	-36.93	kd	CGS001-64215	DNAJC1	Heat shock proteins / DNAJ (HSP40)			
4661	-36.95	oe	ccsbBroad304_06856	RET	Type XIV RTKs: RET			
4662	-36.97	kd	CGS001-10127	ZNF263	Zinc fingers, C2H2-type			
4663	-36.99	oe	ccsbBroad304_03310	LCMT1	-			
4664	-36.99	kd	CGS001-2547	XRCC6	XRCC DNA Repair			
4665	-36.99	kd	CGS001-159296	NKX2-3	Homeoboxes / ANTP class : NKL subclass			
4666	-37.05	cp	BRD-K69328504	L-690488	Inositol monophosphatase inhibitor		IMPA1	Inositol monophosphatase inhibitor
4667	-37.05	cp	BRD-K49448285	bisindolylmaleimide	CDK inhibitor		CCND1, CDK4, LRRK2, PDPK1, PIM1, PRKCA, PRKCB, PRKCI, PRKCZ	CDK inhibitor
4668	-37.06	cp	BRD-K98490050	amsacrine	Topoisomerase inhibitor		TOP2A, KCNH2	Topoisomerase inhibitor
4669	-37.1	cp	BRD-K01624546	docosatrienoic-acid	LTB4 inhibitor			LTB4 inhibitor
4670	-37.1	kd	CGS001-9252	RPS6KA5	MSK subfamily			
4671	-37.12	cp	BRD-K31611373	fluprostenol	Prostanoid receptor agonist		PTGER3, PTGFR, TBXA2R	Prostanoid receptor agonist
4672	-37.12	kd	CGS001-7295	TXN	-			
4673	-37.13	kd	CGS001-351	APP	Endogenous ligands			
4674	-37.14	cp	BRD-K54529596	captopril	ACE inhibitor		ACE, LTA4H, MMP2, MMP9	ACE inhibitor
4675	-37.16	oe	ccsbBroad304_06907	S100A13	S100 calcium binding proteins			
4676	-37.18	cp	BRD-A79237180	ascorbic-acid	Antioxidant		AKR1B1	Antioxidant
4677	-37.18	kd	CGS001-83873	GPR61	GPCR / Class A : Orphans			
4678	-37.19	cp	BRD-K62609077	scoulerine	Adrenergic receptor antagonist		ADRA1D, ADRA2A, GABRA1	Adrenergic receptor antagonist, GABA receptor antagonist, Serotonin receptor antagonist
4679	-37.23	kd	CGS001-23062	GGA2	-			
4680	-37.25	cp	BRD-K28029915	dolasetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
4681	-37.26	kd	CGS001-1611	DAP	-			
4682	-37.27	cc		PRD class homeoboxes and psudogenes LOF	-			
4683	-37.27	oe	ccsbBroad304_07529	AKT3	Akt (Protein kinase B)			
4684	-37.29	cp	BRD-K37798499	etoposide	Topoisomerase inhibitor		TOP2A, CYP2E1, CYP3A5, TOP2B	Topoisomerase inhibitor
4685	-37.34	oe	ccsbBroad304_06048	CRYZ	-			
4686	-37.34	oe	ccsbBroad304_07490	SCRN1	-			
4687	-37.35	kd	CGS001-23325	KIAA1033	-			
4688	-37.52	oe	ccsbBroad304_03853	LSM2	-			
4689	-37.53	kd	CGS001-85004	RERG	-			
4690	-37.55	oe	ccsbBroad304_06773	PRKAR2B	Protein kinase A			
4691	-37.6	cp	BRD-K64606589	apicidin	HDAC inhibitor		HDAC1, HDAC10, HDAC11, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
4692	-37.66	oe	ccsbBroad304_04794	ZFP3	Zinc fingers, C2H2-type			
4693	-37.69	oe	ccsbBroad304_09425	RNF166	RING-type (C3HC4) zinc fingers			
4694	-37.69	oe	ccsbBroad304_08275	TLR8	Toll-like receptor family			
4695	-37.73	oe	ccsbBroad304_05012	CREB3L4	basic leucine zipper proteins			
4696	-37.74	oe	ccsbBroad304_00504	SLC29A1	SLC29 family			
4697	-37.76	cp	BRD-K09436313	prostaglandin	Prostanoid receptor antagonist		AKR1C3, PTGDR, PTGDR2, PTGER1, PTGER2, PTGER4, PTGFR	Prostanoid receptor antagonist
4698	-37.77	kd	CGS001-83448	PUS7L	-			
4699	-37.81	cp	BRD-A47829399	artesunate	DNA synthesis inhibitor			DNA synthesis inhibitor
4700	-37.84	kd	CGS001-256297	PTF1A	Basic helix-loop-helix proteins			
4701	-37.88	kd	CGS001-4726	NDUFS6	Mitochondrial respiratory chain complex / Complex I			
4702	-37.89	cp	BRD-A96107863	nisoldipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA1S, CACNA2D1, CACNB2, CYP3A5	Calcium channel blocker
4703	-37.89	kd	CGS001-8028	MLLT10	Zinc fingers, PHD-type			
4704	-37.9	kd	CGS001-3998	LMAN1	-			
4705	-37.96	kd	CGS001-10957	PNRC1	-			
4706	-38.05	cp	BRD-K64052750	gefitinib	EGFR inhibitor		EGFR, CYP2C19	EGFR inhibitor
4707	-38.15	cp	BRD-K06147391	telenzepine	Acetylcholine receptor antagonist		CHRM1	Acetylcholine receptor antagonist
4708	-38.16	oe	ccsbBroad304_07633	HTATIP2	Short chain dehydrogenase/reductase superfamily / Atypical members			
4709	-38.19	kd	CGS001-54925	ZNF434	-			
4710	-38.34	oe	ccsbBroad304_03945	AKTIP	Ubiquitin-conjugating enzymes E2			
4711	-38.36	oe	ccsbBroad304_06335	GSTP1	Glutathione S-transferases			
4712	-38.36	kd	CGS001-56998	CTNNBIP1	Catenins			
4713	-38.38	kd	CGS001-3791	KDR	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
4714	-38.41	kd	CGS001-116535	MRGPRF	GPCR / Class A : Orphans			
4715	-38.44	kd	CGS001-8315	BRAP	RING-type (C3HC4) zinc fingers			
4716	-38.51	kd	CGS001-57178	ZMIZ1	Zinc fingers, MIZ-type			
4717	-38.61	oe	ccsbBroad304_00060	AMBP	Lipocalins			
4718	-38.63	oe	ccsbBroad304_01720	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4719	-38.63	kd	CGS001-6894	TARBP1	-			
4720	-38.82	kd	CGS001-84527	ZNF559	Zinc fingers, C2H2-type			
4721	-38.87	cp	BRD-K17561142	amiodarone	Potassium channel blocker		KCNH2, ADRB1, CACNA1H, CACNA2D2, CHRM3, CYP2C8, KCNA7, SCN5A	Potassium channel blocker
4722	-38.91	cp	BRD-K29359156	ebselen	H+/K+-ATPase inhibitor		ALB, LTB4R, NOX3	H+/K+-ATPase inhibitor, Cyclooxygenase inhibitor, Glutathione peroxidase agonist, Nitric oxide synthase inhibitor
4723	-39	cp	BRD-A65449987	flunisolide	Cytochrome P450 inhibitor		NR3C1	Cytochrome P450 inhibitor
4724	-39	cp	BRD-A49358627	ciprofibrate	PPAR receptor agonist		PPARA, LPL	PPAR receptor agonist
4725	-39.05	cp	BRD-K30649484	mafenide	Carbonic anhydrase inhibitor		CA6, CA12, CA14, CA2, CA4, CA9	Carbonic anhydrase inhibitor
4726	-39.05	kd	CGS001-56731	SLC2A4RG	-			
4727	-39.06	cp	BRD-K49111258	prazosin	Adrenergic receptor antagonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CDK1, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
4728	-39.11	kd	CGS001-1440	CSF3	Endogenous ligands			
4729	-39.13	cp	BRD-K12002134	megestrol	progesterone receptor agonist		PGR	progesterone receptor agonist
4730	-39.13	kd	CGS001-5793	PTPRG	Receptor tyrosine phosphatases (RTP)			
4731	-39.17	kd	CGS001-9871	SEC24D	-			
4732	-39.21	cp	BRD-K97056771	HY-11007	BCR-ABL kinase inhibitor		ABL1, BCR	BCR-ABL kinase inhibitor
4733	-39.22	kd	CGS001-1613	DAPK3	Death-associated kinase (DAPK) family			
4734	-39.24	kd	CGS001-4616	GADD45B	-			
4735	-39.25	cp	BRD-K26997899	SA-792574	Microtubule inhibitor		TUBB	Microtubule inhibitor
4736	-39.26	kd	CGS001-5599	MAPK8	MAPK:JNK subfamily			
4737	-39.27	kd	CGS001-10574	CCT7	Heat Shock Proteins / Chaperonins			
4738	-39.32	kd	CGS001-5538	PPT1	-			
4739	-39.35	kd	CGS001-11200	CHEK2	CHK1 subfamily			
4740	-39.39	cp	BRD-A72441487	stiripentol	GABA uptake inhibitor		ABAT, SCN1A, SCN3A	GABA uptake inhibitor
4741	-39.46	kd	CGS001-23012	STK38L	NDR family			
4742	-39.46	kd	CGS001-55526	DHTKD1	-			
4743	-39.47	kd	CGS001-5567	PRKACB	Protein kinase A			
4744	-39.5	oe	ccsbBroad304_07935	IFIT5	Tetratricopeptide (TTC) repeat domain containing			
4745	-39.54	oe	ccsbBroad304_05745	CD24	CD molecules			
4746	-39.54	kd	CGS001-9653	HS2ST1	Sulfotransferases, membrane-bound			
4747	-39.57	kd	CGS001-6464	SHC1	SH2 domain containing			
4748	-39.64	oe	ccsbBroad304_02028	SOCS2	SH2 domain containing			
4749	-39.71	cp	BRD-K04710043	hexamethylenebisacetamide	AKT inhibitor			AKT inhibitor, Differentiation inducer, NFkB pathway inhibitor
4750	-39.73	oe	ccsbBroad304_00773	HOXA9	Homeoboxes / ANTP class : HOXL subclass			
4751	-39.75	oe	ccsbBroad304_09831	CERS3	Homeoboxes / CERS class			
4752	-39.76	cp	BRD-A24191444	ifenprodil	Adrenergic receptor antagonist		GRIN1, GRIN2B	Adrenergic receptor antagonist, Glutamate receptor antagonist
4753	-39.78	oe	ccsbBroad304_07140	XPC	-			
4754	-39.8	oe	ccsbBroad304_04718	RPL39L	L ribosomal proteins			
4755	-39.8	kd	CGS001-9406	ZRANB2	Zinc fingers, RAN-binding domain containing			
4756	-39.82	oe	ccsbBroad304_09309	CREB3L1	basic leucine zipper proteins			
4757	-39.82	oe	ccsbBroad304_00117	ATF4	basic leucine zipper proteins			
4758	-39.84	oe	ccsbBroad304_01418	RPL7	L ribosomal proteins			
4759	-39.84	oe	ccsbBroad304_00600	FYN	Src family			
4760	-39.87	cp	BRD-A24543851	nornicotine	Acetylcholine receptor agonist			Acetylcholine receptor agonist
4761	-39.89	cp	BRD-K06895174	cisapride	Serotonin receptor agonist		HTR4, KCNH2, CYP2B6, CYP2C8, CYP3A5, CYP3A7, HTR2A, HTR3A	Serotonin receptor agonist
4762	-39.9	cp	BRD-K30296925	flavokavain-b	Antineoplastic		HIF1A	Antineoplastic
4763	-39.91	kd	CGS001-5105	PCK1	-			
4764	-39.98	cp	BRD-A06352508	SB-218078	CHK inhibitor		CHEK1	CHK inhibitor
4765	-40.06	cp	BRD-K88560311	rucaparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
4766	-40.08	cp	BRD-K76840893	RS-17053	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
4767	-40.09	oe	ccsbBroad304_07145	ZFP161	-			
4768	-40.09	oe	ccsbBroad304_06625	NDUFS4	Mitochondrial respiratory chain complex / Complex I			
4769	-40.1	cp	BRD-A66435872	HTMT	Histamine receptor agonist		HRH4	Histamine receptor agonist
4770	-40.14	cp	BRD-K47150025	KI-8751	VEGFR inhibitor		KDR	VEGFR inhibitor, KIT inhibitor, PDGFR receptor inhibitor
4771	-40.16	kd	CGS001-5710	PSMD4	Proteasome (prosome, macropain) subunits			
4772	-40.21	oe	ccsbBroad304_01825	SLC30A2	SLC30 zinc transporter family			
4773	-40.21	cp	BRD-K42142750	retrorsine	Antimitotic			Antimitotic, Cytotoxic agent, Mutagenic
4774	-40.25	oe	ccsbBroad304_03555	PANK4	-			
4775	-40.25	kd	CGS001-1852	DUSP9	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
4776	-40.28	kd	CGS001-2786	GNG4	-			
4777	-40.29	kd	CGS001-57720	GPR107	GPCR / Unclassified : 7TM orphan receptors			
4778	-40.29	kd	CGS001-196	AHR	Basic helix-loop-helix proteins			
4779	-40.35	oe	ccsbBroad304_07976	RNF167	RING-type (C3HC4) zinc fingers			
4780	-40.36	kd	CGS001-54546	RNF186	RING-type (C3HC4) zinc fingers			
4781	-40.37	kd	CGS001-27154	BRPF3	Non-enzymatic BRD containing proteins			
4782	-40.43	oe	ccsbBroad304_07006	ST14	Serine peptidases / Transmembrane			
4783	-40.45	kd	CGS001-3556	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
4784	-40.52	cp	BRD-A43940795	tetrahydropalmatine	Serotonin release inhibitor			Serotonin release inhibitor
4785	-40.52	kd	CGS001-126295	ZNF57	Zinc fingers, C2H2-type			
4786	-40.53	cp	BRD-K92049597	triamterene	Sodium channel blocker		SCNN1A, SCNN1B, SCNN1G, SCNN1D	Sodium channel blocker
4787	-40.55	kd	CGS001-7090	TLE3	WD repeat domain containing			
4788	-40.59	oe	ccsbBroad304_01377	RARG	Retinoic acid receptors			
4789	-40.64	kd	CGS001-79142	PHF23	Zinc fingers, PHD-type			
4790	-40.7	oe	ccsbBroad304_00991	MDH1	-			
4791	-40.7	kd	CGS001-54941	RNF125	RING-type (C3HC4) zinc fingers			
4792	-40.75	oe	ccsbBroad304_00272	CDC25A	Protein tyrosine phosphatases / Class III Cys-based PTPs			
4793	-40.75	kd	CGS001-5775	PTPN4	Protein tyrosine phosphatases			
4794	-40.77	oe	ccsbBroad304_07531	TANK	-			
4795	-40.94	cp	BRD-K48168960	propylthiouracil	Thyroid peroxidase inhibitor		TPO, DIO1	Thyroid peroxidase inhibitor
4796	-41.03	cp	BRD-A39255369	DCPIB	Chloride channel blocker		SLC1A2	Chloride channel blocker, Gap junction modulator, Glutamate inhibitor
4797	-41.05	kd	CGS001-435	ASL	-			
4798	-41.12	oe	ccsbBroad304_09391	DTX2	RING-type (C3HC4) zinc fingers			
4799	-41.17	kd	CGS001-3718	JAK3	Janus kinase (JakA) family			
4800	-41.18	oe	ccsbBroad304_04190	CCDC92	-			
4801	-41.24	kd	CGS001-7029	TFDP2	-			
4802	-41.28	kd	CGS001-10295	BCKDK	Pyruvate dehydrogenase kinase (PDHK) family			
4803	-41.3	oe	ccsbBroad304_03445	UGT1A1	UDP glucuronosyltransferases			
4804	-41.3	kd	CGS001-85236	HIST1H2BK	Histones / Replication-dependent			
4805	-41.39	cp	BRD-K96037667	norethindrone	Progesterone receptor agonist		PGR	Progesterone receptor agonist, Progestogen hormone
4806	-41.43	oe	ccsbBroad304_01205	PIN1	-			
4807	-41.45	oe	ccsbBroad304_00614	GAMT	-			
4808	-41.5	cp	BRD-K55430733	WAY-629	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
4809	-41.52	oe	ccsbBroad304_00859	IL12A	Interleukins and interleukin receptors			
4810	-41.53	cc		PI3K inhibitor	-			
4811	-41.53	oe	ccsbBroad304_01144	PAK1	PAKA subfamily			
4812	-41.53	kd	CGS001-5727	PTCH1	-			
4813	-41.56	cp	BRD-U25771771	WZ-4-145	EGFR inhibitor		CSF1R, DDR1, EGFR, PDGFRA, TIE1	EGFR inhibitor
4814	-41.61	cp	BRD-A31575449	CGP-20712	Adrenergic receptor antagonist		ADRB1, ADRB3	Adrenergic receptor antagonist
4815	-41.69	cp	BRD-K39462424	dexchlorpheniramine	Histamine receptor antagonist			Histamine receptor antagonist
4816	-41.82	kd	CGS001-10284	SAP18	-			
4817	-41.85	oe	ccsbBroad304_00849	IL4	Interleukins and interleukin receptors			
4818	-41.87	oe	ccsbBroad304_05142	OLIG3	Basic helix-loop-helix proteins			
4819	-41.89	kd	CGS001-638	BIK	-			
4820	-41.92	oe	ccsbBroad304_09934	MKX	Homeoboxes / TALE class			
4821	-42.01	oe	ccsbBroad304_00115	ASPH	-			
4822	-42.03	cp	BRD-A70649075	sulconazole	Sterol demethylase inhibitor			Sterol demethylase inhibitor
4823	-42.05	oe	ccsbBroad304_03271	ECSIT	Mitochondrial respiratory chain complex assembly factors			
4824	-42.09	oe	ccsbBroad304_13847	DUSP3	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
4825	-42.15	kd	CGS001-3706	ITPKA	Inositol 1,4,5-trisphosphate 3-kinases			
4826	-42.19	kd	CGS001-5290	PIK3CA	Phosphatidylinositol kinases			
4827	-42.19	kd	CGS001-2189	FANCG	Fanconi anemia, complementation groups			
4828	-42.22	oe	ccsbBroad304_07183	BRPF1	Non-enzymatic BRD containing proteins			
4829	-42.22	kd	CGS001-9375	TM9SF2	-			
4830	-42.25	cp	BRD-K70557564	zosuquidar	P-glycoprotein inhibitor		ABCB1, ABCB4	P-glycoprotein inhibitor
4831	-42.27	kd	CGS001-5336	PLCG2	Phosphoinositide-specific phospholipase C			
4832	-42.29	oe	ccsbBroad304_08742	ZNF398	Zinc fingers, C2H2-type			
4833	-42.3	cp	BRD-K14888893	minoxidil	KATP activator		KCNJ8, ABCC9, KCNJ1, KCNJ10, KCNJ11, PTGS1, REN	KATP activator, KIR6 channel (KATP) activator, Vasodilator
4834	-42.37	cp	BRD-K48932581	cetraxate	Mucus protecting agent		GAST	Mucus protecting agent
4835	-42.42	kd	CGS001-4088	SMAD3	SMADs			
4836	-42.42	kd	CGS001-10670	RRAGA	-			
4837	-42.45	cp	BRD-K41410256	balsalazide	Cyclooxygenase inhibitor		PTGS1, PTGS2, ALOX5, PPARG	Cyclooxygenase inhibitor
4838	-42.48	oe	ccsbBroad304_05394	ZNF621	Zinc fingers, C2H2-type			
4839	-42.48	kd	CGS001-8720	MBTPS1	Subtilisin			
4840	-42.51	kd	CGS001-208	AKT2	Akt (Protein kinase B)			
4841	-42.52	oe	ccsbBroad304_01261	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4842	-42.55	kd	CGS001-2967	GTF2H3	General transcription factors			
4843	-42.58	kd	CGS001-51569	UFM1	-			
4844	-42.58	kd	CGS001-8905	AP1S2	-			
4845	-42.6	kd	CGS001-9618	TRAF4	RING-type (C3HC4) zinc fingers			
4846	-42.63	oe	ccsbBroad304_06736	PLCG2	Phosphoinositide-specific phospholipase C			
4847	-42.64	cc		Gamma secretase inhibitor	-			
4848	-42.64	kd	CGS001-8850	KAT2B	Histone acetyltransferases (HATs)			
4849	-42.73	kd	CGS001-5321	PLA2G4A	Phospholipase A2			
4850	-42.74	kd	CGS001-4094	MAF	-			
4851	-42.82	oe	ccsbBroad304_09177	EFCAB2	EF-hand domain containing			
4852	-42.84	oe	ccsbBroad304_10901	IGF1R	Type II RTKs: Insulin receptor family			
4853	-42.86	cp	BRD-K60298136	ITE	Aryl hydrocarbon receptor agonist		AHR	Aryl hydrocarbon receptor agonist
4854	-42.86	kd	CGS001-5580	PRKCD	Delta subfamily			
4855	-42.87	cc		Serotonin receptor agonist	-			
4856	-42.87	oe	ccsbBroad304_03554	NAT10	-			
4857	-42.91	cp	BRD-K64610608	EMF-bca1-57	caspase inhibitor		CASP3	caspase inhibitor
4858	-42.91	cp	BRD-A35033682	eriodictyol	Cytochrome P450 inhibitor		CYP1B1, NFE2L2, XDH	Cytochrome P450 inhibitor
4859	-42.93	kd	CGS001-5608	MAP2K6	MAPKK:STE7 family			
4860	-43.04	oe	ccsbBroad304_02822	ARFIP2	-			
4861	-43.05	cp	BRD-K91733562	secoisolariciresinol	Antioxidant			Antioxidant
4862	-43.05	cp	BRD-K36395411	SB-206553	Serotonin receptor antagonist		HTR2B, HTR2C, HTR1A, HTR2A	Serotonin receptor antagonist
4863	-43.07	kd	CGS001-9533	POLR1C	RNA polymerase subunits			
4864	-43.08	cp	BRD-K68392338	ZK-93426	Benzodiazepine receptor antagonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor antagonist
4865	-43.1	cp	BRD-K42500029	CGP-57380	MAP kinase inhibitor		AURKB, LCK, MKNK1, MKNK2, SGK1	MAP kinase inhibitor
4866	-43.14	kd	CGS001-340371	NRBP2	NRBP family			
4867	-43.2	kd	CGS001-11040	PIM2	PIM family			
4868	-43.25	kd	CGS001-2919	CXCL1	Endogenous ligands			
4869	-43.26	cp	BRD-K20742498	RS-39604	Serotonin receptor antagonist		HTR4	Serotonin receptor antagonist
4870	-43.26	kd	CGS001-3685	ITGAV	Integrins			
4871	-43.32	oe	ccsbBroad304_03311	EVL	-			
4872	-43.34	kd	CGS001-1910	EDNRB	Endothelin receptors			
4873	-43.35	cp	BRD-A64479082	quinidine	Sodium channel blocker		SCN5A, ABCB1, CYP2D6, KCNA5, KCNA7, KCNH1, KCNH2, KCNH5, KCNK1, KCNK6, SLC29A4	Sodium channel blocker
4874	-43.38	oe	ccsbBroad304_02801	CASP14	Caspases			
4875	-43.42	cp	BRD-A80638690	floxuridine	DNA synthesis inhibitor		TYMS	DNA synthesis inhibitor
4876	-43.42	cp	BRD-M00539986	formoterol	Adrenergic receptor agonist		ADRB2, CYP2C19	Adrenergic receptor agonist
4877	-43.48	oe	ccsbBroad304_01091	NFIB	-			
4878	-43.49	oe	ccsbBroad304_06462	ITGAE	Integrins			
4879	-43.5	oe	ccsbBroad304_03659	FOXJ2	Forkhead boxes			
4880	-43.51	kd	CGS001-397	ARHGDIB	Endogenous ligands			
4881	-43.52	oe	ccsbBroad304_06619	NCF2	Tetratricopeptide (TTC) repeat domain containing			
4882	-43.52	kd	CGS001-2058	EPRS	Aminoacyl tRNA synthetases / Class I			
4883	-43.54	cp	BRD-A81177136	KN-62	Calcium-calmodulin dependent protein kinase inhibitor		AKT1, CAMK2A, CHEK1, LCK, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, P2RX7, PRKCA, ROCK1, RPS6KB1, SGK1	Calcium-calmodulin dependent protein kinase inhibitor, Purinergic receptor antagonist
4884	-43.54	kd	CGS001-5709	PSMD3	Proteasome (prosome, macropain) subunits			
4885	-43.6	kd	CGS001-190	NR0B1	DAX-like receptors			
4886	-43.7	oe	ccsbBroad304_02045	BUD31	-			
4887	-43.7	oe	ccsbBroad304_03798	PHTF2	-			
4888	-43.74	kd	CGS001-56938	ARNTL2	Basic helix-loop-helix proteins			
4889	-43.75	cp	BRD-K03109492	NSC-663284	CDC inhibitor		CDC25A, CDC25B, CDC25C	CDC inhibitor
4890	-43.79	cp	BRD-K93645900	tadalafil	Phosphodiesterase inhibitor		PDE5A, PDE11A	Phosphodiesterase inhibitor
4891	-43.83	oe	ccsbBroad304_09354	IGSF8	CD molecules			
4892	-43.85	kd	CGS001-8864	PER2	-			
4893	-43.87	cp	BRD-K92678294	irilin-a	Isoflavone			Isoflavone
4894	-43.87	kd	CGS001-6788	STK3	MST subfamily			
4895	-43.94	oe	ccsbBroad304_00580	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
4896	-43.98	kd	CGS001-51097	SCCPDH	-			
4897	-43.99	kd	CGS001-6678	SPARC	-			
4898	-44.06	oe	ccsbBroad304_07605	LYPLA1	-			
4899	-44.06	cp	BRD-A56245458	reichstein	Androgen receptor antagonist		AR	Androgen receptor antagonist
4900	-44.15	oe	ccsbBroad304_02571	TOMM34	Tetratricopeptide (TTC) repeat domain containing			
4901	-44.2	kd	CGS001-5817	PVR	Immunoglobulin superfamily / C2-set domain containing			
4902	-44.23	kd	CGS001-5664	PSEN2	Presenilin			
4903	-44.24	oe	ccsbBroad304_04690	ZNF653	Zinc fingers, C2H2-type			
4904	-44.24	kd	CGS001-6895	TARBP2	-			
4905	-44.28	oe	ccsbBroad304_07667	CGRRF1	RING-type (C3HC4) zinc fingers			
4906	-44.3	oe	ccsbBroad304_05970	CDC20	WD repeat domain containing			
4907	-44.3	kd	CGS001-24149	ZNF318	Zinc fingers, C2H2-type			
4908	-44.35	kd	CGS001-6197	RPS6KA3	RSK subfamily			
4909	-44.36	cp	BRD-K47869605	podophyllotoxin	Microtubule inhibitor		IGF1R, CASP3, TOP2A, TUBA4A, TUBB	Microtubule inhibitor, Tubulin inhibitor
4910	-44.37	cp	BRD-A62025033	temsirolimus	MTOR inhibitor		MTOR, PTEN	MTOR inhibitor
4911	-44.37	kd	CGS001-55278	QRSL1	-			
4912	-44.47	kd	CGS001-81544	GDPD5	-			
4913	-44.51	kd	CGS001-81539	SLC38A1	System A-like transporters			
4914	-44.53	kd	CGS001-488	ATP2A2	Calcium-ATPases			
4915	-44.57	cp	BRD-K25394294	oxaprozin	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
4916	-44.61	cp	BRD-K13566078	BMS-345541	IKK inhibitor		IKBKB, CHUK	IKK inhibitor
4917	-44.63	oe	ccsbBroad304_09233	GPR128	Adhesion Class GPCRs			
4918	-44.63	kd	CGS001-5660	PSAP	Endogenous ligands			
4919	-44.64	oe	ccsbBroad304_00380	CSNK1G2	Casein kinase 1 (CK1) family			
4920	-44.69	oe	ccsbBroad304_03351	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
4921	-44.71	kd	CGS001-7048	TGFBR2	Type II receptor serine/threonine kinases			
4922	-44.71	kd	CGS001-6272	SORT1	-			
4923	-44.74	oe	ccsbBroad304_05868	ATP5C1	ATPases / F-type			
4924	-44.86	oe	ccsbBroad304_00695	CXCL1	Endogenous ligands			
4925	-44.88	cp	BRD-K88568253	iproniazid	Monoamine oxidase inhibitor		MAOA, MAOB	Monoamine oxidase inhibitor
4926	-44.91	kd	CGS001-23224	SYNE2	-			
4927	-44.93	oe	ccsbBroad304_09708	PNLDC1	-			
4928	-44.98	kd	CGS001-4846	NOS3	Nitric oxide synthases			
4929	-45	cp	BRD-K25311561	KU-55933	ATM kinase inhibitor		ATM, PRKDC	ATM kinase inhibitor
4930	-45.1	oe	ccsbBroad304_02423	CD2BP2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
4931	-45.12	kd	CGS001-79174	CRELD2	-			
4932	-45.15	oe	ccsbBroad304_00706	GTF2B	General transcription factors			
4933	-45.23	oe	ccsbBroad304_04379	LZIC	-			
4934	-45.23	cp	BRD-K21733600	rofecoxib	Cyclooxygenase inhibitor		PTGS2, CYP3A4, ELN	Cyclooxygenase inhibitor
4935	-45.25	kd	CGS001-4144	MAT2A	-			
4936	-45.28	oe	ccsbBroad304_06381	HMGB1	High-mobility group / Canonical			
4937	-45.31	oe	ccsbBroad304_08888	ACD	-			
4938	-45.32	oe	ccsbBroad304_13912	NDUFB1	Mitochondrial respiratory chain complex / Complex I			
4939	-45.35	oe	ccsbBroad304_09445	MRGPRX3	GPCR / Class A : Orphans			
4940	-45.46	kd	CGS001-4864	NPC1	-			
4941	-45.47	kd	CGS001-25966	C2CD2	-			
4942	-45.54	kd	CGS001-226	ALDOA	-			
4943	-45.63	oe	ccsbBroad304_02376	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
4944	-45.73	kd	CGS001-440	ASNS	-			
4945	-45.78	kd	CGS001-2118	ETV4	ETS Transcription Factors			
4946	-45.84	cp	BRD-K82983861	GW-0742	PPAR receptor agonist		INS, PPARD	PPAR receptor agonist, Insulin sensitizer
4947	-45.85	oe	ccsbBroad304_02040	NAE1	Ubiquitin-like modifier activating enzymes			
4948	-45.85	kd	CGS001-1019	CDK4	Cyclin-dependent kinases, CDK4 subfamily			
4949	-45.97	oe	ccsbBroad304_02139	HMGN3	High-mobility group / Canonical			
4950	-45.98	kd	CGS001-5782	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
4951	-46.01	cp	BRD-K60640630	mometasone	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist, Immunosuppressant
4952	-46.07	cp	BRD-K65639003	icariin	Phosphodiesterase inhibitor		NMUR2, PDE5A, SORD	Phosphodiesterase inhibitor
4953	-46.09	cp	BRD-K07220430	cinnarizine	Calcium channel blocker		HRH1, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD2, DRD5	Calcium channel blocker
4954	-46.18	oe	ccsbBroad304_02509	GMEB1	-			
4955	-46.23	cp	BRD-K95785537	PP-2	SRC inhibitor		SRC, LCK, ABL1, LYN, RIPK2	SRC inhibitor
4956	-46.25	kd	CGS001-23483	TGDS	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
4957	-46.3	kd	CGS001-5900	RALGDS	-			
4958	-46.3	kd	CGS001-8895	CPNE3	-			
4959	-46.31	oe	ccsbBroad304_01147	PC	Carboxylases			
4960	-46.32	kd	CGS001-7391	USF1	Basic helix-loop-helix proteins			
4961	-46.35	kd	CGS001-595	CCND1	-			
4962	-46.46	oe	ccsbBroad304_06658	NT5E	Adenosine turnover			
4963	-46.46	kd	CGS001-55810	FOXJ2	Forkhead boxes			
4964	-46.47	cc		PKC activator	-			
4965	-46.48	cp	BRD-K54094468	remoxipride	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, SIGMAR1	Dopamine receptor antagonist
4966	-46.51	cp	BRD-A09722536	cyclophosphamide	DNA alkylating agent		BCL2, CYP2B6, CYP2C19, CYP3A5, LGALS1	DNA alkylating agent
4967	-46.56	cp	BRD-K66874953	pifithrin-alpha	TP53 inhibitor		TP53	TP53 inhibitor
4968	-46.57	oe	ccsbBroad304_02121	UBE2L6	Ubiquitin-conjugating enzymes E2			
4969	-46.59	oe	ccsbBroad304_07491	IP6K1	-			
4970	-46.61	oe	ccsbBroad304_01342	PTPN6	Protein tyrosine phosphatases			
4971	-46.66	kd	CGS001-7915	ALDH5A1	Aldehyde dehydrogenases			
4972	-46.68	oe	ccsbBroad304_01443	MRPL12	Mitochondrial ribosomal proteins / large subunits			
4973	-46.7	kd	CGS001-2021	ENDOG	-			
4974	-46.72	cp	BRD-K59369769	tozasertib	Aurora kinase inhibitor		AURKA, AURKB, ABL1, AURKC, BCR, FLT3, JAK2, DDR2, LCK	Aurora kinase inhibitor, BCR-ABL kinase inhibitor, FLT3 inhibitor, JAK inhibitor
4975	-46.77	kd	CGS001-7291	TWIST1	Basic helix-loop-helix proteins			
4976	-46.86	kd	CGS001-5581	PRKCE	Eta subfamily			
4977	-46.87	cc		Akt Signaling GOF	-			
4978	-46.92	kd	CGS001-7024	TFCP2	-			
4979	-46.93	kd	CGS001-81856	ZNF611	Zinc fingers, C2H2-type			
4980	-46.94	oe	ccsbBroad304_04619	GNG8	-			
4981	-46.99	kd	CGS001-6499	SKIV2L	-			
4982	-47.01	oe	ccsbBroad304_00795	HSF2	-			
4983	-47.03	oe	ccsbBroad304_07029	TADA2A	-			
4984	-47.04	kd	CGS001-57117	INTS12	Zinc fingers, PHD-type			
4985	-47.09	oe	ccsbBroad304_02815	SSBP2	-			
4986	-47.1	cp	BRD-K93325701	damnacanthal	SRC inhibitor			SRC inhibitor
4987	-47.18	cp	BRD-K03842655	penitrem-a	Potassium channel blocker		KCNMA1	Potassium channel blocker
4988	-47.21	oe	ccsbBroad304_14291	GDPD5	-			
4989	-47.27	cp	BRD-K01436366	XMD-1150	Leucine rich repeat kinase inhibitor		LRRK2	Leucine rich repeat kinase inhibitor
4990	-47.28	cp	BRD-K67277431	picotamide	Thromboxane receptor antagonist		TBXA2R, TBXAS1	Thromboxane receptor antagonist, Thromboxane synthase inhibitor
4991	-47.28	cp	BRD-K61951118	FG-7142	GABA benzodiazepine site receptor inverse agonist			GABA benzodiazepine site receptor inverse agonist
4992	-47.29	oe	ccsbBroad304_01203	PIM1	PIM family			
4993	-47.29	oe	ccsbBroad304_01267	PPP4C	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
4994	-47.33	kd	CGS001-1969	EPHA2	Type XIII RTKs: Ephrin receptor family			
4995	-47.41	cp	BRD-K67868012	PI-103	MTOR inhibitor		PIK3CA, PIK3CG, MTOR, PIK3CB, PIK3CD, PRKDC	MTOR inhibitor, PI3K inhibitor
4996	-47.46	cc		PKC inhibitor	-			
4997	-47.54	oe	ccsbBroad304_00070	ANXA5	Annexins			
4998	-47.71	cp	BRD-A29437505	RWJ-21757	TLR agonist		TLR7	TLR agonist
4999	-47.75	kd	CGS001-5255	PHKA1	-			
5000	-47.78	cp	BRD-K56343971	vemurafenib	RAF inhibitor		BRAF, CYP2C19, CYP3A4, CYP3A5, RAF1	RAF inhibitor
5001	-47.79	oe	ccsbBroad304_00256	TNFSF8	CD molecules			
5002	-47.79	kd	CGS001-64921	CASD1	-			
5003	-47.83	cp	BRD-K36737713	AG-957	Protein tyrosine kinase inhibitor		ABL1, EGFR	Protein tyrosine kinase inhibitor
5004	-47.96	oe	ccsbBroad304_00728	HBE1	-			
5005	-47.98	kd	CGS001-23596	OPN3	GPCR / Class A : Opsin receptors			
5006	-48	oe	ccsbBroad304_07244	GPR65	GPCR / Class A : Orphans			
5007	-48.02	cp	BRD-K55677650	CO-101244	Ionotropic glutamate receptor antagonist		GRIN2B	Ionotropic glutamate receptor antagonist
5008	-48.04	cc		HRH1 antagonist	-			
5009	-48.04	oe	ccsbBroad304_02063	SLC25A14	Mitochondrial uncoupling proteins			
5010	-48.07	cp	BRD-K77175907	calcifediol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
5011	-48.08	oe	ccsbBroad304_02032	TSC22D1	-			
5012	-48.1	oe	ccsbBroad304_09648	ZNF548	Zinc fingers, C2H2-type			
5013	-48.17	cp	BRD-K28907958	CD-437	Retinoid receptor agonist		RARG	Retinoid receptor agonist
5014	-48.21	oe	ccsbBroad304_01394	RFX4	-			
5015	-48.22	oe	ccsbBroad304_00975	MAT2A	-			
5016	-48.22	cp	BRD-K18194590	mephentermine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3	Adrenergic receptor agonist
5017	-48.25	kd	CGS001-27035	NOX1	-			
5018	-48.33	cp	BRD-K46424862	hymecromone	Monoamine oxidase inhibitor		MAOA	Monoamine oxidase inhibitor
5019	-48.33	cp	BRD-K70881766	solanine	Acetylcholinesterase inhibitor			Acetylcholinesterase inhibitor
5020	-48.37	cp	BRD-K99063460	didanosine	Nucleoside reverse transcriptase inhibitor		PNP	Nucleoside reverse transcriptase inhibitor
5021	-48.42	oe	ccsbBroad304_14242	MCCC2	-			
5022	-48.47	oe	ccsbBroad304_14044	PCGF3	Polycomb group ring fingers			
5023	-48.54	cp	BRD-A50928468	norgestrel	Progesterone receptor agonist		CYP2E1, PGR	Progesterone receptor agonist
5024	-48.57	kd	CGS001-23047	PDS5B	-			
5025	-48.59	oe	ccsbBroad304_01872	DGCR14	-			
5026	-48.6	cp	BRD-K54330070	SB-202190	p38 MAPK inhibitor		MAPK14, AKT1, ALOX5, CHEK1, GSK3B, LCK, MAPK1, MAPK11, MAPK12, MAPK8, PRKCA, ROCK1, RPS6KB1, SGK1	p38 MAPK inhibitor
5027	-48.62	oe	ccsbBroad304_08805	SLC22A23	Orphan or poorly characterized SLC22 family members			
5028	-48.66	kd	CGS001-4833	NME4	-			
5029	-48.71	oe	ccsbBroad304_00077	APEX1	-			
5030	-48.74	oe	ccsbBroad304_00464	DTNA	-			
5031	-48.82	kd	CGS001-2870	GRK6	GRK1/3 subfamily			
5032	-48.83	oe	ccsbBroad304_05049	GPBAR1	Bile acid receptor			
5033	-48.87	kd	CGS001-1184	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
5034	-48.88	kd	CGS001-54541	DDIT4	-			
5035	-48.91	kd	CGS001-5257	PHKB	-			
5036	-49.03	cp	BRD-K94379058	BML-190	Cannabinoid receptor inverse agonist		CNR2	Cannabinoid receptor inverse agonist
5037	-49.05	oe	ccsbBroad304_00956	LYZ	-			
5038	-49.06	kd	CGS001-3337	DNAJB1	Heat shock proteins / DNAJ (HSP40)			
5039	-49.09	kd	CGS001-4436	MSH2	-			
5040	-49.1	oe	ccsbBroad304_06286	GLUL	-			
5041	-49.16	cp	BRD-K04548931	pidorubicine	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
5042	-49.17	oe	ccsbBroad304_10489	CSF3	Endogenous ligands			
5043	-49.23	oe	ccsbBroad304_00867	IMPDH2	Oxidoreductases			
5044	-49.23	kd	CGS001-2634	GBP2	-			
5045	-49.24	oe	ccsbBroad304_00985	MCL1	-			
5046	-49.25	oe	ccsbBroad304_03604	ENOSF1	-			
5047	-49.26	oe	ccsbBroad304_07511	KIF14	Kinesins			
5048	-49.29	cp	BRD-K20197062	SA-94315	Caspase inhibitor		CASP3	Caspase inhibitor
5049	-49.29	kd	CGS001-10097	ACTR2	-			
5050	-49.33	oe	ccsbBroad304_01623	SUPT4H1	-			
5051	-49.35	oe	ccsbBroad304_00329	CLTA	-			
5052	-49.4	cp	BRD-K89210380	biotin	Vitamin B		ACACA, ACACB, HLCS, MCCC1, MCCC2, PC, PCCA, PCCB, SLC5A6	Vitamin B
5053	-49.48	kd	CGS001-7994	KAT6A	Histone acetyltransferases (HATs)			
5054	-49.5	kd	CGS001-9903	KLHL21	BTB/POZ domain containing			
5055	-49.5	kd	CGS001-28964	GIT1	Ankyrin repeat domain containing			
5056	-49.57	oe	ccsbBroad304_08594	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5057	-49.59	cp	BRD-A85280935	quinpirole	Dopamine receptor agonist		DRD2, DRD3, DRD4, DRD1, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor agonist
5058	-49.6	kd	CGS001-9180	OSMR	IL-6 receptor family			
5059	-49.63	kd	CGS001-7494	XBP1	basic leucine zipper proteins			
5060	-49.64	cp	BRD-K86003836	flubendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
5061	-49.69	kd	CGS001-10329	TMEM5	-			
5062	-49.72	cp	BRD-K32412559	morphothebaine	Adrenergic receptor antagonist			Adrenergic receptor antagonist
5063	-49.78	cp	BRD-K02407574	parbendazole	Tubulin inhibitor		TUBB	Tubulin inhibitor
5064	-49.8	oe	ccsbBroad304_00017	ACTN2	EF-hand domain containing			
5065	-49.85	kd	CGS001-1022	CDK7	Cyclin-dependent kinases, CDK7 subfamily			
5066	-49.86	kd	CGS001-27034	ACAD8	-			
5067	-49.88	cp	BRD-K46384212	o-3M3FBS	phospholipase activator			phospholipase activator
5068	-49.98	cp	BRD-K17674993	diflorasone	Corticosteroid agonist		NR3C1, PLA2G1B	Corticosteroid agonist, Glucocorticoid receptor agonist, Cytochrome P450 inhibitor, Immunosuppressant
5069	-49.99	kd	CGS001-1213	CLTC	-			
5070	-50.03	oe	ccsbBroad304_00510	EPHX2	-			
5071	-50.07	oe	ccsbBroad304_04471	C5ORF62	-			
5072	-50.09	cp	BRD-A97730597	hexylcaine	Sodium channel blocker		SCN5A, SCN10A	Sodium channel blocker
5073	-50.09	cp	BRD-K76064317	tyrphostin-AG-1296	FLT3 inhibitor		FLT3	FLT3 inhibitor
5074	-50.11	oe	ccsbBroad304_06481	KCNJ11	Inwardly rectifying potassium channels			
5075	-50.17	oe	ccsbBroad304_06651	NOV	-			
5076	-50.21	cp	BRD-K71799949	carbamazepine	Carboxamide antiepileptic		ABCB1, CYP1A2, CYP3A4, SCN1A, SCN3A, SCN5A	Carboxamide antiepileptic
5077	-50.22	cp	BRD-A66563878	medetomidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
5078	-50.24	cp	BRD-A16478930	amcinonide	Glucocorticoid receptor agonist		NR3C1, ANXA1	Glucocorticoid receptor agonist
5079	-50.26	cp	BRD-A04553218	chlorphenamine	Histamine receptor antagonist		HRH1, SLC6A2, SLC6A3, SLC6A4	Histamine receptor antagonist
5080	-50.31	cp	BRD-K82147103	lofepramine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A4	Norepinephrine reuptake inhibitor, Serotonin reuptake inhibitor
5081	-50.33	oe	ccsbBroad304_10094	ZNF790	Zinc fingers, C2H2-type			
5082	-50.44	cp	BRD-A25067867	benzatropine	Acetylcholine receptor antagonist		CHRM1, HRH1, SLC6A3	Acetylcholine receptor antagonist
5083	-50.45	oe	ccsbBroad304_01372	RALB	-			
5084	-50.49	cp	BRD-A04756508	norgestimate	Progesterone receptor agonist		PGR, ESR1	Progesterone receptor agonist
5085	-50.54	oe	ccsbBroad304_08152	PSAT1	-			
5086	-50.54	kd	CGS001-388	RHOB	-			
5087	-50.56	oe	ccsbBroad304_00862	IL13RA2	IL-2 receptor family			
5088	-50.56	kd	CGS001-1615	DARS	Aminoacyl tRNA synthetases / Class II			
5089	-50.56	cp	BRD-K90027355	spironolactone	Mineralocorticoid receptor antagonist		NR3C2, AR, CACNA1A, CACNA1B, CACNA1C, CACNA1D, CACNA1F, CACNA1G, CACNA1H, CACNA1I, CACNA1S, CACNA2D1, CACNA2D2, CACNA2D3, CACNB1, CACNB2, CACNB3, CACNB4, CACNG1, CYP11B2, KCNA5, KCND3, NR3C1, PGR, SCNN1A, SHBG	Mineralocorticoid receptor antagonist
5090	-50.58	kd	CGS001-54498	SMOX	-			
5091	-50.6	cp	BRD-A78877355	nefopam	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
5092	-50.67	kd	CGS001-958	CD40	Tumour necrosis factor (TNF) receptor family			
5093	-50.7	cp	BRD-K33583600	isoliquiritigenin	Guanylate cyclase activator		AKR1B1, HRH2, SIRT1	Guanylate cyclase activator
5094	-50.7	cp	BRD-K81521265	dicyclohexylurea	Epoxide hydolase inhibitor		EPHX2	Epoxide hydolase inhibitor
5095	-50.74	kd	CGS001-23657	SLC7A11	Solute carriers			
5096	-50.75	cp	BRD-K00234327	RU-24969	Serotonin receptor agonist		HTR1A, HTR1B, HTR6, HTR1D, HTR2A, HTR2B, HTR2C, HTR5A	Serotonin receptor agonist
5097	-50.8	cp	BRD-A25234499	aminoglutethimide	Glucocorticoid receptor antagonist		CYP19A1, CYP11A1, NR3C1	Glucocorticoid receptor antagonist
5098	-50.81	kd	CGS001-79862	ZNF669	Zinc fingers, C2H2-type			
5099	-50.81	cp	BRD-A63998256	helveticoside	ATPase inhibitor		ATP1A1	ATPase inhibitor
5100	-50.83	cp	BRD-K04993501	cefixime	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5101	-50.85	oe	ccsbBroad304_02502	GNA13	-			
5102	-50.88	kd	CGS001-10672	GNA13	-			
5103	-50.91	oe	ccsbBroad304_00747	HLF	-			
5104	-50.96	oe	ccsbBroad304_07888	CBX6	-			
5105	-50.96	cp	BRD-K87142802	veliparib	PARP inhibitor		PARP1, PARP2	PARP inhibitor
5106	-51.03	kd	CGS001-1514	CTSL1	-			
5107	-51.17	cp	BRD-K54233340	dorsomorphin	AMPK inhibitor		ACVR1, BMPR1A, BMPR1B, EPHA2, FKBP1A, FLT1, FLT3, KDR, LCK, MKNK1, PRKAA1, RPS6KA1, SRC	AMPK inhibitor
5108	-51.19	oe	ccsbBroad304_04194	ELL3	-			
5109	-51.31	kd	CGS001-1163	CKS1B	-			
5110	-51.32	oe	ccsbBroad304_03926	SLC39A8	SLC39 family of metal ion transporters			
5111	-51.34	cp	BRD-K94294671	OSI-027	MTOR inhibitor		MTOR	MTOR inhibitor
5112	-51.37	cp	BRD-K83988098	alvespimycin	HSP inhibitor		HSP90AA1	HSP inhibitor
5113	-51.37	oe	ccsbBroad304_09471	CSNK1A1L	Casein kinase 1 (CK1) family			
5114	-51.41	oe	ccsbBroad304_00024	ADCY3	Adenylyl cyclases			
5115	-51.42	oe	ccsbBroad304_07704	SUB1	-			
5116	-51.43	cp	BRD-K53737926	amitriptyline	Norepinephrine inhibitor		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HRH1, HTR6, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRB1, ADRB2, ADRB3, HRH2, HRH4, HTR1A, HTR1B, HTR1D, HTR2A, HTR2C, HTR7, KCNA1, KCND2, KCND3, KCNQ2, KCNQ3, NTRK1, NTRK2, OPRD1, OPRK1, OPRM1, SIGMAR1	Norepinephrine inhibitor, Norepinephrine reuptake inhibitor, Serotonin receptor antagonist, Serotonin reuptake inhibitor
5117	-51.54	kd	CGS001-9706	ULK2	Unc-51-like kinase (ULK) family			
5118	-51.6	kd	CGS001-817	CAMK2D	CAMK2 family			
5119	-51.63	kd	CGS001-10139	ARFRP1	ADP-ribosylation factors			
5120	-51.68	oe	ccsbBroad304_00312	CIRBP	RNA binding motif (RRM) containing			
5121	-51.78	kd	CGS001-8737	RIPK1	Receptor interacting protein kinase (RIPK) family			
5122	-51.8	oe	ccsbBroad304_13985	ZNF200	Zinc fingers, C2H2-type			
5123	-51.83	oe	ccsbBroad304_02956	EHF	-			
5124	-51.86	cp	BRD-K19227686	phenolphthalein	Indicator dye			Indicator dye
5125	-51.95	kd	CGS001-2806	GOT2	-			
5126	-52.03	kd	CGS001-4678	NASP	Tetratricopeptide (TTC) repeat domain containing			
5127	-52.05	oe	ccsbBroad304_07592	CEPT1	-			
5128	-52.06	oe	ccsbBroad304_03544	FAIM	-			
5129	-52.07	cp	BRD-K96319534	phentermine	Dopamine uptake inhibitor		MAOA, MAOB, SLC6A2, SLC6A3, SLC6A4	Dopamine uptake inhibitor, Serotonin reuptake inhibitor
5130	-52.07	cp	BRD-A75402480	desoxycorticosterone	Mineralocorticoid receptor agonist			Mineralocorticoid receptor agonist
5131	-52.09	oe	ccsbBroad304_06336	GSTT1	Glutathione S-transferases / Soluble			
5132	-52.12	oe	ccsbBroad304_01754	UCK2	-			
5133	-52.12	oe	ccsbBroad304_01284	PRKCZ	Iota subfamily			
5134	-52.13	cp	BRD-K81062487	taurocholic-acid	Bile acid		CEL, FXR, NR1H4, FABP6, SLCO1C1	Bile acid
5135	-52.15	oe	ccsbBroad304_08480	PNPO	-			
5136	-52.17	kd	CGS001-1024	CDK8	Cyclin-dependent kinases, CDK8 subfamily			
5137	-52.2	cc		KCNJ11 modulator	-			
5138	-52.31	cp	BRD-A78377521	monastrol	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
5139	-52.32	kd	CGS001-84449	ZNF333	Zinc fingers, C2H2-type			
5140	-52.37	oe	ccsbBroad304_06685	PAH	Amino acid hydroxylases			
5141	-52.4	cp	BRD-K86930074	cediranib	KIT inhibitor		KDR, FLT1, FLT4, KIT, PDGFRB, CSF1R, FLT3, PDGFRA	KIT inhibitor, VEGFR inhibitor
5142	-52.42	oe	ccsbBroad304_00657	GNG4	-			
5143	-52.43	cp	BRD-K17868609	BRL-54443	Serotonin receptor agonist		HTR1E, HTR1F	Serotonin receptor agonist
5144	-52.46	oe	ccsbBroad304_09206	ZGPAT	G patch domain containing			
5145	-52.48	cp	BRD-A48720949	testosterone	androgen receptor agonist		AR, CYP19A1, CYP2C19, CYP2C8, CYP3A5	androgen receptor agonist
5146	-52.48	kd	CGS001-57157	PHTF2	-			
5147	-52.49	oe	ccsbBroad304_13598	NRBP2	NRBP family			
5148	-52.55	kd	CGS001-1384	CRAT	-			
5149	-52.58	oe	ccsbBroad304_01222	PLP2	-			
5150	-52.61	cp	BRD-K68103045	CGS-20625	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5	Benzodiazepine receptor agonist, GABA benzodiazepine site receptor partial agonist
5151	-52.61	kd	CGS001-1605	DAG1	-			
5152	-52.65	oe	ccsbBroad304_09665	SIK1	QIK subfamily			
5153	-52.65	oe	ccsbBroad304_09258	MYLK2	Myosin Light Chain Kinase (MLCK) family			
5154	-52.66	cp	BRD-K48869804	icilin	TRPV agonist		TRPA1, TRPM8	TRPV agonist
5155	-52.72	cp	BRD-K64755930	etazolate	Phosphodiesterase inhibitor		GABRB3, PDE4A	Phosphodiesterase inhibitor
5156	-52.92	kd	CGS001-7037	TFRC	CD molecules			
5157	-52.98	kd	CGS001-6696	SPP1	Endogenous ligands			
5158	-53.03	kd	CGS001-3198	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
5159	-53.03	cp	BRD-A53952395	prilocaine	Local anesthetic		SCN5A	Local anesthetic
5160	-53.07	kd	CGS001-440435	GPR179	GPCR / Class C : Orphans			
5161	-53.11	kd	CGS001-57665	RDH14	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5162	-53.13	cp	BRD-K08998509	fananserin	Dopamine receptor antagonist		HTR2A, DRD4	Dopamine receptor antagonist, Serotonin receptor antagonist
5163	-53.13	kd	CGS001-151126	ZNF385B	-			
5164	-53.14	cp	BRD-K04853698	LDN-193189	Serine/threonine kinase inhibitor		ACVR1, BMPR1A	Serine/threonine kinase inhibitor
5165	-53.21	kd	CGS001-26986	PABPC1	RNA binding motif (RRM) containing			
5166	-53.22	kd	CGS001-5524	PPP2R4	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5167	-53.24	kd	CGS001-2195	FAT1	Cadherins / Cadherin-related			
5168	-53.35	oe	ccsbBroad304_01102	NMT1	-			
5169	-53.36	kd	CGS001-6820	SULT2B1	Sulfotransferases, cytosolic			
5170	-53.43	kd	CGS001-53831	GPR84	GPCR / Class A : Fatty acid receptors			
5171	-53.48	oe	ccsbBroad304_01545	SLC3A2	SLC3 family			
5172	-53.48	cp	BRD-K21853356	RG-14620	EGFR inhibitor		EGFR	EGFR inhibitor
5173	-53.49	kd	CGS001-1959	EGR2	Zinc fingers, C2H2-type			
5174	-53.5	oe	ccsbBroad304_00549	FDX1	-			
5175	-53.5	cp	BRD-K63913457	eicosatrienoic-acid	Vasodilator			Vasodilator
5176	-53.59	cp	BRD-K36740062	GSK-1070916	Aurora kinase inhibitor		AURKB, AURKC, AURKA, CYP2D6, CYP3A4	Aurora kinase inhibitor
5177	-53.61	kd	CGS001-324	APC	Armadillo repeat containing			
5178	-53.64	oe	ccsbBroad304_02140	ZNHIT3	Zinc fingers, HIT-type			
5179	-53.72	oe	ccsbBroad304_02737	JMJD6	-			
5180	-53.72	cp	BRD-K30697463	desoximetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
5181	-53.73	oe	ccsbBroad304_04544	RCCD1	-			
5182	-53.73	oe	ccsbBroad304_00470	DVL2	Dishevelled homologs			
5183	-53.88	oe	ccsbBroad304_07800	EXOSC8	-			
5184	-53.98	cp	BRD-K01192156	tyrphostin-AG-112	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5185	-54	oe	ccsbBroad304_01556	SMARCB1	-			
5186	-54	cp	BRD-K46211610	tolazoline	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, HRH1, HRH2	Adrenergic receptor antagonist
5187	-54.08	oe	ccsbBroad304_04082	SLC52A2	SLC52 family of riboflavin transporters			
5188	-54.15	kd	CGS001-162699	TCEB3C	-			
5189	-54.19	cp	BRD-A96882008	L-732138	Tachykinin antagonist		TACR1, TACR2	Tachykinin antagonist
5190	-54.22	cc		VEGFR inhibitor	-			
5191	-54.35	cp	BRD-K13927029	retinol	Retinoid receptor ligand		ALDH1A1, ALDH1A2, ALDH1A3, DHRS3, DHRS4, LRAT, NR2C2, RBP1, RBP3, RDH11, RDH12, RDH13, RDH14, RDH5, RDH8, RETSAT, RHO, RLBP1, RXRA, RXRB, RXRG	Retinoid receptor ligand
5192	-54.35	kd	CGS001-5359	PLSCR1	-			
5193	-54.35	kd	CGS001-2959	GTF2B	General transcription factors			
5194	-54.53	oe	ccsbBroad304_07427	PIGB	Dolichyl D-mannosyl phosphate dependent mannosyltransferases			
5195	-54.53	kd	CGS001-1465	CSRP1	-			
5196	-54.6	oe	ccsbBroad304_01075	NDUFV1	Mitochondrial respiratory chain complex / Complex I			
5197	-54.61	cp	BRD-K82865713	prostaglandin-b2	cAMP inhibitor			cAMP inhibitor
5198	-54.62	kd	CGS001-1381	CRABP1	Fatty acid-binding proteins			
5199	-54.68	cp	BRD-K51805276	temefos	Cholinesterase inhibitor			Cholinesterase inhibitor
5200	-54.71	oe	ccsbBroad304_02086	PDLIM1	-			
5201	-54.85	oe	ccsbBroad304_08952	E2F8	-			
5202	-54.86	cp	BRD-K92492521	LY-255283	Leukotriene receptor antagonist		LTB4R, LTB4R2	Leukotriene receptor antagonist
5203	-54.87	kd	CGS001-8575	PRKRA	-			
5204	-54.9	kd	CGS001-408	ARRB1	-			
5205	-54.95	oe	ccsbBroad304_07306	TNFRSF10A	Tumour necrosis factor (TNF) receptor family			
5206	-54.99	kd	CGS001-81550	TDRD3	Tudor domain containing			
5207	-55.01	cp	BRD-K51816706	oxindole-I	VEGFR inhibitor		AKT1, KDR, PDPK1, RET	VEGFR inhibitor
5208	-55.03	kd	CGS001-26036	ZNF451	Zinc fingers, C2H2-type			
5209	-55.09	oe	ccsbBroad304_06836	RAD23B	-			
5210	-55.13	kd	CGS001-10051	SMC4	Structural maintenance of chromosomes proteins			
5211	-55.16	kd	CGS001-9380	GRHPR	-			
5212	-55.18	kd	CGS001-55847	CISD1	CDGSH iron sulfur domain containing			
5213	-55.19	kd	CGS001-115727	RASGRP4	EF-hand domain containing			
5214	-55.24	cp	BRD-K93201660	ML-7	Myosin light chain kinase inhibitor		MYLK	Myosin light chain kinase inhibitor
5215	-55.26	cp	BRD-A46393198	tetramisole	Immunostimulant			Immunostimulant
5216	-55.27	cp	BRD-K54411430	robustic-acid	cAMP inhibitor			cAMP inhibitor
5217	-55.28	kd	CGS001-5063	PAK3	PAKA subfamily			
5218	-55.29	cp	BRD-A55416093	colforsin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator, Adenylate cyclase stimulant
5219	-55.38	kd	CGS001-11188	NISCH	-			
5220	-55.44	cp	BRD-K95899059	LY-344864	Serotonin receptor agonist		HTR1F, HTR1A, HTR1B, HTR1D, HTR1E, HTR2A, HTR2B, HTR2C, HTR7	Serotonin receptor agonist
5221	-55.65	kd	CGS001-84539	MCHR2	GPCR / Class A : MCH receptors			
5222	-55.66	kd	CGS001-2261	FGFR3	Type V RTKs: FGF (fibroblast growth factor) receptor family			
5223	-55.74	kd	CGS001-23528	ZNF281	Zinc fingers, C2H2-type			
5224	-55.78	kd	CGS001-4713	NDUFB7	Mitochondrial respiratory chain complex / Complex I			
5225	-55.84	oe	ccsbBroad304_00207	CALM2	EF-hand domain containing			
5226	-55.92	kd	CGS001-3958	LGALS3	Endogenous ligands			
5227	-55.97	oe	ccsbBroad304_04802	COX6B2	Mitochondrial respiratory chain complex / Complex IV			
5228	-56.02	oe	ccsbBroad304_01259	PPP1CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5229	-56.02	kd	CGS001-339403	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
5230	-56.06	cp	BRD-A54490543	pirlindole	Monoamine oxidase inhibitor		MAOA, SLC6A2, SLC6A4	Monoamine oxidase inhibitor
5231	-56.31	kd	CGS001-9870	KIAA0317	-			
5232	-56.37	oe	ccsbBroad304_05420	EIF4E3	Translation Initiation Factor 4E			
5233	-56.38	oe	ccsbBroad304_01148	PCBD1	-			
5234	-56.43	oe	ccsbBroad304_01732	UBA52	L ribosomal proteins			
5235	-56.46	cp	BRD-K62289640	lylamine	Cannabinoid receptor agonist		CNR1	Cannabinoid receptor agonist
5236	-56.48	kd	CGS001-7528	YY1	INO80 complex subunits			
5237	-56.53	oe	ccsbBroad304_02869	ASF1A	-			
5238	-56.56	cp	BRD-K49328571	dasatinib	BCR-ABL kinase inhibitor		ABL1, FYN, LCK, SRC, KIT, YES1, BCR, EPHA2, LYN, PDGFRB, ABL2, BTK, DDR1, DDR2, PDGFRA, STAT5B	BCR-ABL kinase inhibitor, Ephrin inhibitor, KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor, Tyrosine kinase inhibitor
5239	-56.57	kd	CGS001-6723	SRM	-			
5240	-56.57	kd	CGS001-9604	RNF14	RING-type (C3HC4) zinc fingers			
5241	-56.58	oe	ccsbBroad304_02163	MED7	-			
5242	-56.6	oe	ccsbBroad304_02131	ATP6V1F	ATPases / V-type			
5243	-56.7	kd	CGS001-3029	HAGH	-			
5244	-56.73	oe	ccsbBroad304_05471	ABCB5	ATP binding cassette transporters / subfamily B			
5245	-56.74	oe	ccsbBroad304_01406	RNASE4	Ribonucleases, RNase A			
5246	-56.74	oe	ccsbBroad304_06159	CTTN	-			
5247	-56.81	oe	ccsbBroad304_05749	A2M	-			
5248	-56.81	kd	CGS001-5563	PRKAA2	AMPK subfamily			
5249	-56.9	oe	ccsbBroad304_03314	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
5250	-56.94	oe	ccsbBroad304_08681	ADCK3	ABC1-B subfamily			
5251	-57.02	kd	CGS001-162239	ZFP1	Zinc fingers, C2H2-type			
5252	-57.03	cp	BRD-A26032986	zaldaride	Calmodulin antagonist		CALM1	Calmodulin antagonist
5253	-57.03	kd	CGS001-156	ADRBK1	BARK/GRK2 subfamily			
5254	-57.04	cp	BRD-U44618005	WH-4023	SRC inhibitor		ABL1, LCK, SRC	SRC inhibitor
5255	-57.04	cp	BRD-K77677632	SB-200646	Serotonin receptor antagonist		HTR2B, HTR2C	Serotonin receptor antagonist
5256	-57.13	cp	BRD-K66792149	quinoclamine	Algicide			Algicide
5257	-57.13	kd	CGS001-1512	CTSH	Cathepsins			
5258	-57.29	kd	CGS001-4122	MAN2A2	-			
5259	-57.32	kd	CGS001-2241	FER	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5260	-57.34	cp	BRD-K87932577	CDK1-5-inhibitor	CDK inhibitor		CDK1, CDK5, GSK3B	CDK inhibitor, Glycogen synthase kinase inhibitor
5261	-57.49	cc		NFKB Activation GOF	-			
5262	-57.5	oe	ccsbBroad304_09195	MCM8	-			
5263	-57.51	kd	CGS001-339327	ZNF546	Zinc fingers, C2H2-type			
5264	-57.53	kd	CGS001-11136	SLC7A9	SLC7 family			
5265	-57.58	oe	ccsbBroad304_01654	TCTA	-			
5266	-57.58	cp	BRD-K67261995	adipiodone	Contrast agent		ALB	Contrast agent
5267	-57.61	cp	BRD-K52080565	rilmenidine	Imidazoline receptor agonist		NISCH	Imidazoline receptor agonist
5268	-57.63	oe	ccsbBroad304_00379	CSNK1E	Casein kinase 1 (CK1) family			
5269	-57.66	kd	CGS001-23043	TNIK	MSN subfamily			
5270	-57.66	kd	CGS001-94234	FOXQ1	Forkhead boxes			
5271	-57.76	cp	BRD-K18059238	gamma-linolenic-acid	Cyclooxygenase inhibitor		TBXAS1	Cyclooxygenase inhibitor, Prostanoid receptor agonist
5272	-57.8	kd	CGS001-60468	BACH2	BTB/POZ domain containing			
5273	-57.82	cc		DNA Replication LOF	-			
5274	-57.85	cp	BRD-K32292990	CGP-53353	EGFR inhibitor		EGFR, PRKCB	EGFR inhibitor, PKC inhibitor
5275	-57.87	oe	ccsbBroad304_00360	CREB1	basic leucine zipper proteins			
5276	-57.92	cc		Potassium channel activator	-			
5277	-57.99	kd	CGS001-593	BCKDHA	-			
5278	-58.03	kd	CGS001-5894	RAF1	RAF family			
5279	-58.03	kd	CGS001-8543	LMO4	-			
5280	-58.07	cp	BRD-K98548675	parthenolide	NFkB pathway inhibitor		ADIPOR2, IKBKB, RELA	NFkB pathway inhibitor, Adiponectin receptor agonist
5281	-58.09	cp	BRD-A61392169	eliprodil	Glutamate receptor antagonist		GRIN1, GRIN2B	Glutamate receptor antagonist
5282	-58.1	cp	BRD-K33882852	ZK-93423	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	Benzodiazepine receptor agonist
5283	-58.12	kd	CGS001-2324	FLT4	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
5284	-58.15	cp	BRD-A15131297	benazepril	ACE inhibitor		ACE	ACE inhibitor
5285	-58.17	cp	BRD-K53979406	ALX-5407	Glycine transporter inhibitor		SLC6A9	Glycine transporter inhibitor
5286	-58.18	kd	CGS001-57819	LSM2	-			
5287	-58.18	kd	CGS001-4254	KITLG	-			
5288	-58.24	kd	CGS001-2023	ENO1	-			
5289	-58.28	kd	CGS001-10318	TNIP1	-			
5290	-58.3	oe	ccsbBroad304_03842	ZNF317	Zinc fingers, C2H2-type			
5291	-58.32	oe	ccsbBroad304_02345	TXNDC9	-			
5292	-58.33	kd	CGS001-64400	AKTIP	Ubiquitin-conjugating enzymes E2			
5293	-58.35	cp	BRD-K80725821	RS-16566	Serotonin receptor antagonist			Serotonin receptor antagonist
5294	-58.38	kd	CGS001-10906	TRAFD1	-			
5295	-58.41	cp	BRD-K26160755	RS-45041-190	Imidazoline receptor agonist			Imidazoline receptor agonist
5296	-58.44	cp	BRD-K47679368	bromfenac	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5297	-58.5	oe	ccsbBroad304_02889	WWTR1	Hippo Signaling			
5298	-58.52	cp	BRD-K08556791	ethoprop	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5299	-58.54	oe	ccsbBroad304_02766	GPR161	GPCR / Class A : Orphans			
5300	-58.58	oe	ccsbBroad304_07766	RASSF1	-			
5301	-58.61	kd	CGS001-2627	GATA6	GATA zinc finger domain containing			
5302	-58.64	oe	ccsbBroad304_02632	PTP4A3	Protein tyrosine phosphatases			
5303	-58.67	oe	ccsbBroad304_06095	DFFB	-			
5304	-58.68	cp	BRD-K06750613	GSK-1059615	PI3K inhibitor		PIK3CA, PIK3CG	PI3K inhibitor
5305	-58.72	kd	CGS001-5437	POLR2H	RNA polymerase subunits			
5306	-58.83	cc		HDAC inhibitor	-			
5307	-58.89	cp	BRD-K83063356	RS-102895	CCR antagonist		CCR2	CCR antagonist
5308	-58.93	kd	CGS001-2782	GNB1	WD repeat domain containing			
5309	-58.96	cp	BRD-A08709697	heliotrine	Pyrrolizidine alkaloid			Pyrrolizidine alkaloid
5310	-58.96	kd	CGS001-4292	MLH1	-			
5311	-58.99	oe	ccsbBroad304_00446	DKC1	-			
5312	-59.14	cp	BRD-K05528470	L-745870	Dopamine receptor antagonist		DRD4, DRD1, DRD2, DRD3, HTR1A, HTR2A, HTR6, HTR7	Dopamine receptor antagonist
5313	-59.19	oe	ccsbBroad304_13911	NDUFA9	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5314	-59.28	cp	BRD-K70241288	L-692585	Growth hormone releasing peptide ligand agonist		GH1, GHSR	Growth hormone releasing peptide ligand agonist
5315	-59.3	cc		HMGCR inhibitor	-			
5316	-59.36	oe	ccsbBroad304_01070	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
5317	-59.38	kd	CGS001-4751	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
5318	-59.4	cp	BRD-K69690935	curcumin	Cyclooxygenase inhibitor		PTGS1, PTGS2, APP, CA1, CA12, CA14, CA2, CA4, CA6, CA9, CCND1, CYP3A4, DNMT1, DNMT3B, EP300, G6PC, MAPT, MMP13, MMP9, NOS2, XDH	Cyclooxygenase inhibitor, Histone acetyltransferase inhibitor, Lipoxygenase inhibitor, NFkB pathway inhibitor
5319	-59.42	cp	BRD-K76274772	MAPP-D-erythro	Ceramidase inhibitor			Ceramidase inhibitor
5320	-59.45	kd	CGS001-5045	FURIN	Subtilisin			
5321	-59.49	cp	BRD-A91555231	norepinephrine	Adrenergic receptor agonist		ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB3, ADRB2, DRD1, DRD5, PAH, SLC18A1, SLC18A2	Adrenergic receptor agonist
5322	-59.52	oe	ccsbBroad304_00617	GBA	-			
5323	-59.52	kd	CGS001-4773	NFATC2	Nuclear factor of activated T-cells			
5324	-59.62	oe	ccsbBroad304_06831	RAC1	Endogenous ligands			
5325	-59.62	cp	BRD-K61829047	7b-cis	Exportin antagonist		XPO1	Exportin antagonist
5326	-59.62	cp	BRD-A65076780	dihydroergocristine	Adrenergic receptor antagonist		HTR2A, ADRA1A, ADRB1, DRD1, DRD2, DRD3, DRD4, DRD5, HTR1A, HTR3A, HTR4, HTR5A, HTR6, HTR7	Adrenergic receptor antagonist, Prolactin inhibitor
5327	-59.63	kd	CGS001-55612	FERMT1	Fermitins			
5328	-59.74	kd	CGS001-4047	LSS	Lanosterol biosynthesis pathway			
5329	-59.75	kd	CGS001-26994	RNF11	RING-type (C3HC4) zinc fingers			
5330	-59.77	cp	BRD-K10467831	tibolone	Androgen receptor agonist		AR, ESR1, PGR, STS	Androgen receptor agonist, Estrogen receptor agonist, Progesterone receptor agonist
5331	-59.8	cp	BRD-K82823076	RO-15-4513	GABA benzodiazepine site receptor inverse agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRA4, GABRA6, GABRB2, GABRG2	GABA benzodiazepine site receptor inverse agonist
5332	-59.81	kd	CGS001-84435	GPR123	Adhesion Class GPCRs			
5333	-59.84	kd	CGS001-10105	PPIF	-			
5334	-59.92	oe	ccsbBroad304_01168	PDPK1	PDK1 family			
5335	-59.94	oe	ccsbBroad304_00454	DNMT3A	Methyltransferases			
5336	-59.95	cp	BRD-K29653726	topiramate	Carbonic anhydrase inhibitor		CA2, CA4, GRIK1, CA1, CA12, CA7, CYP2C19, CYP3A4, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA1, SCN1A, SCN5A	Carbonic anhydrase inhibitor, Glutamate receptor antagonist, Kainate receptor antagonist
5337	-59.96	cp	BRD-A49765801	fludroxycortide	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
5338	-59.96	cp	BRD-K50660797	epicatechin	Bacterial DNA gyrase inhibitor		FASN, APP, BACE1, SLC5A1	Bacterial DNA gyrase inhibitor, Cyclooxygenase inhibitor, DNA polymerase inhibitor
5339	-59.99	kd	CGS001-80135	RPF1	-			
5340	-60	cp	BRD-K59753853	MDL-29951	Glutamate receptor antagonist		FBP1, GPR17	Glutamate receptor antagonist
5341	-60.02	oe	ccsbBroad304_07124	UROD	-			
5342	-60.03	kd	CGS001-7079	TIMP4	-			
5343	-60.11	oe	ccsbBroad304_06094	DFFA	-			
5344	-60.19	kd	CGS001-5525	PPP2R5A	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
5345	-60.29	cc		C2 domain containing protein kinases LOF	-			
5346	-60.31	cp	BRD-K39987650	bisacodyl	Laxative			Laxative
5347	-60.34	cp	BRD-K07691486	roscovitine	CDK inhibitor		CDK2, CDK9, CDK7, CDK1, CDK5	CDK inhibitor
5348	-60.41	kd	CGS001-6303	SAT1	-			
5349	-60.43	cp	BRD-K04466929	Merck60	HDAC inhibitor		HDAC1, HDAC2	HDAC inhibitor
5350	-60.43	cp	BRD-K15935639	z-leu3-VS	Proteasome inhibitor			Proteasome inhibitor
5351	-60.5	kd	CGS001-51588	PIAS4	Zinc fingers, MIZ-type			
5352	-60.52	oe	ccsbBroad304_08993	DHDDS	-			
5353	-60.57	oe	ccsbBroad304_01640	TAF12	-			
5354	-60.57	cp	BRD-K37312348	kenpaullone	CDK inhibitor		GSK3B, CDK1, CDK5, CCNB1, CDK2, LCK	CDK inhibitor, Glycogen synthase kinase inhibitor
5355	-60.59	cp	BRD-K56301217	ABT-737	BCL inhibitor		BCL2, BCL2L1, BCL2L2	BCL inhibitor
5356	-60.6	oe	ccsbBroad304_07147	ZNF8	Zinc fingers, C2H2-type			
5357	-60.75	cp	BRD-A42553870	L-152804	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
5358	-60.75	cp	BRD-K52397688	amperozide	Dopamine receptor antagonist		HTR2A, DRD2, FAAH	Dopamine receptor antagonist
5359	-60.76	oe	ccsbBroad304_03368	GPRC5B	GPCR / Class C : Orphans			
5360	-60.76	cp	BRD-K51671335	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
5361	-60.77	cp	BRD-K31843556	T-0070907	PPAR receptor antagonist		PPARG	PPAR receptor antagonist
5362	-60.84	kd	CGS001-1647	GADD45A	-			
5363	-60.86	kd	CGS001-7026	NR2F2	COUP-TF-like receptors			
5364	-60.87	cc		EIF Proteins LOF	-			
5365	-60.88	kd	CGS001-2222	FDFT1	Lanosterol biosynthesis pathway			
5366	-60.89	kd	CGS001-51586	MED15	-			
5367	-60.89	kd	CGS001-55033	FKBP14	EF-hand domain containing			
5368	-60.98	oe	ccsbBroad304_06004	CKB	-			
5369	-60.98	kd	CGS001-51131	PHF11	Zinc fingers, PHD-type			
5370	-61.02	oe	ccsbBroad304_00519	ETFB	-			
5371	-61.05	kd	CGS001-27333	GOLIM4	-			
5372	-61.06	oe	ccsbBroad304_02677	PDAP1	-			
5373	-61.08	cp	BRD-K62792802	LY-83583	Guanylyl cyclase inhibitor		GUCY1A2	Guanylyl cyclase inhibitor
5374	-61.12	kd	CGS001-2992	GYG1	Glycosyltransferase family 8 domain containing			
5375	-61.16	cp	BRD-K44442813	pidotimod	Interferon receptor agonist			Interferon receptor agonist, Interleukin receptor agonist
5376	-61.19	cp	BRD-K74501079	azithromycin	Bacterial 50S ribosomal subunit inhibitor		MLNR	Bacterial 50S ribosomal subunit inhibitor
5377	-61.2	kd	CGS001-3480	IGF1R	Type II RTKs: Insulin receptor family			
5378	-61.26	kd	CGS001-57222	ERGIC1	-			
5379	-61.29	kd	CGS001-8295	TRRAP	TRRAP subfamily			
5380	-61.33	kd	CGS001-866	SERPINA6	Serine (or cysteine) peptidase inhibitors			
5381	-61.36	cp	BRD-K90543092	levonorgestrel	Estrogen receptor agonist		PGR, AR, CYP2E1, ESR1, SRD5A1	Estrogen receptor agonist, Glucocorticoid receptor antagonist, Progesterone receptor agonist, Progesterone receptor antagonist
5382	-61.45	cp	BRD-K78084463	W-12	Calmodulin antagonist			Calmodulin antagonist
5383	-61.46	kd	CGS001-4129	MAOB	Catecholamine turnover			
5384	-61.53	cp	BRD-K99029477	prometon	Photosynthesis inhibitor			Photosynthesis inhibitor
5385	-61.56	kd	CGS001-5594	MAPK1	MAPK:ERK subfamily			
5386	-61.57	oe	ccsbBroad304_06952	SKP1	-			
5387	-61.57	cp	BRD-A97674275	ranolazine	Sodium channel blocker		SCN9A, SCN10A, SCN5A, SLC22A2	Sodium channel blocker
5388	-61.58	cp	BRD-K22503835	scriptaid	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5389	-61.59	kd	CGS001-165082	GPR113	Adhesion Class GPCRs			
5390	-61.6	kd	CGS001-1111	CHEK1	CHK1 subfamily			
5391	-61.63	cp	BRD-K19136521	indirubin	CDK inhibitor		CDK1, CDK5, CCNE1, CDK2, CDK4, CDK5R1, CDK9, GSK3A, GSK3B, LCK, LRRK1, LRRK2	CDK inhibitor
5392	-61.64	cp	BRD-K95885906	quercetagetin	PIM inhibitor		PIM1	PIM inhibitor
5393	-61.66	cp	BRD-K59753975	vindesine	Tubulin inhibitor		TUBB, TUBB1	Tubulin inhibitor
5394	-61.66	cp	BRD-K66412701	pazufloxacin	Topoisomerase inhibitor			Topoisomerase inhibitor
5395	-61.67	oe	ccsbBroad304_06862	RGS3	-			
5396	-61.75	oe	ccsbBroad304_02351	DHRS2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5397	-61.79	cp	BRD-K77641333	naphazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A	Adrenergic receptor agonist
5398	-61.8	kd	CGS001-8833	GMPS	-			
5399	-61.88	oe	ccsbBroad304_00391	CTH	Hydrogen sulphide synthesis			
5400	-61.92	oe	ccsbBroad304_01527	SGK1	SGK family			
5401	-61.92	oe	ccsbBroad304_03071	CHMP4A	Charged multivesicular body proteins			
5402	-61.92	kd	CGS001-6794	STK11	LKB subfamily			
5403	-61.95	cp	BRD-A06726973	dibutyrylcyclic-gmp	cGMP analog			cGMP analog
5404	-61.95	kd	CGS001-4728	NDUFS8	Mitochondrial respiratory chain complex / Complex I			
5405	-62.02	kd	CGS001-55631	LRRC40	-			
5406	-62.07	cp	BRD-K71003802	hippeastrine	Plant alkaloid			Plant alkaloid
5407	-62.11	kd	CGS001-9989	PPP4R1	Serine/threonine phosphatases / Protein phosphatase 4, regulatory subunits			
5408	-62.18	kd	CGS001-8091	HMGA2	High-mobility group / Canonical			
5409	-62.19	cp	BRD-A68589262	troxipide	Glucosamine synthetase stimulant			Glucosamine synthetase stimulant
5410	-62.32	cp	BRD-K00312224	PPT	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5411	-62.33	cp	BRD-K59650319	YM-298198	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5412	-62.37	cp	BRD-K96263742	GW-7647	PPAR receptor agonist		PPARA	PPAR receptor agonist
5413	-62.39	oe	ccsbBroad304_00542	FBP1	-			
5414	-62.43	cp	BRD-K63792901	arecaidine	Acetylcholine receptor agonist		CHRM1, CHRM2, CHRM3, CHRM4	Acetylcholine receptor agonist
5415	-62.46	cp	BRD-A36074203	remacemide	Glutamate receptor antagonist		GRIN1	Glutamate receptor antagonist
5416	-62.5	oe	ccsbBroad304_00602	SLC37A4	SLC37 family of phosphosugar/phosphate exchangers			
5417	-62.5	kd	CGS001-1052	CEBPD	basic leucine zipper proteins			
5418	-62.52	oe	ccsbBroad304_00678	GPR37	GPCR / Class A : Orphans			
5419	-62.53	kd	CGS001-116443	GRIN3A	Glutamate receptors			
5420	-62.57	oe	ccsbBroad304_01666	TGFBR1	Type I receptor serine/threonine kinases			
5421	-62.57	kd	CGS001-5571	PRKAG1	AMPK subfamily			
5422	-62.67	cp	BRD-K84175871	pseudoephedrine	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRB1, ADRB2, ATF1, ATF2, ATF3, ATF4, ATF5, ATF6, ATF7, CXCL8, FOS, HRH1, IL2, JDP2, JUN, NFATC1, SLC6A2, SLC6A3, SLC6A4, TNF	Adrenergic receptor agonist
5423	-62.71	kd	CGS001-10427	SEC24B	-			
5424	-62.78	cp	BRD-K70487031	flupentixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, CHRM1, DRD3, DRD5, HTR2A	Dopamine receptor antagonist
5425	-62.81	cp	BRD-K69650333	idarubicin	Topoisomerase inhibitor		TOP2A	Topoisomerase inhibitor
5426	-62.83	kd	CGS001-148327	CREB3L4	basic leucine zipper proteins			
5427	-62.89	oe	ccsbBroad304_02659	SLC6A14	Glycine transporter subfamily			
5428	-62.92	cp	BRD-K17743125	belinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5429	-62.98	oe	ccsbBroad304_00237	CCND3	-			
5430	-62.99	kd	CGS001-930	CD19	CD molecules			
5431	-63	cp	BRD-K93618743	ipriflavone	Bone resorption inhibitor			Bone resorption inhibitor
5432	-63.04	kd	CGS001-7103	TSPAN8	Tetraspanins			
5433	-63.06	cp	BRD-A65597028	RX-821002	Adrenergic receptor antagonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor antagonist
5434	-63.08	cp	BRD-K30563334	rifabutin	Protein synthesis inhibitor		CYP3A4, HSP90AA1, HSP90B1	Protein synthesis inhibitor
5435	-63.09	cp	BRD-K13646352	midostaurin	FLT3 inhibitor		FLT3, KIT, CCNB1, FLT1, KDR, PDGFRB, PRKCA, PRKCG, VEGFA	FLT3 inhibitor, KIT inhibitor, PKC inhibitor
5436	-63.1	cp	BRD-A79903587	tegafur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
5437	-63.1	cp	BRD-A23072235	pheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5438	-63.11	cp	BRD-K04923131	GSK-3-inhibitor-IX	Glycogen synthase kinase inhibitor		ALOX5, GSK3A, GSK3B	Glycogen synthase kinase inhibitor, Lipoxygenase inhibitor
5439	-63.15	oe	ccsbBroad304_06897	RPS6KB2	p70 subfamily			
5440	-63.2	kd	CGS001-5698	PSMB9	Proteasome (prosome, macropain) subunits			
5441	-63.2	kd	CGS001-136	ADORA2B	GPCR / Class A : Adenosine receptors			
5442	-63.27	kd	CGS001-4923	NTSR1	GPCR / Class A : Neurotensin receptors			
5443	-63.28	oe	ccsbBroad304_00046	AKT1	Akt (Protein kinase B)			
5444	-63.3	cp	BRD-A60294240	tribenoside	Anti-inflammatory			Anti-inflammatory, Capillary stabilizing agent
5445	-63.4	cp	BRD-K02123250	JNJ-38877605	Tyrosine kinase inhibitor		MET	Tyrosine kinase inhibitor
5446	-63.47	oe	ccsbBroad304_00283	CDKN2C	Ankyrin repeat domain containing			
5447	-63.52	oe	ccsbBroad304_04801	ZNF543	Zinc fingers, C2H2-type			
5448	-63.55	oe	ccsbBroad304_00990	DNAJB9	Heat shock proteins / DNAJ (HSP40)			
5449	-63.58	cp	BRD-K32536677	AGK-2	SIRT inhibitor		SIRT2	SIRT inhibitor
5450	-63.63	cp	BRD-A51382177	fosinopril	ACE inhibitor		ACE, ABCG2	ACE inhibitor
5451	-63.67	cp	BRD-K34014345	naproxol	Anti-inflammatory		PTGS1, PTGS2	Anti-inflammatory
5452	-63.7	cp	BRD-A00993607	alprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2, HTR1A	Adrenergic receptor antagonist
5453	-63.72	oe	ccsbBroad304_01174	PEX13	-			
5454	-63.77	oe	ccsbBroad304_00644	GCLC	-			
5455	-63.78	cp	BRD-K86434416	selegiline	Monoamine oxidase inhibitor		MAOB, MAOA, CYP2B6, CYP2C19	Monoamine oxidase inhibitor
5456	-63.81	kd	CGS001-283455	KSR2	RAF family			
5457	-63.88	cp	BRD-A36471396	biperiden	Acetylcholine receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA2	Acetylcholine receptor antagonist
5458	-63.91	cp	BRD-K51918615	iodophenpropit	Histamine receptor antagonist		HRH3, HRH4, GRIN2B	Histamine receptor antagonist
5459	-63.95	oe	ccsbBroad304_00038	AGL	-			
5460	-63.98	cp	BRD-K66896231	BRD-K66896231	Acetylcholinesterase inhibitor		ACHE	Acetylcholinesterase inhibitor
5461	-64.04	cp	BRD-K56403959	ZK-756326	CC chemokine receptor ligand		CCR8	CC chemokine receptor ligand
5462	-64.08	cp	BRD-K10016611	pyridine-2-aldoxime	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor
5463	-64.08	cp	BRD-K15592317	CP466722	ATM kinase inhibitor		ATM	ATM kinase inhibitor
5464	-64.09	cp	BRD-A43150328	penicillic-acid	other antibiotic			other antibiotic
5465	-64.09	kd	CGS001-7097	TLR2	Toll-like receptor family			
5466	-64.12	cp	BRD-A53131506	epitestosterone	Inactive testosterone analog		AKR1C1, AKR1C2, AR	Inactive testosterone analog
5467	-64.14	cp	BRD-K84955386	hyperoside	Glucosidase inhibitor		ACE, AKR1B1, GAA	Glucosidase inhibitor
5468	-64.16	oe	ccsbBroad304_01532	SIAH1	-			
5469	-64.16	cp	BRD-K49668410	clarithromycin	Bacterial 50S ribosomal subunit inhibitor		CYP2C19, CYP3A4, CYP3A5, CYP3A7	Bacterial 50S ribosomal subunit inhibitor
5470	-64.2	kd	CGS001-3280	HES1	Basic helix-loop-helix proteins			
5471	-64.25	cp	BRD-K11433652	aspirin	Cyclooxygenase inhibitor		PTGS1, PTGS2, TP53, AKR1C1, ASIC3, EDNRA, HSPA5, IKBKB, NFKB1, NFKB2, NFKBIA, PRKAA1, PRKAA2, PRKAB1, PRKAB2, PRKAG1, PRKAG2, PRKAG3, RPS6KA3	Cyclooxygenase inhibitor
5472	-64.27	kd	CGS001-390980	ZNF805	Zinc fingers, C2H2-type			
5473	-64.4	cp	BRD-K96799727	pifithrin-mu	HSP inhibitor		HSPA1A, TP53	HSP inhibitor
5474	-64.43	kd	CGS001-9140	ATG12	-			
5475	-64.48	kd	CGS001-7054	TH	Amino acid hydroxylases			
5476	-64.51	kd	CGS001-8022	LHX3	Homeoboxes / LIM class			
5477	-64.57	kd	CGS001-2769	GNA15	-			
5478	-64.58	cp	BRD-K20920669	cromoglicic-acid	Immunosuppressant		KCNMA1, S100P	Immunosuppressant
5479	-64.62	kd	CGS001-162979	ZNF296	Zinc fingers, C2H2-type			
5480	-64.67	oe	ccsbBroad304_02219	MORF4L2	-			
5481	-64.68	oe	ccsbBroad304_01376	RARB	Retinoic acid receptors			
5482	-64.7	oe	ccsbBroad304_01247	POU2AF1	-			
5483	-64.7	kd	CGS001-3783	KCNN4	Calcium-activated potassium channels			
5484	-64.73	kd	CGS001-84433	CARD11	-			
5485	-64.76	cp	BRD-K24201553	SB-269970	Serotonin receptor antagonist		HTR7	Serotonin receptor antagonist
5486	-64.77	cp	BRD-K97752965	nicorandil	Nitric oxide donor		ABCC9, KCNJ11, KCNJ8	Nitric oxide donor, Potassium channel activator
5487	-64.79	kd	CGS001-148103	ZNF599	Zinc fingers, C2H2-type			
5488	-64.83	oe	ccsbBroad304_03439	GNB1L	WD repeat domain containing			
5489	-64.88	kd	CGS001-5606	MAP2K3	MAPKK:STE7 family			
5490	-64.95	kd	CGS001-58190	CTDSP1	Serine/threonine phosphatases / CTD aspartate-based phosphatases			
5491	-64.96	oe	ccsbBroad304_06138	EDNRB	Endothelin receptors			
5492	-64.98	cc		SRC inhibitor	-			
5493	-64.99	oe	ccsbBroad304_10437	STMN1	-			
5494	-65.1	oe	ccsbBroad304_00648	GLRX	-			
5495	-65.11	oe	ccsbBroad304_03683	APOM	Apolipoproteins			
5496	-65.13	oe	ccsbBroad304_01423	RPL19	L ribosomal proteins			
5497	-65.14	cp	BRD-K96271548	coumaric-acid	Antioxidant			Antioxidant
5498	-65.15	kd	CGS001-284119	PTRF	-			
5499	-65.18	cp	BRD-K42098891	protriptyline	Tricyclic antidepressant		SLC6A2, SLC6A4	Tricyclic antidepressant
5500	-65.24	kd	CGS001-581	BAX	-			
5501	-65.4	kd	CGS001-205564	SENP5	-			
5502	-65.43	kd	CGS001-126823	KLHDC9	-			
5503	-65.43	kd	CGS001-1675	CFD	Complement system			
5504	-65.52	cp	BRD-A58048407	nimodipine	Calcium channel blocker		CACNA1C, NR3C2, AHR, CACNA1D, CACNA1F, CACNA1S, CACNB1, CACNB2, CACNB3, CACNB4, CFTR	Calcium channel blocker
5505	-65.57	oe	ccsbBroad304_01981	DYNLL1	Cytoplasmic dyneins			
5506	-65.64	cc		DNA synthesis inhibitor	-			
5507	-65.68	kd	CGS001-1803	DPP4	Prolyl oligopeptidase			
5508	-65.69	oe	ccsbBroad304_00099	ARG2	Arginase			
5509	-65.7	oe	ccsbBroad304_08217	SCCPDH	-			
5510	-65.73	kd	CGS001-10559	SLC35A1	SLC35 family of nucleotide sugar transporters			
5511	-65.8	cp	BRD-K21672174	RO-28-1675	Glucokinase activator		GCK	Glucokinase activator
5512	-65.84	oe	ccsbBroad304_00554	FGB	Endogenous ligands			
5513	-65.86	cc		MTOR inhibitor	-			
5514	-65.88	kd	CGS001-23523	CABIN1	-			
5515	-65.89	cc		Proteasome inhibitor	-			
5516	-65.89	cp	BRD-A93659613	GR-89696	Opioid receptor agonist		OPRK1	Opioid receptor agonist
5517	-65.94	kd	CGS001-1736	DKC1	-			
5518	-65.96	oe	ccsbBroad304_00521	ETV5	ETS Transcription Factors			
5519	-66	cp	BRD-K32645441	dipropyl-5ct	Serotonin receptor agonist		HTR1B, HTR1D, HTR1F, HTR7	Serotonin receptor agonist
5520	-66.03	cp	BRD-K15616905	CCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
5521	-66.04	kd	CGS001-699	BUB1	Bub family			
5522	-66.05	cc		Bromodomain Inhibitor	-			
5523	-66.12	oe	ccsbBroad304_06134	ECH1	-			
5524	-66.16	oe	ccsbBroad304_01579	SOX2	SRY (sex determining region Y)-boxes			
5525	-66.16	cp	BRD-K07237224	moclobemide	Monoamine oxidase inhibitor		MAOA, CYP2C19, MAOB	Monoamine oxidase inhibitor
5526	-66.16	kd	CGS001-60493	FASTKD5	-			
5527	-66.21	cp	BRD-K30097969	pitavastatin	HMGCR inhibitor		HMGCR, APOA1, CYP2C8	HMGCR inhibitor
5528	-66.25	cp	BRD-K78637815	LY-320135	Cannabinoid receptor antagonist		CNR1	Cannabinoid receptor antagonist
5529	-66.25	kd	CGS001-11143	KAT7	Histone acetyltransferases (HATs)			
5530	-66.29	oe	ccsbBroad304_06260	GATA3	GATA zinc finger domain containing			
5531	-66.43	kd	CGS001-22930	RAB3GAP1	-			
5532	-66.55	cp	BRD-K79602928	metformin	Insulin sensitizer		ACACB, INS, PRKAB1	Insulin sensitizer
5533	-66.57	cp	BRD-K67783091	haloperidol	Dopamine receptor antagonist		DRD2, DRD1, DRD3, HTR2A, CYP3A7, DRD4, DRD5, GRIN2B, HRH1, HTR1A, HTR1D, HTR2B, HTR7, KCNH1	Dopamine receptor antagonist, Psychoactive drug
5534	-66.61	oe	ccsbBroad304_10014	RXFP4	GPCR / Class A : Relaxin family peptide receptors			
5535	-66.65	cp	BRD-K11158509	tyrphostin-B44	EGFR inhibitor			EGFR inhibitor
5536	-66.79	oe	ccsbBroad304_01216	PLD1	Phosphatidylcholine-specific phospholipase D			
5537	-66.79	cp	BRD-K06753942	nobiletin	MEK inhibitor		ABCB1, MAP2K1, TYR	MEK inhibitor
5538	-66.8	cp	BRD-A43082555	loxoprofen	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor, Prostanoid receptor antagonist
5539	-66.89	cp	BRD-A67605442	tetrahydrobiopterin	Nitric oxide stimulant		PAH, TH, DBH, NOS3, TPH1	Nitric oxide stimulant, Nitric oxide synthase stimulant, Phenylalanine 4-hydroxylase stimulant
5540	-66.94	cp	BRD-A31195449	TCB2	Serotonin receptor agonist		HTR2A	Serotonin receptor agonist
5541	-66.94	kd	CGS001-3155	HMGCL	-			
5542	-66.95	kd	CGS001-9787	DLGAP5	-			
5543	-66.97	oe	ccsbBroad304_06496	KNG1	Endogenous ligands			
5544	-67.04	kd	CGS001-2242	FES	Fer family			
5545	-67.06	cp	BRD-K77998258	ganglioside	SRC activator			SRC activator
5546	-67.19	oe	ccsbBroad304_06041	CRYAA	Heat shock proteins / HSPB			
5547	-67.25	cp	BRD-K14821540	FCCP	Mitochondrial oxidative phosphorylation uncoupler			Mitochondrial oxidative phosphorylation uncoupler
5548	-67.31	cp	BRD-K08502430	angiogenesis-inhibitor	Angiogenesis inhibitor		EGFR	Angiogenesis inhibitor
5549	-67.34	cp	BRD-K93480852	KN-93	Calcium-calmodulin dependent protein kinase inhibitor		CAMK2A	Calcium-calmodulin dependent protein kinase inhibitor
5550	-67.34	kd	CGS001-2321	FLT1	Type IV RTKs: VEGF (vascular endothelial growth factor) receptor family			
5551	-67.36	kd	CGS001-57822	GRHL3	-			
5552	-67.41	kd	CGS001-9710	KIAA0355	-			
5553	-67.42	cp	BRD-K72703948	ZM-447439	Aurora kinase inhibitor		AURKA, AURKB	Aurora kinase inhibitor
5554	-67.42	cp	BRD-K96402602	farnesylthiotriazole	PPMTase inhibitor			PPMTase inhibitor
5555	-67.47	kd	CGS001-84636	GPR174	GPCR / Class A : Orphans			
5556	-67.51	cp	BRD-K69837166	trap-101	Nociceptin/orphanin FQ (NOP) receptor antagonist		OPRL1	Nociceptin/orphanin FQ (NOP) receptor antagonist, Opioid receptor antagonist
5557	-67.54	cp	BRD-K51018020	VAMA-37	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor
5558	-67.54	kd	CGS001-369	ARAF	RAF family			
5559	-67.66	kd	CGS001-5144	PDE4D	Phosphodiesterases			
5560	-67.69	kd	CGS001-6924	TCEB3	-			
5561	-67.7	cp	BRD-K33106058	cytarabine	Ribonucleotide reductase inhibitor		POLB, POLA1	Ribonucleotide reductase inhibitor
5562	-67.75	oe	ccsbBroad304_06317	GPR26	GPCR / Class A : Orphans			
5563	-67.77	kd	CGS001-146434	ZNF597	Zinc fingers, C2H2-type			
5564	-67.81	oe	ccsbBroad304_00322	CLCN5	Ion channels / Chloride channels : Voltage-sensitive			
5565	-67.82	cp	BRD-K72783841	tyrphostin-AG-555	EGFR inhibitor		CDK2, EGFR	EGFR inhibitor
5566	-67.83	cp	BRD-K83972459	JWE-035	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor
5567	-67.87	cp	BRD-A16934955	nalbuphine	Opioid receptor agonist		OPRD1, OPRK1, OPRM1	Opioid receptor agonist, Opioid receptor antagonist
5568	-68.03	cp	BRD-K15600710	obatoclax	BCL inhibitor		BCL2, BCL2L1, MCL1	BCL inhibitor
5569	-68.07	kd	CGS001-7175	TPR	-			
5570	-68.08	kd	CGS001-5499	PPP1CA	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5571	-68.12	oe	ccsbBroad304_00078	BIRC2	Inhibitors of apoptosis (IAP) protein family			
5572	-68.15	kd	CGS001-10681	GNB5	WD repeat domain containing			
5573	-68.19	cc		Tricyclic antidepressant	-			
5574	-68.19	kd	CGS001-7316	UBC	-			
5575	-68.22	cp	BRD-K46556543	canrenoic-acid	Mineralocorticoid receptor antagonist			Mineralocorticoid receptor antagonist
5576	-68.23	kd	CGS001-47	ACLY	-			
5577	-68.29	cp	BRD-K34437622	BRD-K34437622	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
5578	-68.3	oe	ccsbBroad304_06542	LTBR	Tumor necrosis factor receptor superfamily			
5579	-68.3	oe	ccsbBroad304_00161	BID	Endogenous ligands			
5580	-68.31	cp	BRD-A17655518	ibuprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, ASIC1, BCL2, CFTR, CYP2C8, FABP2, PLAT, PPARG, SLC5A8, THBD	Cyclooxygenase inhibitor, NFkB pathway inhibitor
5581	-68.39	oe	ccsbBroad304_06453	ING2	Zinc fingers, PHD-type			
5582	-68.54	cp	BRD-K22828899	TUL-XXI039	Serine/threonine kinase inhibitor			Serine/threonine kinase inhibitor
5583	-68.57	kd	CGS001-8613	PPAP2B	Lipid phosphate phosphatases			
5584	-68.59	cp	BRD-A07824748	flavanone	11-beta-HSD1 inhibitor		ADORA3, HSD11B1	11-beta-HSD1 inhibitor
5585	-68.59	kd	CGS001-4351	MPI	-			
5586	-68.63	cp	BRD-K59331372	SB-366791	TRPV antagonist		TRPV1	TRPV antagonist
5587	-68.65	oe	ccsbBroad304_01962	STK16	NAK family			
5588	-68.65	kd	CGS001-2896	GRN	-			
5589	-68.68	kd	CGS001-90589	ZNF625	Zinc fingers, C2H2-type			
5590	-68.71	cp	BRD-K20655524	mefexamide	Psychoactive drug			Psychoactive drug
5591	-68.73	cc		Aromatase inhibitor	-			
5592	-68.78	oe	ccsbBroad304_11668	TBC1D9B	EF-hand domain containing			
5593	-68.78	kd	CGS001-1062	CENPE	Kinesins			
5594	-68.83	oe	ccsbBroad304_08645	BCCIP	-			
5595	-68.9	kd	CGS001-1431	CS	-			
5596	-68.93	cp	BRD-U97083655	teicoplanin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
5597	-68.93	cp	BRD-A10715913	sulpiride	Dopamine receptor antagonist		DRD2, CA7, DRD3, CA1, CA12	Dopamine receptor antagonist
5598	-68.94	cp	BRD-A64092382	mexiletine	Sodium channel blocker		SCN5A, AHR, CYP2B6, CYP2E1, KCNK2, KCNK3, SCN4A	Sodium channel blocker
5599	-68.95	kd	CGS001-4638	MYLK	Myosin Light Chain Kinase (MLCK) family			
5600	-68.99	kd	CGS001-2015	EMR1	Adhesion Class GPCRs			
5601	-69.02	oe	ccsbBroad304_02398	LANCL1	-			
5602	-69.02	oe	ccsbBroad304_00389	CTBP1	-			
5603	-69.03	cp	BRD-A13807286	HA-14-1	BCL inhibitor		BCL2	BCL inhibitor
5604	-69.04	oe	ccsbBroad304_07079	TSPAN4	Tetraspanins			
5605	-69.04	cp	BRD-K98493452	honokiol	AKT inhibitor		ALOX5, PTGS1, PTGS2	AKT inhibitor
5606	-69.06	oe	ccsbBroad304_06774	PRKCQ	Delta subfamily			
5607	-69.07	cp	BRD-K66353228	zoxazolamine	Myorelaxant			Myorelaxant
5608	-69.08	kd	CGS001-2188	FANCF	Fanconi anemia, complementation groups			
5609	-69.09	oe	ccsbBroad304_00478	S1PR3	GPCR / Class A : Lysophospholipid receptors : Sphingosine 1-phosphate			
5610	-69.1	kd	CGS001-6818	SULT1A3	Sulfotransferases, cytosolic			
5611	-69.13	oe	ccsbBroad304_02421	WFDC2	WAP four-disulfide core domain containing			
5612	-69.2	oe	ccsbBroad304_01379	RBBP6	-			
5613	-69.22	oe	ccsbBroad304_02691	PUF60	RNA binding motif (RRM) containing			
5614	-69.23	cp	BRD-A68929948	DAPT-GSI-IX	Gamma secretase inhibitor			Gamma secretase inhibitor
5615	-69.3	kd	CGS001-29078	NDUFAF4	Mitochondrial respiratory chain complex assembly factors			
5616	-69.37	cp	BRD-A88254928	salbutamol	Adrenergic receptor agonist		ADRB2, ADRB1	Adrenergic receptor agonist
5617	-69.38	cp	BRD-K86887724	dofetilide	Potassium channel blocker		KCNH2, KCNH1, KCNJ12, KCNK2	Potassium channel blocker
5618	-69.49	cp	BRD-A01346607	flumetasone	Glucocorticoid receptor agonist		NR3C1, PLA2G1B	Glucocorticoid receptor agonist
5619	-69.54	cp	BRD-K42452249	EO-1428	p38 MAPK inhibitor		MAPK11, MAPK14	p38 MAPK inhibitor
5620	-69.61	oe	ccsbBroad304_01165	PDK1	-			
5621	-69.65	oe	ccsbBroad304_03658	DCP1A	-			
5622	-69.69	kd	CGS001-11004	KIF2C	Kinesins			
5623	-69.74	kd	CGS001-356	FASLG	Tumour necrosis factor (TNF) receptor family			
5624	-69.76	cp	BRD-K87696786	LY-456236	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5625	-69.86	kd	CGS001-835	CASP2	Caspases			
5626	-69.87	kd	CGS001-9805	SCRN1	-			
5627	-69.87	kd	CGS001-79722	ANKRD55	Ankyrin repeat domain containing			
5628	-69.93	cp	BRD-K21283037	riluzole	Glutamate inhibitor		KCND3, KCNK10, KCNK2, KCNK4, KCNN4, SCN5A, SLC7A11	Glutamate inhibitor
5629	-69.99	oe	ccsbBroad304_03413	SLC38A2	System A-like transporters			
5630	-70.01	cp	BRD-A62809825	thapsigargin	ATPase inhibitor		ATP2A1	ATPase inhibitor
5631	-70.01	cp	BRD-K59637651	NSC-119889	Protein synthesis inhibitor			Protein synthesis inhibitor
5632	-70.03	kd	CGS001-335	APOA1	Apolipoproteins			
5633	-70.05	kd	CGS001-89882	TPD52L3	-			
5634	-70.07	oe	ccsbBroad304_03404	POLE3	DNA polymerases			
5635	-70.12	cp	BRD-A95696066	nisoxetine	Norepinephrine reuptake inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine reuptake inhibitor
5636	-70.18	kd	CGS001-7874	USP7	Ubiquitin-specific peptidases			
5637	-70.25	kd	CGS001-10606	PAICS	-			
5638	-70.33	cp	BRD-K53878242	MMPX	Phosphodiesterase inhibitor			Phosphodiesterase inhibitor
5639	-70.39	oe	ccsbBroad304_00381	CSNK2A1	Casein kinase 2 (CK2) family			
5640	-70.39	oe	ccsbBroad304_00817	IDH2	-			
5641	-70.39	kd	CGS001-29978	UBQLN2	Ubiquilin family			
5642	-70.42	kd	CGS001-11113	CIT	Other DMPK family kinases			
5643	-70.46	oe	ccsbBroad304_06382	HMGCL	-			
5644	-70.46	kd	CGS001-9258	MFHAS1	-			
5645	-70.53	oe	ccsbBroad304_00539	FANCG	Fanconi anemia, complementation groups			
5646	-70.56	oe	ccsbBroad304_00210	CALR	-			
5647	-70.66	oe	ccsbBroad304_01061	NAB2	-			
5648	-70.71	cp	BRD-K10136726	tosyllysyl-chloromethyl-ketone	Chymotrypsin inhibitor			Chymotrypsin inhibitor
5649	-70.75	kd	CGS001-51684	SUFU	-			
5650	-70.77	oe	ccsbBroad304_01470	RXRG	Retinoid X receptors			
5651	-70.78	kd	CGS001-8321	FZD1	GPCR / Class F : Frizzled receptors			
5652	-70.82	kd	CGS001-64241	ABCG8	ATP binding cassette transporters / subfamily G			
5653	-70.94	cp	BRD-K17415526	tyrphostin-AG-835	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
5654	-71.01	kd	CGS001-670	BPHL	-			
5655	-71.06	cp	BRD-K41868777	W-5	Calmodulin antagonist			Calmodulin antagonist
5656	-71.08	cc		Glycogen synthase kinase inhibitor	-			
5657	-71.1	oe	ccsbBroad304_05779	ADK	Adenosine turnover			
5658	-71.22	oe	ccsbBroad304_05939	CBLB	RING-type (C3HC4) zinc fingers			
5659	-71.22	kd	CGS001-5579	PRKCB	Alpha subfamily			
5660	-71.23	cp	BRD-K80396088	gliquidone	Sulfonylurea		ABCC8, KCNJ10, KCNJ11, KCNJ8	Sulfonylurea
5661	-71.26	kd	CGS001-9712	USP6NL	-			
5662	-71.28	oe	ccsbBroad304_05757	ACADS	-			
5663	-71.35	cp	BRD-K73319509	PF-04217903	c-Met inhibitor		MET	c-Met inhibitor
5664	-71.35	kd	CGS001-7702	ZNF143	Zinc fingers, C2H2-type			
5665	-71.36	cp	BRD-K41903098	diphenoxylate	Opioid receptor agonist		OPRM1, OPRD1	Opioid receptor agonist
5666	-71.36	kd	CGS001-26149	ZNF658	Zinc fingers, C2H2-type			
5667	-71.4	cp	BRD-A87848830	bimatoprost	Prostanoid receptor agonist		PTGFR, AKR1C3, PTGER1, PTGER3	Prostanoid receptor agonist
5668	-71.4	cp	BRD-K14441456	tyrphostin-AG-556	EGFR inhibitor		EGFR	EGFR inhibitor
5669	-71.4	kd	CGS001-7867	MAPKAPK3	MAPKAPK subfamily			
5670	-71.46	oe	ccsbBroad304_06679	OXTR	GPCR / Class A : Vasopressin and oxytocin receptors			
5671	-71.5	cc		MCM family LOF	-			
5672	-71.56	cp	BRD-K44432556	VU-0418946-1	HIF modulator		HIF1A	HIF modulator
5673	-71.62	kd	CGS001-3575	IL7R	IL-2 receptor family			
5674	-71.69	oe	ccsbBroad304_02806	OPN3	GPCR / Class A : Opsin receptors			
5675	-71.7	cp	BRD-K68336408	tyrphostin-AG-1478	EGFR inhibitor		EGFR, MAPK14	EGFR inhibitor
5676	-71.7	kd	CGS001-4313	MMP2	Matrix metallopeptidase			
5677	-71.74	cp	BRD-A31801025	formestane	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5678	-71.75	cp	BRD-K79090631	CGP-60474	CDK inhibitor		CDK1, CDK2	CDK inhibitor
5679	-71.75	cp	BRD-K12516989	zaprinast	Phosphodiesterase inhibitor		PDE5A, GPR35, PDE1A, PDE4D, PDE9A	Phosphodiesterase inhibitor
5680	-71.77	oe	ccsbBroad304_01673	TIMP3	-			
5681	-71.83	kd	CGS001-54438	GFOD1	-			
5682	-71.85	cp	BRD-A04706586	bucladesine	Adenosine receptor agonist		PRKACA	Adenosine receptor agonist, cAMP stimulant
5683	-71.91	cp	BRD-K72903603	zidovudine	Reverse transcriptase inhibitor		TERT	Reverse transcriptase inhibitor
5684	-72.01	oe	ccsbBroad304_06413	HSP90AA1	Heat shock proteins / HSPC			
5685	-72.05	cp	BRD-K48722258	dilazep	Adenosine reuptake inhibitor		SLC29A1, CACNA1C	Adenosine reuptake inhibitor
5686	-72.07	kd	CGS001-66008	TRAK2	-			
5687	-72.08	kd	CGS001-57154	SMURF1	-			
5688	-72.11	kd	CGS001-79727	LIN28A	Zinc fingers, CCHC domain containing			
5689	-72.22	kd	CGS001-11245	GPR176	GPCR / Class A : Orphans			
5690	-72.24	cp	BRD-K52394958	GR-159897	Tachykinin antagonist		TACR2, TAC1	Tachykinin antagonist
5691	-72.27	kd	CGS001-54556	ING3	Zinc fingers, PHD-type			
5692	-72.29	cp	BRD-K85266041	DNQX	Glutamate receptor antagonist		GRIA1, GRIA2, GRIK1, GRIN1, GRIN2A, GRIN2B	Glutamate receptor antagonist
5693	-72.39	oe	ccsbBroad304_02332	MBNL2	Zinc fingers, CCCH-type domain containing			
5694	-72.4	kd	CGS001-3821	KLRC1	CD molecules			
5695	-72.43	oe	ccsbBroad304_00146	BAD	-			
5696	-72.45	cp	BRD-K18895904	olanzapine	Dopamine receptor antagonist		DRD2, HTR2A, HTR2C, DRD1, DRD3, DRD4, HRH1, HTR1A, HTR1B, HTR1D, HTR1E, HTR6, HTR7, ADRA1A, ADRA1B, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C8, DRD5, GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, HRH2, HRH4, HTR1F, HTR2B, HTR3A, HTR5A	Dopamine receptor antagonist, Serotonin receptor antagonist
5697	-72.46	oe	ccsbBroad304_02619	PRSS23	Serine peptidases / Serine peptidases			
5698	-72.48	cp	BRD-K92991072	PAC-1	Caspase activator		CASP3	Caspase activator
5699	-72.53	oe	ccsbBroad304_02788	PRAME	-			
5700	-72.54	kd	CGS001-9031	BAZ1B	Zinc fingers, PHD-type			
5701	-72.55	kd	CGS001-25949	SYF2	-			
5702	-72.56	cp	BRD-A14208071	oxyphenonium	Cholinergic receptor antagonist		CHRM1	Cholinergic receptor antagonist
5703	-72.56	kd	CGS001-16	AARS	Aminoacyl tRNA synthetases / Class II			
5704	-72.59	kd	CGS001-5747	PTK2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5705	-72.6	oe	ccsbBroad304_10929	JAK2	Janus kinase (JakA) family			
5706	-72.68	cp	BRD-K82561139	ricinine	Casein kinase inhibitor			Casein kinase inhibitor
5707	-72.68	kd	CGS001-5332	PLCB4	Phosphoinositide-specific phospholipase C			
5708	-72.73	cp	BRD-K99498722	NPI-2358	Tubulin inhibitor			Tubulin inhibitor
5709	-72.74	kd	CGS001-2160	F11	Chymotrypsin			
5710	-72.77	kd	CGS001-35	ACADS	-			
5711	-72.79	cp	BRD-K45988865	tetramethylsilane	Internal standard for NMR spectroscopy			Internal standard for NMR spectroscopy
5712	-72.82	kd	CGS001-5110	PCMT1	-			
5713	-72.84	oe	ccsbBroad304_00490	EIF4EBP1	-			
5714	-72.86	cp	BRD-K00673382	famotidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
5715	-72.98	kd	CGS001-5708	PSMD2	Proteasome subunits			
5716	-73.02	oe	ccsbBroad304_08879	CASD1	-			
5717	-73.1	oe	ccsbBroad304_03191	NOSIP	-			
5718	-73.1	kd	CGS001-10745	PHTF1	-			
5719	-73.15	kd	CGS001-2078	ERG	ETS Transcription Factors			
5720	-73.16	cp	BRD-K39120595	bithionol	Autotaxin inhibitor		ESR1, ESR2, MCL1	Autotaxin inhibitor
5721	-73.18	kd	CGS001-5156	PDGFRA	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
5722	-73.2	kd	CGS001-9318	COPS2	-			
5723	-73.21	oe	ccsbBroad304_07450	RNF7	RING-type (C3HC4) zinc fingers			
5724	-73.22	oe	ccsbBroad304_08089	MAT2B	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5725	-73.23	cp	BRD-A82096673	KU-C103428N	CDC inhibitor		NFE2	CDC inhibitor, Rho associated kinase inhibitor
5726	-73.23	cp	BRD-K74133369	oligomycin-a	ATP synthase inhibitor		ATP5A1	ATP synthase inhibitor, ATPase inhibitor
5727	-73.25	kd	CGS001-27113	BBC3	-			
5728	-73.43	kd	CGS001-29957	SLC25A24	Mitochondrial nucleotide transporter subfamily			
5729	-73.48	kd	CGS001-5427	POLE2	DNA polymerases			
5730	-73.5	cc		BCL inhibitor	-			
5731	-73.5	kd	CGS001-10928	RALBP1	-			
5732	-73.53	kd	CGS001-3098	HK1	-			
5733	-73.6	cp	BRD-K79404599	enzastaurin	PKC inhibitor		PRKCB, AKT1, GSK3B, PRKCA, PRKCD, PRKCG	PKC inhibitor
5734	-73.62	oe	ccsbBroad304_07091	TPM1	Tropomyosins			
5735	-73.64	cp	BRD-K85606544	neratinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, KDR	EGFR inhibitor
5736	-73.65	cc		HIF activator	-			
5737	-73.66	cp	BRD-K81839095	estrone	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist, Estrogenic hormone
5738	-73.67	kd	CGS001-3117	HLA-DQA1	Immunoglobulin superfamily / C1-set domain containing			
5739	-73.7	oe	ccsbBroad304_02419	NDRG1	-			
5740	-73.73	cp	BRD-K60230970	MG-132	Proteasome inhibitor		PSMB1	Proteasome inhibitor
5741	-73.74	cp	BRD-A83326220	brazilin	Nitric oxide production inhibitor			Nitric oxide production inhibitor
5742	-73.76	oe	ccsbBroad304_01008	KITLG	-			
5743	-73.77	cp	BRD-A83892713	rifampicin	RNA polymerase inhibitor		NR1I2, ABCB1, CYP2B6, CYP2C19, CYP2C8, CYP3A4, CYP3A5, SLCO1A2, SLCO1B1, SLCO1B3	RNA polymerase inhibitor
5744	-73.77	cp	BRD-K63430059	methoxsalen	DNA synthesis inhibitor		ACHE, CYP1A2	DNA synthesis inhibitor
5745	-73.78	kd	CGS001-7353	UFD1L	-			
5746	-73.83	kd	CGS001-7099	TLR4	Toll-like receptor family			
5747	-73.85	kd	CGS001-6275	S100A4	EF-hand domain containing			
5748	-73.87	cp	BRD-A64125466	dehydrocholic-acid	choleretic agent			choleretic agent
5749	-73.88	oe	ccsbBroad304_08873	P2RY12	GPCR / Class A : Purinergic receptors, P2Y			
5750	-73.94	cp	BRD-K05181463	L-741626	Dopamine receptor antagonist		DRD2, DRD3, DRD4, HTR2A, HTR2B	Dopamine receptor antagonist
5751	-74.01	kd	CGS001-84634	KISS1R	GPCR / Class A : RF amide peptide receptors			
5752	-74.12	oe	ccsbBroad304_02094	FIBP	-			
5753	-74.12	kd	CGS001-2673	GFPT1	-			
5754	-74.23	cp	BRD-K59058766	chlorprothixene	Dopamine receptor antagonist		DRD2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, DRD1, DRD3, HRH1, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist
5755	-74.33	kd	CGS001-166793	ZBTB49	BTB/POZ domain containing			
5756	-74.34	cp	BRD-A18579359	wiskostatin	Neural Wiskott-Aldrich syndrome protein inhibitor		WAS, WASL	Neural Wiskott-Aldrich syndrome protein inhibitor
5757	-74.35	kd	CGS001-5297	PI4KA	1-phosphatidylinositol 4-kinase family			
5758	-74.5	oe	ccsbBroad304_01519	SET	-			
5759	-74.52	kd	CGS001-26353	HSPB8	Heat shock proteins / HSPB			
5760	-74.55	kd	CGS001-113451	ADC	-			
5761	-74.58	oe	ccsbBroad304_06401	HRH1	Histamine receptors			
5762	-74.58	kd	CGS001-2066	ERBB4	Type I RTKs: ErbB (epidermal growth factor) receptor family			
5763	-74.62	kd	CGS001-57547	ZNF624	Zinc fingers, C2H2-type			
5764	-74.65	kd	CGS001-30001	ERO1L	-			
5765	-74.74	kd	CGS001-10390	CEPT1	-			
5766	-74.76	cp	BRD-A27887842	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
5767	-74.79	oe	ccsbBroad304_01092	NFIL3	basic leucine zipper proteins			
5768	-74.82	oe	ccsbBroad304_09758	APOBEC3H	Apolipoprotein B mRNA editing enzymes			
5769	-74.86	cp	BRD-K45401373	betulinic-acid	Apoptosis stimulant		CASP3, CASP8, GPBAR1, TOP1	Apoptosis stimulant, Caspase activator, Diacylglycerol O acyltransferase inhibitor, HIV integrase inhibitor, NFkB pathway activator, NFkB pathway inhibitor, SARS coronavirus 3C-like protease inhibitor, Topoisomerase inhibitor
5770	-74.96	kd	CGS001-572	BAD	-			
5771	-74.98	cp	BRD-K39111395	BCL2-inhibitor	BCL inhibitor		BCL2	BCL inhibitor
5772	-75.05	oe	ccsbBroad304_01238	POLR2D	RNA polymerase subunits			
5773	-75.08	cp	BRD-K77390737	xanthohumol	ATPase inhibitor		CYP19A1, VCP	ATPase inhibitor
5774	-75.16	cp	BRD-K41445866	alfaxalone	Chloride channel agonist		HSD11B1	Chloride channel agonist, GABA receptor agonist
5775	-75.17	kd	CGS001-54749	EPDR1	-			
5776	-75.22	cp	BRD-A95513702	androsta-1,4-dien-3,17-dione	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
5777	-75.27	kd	CGS001-3156	HMGCR	Lanosterol biosynthesis pathway			
5778	-75.3	cc		Vitamin D receptor agonist	-			
5779	-75.31	kd	CGS001-6772	STAT1	SH2 domain containing			
5780	-75.35	oe	ccsbBroad304_00529	F3	CD molecules			
5781	-75.38	oe	ccsbBroad304_00273	CDC25B	Protein tyrosine phosphatases / Class III Cys-based PTPs			
5782	-75.38	cp	BRD-K85030058	benactyzine	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
5783	-75.49	cp	BRD-K59851896	calycanthine	GABA release inhibitor			GABA release inhibitor
5784	-75.49	kd	CGS001-818	CAMK2G	CAMK2 family			
5785	-75.51	oe	ccsbBroad304_04256	RNF146	RING-type (C3HC4) zinc fingers			
5786	-75.51	kd	CGS001-51284	TLR7	Toll-like receptor family			
5787	-75.52	cp	BRD-A79803969	memantine	Glutamate receptor antagonist		GRIN1, CHRFAM7A, CYP2E1, DRD2, GRIN2A, GRIN2B, GRIN3A, HTR3A	Glutamate receptor antagonist
5788	-75.54	cp	BRD-K78126613	menadione	Mitochondrial DNA polymerase inhibitor		AOX1, BGLAP, F10, F2, F7, F9, GGCX, NQO1, NQO2, PKM, PROC, PROS1, PROZ, VKORC1, VKORC1L1	Mitochondrial DNA polymerase inhibitor, Phosphatase inhibitor
5789	-75.55	cp	BRD-K97399794	quercetin	Polar auxin transport inhibitor		PIK3CG, AKR1B1, ATP5A1, ATP5B, ATP5C1, CYP2C8, EGFR, GAA, HCK, HIBCH, MAOA, PIM1, PTPN1, SCN5A, SIRT1, STK17B, UGT3A1, XDH	Polar auxin transport inhibitor
5790	-75.57	kd	CGS001-51728	POLR3K	RNA polymerase subunits			
5791	-75.6	kd	CGS001-2932	GSK3B	GSK subfamily			
5792	-75.63	oe	ccsbBroad304_11277	HAT1	Histone acetyltransferases (HATs)			
5793	-75.68	kd	CGS001-2834	PRLHR	GPCR / Class A : RF amide peptide receptors			
5794	-75.7	cp	BRD-A18202423	CPCCOEt	Glutamate receptor antagonist		GRM1	Glutamate receptor antagonist
5795	-75.7	kd	CGS001-55958	KLHL9	BTB/POZ domain containing			
5796	-75.73	cp	BRD-K64341947	CFM-1571	Guanylate cyclase activator			Guanylate cyclase activator
5797	-75.75	kd	CGS001-8741	TNFSF13	CD molecules			
5798	-75.77	kd	CGS001-8477	GPR65	GPCR / Class A : Orphans			
5799	-75.82	cp	BRD-K21806131	tegaserod	Serotonin receptor partial agonist		HTR4, HTR2B, HTR2A, HTR2C	Serotonin receptor partial agonist
5800	-75.98	cp	BRD-K34608650	BRD-K34608650	Cannabinoid receptor agonist		CNR2	Cannabinoid receptor agonist
5801	-75.98	kd	CGS001-7693	ZNF134	Zinc fingers, C2H2-type			
5802	-76	oe	ccsbBroad304_06374	HLA-DRA	Immunoglobulin superfamily / C1-set domain containing			
5803	-76	kd	CGS001-5245	PHB	-			
5804	-76.02	oe	ccsbBroad304_11054	PRKAR2A	Protein kinase A			
5805	-76.04	cp	BRD-K93034159	cladribine	Adenosine deaminase inhibitor		ADA, PNP, POLA1, POLE, POLE2, POLE3, POLE4, RRM1, RRM2, RRM2B	Adenosine deaminase inhibitor, Ribonucleoside reductase inhibitor
5806	-76.08	kd	CGS001-137209	ZNF572	Zinc fingers, C2H2-type			
5807	-76.09	kd	CGS001-10285	SMNDC1	Tudor domain containing			
5808	-76.14	cp	BRD-K00603606	ticlopidine	Purinergic receptor antagonist		P2RY12, CYP2B6, CYP2C19	Purinergic receptor antagonist
5809	-76.15	oe	ccsbBroad304_01841	BAG6	-			
5810	-76.16	oe	ccsbBroad304_01155	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
5811	-76.18	kd	CGS001-678	ZFP36L2	RING-type (C3HC4) zinc fingers			
5812	-76.19	cp	BRD-K47631482	bromhexine	Mucolytic agent			Mucolytic agent
5813	-76.2	oe	ccsbBroad304_01001	MEST	-			
5814	-76.2	kd	CGS001-55825	PECR	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 1			
5815	-76.3	cp	BRD-K72726508	arcyriaflavin-a	CDK inhibitor		CCND1, CCNE1, CDK2, CDK4	CDK inhibitor
5816	-76.34	kd	CGS001-5550	PREP	Prolyl oligopeptidase			
5817	-76.38	cp	BRD-K85015012	NNC-05-2090	GAT inhibitor		SLC6A11, SLC6A12, SLC6A13	GAT inhibitor, GABA uptake inhibitor
5818	-76.46	cp	BRD-K30240666	clemastine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
5819	-76.46	kd	CGS001-29880	ALG5	Glycosyltransferase family 2 domain containing			
5820	-76.48	kd	CGS001-51203	NUSAP1	-			
5821	-76.49	oe	ccsbBroad304_01262	PPP2CB	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
5822	-76.5	cp	BRD-K87573634	propylpyrazole	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
5823	-76.54	cp	BRD-K67445247	flurofamide	Urease inhibitor			Urease inhibitor
5824	-76.56	oe	ccsbBroad304_06081	DGKA	EF-hand domain containing			
5825	-76.57	kd	CGS001-53836	GPR87	GPCR / Class A : Orphans			
5826	-76.63	cp	BRD-K26801045	pipamperone	Dopamine receptor antagonist		DRD2, HTR2A, HRH1, HTR1A, HTR1B, HTR1D	Dopamine receptor antagonist
5827	-76.64	kd	CGS001-23585	TMEM50A	-			
5828	-76.65	cp	BRD-K08640512	RS-100329	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
5829	-76.66	cp	BRD-K55424922	anpirtoline	Serotonin receptor agonist		HTR1B, HTR3A	Serotonin receptor agonist
5830	-76.69	kd	CGS001-5327	PLAT	Chymotrypsin			
5831	-76.7	cp	BRD-K50422030	clomethiazole	GABA receptor antagonist		GABRA1	GABA receptor antagonist, GABA receptor modulator
5832	-76.8	cp	BRD-K85013741	auraptene	Nitric oxide production inhibitor		MAOB	Nitric oxide production inhibitor
5833	-76.83	cp	BRD-K62810658	PD-98059	MEK inhibitor		MAP2K1, AKT1, CHEK1, GSK3B, LCK, MAP2K2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK3, MAPK8, PRKCA, RAF1, ROCK1, RPS6KB1, SGK1	MEK inhibitor, MAP kinase inhibitor
5834	-76.83	kd	CGS001-5325	PLAGL1	Zinc fingers, C2H2-type			
5835	-76.88	kd	CGS001-9695	EDEM1	-			
5836	-76.94	oe	ccsbBroad304_10428	ETS2	ETS Transcription Factors			
5837	-77.01	cp	BRD-A56892734	esomeprazole	ATPase inhibitor		ATP4A, CYP2C19, CYP3A4	ATPase inhibitor
5838	-77.1	cp	BRD-K31633810	DAU-5884	Acetylcholine receptor antagonist		CHRM1, CHRM3	Acetylcholine receptor antagonist
5839	-77.17	oe	ccsbBroad304_04454	FBXL20	F-boxes / Leucine-rich repeats			
5840	-77.18	cp	BRD-K70330367	amantadine	Glutamate receptor antagonist		DRD2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A	Glutamate receptor antagonist
5841	-77.18	kd	CGS001-26762	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
5842	-77.2	kd	CGS001-6307	MSMO1	Fatty acid hydroxylase domain containing			
5843	-77.25	cp	BRD-K78122587	NNC-55-0396	T-type calcium channel blocker		CATSPER1, CATSPER2, CATSPER3, CATSPER4	T-type calcium channel blocker
5844	-77.26	kd	CGS001-5013	OTX1	Homeoboxes / PRD class			
5845	-77.29	cp	BRD-K99451608	lopinavir	HIV protease inhibitor			HIV protease inhibitor
5846	-77.29	kd	CGS001-4609	MYC	Basic helix-loop-helix proteins			
5847	-77.3	cp	BRD-K15409150	penfluridol	T-type calcium channel blocker		CACNA1G, DRD1, DRD2	T-type calcium channel blocker
5848	-77.35	kd	CGS001-5583	PRKCH	Eta subfamily			
5849	-77.35	kd	CGS001-79139	DERL1	-			
5850	-77.4	cp	BRD-K31987754	oleylethanolamide	Cannabinoid receptor agonist		GPR119, CNR1, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Potassium channel blocker, Glucose dependent insulinotropic receptor agonist
5851	-77.41	oe	ccsbBroad304_00709	GUK1	-			
5852	-77.42	cp	BRD-K54142781	cirazoline	Adrenergic receptor agonist		ADRA1A	Adrenergic receptor agonist
5853	-77.45	cp	BRD-A93477898	PETCM	Caspase activator		CASP3	Caspase activator
5854	-77.56	cp	BRD-K73293050	WZ-3146	EGFR inhibitor		EGFR	EGFR inhibitor
5855	-77.58	oe	ccsbBroad304_09656	ZNF555	Zinc fingers, C2H2-type			
5856	-77.58	kd	CGS001-2235	FECH	-			
5857	-77.59	kd	CGS001-29965	C16ORF5	-			
5858	-77.64	kd	CGS001-3017	HIST1H2BD	Histones / Replication-dependent			
5859	-77.65	kd	CGS001-3516	RBPJ	-			
5860	-77.66	oe	ccsbBroad304_05422	VN1R5	GPCR / Unclassified : Vomeronasal receptors, type 1			
5861	-77.69	kd	CGS001-121599	SPIC	ETS Transcription Factors			
5862	-77.7	cp	BRD-K00206590	P-1075	ATP channel activator		KCNJ8	ATP channel activator, Potassium channel activator
5863	-77.73	oe	ccsbBroad304_00611	GALE	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
5864	-77.73	cp	BRD-K67637637	olopatadine	Histamine receptor antagonist		HRH1, S100A1, S100A12, S100A13, S100A2, S100B	Histamine receptor antagonist
5865	-77.75	oe	ccsbBroad304_00755	HMGCR	Lanosterol biosynthesis pathway			
5866	-77.8	kd	CGS001-3985	LIMK2	LIMK subfamily			
5867	-77.84	oe	ccsbBroad304_08534	STRADB	STLK subfamily			
5868	-77.85	kd	CGS001-780	DDR1	Type XVI RTKs: DDR (collagen receptor) family			
5869	-77.86	oe	ccsbBroad304_02500	RRAGA	-			
5870	-77.87	oe	ccsbBroad304_03761	LHX9	Homeoboxes / LIM class			
5871	-77.87	cp	BRD-K47780086	penciclovir	DNA directed DNA polymerase inhibitor			DNA directed DNA polymerase inhibitor
5872	-77.92	oe	ccsbBroad304_01283	PRKCE	Eta subfamily			
5873	-77.99	cp	BRD-K69032158	diprotin-a	Dipeptidyl peptidase inhibitor		DPP4	Dipeptidyl peptidase inhibitor
5874	-78.02	kd	CGS001-6670	SP3	Specificity protein transcription factors			
5875	-78.03	oe	ccsbBroad304_08734	ZNF490	Zinc fingers, C2H2-type			
5876	-78.03	oe	ccsbBroad304_07632	PROCR	CD molecules			
5877	-78.11	oe	ccsbBroad304_05183	TXLNA	-			
5878	-78.12	cp	BRD-A59303141	quinethazone	Thiazide diuretic		CA1, CA2, SLC12A1, SLC12A2, SLC12A3	Thiazide diuretic
5879	-78.13	cp	BRD-A21858158	praziquantel	Anthelmintic			Anthelmintic
5880	-78.13	kd	CGS001-6428	SRSF3	RNA binding motif (RRM) containing			
5881	-78.14	oe	ccsbBroad304_03939	RNF25	RING-type (C3HC4) zinc fingers			
5882	-78.15	oe	ccsbBroad304_01894	HIST1H2AC	Histones / Replication-dependent			
5883	-78.21	oe	ccsbBroad304_04567	ZNF300	Zinc fingers, C2H2-type			
5884	-78.23	kd	CGS001-55191	NADSYN1	-			
5885	-78.25	cp	BRD-K44497846	enalapril	ACE inhibitor		ACE	ACE inhibitor
5886	-78.26	cp	BRD-A35623999	CGP-37157	L-type calcium channel blocker		SLC8A1	L-type calcium channel blocker, Mitochondrial Na+/Ca2+ exchanger antagonist, Sodium/calcium exchange inhibitor
5887	-78.28	kd	CGS001-26993	AKAP8L	-			
5888	-78.34	oe	ccsbBroad304_05796	AK1	Adenylate kinases			
5889	-78.36	kd	CGS001-124641	OVCA2	-			
5890	-78.39	kd	CGS001-2690	GHR	Prolactin receptor family			
5891	-78.48	cp	BRD-K76907295	VU-0418947-2	HIF modulator			HIF modulator
5892	-78.51	kd	CGS001-11212	PROSC	-			
5893	-78.53	cp	BRD-A37347161	BRL-52537	Opioid receptor agonist		OPRK1	Opioid receptor agonist
5894	-78.55	kd	CGS001-2760	GM2A	-			
5895	-78.59	kd	CGS001-266977	GPR110	Adhesion Class GPCRs			
5896	-78.6	cp	BRD-A86044036	flurbiprofen	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
5897	-78.61	kd	CGS001-10954	PDIA5	Protein disulfide isomerases			
5898	-78.73	kd	CGS001-3119	HLA-DQB1	Immunoglobulin superfamily / C1-set domain containing			
5899	-78.74	cc		Toll like receptors LOF	-			
5900	-78.8	cp	BRD-A63667919	methylergometrine	Dopamine receptor antagonist		DRD1, HTR1E, HTR1F, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
5901	-78.82	oe	ccsbBroad304_02469	SLC35A1	SLC35 family of nucleotide sugar transporters			
5902	-78.83	oe	ccsbBroad304_00564	FGR	Src family			
5903	-78.84	kd	CGS001-6909	TBX2	T-boxes			
5904	-78.93	cc		CDK inhibitor	-			
5905	-78.97	kd	CGS001-5352	PLOD2	-			
5906	-78.98	oe	ccsbBroad304_03323	LARS	Aminoacyl tRNA synthetases / Class I			
5907	-79	cp	BRD-A41555725	chlortetracycline	Protein synthesis inhibitor			Protein synthesis inhibitor
5908	-79.03	oe	ccsbBroad304_01858	FOSL1	basic leucine zipper proteins			
5909	-79.05	kd	CGS001-8536	CAMK1	CAMK1 family			
5910	-79.07	cp	BRD-A00267231	hemado	Adenosine receptor agonist		ADORA3, ADORA1, ADORA2A, ADORA2B	Adenosine receptor agonist
5911	-79.08	kd	CGS001-4547	MTTP	-			
5912	-79.09	oe	ccsbBroad304_00156	BCL2L1	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
5913	-79.1	cp	BRD-K85090592	pilocarpine	Acetylcholine receptor agonist		CHRM3, CHRM1, CHRM2, CHRM4, CHRM5	Acetylcholine receptor agonist
5914	-79.1	cp	BRD-K11399644	phenformin	AMPK activator		KCNJ8, PRKAA1	AMPK activator
5915	-79.1	cp	BRD-K76568384	PHTPP	Estrogen receptor antagonist		ESR2	Estrogen receptor antagonist
5916	-79.12	cc		Beta-adrenergic receptor agonist	-			
5917	-79.14	kd	CGS001-7083	TK1	-			
5918	-79.25	kd	CGS001-85315	PAQR8	-			
5919	-79.26	cp	BRD-K80639402	SB-258585	Serotonin receptor antagonist		HTR6	Serotonin receptor antagonist
5920	-79.26	cp	BRD-K36616567	doxepin	Histamine receptor antagonist		HRH1, HRH2, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH4, HTR1A, HTR2A, HTR2B, HTR2C, HTR6, KCNH2, SLC6A3	Histamine receptor antagonist
5921	-79.27	cp	BRD-K22878149	SB-205607	Delta 1 opioid receptor agonist		OPRD1, OPRK1, OPRM1	Delta 1 opioid receptor agonist
5922	-79.28	kd	CGS001-23061	TBC1D9B	EF-hand domain containing			
5923	-79.29	cp	BRD-A39052811	mosapride	Serotonin receptor agonist		HTR4, HTR3A	Serotonin receptor agonist
5924	-79.31	cp	BRD-A87479750	tenidap	Cyclooxygenase inhibitor		ALOX5, KCNJ4, PTGS1	Cyclooxygenase inhibitor
5925	-79.31	cp	BRD-K31627533	rimexolone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist
5926	-79.37	kd	CGS001-546	ATRX	-			
5927	-79.37	kd	CGS001-5763	PTMS	-			
5928	-79.38	kd	CGS001-29888	STRN4	WD repeat domain containing			
5929	-79.39	kd	CGS001-23378	RRP8	-			
5930	-79.4	kd	CGS001-23212	RRS1	-			
5931	-79.53	cp	BRD-K28761384	zuclopenthixol	Dopamine receptor antagonist		DRD2, DRD1, ADRA1A, ADRA2A, DRD5, HRH1, HTR2A	Dopamine receptor antagonist
5932	-79.55	oe	ccsbBroad304_00977	MAX	Basic helix-loop-helix proteins			
5933	-79.55	kd	CGS001-4835	NQO2	-			
5934	-79.56	cp	BRD-A29485665	bicalutamide	Androgen receptor antagonist		AR, CYP2C19	Androgen receptor antagonist
5935	-79.57	kd	CGS001-23588	KLHDC2	-			
5936	-79.58	oe	ccsbBroad304_04095	CHMP6	Charged multivesicular body proteins			
5937	-79.61	kd	CGS001-7013	TERF1	-			
5938	-79.72	oe	ccsbBroad304_00846	IL2	Interleukins and interleukin receptors			
5939	-79.8	kd	CGS001-64343	AZI2	-			
5940	-79.82	kd	CGS001-53632	PRKAG3	AMPK subfamily			
5941	-79.82	kd	CGS001-338	APOB	Apolipoproteins			
5942	-79.83	cp	BRD-K95435023	PHA-665752	c-Met inhibitor		MET	c-Met inhibitor
5943	-79.88	cp	BRD-K52850071	JAK3-Inhibitor-II	JAK inhibitor		EGFR, ALK, JAK1, JAK2, JAK3	JAK inhibitor
5944	-79.93	kd	CGS001-3336	HSPE1	Heat Shock Proteins / Chaperonins			
5945	-79.94	kd	CGS001-6659	SOX4	SRY (sex determining region Y)-boxes			
5946	-79.95	cp	BRD-K50168500	canertinib	EGFR inhibitor		EGFR, ERBB2, ERBB4, AKT1	EGFR inhibitor
5947	-79.97	cp	BRD-A68888262	azelastine	Histamine receptor antagonist		HRH1, CYP2C19	Histamine receptor antagonist
5948	-80.01	cp	BRD-K44067360	flufenamic-acid	Chloride channel blocker		AKR1C3, AR, PTGS1, PTGS2, ANO1, GJA1, GJA10, GJA3, GJA4, GJA5, GJA8, GJA9, GJB1, GJB2, GJB3, GJB4, GJB5, GJB6, GJB7, GJC1, GJC2, GJC3, GJD2, GJD3, GJD4, GJE1, PANX1, PANX2, PANX3, PKD2L1, TRPC5, TRPM2, TRPM5	Chloride channel blocker
5949	-80.04	cp	BRD-A02990301	lofexidine	Adrenergic receptor agonist		ADRA2A	Adrenergic receptor agonist
5950	-80.07	oe	ccsbBroad304_03382	ZAK	MLK subfamily			
5951	-80.07	oe	ccsbBroad304_02497	YKT6	-			
5952	-80.12	cc		Canonical high mobility group proteins LOF	-			
5953	-80.13	oe	ccsbBroad304_02761	SIRT3	Histone deacetylases (HDACs)			
5954	-80.13	cp	BRD-K98530306	clonidine	Adrenergic receptor agonist		ADRA2A, ADRA2B, ADRA2C, ADRA1A, ADRA1B, ADRA1D	Adrenergic receptor agonist
5955	-80.16	oe	ccsbBroad304_01662	TFDP2	-			
5956	-80.17	kd	CGS001-6821	SUOX	-			
5957	-80.17	kd	CGS001-2000	ELF4	ETS Transcription Factors			
5958	-80.17	kd	CGS001-837	CASP4	Caspases			
5959	-80.18	cp	BRD-A90131694	alclometasone	Glucocorticoid receptor agonist		NR3C1, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
5960	-80.2	kd	CGS001-7384	UQCRC1	Mitochondrial respiratory chain complex / Complex III			
5961	-80.26	cp	BRD-K37206356	rhamnetin	HDAC inhibitor		ALOX5, MAPK8	HDAC inhibitor
5962	-80.28	kd	CGS001-23647	ARFIP2	-			
5963	-80.29	kd	CGS001-27	ABL2	Abl family			
5964	-80.31	cp	BRD-K65417056	meprylcaine	Local anesthetic			Local anesthetic
5965	-80.33	cp	BRD-K62353524	DY-131	Estrogen receptor agonist		ESR2, ESRRB, ESRRG	Estrogen receptor agonist
5966	-80.34	cp	BRD-A78295502	hydroquinine	Antiarrhythmic			Antiarrhythmic
5967	-80.35	kd	CGS001-56993	TOMM22	-			
5968	-80.41	cp	BRD-K17075857	chloroxine	Opioid receptor antagonist		OPRK1	Opioid receptor antagonist
5969	-80.48	kd	CGS001-26191	PTPN22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
5970	-80.51	cp	BRD-K34092021	arvanil	TRPV agonist		CNR1, TRPV1	TRPV agonist
5971	-80.52	kd	CGS001-6184	RPN1	-			
5972	-80.54	cp	BRD-K02130563	panobinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC4, HDAC6, HDAC7, HDAC8, HDAC9	HDAC inhibitor
5973	-80.6	oe	ccsbBroad304_00651	GNAI3	-			
5974	-80.6	oe	ccsbBroad304_07548	TSSC4	-			
5975	-80.6	kd	CGS001-3566	IL4R	IL-2 receptor family			
5976	-80.65	cp	BRD-K94144010	cotinine	Nicotine metabolite			Nicotine metabolite
5977	-80.68	oe	ccsbBroad304_02306	PQBP1	-			
5978	-80.68	oe	ccsbBroad304_02565	RALBP1	-			
5979	-80.74	kd	CGS001-285601	GPR150	GPCR / Class A : Orphans			
5980	-80.75	oe	ccsbBroad304_09316	ISX	Homeoboxes / PRD class			
5981	-80.76	oe	ccsbBroad304_08128	ALG5	Glycosyltransferase family 2 domain containing			
5982	-80.78	cp	BRD-A42831637	tetrahydrocannabinol-7-oic-acid	Anti-inflammatory			Anti-inflammatory, Cannabinoid metabolite
5983	-80.8	cp	BRD-A50157456	terbutaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
5984	-80.8	kd	CGS001-9337	CNOT8	-			
5985	-80.88	cp	BRD-K83289131	CAY-10618	NAMPT inhibitor		NAMPT	NAMPT inhibitor
5986	-80.9	kd	CGS001-5993	RFX5	-			
5987	-80.93	cp	BRD-K52735702	cefdinir	Bacterial cell wall synthesis inhibitor		MPO	Bacterial cell wall synthesis inhibitor
5988	-80.93	cp	BRD-K14765469	vesamicol	Acetylcholinesterase inhibitor		SLC18A3	Acetylcholinesterase inhibitor
5989	-80.98	oe	ccsbBroad304_01672	TIMP2	-			
5990	-81.06	cp	BRD-K64514229	toltrazuril	Antiprotozoal			Antiprotozoal
5991	-81.08	cc		Topoisomerase inhibitor	-			
5992	-81.1	oe	ccsbBroad304_09497	ZNF57	Zinc fingers, C2H2-type			
5993	-81.13	cp	BRD-K34415467	trimethobenzamide	Histamine receptor antagonist		DRD2	Histamine receptor antagonist
5994	-81.24	cp	BRD-K16485616	mocetinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC11	HDAC inhibitor
5995	-81.32	kd	CGS001-3656	IRAK2	Interleukin-1 receptor-associated kinase (IRAK) family			
5996	-81.39	kd	CGS001-5777	PTPN6	Protein tyrosine phosphatases			
5997	-81.49	cp	BRD-K19533706	tranilast	Angiogenesis inhibitor		HPGDS, HRH1, IDO1, IFNG, IL10, IL2, IL4, SLC22A12, TGFB1, TNF, TRPV2	Angiogenesis inhibitor
5998	-81.51	kd	CGS001-8089	YEATS4	-			
5999	-81.52	oe	ccsbBroad304_03652	EXOC2	-			
6000	-81.56	oe	ccsbBroad304_01234	POLB	DNA polymerases			
6001	-81.56	cp	BRD-A82371568	clofarabine	Ribonucleoside reductase inhibitor		RRM1, POLA1, RRM2, SLC22A8	Ribonucleoside reductase inhibitor
6002	-81.56	kd	CGS001-7697	ZNF138	Zinc fingers, C2H2-type			
6003	-81.59	kd	CGS001-4601	MXI1	Basic helix-loop-helix proteins			
6004	-81.61	oe	ccsbBroad304_04117	SLC25A22	Mitochondrial amino acid transporter subfamily			
6005	-81.64	cp	BRD-K41996876	tyrphostin-1	EGFR inhibitor		EGFR	EGFR inhibitor
6006	-81.66	cp	BRD-K01253243	SB-590885	RAF inhibitor		BRAF	RAF inhibitor
6007	-81.8	oe	ccsbBroad304_07662	NPRL2	-			
6008	-81.8	cp	BRD-K01095011	finasteride	5-alpha reductase inhibitor		SRD5A2, SRD5A1, AKR1D1, AR	5-alpha reductase inhibitor
6009	-81.8	kd	CGS001-25797	QPCT	Aminopeptidase Y			
6010	-81.84	cp	BRD-K24526313	levcromakalim	Potassium channel activator		KCNJ8, ABCC9, KCNJ5	Potassium channel activator
6011	-81.89	oe	ccsbBroad304_00394	CTSD	Cathepsins			
6012	-81.89	cp	BRD-K38903228	hesperidin	Flavanone glycoside		CACNA1B	Flavanone glycoside
6013	-81.91	kd	CGS001-25839	COG4	Components of oligomeric golgi complex			
6014	-81.93	kd	CGS001-29850	TRPM5	Transient Receptor Potential channels			
6015	-81.94	cp	BRD-K12260308	xanthoxyline	Antifungal			Antifungal
6016	-82.01	cp	BRD-K09485525	GANT-61	GLI antagonist		DHH, IHH	GLI antagonist
6017	-82.01	kd	CGS001-775	CACNA1C	Calcium channel subunits			
6018	-82.04	cp	BRD-K71035033	masitinib	KIT inhibitor		KIT, FGFR3, LYN, PDGFRA, PDGFRB	KIT inhibitor, PDGFR receptor inhibitor, SRC inhibitor
6019	-82.08	oe	ccsbBroad304_06282	GLDC	-			
6020	-82.13	oe	ccsbBroad304_00810	HYAL1	-			
6021	-82.17	cp	BRD-A43671941	oxprenolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6022	-82.18	kd	CGS001-11044	PAPD7	-			
6023	-82.27	cc		IL4 Pathway LOF	-			
6024	-82.27	oe	ccsbBroad304_01664	TGFA	-			
6025	-82.38	kd	CGS001-79724	ZNF768	Zinc fingers, C2H2-type			
6026	-82.43	cp	BRD-A41450521	tosufloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6027	-82.44	kd	CGS001-9261	MAPKAPK2	MAPKAPK subfamily			
6028	-82.49	oe	ccsbBroad304_08715	SALL4	Zinc fingers, C2H2-type			
6029	-82.63	cp	BRD-K49810818	sorafenib	FLT3 inhibitor		RET, BRAF, FLT3, KDR, RAF1, FLT1, FLT4, KIT, DDR2, FGFR1, PDGFRB, CYP2B6, CYP2C8, CYP3A5, PDGFB, SLCO1B3	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor, RAF inhibitor, VEGFR inhibitor, RET tyrosine kinase inhibitor
6030	-82.65	kd	CGS001-6657	SOX2	SRY (sex determining region Y)-boxes			
6031	-82.65	kd	CGS001-140609	NEK7	NIMA (never in mitosis gene a)- related kinase (NEK) family			
6032	-82.67	kd	CGS001-84844	PHF5A	Zinc fingers, PHD-type			
6033	-82.68	oe	ccsbBroad304_00003	ABAT	GABA turnover			
6034	-82.7	kd	CGS001-3074	HEXB	-			
6035	-82.73	kd	CGS001-3988	LIPA	-			
6036	-82.74	oe	ccsbBroad304_06410	HSPA8	Heat shock proteins / HSP70			
6037	-82.74	kd	CGS001-11320	MGAT4A	-			
6038	-82.81	kd	CGS001-56647	BCCIP	-			
6039	-82.82	cp	BRD-A85234536	N6-cyclopentyladenosine	Adenosine receptor agonist		ADORA1, ADORA2A, ADORA2B, ADORA3, SLC29A1	Adenosine receptor agonist
6040	-82.83	cp	BRD-K09497549	kawain	Calcium channel modulator		MTOR	Calcium channel modulator, MTOR inhibitor, Sodium channel blocker
6041	-82.89	kd	CGS001-9655	SOCS5	SH2 domain containing			
6042	-82.92	cp	BRD-K60460488	nelfinavir	HIV protease inhibitor		CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
6043	-82.94	kd	CGS001-6093	ROCK1	Pleckstrin homology (PH) domain containing			
6044	-82.95	kd	CGS001-7541	ZFP161	-			
6045	-83	cp	BRD-A03623303	metoprolol	Adrenergic receptor antagonist		ADRB1, ADRB2	Adrenergic receptor antagonist
6046	-83.01	kd	CGS001-115560	ZNF501	Zinc fingers, C2H2-type			
6047	-83.02	cp	BRD-A01643550	prednisolone	Glucocorticoid receptor agonist		NR3C1, NR3C2, SERPINA6	Glucocorticoid receptor agonist
6048	-83.02	cp	BRD-A97739905	ketoprofen	Cyclooxygenase inhibitor		PTGS2, PTGS1, CXCR1, SLC5A8	Cyclooxygenase inhibitor
6049	-83.02	kd	CGS001-5585	PKN1	Protein kinase N (PKN) family			
6050	-83.02	kd	CGS001-56882	CDC42SE1	-			
6051	-83.04	cp	BRD-A39172021	ampiroxicam	Cyclooxygenase inhibitor		PTGS1, PTGS2	Cyclooxygenase inhibitor
6052	-83.05	kd	CGS001-29883	CNOT7	-			
6053	-83.09	cc		Lysine acetyltransferases LOF	-			
6054	-83.09	kd	CGS001-4869	NPM1	-			
6055	-83.14	kd	CGS001-54899	PXK	Slob family			
6056	-83.2	oe	ccsbBroad304_02108	AURKB	Aurora kinase			
6057	-83.2	cp	BRD-K78485176	olmesartan	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
6058	-83.22	kd	CGS001-3109	HLA-DMB	Immunoglobulin superfamily / C1-set domain containing			
6059	-83.25	cp	BRD-K12357156	AG-490	EGFR inhibitor		JAK2, JAK3, EGFR, STAT3	EGFR inhibitor, ErbB2 inhibitor, JAK inhibitor
6060	-83.29	cp	BRD-K64044582	linoleamide	ACAT inhibitor		SOAT1, SOAT2	ACAT inhibitor
6061	-83.32	kd	CGS001-36	ACADSB	-			
6062	-83.33	oe	ccsbBroad304_00654	GNB1	WD repeat domain containing			
6063	-83.35	cc		T-type calcium channel blocker	-			
6064	-83.36	kd	CGS001-4938	OAS1	-			
6065	-83.4	cp	BRD-K50891186	GR-103691	Dopamine receptor antagonist			Dopamine receptor antagonist
6066	-83.42	cp	BRD-K89997465	chlorpromazine	Dopamine receptor antagonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HRH1, HTR1A, HTR2A, HTR2C, HTR6, HTR7, ADRA1A, ADRA1B, ADRA1D, CALM1, CHRM1, CHRM3, HRH4, HTR2B, KCNH2, KIF11, ORM1, ORM2, SMPD1, TRPC5	Dopamine receptor antagonist
6067	-83.43	kd	CGS001-51701	NLK	nmo subfamily			
6068	-83.44	cc		Aldehyde dehydrogenases LOF	-			
6069	-83.45	cp	BRD-K06593056	LE-135	Retinoid receptor agonist		RARB	Retinoid receptor agonist
6070	-83.5	cp	BRD-K16195444	oxymetazoline	Adrenergic receptor agonist		ADRA1A, ADRA2A, ADRA1B, ADRA1D, ADRA2B, ADRA2C, CYP2C19, HTR1B, HTR1D, HTR2C	Adrenergic receptor agonist
6071	-83.51	cp	BRD-K50495309	SRC-kinase-inhibitor-I	SRC inhibitor		CSK, LCK, RIPK2	SRC inhibitor
6072	-83.52	cp	BRD-K10974103	diloxanide	Protein synthesis inhibitor			Protein synthesis inhibitor
6073	-83.54	cc		EGFR inhibitor	-			
6074	-83.57	kd	CGS001-4069	LYZ	-			
6075	-83.59	oe	ccsbBroad304_06340	GTF2H3	General transcription factors			
6076	-83.63	oe	ccsbBroad304_01684	TNF	Tumor necrosis factor (ligand) superfamily			
6077	-83.65	cp	BRD-K57718010	pentylenetetrazol	GABA receptor antagonist			GABA receptor antagonist
6078	-83.67	oe	ccsbBroad304_05767	ACVR1	Type I receptor serine/threonine kinases			
6079	-83.69	oe	ccsbBroad304_04752	IKBIP	-			
6080	-83.69	kd	CGS001-5999	RGS4	Regulators of G-protein signaling			
6081	-83.69	kd	CGS001-56654	NPDC1	-			
6082	-83.7	oe	ccsbBroad304_01642	TAL2	Basic helix-loop-helix proteins			
6083	-83.71	oe	ccsbBroad304_06120	DRD1	Dopamine receptors			
6084	-83.75	cp	BRD-K68558722	deracoxib	Cyclooxygenase inhibitor		PTGS2	Cyclooxygenase inhibitor
6085	-83.79	oe	ccsbBroad304_02242	SNX17	Sorting nexins			
6086	-83.8	cp	BRD-A02176148	tubaic-acid	Mitochondrial complex I inhibitor		MT-ND1	Mitochondrial complex I inhibitor, NADH-ubiquinone oxidoreductase (Complex I) inhibitor
6087	-83.83	oe	ccsbBroad304_04064	PRR15L	-			
6088	-83.85	kd	CGS001-28985	MCTS1	-			
6089	-83.86	cp	BRD-A36217750	sulfinpyrazone	Uricosuric blocker		ABCC1, ABCC2, FPR1, SLC22A12	Uricosuric blocker
6090	-83.89	kd	CGS001-1482	NKX2-5	Homeoboxes / ANTP class : NKL subclass			
6091	-83.9	oe	ccsbBroad304_05192	SPRED2	-			
6092	-83.9	cp	BRD-K64890080	BI-2536	PLK inhibitor		PLK1, BRD4, PLK2, PLK3	PLK inhibitor
6093	-83.9	kd	CGS001-9887	SMG7	-			
6094	-83.94	cp	BRD-K90864987	cobalt(II)-chloride	HSP inducer		HIF1A	HSP inducer
6095	-83.95	cp	BRD-A77118605	BML-ST330	Phospholipase inhibitor			Phospholipase inhibitor
6096	-84	cp	BRD-A65767837	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6097	-84.03	kd	CGS001-5440	POLR2K	RNA polymerase subunits			
6098	-84.04	cp	BRD-K64746805	MBCQ	Phosphodiesterase inhibitor		PDE5A	Phosphodiesterase inhibitor
6099	-84.05	cp	BRD-K53913732	SB-408124	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
6100	-84.06	cp	BRD-K62996583	lidoflazine	Calcium channel blocker		SCN1A, SCN3A, SLC29A1	Calcium channel blocker
6101	-84.07	oe	ccsbBroad304_02187	POLR1C	RNA polymerase subunits			
6102	-84.09	kd	CGS001-3895	KTN1	-			
6103	-84.12	cp	BRD-A75479906	rimantadine	Antiviral			Antiviral, RNA synthesis inhibitor
6104	-84.17	oe	ccsbBroad304_00845	IL1RAP	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6105	-84.19	cp	BRD-K15108141	gemcitabine	Ribonucleotide reductase inhibitor		RRM1, CMPK1, RRM2, TYMS	Ribonucleotide reductase inhibitor
6106	-84.19	kd	CGS001-7357	UGCG	Glycosyltransferase family 2 domain containing			
6107	-84.23	oe	ccsbBroad304_03858	SRPRB	-			
6108	-84.32	kd	CGS001-9275	BCL7B	-			
6109	-84.36	kd	CGS001-388677	NOTCH2NL	-			
6110	-84.37	cp	BRD-A70449690	forskolin	Adenylyl cyclase activator		ADCY2, ADCY5, GNAS	Adenylyl cyclase activator
6111	-84.4	kd	CGS001-5252	PHF1	Zinc fingers, PHD-type			
6112	-84.43	cc		Angiotensin receptor antagonist	-			
6113	-84.44	cp	BRD-K76698671	HNHA	HDAC inhibitor		HDAC1	HDAC inhibitor
6114	-84.45	kd	CGS001-5577	PRKAR2B	Protein kinase A			
6115	-84.45	kd	CGS001-23223	RRP12	-			
6116	-84.46	cp	BRD-A55946879	BW-B70C	Lipoxygenase inhibitor		ALOX5	Lipoxygenase inhibitor
6117	-84.48	cc		Tachykinin antagonist	-			
6118	-84.53	oe	ccsbBroad304_00262	CD59	CD molecules			
6119	-84.53	kd	CGS001-1201	CLN3	-			
6120	-84.54	kd	CGS001-7580	ZNF32	Zinc fingers, C2H2-type			
6121	-84.54	cp	BRD-A47513740	calyculin	Protein phosphatase inhibitor		PPP1CA, PPP1CC, PPP2CA	Protein phosphatase inhibitor
6122	-84.56	kd	CGS001-64863	METTL4	-			
6123	-84.6	cp	BRD-K11630072	carmofur	Thymidylate synthase inhibitor		TYMS	Thymidylate synthase inhibitor
6124	-84.6	kd	CGS001-3398	ID2	Basic helix-loop-helix proteins			
6125	-84.64	cp	BRD-K01555864	dibenzoylmethane	Antineoplastic			Antineoplastic
6126	-84.64	kd	CGS001-10270	AKAP8	A-kinase anchor proteins			
6127	-84.65	cp	BRD-A06352418	terfenadine	Histamine receptor antagonist		HRH1, KCNH2, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, KCNH1	Histamine receptor antagonist
6128	-84.66	oe	ccsbBroad304_07178	ZFP112	-			
6129	-84.69	cp	BRD-A65440446	cimaterol	Adrenergic receptor agonist			Adrenergic receptor agonist
6130	-84.69	cp	BRD-K28806945	L-750667	Dopamine receptor antagonist		DRD4	Dopamine receptor antagonist
6131	-84.73	oe	ccsbBroad304_06814	PTPN12	Protein tyrosine phosphatases / Class I Cys-based PTPs : Non-receptor			
6132	-84.73	cp	BRD-K73196317	urapidil	Adrenergic receptor antagonist		HTR1A	Adrenergic receptor antagonist
6133	-84.74	oe	ccsbBroad304_01356	QDPR	Short chain dehydrogenase/reductase superfamily / Atypical members			
6134	-84.76	kd	CGS001-9112	MTA1	GATA zinc finger domain containing			
6135	-84.78	kd	CGS001-10400	PEMT	-			
6136	-84.79	oe	ccsbBroad304_05560	AMIGO3	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6137	-84.79	cp	BRD-K40919711	BAPTA-AM	Potassium channel blocker		KCNA3, KCNA5, KCNH2	Potassium channel blocker
6138	-84.79	kd	CGS001-6906	SERPINA7	Serine (or cysteine) peptidase inhibitors			
6139	-84.83	oe	ccsbBroad304_03878	SENP2	-			
6140	-84.83	oe	ccsbBroad304_01164	PDHB	-			
6141	-84.85	cp	BRD-K72895815	SSR-69071	Leukocyte elastase inhibitor		ELANE	Leukocyte elastase inhibitor
6142	-84.85	kd	CGS001-966	CD59	CD molecules			
6143	-84.91	kd	CGS001-716	C1S	Complement system			
6144	-84.93	cp	BRD-A51182606	chloramphenicol	Protein synthesis inhibitor		CD55, CYP2C19	Protein synthesis inhibitor, Bacterial 50S ribosomal subunit inhibitor
6145	-84.93	cp	BRD-K78431006	crizotinib	ALK inhibitor		ALK, MET, CYP2B6, CYP3A5, MST1R, ROS1	ALK inhibitor
6146	-84.93	kd	CGS001-1196	CLK2	CDC-like kinases			
6147	-85	kd	CGS001-23236	PLCB1	Phosphoinositide-specific phospholipase C			
6148	-85.03	kd	CGS001-23384	SPECC1L	-			
6149	-85.04	cc		Bacterial DNA gyrase inhibitor	-			
6150	-85.04	oe	ccsbBroad304_07363	AIFM1	-			
6151	-85.05	oe	ccsbBroad304_00527	F2RL1	GPCR / Class A : Protease activated receptors			
6152	-85.1	kd	CGS001-170463	SSBP4	-			
6153	-85.11	kd	CGS001-847	CAT	-			
6154	-85.14	kd	CGS001-2037	EPB41L2	-			
6155	-85.21	kd	CGS001-2171	FABP5	Fatty acid-binding proteins			
6156	-85.26	cp	BRD-K18036262	L-168049	Glucagon receptor antagonist		GCGR	Glucagon receptor antagonist
6157	-85.27	kd	CGS001-29994	BAZ2B	Zinc fingers, PHD-type			
6158	-85.29	cp	BRD-K39391626	ethylestrenol	Progesterone receptor agonist		AR	Progesterone receptor agonist
6159	-85.3	cc		Ribonucleotide reductase inhibitor	-			
6160	-85.31	oe	ccsbBroad304_06681	P2RY2	GPCR / Class A : Purinergic receptors, P2Y			
6161	-85.35	kd	CGS001-6857	SYT1	Synaptotagmins			
6162	-85.36	kd	CGS001-3163	HMOX2	Haem oxygenase			
6163	-85.43	kd	CGS001-9246	UBE2L6	Ubiquitin-conjugating enzymes E2			
6164	-85.47	cp	BRD-K43245338	MDL-28170	Calpain inhibitor		CAPN1, CTSB, CTSL	Calpain inhibitor
6165	-85.5	oe	ccsbBroad304_07026	SYT1	Synaptotagmins			
6166	-85.59	cp	BRD-K30020243	aliskiren	Antihypertensive		REN	Antihypertensive, Peptidase inhibitor, Protease inhibitor, Renin inhibitor
6167	-85.6	kd	CGS001-3767	KCNJ11	Inwardly rectifying potassium channels			
6168	-85.62	kd	CGS001-5211	PFKL	-			
6169	-85.64	cp	BRD-K76775527	nimesulide	Cyclooxygenase inhibitor		PTGS2, LTF, PLA2G2E, PTGS1	Cyclooxygenase inhibitor
6170	-85.64	kd	CGS001-4143	MAT1A	-			
6171	-85.68	kd	CGS001-5562	PRKAA1	AMPK subfamily			
6172	-85.68	kd	CGS001-929	CD14	CD molecules			
6173	-85.7	cp	BRD-K66206289	lobeline	Acetylcholine receptor antagonist		SLC18A2, CHRNA10, CHRNA4, CHRNA9, CHRNB2, OPRM1	Acetylcholine receptor antagonist
6174	-85.71	cp	BRD-A94709349	metaxalone	Muscle relaxant			Muscle relaxant
6175	-85.71	kd	CGS001-10914	PAPOLA	-			
6176	-85.73	oe	ccsbBroad304_00270	CDK1	Cyclin-dependent kinases, CDK1 subfamily			
6177	-85.77	cp	BRD-K29582677	flunarizine	Calcium channel blocker		CACNA1G, CACNA1H, CACNA1I, CALM1, CYP2J2, HRH1	Calcium channel blocker
6178	-85.8	kd	CGS001-2064	ERBB2	Type I RTKs: ErbB (epidermal growth factor) receptor family			
6179	-85.83	cp	BRD-K46469693	SCH-442416	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
6180	-85.88	cc		Purinergic receptors P2Y GOF	-			
6181	-85.89	cp	BRD-K63630713	etacrynic-acid	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, SLC12A2	Sodium/potassium/chloride transporter inhibitor
6182	-85.99	oe	ccsbBroad304_09446	MRGPRX4	GPCR / Class A : Orphans			
6183	-86	kd	CGS001-4233	MET	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
6184	-86.04	oe	ccsbBroad304_07362	NMI	-			
6185	-86.05	cp	BRD-K14618467	IKK-16	IKK inhibitor		IKBKB	IKK inhibitor
6186	-86.06	cp	BRD-K64451768	GANT-58	GLI antagonist		DHH, GLI1, IHH	GLI antagonist
6187	-86.07	cp	BRD-K51677086	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
6188	-86.08	oe	ccsbBroad304_03510	FKBP14	EF-hand domain containing			
6189	-86.08	kd	CGS001-5292	PIM1	PIM family			
6190	-86.09	oe	ccsbBroad304_08461	CDCA4	-			
6191	-86.09	kd	CGS001-586	BCAT1	-			
6192	-86.15	cp	BRD-K77947974	fluspirilene	Dopamine receptor antagonist		DRD2, HTR2A, CACNG1, HRH1, HTR1A, HTR1D, HTR1E	Dopamine receptor antagonist
6193	-86.16	kd	CGS001-9971	NR1H4	Liver X receptor-like receptors			
6194	-86.24	oe	ccsbBroad304_08878	METTL4	-			
6195	-86.25	cp	BRD-K34330170	rotenonic-acid	Retinoid receptor antagonist			Retinoid receptor antagonist
6196	-86.31	cp	BRD-K60174629	z-prolyl-prolinal	Prolyl endopeptidase inhibitor		PREP	Prolyl endopeptidase inhibitor
6197	-86.34	cp	BRD-A09094913	strychnine	Acetylcholine receptor antagonist		GLRA1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CHRNA10, CHRNA9, GLRA2, GLRA3, GLRB	Acetylcholine receptor antagonist
6198	-86.35	kd	CGS001-6416	MAP2K4	MAPKK:STE7 family			
6199	-86.4	cp	BRD-K10177585	PSB-11	Adenosine receptor antagonist		ADORA3, ADORA1, ADORA2A	Adenosine receptor antagonist
6200	-86.4	cp	BRD-K40992116	parachlorophenol	Anti-infective			Anti-infective
6201	-86.47	oe	ccsbBroad304_03040	NKIRAS2	-			
6202	-86.5	cp	BRD-K52989797	clomipramine	Serotonin transporter inhibitor (SERT)		SLC6A4, SLC6A2, CYP2C19, GSTP1, HTR2A, HTR2B, HTR2C, SLC6A3	Serotonin transporter inhibitor (SERT)
6203	-86.55	kd	CGS001-10775	POP4	-			
6204	-86.56	kd	CGS001-826	CAPNS1	EF-hand domain containing			
6205	-86.67	cp	BRD-K04210847	tamoxifen	Estrogen receptor antagonist		ESR1, ESR2, CYP3A5, EBP, GPER1, PRKCA, PRKCB, PRKCD, PRKCE, PRKCG, PRKCI, PRKCQ, PRKCZ	Estrogen receptor antagonist, Selective estrogen receptor modulator (SERM)
6206	-86.67	kd	CGS001-2266	FGG	Endogenous ligands			
6207	-86.68	kd	CGS001-5230	PGK1	-			
6208	-86.71	oe	ccsbBroad304_04909	ZNF572	Zinc fingers, C2H2-type			
6209	-86.72	cp	BRD-K13356952	methazolamide	Carbonic anhydrase inhibitor		CA1, CA2, CA4, CA7, CA12, CA14, INS	Carbonic anhydrase inhibitor
6210	-86.75	kd	CGS001-6259	RYK	Type XV RTKs: RYK			
6211	-86.78	oe	ccsbBroad304_10507	SNX7	Sorting nexins			
6212	-86.82	cp	BRD-U68942961	JW-7-24-1	LCK Inhibitor		LCK	LCK Inhibitor
6213	-86.83	cp	BRD-A81402010	KU-C103443N	CDC inhibitor			CDC inhibitor, Rho associated kinase inhibitor
6214	-86.84	cp	BRD-K33572481	taurodeoxycholic-acid	Bile acid			Bile acid
6215	-86.85	kd	CGS001-83737	ITCH	-			
6216	-86.86	oe	ccsbBroad304_00769	HOXA1	Homeoboxes / ANTP class : HOXL subclass			
6217	-86.88	kd	CGS001-3226	HOXC10	Homeoboxes / ANTP class : HOXL subclass			
6218	-86.9	kd	CGS001-23770	FKBP8	Tetratricopeptide (TTC) repeat domain containing			
6219	-86.91	kd	CGS001-9326	ZNHIT3	Zinc fingers, HIT-type			
6220	-86.94	kd	CGS001-10001	MED6	-			
6221	-86.94	kd	CGS001-3689	ITGB2	Integrins			
6222	-87	cp	BRD-A31159102	fluoxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, ANO1, CYP2C19, HTR2B	Selective serotonin reuptake inhibitor (SSRI)
6223	-87	cp	BRD-K06980535	promazine	Dopamine receptor antagonist		CHRM5, DRD2, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, CHRM4, DRD1, DRD3, DRD4, HRH1, HTR2A, HTR2C	Dopamine receptor antagonist
6224	-87.04	kd	CGS001-9568	GABBR2	GABA receptors			
6225	-87.1	cp	BRD-K66956375	oleoylethanolamide	Cannabinoid receptor agonist		CNR1, GPR119, GPR55, KCND3, PPARA	Cannabinoid receptor agonist, Glucose dependent insulinotropic receptor agonist, Potassium channel blocker, PPAR receptor agonist
6226	-87.12	cp	BRD-K60923938	veratridine	Sodium channel activator		SCN1A, SCN3A, SCN8A, SCN9A	Sodium channel activator
6227	-87.13	oe	ccsbBroad304_06088	AKR1C1	Aldo-keto reductases			
6228	-87.15	cp	BRD-K77286328	reversine	Aurora kinase inhibitor		AURKB, ADORA3, AURKA, INCENP, MAP2K1	Aurora kinase inhibitor
6229	-87.2	cp	BRD-K20755323	SA-792728	Sphingosine kinase inhibitor		SPHK1, VCP	Sphingosine kinase inhibitor
6230	-87.22	kd	CGS001-217	ALDH2	Aldehyde dehydrogenases			
6231	-87.24	kd	CGS001-10797	MTHFD2	-			
6232	-87.25	oe	ccsbBroad304_07017	SUOX	-			
6233	-87.27	kd	CGS001-1455	CSNK1G2	Casein kinase 1 (CK1) family			
6234	-87.27	kd	CGS001-167826	OLIG3	Basic helix-loop-helix proteins			
6235	-87.35	kd	CGS001-6647	SOD1	-			
6236	-87.36	cp	BRD-K43149758	myricetin	Androgen receptor agonist		PIK3CG, AR, CYP3A4	Androgen receptor agonist, Cytochrome P450 inhibitor
6237	-87.36	cp	BRD-K50417881	eticlopride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
6238	-87.36	cp	BRD-K98521173	desoxycortone	Mineralocorticoid receptor agonist		NR3C1, NR3C2	Mineralocorticoid receptor agonist
6239	-87.39	kd	CGS001-5714	PSMD8	Proteasome (prosome, macropain) subunits			
6240	-87.4	kd	CGS001-25824	PRDX5	-			
6241	-87.4	kd	CGS001-87	ACTN1	EF-hand domain containing			
6242	-87.48	oe	ccsbBroad304_10758	CTBP2	-			
6243	-87.48	cp	BRD-K75532464	FTI-276	Farnesyltransferase inhibitor		FNTA, FNTB	Farnesyltransferase inhibitor
6244	-87.5	cp	BRD-K77987382	mebendazole	Tubulin inhibitor		TUBA1A, TUBB, TUBB4B	Tubulin inhibitor
6245	-87.51	kd	CGS001-23102	TBC1D2B	-			
6246	-87.52	kd	CGS001-4000	LMNA	Intermediate filaments type V, lamins			
6247	-87.52	kd	CGS001-8678	BECN1	-			
6248	-87.53	oe	ccsbBroad304_01128	OTX2	Homeoboxes / PRD class			
6249	-87.53	kd	CGS001-7296	TXNRD1	-			
6250	-87.56	cp	BRD-K46137903	prednicarbate	Phospholipase activator		NR3C1, PLA2G1B	Phospholipase activator
6251	-87.58	oe	ccsbBroad304_02843	FTSJ1	-			
6252	-87.59	cp	BRD-A53576514	orphenadrine	Acetylcholine receptor antagonist		CYP2B6, GRIN1, GRIN2D, GRIN3A, GRIN3B, HRH1, SCN10A, SLC6A2	Acetylcholine receptor antagonist
6253	-87.59	kd	CGS001-10955	SERINC3	-			
6254	-87.59	cp	BRD-K10995081	perphenazine	Dopamine receptor antagonist		DRD2, CALM1, DRD1, HRH1, HTR2A, HTR2C, HTR6, HTR7	Dopamine receptor antagonist
6255	-87.61	oe	ccsbBroad304_00348	MAP3K8	MAPKKK:STE-unique family			
6256	-87.62	kd	CGS001-2194	FASN	Short chain dehydrogenase/reductase superfamily / Atypical members			
6257	-87.75	cp	BRD-A29901043	KIN001-127	ITK inhibitor		ITK	ITK inhibitor
6258	-87.78	kd	CGS001-1456	CSNK1G3	Casein kinase 1 (CK1) family			
6259	-87.82	kd	CGS001-2534	FYN	Src family			
6260	-87.83	kd	CGS001-23499	MACF1	EF-hand domain containing			
6261	-87.85	kd	CGS001-54659	UGT1A3	UDP glucuronosyltransferases			
6262	-87.95	oe	ccsbBroad304_13848	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
6263	-87.95	kd	CGS001-2237	FEN1	-			
6264	-87.97	kd	CGS001-5164	PDK2	PDHK family			
6265	-88	kd	CGS001-5646	PRSS3	Serine peptidases / Serine peptidases			
6266	-88.03	cp	BRD-A19661776	mianserin	Serotonin receptor antagonist		HTR2A, HTR2C, ADRA1A, ADRA1B, ADRA1D, HRH1, HTR2B, HTR6, HTR7, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD2, DRD3, DRD5, HRH2, HRH4, HTR1A, HTR1F, OPRK1, SLC6A2, SLC6A3, SLC6A4	Serotonin receptor antagonist
6267	-88.03	kd	CGS001-2048	EPHB2	Type XIII RTKs: Ephrin receptor family			
6268	-88.04	cp	BRD-A99411506	esculin	Antioxidant			Antioxidant
6269	-88.06	cp	BRD-A14966924	alaproclate	Serotonin receptor antagonist		SLC6A4	Serotonin receptor antagonist
6270	-88.19	oe	ccsbBroad304_00784	HRAS	RAS subfamily			
6271	-88.19	cp	BRD-K17140735	SCH-79797	Proteasome inhibitor		F2R	Proteasome inhibitor
6272	-88.2	kd	CGS001-3199	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
6273	-88.25	cc		Thymidylate synthase inhibitor	-			
6274	-88.26	oe	ccsbBroad304_03732	NPDC1	-			
6275	-88.3	oe	ccsbBroad304_01797	ZNF32	Zinc fingers, C2H2-type			
6276	-88.32	cp	BRD-A46186775	hydrocortisone	Glucocorticoid receptor agonist		ANXA1, NOS2, NR3C1, NR3C2	Glucocorticoid receptor agonist
6277	-88.33	oe	ccsbBroad304_00819	IDH3B	-			
6278	-88.36	kd	CGS001-84365	MKI67IP	-			
6279	-88.37	kd	CGS001-10769	PLK2	Polo-like kinase (PLK) family			
6280	-88.38	kd	CGS001-9774	BCLAF1	-			
6281	-88.42	cp	BRD-A10969569	ambelline	Plant alkaloid			Plant alkaloid
6282	-88.44	kd	CGS001-10450	PPIE	RNA binding motif (RRM) containing			
6283	-88.47	kd	CGS001-7272	TTK	TTK family			
6284	-88.54	oe	ccsbBroad304_05425	SNAI3	Snail homologs			
6285	-88.54	cp	BRD-K24675965	LY-288513	CCK receptor antagonist		CCKBR	CCK receptor antagonist
6286	-88.59	kd	CGS001-8764	TNFRSF14	Tumour necrosis factor (TNF) receptor family			
6287	-88.59	kd	CGS001-5037	PEBP1	-			
6288	-88.63	oe	ccsbBroad304_03177	FIS1	-			
6289	-88.66	oe	ccsbBroad304_00899	KCNK2	Two-P potassium channels			
6290	-88.67	cp	BRD-A95096829	PNU-96415E	Dopamine receptor antagonist			Dopamine receptor antagonist
6291	-88.8	oe	ccsbBroad304_07337	TAF1B	-			
6292	-88.82	oe	ccsbBroad304_00860	IL13	Interleukins and interleukin receptors			
6293	-88.82	cp	BRD-K73824630	skatole	Thrombin inhibitor		F2	Thrombin inhibitor
6294	-88.87	oe	ccsbBroad304_06995	SREBF1	Basic helix-loop-helix proteins			
6295	-88.89	oe	ccsbBroad304_06144	EFNB3	Ephrins			
6296	-88.9	oe	ccsbBroad304_02875	BRP44	-			
6297	-88.91	kd	CGS001-83637	ZMIZ2	Zinc fingers, MIZ-type			
6298	-88.91	kd	CGS001-84923	FAM104A	-			
6299	-88.94	cp	BRD-K10870738	CDC	Lipoxygenase inhibitor		ALOX12, ALOX5	Lipoxygenase inhibitor
6300	-89.04	cp	BRD-K63675182	triflupromazine	Dopamine receptor antagonist		HTR2B, CHRM1, CHRM2, CHRNA7, DRD1, DRD2	Dopamine receptor antagonist
6301	-89.06	cp	BRD-K54708045	nTZDpa	PPAR receptor agonist		PPARG	PPAR receptor agonist
6302	-89.13	kd	CGS001-57048	PLSCR3	-			
6303	-89.22	kd	CGS001-3251	HPRT1	-			
6304	-89.25	oe	ccsbBroad304_06908	S100B	EF-hand domain containing			
6305	-89.26	oe	ccsbBroad304_01789	SF1	Zinc fingers, CCHC domain containing			
6306	-89.28	cp	BRD-K11911061	GR-127935	Serotonin receptor antagonist		HTR1B, HTR1D, HTR1A, HTR2A, HTR2C, HTR1E, HTR1F, HTR2B, HTR6	Serotonin receptor antagonist
6307	-89.31	oe	ccsbBroad304_01889	FZD4	GPCR / Class F : Frizzled receptors			
6308	-89.33	cp	BRD-K37080523	isoreserpine	Vesicular monoamine transporter inhibitor		SLC18A2, SLC18A1, SIAH1	Vesicular monoamine transporter inhibitor
6309	-89.35	cp	BRD-K09537769	NU-7026	DNA dependent protein kinase inhibitor		PRKDC	DNA dependent protein kinase inhibitor, MTOR inhibitor, PI3K inhibitor
6310	-89.36	cp	BRD-K97564742	mepyramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
6311	-89.4	oe	ccsbBroad304_01094	NFKBIB	Ankyrin repeat domain containing			
6312	-89.42	kd	CGS001-221188	GPR114	Adhesion Class GPCRs			
6313	-89.44	oe	ccsbBroad304_09344	ZNF764	Zinc fingers, C2H2-type			
6314	-89.45	oe	ccsbBroad304_07131	VRK1	Vaccina related kinase (VRK) family			
6315	-89.47	cc		Kruppel like transcription factors LOF	-			
6316	-89.48	cp	BRD-A94669766	naringenin	Aromatase inhibitor		CYP19A1, ESR2, CYP1B1, GLO1, HSD17B1	Aromatase inhibitor, TRPV antagonist
6317	-89.5	cp	BRD-K26664453	cytochalasin-b	Microtubule inhibitor		ACTB	Microtubule inhibitor
6318	-89.52	cp	BRD-K33551950	radicicol	HSP inhibitor		ACLY, DLAT, HSP90AB1, HSP90B1, MAP3K7, OPRM1, PDK3	HSP inhibitor
6319	-89.52	cp	BRD-K82577285	dipropyl-dopamine	Dopamine receptor agonist			Dopamine receptor agonist
6320	-89.54	kd	CGS001-2494	NR5A2	Fushi tarazu F1-like receptors			
6321	-89.55	cp	BRD-K68756823	FR-180204	-666		MAPK1, MAPK3	-666
6322	-89.55	cp	BRD-A39230911	chlorphensin	Muscle relaxant			Muscle relaxant
6323	-89.55	cp	BRD-A35511923	L-803087	Somatostatin receptor agonist		SSTR4	Somatostatin receptor agonist
6324	-89.6	kd	CGS001-1591	CYP24A1	Cytochrome P450s			
6325	-89.63	cp	BRD-K23583188	lavendustin-a	EGFR inhibitor		EGFR, LCK	EGFR inhibitor
6326	-89.68	cp	BRD-A43849199	karakoline	Phytotoxin			Phytotoxin
6327	-89.72	oe	ccsbBroad304_02285	MED6	-			
6328	-89.72	kd	CGS001-4507	MTAP	-			
6329	-89.74	kd	CGS001-302	ANXA2	Annexins			
6330	-89.75	kd	CGS001-375133	PI4KAP2	-			
6331	-89.76	kd	CGS001-29763	PACSIN3	-			
6332	-89.78	oe	ccsbBroad304_00756	HMGCS2	Lanosterol biosynthesis pathway			
6333	-89.79	cp	BRD-A27143604	DPN	Estrogen receptor agonist		ESR2	Estrogen receptor agonist
6334	-89.79	kd	CGS001-5564	PRKAB1	AMPK subfamily			
6335	-89.84	kd	CGS001-51056	LAP3	Leucyl aminopeptidase			
6336	-89.85	cp	BRD-K84566043	fenpiverinium	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
6337	-89.86	cp	BRD-U37049823	HG-6-64-01	RAF inhibitor		ABL1, BRAF, CSF1R, EGFR, FGFR1, FLT3, KIT, MAPK11, PDGFRB, RET	RAF inhibitor
6338	-89.88	cp	BRD-K79425933	benperidol	Dopamine receptor antagonist		DRD2	Dopamine receptor antagonist
6339	-89.92	oe	ccsbBroad304_01269	PPP3R2	EF-hand domain containing			
6340	-89.96	oe	ccsbBroad304_01966	RUVBL1	ATPases / AAA-type			
6341	-89.99	cp	BRD-A72711497	lasalocid	Bacterial permeability inducer			Bacterial permeability inducer
6342	-90.01	kd	CGS001-5335	PLCG1	Phosphoinositide-specific phospholipase C			
6343	-90.05	cp	BRD-K38477985	malonoben	Protein tyrosine kinase inhibitor		EGFR	Protein tyrosine kinase inhibitor
6344	-90.07	cp	BRD-A50684349	fenoldopam	Dopamine receptor agonist		DRD1, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, DRD4, DRD5	Dopamine receptor agonist
6345	-90.08	cp	BRD-K87919739	tyrphostin-AG-825	Receptor tyrosine protein kinase inhibitor		ERBB2	Receptor tyrosine protein kinase inhibitor
6346	-90.09	oe	ccsbBroad304_07764	SLC2A6	Solute carriers			
6347	-90.15	cp	BRD-K39670393	amthamine	Histamine receptor agonist		HRH2	Histamine receptor agonist
6348	-90.22	kd	CGS001-2752	GLUL	-			
6349	-90.22	kd	CGS001-25861	DFNB31	-			
6350	-90.23	kd	CGS001-1312	COMT	Catecholamine turnover			
6351	-90.25	cp	BRD-K99447003	enalaprilat	ACE inhibitor		ACE	ACE inhibitor
6352	-90.29	cp	BRD-K19462402	buflomedil	Adrenergic receptor antagonist		CACNA1C	Adrenergic receptor antagonist, Calcium channel blocker
6353	-90.32	cp	BRD-K71266197	PSB-06126	NTPDase inhibitor		ENTPD3	NTPDase inhibitor
6354	-90.33	kd	CGS001-26996	GPR160	GPCR / Class A : Orphans			
6355	-90.36	cp	BRD-K62929068	6-benzylaminopurine	Purinergic receptor activator			Purinergic receptor activator
6356	-90.43	kd	CGS001-6421	SFPQ	RNA binding motif (RRM) containing			
6357	-90.44	cp	BRD-K29950728	clomifene	Estrogen receptor antagonist		ESR1, AR	Estrogen receptor antagonist
6358	-90.48	cp	BRD-K46056750	AZD-7762	CHK inhibitor		CHEK1, CHEK2	CHK inhibitor
6359	-90.49	kd	CGS001-64376	IKZF5	IKAROS zinc fingers			
6360	-90.54	cp	BRD-A92585442	RU-28318	Cytochrome P450 inhibitor		NR3C2	Cytochrome P450 inhibitor
6361	-90.55	kd	CGS001-23139	MAST2	MAST family			
6362	-90.57	cp	BRD-K62056274	quipazine	Serotonin receptor agonist		HTR2A, HTR3A, HTR3B, HTR1A, HTR1D, HTR2B, HTR2C, HTR6, SLC6A4	Serotonin receptor agonist
6363	-90.58	oe	ccsbBroad304_08825	LHPP	-			
6364	-90.59	kd	CGS001-1460	CSNK2B	Casein kinase 2 (CK2) family			
6365	-90.6	kd	CGS001-6392	SDHD	Mitochondrial respiratory chain complex / Complex II			
6366	-90.6	kd	CGS001-5422	POLA1	DNA polymerases			
6367	-90.65	cp	BRD-K80451230	zamifenacin	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
6368	-90.65	cp	BRD-A39969961	eplerenone	Cytochrome P450 inhibitor		NR3C2, CYP3A5	Cytochrome P450 inhibitor
6369	-90.66	cp	BRD-K19540840	saracatinib	SRC inhibitor		SRC, ABL1, LCK, YES1	SRC inhibitor
6370	-90.68	kd	CGS001-3845	KRAS	RAS subfamily			
6371	-90.7	cp	BRD-K41567364	SB-334867	Orexin receptor antagonist		HCRTR1, HCRTR2	Orexin receptor antagonist
6372	-90.74	kd	CGS001-9589	WTAP	-			
6373	-90.83	kd	CGS001-5721	PSME2	Proteasome (prosome, macropain) subunits			
6374	-90.86	cp	BRD-K05737787	isoeugenol	Nitric oxide production inhibitor			Nitric oxide production inhibitor
6375	-90.9	cp	BRD-K33308633	INCA-6	Calcineurin inhibitor		NFATC1	Calcineurin inhibitor
6376	-90.96	kd	CGS001-3596	IL13	Interleukins and interleukin receptors			
6377	-90.98	oe	ccsbBroad304_02092	SYNGR3	-			
6378	-91	kd	CGS001-3249	HPN	Serine peptidases / Transmembrane			
6379	-91.03	cp	BRD-K63265447	docetaxel	Tubulin inhibitor		TUBB, BCL2, MAP2, MAP4, MAPT, NR1I2, TUBB1	Tubulin inhibitor
6380	-91.12	kd	CGS001-285220	EPHA6	Type XIII RTKs: Ephrin receptor family			
6381	-91.13	cc		Dopamine receptor antagonist	-			
6382	-91.14	cc		RAF inhibitor	-			
6383	-91.14	kd	CGS001-9638	FEZ1	-			
6384	-91.22	kd	CGS001-5819	PVRL2	Immunoglobulin superfamily / C2-set domain containing			
6385	-91.27	cp	BRD-A10070317	propranolol	Adrenergic receptor antagonist		ADRB2, ADRB3, ADRB1, CYP2C19, HTR1A, HTR1B	Adrenergic receptor antagonist
6386	-91.28	kd	CGS001-4522	MTHFD1	-			
6387	-91.31	cp	BRD-K92758126	gibberellic-acid	NFkB pathway inhibitor		AADACL2	NFkB pathway inhibitor
6388	-91.32	kd	CGS001-8548	BLZF1	-			
6389	-91.37	cp	BRD-A22707317	SB-205384	GABA receptor modulator		GABRA3, GABRA5, GABRA6	GABA receptor modulator
6390	-91.39	cp	BRD-K95992530	Cyclo-[Arg-Gly-Asp-D-Phe-Val]	integrin antagonist		ITGAV, ITGB3	integrin antagonist
6391	-91.46	cp	BRD-K84595254	strophanthidin	ATPase inhibitor		ATP1A1, ATP1A2, ATP1A3, ATP1A4, ATP1B1, ATP1B2, ATP1B3, ATP1B4, FXYD2	ATPase inhibitor
6392	-91.47	cp	BRD-K83636919	entacapone	Catechol O methyltransferase inhibitor		COMT	Catechol O methyltransferase inhibitor
6393	-91.49	cp	BRD-K52172416	anastrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
6394	-91.49	cp	BRD-K60274257	dephostatin	Tyrosine phosphatase inhibitor		PTPN1, PTPN6	Tyrosine phosphatase inhibitor
6395	-91.49	cp	BRD-K12906962	dichlorobenzamil	Sodium/calcium exchange inhibitor			Sodium/calcium exchange inhibitor
6396	-91.53	kd	CGS001-183	AGT	Endogenous ligands			
6397	-91.54	kd	CGS001-83440	ADPGK	-			
6398	-91.58	cp	BRD-K62221994	T-98475	Gonadotropin releasing factor hormone receptor antagonist		GNRH1, GNRHR	Gonadotropin releasing factor hormone receptor antagonist
6399	-91.59	kd	CGS001-7128	TNFAIP3	OTU domain containing			
6400	-91.6	kd	CGS001-23408	SIRT5	Histone deacetylases			
6401	-91.6	cp	BRD-K26818574	BIX-01294	Histone lysine methyltransferase inhibitor		EHMT1, EHMT2	Histone lysine methyltransferase inhibitor, DNA methyltransferase inhibitor
6402	-91.62	kd	CGS001-1975	EIF4B	RNA binding motif (RRM) containing			
6403	-91.63	kd	CGS001-6675	UAP1	-			
6404	-91.65	cp	BRD-K40255344	tyrphostin-A9	Protein tyrosine kinase inhibitor			Protein tyrosine kinase inhibitor, Tyrosine kinase inhibitor
6405	-91.65	kd	CGS001-2625	GATA3	GATA zinc finger domain containing			
6406	-91.65	kd	CGS001-4486	MST1R	Type X RTKs: HGF (hepatocyte growth factor) receptor family			
6407	-91.67	cp	BRD-K73589401	corticosterone	mineralocorticoid receptor agonist		HSD11B1, NR3C2, NCOA1	mineralocorticoid receptor agonist
6408	-91.67	cp	BRD-K93441486	diphemanil	Acetylcholine receptor antagonist		CHRM3	Acetylcholine receptor antagonist
6409	-91.69	cp	BRD-K28296557	AKT-inhibitor-IV	AKT inhibitor		AKT1	AKT inhibitor
6410	-91.69	kd	CGS001-5663	PSEN1	Presenilin			
6411	-91.7	kd	CGS001-10165	SLC25A13	Mitochondrial amino acid transporter subfamily			
6412	-91.71	kd	CGS001-2056	EPO	Endogenous ligands			
6413	-91.71	kd	CGS001-645	BLVRB	Short chain dehydrogenase/reductase superfamily / Atypical members			
6414	-91.74	cp	BRD-K76534306	enrofloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6415	-91.75	kd	CGS001-27199	OXGR1	GPCR / Class A : Orphans, Oxoglutarate receptor			
6416	-91.75	kd	CGS001-55897	MESP1	Basic helix-loop-helix proteins			
6417	-91.78	oe	ccsbBroad304_02447	ATP5H	ATPases / F-type			
6418	-91.78	cp	BRD-A24817035	laudanosine	Central nervous system agent			Central nervous system agent
6419	-91.78	cp	BRD-K88868628	iodoacetic-acid	Cysteine peptidase inhibitor			Cysteine peptidase inhibitor
6420	-91.83	oe	ccsbBroad304_07861	COBL	-			
6421	-91.84	cp	BRD-K28936863	ketotifen	Histamine receptor agonist		HRH1, PDE4A, PDE4B, PDE4C, PDE4D, PDE7A, PDE7B, PDE8A, PDE8B, PGD	Histamine receptor agonist, Histamine receptor ligand, Leukotriene receptor antagonist, Phosphodiesterase inhibitor
6422	-91.89	cp	BRD-K75641298	metoclopramide	Dopamine receptor antagonist		DRD2, HTR3A, HTR4, CHRM1, HTR3B	Dopamine receptor antagonist, Serotonin receptor antagonist
6423	-91.9	cp	BRD-A97437073	rosiglitazone	Insulin sensitizer		PPARG, ACSL4, CYP2C8, FFAR1, INS, TRPC5, TRPM3	Insulin sensitizer, PPAR receptor agonist
6424	-91.92	cp	BRD-K58299615	RO-90-7501	Beta amyloid inhibitor		APP	Beta amyloid inhibitor
6425	-91.94	cc		Adenosine receptor agonist	-			
6426	-91.96	cp	BRD-A32164164	methyllycaconitine	Acetylcholine receptor antagonist		CHRNA7	Acetylcholine receptor antagonist
6427	-91.97	cp	BRD-K09499853	KU-0060648	DNA dependent protein kinase inhibitor		PIK3CA, PIK3CB, PIK3CD, PIK3CG, PRKDC	DNA dependent protein kinase inhibitor, PI3K inhibitor
6428	-92.01	kd	CGS001-1719	DHFR	Oxidoreductases			
6429	-92.04	cc		Na-K-Cl transporter inhibitor	-			
6430	-92.05	oe	ccsbBroad304_07018	SUPT5H	-			
6431	-92.05	oe	ccsbBroad304_06852	RBP4	Lipocalins			
6432	-92.11	cp	BRD-K17823458	danoprevir	HCV inhibitor			HCV inhibitor
6433	-92.13	oe	ccsbBroad304_03618	OSGEP	-			
6434	-92.14	cp	BRD-K16508793	diazepam	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, ADRA1A, CYP2C19, GABRA4, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GABRR1, GABRR2, GABRR3, TSPO	Benzodiazepine receptor agonist
6435	-92.17	kd	CGS001-2810	SFN	-			
6436	-92.21	kd	CGS001-10078	TSSC4	-			
6437	-92.24	cp	BRD-K66788707	fludarabine	DNA synthesis inhibitor		ADA, DCK, POLA1, RRM1, RRM2	DNA synthesis inhibitor, DNA repair enzyme inhibitor, Purine antagonist
6438	-92.24	cp	BRD-A22143024	estropipate	Estrogen receptor agonist		ESR1, ESR2	Estrogen receptor agonist
6439	-92.24	kd	CGS001-1635	DCTD	-			
6440	-92.28	cp	BRD-A41519720	ezetimibe	Niemann-Pick C1-like 1 protein antagonist		NPC1L1, ANPEP, SOAT1	Niemann-Pick C1-like 1 protein antagonist, Cholesterol inhibitor
6441	-92.3	cp	BRD-K13261168	LY-16350	Dopamine receptor agonist		DRD2, DRD3	Dopamine receptor agonist
6442	-92.31	cp	BRD-K06426971	ryuvidine	Histone lysine methyltransferase inhibitor		CDK4, CDK2	Histone lysine methyltransferase inhibitor
6443	-92.32	cp	BRD-K25186396	tangeritin	Cell cycle inhibitor			Cell cycle inhibitor
6444	-92.32	kd	CGS001-1633	DCK	-			
6445	-92.33	oe	ccsbBroad304_05439	O3FAR1	-			
6446	-92.35	cp	BRD-A74980173	gatifloxacin	Bacterial DNA gyrase inhibitor			Bacterial DNA gyrase inhibitor
6447	-92.42	kd	CGS001-9467	SH3BP5	-			
6448	-92.43	cp	BRD-A09828896	SKF-81297	Dopamine receptor agonist		DRD1, DRD5	Dopamine receptor agonist
6449	-92.43	cp	BRD-K36862742	hydroflumethiazide	Sodium/potassium/chloride transporter inhibitor		SLC12A1, ATP1A1, CA1, CA12, CA2, CA4, CA9, KCNMA1	Sodium/potassium/chloride transporter inhibitor
6450	-92.45	oe	ccsbBroad304_00902	KCNN4	Calcium-activated potassium channels			
6451	-92.45	cp	BRD-K94832621	Y-134	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
6452	-92.48	kd	CGS001-10525	HYOU1	Heat shock proteins / HSP70			
6453	-92.5	oe	ccsbBroad304_00734	HDAC1	Histone deacetylases			
6454	-92.53	kd	CGS001-7832	BTG2	-			
6455	-92.54	cc		Estrogen receptor antagonist	-			
6456	-92.57	cp	BRD-K11853856	PJ-34	PARP inhibitor		EEF2, PARP1, PARP15, PARP3	PARP inhibitor
6457	-92.58	oe	ccsbBroad304_01480	S100P	EF-hand domain containing			
6458	-92.6	cp	BRD-A73909368	dactinomycin	RNA polymerase inhibitor		POLR2A	RNA polymerase inhibitor
6459	-92.62	cp	BRD-K81209159	herniarin	Acetylcholinesterase inhibitor		ACHE, CA1, CA12, CA14, CA4, CA6, CA9	Acetylcholinesterase inhibitor
6460	-92.64	oe	ccsbBroad304_14020	SH3BP5	-			
6461	-92.64	kd	CGS001-22978	NT5C2	Adenosine turnover			
6462	-92.65	kd	CGS001-29959	NRBP1	NRBP family			
6463	-92.71	kd	CGS001-3716	JAK1	Janus kinase (JakA) family			
6464	-92.73	kd	CGS001-135	ADORA2A	GPCR / Class A : Adenosine receptors			
6465	-92.78	oe	ccsbBroad304_03387	NUDT9	Nudix motif containing			
6466	-92.79	kd	CGS001-7100	TLR5	Toll-like receptor family			
6467	-92.83	cp	BRD-A28856712	tetryzoline	Adrenergic receptor agonist			Adrenergic receptor agonist
6468	-92.86	oe	ccsbBroad304_06824	PVR	Immunoglobulin superfamily / C2-set domain containing			
6469	-92.88	oe	ccsbBroad304_06783	LGMN	Legumain			
6470	-92.9	kd	CGS001-5160	PDHA1	-			
6471	-92.92	kd	CGS001-6195	RPS6KA1	RSK subfamily			
6472	-92.93	cp	BRD-K50388907	fenofibrate	PPAR receptor agonist		PPARA, APOA1, CYP2C19, CYP2C8, MMP25	PPAR receptor agonist
6473	-92.93	cp	BRD-K51318897	fenbendazole	Tubulin inhibitor		CYP2C19, CYP2D6, CYP2J2, CYP3A4, TUBB	Tubulin inhibitor
6474	-92.93	cp	BRD-A41250306	cyclopenthiazide	Thiazide diuretic			Thiazide diuretic
6475	-92.93	kd	CGS001-23028	KDM1A	Histone demethylase			
6476	-92.94	kd	CGS001-6558	SLC12A2	SLC12 family of cation-coupled chloride transporters			
6477	-92.97	kd	CGS001-5947	RBP1	Fatty acid binding protein family			
6478	-92.98	kd	CGS001-5696	PSMB8	Proteasome (prosome, macropain) subunits			
6479	-93.03	cp	BRD-K94176593	TWS-119	Glycogen synthase kinase inhibitor		GSK3B, JUN, MYC	Glycogen synthase kinase inhibitor
6480	-93.03	cp	BRD-K35629949	SR-27897	CCK receptor antagonist		CCKAR	CCK receptor antagonist
6481	-93.03	kd	CGS001-1105	CHD1	-			
6482	-93.07	kd	CGS001-3705	ITPK1	-			
6483	-93.11	cp	BRD-A68723818	brompheniramine	Histamine receptor antagonist		HRH1, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5	Histamine receptor antagonist
6484	-93.26	cp	BRD-K26117720	gingerol	Nitric oxide synthase inhibitor			Nitric oxide synthase inhibitor
6485	-93.33	kd	CGS001-7264	TSTA3	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6486	-93.35	cc		Trace amine receptors LOF	-			
6487	-93.41	oe	ccsbBroad304_03772	CCNL1	-			
6488	-93.45	oe	ccsbBroad304_02621	PRDM7	Zinc fingers, C2H2-type			
6489	-93.45	kd	CGS001-63929	XPNPEP3	Methionyl aminopeptidase			
6490	-93.45	oe	ccsbBroad304_02019	IL18RAP	CD molecules			
6491	-93.47	kd	CGS001-4439	MSH5	-			
6492	-93.48	cp	BRD-A84389633	tropanyl-3,5-dimethylbenzoate	Serotonin receptor antagonist			Serotonin receptor antagonist
6493	-93.49	oe	ccsbBroad304_07565	RBM6	G patch domain containing			
6494	-93.52	cp	BRD-K39823328	VU-0366037-2	Glutamate receptor modulator		GRM4	Glutamate receptor modulator
6495	-93.57	cp	BRD-K50836978	purvalanol-a	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CSNK1G3, RPS6KA1, SRC	CDK inhibitor, DYRK inhibitor
6496	-93.59	cc		JAK inhibitor	-			
6497	-93.59	kd	CGS001-8428	STK24	YSK subfamily			
6498	-93.61	cc		PDGFR/KIT inhibitor	-			
6499	-93.61	kd	CGS001-1123	CHN1	Rho GTPase activating proteins			
6500	-93.62	oe	ccsbBroad304_06398	HPN	Serine peptidases / Transmembrane			
6501	-93.69	oe	ccsbBroad304_06609	MYL6	EF-hand domain containing			
6502	-93.69	cp	BRD-A64297288	amlodipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, ABCG2, CA1, CACNA1B, CACNA1S, CACNA2D3, CACNB1, CACNB2, SMPD1	Calcium channel blocker
6503	-93.71	kd	CGS001-79885	HDAC11	Histone deacetylases			
6504	-93.72	oe	ccsbBroad304_02759	DICER1	-			
6505	-93.72	oe	ccsbBroad304_02128	GPR55	GPCR / Class A : Orphans			
6506	-93.72	cp	BRD-K17743697	KB-R7943	Sodium/calcium exchange inhibitor		SLC8A1, TRPC3, TRPC5, TRPC6	Sodium/calcium exchange inhibitor
6507	-93.72	cp	BRD-A13650332	flucloxacillin	Bacterial cell wall synthesis inhibitor			Bacterial cell wall synthesis inhibitor
6508	-93.72	kd	CGS001-3980	LIG3	-			
6509	-93.78	kd	CGS001-124626	ZPBP2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
6510	-93.83	cc		DNA dependent protein kinase inhibitor	-			
6511	-93.84	cp	BRD-A35912562	pregnenolone	Glutamate receptor modulator		CYP17A1, PGR, SULT2B1	Glutamate receptor modulator, Acetylcholine release enhancer, Dopamine release enhancer, GABA receptor negative allosteric modulator
6512	-93.87	cp	BRD-A28105619	cucurbitacin-i	JAK inhibitor		JAK2, STAT3	JAK inhibitor, Lipocortin synthesis stimulant, STAT inhibitor
6513	-93.87	kd	CGS001-55229	PANK4	-			
6514	-93.92	cp	BRD-K55344148	BU-224	Imidazoline receptor ligand		MAOA, MAOB	Imidazoline receptor ligand
6515	-93.92	kd	CGS001-64223	MLST8	WD repeat domain containing			
6516	-93.96	oe	ccsbBroad304_00762	FOXA3	Forkhead boxes			
6517	-93.96	cp	BRD-K88551539	CAY-10585	HIF modulator		HIF1A	HIF modulator
6518	-93.98	cp	BRD-A67748489	K3644	Kinesin-like spindle protein inhibitor		KIF11	Kinesin-like spindle protein inhibitor
6519	-93.99	oe	ccsbBroad304_00957	M6PR	-			
6520	-93.99	kd	CGS001-6897	TARS	Aminoacyl tRNA synthetases / Class II			
6521	-94.03	kd	CGS001-4552	MTRR	-			
6522	-94.06	kd	CGS001-79258	MMEL1	-			
6523	-94.08	cp	BRD-K37691127	hinokitiol	Tyrosinase inhibitor		TYR	Tyrosinase inhibitor
6524	-94.11	cp	BRD-K82688027	RG-13022	PDGFR receptor inhibitor		EGFR, PDGFRA, PDGFRB	PDGFR receptor inhibitor
6525	-94.11	kd	CGS001-5629	PROX1	Homeoboxes / PROS class			
6526	-94.12	kd	CGS001-4717	NDUFC1	Mitochondrial respiratory chain complex / Complex I			
6527	-94.13	oe	ccsbBroad304_02612	DUSP14	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
6528	-94.14	cp	BRD-A59174698	ritodrine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6529	-94.15	kd	CGS001-51330	TNFRSF12A	Tumour necrosis factor (TNF) receptor family			
6530	-94.19	kd	CGS001-10062	NR1H3	Liver X receptor-like receptors			
6531	-94.2	oe	ccsbBroad304_03097	CNOT7	-			
6532	-94.2	kd	CGS001-3590	IL11RA	IL-6 receptor family			
6533	-94.22	cp	BRD-K03406345	azacitidine	DNA methyltransferase inhibitor		DNMT1	DNA methyltransferase inhibitor
6534	-94.23	kd	CGS001-83550	GPR101	GPCR / Class A : Orphans			
6535	-94.24	oe	ccsbBroad304_02173	ATG5	-			
6536	-94.26	kd	CGS001-7314	UBB	-			
6537	-94.27	cp	BRD-A63546914	RO-04-5595	Glutamate receptor antagonist			Glutamate receptor antagonist
6538	-94.29	oe	ccsbBroad304_08849	ABCG8	ATP binding cassette transporters / subfamily G			
6539	-94.3	kd	CGS001-55256	ADI1	-			
6540	-94.31	kd	CGS001-50943	FOXP3	Forkhead boxes			
6541	-94.36	cp	BRD-K68202742	trichostatin-a	HDAC inhibitor		HDAC7, HDAC8, HDAC1, HDAC10, HDAC2, HDAC3, HDAC4, HDAC5, HDAC6, HDAC9	HDAC inhibitor, CDK activator, ID1 inhibitor
6542	-94.38	kd	CGS001-5937	RBMS1	RNA binding motif (RRM) containing			
6543	-94.42	cp	BRD-A89672324	CGP-55845	GABA receptor antagonist		GABBR1, GABBR2, KCTD12, KCTD16, KCTD8	GABA receptor antagonist
6544	-94.43	kd	CGS001-949	SCARB1	-			
6545	-94.44	cp	BRD-K29555132	arachidonamide	Cannabinoid receptor agonist		CNR1, CNR2	Cannabinoid receptor agonist
6546	-94.45	cp	BRD-A00758722	noretynodrel	Progestogen hormone		PGR	Progestogen hormone
6547	-94.46	cp	BRD-K15588452	R-96544	Serotonin receptor antagonist		HTR2A	Serotonin receptor antagonist
6548	-94.46	kd	CGS001-7803	PTP4A1	Protein tyrosine phosphatases / Class I Cys-based PTPs : PRLs			
6549	-94.47	kd	CGS001-10048	RANBP9	-			
6550	-94.48	cp	BRD-A10977446	carvedilol	Adrenergic receptor antagonist		ADRB1, ADRB2, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB3, CYP2C19, CYP2E1, GJA1, HIF1A, KCNH2, NDUFC2, NPPB, RYR2, SELE, VCAM1, VEGFA	Adrenergic receptor antagonist
6551	-94.5	cp	BRD-A13188892	doxazosin	Adrenergic receptor antagonist		ADRA1D, ADRA1A, ADRA1B, CYP2C19, KCNH2, KCNH6, KCNH7	Adrenergic receptor antagonist
6552	-94.52	cc		Interleukin receptors LOF	-			
6553	-94.53	oe	ccsbBroad304_00240	CCNH	General transcription factor IIH complex subunits			
6554	-94.53	cp	BRD-A72988804	tiaprofenic-acid	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
6555	-94.54	cp	BRD-K45296539	ZD-7114	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
6556	-94.55	kd	CGS001-51752	ERAP1	Aminopeptidase N			
6557	-94.56	cp	BRD-K54665485	R-59022	Diacylglycerol kinase inhibitor		DGKA	Diacylglycerol kinase inhibitor, Protein kinase inhibitor
6558	-94.56	kd	CGS001-5373	PMM2	-			
6559	-94.58	oe	ccsbBroad304_07328	PRPF4B	PRP4 subfamily			
6560	-94.59	kd	CGS001-10166	SLC25A15	Mitochondrial amino acid transporter subfamily			
6561	-94.6	kd	CGS001-50814	NSDHL	Short chain dehydrogenase/reductase superfamily / Extended SDR fold			
6562	-94.6	kd	CGS001-29940	DSE	-			
6563	-94.61	kd	CGS001-5347	PLK1	Polo-like kinase (PLK) family			
6564	-94.63	kd	CGS001-1622	DBI	-			
6565	-94.64	cp	BRD-K55468218	spiperone	Dopamine receptor antagonist		ADRA1A, DRD2, DRD3, DRD4, HTR1A, HTR2A, HTR7, ADRA1B, ADRA1D, DRD1, DRD5, HTR1D, HTR2B, HTR2C, HTR6	Dopamine receptor antagonist
6566	-94.64	kd	CGS001-91304	C19ORF6	-			
6567	-94.69	cp	BRD-A39747742	estradiol-valerate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6568	-94.69	kd	CGS001-64422	ATG3	-			
6569	-94.7	cp	BRD-K40902647	vincamine	Adrenergic receptor antagonist		CHRM1, CHRM2, CHRM3, CHRM4	Adrenergic receptor antagonist
6570	-94.71	oe	ccsbBroad304_00120	ATOX1	-			
6571	-94.74	cp	BRD-A18917088	estradiol	Contraceptive agent		ESR1, ESR2, NR1I2, CYP2B6, CYP2C19, CYP2C8, CYP2E1, CYP3A5, CYP3A7, GPER1, KCNMA1	Contraceptive agent, Estrogen receptor agonist
6572	-94.75	kd	CGS001-10451	VAV3	Rho guanine nucleotide exchange factors			
6573	-94.77	kd	CGS001-147837	ZNF563	Zinc fingers, C2H2-type			
6574	-94.8	cp	BRD-K07212038	selinidin	Mast cell stabilizer			Mast cell stabilizer
6575	-94.8	cp	BRD-K26521938	dinoprostone	Prostanoid receptor agonist		PTGER2, PTGER1, PTGER3, PTGER4, CATSPER1, CATSPER2, CATSPER3, CATSPER4, PTGDR, PTGDR2, PTGFR, TBXA2R	Prostanoid receptor agonist
6576	-94.81	cp	BRD-K05653692	DL-PDMP	Glucosyltransferase inhibitor		ASAH1, UGCG	Glucosyltransferase inhibitor
6577	-94.81	kd	CGS001-7862	BRPF1	Non-enzymatic BRD containing proteins			
6578	-94.83	cp	BRD-K19796430	erismodegib	Smoothened receptor antagonist		SMO	Smoothened receptor antagonist
6579	-94.83	kd	CGS001-51347	TAOK3	TAO subfamily			
6580	-94.84	oe	ccsbBroad304_01970	RFXANK	Ankyrin repeat domain containing			
6581	-94.86	kd	CGS001-57512	GPR158	GPCR / Class C : Orphans			
6582	-94.88	oe	ccsbBroad304_02168	GGPS1	Lanosterol biosynthesis pathway			
6583	-94.88	kd	CGS001-3265	HRAS	RAS subfamily			
6584	-94.88	cp	BRD-K71512533	SNS-314	Aurora kinase inhibitor		AURKA, AURKB, AURKC	Aurora kinase inhibitor
6585	-94.91	kd	CGS001-4087	SMAD2	SMADs			
6586	-94.93	cp	BRD-A69960130	bromocriptine	Dopamine receptor agonist		DRD2, ADRA2A, ADRA2B, ADRA2C, DRD1, DRD3, DRD4, DRD5, HTR1A, HTR1B, HTR1D, HTR2A, HTR2B, HTR2C, ADRA1A, ADRA1B, ADRA1D, HTR6, HTR7, PRL	Dopamine receptor agonist
6587	-94.95	cp	BRD-M86331534	pyrvinium-pamoate	AKT inhibitor		AR	AKT inhibitor
6588	-94.96	cp	BRD-K89839824	raltitrexed	Thymidylate synthase inhibitor		TYMS, FPGS	Thymidylate synthase inhibitor
6589	-94.98	oe	ccsbBroad304_00184	C2	Complement system			
6590	-94.98	kd	CGS001-10198	MPHOSPH9	-			
6591	-95.01	cp	BRD-K94689771	pinocembrin	CYP1B1 inhibitor		AR, CYP1B1, SRD5A1, SRD5A2	CYP1B1 inhibitor
6592	-95.05	kd	CGS001-6217	RPS16	S ribosomal proteins			
6593	-95.05	kd	CGS001-1429	CRYZ	-			
6594	-95.09	kd	CGS001-57018	CCNL1	-			
6595	-95.11	cp	BRD-K05104363	PD-184352	MEK inhibitor		MAP2K1, MAP2K2, MAP3K1, MAP3K2	MEK inhibitor
6596	-95.12	oe	ccsbBroad304_00009	ACLY	-			
6597	-95.14	kd	CGS001-2539	G6PD	-			
6598	-95.18	cp	BRD-K03816923	rottlerin	MAP kinase inhibitor		KCNH2, PRKCD, TGM2	MAP kinase inhibitor, Protein kinase inhibitor
6599	-95.18	cp	BRD-A95869247	indapamide	Thiazide diuretic		KCNQ1, CA7, KCNE1, SLC12A3	Thiazide diuretic
6600	-95.19	cp	BRD-K13211965	L-741742	Dopamine receptor antagonist		DRD4, DRD3, SCN1A, SCN3A	Dopamine receptor antagonist
6601	-95.2	cp	BRD-K17705806	JTC-801	Opioid receptor antagonist		OPRL1	Opioid receptor antagonist
6602	-95.22	oe	ccsbBroad304_01933	TEAD2	-			
6603	-95.26	kd	CGS001-9641	IKBKE	IKK family			
6604	-95.27	kd	CGS001-8639	AOC3	Oxidoreductases			
6605	-95.28	cp	BRD-K02581333	protein-tyrosine-phosphatase-inhibitor-IV	Tyrosine phosphatase inhibitor		PTPN1, PTPN11	Tyrosine phosphatase inhibitor
6606	-95.28	cp	BRD-K59469039	AG-879	Angiogenesis inhibitor		ERBB2, KDR, NTRK1	Angiogenesis inhibitor, Tyrosine kinase inhibitor, VEGFR inhibitor
6607	-95.29	kd	CGS001-2042	EPHA3	Type XIII RTKs: Ephrin receptor family			
6608	-95.31	kd	CGS001-3832	KIF11	Kinesins			
6609	-95.34	cc		X linked mental retardation group 1 LOF	-			
6610	-95.34	oe	ccsbBroad304_02230	HERPUD1	-			
6611	-95.34	cp	BRD-K62959606	sphingosine	Ceramidase inhibitor		GLTP, PVR, TRPM3	Ceramidase inhibitor
6612	-95.34	cp	BRD-K56001384	antimycin-a	ATP synthase inhibitor		CYCS	ATP synthase inhibitor
6613	-95.35	cp	BRD-K47207162	zimelidine	Serotonin reuptake inhibitor		SLC6A4, MAOA, MAOB	Serotonin reuptake inhibitor
6614	-95.37	kd	CGS001-337867	UBAC2	-			
6615	-95.37	kd	CGS001-10095	ARPC1B	Actin related protein 2/3 complex subunits			
6616	-95.39	oe	ccsbBroad304_08113	DNAJC15	Heat shock proteins / DNAJ (HSP40)			
6617	-95.4	kd	CGS001-339500	ZNF678	Zinc fingers, C2H2-type			
6618	-95.41	cp	BRD-A58564983	selamectin	Nematocide			Nematocide
6619	-95.42	cp	BRD-A41833852	naloxone	Opioid receptor antagonist		OPRM1, OPRK1, OPRD1, CREB1, ESR1, TLR4	Opioid receptor antagonist
6620	-95.43	oe	ccsbBroad304_00113	ASNS	-			
6621	-95.43	kd	CGS001-4729	NDUFV2	Mitochondrial respiratory chain complex / Complex I			
6622	-95.44	cp	BRD-K40656405	L-165041	PPAR receptor agonist		PPARD	PPAR receptor agonist
6623	-95.44	kd	CGS001-84936	ZFYVE19	Zinc fingers, FYVE domain containing			
6624	-95.46	kd	CGS001-9517	SPTLC2	Serine palmitoyltransferase			
6625	-95.49	cp	BRD-A91452556	estradiol-cypionate	Estrogen receptor agonist		ESR1	Estrogen receptor agonist
6626	-95.49	kd	CGS001-558	AXL	Fibronectin type III domain containing			
6627	-95.5	cp	BRD-K27184429	levocetirizine	Histamine receptor antagonist		HRH1, CXCL8	Histamine receptor antagonist
6628	-95.51	oe	ccsbBroad304_01927	NR0B2	DAX-like receptors			
6629	-95.52	cp	BRD-K14920963	erythrosine	Coloring agent			Coloring agent
6630	-95.52	kd	CGS001-55366	LGR4	GPCR / Class A : Orphans			
6631	-95.52	kd	CGS001-1045	CDX2	Homeoboxes / ANTP class : HOXL subclass			
6632	-95.56	cp	BRD-K24681473	YM-155	Survivin inhibitor		BIRC5	Survivin inhibitor
6633	-95.56	kd	CGS001-91464	ISX	Homeoboxes / PRD class			
6634	-95.58	cp	BRD-A73581086	ergometrine	Adrenergic receptor agonist		ADRA1A, HTR1E, HTR2A	Adrenergic receptor agonist, Serotonin receptor agonist
6635	-95.6	oe	ccsbBroad304_01291	MAP2K6	MAPKK:STE7 family			
6636	-95.6	cp	BRD-K65814004	diphenyleneiodonium	Nitric oxide synthase inhibitor		ALDH1A2, ALDH2, ALDH5A1, ALDH7A1, NOX3, XDH	Nitric oxide synthase inhibitor
6637	-95.62	kd	CGS001-7077	TIMP2	-			
6638	-95.62	kd	CGS001-2592	GALT	-			
6639	-95.63	cp	BRD-K39733634	L-161982	Prostanoid receptor antagonist		PTGER4	Prostanoid receptor antagonist, Angiotensin receptor antagonist
6640	-95.64	cp	BRD-K80738081	resveratrol	Cytochrome P450 inhibitor		PTGS1, PTGS2, SIRT1, APOA1, BACE1, CSNK2A1, MAOA, NQO2, SCN5A, TXNRD1, TXNRD2, XDH	Cytochrome P450 inhibitor, SIRT activator
6641	-95.67	oe	ccsbBroad304_07520	USP15	Ubiquitin-specific peptidases			
6642	-95.67	kd	CGS001-900	CCNG1	-			
6643	-95.68	cc		FLT3 inhibitor	-			
6644	-95.68	oe	ccsbBroad304_06234	G6PC	-			
6645	-95.68	oe	ccsbBroad304_01166	PDK2	PDHK family			
6646	-95.72	oe	ccsbBroad304_10012	ZNF546	Zinc fingers, C2H2-type			
6647	-95.75	kd	CGS001-350	APOH	Apolipoproteins			
6648	-95.78	oe	ccsbBroad304_01398	RHEB	-			
6649	-95.8	kd	CGS001-1662	DDX10	DEAD-boxes			
6650	-95.81	cp	BRD-K51223576	AG-99	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
6651	-95.81	cp	BRD-A34205397	suloctidil	Adrenergic receptor antagonist			Adrenergic receptor antagonist
6652	-95.84	oe	ccsbBroad304_02741	PDS5A	-			
6653	-95.85	oe	ccsbBroad304_03696	C19ORF10	-			
6654	-95.88	oe	ccsbBroad304_01302	KLK6	Chymotrypsin			
6655	-95.88	kd	CGS001-57057	TBX20	T-boxes			
6656	-95.89	cp	BRD-A08003242	rhodomyrtoxin-b	sodium fluorescein uptake inhibitor			sodium fluorescein uptake inhibitor
6657	-95.89	cp	BRD-K05901394	terguride	Dopamine receptor agonist		DRD2, HTR2A, HTR2B, ADRA1A, ADRA2A, ADRA2B, ADRA2C, DRD3, DRD4, HTR1A, HTR1B, HTR1D, HTR2C, PRL	Dopamine receptor agonist, Serotonin receptor antagonist
6658	-95.93	cc		FOS transcription factor family GOF	-			
6659	-95.93	cp	BRD-K08417745	SID-26681509	Cathepsin inhibitor		CTSL	Cathepsin inhibitor
6660	-95.94	cp	BRD-K00662280	CL-218872	GABA receptor agonist		GABRA1, GABRA2, GABRA3, GABRA5, GABRB2, GABRG2	GABA receptor agonist
6661	-95.97	cc		ATP synthase inhibitor	-			
6662	-95.98	kd	CGS001-5361	PLXNA1	Plexins			
6663	-96	cc		HIV protease inhibitor	-			
6664	-96	cp	BRD-K67578145	GDC-0879	RAF inhibitor		BRAF	RAF inhibitor
6665	-96.03	cc		Estrogen receptor agonist	-			
6666	-96.03	kd	CGS001-55837	EAPP	-			
6667	-96.04	oe	ccsbBroad304_03005	HCAR1	GPCR / Class A : Hydroxy-carboxylic acid receptors			
6668	-96.05	cp	BRD-K14791739	fluticasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, CYP3A7, NR3C2, PGR, PLA2G4A	Glucocorticoid receptor agonist
6669	-96.05	cp	BRD-K42748308	XE-991	Potassium channel blocker		KCNQ1, KCNQ2, KCNQ3, KCNQ4, KCNQ5	Potassium channel blocker
6670	-96.06	kd	CGS001-55176	SEC61A2	-			
6671	-96.06	kd	CGS001-663	BNIP2	-			
6672	-96.1	cp	BRD-K07403598	CAY-10470	NFkB pathway inhibitor		NFKB1, TNF	NFkB pathway inhibitor
6673	-96.12	oe	ccsbBroad304_00998	MEIS2	Homeoboxes / TALE class			
6674	-96.13	cp	BRD-K15715913	fluperlapine	Serotonin receptor antagonist		DRD2, HTR2A, HTR6, HTR7	Serotonin receptor antagonist
6675	-96.16	cp	BRD-K04430056	7-nitroindazole	nitric oxide synthase inhibitor		NOS1, NOS2, NOS3	nitric oxide synthase inhibitor
6676	-96.17	cp	BRD-K08924299	palonosetron	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
6677	-96.17	kd	CGS001-6193	RPS5	S ribosomal proteins			
6678	-96.17	kd	CGS001-54583	EGLN1	2-oxoglutarate oxygenases			
6679	-96.18	cp	BRD-K36198571	WAY-170523	Metalloproteinase inhibitor		MMP13	Metalloproteinase inhibitor
6680	-96.21	kd	CGS001-55662	HIF1AN	-			
6681	-96.21	kd	CGS001-527	ATP6V0C	ATPases / V-type			
6682	-96.23	cp	BRD-K82562631	tolmetin	Cyclooxygenase inhibitor		PTGS2, PTGS1	Cyclooxygenase inhibitor
6683	-96.24	cp	BRD-K07736136	VX-702	p38 MAPK inhibitor		MAPK14, MAPK11, MAPK12	p38 MAPK inhibitor
6684	-96.28	cp	BRD-K36009368	NNC-63-0532	Opioid receptor agonist		OPRL1	Opioid receptor agonist
6685	-96.29	cp	BRD-A84327315	calcitriol	Vitamin D receptor agonist		VDR, CYP3A5	Vitamin D receptor agonist
6686	-96.29	cp	BRD-K56429665	calcipotriol	Vitamin D receptor agonist		VDR	Vitamin D receptor agonist
6687	-96.29	cp	BRD-A99449986	MT-21	Caspase activator		CYCS, SLC25A4	Caspase activator
6688	-96.31	kd	CGS001-23581	CASP14	Caspases			
6689	-96.35	oe	ccsbBroad304_07834	GGA2	-			
6690	-96.36	kd	CGS001-6203	RPS9	S ribosomal proteins			
6691	-96.38	cp	BRD-A23637604	oxymetholone	Androgen receptor agonist		AR	Androgen receptor agonist
6692	-96.39	oe	ccsbBroad304_00792	HSD17B2	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6693	-96.39	kd	CGS001-9897	KIAA0196	-			
6694	-96.41	oe	ccsbBroad304_01183	PGD	-			
6695	-96.42	oe	ccsbBroad304_06319	GPR35	GPCR / Class A : Orphans			
6696	-96.46	cp	BRD-K41707108	ceramide	Phosphoenolpyruvate carboxylase activator			Phosphoenolpyruvate carboxylase activator, Serine/threonine protein phosphatase activator
6697	-96.46	kd	CGS001-57541	ZNF398	Zinc fingers, C2H2-type			
6698	-96.47	cp	BRD-K88742110	BRD-K88742110	HDAC inhibitor		HDAC8, IL1B	HDAC inhibitor
6699	-96.48	oe	ccsbBroad304_00931	LCN2	Lipocalins			
6700	-96.48	cp	BRD-K05350981	oligomycin-c	ATPase inhibitor		ATP5A1	ATPase inhibitor, ATP synthase inhibitor
6701	-96.5	kd	CGS001-57693	ZNF317	Zinc fingers, C2H2-type			
6702	-96.52	cp	BRD-A45498368	WYE-125132	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor
6703	-96.54	cc		Lipocalins GOF	-			
6704	-96.56	oe	ccsbBroad304_01495	CCL2	Chemokine ligands			
6705	-96.57	kd	CGS001-5355	PLP2	-			
6706	-96.59	oe	ccsbBroad304_00094	ARF1	ADP-ribosylation factors			
6707	-96.59	kd	CGS001-1345	COX6C	Mitochondrial respiratory chain complex			
6708	-96.6	kd	CGS001-7775	ZNF232	Zinc fingers, C2H2-type			
6709	-96.63	oe	ccsbBroad304_03268	GMPR2	-			
6710	-96.65	cp	BRD-K28912512	nicotinamide	Protein synthesis stimulant		PARP1, AOX1, BST1, CYP2E1, LDHA, SIRT5	Protein synthesis stimulant
6711	-96.65	kd	CGS001-9867	PJA2	RING-type (C3HC4) zinc fingers			
6712	-96.66	kd	CGS001-4097	MAFG	-			
6713	-96.67	cp	BRD-A93206962	L-755507	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
6714	-96.68	cp	BRD-K31792052	pifithrin	Interleukin receptor antagonist			Interleukin receptor antagonist
6715	-96.69	cp	BRD-K70914287	BIBX-1382	EGFR inhibitor		EGFR, ERBB2	EGFR inhibitor, Tyrosine kinase inhibitor
6716	-96.71	oe	ccsbBroad304_07101	TSC2	-			
6717	-96.71	oe	ccsbBroad304_03687	NSFL1C	UBX domain containing			
6718	-96.71	cp	BRD-K54771420	glycocholic-acid	Cholesterol inhibitor		FABP6	Cholesterol inhibitor
6719	-96.72	kd	CGS001-7188	TRAF5	RING-type (C3HC4) zinc fingers			
6720	-96.72	kd	CGS001-3957	LGALS2	Lectins, galactoside-binding			
6721	-96.75	cp	BRD-K97354755	SU-6656	SRC inhibitor		LYN, AURKB, AURKC, BRSK2, CALM1, CAMK2D, LCK, RET, SRC, YES1	SRC inhibitor
6722	-96.75	kd	CGS001-120892	LRRK2	Leucine-rich repeat kinase (LRRK) family			
6723	-96.76	cp	BRD-K64310881	MW-STK33-3B	Potassium channel activator			Potassium channel activator
6724	-96.76	cp	BRD-K96084870	DMBI	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor, VEGFR inhibitor
6725	-96.77	oe	ccsbBroad304_14143	NUSAP1	-			
6726	-96.78	cp	BRD-K12502280	TG-101348	FLT3 inhibitor		JAK2, FLT3, BRD4, JAK1, JAK3, RET, TYK2	FLT3 inhibitor, JAK inhibitor
6727	-96.79	kd	CGS001-10616	RBCK1	RING-type (C3HC4) zinc fingers			
6728	-96.83	kd	CGS001-185	AGTR1	Angiotensin receptors			
6729	-96.84	kd	CGS001-57616	TSHZ3	Teashirt zinc fingers			
6730	-96.84	kd	CGS001-7056	THBD	CD molecules			
6731	-96.87	kd	CGS001-390212	GPR152	GPCR / Class A : Orphans			
6732	-96.88	kd	CGS001-10962	MLLT11	-			
6733	-96.89	cp	BRD-K26863634	BIX-01338	Histone lysine methyltransferase inhibitor			Histone lysine methyltransferase inhibitor
6734	-96.89	kd	CGS001-8019	BRD3	Bromodomain kinase (BRDK) family			
6735	-96.89	kd	CGS001-10254	STAM2	-			
6736	-96.9	oe	ccsbBroad304_07820	SNW1	-			
6737	-96.91	oe	ccsbBroad304_09657	PHF13	Zinc fingers, PHD-type			
6738	-96.92	cp	BRD-K07507905	BRL-37344	Adrenergic receptor agonist		ADRB3, ADRB1, ADRB2	Adrenergic receptor agonist
6739	-96.93	oe	ccsbBroad304_00577	FOXO3	Forkhead boxes			
6740	-96.93	oe	ccsbBroad304_00238	CCNE1	-			
6741	-96.93	kd	CGS001-204851	HIPK1	HIPK subfamily			
6742	-96.94	kd	CGS001-6598	SMARCB1	-			
6743	-96.95	cp	BRD-K05658747	raltegravir	HIV integrase inhibitor			HIV integrase inhibitor
6744	-96.97	oe	ccsbBroad304_00834	IFNGR1	Interferon receptor family			
6745	-96.98	oe	ccsbBroad304_09006	RPF1	-			
6746	-96.98	cp	BRD-K53414658	tivozanib	VEGFR inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, PDGFRB	VEGFR inhibitor
6747	-97	cp	BRD-K55748775	SCH-28080	ATPase inhibitor		ATP4A	ATPase inhibitor
6748	-97.03	cp	BRD-K05151076	ZK-164015	Estrogen receptor antagonist		ESR1, ESR2	Estrogen receptor antagonist
6749	-97.04	oe	ccsbBroad304_02958	HSPB8	Heat shock proteins / HSPB			
6750	-97.04	kd	CGS001-1831	TSC22D3	-			
6751	-97.05	cc		Serine proteases GOF	-			
6752	-97.05	cp	BRD-K10065684	dantron	Laxative			Laxative
6753	-97.06	kd	CGS001-10094	ARPC3	Actin related protein 2/3 complex subunits			
6754	-97.07	cp	BRD-K10860596	granisetron	Serotonin receptor antagonist		HTR3A, CYP3A5	Serotonin receptor antagonist
6755	-97.09	kd	CGS001-5287	PIK3C2B	Phosphatidylinositol-4-phosphate 3-kinase family			
6756	-97.09	cp	BRD-A07780951	orciprenaline	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
6757	-97.1	kd	CGS001-4175	MCM6	-			
6758	-97.11	kd	CGS001-6885	MAP3K7	MAPKKK:TAK1 subfamily			
6759	-97.12	cc		NFkB pathway inhibitor	-			
6760	-97.12	kd	CGS001-83933	HDAC10	Histone deacetylases			
6761	-97.16	oe	ccsbBroad304_05309	OR52B2	GPCR / Class A : Olfactory receptors			
6762	-97.18	oe	ccsbBroad304_02133	CD83	CD molecules			
6763	-97.18	cp	BRD-A62021152	WAY-161503	Serotonin receptor agonist		HTR2C	Serotonin receptor agonist
6764	-97.22	oe	ccsbBroad304_07277	RTCD1	-			
6765	-97.22	kd	CGS001-57147	SCYL3	-			
6766	-97.22	kd	CGS001-8986	RPS6KA4	MSK subfamily			
6767	-97.22	oe	ccsbBroad304_02197	VPS26A	-			
6768	-97.23	kd	CGS001-7570	ZNF22	Zinc fingers, C2H2-type			
6769	-97.24	kd	CGS001-7431	VIM	Intermediate filaments type III			
6770	-97.25	oe	ccsbBroad304_02218	IKBKE	IKK family			
6771	-97.25	oe	ccsbBroad304_04399	PGBD1	-			
6772	-97.26	cp	BRD-A15415227	GW-1929	PPAR receptor agonist		INS, PPARG	PPAR receptor agonist, Insulin sensitizer
6773	-97.27	cp	BRD-K54256913	MK-1775	WEE1 kinase inhibitor		WEE1	WEE1 kinase inhibitor
6774	-97.3	cc		Baculoviral IAP repeat domain containing LOF	-			
6775	-97.3	kd	CGS001-6469	SHH	-			
6776	-97.31	kd	CGS001-26574	AATF	-			
6777	-97.33	oe	ccsbBroad304_00770	HOXA2	Homeoboxes / ANTP class : HOXL subclass			
6778	-97.33	cp	BRD-K37447567	hydrocotarnine	Opioid receptor antagonist			Opioid receptor antagonist
6779	-97.33	kd	CGS001-7917	BAG6	-			
6780	-97.34	kd	CGS001-84290	CAPNS2	EF-hand domain containing			
6781	-97.35	oe	ccsbBroad304_00118	ATIC	-			
6782	-97.35	kd	CGS001-5522	PPP2R2C	Serine/threonine phosphatases / Protein phosphatase 2, regulatory subunits			
6783	-97.35	oe	ccsbBroad304_06028	CPE	Carboxypeptidase A			
6784	-97.36	oe	ccsbBroad304_02239	RASSF2	-			
6785	-97.36	kd	CGS001-11243	PMF1	-			
6786	-97.38	kd	CGS001-3635	INPP5D	Inositol polyphosphate phosphatases			
6787	-97.39	oe	ccsbBroad304_06975	SMARCC2	-			
6788	-97.41	oe	ccsbBroad304_00489	EHHADH	-			
6789	-97.41	kd	CGS001-1314	COPA	Endogenous ligands			
6790	-97.47	cp	BRD-K12102668	nialamide	Monoamine oxidase inhibitor		COMT, MAOA, MAOB	Monoamine oxidase inhibitor
6791	-97.48	oe	ccsbBroad304_03961	SMURF2	-			
6792	-97.48	oe	ccsbBroad304_08853	RGS18	Regulators of G-protein signaling			
6793	-97.48	kd	CGS001-25888	ZNF473	Zinc fingers, C2H2-type			
6794	-97.49	kd	CGS001-10915	TCERG1	-			
6795	-97.5	oe	ccsbBroad304_01289	MAPK13	MAPK:p38 subfamily			
6796	-97.5	oe	ccsbBroad304_02313	ACTR3	-			
6797	-97.5	cp	BRD-K84266862	BRL-50481	Phosphodiesterase inhibitor		PDE7A, PDE7B	Phosphodiesterase inhibitor
6798	-97.5	kd	CGS001-330	BIRC3	Inhibitors of apoptosis (IAP) protein family			
6799	-97.51	oe	ccsbBroad304_02485	STAMBP	-			
6800	-97.51	cp	BRD-K91263825	nortriptyline	Tricyclic antidepressant		KCNJ10, SLC6A2, SLC6A4, ADRA1A, ADRA1B, ADRA1D, ADRA2A, ADRA2B, ADRA2C, ADRB1, ADRB2, ADRB3, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, CYP2C19, DRD2, HRH1, HTR1A, HTR2A, HTR2C, HTR6, PGRMC1, PIK3CD, SIGMAR1	Tricyclic antidepressant
6801	-97.51	kd	CGS001-54623	PAF1	-			
6802	-97.52	kd	CGS001-6004	RGS16	Regulators of G-protein signaling			
6803	-97.53	kd	CGS001-5294	PIK3CG	Phosphatidylinositol kinases			
6804	-97.54	cp	BRD-A49734948	foliosidine	Plant alkaloid			Plant alkaloid
6805	-97.55	kd	CGS001-5471	PPAT	Phosphoribosyl pyrophosphate amidotransferase			
6806	-97.55	kd	CGS001-54512	EXOSC4	-			
6807	-97.57	kd	CGS001-2864	FFAR1	Fatty acid receptors			
6808	-97.58	kd	CGS001-3932	LCK	Src family			
6809	-97.59	oe	ccsbBroad304_00415	CYP24A1	Cytochrome P450s			
6810	-97.6	oe	ccsbBroad304_02784	SUZ12	Zinc fingers, C2H2-type			
6811	-97.6	oe	ccsbBroad304_09503	KLHDC9	-			
6812	-97.6	kd	CGS001-8611	PPAP2A	Lipid phosphate phosphatases			
6813	-97.61	kd	CGS001-4709	NDUFB3	Mitochondrial respiratory chain complex / Complex I			
6814	-97.62	oe	ccsbBroad304_02319	PREB	WD repeat domain containing			
6815	-97.63	oe	ccsbBroad304_03173	TMED7	-			
6816	-97.64	oe	ccsbBroad304_08296	UBE2J1	Ubiquitin-conjugating enzymes E2			
6817	-97.66	cp	BRD-A39268308	epibatidine	Acetylcholine receptor agonist		CHRFAM7A, CHRNA2, CHRNA3, CHRNA4, CHRNA7	Acetylcholine receptor agonist
6818	-97.66	kd	CGS001-10694	CCT8	Heat Shock Proteins / Chaperonins			
6819	-97.67	oe	ccsbBroad304_01478	S100A11	EF-hand domain containing			
6820	-97.67	cp	BRD-K43068349	AMG-9810	TRPV antagonist		TRPV1	TRPV antagonist
6821	-97.67	kd	CGS001-9748	SLK	SLK subfamily			
6822	-97.69	oe	ccsbBroad304_01658	PRDX2	-			
6823	-97.69	kd	CGS001-6282	S100A11	EF-hand domain containing			
6824	-97.7	kd	CGS001-501	ALDH7A1	Aldehyde dehydrogenases			
6825	-97.72	kd	CGS001-378	ARF4	ADP-ribosylation factors			
6826	-97.73	cp	BRD-A44448661	pentobarbital	Barbiturate antiepileptic		GABRA1, CHRNA4, CHRNA7, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ, GRIA2, GRIK2, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Barbiturate antiepileptic, GABA receptor modulator
6827	-97.73	kd	CGS001-5879	RAC1	Endogenous ligands			
6828	-97.75	cp	BRD-K60623809	SU-11652	Tyrosine kinase inhibitor		KDR, PDGFRB, CAMK1G, FGF2, FGFR1, FLT1, KIT, PDGFRA	Tyrosine kinase inhibitor
6829	-97.75	cp	BRD-K76304753	phenazopyridine	Local anesthetic		SCN1A	Local anesthetic
6830	-97.75	kd	CGS001-4055	LTBR	Tumor necrosis factor receptor superfamily			
6831	-97.78	kd	CGS001-9324	HMGN3	High-mobility group / Canonical			
6832	-97.78	kd	CGS001-10552	ARPC1A	Actin related protein 2/3 complex subunits			
6833	-97.79	cp	BRD-K28849549	mesalazine	Cyclooxygenase inhibitor		PTGS1, PPARG, PTGS2, ALOX5, CHUK, CTNNB1, IKBKB, MPO, NAT1	Cyclooxygenase inhibitor, Lipoxygenase inhibitor, Prostanoid receptor antagonist
6834	-97.8	kd	CGS001-117195	MRGPRX3	GPCR / Class A : Orphans			
6835	-97.8	kd	CGS001-56616	DIABLO	-			
6836	-97.81	cc		LIM class homeoboxes GOF	-			
6837	-97.81	cp	BRD-K51290057	SA-792709	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
6838	-97.83	oe	ccsbBroad304_14174	CDKAL1	-			
6839	-97.83	kd	CGS001-56670	SUCNR1	GPCR / Class A : Orphans			
6840	-97.84	kd	CGS001-55746	NUP133	-			
6841	-97.85	oe	ccsbBroad304_07783	PMF1-BGLAP	-			
6842	-97.85	kd	CGS001-10657	KHDRBS1	-			
6843	-97.88	oe	ccsbBroad304_05982	CDX2	Homeoboxes / ANTP class : HOXL subclass			
6844	-97.88	kd	CGS001-4849	CNOT3	-			
6845	-97.89	oe	ccsbBroad304_01484	SATB1	Homeoboxes / CUT class			
6846	-97.89	kd	CGS001-10668	CGRRF1	RING-type (C3HC4) zinc fingers			
6847	-97.9	oe	ccsbBroad304_00774	HOXA10	Homeoboxes / ANTP class : HOXL subclass			
6848	-97.91	cp	BRD-K83963101	MLN-8054	Aurora kinase inhibitor		AURKA	Aurora kinase inhibitor, Mitotic inhibitor, Protein kinase inhibitor
6849	-97.92	oe	ccsbBroad304_04261	RAB1B	RAB, member RAS oncogene			
6850	-97.92	kd	CGS001-63027	SLC22A23	Orphan or poorly characterized SLC22 family members			
6851	-97.93	cp	BRD-K91699951	benzonatate	Local anesthetic		SCN5A	Local anesthetic
6852	-97.94	oe	ccsbBroad304_05979	CDK9	Cyclin-dependent kinases, CDK9 subfamily			
6853	-97.94	cp	BRD-A28970875	puromycin	Protein synthesis inhibitor		NHP2L1, RPL10L, RPL11, RPL13A, RPL15, RPL19, RPL23, RPL23A, RPL26L1, RPL3, RPL37, RPL8, RSL24D1	Protein synthesis inhibitor
6854	-97.95	oe	ccsbBroad304_01515	SDHD	Mitochondrial respiratory chain complex / Complex II			
6855	-97.97	oe	ccsbBroad304_05856	ASAH1	Acid ceramidase			
6856	-97.97	kd	CGS001-56889	TM9SF3	-			
6857	-97.98	cp	BRD-K32526544	DCEBIO	Potassium channel activator		KCNN2, KCNN3, KCNN4	Potassium channel activator
6858	-97.98	kd	CGS001-8751	ADAM15	ADAM metallopeptidase domain containing			
6859	-97.99	cp	BRD-K92870997	pterostilbene	Cyclooxygenase inhibitor		FAAH, PPARA, PTGS1, PTGS2	Cyclooxygenase inhibitor, PPAR receptor agonist
6860	-97.99	kd	CGS001-634	CEACAM1	CD molecules			
6861	-98	oe	ccsbBroad304_00398	CTSL2	-			
6862	-98	oe	ccsbBroad304_06022	COX7B	Mitochondrial respiratory chain complex			
6863	-98.01	cc		Vesicular Transport LOF	-			
6864	-98.01	oe	ccsbBroad304_02175	MAGED1	-			
6865	-98.01	kd	CGS001-537	ATP6AP1	-			
6866	-98.02	kd	CGS001-5193	PEX12	-			
6867	-98.03	oe	ccsbBroad304_00781	HPD	Oxidoreductases			
6868	-98.03	kd	CGS001-22818	COPZ1	-			
6869	-98.03	kd	CGS001-509	ATP5C1	ATPases / F-type			
6870	-98.04	kd	CGS001-8505	PARG	-			
6871	-98.04	kd	CGS001-5053	PAH	Amino acid hydroxylases			
6872	-98.04	kd	CGS001-2909	ARHGAP35	Rho GTPase activating proteins			
6873	-98.05	kd	CGS001-5209	PFKFB3	-			
6874	-98.05	cp	BRD-K89732114	trifluoperazine	Dopamine receptor antagonist		DRD2, ABCG2, ADRA1A, CALM1, CALY, CAMK2A, DRD4, HRH1, HTR2A, HTR2C, S100A4, SCN4A, SCN9A, TNNC1	Dopamine receptor antagonist
6875	-98.06	cp	BRD-K99922388	DPO-1	Potassium channel blocker		KCNA5	Potassium channel blocker
6876	-98.06	kd	CGS001-23522	KAT6B	Histone acetyltransferases (HATs)			
6877	-98.07	oe	ccsbBroad304_00832	IFNB1	Interferons			
6878	-98.07	cp	BRD-K06543683	bisindolylmaleimide-ix	CDK inhibitor		SIRT1, AKT1, GSK3B, LCK, LRRK2, MAPK1, MAPK11, MAPK12, MAPK14, MAPK8, PRKCA, ROCK1, RPS6KB1, SIRT2	CDK inhibitor, PKC inhibitor
6879	-98.09	cp	BRD-K13087974	4,5-dianilinophthalimide	EGFR inhibitor		EGFR	EGFR inhibitor
6880	-98.1	cp	BRD-U66370498	androstanol	CAR antagonist		NR1I3	CAR antagonist
6881	-98.1	kd	CGS001-2122	MECOM	Zinc fingers, C2H2-type			
6882	-98.1	kd	CGS001-147183	KRT25	Intermediate filaments type I, keratins (acidic)			
6883	-98.12	cp	BRD-K36627727	tamibarotene	Retinoid receptor agonist		RARA, RARB	Retinoid receptor agonist
6884	-98.12	cp	BRD-K75958195	pizotifen	Serotonin receptor antagonist		HTR2A, HTR1A, HTR2C	Serotonin receptor antagonist
6885	-98.13	cp	BRD-K00627859	tubastatin-a	HDAC inhibitor		HDAC6	HDAC inhibitor
6886	-98.14	kd	CGS001-8092	ALX1	Homeoboxes / PRD class			
6887	-98.16	cp	BRD-K35960502	niclosamide	DNA replication inhibitor		STAT3	DNA replication inhibitor, STAT inhibitor
6888	-98.17	cp	BRD-K52020312	metronidazole	DNA inhibitor		CYP2C8, CYP2E1, CYP3A5, CYP3A7	DNA inhibitor, Antiprotozoal
6889	-98.17	cp	BRD-K81272440	dantrolene	Calcium channel blocker		RYR1, RYR3	Calcium channel blocker
6890	-98.17	kd	CGS001-3815	KIT	Type III RTKs: PDGFR, CSFR, Kit, FLT3 receptor family			
6891	-98.18	kd	CGS001-6927	HNF1A	Homeoboxes / HNF class			
6892	-98.19	kd	CGS001-9212	AURKB	Aurora kinase			
6893	-98.23	oe	ccsbBroad304_09756	PAQR7	-			
6894	-98.23	kd	CGS001-7849	PAX8	Paired boxes			
6895	-98.23	kd	CGS001-2936	GSR	Oxidoreductases			
6896	-98.23	kd	CGS001-5167	ENPP1	-			
6897	-98.24	cp	BRD-K32696739	noreleagnine	Monoamine oxidase inhibitor		ADRA2A, ADRA2B, ADRA2C, HTR2A, MAOA, MAOB	Monoamine oxidase inhibitor, Serotonin receptor agonist
6898	-98.25	oe	ccsbBroad304_06855	RDX	-			
6899	-98.25	cp	BRD-K68065987	MK-2206	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
6900	-98.27	oe	ccsbBroad304_00101	RHOC	-			
6901	-98.27	cp	BRD-K49027941	PSB-1115	Adenosine receptor antagonist		ADORA2B, ADORA1, ADORA3	Adenosine receptor antagonist
6902	-98.27	cp	BRD-A03816571	CP-55940	Cannabinoid receptor agonist		CNR1, CNR2, CXCR4, GPR55	Cannabinoid receptor agonist
6903	-98.27	cp	BRD-K29668683	BD-1063	Sigma receptor antagonist		SIGMAR1	Sigma receptor antagonist
6904	-98.27	kd	CGS001-23326	USP22	Ubiquitin-specific peptidases			
6905	-98.27	kd	CGS001-3601	IL15RA	IL-2 receptor family			
6906	-98.29	cp	BRD-K87510569	RS-504393	CC chemokine receptor antagonist		CCR2, CCL2	CC chemokine receptor antagonist
6907	-98.29	kd	CGS001-79017	GGCT	Leukotriene and lipoxin metabolism			
6908	-98.3	cp	BRD-K72676686	fluvoxamine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CYP2C19	Selective serotonin reuptake inhibitor (SSRI)
6909	-98.32	cc		Calcium channel blocker	-			
6910	-98.32	kd	CGS001-9341	VAMP3	Vesicle-associated membrane proteins			
6911	-98.33	oe	ccsbBroad304_00509	EPHX1	-			
6912	-98.34	oe	ccsbBroad304_00180	BTK	Pleckstrin homology (PH) domain containing			
6913	-98.34	kd	CGS001-132	ADK	Adenosine turnover			
6914	-98.34	oe	ccsbBroad304_06383	HMMR	CD molecules			
6915	-98.36	oe	ccsbBroad304_08536	PARL	-			
6916	-98.36	kd	CGS001-51478	HSD17B7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 2			
6917	-98.36	kd	CGS001-2745	GLRX	-			
6918	-98.37	kd	CGS001-5523	PPP2R3A	EF-hand domain containing			
6919	-98.38	kd	CGS001-2002	ELK1	ETS Transcription Factors			
6920	-98.38	cp	BRD-K64517075	heliomycin	ATP synthase inhibitor			ATP synthase inhibitor
6921	-98.39	cp	BRD-K51485625	ritonavir	HIV protease inhibitor		CYP3A4, CYP1A2, CYP2B6, CYP2C19, CYP3A5, CYP3A7	HIV protease inhibitor
6922	-98.39	kd	CGS001-10473	HMGN4	High-mobility group / Canonical			
6923	-98.4	cc		Histone deacetylases LOF	-			
6924	-98.41	cp	BRD-K86958018	olvanil	TRPV agonist		TRPV1, CNR1, GPR119	TRPV agonist
6925	-98.42	oe	ccsbBroad304_07889	QPRT	-			
6926	-98.42	oe	ccsbBroad304_05947	CCNC	-			
6927	-98.42	kd	CGS001-6541	SLC7A1	SLC7 family			
6928	-98.43	kd	CGS001-122011	CSNK1A1L	Casein kinase 1 (CK1) family			
6929	-98.43	cp	BRD-K94830329	ataluren	CFTR channel agonist		CFTR, DMD, F8, F9	CFTR channel agonist, Dystrophin stimulant
6930	-98.44	cc		Protein synthesis inhibitor	-			
6931	-98.45	kd	CGS001-4605	MYBL2	-			
6932	-98.47	cc		PPAR receptor agonist	-			
6933	-98.47	cp	BRD-K49372556	mofezolac	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
6934	-98.47	cp	BRD-K80970344	pyrrolidine-dithiocarbamate	NFkB pathway inhibitor		HSD11B1, RELA	NFkB pathway inhibitor
6935	-98.47	kd	CGS001-4323	MMP14	Matrix metallopeptidase			
6936	-98.49	kd	CGS001-1153	CIRBP	RNA binding motif (RRM) containing			
6937	-98.5	kd	CGS001-10645	CAMKK2	Meta subfamily			
6938	-98.5	kd	CGS001-253430	IPMK	-			
6939	-98.51	kd	CGS001-56997	ADCK3	ABC1-B subfamily			
6940	-98.54	cp	BRD-K01649396	indatraline	Norepinephrine transporter inhibitor		SLC6A2, SLC6A3, SLC6A4	Norepinephrine transporter inhibitor
6941	-98.54	cp	BRD-K74305673	IKK-2-inhibitor-V	IKK inhibitor		IKBKB	IKK inhibitor, NFkB pathway inhibitor
6942	-98.54	kd	CGS001-8226	HDHD1	-			
6943	-98.56	oe	ccsbBroad304_06393	HOXC4	Homeoboxes / ANTP class : HOXL subclass			
6944	-98.58	oe	ccsbBroad304_00392	CTLA4	CD molecules			
6945	-98.58	kd	CGS001-391013	PLA2G2C	-			
6946	-98.6	cp	BRD-K08206212	entecavir	Reverse transcriptase inhibitor			Reverse transcriptase inhibitor, DNA replication inhibitor
6947	-98.6	cp	BRD-A17065207	brefeldin-a	Protein synthesis inhibitor		ARF1, ARFGEF1, ARFGEF2, CYTH2, GBF1, SAR1A	Protein synthesis inhibitor, Brefeldin A inhibited guanine nucleotide exchange protein inhibitor, Golgi-specific brefeldin A-resistance guanine nucleotide exchange factor inhibitor
6948	-98.6	kd	CGS001-10482	NXF1	-			
6949	-98.62	cp	BRD-K40624912	ZM-39923	JAK inhibitor		JAK1, JAK3	JAK inhibitor
6950	-98.62	cp	BRD-K67352070	TC-2559	Acetylcholine receptor agonist		CHRNA4	Acetylcholine receptor agonist
6951	-98.62	kd	CGS001-29915	HCFC2	-			
6952	-98.63	oe	ccsbBroad304_01777	WNT1	Endogenous ligands			
6953	-98.63	cp	BRD-K17110974	aristolochic-acid	Phospholipase inhibitor			Phospholipase inhibitor
6954	-98.63	cp	BRD-K31912990	CGP-71683	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
6955	-98.63	kd	CGS001-84669	USP32	EF-hand domain containing			
6956	-98.64	cp	BRD-A94413429	NTNCB	Neuropeptide receptor antagonist		NPY5R	Neuropeptide receptor antagonist
6957	-98.65	kd	CGS001-3034	HAL	-			
6958	-98.67	oe	ccsbBroad304_01038	MSRA	-			
6959	-98.67	cp	BRD-A27489425	rolitetracycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
6960	-98.67	kd	CGS001-3091	HIF1A	Basic helix-loop-helix proteins			
6961	-98.67	kd	CGS001-406	ARNTL	Basic helix-loop-helix proteins			
6962	-98.67	cp	BRD-K10573841	tunicamycin	GLCNAC phosphotransferase inhibitor		GNPTAB	GLCNAC phosphotransferase inhibitor
6963	-98.7	kd	CGS001-5170	PDPK1	PDK1 family			
6964	-98.71	cp	BRD-A71157293	fursultiamine	Vitamin B			Vitamin B
6965	-98.71	kd	CGS001-8649	LAMTOR3	-			
6966	-98.72	cp	BRD-A49370193	RO-60-0175	Serotonin receptor agonist		HTR2C, HTR2A, HTR2B	Serotonin receptor agonist
6967	-98.73	cp	BRD-K04546108	JAK3-inhibitor-VI	JAK inhibitor		JAK3	JAK inhibitor
6968	-98.73	kd	CGS001-5511	PPP1R8	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
6969	-98.73	kd	CGS001-563	AZGP1	Immunoglobulin superfamily / C1-set domain containing			
6970	-98.74	cp	BRD-K98157055	SIB-1757	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
6971	-98.74	cp	BRD-K47598052	PP-1	SRC inhibitor		HCK, RET, SRC	SRC inhibitor, ABL inhibitor
6972	-98.74	cp	BRD-K33204703	AG-370	PDGFR receptor inhibitor		PDGFRB	PDGFR receptor inhibitor
6973	-98.75	oe	ccsbBroad304_03420	TOLLIP	-			
6974	-98.76	kd	CGS001-7376	NR1H2	Liver X receptor-like receptors			
6975	-98.77	cp	BRD-A82590476	SDZ-NKT-343	Tachykinin antagonist		TACR1	Tachykinin antagonist
6976	-98.78	kd	CGS001-2647	BLOC1S1	Biogenesis of lysosomal organelles complex-1 subunits			
6977	-98.79	oe	ccsbBroad304_10240	CROT	-			
6978	-98.79	oe	ccsbBroad304_04649	ADC	-			
6979	-98.8	cp	BRD-A19248578	latrunculin-b	Actin polymerization inhibitor		ACTA1, MKL1, SPIRE2	Actin polymerization inhibitor, Unidentified pharmacological activity
6980	-98.8	cp	BRD-K63550407	erythromycin	NFkB pathway inhibitor		CYP3A4, MLNR	NFkB pathway inhibitor
6981	-98.81	oe	ccsbBroad304_12885	ZFYVE19	Zinc fingers, FYVE domain containing			
6982	-98.82	oe	ccsbBroad304_02367	CALCOCO2	-			
6983	-98.82	oe	ccsbBroad304_00126	ATP5A1	ATPases / F-type			
6984	-98.82	cp	BRD-K68437527	EMF-bca1-60	caspase inhibitor			caspase inhibitor
6985	-98.82	kd	CGS001-27097	TAF5L	WD repeat domain containing			
6986	-98.84	oe	ccsbBroad304_00752	HMGB3	High-mobility group / Canonical			
6987	-98.84	oe	ccsbBroad304_00378	CSNK1D	Casein kinase 1 (CK1) family			
6988	-98.84	cp	BRD-A44780397	mifepristone	Glucocorticoid receptor antagonist		PGR, NR3C1, AR, CYP2B6, CYP2C8, CYP3A5, CYP3A7, NR1I2	Glucocorticoid receptor antagonist, Progesterone receptor antagonist
6989	-98.86	oe	ccsbBroad304_00512	EPO	Endogenous ligands			
6990	-98.86	oe	ccsbBroad304_01290	MAP2K5	MAPKK:STE7 family			
6991	-98.86	cp	BRD-A02481876	importazole	Importin-beta transport receptor inhibitor		KPNB1	Importin-beta transport receptor inhibitor
6992	-98.86	cp	BRD-K06854232	AM-580	Retinoid receptor agonist		RARA	Retinoid receptor agonist
6993	-98.86	kd	CGS001-9978	RBX1	RING-type (C3HC4) zinc fingers			
6994	-98.87	kd	CGS001-10544	PROCR	CD molecules			
6995	-98.88	oe	ccsbBroad304_09983	ZNF454	Zinc fingers, C2H2-type			
6996	-98.88	kd	CGS001-8667	EIF3H	-			
6997	-98.91	oe	ccsbBroad304_00249	CD14	CD molecules			
6998	-98.91	cp	BRD-A32349859	methyl-angolensate	Apoptosis inhibitor		HTR2B	Apoptosis inhibitor
6999	-98.91	kd	CGS001-7276	TTR	-			
7000	-98.92	oe	ccsbBroad304_02213	TRAF4	RING-type (C3HC4) zinc fingers			
7001	-98.92	kd	CGS001-178	AGL	-			
7002	-98.93	cp	BRD-A77050075	heraclenol	Vitamin K antagonist			Vitamin K antagonist
7003	-98.93	cp	BRD-K18855837	varenicline	Acetylcholine receptor agonist		CHRNA4, CHRNA3, CHRNA6, CHRNA7, CHRNB2	Acetylcholine receptor agonist
7004	-98.93	cp	BRD-K28143534	cyproheptadine	Histamine receptor antagonist		HRH1, ADRA1A, ADRA1B, ADRA1D, CHRM1, CHRM2, CHRM3, HTR2A, HTR2B, HTR2C, HTR6, HTR7	Histamine receptor antagonist
7005	-98.93	cp	BRD-K34154330	tracazolate	GABA receptor modulator		GABRA1	GABA receptor modulator
7006	-98.94	cp	BRD-A84134924	pancuronium	Acetylcholine receptor antagonist		CHRM2, CHRM3, CHRNA1, CHRNA2	Acetylcholine receptor antagonist
7007	-98.94	kd	CGS001-7301	TYRO3	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
7008	-98.95	cp	BRD-A15079084	phorbol-12-myristate-13-acetate	PKC activator		CD4, KCNT2, PRKCA, TRPV4	PKC activator
7009	-98.95	cp	BRD-K37991163	paroxetine	Selective serotonin reuptake inhibitor (SSRI)		SLC6A4, CHRM1, CHRM2, CHRM3, CHRM4, CHRM5, HTR2A, SLC6A2	Selective serotonin reuptake inhibitor (SSRI)
7010	-98.95	kd	CGS001-11315	PARK7	Parkinson disease			
7011	-98.95	kd	CGS001-283150	FOXR1	Forkhead boxes			
7012	-98.97	oe	ccsbBroad304_02311	ARPC3	Actin related protein 2/3 complex subunits			
7013	-98.97	cp	BRD-K19295594	gossypol	BCL inhibitor		BCL2, BCL2L1, MCL1, BCL2L2, CTGF, EGF	BCL inhibitor, MCL1 inhibitor
7014	-98.98	oe	ccsbBroad304_01312	PSMB8	Proteasome (prosome, macropain) subunits			
7015	-98.98	kd	CGS001-3303	HSPA1A	Heat shock proteins / HSP70			
7016	-98.99	oe	ccsbBroad304_06188	F10	Chymotrypsin			
7017	-98.99	cp	BRD-K43468059	byssochlamic-acid	Mycotoxin			Mycotoxin
7018	-98.99	kd	CGS001-1848	DUSP6	Protein tyrosine phosphatases / Class I Cys-based PTPs : MAP kinase phosphatases			
7019	-99.01	cp	BRD-K48029790	OBAA	Phospholipase inhibitor		PLA2G1B	Phospholipase inhibitor
7020	-99.02	cp	BRD-A89337244	PD-102807	Acetylcholine receptor antagonist		CHRM4	Acetylcholine receptor antagonist
7021	-99.02	kd	CGS001-4089	SMAD4	SMADs			
7022	-99.03	kd	CGS001-84547	PGBD1	-			
7023	-99.04	cp	BRD-K81225797	SCH-58261	Adenosine receptor antagonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor antagonist
7024	-99.04	kd	CGS001-2152	F3	CD molecules			
7025	-99.06	oe	ccsbBroad304_04754	SPIC	ETS Transcription Factors			
7026	-99.06	cp	BRD-K47761761	PD-168077	Dopamine receptor agonist		DRD2, DRD4	Dopamine receptor agonist
7027	-99.06	cp	BRD-K21667562	AM-404	Cyclooxygenase inhibitor		TRPV1, CNR1, CNR2, FAAH	Cyclooxygenase inhibitor, FAAH inhibitor, TRPV antagonist
7028	-99.06	oe	ccsbBroad304_01288	MAPK9	MAPK:JNK subfamily			
7029	-99.07	oe	ccsbBroad304_00145	BACH1	BTB/POZ domain containing			
7030	-99.07	kd	CGS001-7771	ZFP112	-			
7031	-99.07	kd	CGS001-10298	PAK4	PAKB subfamily			
7032	-99.08	oe	ccsbBroad304_08670	DUSP22	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7033	-99.08	cp	BRD-K02227374	milnacipran	Serotonin reuptake inhibitor		SLC6A2, SLC6A4, GRIN1, GRIN2A, GRIN2B, GRIN2C, GRIN2D, GRIN3A, GRIN3B	Serotonin reuptake inhibitor
7034	-99.08	cp	BRD-K94270326	ecopipam	Dopamine receptor antagonist		DRD1, DRD5, DRD2	Dopamine receptor antagonist
7035	-99.08	kd	CGS001-7360	UGP2	-			
7036	-99.1	oe	ccsbBroad304_05390	DUSP28	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7037	-99.1	cp	BRD-K21680192	mitoxantrone	Topoisomerase inhibitor		TOP2A, PIM1	Topoisomerase inhibitor
7038	-99.1	cp	BRD-A98283014	calmidazolium	Calcium channel blocker		ATP2B1, PDE1A	Calcium channel blocker, Calmodulin antagonist
7039	-99.1	kd	CGS001-7433	VIPR1	GPCR / Class B : VIP and PACAP (ADCYAP1) receptors			
7040	-99.1	kd	CGS001-1462	VCAN	Immunoglobulin superfamily / V-set domain containing			
7041	-99.1	kd	CGS001-6429	SRSF4	RNA binding motif (RRM) containing			
7042	-99.1	kd	CGS001-55274	PHF10	Zinc fingers, PHD-type			
7043	-99.12	cc		SMAD family LOF	-			
7044	-99.12	cp	BRD-A02189320	met-leu-phe	-666			-666
7045	-99.12	kd	CGS001-8635	RNASET2	-			
7046	-99.14	kd	CGS001-94235	GNG8	-			
7047	-99.15	cp	BRD-K18779551	bifemelane	Acetylcholine release stimulant		SLC6A2	Acetylcholine release stimulant, Adrenergic transmitter uptake inhibitor, Reducing agent
7048	-99.15	kd	CGS001-4602	MYB	-			
7049	-99.15	kd	CGS001-3755	KCNG1	Voltage-gated potassium channels			
7050	-99.16	kd	CGS001-51727	CMPK1	-			
7051	-99.17	oe	ccsbBroad304_00818	IDH3A	-			
7052	-99.17	kd	CGS001-6773	STAT2	SH2 domain containing			
7053	-99.21	kd	CGS001-9491	PSMF1	Proteasome (prosome, macropain) subunits			
7054	-99.21	kd	CGS001-2645	GCK	Hexokinases			
7055	-99.23	oe	ccsbBroad304_07506	UBAP2L	-			
7056	-99.23	oe	ccsbBroad304_00100	RHOA	-			
7057	-99.23	cp	BRD-K36377456	marmesin	Angiogenesis inhibitor			Angiogenesis inhibitor
7058	-99.23	cp	BRD-K26573499	DMAB-anabaseine	Adrenergic receptor agonist		CHRNA7	Adrenergic receptor agonist
7059	-99.23	kd	CGS001-7150	TOP1	DNA Topoisomerases			
7060	-99.25	oe	ccsbBroad304_00486	EFNB2	Ephrins			
7061	-99.25	cp	BRD-A83937277	mephenytoin	Hydantoin antiepileptic		SCN5A, CYP2C19	Hydantoin antiepileptic
7062	-99.25	kd	CGS001-9322	TRIP10	-			
7063	-99.26	oe	ccsbBroad304_06562	MAT1A	-			
7064	-99.26	oe	ccsbBroad304_00874	INS	-			
7065	-99.26	cp	BRD-K49049886	CGS-15943	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
7066	-99.26	cp	BRD-A36267905	buphenine	Adrenergic receptor agonist		ADRB2	Adrenergic receptor agonist
7067	-99.26	kd	CGS001-6721	SREBF2	Basic helix-loop-helix proteins			
7068	-99.26	kd	CGS001-10461	MERTK	Type XI RTKs: TAM (TYRO3-, AXL- and MER-TK) receptor family			
7069	-99.27	kd	CGS001-4329	ALDH6A1	Aldehyde dehydrogenases			
7070	-99.28	oe	ccsbBroad304_06220	FOS	basic leucine zipper proteins			
7071	-99.28	kd	CGS001-255738	PCSK9	Subtilisin			
7072	-99.3	kd	CGS001-118442	GPR62	GPCR / Class A : Orphans			
7073	-99.32	oe	ccsbBroad304_00655	GNB2	WD repeat domain containing			
7074	-99.32	cp	BRD-K99616396	motesanib	KIT inhibitor		FLT1, FLT4, KDR, KIT, PDGFRA, RET	KIT inhibitor, PDGFR receptor inhibitor, VEGFR inhibitor
7075	-99.32	cp	BRD-K86595100	chlordiazepoxide	Benzodiazepine receptor agonist		GABRA1, GABRA2, GABRA3, GABRA4, GABRA5, GABRA6, GABRB1, GABRB2, GABRB3, GABRD, GABRE, GABRG1, GABRG2, GABRG3, GABRP, GABRQ	Benzodiazepine receptor agonist
7076	-99.32	kd	CGS001-10161	LPAR6	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7077	-99.32	kd	CGS001-11019	LIAS	-			
7078	-99.32	kd	CGS001-3956	LGALS1	Endogenous ligands			
7079	-99.32	kd	CGS001-9289	GPR56	Adhesion Class GPCRs			
7080	-99.34	oe	ccsbBroad304_04525	TGIF2LY	Homeoboxes / TALE class			
7081	-99.34	oe	ccsbBroad304_06678	OTX1	Homeoboxes / PRD class			
7082	-99.34	cp	BRD-K81528515	nilotinib	ABL inhibitor		ABL1, KIT, BCR, CYP2B6, CYP2C8, DDR1, DDR2, PDGFRA	ABL inhibitor, BCR-ABL kinase inhibitor
7083	-99.34	cp	BRD-K66296774	fluvastatin	HMGCR inhibitor		HMGCR, CYP2C8	HMGCR inhibitor
7084	-99.34	cp	BRD-A93000692	ciglitazone	PPAR receptor agonist		PPARG, INS	PPAR receptor agonist
7085	-99.35	cp	BRD-A81866333	CGS-21680	Adenosine receptor agonist		ADORA2A, ADORA1, ADORA2B, ADORA3	Adenosine receptor agonist
7086	-99.35	kd	CGS001-122809	SOCS4	SH2 domain containing			
7087	-99.35	kd	CGS001-10267	RAMP1	Receptor (G protein-coupled) activity modifying proteins			
7088	-99.37	oe	ccsbBroad304_00889	JUNB	basic leucine zipper proteins			
7089	-99.37	cp	BRD-K27737647	H-89	PKA inhibitor		PRKACA, GSG2, KCNA2, KCNA3, KCNA5, KCNAB2, KCNC1, KCNC2, KCNC3, KCNE1, KCNE2, KCNE3, KCNE4, KCNH1, KCNH2, KCNQ1, KCNQ2, KCNQ3, KCNQ5, KCNS3, PKIA	PKA inhibitor
7090	-99.37	kd	CGS001-51750	RTEL1	-			
7091	-99.37	cp	BRD-A75368507	demeclocycline	Bacterial 30S ribosomal subunit inhibitor			Bacterial 30S ribosomal subunit inhibitor
7092	-99.39	oe	ccsbBroad304_04613	HSPB9	Heat shock proteins / HSPB			
7093	-99.39	kd	CGS001-29110	TBK1	IKK family			
7094	-99.39	cp	BRD-A09539288	homatropine	Acetylcholine receptor antagonist		CES1, CHRM1	Acetylcholine receptor antagonist
7095	-99.39	cp	BRD-A47494775	dipivefrine	Adrenergic receptor agonist		ADRA1A, ACHE, ADRA2A, ADRB2, BCHE	Adrenergic receptor agonist
7096	-99.4	cp	BRD-K30990140	FR-122047	Cyclooxygenase inhibitor			Cyclooxygenase inhibitor
7097	-99.41	oe	ccsbBroad304_02990	LYPD3	-			
7098	-99.41	cp	BRD-A83431637	resmethrin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7099	-99.41	kd	CGS001-112858	TP53RK	Bud32 family			
7100	-99.41	kd	CGS001-5228	PGF	-			
7101	-99.41	cp	BRD-A84481105	thioridazine	Dopamine receptor antagonist		DRD1, DRD2, HTR2A, ADRA1A, ADRA1B, CHRNA7, DRD5, HRH1, HTR1A, HTR2C, HTR6, HTR7, KCNH2, MALT1	Dopamine receptor antagonist
7102	-99.42	cp	BRD-K04877770	FTase-inhibitor-B581	Farnesyltransferase inhibitor			Farnesyltransferase inhibitor
7103	-99.42	kd	CGS001-637	BID	Endogenous ligands			
7104	-99.43	cp	BRD-K14536225	piceid	Glucosidase inhibitor		GAA, XDH	Glucosidase inhibitor
7105	-99.43	cp	BRD-K96809896	SKF-86002	p38 MAPK inhibitor		ALOX5, MAPK14	p38 MAPK inhibitor
7106	-99.43	kd	CGS001-5217	PFN2	-			
7107	-99.43	kd	CGS001-2167	FABP4	Fatty acid binding protein family			
7108	-99.44	cp	BRD-A54029483	IRL-2500	Endothelin receptor antagonist		EDNRB	Endothelin receptor antagonist
7109	-99.44	cp	BRD-K88789588	letrozole	Aromatase inhibitor		CYP19A1	Aromatase inhibitor
7110	-99.45	cc		Minor histocompatibility antigens LOF	-			
7111	-99.45	cp	BRD-U33728988	QL-X-138	MTOR inhibitor		BTK, JAK3, MKNK2, MTOR, PRKDC	MTOR inhibitor
7112	-99.45	cp	BRD-K87990216	piretanide	Glucocorticoid receptor agonist		SLC12A1, SLC12A2	Glucocorticoid receptor agonist
7113	-99.45	kd	CGS001-10481	HOXB13	Homeoboxes / ANTP class : HOXL subclass			
7114	-99.45	kd	CGS001-5127	CDK16	Cyclin-dependent kinases, TAIRE subfamily			
7115	-99.45	kd	CGS001-433	ASGR2	C-type lectin domain containing			
7116	-99.46	cp	BRD-K21936341	oxotremorine	Acetylcholine receptor agonist		CHRM2, CHRM1, CHRM3, CHRM4	Acetylcholine receptor agonist, Cholinergic receptor agonist
7117	-99.46	kd	CGS001-350383	GPR142	GPCR / Class A : Orphans			
7118	-99.47	oe	ccsbBroad304_07267	PDLIM4	-			
7119	-99.47	oe	ccsbBroad304_07634	AGPAT2	1-acylglycerol-3-phosphate O-acyltransferases			
7120	-99.47	kd	CGS001-6240	RRM1	Ribonucleoside-diphosphate reductases			
7121	-99.47	kd	CGS001-8334	HIST1H2AC	Histones / Replication-dependent			
7122	-99.48	oe	ccsbBroad304_03308	YTHDF2	-			
7123	-99.5	cp	BRD-A55913614	primaquine	Antimalarial		KRT7, NQO2	Antimalarial, DNA inhibitor
7124	-99.5	cp	BRD-A07875874	cilnidipine	Calcium channel blocker		CACNA1B, CACNA1C	Calcium channel blocker
7125	-99.5	kd	CGS001-5295	PIK3R1	Phosphatidylinositol kinases			
7126	-99.5	kd	CGS001-6194	RPS6	S ribosomal proteins			
7127	-99.5	kd	CGS001-9020	MAP3K14	MAPKKK:STE-unique family			
7128	-99.51	cp	BRD-K19220233	JNK-9L	JNK inhibitor		MAPK8	JNK inhibitor
7129	-99.52	oe	ccsbBroad304_08782	SNX6	Sorting nexins			
7130	-99.52	cp	BRD-K40175214	torin-1	MTOR inhibitor		MTOR, PIK3CA	MTOR inhibitor, PI3K inhibitor
7131	-99.52	cp	BRD-K13810148	givinostat	HDAC inhibitor		HDAC2, HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, HDAC9, IL1B, IL1R2, IL6R, TNF	HDAC inhibitor
7132	-99.54	oe	ccsbBroad304_01660	TFAP4	Basic helix-loop-helix proteins			
7133	-99.54	oe	ccsbBroad304_02702	MSRB2	-			
7134	-99.54	cp	BRD-A12560204	nitrendipine	Calcium channel blocker		CACNA1C, CACNA1D, CACNA2D1, CACNA1H, CACNA1S, CACNA2D2, CACNB2, CACNG1, KCNN4	Calcium channel blocker
7135	-99.54	cp	BRD-K13032584	procarbazine	Monoamine oxidase inhibitor			Monoamine oxidase inhibitor
7136	-99.54	kd	CGS001-89910	UBE3B	-			
7137	-99.54	kd	CGS001-1728	NQO1	-			
7138	-99.55	kd	CGS001-55907	CMAS	-			
7139	-99.56	oe	ccsbBroad304_06126	TSC22D3	-			
7140	-99.56	cp	BRD-A01787639	naftopidil	Adrenergic receptor antagonist		ADRA1A, ADRA1D	Adrenergic receptor antagonist
7141	-99.56	kd	CGS001-57761	TRIB3	Trbl family			
7142	-99.56	kd	CGS001-55876	GSDMB	-			
7143	-99.57	kd	CGS001-51385	ZNF589	Zinc fingers, C2H2-type			
7144	-99.57	kd	CGS001-3458	IFNG	Interferons			
7145	-99.58	oe	ccsbBroad304_00840	IGFBP7	insulin-like growth factor (IGF) binding proteins			
7146	-99.58	oe	ccsbBroad304_01769	VEGFB	-			
7147	-99.58	cp	BRD-K73397362	purmorphamine	Smoothened receptor agonist		SMO, DHH, IHH, PTCH1	Smoothened receptor agonist
7148	-99.58	kd	CGS001-51776	ZAK	MLK subfamily			
7149	-99.58	kd	CGS001-5460	POU5F1	Homeoboxes / POU class			
7150	-99.58	kd	CGS001-4199	ME1	-			
7151	-99.58	kd	CGS001-863	CBFA2T3	A-kinase anchor proteins			
7152	-99.58	kd	CGS001-111	ADCY5	Adenylate cyclases			
7153	-99.58	cp	BRD-A70407468	PSB-36	Adenosine receptor antagonist		ADORA1, ADORA2A, ADORA2B, ADORA3	Adenosine receptor antagonist
7154	-99.6	oe	ccsbBroad304_00140	ATP6V0A1	ATPases / V-type			
7155	-99.6	cp	BRD-K15842202	eudesmic-acid	-666			-666
7156	-99.6	kd	CGS001-319100	TAAR6	GPCR / Class A : Trace amine associated receptors			
7157	-99.6	kd	CGS001-1642	DDB1	-			
7158	-99.61	oe	ccsbBroad304_03594	TNFRSF19	Tumour necrosis factor (TNF) receptor family			
7159	-99.61	oe	ccsbBroad304_01723	TTK	TTK family			
7160	-99.61	oe	ccsbBroad304_02026	NRP1	CD molecules			
7161	-99.61	oe	ccsbBroad304_13499	KSR2	RAF family			
7162	-99.61	oe	ccsbBroad304_03574	FBXW7	F-boxes / WD-40 domains			
7163	-99.61	cp	BRD-K77908580	entinostat	HDAC inhibitor		HDAC1, HDAC2, HDAC3, HDAC9	HDAC inhibitor
7164	-99.61	cp	BRD-K31471398	dihydrexidine	Dopamine receptor agonist		DRD1, DRD2, DRD3, DRD4, DRD5	Dopamine receptor agonist
7165	-99.61	cp	BRD-A45889380	mepacrine	Cytokine production inhibitor		TP53, AKT1, MTOR, NFKB1, PLA2G1B, PLA2G2A, PLA2G2D, PLA2G4A, PLA2G6, PLCL1	Cytokine production inhibitor, NFkB pathway inhibitor, TP53 activator
7166	-99.61	cp	BRD-A52588987	SKF-83566	Dopamine receptor antagonist		DRD1, DRD5	Dopamine receptor antagonist
7167	-99.61	kd	CGS001-11254	SLC6A14	Glycine transporter subfamily			
7168	-99.61	kd	CGS001-6233	RPS27A	S ribosomal proteins			
7169	-99.61	cp	BRD-A09925278	etilefrine	Adrenergic receptor agonist		ADRA1A, ADRB1	Adrenergic receptor agonist
7170	-99.63	oe	ccsbBroad304_02205	WTAP	-			
7171	-99.63	oe	ccsbBroad304_00789	HSBP1	-			
7172	-99.63	oe	ccsbBroad304_05881	BCL2L2	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7173	-99.63	cp	BRD-K89162000	tandutinib	FLT3 inhibitor		FLT3, KIT, PDGFRA, PDGFRB, CSF1R, PDGFD	FLT3 inhibitor, KIT inhibitor, PDGFR receptor inhibitor
7174	-99.63	cp	BRD-A38030642	cyclosporin-a	Calcineurin inhibitor		PPIA, ABCB11, CAMLG, CYP3A5, CYP3A7, FPR1, PPID, PPIF, PPP3CA, PPP3R2, SLC10A1, SLCO1B1, SLCO1B3	Calcineurin inhibitor
7175	-99.63	cp	BRD-K89402695	L-655240	Thromboxane receptor antagonist		PTGES	Thromboxane receptor antagonist
7176	-99.63	cp	BRD-K67860401	AR-A014418	Glycogen synthase kinase inhibitor		GSK3B	Glycogen synthase kinase inhibitor
7177	-99.63	kd	CGS001-2877	GPX2	-			
7178	-99.64	kd	CGS001-10600	USP16	Ubiquitin-specific peptidases			
7179	-99.64	kd	CGS001-3125	HLA-DRB3	Immunoglobulin superfamily / C1-set domain containing			
7180	-99.65	oe	ccsbBroad304_06304	GPC1	Proteoglycans / Cell Surface : Glypicans			
7181	-99.65	oe	ccsbBroad304_02840	PISD	Decarboxylases			
7182	-99.65	kd	CGS001-3306	HSPA2	Heat shock proteins / HSP70			
7183	-99.65	kd	CGS001-1182	CLCN3	Ion channels / Chloride channels : Voltage-sensitive			
7184	-99.65	kd	CGS001-327	APEH	Prolyl oligopeptidase			
7185	-99.66	kd	CGS001-382	ARF6	ADP-ribosylation factors			
7186	-99.67	oe	ccsbBroad304_05985	CFL1	-			
7187	-99.67	cp	BRD-K04887706	AKT-inhibitor-1-2	AKT inhibitor		AKT1, AKT2, AKT3	AKT inhibitor
7188	-99.67	cp	BRD-K66782112	BRD-K66782112	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
7189	-99.67	kd	CGS001-3084	NRG1	Immunoglobulin superfamily / I-set domain containing			
7190	-99.67	kd	CGS001-3428	IFI16	-			
7191	-99.67	kd	CGS001-27161	EIF2C2	-			
7192	-99.69	oe	ccsbBroad304_10423	BMPR1A	Type I receptor serine/threonine kinases			
7193	-99.69	cp	BRD-A25569250	KI-16425	Lysophosphatidic acid receptor antagonist		LPAR1, LPAR3	Lysophosphatidic acid receptor antagonist
7194	-99.69	cp	BRD-K19284129	salvinorin-a	Opioid receptor agonist		OPRK1, OPRD1, OPRM1	Opioid receptor agonist
7195	-99.69	cp	BRD-K19352500	prochlorperazine	Dopamine receptor antagonist		DRD2, DRD1, DRD3, DRD4	Dopamine receptor antagonist
7196	-99.69	kd	CGS001-6119	RPA3	-			
7197	-99.69	kd	CGS001-4697	NDUFA4	-			
7198	-99.69	kd	CGS001-9415	FADS2	Fatty acid desaturases			
7199	-99.69	kd	CGS001-2050	EPHB4	Type XIII RTKs: Ephrin receptor family			
7200	-99.7	kd	CGS001-51433	ANAPC5	Anaphase promoting complex subunits			
7201	-99.72	oe	ccsbBroad304_00390	CTGF	-			
7202	-99.72	cp	BRD-A37052580	physostigmine	Acetylcholinesterase inhibitor		ACHE, BCHE	Acetylcholinesterase inhibitor, Cholinesterase inhibitor
7203	-99.72	cp	BRD-K54987996	CAY-10578	Casein kinase inhibitor			Casein kinase inhibitor
7204	-99.72	cp	BRD-A68281735	REV-5901	Leukotriene receptor antagonist		ALOX5	Leukotriene receptor antagonist, Lipoxygenase inhibitor
7205	-99.72	kd	CGS001-7280	TUBB2A	Tubulins			
7206	-99.72	kd	CGS001-1029	CDKN2A	-			
7207	-99.73	kd	CGS001-2057	EPOR	Prolactin receptor family			
7208	-99.74	oe	ccsbBroad304_01514	SDHC	Mitochondrial respiratory chain complex / Complex II			
7209	-99.74	oe	ccsbBroad304_08511	RFK	-			
7210	-99.74	oe	ccsbBroad304_04678	GPR146	GPCR / Class A : Orphans			
7211	-99.74	oe	ccsbBroad304_00170	BNIP1	-			
7212	-99.74	oe	ccsbBroad304_00116	ASS1	-			
7213	-99.74	cp	BRD-A71657825	2-(biphenyl-4-ylsulfonamido)pentanedioic-acid	Matrix metalloprotease inhibitor		MMP13, MMP8, MMP9	Matrix metalloprotease inhibitor
7214	-99.74	cp	BRD-K41564320	purvalanol-b	Tyrosine kinase inhibitor		CDK2, CDK4, MAPK1, MAPK3, CDK5, SRPK2	Tyrosine kinase inhibitor
7215	-99.74	cp	BRD-K54095730	CMPD-1	p38 MAPK inhibitor		GNRHR, MAPK14	p38 MAPK inhibitor
7216	-99.74	cp	BRD-K49294207	BIBU-1361	EGFR inhibitor		EGFR	EGFR inhibitor
7217	-99.74	kd	CGS001-7226	TRPM2	Transient Receptor Potential channels			
7218	-99.74	kd	CGS001-6776	STAT5A	SH2 domain containing			
7219	-99.74	kd	CGS001-51601	LIPT1	-			
7220	-99.74	kd	CGS001-51135	IRAK4	Interleukin-1 receptor-associated kinase (IRAK) family			
7221	-99.74	kd	CGS001-3030	HADHA	-			
7222	-99.74	kd	CGS001-2289	FKBP5	Tetratricopeptide (TTC) repeat domain containing			
7223	-99.74	kd	CGS001-25842	ASF1A	-			
7224	-99.76	oe	ccsbBroad304_03175	MRPS16	Mitochondrial ribosomal proteins / small subunits			
7225	-99.76	cp	BRD-K68174511	torin-2	MTOR inhibitor		MTOR	MTOR inhibitor
7226	-99.76	cp	BRD-A59985574	topotecan	Topoisomerase inhibitor		TOP1, TOP1MT	Topoisomerase inhibitor
7227	-99.76	cp	BRD-A33833419	TER-14687	Inhibitor of translocation of PKCq in T cells		PRKCQ	Inhibitor of translocation of PKCq in T cells
7228	-99.76	cp	BRD-K34820100	tebuthiuron	Photosynthesis inhibitor			Photosynthesis inhibitor
7229	-99.76	cp	BRD-K15567136	papaverine	Phosphodiesterase inhibitor		PDE10A, PDE4B, PDE5A	Phosphodiesterase inhibitor
7230	-99.76	cp	BRD-K81709173	halcinonide	Glucocorticoid receptor agonist		NR3C1	Glucocorticoid receptor agonist
7231	-99.76	kd	CGS001-126375	ZNF792	Zinc fingers, C2H2-type			
7232	-99.76	kd	CGS001-23678	SGK3	SGK family			
7233	-99.76	kd	CGS001-3419	IDH3A	-			
7234	-99.78	oe	ccsbBroad304_09095	PUS7L	-			
7235	-99.78	oe	ccsbBroad304_00492	EIF5A	-			
7236	-99.78	cp	BRD-A18497530	5-iodotubercidin	Adenosine kinase inhibitor		MAPK3, ADK, CSNK1G2, GSG2, LRRK2	Adenosine kinase inhibitor
7237	-99.78	cp	BRD-K52911425	GDC-0941	PI3K inhibitor		PIK3CG, PIK3CA, PIK3CB, PIK3CD	PI3K inhibitor
7238	-99.78	cp	BRD-K63343048	orlistat	Lipase inhibitor		PNLIP, DAGLA, FASN, LIPF, CNR1, DAGLB	Lipase inhibitor
7239	-99.78	cp	BRD-A64933752	CV-1808	Adenosine receptor agonist		ADORA2A, ADORA2B	Adenosine receptor agonist
7240	-99.78	cp	BRD-K20482099	rutin	Antioxidant		AKR1C3, AKR1B1, F10	Antioxidant, Capillary stabilizing agent, Nitric oxide scavenger
7241	-99.78	kd	CGS001-64127	NOD2	Nucleotide-binding domain and leucine rich repeat containing			
7242	-99.78	kd	CGS001-823	CAPN1	EF-hand domain containing			
7243	-99.8	oe	ccsbBroad304_05773	ADCY9	Adenylyl cyclases			
7244	-99.8	oe	ccsbBroad304_02572	SERINC3	-			
7245	-99.8	cp	BRD-A85025557	NCS-382	GABA receptor antagonist		GABBR1, GABBR2, SLC52A2	GABA receptor antagonist
7246	-99.8	cp	BRD-A12016240	LY-278584	Serotonin receptor antagonist		HTR3A	Serotonin receptor antagonist
7247	-99.8	cp	BRD-A09056319	alfuzosin	Adrenergic receptor antagonist		ADRA1A, ADRA1D, ADRA1B, KCNH2	Adrenergic receptor antagonist
7248	-99.8	kd	CGS001-25800	SLC39A6	SLC39 family of metal ion transporters			
7249	-99.8	kd	CGS001-6500	SKP1	-			
7250	-99.8	kd	CGS001-4718	NDUFC2	Mitochondrial respiratory chain complex / Complex I			
7251	-99.8	kd	CGS001-7976	FZD3	GPCR / Class F : Frizzled receptors			
7252	-99.8	kd	CGS001-3171	FOXA3	Forkhead boxes			
7253	-99.8	oe	ccsbBroad304_05972	CDC25C	Serine/threonine phosphatases / Protein phosphatase 1, regulatory subunits			
7254	-99.82	oe	ccsbBroad304_01065	NDUFA3	Mitochondrial respiratory chain complex / Complex I			
7255	-99.82	oe	ccsbBroad304_02373	SPRY2	-			
7256	-99.82	oe	ccsbBroad304_05348	FOXR1	Forkhead boxes			
7257	-99.82	oe	ccsbBroad304_00518	ETFA	-			
7258	-99.82	cp	BRD-A01317026	7,8-dihydro-L-biopterin	Dihydroneopterin aldolase inhibitor		NOS2, TPH1	Dihydroneopterin aldolase inhibitor
7259	-99.82	cp	BRD-U86922168	QL-XII-47	BTK inhibitor		BMX, BTK	BTK inhibitor, Cytoplasmic tyrosine protein kinase BMX inhibitor
7260	-99.82	cp	BRD-K23383398	T-0901317	LXR agonist		NR1H3, NR1H2, ABCA1, NCOA1, NCOA2, NR1I2, RORA, RORC, RXRB	LXR agonist, ABC transporter expression enhancer, ROR inverse agonist
7261	-99.82	cp	BRD-K35941380	methysergide	Serotonin receptor antagonist		HTR2C, HTR1B, HTR1E, HTR1F, HTR2A, HTR2B, HTR7, HTR1A, HTR1D, HTR5A, HTR6	Serotonin receptor antagonist
7262	-99.82	cp	BRD-A30437061	camptothecin	Topoisomerase inhibitor		TOP1, HIF1A	Topoisomerase inhibitor
7263	-99.82	cp	BRD-K13642330	cosmosiin	Cytochrome P450 inhibitor			Cytochrome P450 inhibitor
7264	-99.82	kd	CGS001-116512	MRGPRD	GPCR / Class A : Orphans			
7265	-99.82	kd	CGS001-79618	HMBOX1	Homeoboxes / HNF class			
7266	-99.82	kd	CGS001-55869	HDAC8	Histone deacetylases			
7267	-99.82	kd	CGS001-2224	FDPS	Lanosterol biosynthesis pathway			
7268	-99.82	kd	CGS001-2150	F2RL1	GPCR / Class A : Protease activated receptors			
7269	-99.82	oe	ccsbBroad304_02506	EBP	-			
7270	-99.82	cp	BRD-K22662435	ganciclovir	DNA polymerase inhibitor			DNA polymerase inhibitor
7271	-99.84	oe	ccsbBroad304_01455	RPS16	S ribosomal proteins			
7272	-99.84	kd	CGS001-8732	RNGTT	Protein tyrosine phosphatases / Class I Cys-based PTPs : Atypical dual specificity phosphatases			
7273	-99.85	oe	ccsbBroad304_00488	EGR3	Zinc fingers, C2H2-type			
7274	-99.85	oe	ccsbBroad304_02751	SATB2	Homeoboxes / CUT class			
7275	-99.85	oe	ccsbBroad304_00223	CASP9	Caspases			
7276	-99.85	cp	BRD-K64800655	PHA-793887	CDK inhibitor		CDK1, CDK2, CDK4, CDK5, CCND1, CCNE1, CDK7, CDK9	CDK inhibitor
7277	-99.85	kd	CGS001-431707	LHX8	Homeoboxes / LIM class			
7278	-99.85	kd	CGS001-8805	TRIM24	TIF1 family			
7279	-99.85	kd	CGS001-6660	SOX5	SRY (sex determining region Y)-boxes			
7280	-99.85	kd	CGS001-6223	RPS19	S ribosomal proteins			
7281	-99.85	kd	CGS001-23566	LPAR3	GPCR / Class A : Lysophospholipid receptors : Lysophosphatidic acid			
7282	-99.85	kd	CGS001-486	FXYD2	Ion transport regulator			
7283	-99.85	kd	CGS001-24140	FTSJ1	-			
7284	-99.85	kd	CGS001-51635	DHRS7	Short chain dehydrogenase/reductase superfamily / Classical SDR fold cluster 3			
7285	-99.85	kd	CGS001-31	ACACA	Carboxylases			
7286	-99.86	cp	BRD-K28183345	proguanil	Dihydrofolate reductase inhibitor		CYP2C19, DHFR	Dihydrofolate reductase inhibitor
7287	-99.87	oe	ccsbBroad304_06683	FURIN	Subtilisin			
7288	-99.87	oe	ccsbBroad304_00232	SERPINA6	Serine (or cysteine) peptidase inhibitors			
7289	-99.87	oe	ccsbBroad304_01967	PPAP2A	Lipid phosphate phosphatases			
7290	-99.87	oe	ccsbBroad304_07287	HYAL2	-			
7291	-99.87	cp	BRD-A96799240	4-hydroxyretinoic-acid	Retinoid receptor binder			Retinoid receptor binder
7292	-99.87	cp	BRD-K49481516	galantamine	Acetylcholinesterase inhibitor		ACHE, BCHE, CHRNA1, CHRNA10, CHRNA2, CHRNA3, CHRNA4, CHRNA5, CHRNA6, CHRNA7, CHRNA9, CHRNB1, CHRNB2, CHRNB3, CHRNB4, CHRND, CHRNE, CHRNG	Acetylcholinesterase inhibitor
7293	-99.87	cp	BRD-K64157027	ZD-2079	Adrenergic receptor agonist		ADRB3	Adrenergic receptor agonist
7294	-99.87	cp	BRD-K66019333	oxantel	Anthelmintic			Anthelmintic
7295	-99.87	cp	BRD-K84709232	caffeic-acid	Lipoxygenase inhibitor		ALOX5, MIF, RELA, TNF	Lipoxygenase inhibitor, HIV integrase inhibitor, NFkB pathway inhibitor, Nitric oxide production inhibitor, PPAR receptor modulator, TNF production inhibitor, Tumor necrosis factor production inhibitor
7296	-99.87	cp	BRD-K97810537	beclometasone	Glucocorticoid receptor agonist		NR3C1, CYP3A5, GPR97, SERPINA6	Glucocorticoid receptor agonist, Immunosuppressant
7297	-99.87	kd	CGS001-84231	TRAF7	RING-type (C3HC4) zinc fingers			
7298	-99.87	kd	CGS001-5586	PKN2	Protein kinase N (PKN) family			
7299	-99.87	kd	CGS001-8554	PIAS1	Zinc fingers, MIZ-type			
7300	-99.87	kd	CGS001-4149	MAX	Basic helix-loop-helix proteins			
7301	-99.87	kd	CGS001-2621	GAS6	-			
7302	-99.89	oe	ccsbBroad304_06637	NFKB1	NFkappaB transcription factor family			
7303	-99.89	oe	ccsbBroad304_07158	ZNF74	Zinc fingers, C2H2-type			
7304	-99.89	oe	ccsbBroad304_01958	YARS	Aminoacyl tRNA synthetases / Class I			
7305	-99.89	oe	ccsbBroad304_07802	TWF2	Twinfilin subfamily			
7306	-99.89	oe	ccsbBroad304_02674	STK38	NDR family			
7307	-99.89	oe	ccsbBroad304_01401	RIT1	-			
7308	-99.89	oe	ccsbBroad304_01373	RAN	-			
7309	-99.89	cp	BRD-K13390322	AT-7519	CDK inhibitor		CDK2, CDK5, CDK1, CDK4, CDK6, CDK9	CDK inhibitor, Cell cycle inhibitor
7310	-99.89	cp	BRD-K15086322	JNJ-10191584	Histamine receptor antagonist		HRH4	Histamine receptor antagonist
7311	-99.89	cp	BRD-A48570745	ivermectin	GABA receptor agonist		CHRNA7, GABRB3, GLRA3, P2RX7	GABA receptor agonist
7312	-99.89	cp	BRD-K41160163	fenobam	Glutamate receptor antagonist		GRM5	Glutamate receptor antagonist
7313	-99.89	cp	BRD-A90311807	cilastatin	Dehydropeptidase inhibitor		DPEP1	Dehydropeptidase inhibitor
7314	-99.89	kd	CGS001-83439	TCF7L1	-			
7315	-99.89	kd	CGS001-83999	KREMEN1	-			
7316	-99.89	kd	CGS001-94239	H2AFV	Histones / Replication-independent			
7317	-99.89	kd	CGS001-51053	GMNN	-			
7318	-99.89	kd	CGS001-2079	ERH	-			
7319	-99.89	kd	CGS001-1892	ECHS1	-			
7320	-99.89	kd	CGS001-6790	AURKA	Aurora kinase			
7321	-99.91	cc		Thromboxane receptor antagonist	-			
7322	-99.91	oe	ccsbBroad304_07322	SGPL1	Sphingosine 1-phosphate lyase			
7323	-99.91	oe	ccsbBroad304_03917	RBKS	-			
7324	-99.91	oe	ccsbBroad304_04216	PBX4	Homeoboxes / TALE class			
7325	-99.91	oe	ccsbBroad304_05135	PARP15	-			
7326	-99.91	oe	ccsbBroad304_05523	KRT26	Intermediate filaments type I, keratins (acidic)			
7327	-99.91	oe	ccsbBroad304_03859	ENOPH1	-			
7328	-99.91	oe	ccsbBroad304_02048	BCL10	-			
7329	-99.91	cp	BRD-A80960055	celastrol	Anti-inflammatory		IL1B, TNF	Anti-inflammatory, Antioxidant, NFkB pathway inhibitor, HSP inhibitor, Topoisomerase inhibitor
7330	-99.91	cp	BRD-A58157837	butabindide	Tripeptidyl peptidase inhibitor		TPP2	Tripeptidyl peptidase inhibitor
7331	-99.91	kd	CGS001-84765	ZNF577	Zinc fingers, C2H2-type			
7332	-99.91	kd	CGS001-124961	ZFP3	Zinc fingers, C2H2-type			
7333	-99.91	kd	CGS001-6207	RPS13	S ribosomal proteins			
7334	-99.91	kd	CGS001-4141	MARS	Aminoacyl tRNA synthetases / Class I			
7335	-99.91	kd	CGS001-3421	IDH3G	-			
7336	-99.91	kd	CGS001-9156	EXO1	-			
7337	-99.91	kd	CGS001-54505	DHX29	DEAH-boxes			
7338	-99.91	kd	CGS001-604	BCL6	BTB/POZ domain containing			
7339	-99.91	kd	CGS001-8313	AXIN2	-			
7340	-99.92	oe	ccsbBroad304_02625	SLC7A9	SLC7 family			
7341	-99.93	oe	ccsbBroad304_01716	TSN	-			
7342	-99.93	oe	ccsbBroad304_06934	SFPQ	RNA binding motif (RRM) containing			
7343	-99.93	oe	ccsbBroad304_06663	OAS1	-			
7344	-99.93	oe	ccsbBroad304_00851	IL6R	IL-6 receptor family			
7345	-99.93	oe	ccsbBroad304_00833	IFNG	Interferons			
7346	-99.93	oe	ccsbBroad304_01808	ZNF134	Zinc fingers, C2H2-type			
7347	-99.93	oe	ccsbBroad304_09043	TSEN2	tRNA splicing endonuclease subunits			
7348	-99.93	oe	ccsbBroad304_07320	SQSTM1	-			
7349	-99.93	oe	ccsbBroad304_02709	SCMH1	Sterile alpha motif (SAM) domain containing			
7350	-99.93	oe	ccsbBroad304_00034	AES	-			
7351	-99.93	cp	BRD-K11636097	JNJ-7706621	CDK inhibitor		CDK1, CDK2, AURKA, AURKB	CDK inhibitor
7352	-99.93	cp	BRD-K81855038	roxatidine	Histamine receptor antagonist		HRH2	Histamine receptor antagonist
7353	-99.93	cp	BRD-A16311756	profenamine	Butyrylcholinesterase inhibitor		CHRM1, BCHE, CHRM2, GRIN3A	Butyrylcholinesterase inhibitor, Cholinergic receptor antagonist
7354	-99.93	cp	BRD-K00486786	RO-08-2750	NGF binding inhibitor		NGFR, NGF	NGF binding inhibitor
7355	-99.93	cp	BRD-K56596464	QX-314	Sodium channel blocker		MAPK14, TGFBR1	Sodium channel blocker
7356	-99.93	cp	BRD-K02283807	GR-32191	Thromboxane receptor antagonist		TBXA2R	Thromboxane receptor antagonist
7357	-99.93	kd	CGS001-6493	SIM2	Basic helix-loop-helix proteins			
7358	-99.93	kd	CGS001-5378	PMS1	-			
7359	-99.93	kd	CGS001-8566	PDXK	-			
7360	-99.93	kd	CGS001-4926	NUMA1	-			
7361	-99.93	kd	CGS001-2618	GART	Ribosyl transferases			
7362	-99.93	kd	CGS001-2263	FGFR2	Type V RTKs: FGF (fibroblast growth factor) receptor family			
7363	-99.93	kd	CGS001-2181	ACSL3	Acyl-CoA synthetase family			
7364	-99.93	kd	CGS001-18	ABAT	GABA turnover			
7365	-99.93	oe	ccsbBroad304_00175	ZFP36L1	RING-type (C3HC4) zinc fingers			
7366	-99.93	oe	ccsbBroad304_00233	CBR1	Prostaglandin synthases			
7367	-99.94	kd	CGS001-5162	PDHB	-			
7368	-99.95	oe	ccsbBroad304_00888	ITPK1	-			
7369	-99.95	kd	CGS001-665	BNIP3L	-			
7370	-99.96	cc		GATA Zinc finger domain containing LOF	-			
7371	-99.96	oe	ccsbBroad304_10994	NEK2	NIMA (never in mitosis gene a)- related kinase (NEK) family			
7372	-99.96	oe	ccsbBroad304_02432	IFI30	-			
7373	-99.96	oe	ccsbBroad304_06649	CNOT4	RNA binding motif (RRM) containing			
7374	-99.96	oe	ccsbBroad304_08313	ZNF581	Zinc fingers, C2H2-type			
7375	-99.96	oe	ccsbBroad304_07164	ZNF133	Zinc fingers, C2H2-type			
7376	-99.96	oe	ccsbBroad304_03736	SUCNR1	GPCR / Class A : Orphans			
7377	-99.96	oe	ccsbBroad304_01610	STAT4	SH2 domain containing			
7378	-99.96	oe	ccsbBroad304_01475	S100A6	EF-hand domain containing			
7379	-99.96	oe	ccsbBroad304_06888	RPN1	-			
7380	-99.96	oe	ccsbBroad304_09703	RNF145	RING-type (C3HC4) zinc fingers			
7381	-99.96	oe	ccsbBroad304_07961	RCHY1	RING-type (C3HC4) zinc fingers			
7382	-99.96	oe	ccsbBroad304_02864	PRDX5	-			
7383	-99.96	oe	ccsbBroad304_07272	PPAP2B	Lipid phosphate phosphatases			
7384	-99.96	oe	ccsbBroad304_02208	PDIA4	Protein disulfide isomerases			
7385	-99.96	oe	ccsbBroad304_00944	LIMK2	LIMK subfamily			
7386	-99.96	oe	ccsbBroad304_10157	LHX8	Homeoboxes / LIM class			
7387	-99.96	oe	ccsbBroad304_02249	KIAA0494	-			
7388	-99.96	oe	ccsbBroad304_02974	HAVCR1	Immunoglobulin superfamily / V-set domain containing			
7389	-99.96	oe	ccsbBroad304_00563	FGG	Endogenous ligands			
7390	-99.96	oe	ccsbBroad304_00796	DNAJB2	Heat shock proteins / DNAJ (HSP40)			
7391	-99.96	oe	ccsbBroad304_05944	CCBL1	Hydrogen sulphide synthesis			
7392	-99.96	oe	ccsbBroad304_00138	ATP6V0B	ATPases / V-type			
7393	-99.96	oe	ccsbBroad304_07273	ASMTL	Pseudoautosomal regions / PAR1			
7394	-99.96	oe	ccsbBroad304_03469	ANKRD49	Ankyrin repeat domain containing			
7395	-99.96	oe	ccsbBroad304_00053	ALDOA	-			
7396	-99.96	cp	BRD-A26002865	verrucarin-a	Protein synthesis inhibitor			Protein synthesis inhibitor
7397	-99.96	cp	BRD-K44353683	nateglinide	Insulin secretagogue		ABCC8, KCNJ11, CYP3A4, INS, KCNJ10, PPARG	Insulin secretagogue
7398	-99.96	cp	BRD-K22947005	dexbrompheniramine	Histamine receptor antagonist		HRH1	Histamine receptor antagonist
7399	-99.96	cp	BRD-A81772229	simvastatin	HMGCR inhibitor		HMGCR, CYP2C8, CYP3A4, CYP3A5, ITGB2	HMGCR inhibitor
7400	-99.96	cp	BRD-A92161634	scopoline	Acetylcholine receptor antagonist			Acetylcholine receptor antagonist
7401	-99.96	cp	BRD-K68402494	ML-9	Myosin light chain kinase inhibitor		MLCK, TRPC6, PKA, PKC	Myosin light chain kinase inhibitor
7402	-99.96	cp	BRD-A17535965	gelsemine	Acetylcholine receptor antagonist		GLRA3	Acetylcholine receptor antagonist, Glycine receptor antagonist
7403	-99.96	cp	BRD-K43389675	daunorubicin	RNA synthesis inhibitor		TOP2A, TOP2B	RNA synthesis inhibitor, Topoisomerase inhibitor
7404	-99.96	cp	BRD-K11373525	ZD-7155	Angiotensin receptor antagonist		AGTR1	Angiotensin receptor antagonist
7405	-99.96	cp	BRD-A56012032	thiorphan	Membrane metalloendopeptidase inhibitor		MME	Membrane metalloendopeptidase inhibitor
7406	-99.96	cp	BRD-K60184833	tyrphostin-46	Tyrosine kinase inhibitor		EGFR	Tyrosine kinase inhibitor
7407	-99.96	cp	BRD-A77349281	RK-682	Tyrosine phosphatase inhibitor		HPSE, PTPN1	Tyrosine phosphatase inhibitor
7408	-99.96	cp	BRD-A66927094	nemonapride	Dopamine receptor antagonist		DRD2, DRD3, DRD4	Dopamine receptor antagonist
7409	-99.96	cp	BRD-K93460210	lamotrigine	Serotonin receptor antagonist		SCN1A, SCN2A, SCN3A	Serotonin receptor antagonist, Sodium channel blocker
7410	-99.96	cp	BRD-K78838262	austricine	Hypolipidemic			Hypolipidemic
7411	-99.96	cp	BRD-K94512704	spiramide	Dopamine receptor antagonist		DRD2, HTR1A, HTR2A, HTR2B, HTR2C	Dopamine receptor antagonist, Serotonin receptor antagonist
7412	-99.96	cp	BRD-K89055274	alverine	Muscle relaxant		HTR1A	Muscle relaxant
7413	-99.96	kd	CGS001-375449	MAST4	MAST family			
7414	-99.96	kd	CGS001-167465	ZNF366	Zinc fingers, C2H2-type			
7415	-99.96	kd	CGS001-7511	XPNPEP1	Methionyl aminopeptidase			
7416	-99.96	kd	CGS001-23475	QPRT	-			
7417	-99.96	kd	CGS001-5720	PSME1	Proteasome (prosome, macropain) subunits			
7418	-99.96	kd	CGS001-55011	PIH1D1	-			
7419	-99.96	kd	CGS001-3651	PDX1	Homeoboxes / ANTP class : HOXL subclass			
7420	-99.96	kd	CGS001-64710	NUCKS1	-			
7421	-99.96	kd	CGS001-4714	NDUFB8	Mitochondrial respiratory chain complex / Complex I			
7422	-99.96	kd	CGS001-9643	MORF4L2	-			
7423	-99.96	kd	CGS001-6300	MAPK12	MAPK:p38 subfamily			
7424	-99.96	kd	CGS001-3149	HMGB3	High-mobility group / Canonical			
7425	-99.96	kd	CGS001-2580	GAK	Heat shock proteins / DNAJ (HSP40)			
7426	-99.96	kd	CGS001-9700	ESPL1	-			
7427	-99.96	kd	CGS001-1869	E2F1	-			
7428	-99.96	kd	CGS001-1454	CSNK1E	Casein kinase 1 (CK1) family			
7429	-99.96	kd	CGS001-998	CDC42	-			
7430	-99.96	kd	CGS001-8659	ALDH4A1	Aldehyde dehydrogenases			
7431	-99.96	kd	CGS001-6868	ADAM17	ADAM metallopeptidase domain containing			
7432	-99.96	kd	CGS001-1956	EGFR	Type I RTKs: ErbB (epidermal growth factor) receptor family			
7433	-99.96	oe	ccsbBroad304_00487	EGR1	Zinc fingers, C2H2-type			
7434	-99.96	cp	BRD-K31283835	tofacitinib	JAK inhibitor		JAK3, JAK1, JAK2, CYP2C19, TYK2	JAK inhibitor
7435	-99.96	cp	BRD-K71823332	epothilone-a	Microtubule stabilizing agent			Microtubule stabilizing agent
7436	-99.96	cp	BRD-A30205217	ethotoin	Hydantoin antiepileptic		SCN5A	Hydantoin antiepileptic
7437	-99.97	kd	CGS001-23355	VPS8	-			
7438	-99.98	oe	ccsbBroad304_02018	SUCLA2	-			
7439	-99.98	cp	BRD-A11702965	chromomycin-a3	DNA binding agent			DNA binding agent
7440	-99.98	kd	CGS001-26137	ZBTB20	BTB/POZ domain containing			
7441	-99.98	kd	CGS001-9121	SLC16A5	SLC16 family of monocarboxylate transporters			
7442	-99.98	kd	CGS001-390148	OR5W2	GPCR / Class A : Olfactory receptors			
7443	-99.98	kd	CGS001-3897	L1CAM	CD molecules			
7444	-99.98	kd	CGS001-27201	GPR78	GPCR / Class A : Orphans			
7445	-99.98	kd	CGS001-1677	DFFB	-			
7446	-99.98	kd	CGS001-1490	CTGF	-			
7447	-99.98	kd	CGS001-573	BAG1	-			
7448	-100	cc		Ribosomal 40s Subunit LOF	-			
7449	-100	cp	BRD-K38615104	A-443644	AKT inhibitor		AKT1, AKT2, AKT3, CDC42BPB, GSK3B, PHKG1, PKIA, PRKACA	AKT inhibitor
7450	-100	cp	BRD-K87909389	alvocidib	CDK inhibitor		CDK2, CDK4, CDK1, CDK6, CDK7, CDK9, CDK5, CDK8, EGFR, PYGM, BCL2, BIRC5, CCNT1, MCL1, XIAP	CDK inhibitor
7451	-100	cp	BRD-K06792661	narciclasine	Coflilin signaling pathway activator		RHOA	Coflilin signaling pathway activator, LIM kinase activator, Rho associated kinase activator
7452	-100	cp	BRD-K11927976	ER-27319	Mediator release inhibitor		SYK	Mediator release inhibitor, SYK inhibitor
7453	-100	kd	CGS001-127396	ZNF684	Zinc fingers, C2H2-type			
7454	-100	kd	CGS001-147807	ZNF524	Zinc fingers, C2H2-type			
7455	-100	kd	CGS001-114026	ZIM3	Zinc fingers, C2H2-type			
7456	-100	kd	CGS001-54469	ZFAND6	Zinc fingers, AN1-type domain containing			
7457	-100	kd	CGS001-10352	WARS2	Aminoacyl tRNA synthetases / Class I			
7458	-100	kd	CGS001-51271	UBAP1	-			
7459	-100	kd	CGS001-7298	TYMS	Methyltransferases			
7460	-100	kd	CGS001-7227	TRPS1	GATA zinc finger domain containing			
7461	-100	kd	CGS001-7186	TRAF2	RING-type (C3HC4) zinc fingers			
7462	-100	kd	CGS001-10452	TOMM40	-			
7463	-100	kd	CGS001-6871	TADA2A	-			
7464	-100	kd	CGS001-6856	SYPL1	-			
7465	-100	kd	CGS001-9900	SV2A	Major facilitator superfamily (MFS) of transporters			
7466	-100	kd	CGS001-5979	RET	Type XIV RTKs: RET			
7467	-100	kd	CGS001-5686	PSMA5	Proteasome subunits			
7468	-100	kd	CGS001-3275	PRMT2	Protein arginine N-methyltransferases			
7469	-100	kd	CGS001-5533	PPP3CC	Serine/threonine phosphatases / Protein phosphatase, catalytic subunits			
7470	-100	kd	CGS001-133522	PPARGC1B	RNA binding motif (RRM) containing			
7471	-100	kd	CGS001-55193	PBRM1	Non-enzymatic BRD containing proteins			
7472	-100	kd	CGS001-4916	NTRK3	Type VII RTKs: Neurotrophin receptor/Trk family			
7473	-100	kd	CGS001-4171	MCM2	-			
7474	-100	kd	CGS001-8550	MAPKAPK5	MAPKAPK subfamily			
7475	-100	kd	CGS001-55379	LRRC59	-			
7476	-100	kd	CGS001-51520	LARS	Aminoacyl tRNA synthetases / Class I			
7477	-100	kd	CGS001-3880	KRT19	Intermediate filaments type I, keratins (acidic)			
7478	-100	kd	CGS001-85442	KNDC1	-			
7479	-100	kd	CGS001-51274	KLF3	Kruppel-like transcription factors			
7480	-100	kd	CGS001-8462	KLF11	Kruppel-like transcription factors			
7481	-100	kd	CGS001-64147	KIF9	Kinesins			
7482	-100	kd	CGS001-79711	IPO4	Importins			
7483	-100	kd	CGS001-50604	IL20	Interleukins and interleukin receptors			
7484	-100	kd	CGS001-3586	IL10	Interleukins and interleukin receptors			
7485	-100	kd	CGS001-3485	IGFBP2	insulin-like growth factor (IGF) binding proteins			
7486	-100	kd	CGS001-3476	IGBP1	-			
7487	-100	kd	CGS001-3339	HSPG2	Immunoglobulin superfamily / Immunoglobulin-like domain containing			
7488	-100	kd	CGS001-3281	HSBP1	-			
7489	-100	kd	CGS001-3158	HMGCS2	Lanosterol biosynthesis pathway			
7490	-100	kd	CGS001-10614	HEXIM1	-			
7491	-100	kd	CGS001-165829	GPR156	GPCR / Class C : Orphans			
7492	-100	kd	CGS001-2538	G6PC	-			
7493	-100	kd	CGS001-10023	FRAT1	-			
7494	-100	kd	CGS001-55770	EXOC2	-			
7495	-100	kd	CGS001-51295	ECSIT	Mitochondrial respiratory chain complex assembly factors			
7496	-100	kd	CGS001-1837	DTNA	-			
7497	-100	kd	CGS001-1649	DDIT3	-			
7498	-100	kd	CGS001-1491	CTH	Hydrogen sulphide synthesis			
7499	-100	kd	CGS001-51380	CSAD	-			
7500	-100	kd	CGS001-840	CASP7	Caspases			
7501	-100	kd	CGS001-8945	BTRC	F-boxes / WD-40 domains			
7502	-100	kd	CGS001-271	AMPD2	-			
7503	-100	kd	CGS001-10327	AKR1A1	Aldo-keto reductases			
7504	-100	kd	CGS001-95	ACY1	-			
7505	-100	kd	CGS001-5244	ABCB4	ATP binding cassette transporters / subfamily B			
7506	-100	cp	BRD-A80213327	NSC-23766	Ras GTPase inhibitor			Ras GTPase inhibitor
